Compile Data Set for Download or QSAR
Report error Found 443 Enz. Inhib. hit(s) with Target = 'Motilin receptor'
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599720(H-Motilin | CHEMBL525634)
Affinity DataEC50:  0.970nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50292978(GSK-962040 | N-(3-Fluorophenyl)-1-[(4-([(3S)-3-met...)
Affinity DataEC50:  970nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50255062({3-[4-((3R,5S)-3,5-Dimethyl-piperazin-1-ylmethyl)-...)
Affinity DataEC50:  51nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599721(CHEMBL5175905)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599722(CHEMBL5187975)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599723(CHEMBL5197045)
Affinity DataEC50:  55nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599724(CHEMBL5187776)
Affinity DataEC50:  240nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599725(CHEMBL5187928)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599726(CHEMBL5179543)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599727(CHEMBL5179463)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599728(CHEMBL5179060)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599729(CHEMBL5184722)
Affinity DataEC50:  4.60nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599730(CHEMBL5196819)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599731(CHEMBL5201797)
Affinity DataEC50:  5.30nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599732(CHEMBL5190786)
Affinity DataEC50:  7.5nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599733(CHEMBL5203126)
Affinity DataEC50:  5.60nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599734(CHEMBL5179573)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599735(CHEMBL5192584)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599736(CHEMBL5196982)
Affinity DataEC50:  4.70nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599737(CHEMBL5171964)
Affinity DataEC50:  4.30nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599738(CHEMBL5192530)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50599739(CHEMBL5181246)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR38 expressed in COS-7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  1.67E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50652792(CHEMBL3752910)
Affinity DataKd:  5.95E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50412520(CHEMBL14581)
Affinity DataEC50:  251nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50412521(CHEMBL465104)
Affinity DataEC50:  398nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50254851(3-cyclohexyl-1-((4'-(((3S,5R)-3,5-dimethylpiperazi...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50344942(CHEMBL532 | ERYTHROMYCIN | Erycette | Erymax | Ery...)
Affinity DataEC50:  50.1nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50254851(3-cyclohexyl-1-((4'-(((3S,5R)-3,5-dimethylpiperazi...)
Affinity DataEC50:  50.1nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50254852(N-[4'-((3R,5S)-3,5-Dimethyl-piperazin-1-ylmethyl)-...)
Affinity DataEC50:  79.4nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50254853(N-[4'-((3R,5S)-3,5-Dimethyl-piperazin-1-ylmethyl)-...)
Affinity DataEC50:  31.6nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50412522(CHEMBL465940)
Affinity DataEC50:  50.1nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50254892(2-(3-Chloro-phenyl)-N-[4'-((3R,5S)-3,5-dimethyl-pi...)
Affinity DataEC50:  79.4nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50412523(CHEMBL465271)
Affinity DataEC50:  3.16nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50254893(2-Benzenesulfonyl-N-[4'-((3R,5S)-3,5-dimethyl-pipe...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50412524(CHEMBL464247)
Affinity DataEC50:  19.9nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50412525(CHEMBL517934)
Affinity DataEC50:  251nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50254930(N-[4'-((3R,5S)-3,5-Dimethyl-piperazin-1-ylmethyl)-...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50254931(4'-((3R,5S)-3,5-Dimethyl-piperazin-1-ylmethyl)-bip...)
Affinity DataEC50:  7.94nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50254968([4'-((3R,5S)-3,5-Dimethyl-piperazin-1-ylmethyl)-bi...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50254969([4'-((3R,5S)-3,5-Dimethyl-piperazin-1-ylmethyl)-bi...)
Affinity DataEC50:  63.1nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50254970([4'-((3R,5S)-3,5-Dimethyl-piperazin-1-ylmethyl)-bi...)
Affinity DataEC50:  5.01nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50254971([4-(4-Chloro-phenylamino)-piperidin-1-yl]-[4'-((3R...)
Affinity DataEC50:  50.1nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50412526(CHEMBL518618)
Affinity DataEC50:  2.51nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50254999([4'-((3R,5S)-3,5-Dimethyl-piperazin-1-ylmethyl)-bi...)
Affinity DataEC50:  63.1nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50412527(CHEMBL473853)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50412528(CHEMBL481001)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50412529(CHEMBL481192)
Affinity DataEC50:  398nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50247157((3-(4-(((3R,5S)-3,5-dimethylpiperazin-1-yl)methyl)...)
Affinity DataEC50:  19.9nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50255029({1-[4-((3R,5S)-3,5-Dimethyl-piperazin-1-ylmethyl)-...)
Affinity DataEC50:  15.8nMAssay Description:Agonist activity at human recombinant motilin receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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