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Report error Found 119 Enz. Inhib. hit(s) with Target = 'Peptidase'
TargetPeptidase(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50611988(CEFTAROLINE | Ceftaroline | T 91825 | T-91825)
Affinity DataIC50: 0.160nMAssay Description:Binding affinity to methicillin resistant Staphylococcus aureus PBP2aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPeptidase(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50611989(CHEMBL5271107)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [3H]-penicillin from Staphylococcus aureus PBP2aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031688(CHEMBL3360299)
Affinity DataIC50: 3nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031689(CHEMBL3360298)
Affinity DataIC50: 3nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031695(CHEMBL3360292)
Affinity DataIC50: 4nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031685(CHEMBL3360301)
Affinity DataIC50: 4nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031687(CHEMBL3360300)
Affinity DataIC50: 4nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031684(CHEMBL3360302)
Affinity DataIC50: 4nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031690(CHEMBL3360297)
Affinity DataIC50: 5nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031635(CHEMBL3359786)
Affinity DataIC50: 6nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031632(CHEMBL3359790)
Affinity DataIC50: 6nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031693(CHEMBL3360294)
Affinity DataIC50: 6nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031713(CHEMBL3360282)
Affinity DataIC50: 6nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM103023(US8541363, PVA-039)
Affinity DataIC50: 6.30nMAssay Description:The fluorogenic substrate used for measuring Der p 1 proteolytic activity was 2-aminobenzoylvalylalanylnorleucylseryl-(3-nitro)tyrosinyl aspartamide....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2013
Entry Details
Go to US Patent

TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031668(CHEMBL3359782)
Affinity DataIC50: 7nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM103022(US8541363, PVA-037)
Affinity DataIC50: 7.85nMAssay Description:The fluorogenic substrate used for measuring Der p 1 proteolytic activity was 2-aminobenzoylvalylalanylnorleucylseryl-(3-nitro)tyrosinyl aspartamide....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2013
Entry Details
Go to US Patent

TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031719(CHEMBL3359772)
Affinity DataIC50: 8nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031711(CHEMBL3360284)
Affinity DataIC50: 8nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031697(CHEMBL3360290)
Affinity DataIC50: 9nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031714(CHEMBL3360281)
Affinity DataIC50: 9nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031694(CHEMBL3360293)
Affinity DataIC50: 10nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031700(CHEMBL3360287)
Affinity DataIC50: 11nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031682(CHEMBL3359775)
Affinity DataIC50: 12nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031673(CHEMBL3359780)
Affinity DataIC50: 13nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM103021(US8541363, PVA-038)
Affinity DataIC50: 13nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM103021(US8541363, PVA-038)
Affinity DataIC50: 13.3nMAssay Description:The fluorogenic substrate used for measuring Der p 1 proteolytic activity was 2-aminobenzoylvalylalanylnorleucylseryl-(3-nitro)tyrosinyl aspartamide....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2013
Entry Details
Go to US Patent

TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031696(CHEMBL3360291)
Affinity DataIC50: 14nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM103020(US8541363, PVA-026)
Affinity DataIC50: 14nMAssay Description:The fluorogenic substrate used for measuring Der p 1 proteolytic activity was 2-aminobenzoylvalylalanylnorleucylseryl-(3-nitro)tyrosinyl aspartamide....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2013
Entry Details
Go to US Patent

TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM103020(US8541363, PVA-026)
Affinity DataIC50: 14nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031698(CHEMBL3360289)
Affinity DataIC50: 14nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031699(CHEMBL3360288)
Affinity DataIC50: 14nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50482776(CHEBI:70718 | Ceftaroline Fosamil | PPI-0903 | TAK...)
Affinity DataIC50: 14.6nMAssay Description:Binding affinity to against methicillin-, daptomycin-resistant, vancomycin-intermediate, beta-lactamase-positive Staphylococcus aureus 25 PBP2a by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031719(CHEMBL3359772)
Affinity DataIC50: 17nMAssay Description:Reversible inhibition of house dust mite Derp-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031692(CHEMBL3360295)
Affinity DataIC50: 17nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031633(CHEMBL3359789)
Affinity DataIC50: 17nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031710(CHEMBL3360285)
Affinity DataIC50: 17nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031683(CHEMBL3359773)
Affinity DataIC50: 18nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031670(CHEMBL3359781)
Affinity DataIC50: 18nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031691(CHEMBL3360296)
Affinity DataIC50: 20nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031678(CHEMBL3359779)
Affinity DataIC50: 20nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031715(CHEMBL3359791)
Affinity DataIC50: 24nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031681(CHEMBL3359777)
Affinity DataIC50: 42nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031712(CHEMBL3360283)
Affinity DataIC50: 47nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031634(CHEMBL3359787)
Affinity DataIC50: 55nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031722(CHEMBL3359770)
Affinity DataIC50: 65nMAssay Description:Reversible inhibition of house dust mite Derp-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031717(CHEMBL3359784)
Affinity DataIC50: 67nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031716(CHEMBL3359788)
Affinity DataIC50: 115nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase 1(European house dust mite)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031701(CHEMBL3360286)
Affinity DataIC50: 117nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetPeptidase, M28 family(Bacteroides forsythus)
Fraunhofer-Gesellschaft Zur Forderung Der Angewandten Forschung

US Patent
LigandPNGBDBM667852(US11958871, Example 17)
Affinity DataKi:  123nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2024
Entry Details
Go to US Patent

TargetPeptidase(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50569542(CHEMBL4847813)
Affinity DataKd:  129nMAssay Description:Binding affinity to Staphylococcus aureus PBP2a assessed as equilibrium dissociation constant by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
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