Compile Data Set for Download or QSAR
Report error Found 157 Enz. Inhib. hit(s) with Target = 'Urokinase plasminogen activator surface receptor'
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402366(CHEMBL2206696)
Affinity DataKi:  0.00100nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50005398(CHEMBL2206694)
Affinity DataKi:  0.00100nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402361(CHEMBL2206680)
Affinity DataKi:  0.00200nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402378(CHEMBL2206685)
Affinity DataKi:  0.00200nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402373(CHEMBL2206691)
Affinity DataKi:  0.00200nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402360(CHEMBL2206681)
Affinity DataKi:  0.00200nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402372(CHEMBL2206692)
Affinity DataKi:  0.00300nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402371(CHEMBL2206693)
Affinity DataKi:  0.00300nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402374(CHEMBL2206690)
Affinity DataKi:  0.00300nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402362(CHEMBL2206700)
Affinity DataKi:  0.00400nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402363(CHEMBL2206699)
Affinity DataKi:  0.00400nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402375(CHEMBL2206689)
Affinity DataKi:  0.00400nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402370(CHEMBL2206683)
Affinity DataKi:  0.00600nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402367(CHEMBL2206695)
Affinity DataKi:  0.00700nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402376(CHEMBL2206688)
Affinity DataKi:  0.00800nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402364(CHEMBL2206698)
Affinity DataKi:  0.0110nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402365(CHEMBL2206697)
Affinity DataKi:  0.0120nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402377(CHEMBL2206687)
Affinity DataKi:  0.0330nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402379(CHEMBL2206686)
Affinity DataKi:  0.296nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402368(CHEMBL2206682)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98600((2S)-2-[[(2R)-2-(benzylsulfonylamino)-3-hydroxy-pr...)
Affinity DataKi:  8.90nM ΔG°:  -45.8kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
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TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402369(CHEMBL1652555)
Affinity DataKi:  20.8nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98599((2S)-6-amino-2-[[(2R)-2-(benzylsulfonylamino)-3-hy...)
Affinity DataKi:  24nM ΔG°:  -43.3kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
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TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM50231520(CHEMBL252937 | US8476306, 6.12 | (R)-N-[(S)-1-(4-c...)
Affinity DataKi:  25nM ΔG°:  -43.2kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
Go to US Patent

TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98587((2R)-N-[(1S)-1-(benzyloxymethyl)-2-[(4-carbamimido...)
Affinity DataKi:  28nM ΔG°:  -43.0kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
Go to US Patent

TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98584(3-[[(1R)-2-[[(1S)-2-[(4-carbamimidoylphenyl)methyl...)
Affinity DataKi:  30nM ΔG°:  -42.8kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
Go to US Patent

TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98596((2R)-N-[2-[(4-carbamimidoylphenyl)methylamino]-2-o...)
Affinity DataKi:  31nM ΔG°:  -42.7kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
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TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98594((2R)-N-[2-[(4-carbamimidoylphenyl)methylamino]-2-o...)
Affinity DataKi:  32nM ΔG°:  -42.6kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
Go to US Patent

TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM50110015(N-(BENZYLSULFONYL)SERYL-N~1~-{4-[AMINO(IMINO)METHY...)
Affinity DataKi:  36nM ΔG°:  -42.3kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
Go to US Patent

TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98588((2S)-3-amino-2-[[(2R)-2-(benzylsulfonylamino)-3-hy...)
Affinity DataKi:  36nM ΔG°:  -42.3kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
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TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98583(4-[[(1R)-2-[[(1S)-2-[(4-carbamimidoylphenyl)methyl...)
Affinity DataKi:  38nM ΔG°:  -42.2kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
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TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50120747(cyclic uPA-derived peptide | CHEMBL412236)
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against human Urokinase plasminogen activator receptor (uPAR) was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98601((2S)-6-[[2-[2-[2-[2-[2-[2-[2-[2-[2-(2-aminoethoxy)...)
Affinity DataKi:  42nM ΔG°:  -42.0kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
Go to US Patent

TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50120746(cyclic uPA-derived peptide | CHEMBL405302)
Affinity DataIC50: 50nMAssay Description:Inhibitory activity against human Urokinase plasminogen activator receptor (uPAR) was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98595((2R)-N-[2-[(4-carbamimidoylphenyl)methylamino]-2-o...)
Affinity DataKi:  58nM ΔG°:  -41.2kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
Go to US Patent

TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50120740(cyclic uPA-derived peptide | CHEMBL405999)
Affinity DataIC50: 60nMAssay Description:Inhibitory activity against human Urokinase plasminogen activator receptor (uPAR) was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98590((2S)-3-benzyloxy-2-[[(2R)-2-(benzylsulfonylamino)-...)
Affinity DataKi:  61nM ΔG°:  -41.0kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
Go to US Patent

TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98591(3-[[(1R)-2-[[(1S)-2-[(4-carbamimidoylphenyl)methyl...)
Affinity DataKi:  75nM ΔG°:  -40.5kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
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TargetUrokinase plasminogen activator surface receptor(Human)
National Research Center

Curated by ChEMBL
LigandPNGBDBM50120745(cyclic uPA-derived peptide | CHEMBL263158)
Affinity DataIC50: 80nMAssay Description:Inhibitory activity against human Urokinase plasminogen activator receptor (uPAR) was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98581(methyl 2-[[(1R)-2-[[2-[(4-carbamimidoylphenyl)meth...)
Affinity DataKi:  83nM ΔG°:  -40.3kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
Go to US Patent

TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98585((2R)-N-[(1S)-2-[(4-carbamimidoylphenyl)methylamino...)
Affinity DataKi:  89nM ΔG°:  -40.1kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
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TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98598((2R)-N-[2-[(4-carbamimidoylphenyl)methylamino]-2-o...)
Affinity DataKi:  100nM ΔG°:  -39.8kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
Go to US Patent

TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98589((2S)-2-[[(2R)-2-(benzylsulfonylamino)-3-hydroxy-pr...)
Affinity DataKi:  110nM ΔG°:  -39.6kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
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TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98597((2R)-N-[2-[(4-carbamimidoylphenyl)methylamino]-2-o...)
Affinity DataKi:  110nM ΔG°:  -39.6kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
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TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98603(3-amino-N-[4-[[(2S)-2-[[(2R)-2-(benzylsulfonylamin...)
Affinity DataKi:  110nM ΔG°:  -39.6kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
Go to US Patent

TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM50110015(N-(BENZYLSULFONYL)SERYL-N~1~-{4-[AMINO(IMINO)METHY...)
Affinity DataKi:  120nM ΔG°:  -39.4kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
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TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98586((2R)-2-[[4-(aminomethyl)phenyl]methylsulfonylamino...)
Affinity DataKi:  120nM ΔG°:  -39.4kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
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TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98604(2-[4-[[(1R)-2-[[2-[4-[(3-amino-4-methoxy-benzoyl)a...)
Affinity DataKi:  130nM ΔG°:  -39.2kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
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TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98580(4-[[(1R)-2-[[2-[(4-carbamimidoylphenyl)methylamino...)
Affinity DataKi:  150nM ΔG°:  -38.8kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
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TargetUrokinase plasminogen activator surface receptor(Rat)
The Medicines

US Patent
LigandPNGBDBM98578(3-[[(1R)-2-[[2-[(4-carbamimidoylphenyl)methylamino...)
Affinity DataKi:  160nM ΔG°:  -38.7kJ/moleT: 2°CAssay Description:Inhibition constant of the compound against Plasminogen activator urokinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2013
Entry Details
Go to US Patent

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