Compile Data Set for Download or QSAR
Report error Found 1205 Enz. Inhib. hit(s) with Target = 'Protein kinase C delta type'
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31099(CHEMBL45741 | Flavopiridol | cid_24867231 | 2-(2-c...)
Affinity DataKd:  590nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2011
Entry Details
PCBioAssay
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM6866(1-Acyl-1H-[1,2,4]triazole-3,5-diamine Analogue 3b ...)
Affinity DataKd:  4.50E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2011
Entry Details
PCBioAssay
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM17055((9S)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydr...)
Affinity DataKd:  3.60nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2011
Entry Details
PCBioAssay
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31094(PKC-412 | cid_24202429)
Affinity DataKd:  320nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2011
Entry Details
PCBioAssay
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31096(CHEMBL290084 | Staurosporine | cid_451705 | US2024...)
Affinity DataKd:  1.5nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2011
Entry Details
PCBioAssay
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM92594(Phorbol ester (PDBU))
Affinity DataKd:  0.177nMpH: 7.4 T: 2°CAssay Description:[3H]PDBu binding to the C1 domains of MRCK alpha/beta and PKC alpha/delta was measured using the polyethylene glycol precipitation assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50092014(Butyric acid (1aS,1bS,4aS,7aS,8R,9S,9aR)-9-butyryl...)
Affinity DataKd:  0.330nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2013
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50258529(CHEMBL449158 | bryostatin 1)
Affinity DataKd:  0.260nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2013
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM102423(Bryostatin | Bryostatin 7)
Affinity DataKd:  0.210nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2013
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM239072(US9409931, 5)
Affinity DataEC50:  1.11E+3nMpH: 7.4Assay Description:On the day at experiment Human Protein Kinase C delta (PKCδ, Millipore cat#14-504) was diluted in 20 mM HEPES, 0.03% Triton X-100. Amount of enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2017
Entry Details
US Patent

TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM239070(US9409931, 6)
Affinity DataEC50:  80nMpH: 7.4Assay Description:On the day at experiment Human Protein Kinase C delta (PKCδ, Millipore cat#14-504) was diluted in 20 mM HEPES, 0.03% Triton X-100. Amount of enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2017
Entry Details
US Patent

TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM239071(US9409931, 7)
Affinity DataEC50:  154nMpH: 7.4Assay Description:On the day at experiment Human Protein Kinase C delta (PKCδ, Millipore cat#14-504) was diluted in 20 mM HEPES, 0.03% Triton X-100. Amount of enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2017
Entry Details
US Patent

TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM239069(US9409931, 8)
Affinity DataEC50:  7nMpH: 7.4Assay Description:On the day at experiment Human Protein Kinase C delta (PKCδ, Millipore cat#14-504) was diluted in 20 mM HEPES, 0.03% Triton X-100. Amount of enz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/24/2017
Entry Details
US Patent

TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50280749(CHEMBL4169454)
Affinity DataEC50:  8.03E+3nMAssay Description:Activation of PKCdelta (unknown origin) expressed in human LNCAP cells harboring GFP-tagged RasGRP1 assessed as phosphorylation at ser299 residues af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50280749(CHEMBL4169454)
Affinity DataEC50:  8.28E+3nMAssay Description:Activation of PKCdelta (unknown origin) expressed in human LNCAP cells harboring GFP-tagged RasGRP3 assessed as phosphorylation at ser299 residues af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50280749(CHEMBL4169454)
Affinity DataEC50:  1.69E+4nMAssay Description:Activation of PKCdelta (unknown origin) expressed in HEK293 cells harboring GFP-tagged RasGRP3 assessed as phosphorylation at ser299 residues after 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50280749(CHEMBL4169454)
Affinity DataEC50:  2.46E+4nMAssay Description:Activation of PKCdelta in human Ramos cells expressing RasGRP3 assessed as phosphorylation at ser299 residues after 30 mins by immunoblot methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50099066(phorbol 13-acetate 12-myristate | CHEMBL279115)
Affinity DataEC50:  290nMAssay Description:Activation of PKCdelta (unknown origin) expressed in HEK293 cells harboring GFP-tagged RasGRP3 assessed as phosphorylation at ser299 residues after 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50280749(CHEMBL4169454)
Affinity DataEC50:  1.26E+4nMAssay Description:Activation of PKCdelta (unknown origin) expressed in HEK293 cells harboring GFP-tagged RasGRP1 assessed as phosphorylation at ser299 residues after 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50493440(CHEMBL2430127)
Affinity DataEC50:  4.70nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50493441(CHEMBL2430122)
Affinity DataEC50:  2.90nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50493442(CHEMBL2430115)
Affinity DataEC50:  4.5nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50493443(CHEMBL2430141)
Affinity DataEC50:  5.30nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50493444(CHEMBL2430126)
Affinity DataEC50:  5.30nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50470108(AGN 204332 | Ingenol Mebutate | PEP-005 | PEP005 |...)
Affinity DataEC50:  4.10nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50493445(CHEMBL2430124)
Affinity DataEC50:  11nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50493446(CHEMBL2430142)
Affinity DataEC50:  5.20nMAssay Description:Activation of PKCdelta (unknown origin) using phosphatidylserine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50495188(CHEMBL3105106)
Affinity DataEC50:  8nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50470108(AGN 204332 | Ingenol Mebutate | PEP-005 | PEP005 |...)
Affinity DataEC50:  4.10nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50495189(CHEMBL3105094)
Affinity DataEC50:  3.30nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50495190(CHEMBL3105092)
Affinity DataEC50:  26nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50495191(CHEMBL2430121)
Affinity DataEC50:  6.10nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50495192(CHEMBL3105098)
Affinity DataEC50:  2.5nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50495193(CHEMBL3105103)
Affinity DataEC50:  156nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50495194(CHEMBL3105104)
Affinity DataEC50:  20nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50495195(CHEMBL3105026)
Affinity DataEC50:  988nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50495196(CHEMBL3105095)
Affinity DataEC50:  13nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50495197(CHEMBL3105027)
Affinity DataEC50:  3.70nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50495198(CHEMBL3105088)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50495199(CHEMBL3105102)
Affinity DataEC50:  11nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50495200(CHEMBL3105089)
Affinity DataEC50:  3.80nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50495201(CHEMBL3105096)
Affinity DataEC50:  4.20nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50495202(CHEMBL3105110)
Affinity DataEC50:  13nMAssay Description:Activation of PKCdelta (unknown origin) after 40 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50505541(CHEMBL4465866)
Affinity DataKd:  13nMAssay Description:Binding affinity to recombinant human full length N-terminal GST-tagged PRKCD expressed in baculovirus expression system using PKC peptide as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50505542(CHEMBL4576489)
Affinity DataKd:  3nMAssay Description:Binding affinity to recombinant human full length N-terminal GST-tagged PRKCD expressed in baculovirus expression system using PKC peptide as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKd:  273nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1a domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKd:  1nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKd:  0.530nMAssay Description:Binding affinity for protein kinase C Delta-C1B domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKd:  52nMAssay Description:Binding affinity for protein kinase C Delta-C1A domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50133236(Tetradecanedioic acid ((S)-5-hydroxymethyl-2-isopr...)
Affinity DataKd:  1nMAssay Description:Binding affinity for human Protein kinase C deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Displayed 1 to 50 (of 1205 total ) | Next | Last >>
Jump to: