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Report error Found 1450 Enz. Inhib. hit(s) with Target = 'Somatostatin receptor type 1'
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50473329(CHEMBL311789)
Affinity DataKd:  1.32E+4nMAssay Description:Binding assay at human somatostatin receptor 1 (hsst1) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKd:  0.832nMAssay Description:Binding assay at human somatostatin receptor 1 (hsst1) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50473330(CHEMBL309948)
Affinity DataKd: <1.00E+5nMAssay Description:Binding assay at human somatostatin receptor 1 (hsst1) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50473331(CHEMBL420948)
Affinity DataKd: <1.00E+5nMAssay Description:Binding assay at human somatostatin receptor 1 (hsst1) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50192018(CHEMBL3350037)
Affinity DataKd:  389nMAssay Description:Binding assay at human somatostatin receptor 1 (hsst1) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50065451(2-Amino-N-{4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-(...)
Affinity DataKd:  3.55E+3nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst1) expressed in hSF6 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50065452(2-Amino-N-{4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-(...)
Affinity DataKd:  1.32E+4nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst1) expressed in hSF6 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50065450(2-Amino-3-phenyl-N-{4-[(2S,5S,8S,14S,17R)-8,10,14-...)
Affinity DataKd:  7.08E+3nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst1) expressed in hSF6 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50065453(CHEMBL421362 | L-361,301 | L-363,301 | L-363301 | ...)
Affinity DataKd:  4.57E+3nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst1) expressed in hSF6 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50537061(CHEMBL4527856)
Affinity DataKd:  310nMAssay Description:Displacement of [125I]somatostatin from human SSTR1 expressed in CHO-K1 cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50537072(CHEMBL440072)
Affinity DataKd:  0.290nMAssay Description:Displacement of [125I]somatostatin from human SSTR1 expressed in CHO-K1 cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098602(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098610(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  1.26E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098612(10-(4-Amino-butyl)-16-benzyl-7-(1-hydroxy-ethyl)-1...)
Affinity DataKd:  316nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098617(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  611nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098616(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  867nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098604(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  862nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098609(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098618(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098613(10-(4-Amino-butyl)-16-benzyl-7-(1-hydroxy-ethyl)-1...)
Affinity DataKd:  811nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098607(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  956nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098611(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098619(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  761nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098603(10-(4-Amino-butyl)-19-[(2-amino-3-phenyl-propionyl...)
Affinity DataKd:  378nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098606(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  653nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098615(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  1.20E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098614(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  622nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098605(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098608(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50546560(CHEMBL4778342)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human SST1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592194(CHEMBL5195355)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human SST1More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592196(CHEMBL5174433)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human SST1More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592194(CHEMBL5195355)
Affinity DataEC50: <1.00E+3nMAssay Description:Agonist activity at human SST1More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592196(CHEMBL5174433)
Affinity DataEC50: <1.00E+3nMAssay Description:Agonist activity at human SST1More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50294254((4R,7S,10S,13R,16S,19R)-19-((R)-2-amino-3-(4-hydro...)
Affinity DataEC50:  0.370nMAssay Description:Agonist activity at human sst1 receptor expressed in Chinese hamster CCL39 cells by luciferase reporter gene assay relative to somatostatin-14More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50294252((4R,7S,10S,13R,16S,19R)-19-amino-N-((2S,3R)-1-amin...)
Affinity DataEC50:  3.90nMAssay Description:Agonist activity at human sst1 receptor expressed in Chinese hamster CCL39 cells by luciferase reporter gene assay relative to somatostatin-14More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50294231((4R,7S,10S,13S,16S,19S,22R,25S,28S,31S,34R)-22-((1...)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human sst1 receptor expressed in Chinese hamster CCL39 cells by luciferase reporter gene assay relative to somatostatin-14More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50294255((4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-31...)
Affinity DataEC50:  0.930nMAssay Description:Agonist activity at human sst1 receptor expressed in Chinese hamster CCL39 cells by luciferase reporter gene assay relative to somatostatin-14More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423296(CHEMBL248716)
Affinity DataKd:  4.60nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423297(Obelin | CHEMBL251541)
Affinity DataKd:  0.708nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423298(CHEMBL251334)
Affinity DataKd:  17nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423299(CHEMBL401290)
Affinity DataKd:  0.214nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423300(CHEMBL401091)
Affinity DataKd:  16nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423302(CHEMBL248715)
Affinity DataKd:  1.20nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423305(CHEMBL251335)
Affinity DataKd:  158nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423306(CHEMBL249112)
Affinity DataKd:  1.32E+3nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423307(CHEMBL399464)
Affinity DataKd:  1.20nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423294(CHEMBL248908)
Affinity DataKd:  0.832nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423309(CHEMBL399843)
Affinity DataKd:  1.60nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Rat)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423310(CHEMBL251543)
Affinity DataKd:  19nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
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