Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Neurotensin receptor type 1/2'
TargetNeurotensin receptor type 1/2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280251(UK-73093 | 4-Methyl-N-[2-(3-oxo-1-phenyl-1,3-dihyd...)
Affinity DataIC50: 5.50E+3nMAssay Description:Compound was evaluated for its ability to displace [3H]NT from the neurotensin receptor of bovine brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1/2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50086639(Arg-Pro-Tyr-Ile-Leu | (S)-2-{(2S,3S)-2-[(S)-2-{[(S...)
Affinity DataKi:  28nMAssay Description:Binding ability to compete with [125I]Tyr3-NT (0.15 nM) for human NT receptors cloned in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details Article
PubMed
TargetNeurotensin receptor type 1/2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50217111(CHEMBL1790704)
Affinity DataKi:  450nMAssay Description:Binding ability to compete with [125I]Tyr3-NT (0.15 nM) for human NT receptors cloned in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details Article
PubMed
TargetNeurotensin receptor type 1/2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50217110(CHEMBL1790701)
Affinity DataKi: >2.00E+3nMAssay Description:Binding ability to compete with [125I]Tyr3-NT (0.15 nM) for human NT receptors cloned in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details Article
PubMed