Report error Found 1076 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-3/beta-4'
Affinity DataEC50: 2.30E+4nMAssay Description:The functional properties of the ligands were determined by 86Rb+ efflux assays in cells expressing α3β4 and α4β2 nAChR subtypes....More data for this Ligand-Target Pair
Affinity DataEC50: 2.20E+4nMAssay Description:The functional properties of the ligands were determined by 86Rb+ efflux assays in cells expressing α3β4 and α4β2 nAChR subtypes....More data for this Ligand-Target Pair
Affinity DataEC50: 2.40E+4nMAssay Description:The functional properties of the ligands were determined by 86Rb+ efflux assays in cells expressing α3β4 and α4β2 nAChR subtypes....More data for this Ligand-Target Pair
Affinity DataEC50: 3.51E+3nMAssay Description:Agonist activity at rat alpha3beta4 nAChR expressed in HEK cells assessed as induction of Ca2+ fluxMore data for this Ligand-Target Pair
Affinity DataEC50: 2.54E+3nMAssay Description:Agonist activity at rat alpha3beta4 nAChR expressed in HEK cells assessed as induction of Ca2+ fluxMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Affinity DataEC50: 2.90E+3nMAssay Description:Agonist activity at human alpha3beta4 nAChR expressed in rat GH4C1 cells assessed as inward channel current amplitude at -70 mV holding potential by ...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human alpha3beta4 nAChR expressed in rat GH4C1 cells assessed as inward channel current amplitude at -70 mV holding potential by ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at rat alpha3beta4 nAChR expressed in HEK293 cells assessed as increase in calcium flux measured for 2 mins by Fluo-4-AM dye based F...More data for this Ligand-Target Pair
Affinity DataEC50: 41nMAssay Description:Agonist activity at rat alpha3beta4 nAChR by cell-based rubidium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70E+4nMAssay Description:Agonist activity at rat alpha3beta4 nAChR by cell-based rubidium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70E+4nMAssay Description:Agonist activity at rat alpha3beta4 nAChR by cell-based rubidium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 750nMAssay Description:Agonist activity at rat alpha3beta4 nAChR by cell-based rubidium flux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 570nMAssay Description:Agonist activity at rat alpha3beta4 nAChR by cell-based rubidium flux assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.300nMAssay Description:Tested for binding affinity against Nicotinic acetylcholine receptor alpha3-beta4More data for this Ligand-Target Pair
Affinity DataEC50: 2.09E+5nMAssay Description:Effective concentration against alpha3-beta4 Nicotinic acetylcholine receptor (nAChR)More data for this Ligand-Target Pair
Affinity DataEC50: 700nMAssay Description:Effective concentration against alpha3-beta4 nicotinic acetylcholine receptor expressed in IMR32 cellMore data for this Ligand-Target Pair
Affinity DataEC50: 510nMAssay Description:Effective concentration against alpha3-beta4 nicotinic acetylcholine receptor (nAChR) expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 510nMAssay Description:Effective concentration against alpha3-beta4 nicotinic acetylcholine receptor (nAChR) expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 6.30E+4nMAssay Description:Effective concentration against alpha3-beta4 nicotinic acetylcholine receptor (nAChR) expressed in IMR32 cell More data for this Ligand-Target Pair
Affinity DataEC50: 700nMAssay Description:Effective concentration against alpha3-beta4 nicotinic acetylcholine receptor (nAChR) expressed in IMR32 cell More data for this Ligand-Target Pair
Affinity DataEC50: 3.50E+4nMAssay Description:Agonist activity at rat alpha3beta4 nACHR expressed in human HEK293 cells by rubidium efflux assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+4nMAssay Description:Agonist activity at rat alpha3beta4 nACHR expressed in human HEK293 cells by rubidium efflux assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at alpha-3-beta-4 nAChR in KXalpha-3-beta-4R2 cells by rubidium efflux assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at alpha-3-beta-4 nAChR in KXalpha-3-beta-4R2 cells by rubidium efflux assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Affinity DataEC50: 1.82E+4nMAssay Description:Agonist activity at alpha-3-beta-4 nAChR in KXalpha-3-beta-4R2 cells by rubidium efflux assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at alpha-3-beta-4 nAChR in KXalpha-3-beta-4R2 cells by rubidium efflux assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at alpha-3-beta-4 nAChR in KXalpha-3-beta-4R2 cells by rubidium efflux assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Affinity DataEC50: 1.98E+4nMAssay Description:Agonist activity at alpha-3-beta-4 nAChR in KXalpha-3-beta-4R2 cells by rubidium efflux assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Affinity DataEC50: 28nMAssay Description:Agonist activity at alpha-3-beta-4 nAChR in KXalpha-3-beta-4R2 cells by rubidium efflux assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Affinity DataEC50: 2.08E+4nMAssay Description:Agonist activity at alpha-3-beta-4 nAChR in KXalpha-3-beta-4R2 cells by rubidium efflux assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Affinity DataEC50: 1.38E+4nMAssay Description:Agonist activity at alpha-3-beta-4 nAChR in KXalpha-3-beta-4R2 cells by rubidium efflux assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Affinity DataEC50: 2.64E+4nMAssay Description:Agonist activity at alpha-3-beta-4 nAChR in KXalpha-3-beta-4R2 cells by rubidium efflux assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Affinity DataEC50: 1.32E+5nMAssay Description:Inhibition of human alpha3beta4 nAChR assessed as increase in acetylcholine-induced normalized current at 2 uM (Rvb = 78.5 +/- 10 uM)More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Affinity DataEC50: 2.00E+3nMAssay Description:Agonist activity at human alpha3beta4 nAChR expressed in CHO cells assessed as calcium influx by calcium-4 based FLIPR analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Affinity DataEC50: 3.00E+3nMAssay Description:Agonist activity at human alpha3beta4 nAChR expressed in CHO cells assessed as calcium influx by calcium-4 based FLIPR analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Affinity DataEC50: 9.00E+3nMAssay Description:Agonist activity at human alpha3beta4 nAChR expressed in CHO cells assessed as calcium influx by calcium-4 based FLIPR analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human alpha3beta4 nAChR expressed in CHO cells assessed as calcium influx by calcium-4 based FLIPR analysisMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Istituto Di Chimica Biomolecolare
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human alpha3beta4 nAChR expressed in CHO cells assessed as calcium influx by calcium-4 based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 1.51E+3nMAssay Description:Agonist activity at rat neuronal acetylcholine receptor subunit alpha3beta4 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+6nMAssay Description:Agonist activity at rat neuronal acetylcholine receptor subunit alpha3beta4 expressed in HEK293 cells at 1 mM by FMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+3nMAssay Description:Agonist activity at rat neuronal acetylcholine receptor subunit alpha3beta4 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+5nMAssay Description:Agonist activity at rat neuronal acetylcholine receptor subunit alpha3beta4 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+5nMAssay Description:Agonist activity at rat neuronal acetylcholine receptor subunit alpha3beta4 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+5nMAssay Description:Agonist activity at rat neuronal acetylcholine receptor subunit alpha3beta4 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at rat neuronal acetylcholine receptor subunit alpha3beta4 expressed in HEK293 cells at 1 mM by FMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+6nMAssay Description:Agonist activity at rat neuronal acetylcholine receptor subunit alpha3beta4 expressed in HEK293 cells at 1 mM by FMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at rat neuronal acetylcholine receptor subunit alpha3beta4 expressed in HEK293 cells at 1 mM by FMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+6nMAssay Description:Agonist activity at rat neuronal acetylcholine receptor subunit alpha3beta4 expressed in HEK293 cells at 1 mM by FMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.24E+4nMAssay Description:Agonist activity at rat neuronal acetylcholine receptor subunit alpha3beta4 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+5nMAssay Description:Agonist activity at rat neuronal acetylcholine receptor subunit alpha3beta4 expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair





































