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Report error Found 293 Enz. Inhib. hit(s) with Target = 'Regulator of G-protein signaling 4'
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384752(CHEMBL2037351)
Affinity DataIC50: 5.40nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384751(CHEMBL2037350)
Affinity DataIC50: 7.20nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384755(CHEMBL2037352)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384777(CHEMBL2037229)
Affinity DataIC50: 11nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384754(CHEMBL2037234)
Affinity DataIC50: 13nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM7779(4-butyl-2-ethyl-1,2,4-thiadiazolidine-3,5-dione | ...)
Affinity DataIC50: 14nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384767(CHEMBL2037365)
Affinity DataIC50: 14nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384776(CHEMBL2037228)
Affinity DataIC50: 14nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384743(CHEMBL2037235)
Affinity DataIC50: 14nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384757(CHEMBL2037354)
Affinity DataIC50: 15nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384775(CHEMBL2037227)
Affinity DataIC50: 16nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384760(CHEMBL2035006)
Affinity DataIC50: 16nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384756(CHEMBL2037353)
Affinity DataIC50: 17nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384761(CHEMBL2037358)
Affinity DataIC50: 19nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384764(CHEMBL2037362)
Affinity DataIC50: 20nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM47740(cid_12005086 | 1-ethyl-4-(4-fluoranyl-2-nitro-5-py...)
Affinity DataEC50:  20nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM47800(MLS000736409 | N'-[(E)-(2-fluorophenyl)methyli...)
Affinity DataEC50:  20nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM47728((2E)-3-(2-chloroanilino)-2-(3,3-dimethyl-2,4-dihyd...)
Affinity DataEC50:  20nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384739(CHEMBL2037357)
Affinity DataIC50: 22nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384762(CHEMBL2037359)
Affinity DataIC50: 22nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384746(CHEMBL2037238)
Affinity DataIC50: 24nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384763(CHEMBL2037360)
Affinity DataIC50: 24nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384744(CHEMBL2037236)
Affinity DataIC50: 24nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384768(CHEMBL2037366)
Affinity DataIC50: 26nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384753(CHEMBL2037361)
Affinity DataIC50: 28nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384770(CHEMBL2037368)
Affinity DataIC50: 29nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384745(CHEMBL2037237)
Affinity DataIC50: 29nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384765(CHEMBL2037363)
Affinity DataIC50: 30nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384774(CHEMBL1917204 | US20230414581, Compound 6)
Affinity DataIC50: 30nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384774(CHEMBL1917204 | US20230414581, Compound 6)
Affinity DataIC50: 30nMAssay Description:FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2015
Entry Details
Go to US Patent

TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384750(CHEMBL2037349)
Affinity DataIC50: 33nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384759(CHEMBL2037356)
Affinity DataIC50: 34nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384778(CHEMBL2037230)
Affinity DataIC50: 36nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384749(CHEMBL2037348)
Affinity DataIC50: 38nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384769(CHEMBL2037367)
Affinity DataIC50: 39nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384742(CHEMBL2037233)
Affinity DataIC50: 52nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384766(CHEMBL2037364)
Affinity DataIC50: 54nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384771(CHEMBL2037369)
Affinity DataIC50: 54nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384748(CHEMBL2037347)
Affinity DataIC50: 57nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM47709(9-thiophen-2-yl-5,6,7,9-tetrahydro-1H-[1,2,4]triaz...)
Affinity DataEC50:  60nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2011
Entry Details
PCBioAssay
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384740(CHEMBL2037231)
Affinity DataIC50: 79nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384747(CHEMBL2037346)
Affinity DataIC50: 89nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM46667(2-phenyl-1,2-benzothiazol-3-one (1) | cid_164981 |...)
Affinity DataKi:  110nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2011
Entry Details
PCBioAssay
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384741(CHEMBL2037232)
Affinity DataIC50: 121nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM46667(2-phenyl-1,2-benzothiazol-3-one (1) | cid_164981 |...)
Affinity DataEC50:  135nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2011
Entry Details
PCBioAssay
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM40728(N''-[(Z)-(3-hydroxy-4-oxo-1-cyclohexa-2,5-dienylid...)
Affinity DataKi:  140nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2011
Entry Details
PCBioAssay
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM40728(N''-[(Z)-(3-hydroxy-4-oxo-1-cyclohexa-2,5-dienylid...)
Affinity DataEC50:  164nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2011
Entry Details
PCBioAssay
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50384758(CHEMBL2037355)
Affinity DataIC50: 176nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM43363(MLS000550549 | 2,5-dichloro-3-(1-piperidinyl)-6-[2...)
Affinity DataKi:  230nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2011
Entry Details
PCBioAssay
TargetRegulator of G-protein signaling 4(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM47719(MLS000539990 | 4-chloro-N-(4-chloro-2-methylphenyl...)
Affinity DataKi:  260nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH R21NS057014 HTS to identify small molecule regulators of RGS family protein interaction...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2011
Entry Details
PCBioAssay
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