Compile Data Set for Download or QSAR
Report error Found 722 Enz. Inhib. hit(s) with Target = 'Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1'
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481978(CHEMBL1089622)
Affinity DataKd:  47nMAssay Description:Binding affinity to human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by isothermal titration colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481983(CHEMBL1089623)
Affinity DataKd:  48nMAssay Description:Binding affinity to human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by isothermal titration colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481980(CHEMBL1089627)
Affinity DataKd:  170nMAssay Description:Binding affinity to human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by isothermal titration colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481981(CHEMBL1089628)
Affinity DataKd:  980nMAssay Description:Binding affinity to human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by isothermal titration colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481984(CHEMBL1089626)
Affinity DataKd:  33nMAssay Description:Binding affinity to human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by isothermal titration colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481987(CHEMBL1089624)
Affinity DataKd:  920nMAssay Description:Binding affinity to human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by isothermal titration colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM34010(benzothiophene carboxamide, 18b)
Affinity DataKd:  72nMAssay Description:Binding affinity to full length Pin 1 (unknown origin) by isothermal titration calorimetry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50561320(CHEMBL4758488)
Affinity DataKd: >4.00E+3nMAssay Description:Binding affinity to full length Pin 1 (unknown origin) by isothermal titration calorimetry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKd:  800nMAssay Description:Binding affinity to Pin1 (unknown origin) preincubated for 2 hrs followed by UV irradiation for 15 mins by SDS-PAGE gel based photoaffinity labelling...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170728((R)-Phosphoric acid mono-[(1S,2S)-2-acetylamino-3-...)
Affinity DataKd:  1.40E+5nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170729(Phosphoric acid mono-[(S)-3-(2-carbamoyl-pyrrolidi...)
Affinity DataKd:  3.50E+4nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170731(Phosphoric acid mono-[(1R,2S)-2-acetylamino-3-((S)...)
Affinity DataKd:  8.00E+5nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170730(Phosphoric acid mono-[(1R,2S)-2-[4,4-bis-(4-hydrox...)
Affinity DataKd:  5.00E+3nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170732([1-((S)-2-Carbamoyl-pyrrolidine-1-carbonyl)-4-((S)...)
Affinity DataKd:  9.10E+5nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170733(Phosphoric acid mono-[(1S,3S)-3-(2-carbamoyl-pyrro...)
Affinity DataKd:  3.20E+4nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170734((S)-1-(3-Trifluoromethanesulfonylamino-propionyl)-...)
Affinity DataKd: >2.00E+6nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170735(Phosphoric acid mono-[(1S,3S)-3-(2-carbamoyl-pyrro...)
Affinity DataKd:  3.80E+4nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170736(Phosphoric acid mono-[(1R,2S)-2-acetylamino-3-((R)...)
Affinity DataKd:  4.00E+5nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170737([(S)-1-((S)-2-Carbamoyl-pyrrolidine-1-carbonyl)-2-...)
Affinity DataKd:  1.50E+4nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170742([(S)-1-((S)-2-Carbamoyl-2,5-dihydro-pyrrole-1-carb...)
Affinity DataKd:  6.60E+4nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170738(Phosphoric acid mono-[(1R,2S)-2-acetylamino-3-((S)...)
Affinity DataKd:  4.20E+5nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170739([3-((S)-2-Carbamoyl-pyrrolidin-1-yl)-3-oxo-propyl]...)
Affinity DataKd: >2.00E+6nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170741(5-((S)-2-Carbamoyl-pyrrolidin-1-yl)-5-oxo-pentanoi...)
Affinity DataKd: >2.00E+6nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170740(Phosphoric acid mono-[(1S,3S)-3-(2-carbamoyl-pyrro...)
Affinity DataKd:  4.80E+4nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170743((R)-Phosphoric acid mono-[(1S,2S)-2-acetylamino-3-...)
Affinity DataKd:  1.60E+5nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170744(Phosphoric acid mono-[(1R,2S)-2-acetylamino-3-((S)...)
Affinity DataKd:  3.60E+4nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170746(4-Acetylamino-5-((S)-2-carbamoyl-pyrrolidin-1-yl)-...)
Affinity DataKd: >2.00E+6nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170747(Phosphoric acid mono-[(1R,2S)-2-acetylamino-3-((S)...)
Affinity DataKd:  1.80E+4nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170745(Phosphoric acid mono-[(S)-3-(2-carbamoyl-2,5-dihyd...)
Affinity DataKd:  2.80E+4nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170749(Phosphoric acid mono-[(1S,3S)-3-(2-carbamoyl-pyrro...)
Affinity DataKd:  3.00E+4nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170750(4-((S)-2-Carbamoyl-pyrrolidin-1-yl)-4-oxo-butyric ...)
Affinity DataKd: >2.00E+6nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170751(Phosphoric acid mono-[(1R,2S)-2-acetylamino-3-((R)...)
Affinity DataKd:  1.00E+5nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170748([(S)-1-((S)-2-Carbamoyl-pyrrolidine-1-carbonyl)-5-...)
Affinity DataKd:  5.40E+5nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50170752(1-[(S)-3-(2-Hydroxy-3,4-dioxo-cyclobut-1-enylamino...)
Affinity DataKd: >2.00E+6nMAssay Description:Dissociation constant for human peptidyl-prolyl cis-trans isomerase NIMA-interacting 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50613630(BETAMETHASONE PHOSPHORIC ACID | CHEBI:68603 | Beta...)
Affinity DataKd:  2.20E+3nMAssay Description:Binding affinity to Pin1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKd:  800nMAssay Description:Binding affinity to Pin1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50618850(CHEMBL5423483)
Affinity DataKd:  72nMAssay Description:Inhibition of full length human Pin1 expressed in Escherichia coli assessed as dissociation constant by fluorescence anisotropy binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50618851(CHEMBL5408440)
Affinity DataKd:  620nMAssay Description:Inhibition of full length human Pin1 expressed in Escherichia coli assessed as dissociation constant by fluorescence anisotropy binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50648152(CHEMBL5598464)
Affinity DataKd:  430nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50648153(CHEMBL5596137)
Affinity DataKd:  230nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50648154(CHEMBL5590641)
Affinity DataKd: >5.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50648155(CHEMBL5598139)
Affinity DataKd:  920nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50648156(CHEMBL5596339)
Affinity DataKd:  1.22E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50648157(CHEMBL5598164)
Affinity DataKd:  2.03E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50648158(CHEMBL5597865)
Affinity DataKd:  120nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50648159(CHEMBL5590510)
Affinity DataKd:  2.72E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50648160(CHEMBL5590507)
Affinity DataKd:  370nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50648161(CHEMBL5597961)
Affinity DataKd:  780nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50648162(CHEMBL5596995)
Affinity DataKd:  3.05E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50648163(CHEMBL5597013)
Affinity DataKd:  3.10E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
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