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Report error Found 114 Enz. Inhib. hit(s) with Target = 'Nucleosome-remodeling factor subunit BPTF'
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50539801(CHEMBL4648912 | US11840533, Compound 70)
Affinity DataKd: <1nMAssay Description:Binding affinity to human partial length FALZ (S2791 to H2911 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573197(CHEMBL4872300)
Affinity DataKd:  6.30nMAssay Description:Binding affinity to BPTF (unknown origin) by by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573200(CHEMBL4861491)
Affinity DataKd:  9.30nMAssay Description:Binding affinity to BPTF (unknown origin) by by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573840(CHEMBL4860578)
Affinity DataIC50: 16nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50571296(CHEMBL4873093)
Affinity DataIC50: 16nMAssay Description:Inhibition of BPTF in human HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573844(CHEMBL4873042)
Affinity DataIC50: 27nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573839(CHEMBL4870170)
Affinity DataIC50: 29nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50571296(CHEMBL4873093)
Affinity DataIC50: 30nMAssay Description:Inhibition of BPTF (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573837(CHEMBL4867072)
Affinity DataIC50: 33nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573200(CHEMBL4861491)
Affinity DataIC50: 36nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573838(CHEMBL4868713)
Affinity DataIC50: 37nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573201(CHEMBL4848701)
Affinity DataIC50: 56nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573845(CHEMBL4851594)
Affinity DataIC50: 59nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573849(CHEMBL4866637)
Affinity DataIC50: 59nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573848(CHEMBL4862619)
Affinity DataIC50: 64nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573197(CHEMBL4872300)
Affinity DataIC50: 67nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573201(CHEMBL4848701)
Affinity DataKd:  70nMAssay Description:Binding affinity to BPTF (unknown origin) by by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573852(CHEMBL4780673)
Affinity DataKd:  71nMAssay Description:Binding affinity to BPTF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50571296(CHEMBL4873093)
Affinity DataKd:  71nMAssay Description:Binding affinity to BPTF (unknown origin) by BLI assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50183448(CHEMBL3823478 | US11773085, Compound B2)
Affinity DataKd:  100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573841(CHEMBL4852588)
Affinity DataIC50: 114nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573844(CHEMBL4873042)
Affinity DataEC50:  120nMAssay Description:Displacement of Halo-tagged histone H4 from NanoLuc-tagged BPTF (unknown origin) expressed in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50514899(CHEMBL4461619)
Affinity DataKd:  120nMAssay Description:Binding affinity to BPTF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573846(CHEMBL4853486)
Affinity DataIC50: 145nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573850(CHEMBL4861221)
Affinity DataIC50: 157nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573198(CHEMBL4848138)
Affinity DataIC50: 170nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573203(CHEMBL4863631)
Affinity DataKd:  200nMAssay Description:Binding affinity to BPTF (unknown origin) by by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50514899(CHEMBL4461619)
Affinity DataKd:  200nMAssay Description:Binding affinity to BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50234940(CHEMBL4101756)
Affinity DataIC50: 220nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573192(CHEMBL4850516)
Affinity DataIC50: 250nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573842(CHEMBL4863921)
Affinity DataIC50: 288nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573190(CHEMBL4866748)
Affinity DataIC50: 290nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573191(CHEMBL4870218)
Affinity DataIC50: 310nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50584925(CHEMBL5079885)
Affinity DataKd: <316nMAssay Description:Binding affinity to human FALZ bromodomain by BROMOscan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50514899(CHEMBL4461619)
Affinity DataIC50: 350nMAssay Description:Inhibition of BPTF (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573193(CHEMBL4848082)
Affinity DataIC50: 370nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573203(CHEMBL4863631)
Affinity DataIC50: 380nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50571297(CHEMBL4846718)
Affinity DataKd:  428nMAssay Description:Binding affinity to BPTF (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573202(CHEMBL4877696)
Affinity DataIC50: 550nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573836(CHEMBL4861375)
Affinity DataIC50: 698nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573188(CHEMBL4850913)
Affinity DataIC50: 700nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573204(CHEMBL4863529)
Affinity DataIC50: 790nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573195(CHEMBL4855881)
Affinity DataIC50: 800nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50512964(CHEMBL4574669)
Affinity DataKd:  917nMAssay Description:Binding affinity to human N-terminal His-tagged FALZ by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50234924(CHEMBL4065579)
Affinity DataIC50: 950nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573196(CHEMBL4877118)
Affinity DataIC50: 970nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50157606(CHEMBL3785432)
Affinity DataIC50: 1.46E+3nMAssay Description:Alphascreen assay. Binding to FALZA (domain start/stop: S2791-H2911) by alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50234923(CHEMBL4069412)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50443230(CHEMBL3086885)
Affinity DataKi:  1.62E+3nMAssay Description:Displacement of fluorescein-labeled MS239 from recombinant human BPTF after 1 hr by fluorescence anisotropy assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50573835(CHEMBL4872350)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
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