Compile Data Set for Download or QSAR
Report error Found 139 Enz. Inhib. hit(s) with Target = 'Type 1 fimbrin D-mannose specific adhesin'
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50507926(CHEMBL4530691)
Affinity DataKd:  89nMAssay Description:Binding affinity to Escherichia coli FmlH lectin domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570115(CHEMBL4874004)
Affinity DataKd:  107nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570116(CHEMBL4858700)
Affinity DataKd:  356nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570117(CHEMBL4859663)
Affinity DataKd:  178nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570118(CHEMBL4876354)
Affinity DataKd:  79nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570119(CHEMBL4865920)
Affinity DataKd:  56nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570120(CHEMBL4876104)
Affinity DataKd:  533nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570121(CHEMBL4875319)
Affinity DataKd: >1.00E+3nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570122(CHEMBL4869236)
Affinity DataKd:  61nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570123(CHEMBL4854190)
Affinity DataKd:  51nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570124(CHEMBL4871009)
Affinity DataKd:  33nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570125(CHEMBL4860442)
Affinity DataKd:  7.60nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570126(CHEMBL4850273)
Affinity DataKd:  43nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570127(CHEMBL4849750)
Affinity DataKd:  171nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570128(CHEMBL4862296)
Affinity DataKd:  63nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570129(CHEMBL4866868)
Affinity DataKd:  49nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570130(CHEMBL4866323)
Affinity DataKd:  37nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570131(CHEMBL4855544)
Affinity DataKd:  38nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570132(CHEMBL4871616)
Affinity DataKd:  45nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570133(CHEMBL4846188)
Affinity DataKd:  175nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570134(CHEMBL4874752)
Affinity DataKd:  143nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570135(CHEMBL4874782)
Affinity DataKd:  65nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570136(CHEMBL4849805)
Affinity DataKd:  49nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570137(CHEMBL4847223)
Affinity DataKd:  69nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50357421(CHEMBL1917476)
Affinity DataKd:  336nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50570138(CHEMBL4846063)
Affinity DataKd:  66nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50347460(CHEMBL1170455)
Affinity DataKd:  37nMAssay Description:Antagonist activity at recombinant 6His-tagged thrombin cleavage site of FimH Lectin domain expressed in Escherichia coli HM125 assessed as dissociat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50166886(methyl alpha-D-mannoside | CHEMBL195368)
Affinity DataKd:  2.20E+3nMAssay Description:Binding affinity to Escherichia coli FimH assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50467903(CHEBI:28729 | CHEMBL365590)
Affinity DataKd:  2.30E+3nMAssay Description:Binding affinity to Escherichia coli FimH assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50347460(CHEMBL1170455)
Affinity DataKd:  5nMAssay Description:Binding affinity to Escherichia coli FimH assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50076331(CHEMBL5555901)
Affinity DataKd:  3.18E+4nMAssay Description:Binding affinity for estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details PDB3D3D Structure (crystal)
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50076332(CHEMBL5518062)
Affinity DataKd:  4.17E+5nMAssay Description:Binding affinity for estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50081076(CHEMBL5532605)
Affinity DataKd:  1.25E+5nMAssay Description:Binding affinity for estrogen receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50081077(CHEMBL5558248)
Affinity DataKd:  4.23E+4nMAssay Description:Inhibition of [3H]spiperone binding to human dopamine receptor D4.4 expressed in Chinese hamster ovary cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50081078(CHEMBL5556913)
Affinity DataKd:  6.31E+4nMAssay Description:Inhibition of [3H]spiperone binding to human dopamine receptor D2 short expressed in Chinese hamster ovary cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50135510(CHEMBL5505893)
Affinity DataKd:  1.16E+5nMAssay Description:Inhibition of [3H]spiperone binding to human dopamine receptor D2 long expressed in Chinese hamster ovary cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50135511(CHEMBL5532476)
Affinity DataKd:  1.10E+5nMAssay Description:Inhibition of [3H]-SCH- 23390 binding to dopamine receptor D1 of porcine striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50135512(CHEMBL5512541)
Affinity DataKd:  6.99E+3nMAssay Description:Inhibition of [3H]spiperone binding to human dopamine receptor D3 expressed in Chinese hamster ovary cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50135513(CHEMBL5556815)
Affinity DataKd:  7.34E+3nMAssay Description:Binding affinity towards porcine serotonin receptor 5-HT1A using [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50135514(CHEMBL5505945)
Affinity DataKd:  6.11E+3nMAssay Description:Inhibitory activity contractions of electrically stimulated mouse vas deferens was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50135515(CHEMBL5557754)
Affinity DataKd:  3.78E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50135516(CHEMBL5505793)
Affinity DataKd:  3.55E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50135517(CHEMBL5527985)
Affinity DataKd:  5.94E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50347460(CHEMBL1170455)
Affinity DataKd:  3.60E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50167930(CHEMBL1169700)
Affinity DataKd:  208nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50404815(CHEMBL3417103)
Affinity DataKd:  240nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50634636(CHEMBL1170072)
Affinity DataKd:  1.10E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50634637(CHEMBL3417101)
Affinity DataKd:  84nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50634638(CHEMBL5556130)
Affinity DataKd:  86nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
Washington University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50634639(CHEMBL4085991)
Affinity DataKd:  458nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
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