Compile Data Set for Download or QSAR
Report error Found 872 Enz. Inhib. hit(s) with Target = 'Neuropeptide Y receptor type 4'
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50240829(CHEMBL3559801)
Affinity DataEC50:  0.0300nMAssay Description:Positive allosteric modulation of human NY4 receptor expressed in African green monkey COS7 cells co-expressing delta6Galphaqi4-myr assessed as poten...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50240829(CHEMBL3559801)
Affinity DataEC50:  0.5nMAssay Description:Positive allosteric modulation of human NY4 receptor expressed in African green monkey COS7 cells co-expressing delta6Galphaqi4-myr assessed as poten...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50240829(CHEMBL3559801)
Affinity DataEC50:  4.5nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-tagged NY4 receptor expressed in HEK293 cells assessed as potentiation of pancreatic polypept...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50240829(CHEMBL3559801)
Affinity DataEC50:  443nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-tagged NY4 receptor expressed in HEK293 cells assessed as potentiation of neuropeptide Y-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50240829(CHEMBL3559801)
Affinity DataEC50:  0.0398nMAssay Description:Positive allosteric modulation of human NY4 receptor expressed in African green monkey COS7 cells co-expressing delta6Galphaqi4-myr assessed as poten...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50240829(CHEMBL3559801)
Affinity DataEC50:  0.398nMAssay Description:Positive allosteric modulation of human NY4 receptor expressed in African green monkey COS7 cells co-expressing delta6Galphaqi4-myr assessed as poten...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50240829(CHEMBL3559801)
Affinity DataEC50:  4nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-tagged NY4 receptor expressed in HEK293 cells assessed as potentiation of pancreatic polypept...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50240829(CHEMBL3559801)
Affinity DataEC50:  794nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-tagged NY4 receptor expressed in HEK293 cells assessed as potentiation of peptide YY-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50240829(CHEMBL3559801)
Affinity DataEC50:  5.10E+3nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-fused human NY4 receptor expressed in African green monkey COS7 cells co-expressing delta6Gal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50240829(CHEMBL3559801)
Affinity DataEC50:  0.400nMAssay Description:Positive allosteric modulation of human NY4 receptor expressed in African green monkey COS7 cells co-expressing delta6Galphaqi4-myr assessed as poten...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50240829(CHEMBL3559801)
Affinity DataEC50:  845nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-tagged NY4 receptor expressed in HEK293 cells assessed as potentiation of peptide YY-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50240829(CHEMBL3559801)
Affinity DataEC50:  0.501nMAssay Description:Positive allosteric modulation of human NY4 receptor expressed in African green monkey COS7 cells co-expressing delta6Galphaqi4-myr assessed as poten...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50240829(CHEMBL3559801)
Affinity DataEC50:  398nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-tagged NY4 receptor expressed in HEK293 cells assessed as potentiation of neuropeptide Y-indu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50240829(CHEMBL3559801)
Affinity DataEC50:  5.01E+3nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-fused human NY4 receptor expressed in African green monkey COS7 cells co-expressing delta6Gal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Rat)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50450993(CHEMBL4210786)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at rat neuropeptide Y4 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50466542(CHEMBL4290445)
Affinity DataEC50:  1.00E+4nMAssay Description:Displacement of [125I]-PYY(1 to 36 residues) from mouse Y4R expressed in HEK293 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466538(CHEMBL4284905)
Affinity DataEC50:  10nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466534(CHEMBL4288294)
Affinity DataEC50: <1.00E+3nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466524(CHEMBL4277676)
Affinity DataEC50: <1.00E+3nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466532(CHEMBL4281479)
Affinity DataEC50:  4nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50466532(CHEMBL4281479)
Affinity DataEC50:  790nMAssay Description:Displacement of [125I]-PYY(1 to 36 residues) from mouse Y4R expressed in HEK293 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466532(CHEMBL4281479)
Affinity DataEC50:  4nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50466532(CHEMBL4281479)
Affinity DataEC50:  794nMAssay Description:Displacement of [125I]-PYY(1 to 36 residues) from mouse Y4R expressed in HEK293 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466533(CHEMBL4292105)
Affinity DataEC50: >30nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50466533(CHEMBL4292105)
Affinity DataEC50: >1.00E+3nMAssay Description:Displacement of [125I]-PYY(1 to 36 residues) from mouse Y4R expressed in HEK293 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466529(CHEMBL4283257)
Affinity DataEC50: <1.00E+3nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50466529(CHEMBL4283257)
Affinity DataEC50: <1.00E+4nMAssay Description:Displacement of [125I]-PYY(1 to 36 residues) from mouse Y4R expressed in HEK293 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466538(CHEMBL4284905)
Affinity DataEC50:  10nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466535(CHEMBL4280392)
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466535(CHEMBL4280392)
Affinity DataEC50: <1.00E+3nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50466535(CHEMBL4280392)
Affinity DataEC50: <1.00E+4nMAssay Description:Displacement of [125I]-PYY(1 to 36 residues) from mouse Y4R expressed in HEK293 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466536(CHEMBL4279973)
Affinity DataEC50:  0.5nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466536(CHEMBL4279973)
Affinity DataEC50:  0.501nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466543(CHEMBL4276961)
Affinity DataEC50:  0.200nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466540(CHEMBL4287058)
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50466540(CHEMBL4287058)
Affinity DataEC50: >1.00E+4nMAssay Description:Displacement of [125I]-PYY(1 to 36 residues) from mouse Y4R expressed in HEK293 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466540(CHEMBL4287058)
Affinity DataEC50: <1.00E+3nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50466540(CHEMBL4287058)
Affinity DataEC50: <1.00E+4nMAssay Description:Displacement of [125I]-PYY(1 to 36 residues) from mouse Y4R expressed in HEK293 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466544(CHEMBL4294277)
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466544(CHEMBL4294277)
Affinity DataEC50: <1.00E+3nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466524(CHEMBL4277676)
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466525(CHEMBL4285633)
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466525(CHEMBL4285633)
Affinity DataEC50: <1.00E+3nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50466533(CHEMBL4292105)
Affinity DataEC50: <1.00E+3nMAssay Description:Displacement of [125I]-PYY(1 to 36 residues) from mouse Y4R expressed in HEK293 cell membranes after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466547(CHEMBL4278700)
Affinity DataEC50:  0.200nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466553(CHEMBL4279794)
Affinity DataEC50:  501nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466542(CHEMBL4290445)
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466542(CHEMBL4290445)
Affinity DataEC50: <1.00E+3nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466529(CHEMBL4283257)
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Leipzig University

Curated by ChEMBL
LigandPNGBDBM50466554(CHEMBL4286615)
Affinity DataEC50:  0.160nMAssay Description:Activation of human Y4R expressed in HEK293 cells assessed as inhibition of isoproterenol-induced increase in intracellular cAMP levels by calcium 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
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