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Report error Found 1887 Enz. Inhib. hit(s) with Target = 'Somatostatin receptor type 5'
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50192018(CHEMBL3350037)
Affinity DataKd:  49nMAssay Description:Binding assay at human somatostatin receptor 5 (hsst5) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50473329(CHEMBL311789)
Affinity DataKd: <1.00E+4nMAssay Description:Binding assay at human somatostatin receptor 5 (hsst5) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50473330(CHEMBL309948)
Affinity DataKd: <1.00E+5nMAssay Description:Binding assay at human somatostatin receptor 5 (hsst5) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKd:  0.977nMAssay Description:Binding assay at human somatostatin receptor 5 (hsst5) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50473331(CHEMBL420948)
Affinity DataKd: <1.00E+5nMAssay Description:Binding assay at human somatostatin receptor 5 (hsst5) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50065450(2-Amino-3-phenyl-N-{4-[(2S,5S,8S,14S,17R)-8,10,14-...)
Affinity DataKd:  69nMAssay Description:In vitro inhibition of radioligand binding to human Somatostatin receptor type 5 expressed in CCL-39 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50065451(2-Amino-N-{4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-(...)
Affinity DataKd:  407nMAssay Description:In vitro inhibition of radioligand binding to human Somatostatin receptor type 5 expressed in CCL-39 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50065453(CHEMBL421362 | L-361,301 | L-363,301 | L-363301 | ...)
Affinity DataKd:  7.60nMAssay Description:In vitro inhibition of radioligand binding to human Somatostatin receptor type 5 expressed in CCL-39 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50065452(2-Amino-N-{4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-(...)
Affinity DataKd:  6.17nMAssay Description:In vitro inhibition of radioligand binding to human Somatostatin receptor type 5 expressed in CCL-39 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50537072(CHEMBL440072)
Affinity DataKd:  0.320nMAssay Description:Displacement of [125I]somatostatin from human SSTR5 expressed in CHO-K1 cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50537061(CHEMBL4527856)
Affinity DataKd:  9.60nMAssay Description:Displacement of [125I]somatostatin from human SSTR5 expressed in CHO-K1 cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098604(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  114nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098607(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  629nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098617(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  71.8nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098608(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  83.2nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098616(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  8.41nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098614(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  28.4nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098619(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  8.35nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098613(10-(4-Amino-butyl)-16-benzyl-7-(1-hydroxy-ethyl)-1...)
Affinity DataKd:  27nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098618(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  33.0nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098612(10-(4-Amino-butyl)-16-benzyl-7-(1-hydroxy-ethyl)-1...)
Affinity DataKd:  4.89nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098611(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  50.4nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098609(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  313nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098610(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  16.9nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098602(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098606(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  95.0nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098605(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  92.8nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098615(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  0.610nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50098603(10-(4-Amino-butyl)-19-[(2-amino-3-phenyl-propionyl...)
Affinity DataKd:  23.7nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50546560(CHEMBL4778342)
Affinity DataEC50: <1.00E+3nMAssay Description:Agonist activity at human SST5More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592167(CHEMBL5182561)
Affinity DataEC50:  5.60nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592168(CHEMBL5181646)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592169(CHEMBL5193208)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592170(CHEMBL5180721)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592171(CHEMBL5190580)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592172(CHEMBL5200958)
Affinity DataEC50:  400nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592173(CHEMBL5195986)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592174(CHEMBL5189678)
Affinity DataEC50:  6.10nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592175(CHEMBL5188855)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592176(CHEMBL5188516)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592177(CHEMBL5200338)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592178(CHEMBL5170249)
Affinity DataEC50:  0.360nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592179(CHEMBL5182636)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592180(CHEMBL5184298)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592181(CHEMBL5178891)
Affinity DataEC50:  0.0770nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592182(CHEMBL5180885)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592183(CHEMBL5192315)
Affinity DataEC50:  0.270nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592184(CHEMBL5186952)
Affinity DataEC50:  0.320nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592185(CHEMBL5169724)
Affinity DataEC50:  0.0880nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetSomatostatin receptor type 5(Human)
Eth Zurich

Curated by ChEMBL
LigandPNGBDBM50592186(CHEMBL5177695)
Affinity DataEC50:  5.40nMAssay Description:Agonist activity at human SST5 expressed in CHO-K1 cells assessed as reduction in NKH477-induced intracellular cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
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