Compile Data Set for Download or QSAR
Report error Found 461 Enz. Inhib. hit(s) with Target = 'Protein kinase C eta type'
TargetProtein kinase C eta type(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50064089(teleocidin B-4 | telocidinB-4 4-hydroxymethyl-7,10...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of [3H]- PDBu binding to peptide D of mouse skin Protein kinase C etaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391386(CHEMBL2148106)
Affinity DataKi:  0.110nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50493217(DEMETHOXYDEBROMOAPLYSIATOXIN)
Affinity DataKi:  0.180nMAssay Description:Displacement of [3H]PDBu from PKCeta C1B domain (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 0.251nMAssay Description:Inhibition of human PKCeta using ERMRPRKRQGSVRRRV as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]PDBu from PKCeta C1B domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50097750(Butyric acid (1aR,1bS,4aS,7aR,7bR,8R,9R,9aS)-9-but...)
Affinity DataKi:  0.350nMAssay Description:Displacement of 3[H]PDBu from Protein kinase C eta C1b domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50327943(Aplysiatoxin | CHEMBL1256416)
Affinity DataKi:  0.360nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKd:  0.450nMAssay Description:Binding affinity for protein kinase C eta-C1B domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKd:  0.450nMAssay Description:Binding affinity for Protein kinase C eta C1b domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKd:  0.450nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B peptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKd:  0.450nMAssay Description:Binding affinity to PKCeta-C1B domain peptide using [3H]-labeled compoundMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391388(CHEMBL2148108)
Affinity DataKi:  0.450nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM3153(CHEMBL52529 | 2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4...)
Affinity DataIC50: 0.600nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/25/2005
Entry Details Article

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM3153(CHEMBL52529 | 2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of human Protein Kinase C etaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM3153(CHEMBL52529 | 2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of Protein kinase C etaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM3183(2-({2,6-dihydroxy-4-[({2-[(4-hydroxybenzene)amido]...)
Affinity DataIC50: 0.600nMpH: 7.5 T: 2°CAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM3153(CHEMBL52529 | 2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4...)
Affinity DataIC50: 0.600nMAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2005
Entry Details Article

TargetProtein kinase C eta type(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of [3H]- PDBu binding to peptide D of mouse skin Protein kinase C etaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKd:  0.900nMAssay Description:Displacement of [3H]PDBu from protein kinase C eta C1b domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)
Affinity DataKi:  0.950nMAssay Description:Displacement of 3[H]PDBu from Protein kinase C eta C1b domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50393218(CHEMBL1996510)
Affinity DataIC50: 1nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50285250(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50: 1nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/24/2005
Entry Details Article

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM3153(CHEMBL52529 | 2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4...)
Affinity DataIC50: 1nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C eta isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM3153(CHEMBL52529 | 2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4...)
Affinity DataIC50: 1nMAssay Description:Inhibition of protein kinase C etaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM3153(CHEMBL52529 | 2-{[2,6-dihydroxy-4-({[(1R,2R)-2-[(4...)
Affinity DataIC50: 1nMAssay Description:Inhibition of Protein kinase C etaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human PKCeta using ERMRPRKRQGSVRRRV as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50393214(CHEMBL2151411)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50393228(CHEMBL2153750)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of PKCeta by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50285239(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human Protein Kinase C etaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50055672(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C eta isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50285240(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human Protein Kinase C etaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391897(CHEMBL2147537)
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human PKCeta assessed as [33P]-ATP incorporation into tridecapeptide substrate after 60 mins by scintillation proximity ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM25013(4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3S...)
Affinity DataKd:  2.40nMAssay Description:Binding constant for PRKCH kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM185384(US9156845, 28)
Affinity DataKi:  2.40nMAssay Description:Inhibition of full length human recombinant PKCeta expessed in baculovirus infected insect cells using 5-FAM-RFARKGSLRQKNV-COOH peptide as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM130909(US8822500, Stauro- sporine | US9920060, Staurospor...)
Affinity DataIC50: 2.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM3199(2-{[2,6-dihydroxy-4-({[(1R,2S)-2-[(4-hydroxyphenyl...)
Affinity DataIC50: 3nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50055677(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50: 3nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C eta isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM3186(2-[(4-{[(2S)-2-benzenesulfonamido-3-(4-hydroxyphen...)
Affinity DataIC50: 3nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM3149(Acyclic Balanol Analog (-)-1 | 2-{[2,6-dihydroxy-4...)
Affinity DataIC50: 3nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/31/2005
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50285242(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human Protein Kinase C etaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50285241(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human Protein Kinase C etaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM3199(2-{[2,6-dihydroxy-4-({[(1R,2S)-2-[(4-hydroxyphenyl...)
Affinity DataIC50: 3nMAssay Description:Inhibition of protein kinase C etaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50055668(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50: 3nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C eta isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM3149(Acyclic Balanol Analog (-)-1 | 2-{[2,6-dihydroxy-4...)
Affinity DataIC50: 3nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C eta isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM3149(Acyclic Balanol Analog (-)-1 | 2-{[2,6-dihydroxy-4...)
Affinity DataIC50: 3nMAssay Description:Inhibition of Protein kinase C etaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50285087((R)-2-{2,6-Dihydroxy-4-[(3R,4R)-4-(4-hydroxy-benzo...)
Affinity DataIC50: 3nMAssay Description:Inhibition of Protein kinase C etaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM3149(Acyclic Balanol Analog (-)-1 | 2-{[2,6-dihydroxy-4...)
Affinity DataIC50: 3nMAssay Description:Inhibition of Protein kinase C etaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50366386(CHEMBL1794808)
Affinity DataIC50: 3nMAssay Description:Inhibition of human Protein Kinase C etaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM3199(2-{[2,6-dihydroxy-4-({[(1R,2S)-2-[(4-hydroxyphenyl...)
Affinity DataIC50: 3nMAssay Description:Inhibition of protein kinase C etaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50055684(4-(2-Carboxy-6-hydroxy-benzoyl)-3,5-dihydroxy-benz...)
Affinity DataIC50: 3nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C eta isozymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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