Report error Found 640 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor RXR-beta'
Affinity DataEC50: 770nMAssay Description:Agonist activity at RXRbeta (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 24nMAssay Description:Agonist activity at RXRbeta (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 2.40E+3nMAssay Description:Agonist activity at RXRbeta (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 2.71E+4nMAssay Description:Transactivation of human Gal4-fused RXRbeta LBD expressed in HEK293T cells after 12 to 14 hrs by dual-glo luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.20E+3nMAssay Description:Transactivation of human Gal4-fused RXRbeta LBD expressed in HEK293T cells after 12 to 14 hrs by dual-glo luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.60E+3nMAssay Description:Transactivation of human Gal4-fused RXRbeta LBD expressed in HEK293T cells after 12 to 14 hrs by dual-glo luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.50E+3nMAssay Description:Transactivation of human Gal4-fused RXRbeta LBD expressed in HEK293T cells after 12 to 14 hrs by dual-glo luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.39E+4nMAssay Description:Transactivation of human Gal4-fused RXRbeta LBD expressed in HEK293T cells after 12 to 14 hrs by dual-glo luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60E+4nMAssay Description:Transactivation of human Gal4-fused RXRbeta LBD expressed in HEK293T cells after 12 to 14 hrs by dual-glo luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+4nMAssay Description:Transactivation of human Gal4-fused RXRbeta LBD expressed in HEK293T cells after 12 to 14 hrs by dual-glo luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.20E+4nMAssay Description:Transactivation of human Gal4-fused RXRbeta LBD expressed in HEK293T cells after 12 to 14 hrs by dual-glo luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.20E+4nMAssay Description:Transactivation of human Gal4-fused RXRbeta LBD expressed in HEK293T cells after 12 to 14 hrs by dual-glo luciferase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.20E+3nMAssay Description:Transactivation of human Gal4-fused RXRbeta LBD expressed in HEK293T cells after 12 to 14 hrs by dual-glo luciferase assayMore data for this Ligand-Target Pair
Affinity DataKd: 3nMAssay Description:Binding affinity to Retinoic acid receptor RXR-beta was determined in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataEC50: 67nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-beta was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-beta was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataKd: 853nMAssay Description:Binding affinity to Retinoic acid receptor RXR-beta was determined in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataEC50: 310nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-beta was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to Retinoic acid receptor RXR-beta was determined in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataEC50: 280nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-beta was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to Retinoic acid receptor RXR-beta was determined in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to Retinoic acid receptor RXR-beta was determined in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-beta was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to Retinoic acid receptor RXR-beta was determined in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataEC50: 213nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-beta was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataEC50: 130nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-beta was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataKd: 61nMAssay Description:Binding affinity to Retinoic acid receptor RXR-beta was determined in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataKd: 770nMAssay Description:Binding affinity to Retinoic acid receptor RXR-beta was determined in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+3nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-beta was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataKd: 70nMAssay Description:Binding affinity to Retinoic acid receptor RXR-beta was determined in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataKd: 160nMAssay Description:Binding affinity to Retinoic acid receptor RXR-beta was determined in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+3nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-beta was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataEC50: 2.40E+3nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-beta was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataKd: 150nMAssay Description:Binding affinity to Retinoic acid receptor RXR-beta was determined in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-beta was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataEC50: 770nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-beta was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to Retinoic acid receptor RXR-beta was determined in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataKd: 291nMAssay Description:Binding affinity to Retinoic acid receptor RXR-beta was determined in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataKd: 190nMAssay Description:Binding affinity to Retinoic acid receptor RXR-beta was determined in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-beta was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-beta was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+3nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-beta was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataKd: 191nMAssay Description:Binding affinity to Retinoic acid receptor RXR-beta was determined in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataEC50: 9nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-beta was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataKd: 21nMAssay Description:Binding affinity to Retinoic acid receptor RXR-beta was determined in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:Effective concentrations against Retinoic acid receptor RXR-betaMore data for this Ligand-Target Pair
Affinity DataEC50: 360nMAssay Description:Effective concentrations against Retinoic acid receptor RXR-betaMore data for this Ligand-Target Pair
Affinity DataEC50: 33nMAssay Description:Effective concentrations against Retinoic acid receptor RXR-betaMore data for this Ligand-Target Pair
Affinity DataEC50: 3.20E+3nMAssay Description:Effective concentrations against Retinoic acid receptor RXR-betaMore data for this Ligand-Target Pair
Affinity DataEC50: 2.60nMAssay Description:Effective concentrations against Retinoic acid receptor RXR-betaMore data for this Ligand-Target Pair


3D Structure (crystal)


























