Report error Found 95 Enz. Inhib. hit(s) with Target = 'Threonine--tRNA ligase'
Affinity DataKd: 49nMAssay Description:Inhibition of human cytosolic ThrRS assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKd: 126nMAssay Description:Inhibition of human cytosolic ThrRS assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKd: 115nMAssay Description:Inhibition of human cytosolic ThrRS assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKd: 37nMAssay Description:Binding affinity to full length recombinant salmonella enterica threonyl-tRNA synthetase assessed as dissociation constant in presence of tRNA Leucin...More data for this Ligand-Target Pair
Affinity DataKd: 166nMAssay Description:Binding affinity to full length recombinant salmonella enterica threonyl-tRNA synthetase assessed as dissociation constant in presence of tRNA Threon...More data for this Ligand-Target Pair
Affinity DataKd: 44nMAssay Description:Binding affinity to full length recombinant salmonella enterica threonyl-tRNA synthetase assessed as dissociation constant in presence of glycine by ...More data for this Ligand-Target Pair
Affinity DataKd: 290nMAssay Description:Binding affinity to full length recombinant salmonella enterica threonyl-tRNA synthetase assessed as dissociation constant in presence of L-threonine...More data for this Ligand-Target Pair
Affinity DataKd: 75nMAssay Description:Binding affinity to full length recombinant salmonella enterica threonyl-tRNA synthetase assessed as dissociation constant in presence of ATP by isot...More data for this Ligand-Target Pair
Affinity DataKd: 35nMAssay Description:Binding affinity to full length recombinant salmonella enterica threonyl-tRNA synthetase assessed as dissociation constant by isothermal titration ca...More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against cognate Staphylococcus aureus threonyl tRNA synthetaseMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
Targetthreonine--tRNA ligase(Plasmodium falciparum (isolate 3D7))
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibition of Plasmodium falciparum Threonyl tRNA synthetaseMore data for this Ligand-Target Pair
Targetthreonine--tRNA ligase(Plasmodium falciparum (isolate 3D7))
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of Plasmodium falciparum Threonyl tRNA synthetaseMore data for this Ligand-Target Pair
Targetthreonine--tRNA ligase(Plasmodium falciparum (isolate 3D7))
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of 6xHis-tag recombinant Plasmodium falciparum threonyl tRNA synthetase expressed in Escherichia using L-threonine and total tRNA by lumin...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 103nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
Targetthreonine--tRNA ligase(Plasmodium falciparum (isolate 3D7))
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of Plasmodium falciparum Threonyl tRNA synthetaseMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
Affinity DataIC50: 194nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
Targetthreonine--tRNA ligase(Plasmodium falciparum (isolate 3D7))
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Inhibition of Plasmodium falciparum Threonyl tRNA synthetaseMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 480nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
Affinity DataIC50: 520nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
Affinity DataIC50: 550nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
Affinity DataIC50: 580nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
Targetthreonine--tRNA ligase(Plasmodium falciparum (isolate 3D7))
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of 6xHis-tag recombinant Plasmodium falciparum threonyl tRNA synthetase expressed in Escherichia using L-threonine and total tRNA by lumin...More data for this Ligand-Target Pair
Ligand InfoSimilars
Targetthreonine--tRNA ligase(Plasmodium falciparum (isolate 3D7))
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of 6xHis-tag recombinant Plasmodium falciparum threonyl tRNA synthetase expressed in Escherichia using L-threonine and total tRNA by lumin...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
Affinity DataIC50: 1.86E+3nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
Affinity DataIC50: 2.99E+3nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
Affinity DataIC50: 3.29E+3nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
Affinity DataIC50: 3.71E+3nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
Affinity DataIC50: 5.07E+3nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
Affinity DataIC50: 5.68E+3nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
Affinity DataIC50: 6.63E+3nMAssay Description:Inhibition of recombinant salmonella enterica threonyl-tRNA synthetase assessed as reduction in enzyme activity incubated for 20 min by Kinase Glo lu...More data for this Ligand-Target Pair
TargetThreonine--tRNA ligase(Soybean stem and root rot agent)
Northeast Agricultural University
Curated by ChEMBL
Northeast Agricultural University
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of C-terminal His6-tagged Phytophthora sojae race 1 recombinant ThrRS expressed in Escherichia coli BL21 (Codonplus DE3) assessed as reduc...More data for this Ligand-Target Pair
Targetthreonine--tRNA ligase(Plasmodium falciparum (isolate 3D7))
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of 6xHis-tag recombinant Plasmodium falciparum threonyl tRNA synthetase expressed in Escherichia using L-threonine and total tRNA by lumin...More data for this Ligand-Target Pair
Ligand InfoSimilars
Targetthreonine--tRNA ligase(Plasmodium falciparum (isolate 3D7))
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of Plasmodium falciparum Threonyl tRNA synthetaseMore data for this Ligand-Target Pair
Ligand InfoSimilars
Targetthreonine--tRNA ligase(Plasmodium falciparum (isolate 3D7))
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of 6xHis-tag recombinant Plasmodium falciparum threonyl tRNA synthetase expressed in Escherichia using L-threonine and total tRNA by lumin...More data for this Ligand-Target Pair
Ligand InfoSimilars
Targetthreonine--tRNA ligase(Plasmodium falciparum (isolate 3D7))
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibition of 6xHis-tag recombinant Plasmodium falciparum threonyl tRNA synthetase expressed in Escherichia using L-threonine and total tRNA by lumin...More data for this Ligand-Target Pair
Ligand InfoSimilars
Targetthreonine--tRNA ligase(Plasmodium falciparum (isolate 3D7))
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibition of 6xHis-tag recombinant Plasmodium falciparum threonyl tRNA synthetase expressed in Escherichia using L-threonine and total tRNA by lumin...More data for this Ligand-Target Pair
Ligand InfoSimilars
Targetthreonine--tRNA ligase(Plasmodium falciparum (isolate 3D7))
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Latvian Institute of Organic Synthesis
Curated by ChEMBL
Affinity DataIC50: 7.10E+4nMAssay Description:Inhibition of 6xHis-tag recombinant Plasmodium falciparum threonyl tRNA synthetase expressed in Escherichia using L-threonine and total tRNA by lumin...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 0.700nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair


































3D Structure (crystal)