Compile Data Set for Download or QSAR
Report error Found 162 Enz. Inhib. hit(s) with Target = 'cAMP-specific 3',5'-cyclic phosphodiesterase 4B [122-736]'
LigandPNGBDBM577157(US11472805, Example 62 | 8-Cyclopropyl-10-(5-fluor...)
Affinity DataIC50: 332nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM577156(US11472805, Example 61 | 4-(11-Oxo-6a,7,8,9-tetrah...)
Affinity DataIC50: 39nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399956(US10323042, Example 36 | US10738063, Example 36)
Affinity DataIC50: 838nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577158(US11472805, Example 63 | 13-(4-Chlorophenyl)-6a,7,...)
Affinity DataIC50: 32.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399955(US10323042, Example 35 | US10738063, Example 35)
Affinity DataIC50: 2.30E+3nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577160(US11472805, Example 64 | 8-Cyclopropyl-10-(furo[3,...)
Affinity DataIC50: 11.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399954(US10323042, Example 34 | US10738063, Example 34)
Affinity DataIC50: 979nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577161(US11472805, Example 65 | 8-Cyclopropyl-10-(2,4-dim...)
Affinity DataIC50: 6.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399953(US10323042, Example 33 | US10738063, Example 33)
Affinity DataIC50: 1.08E+3nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577152(US11472805, Example 57 | 10-(4-Chlorophenyl)-8-(5-...)
Affinity DataIC50: 3.81nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399960(US10323042, Example 40 | US10738063, Example 40)
Affinity DataIC50: 53.2nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577153(US11472805, Example 58 | 8-Cyclopropyl-10-([1,2,4]...)
Affinity DataIC50: 24nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399959(US10323042, Example 39 | US10738063, Example 39)
Affinity DataIC50: 1.26E+3nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577154(US11472805, Example 59 | 8-Cyclopropyl-10-(3,5-dif...)
Affinity DataIC50: 9.73nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399958(US10323042, Example 38 | US10738063, Example 38)
Affinity DataIC50: 168nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577155(US11472805, Example 60 | 3-(8-Cyclopropyl-9-oxo-6,...)
Affinity DataIC50: 11.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399957(US10323042, Example 37 | US10738063, Example 37)
Affinity DataIC50: 918nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577166(US11472805, Example 70 | 4-(8-Cyclopropyl-9-oxo-8,...)
Affinity DataIC50: 2.67nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399964(US10323042, Example 44 | US10738063, Example 44)
Affinity DataIC50: 55.6nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577167(US11472805, Example 71 | 5-(7-Cyclopropyl-8-oxo-5,...)
Affinity DataIC50: 43.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399963(US10323042, Example 43 | US10738063, Example 43)
Affinity DataIC50: 86.2nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577076(US11472805, Example 1 | 10-(4-Chlorophenyl)-8-(pyr...)
Affinity DataIC50: 16.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM577168(US11472805, Example 72 | 4-(7-Cyclopropyl-8-oxo-5,...)
Affinity DataIC50: 4.36nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399962(US10323042, Example 42 | US10738063, Example 42)
Affinity DataIC50: 2.05E+3nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577169(US11472805, Example 73 | 10-(4-Chloro-2-methylphen...)
Affinity DataIC50: 25.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399961(US10323042, Example 41 | US10738063, Example 41)
Affinity DataIC50: 1.65E+3nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577162(US11472805, Example 66 | 8-Cyclopropyl-10-(2,4-dim...)
Affinity DataIC50: 6.87nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399968(US10323042, Example 48 | US10738063, Example 48)
Affinity DataIC50: 65nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM399967(US10323042, Example 47 | US10738063, Example 47)
Affinity DataIC50: 90nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577163(US11472805, Example 67 | US11472805, Example 69 | ...)
Affinity DataIC50: 4.93nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM577163(US11472805, Example 67 | US11472805, Example 69 | ...)
Affinity DataIC50: 18.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399966(US10323042, Example 46 | US10738063, Example 46)
Affinity DataIC50: 471nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577163(US11472805, Example 67 | US11472805, Example 69 | ...)
Affinity DataIC50: 16.3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399965(US10323042, Example 45 | US10738063, Example 45)
Affinity DataIC50: 363nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577175(US11472805, Example 79 | 10-(4-Chlorophenyl)-8-(me...)
Affinity DataIC50: 212nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM577091(US11472805, Example 8 | 10-(4-Chloro-3-fluoropheny...)
Affinity DataIC50: 1.27nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399972(US10323042, Example 52 | US10738063, Example 52)
Affinity DataIC50: 3.09E+3nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577176(US11472805, Example 80 | 10-(4-Chlorophenyl)-N-eth...)
Affinity DataIC50: 66.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399971(US10323042, Example 51 | US10738063, Example 51)
Affinity DataIC50: 26.7nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577092(US11472805, Example 9 | 5-(4-Chlorophenyl)-7-cyclo...)
Affinity DataIC50: 298nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM577177(US11472805, Example 81 | 8-Cyclopropyl-10-(2-methy...)
Affinity DataIC50: 3.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM577093(US11472805, Example 10 | (7R)-10-(4-Chlorophenyl)-...)
Affinity DataIC50: 12.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399970(US10323042, Example 50 | US10738063, Example 50)
Affinity DataIC50: 172nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577178(US11472805, Example 82 | 8-Cyclopropyl-10-(4-methy...)
Affinity DataIC50: 1.85E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399969(US10323042, Example 49 | US10738063, Example 49)
Affinity DataIC50: 111nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577170(US11472805, Example 74 | 10-(4-Chloro-3-fluorophen...)
Affinity DataIC50: 27nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM399976(US10323042, Example 55 | US10738063, Example 55)
Affinity DataIC50: 3.61E+3nMAssay Description:Human PDE4B1 coding sequence (amino acids 122 to 736 from the sequence with accession number Q07343) with the mutations resulting in the amino acid s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/4/2021
Entry Details
US Patent

LigandPNGBDBM577078(US11472805, Example 3 | (6aR)-12-(4-Chlorophenyl)-...)
Affinity DataIC50: 1.38nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM577080(US11472805, Example 5 | 10-(4-Chlorophenyl)-8-(4H-...)
Affinity DataIC50: 5.87nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

LigandPNGBDBM577171(US11472805, Example 75 | 10-(4-Chlorophenyl)-8-cyc...)
Affinity DataIC50: 3.99nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

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