Compile Data Set for Download or QSAR
Report error Found 565 Enz. Inhib. hit(s) with Target = 'Neuropeptides B/W receptor type 1'
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362418(CHEMBL1938418)
Affinity DataIC50: 0.180nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362419(CHEMBL1940544)
Affinity DataIC50: 0.200nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362420(CHEMBL1940540)
Affinity DataIC50: 0.330nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362417(CHEMBL1940545)
Affinity DataIC50: 0.420nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362409(CHEMBL1940543)
Affinity DataIC50: 0.430nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362417(CHEMBL1940545)
Affinity DataIC50: 0.660nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362414(CHEMBL1940537)
Affinity DataIC50: 0.690nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362419(CHEMBL1940544)
Affinity DataIC50: 0.860nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362412(CHEMBL1940539)
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362418(CHEMBL1938418)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362420(CHEMBL1940540)
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362415(CHEMBL1940536)
Affinity DataIC50: 1.90nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362411(CHEMBL1940541)
Affinity DataIC50: 2.20nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362413(CHEMBL1940538)
Affinity DataIC50: 2.40nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362410(CHEMBL1940542)
Affinity DataIC50: 2.60nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603459(CHEMBL5187335)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO cells measured by LANCE Ultra cAMP kit-based TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362437(CHEMBL1940367)
Affinity DataIC50: 2.80nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362412(CHEMBL1940539)
Affinity DataIC50: 3nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362430(CHEMBL1940526)
Affinity DataIC50: 3.10nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603429(CHEMBL5170622)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO cells measured by LANCE Ultra cAMP kit-based TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362409(CHEMBL1940543)
Affinity DataIC50: 3.90nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50362414(CHEMBL1940537)
Affinity DataIC50: 4.20nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362438(CHEMBL1940366)
Affinity DataIC50: 4.5nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362435(CHEMBL1940369)
Affinity DataIC50: 4.5nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362413(CHEMBL1940538)
Affinity DataIC50: 4.60nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603433(CHEMBL5204006)
Affinity DataEC50:  5.10nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO cells measured by LANCE Ultra cAMP kit-based TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603467(CHEMBL5197385)
Affinity DataEC50:  5.5nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO cells measured by LANCE Ultra cAMP kit-based TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362414(CHEMBL1940537)
Affinity DataIC50: 5.90nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50362412(CHEMBL1940539)
Affinity DataIC50: 5.90nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50362409(CHEMBL1940543)
Affinity DataIC50: 6nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50013388(CHEMBL350384 | BREMAZOCINE(-) | 6-Ethyl-3-(1-hydro...)
In Depth
Date in BDB:
12/21/2011
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603459(CHEMBL5187335)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603429(CHEMBL5170622)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362436(CHEMBL1940368)
Affinity DataIC50: 8.30nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362415(CHEMBL1940536)
Affinity DataIC50: 9.20nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603428(CHEMBL5194519)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603446(CHEMBL5178929)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50362412(CHEMBL1940539)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362432(CHEMBL1940372)
Affinity DataIC50: 11nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362410(CHEMBL1940542)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603430(CHEMBL5172042)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603431(CHEMBL5206425)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362411(CHEMBL1940541)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362440(CHEMBL1940364)
Affinity DataIC50: 14nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50603469(CHEMBL5177662)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human NPBWR1 expressed in CHO-RD-HGA16 cells measured by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362421(CHEMBL1940535)
Affinity DataIC50: 16nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362422(CHEMBL1940534)
Affinity DataIC50: 17nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Human)
Rti International

Curated by ChEMBL
LigandPNGBDBM50362410(CHEMBL1940542)
Affinity DataIC50: 18nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362436(CHEMBL1940368)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuropeptides B/W receptor type 1(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50362444(CHEMBL1940360)
Affinity DataIC50: 18nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
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