Report error Found 621 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase 12'
Displayed 1 to 50 (of 621 total ) | Next | Last >>
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 0.110nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 0.120nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 0.170nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 0.200nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 0.210nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 0.240nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 0.290nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 0.290nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 0.290nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 0.300nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 0.310nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 0.360nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 0.360nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 0.360nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 0.390nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 0.400nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 0.5nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: <0.5nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
3D Structure (crystal)TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 0.5nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 0.620nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 0.620nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 0.700nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 0.735nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 0.740nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 0.850nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 0.900nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 0.950nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 1nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 1nMAssay Description:Binding affinity to N-terminally GST-tagged wild type human DLK (1 to 520 residues) expressed in sf21 insect cells using N-terminally His-tagged MKK4...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 1nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 1nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 1.10nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 1.25nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 1.59nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 1.60nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 1.60nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 1.64nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 1.72nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 1.90nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human DLK (9 to 111 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human DLK (9 to 111 residues) expressed in Sf21 cells assessed as reduction in substrate phosphorylat...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataIC50: 2nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 2nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 2.10nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 2.20nMAssay Description:A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 2.20nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 2.23nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 2.30nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKi: 2.30nMAssay Description:Binding affinity to N-terminally GST-tagged wild type human DLK (1 to 520 residues) expressed in sf21 insect cells using N-terminally His-tagged MKK4...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System
US Patent
The University of Texas System
US Patent
Affinity DataKd: 2.40nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair