2543 SMILES Strings for Focal adhesion kinase 1

Compound Name
SMILES String
Cn1ncc2c(cccc12)-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12
CN(C)C(=O)N1CCc2ccc(Nc3nc4c(cccn4n3)-c3cc(Cl)ccc3OCC(F)F)cc2CC1
Cn1ncc2c(cccc12)-c1cccn2nc(Nc3ccc4CCN(CCc4c3)C(=O)OC(C)(C)C)nc12
CS(=O)(=O)c1ccc(cc1)C(=C)n1nc(NC(=O)Nc2ccc(cc2)N2CCNCC2)nc1C=C
C[C@H](Nc1cc2n(nc(C)c2cn1)-c1cc(Cl)cc(CCC(N)=O)c1)c1ccccc1 |r|
C[C@H](Nc1cc2n(nc(C)c2cn1)-c1cc(Cl)cc(c1)-c1ccccc1NC(C)=O)c1ccccc1 |r|
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(Cl)cc23)c1F
Cc1[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c(C)c1C(=O)NC[C@H](O)CN1CCOCC1
CN[C@H]1C[C@@H]2O[C@](C)([C@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13
CCN(CC)CCNC(=O)c1c(C)[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c1C
CCOC(=O)CSc1nc(nc2ccccc12)C1CC1
COCCOC(=O)C1C(c2ccsc2)C2=C(CC(CC2=O)c2cccs2)N=C1C |c:29,t:15|
C1Cc2c([nH]c3ccccc23)-c2n[nH]cc12
CN1CCN(CC1)c1ccc(N)c(c1)N1CCN(C)CC1
CC(C)c1nc(SCC(=O)N2CCCC2)c2ccccc2n1
Cc1ccccc1-c1ccc(Nc2ccc(cc2)N2CCOCC2)nn1
Oc1c(C(=O)Nc2cccnc2)c(=O)c2cccc3CCn1c23
COC(=O)c1cccc2C(N=O)c3ccccc3-c12
COC(=O)CSc1nc(nc2ccccc12)C(C)C
O=C(OCCN=C1NS(=O)(=O)c2ccccc12)c1cccnc1 |w:5.4|
CCc1nc(SCC(=O)N2CCCC2)c2ccccc2n1
Cc1ccc2nsnc2c1S(=O)(=O)Nc1cccc2nsnc12
CCN(CC)C(=O)CSc1nc2ccc(CC)cc2cc1C#N
CCn1c2ccccc2c(O)c(C(=O)Nc2nc3ccccc3[nH]2)c1=O
OP(O)(=O)C(=C)c1cccc2ccccc12
CC(C)c1nc2n[nH]c(N)c2c2CCCCc12
COC(=O)c1[nH]c2ccc(C)cc2c1NC(=O)CN1CCCc2ccccc12
COCCN(Cc1ccccc1)P(O)(=O)c1ccccc1OCC(O)=O
CN1CCc2c(C1)sc1N=CN3N\C(N=C3c21)=C1/C=CC=CC1=O |c:10,15,22,24|
OP(O)(=O)c1cccc(Cl)c1C(=O)Oc1ccccc1
CC(C)c1nc2n[nH]c(N)c2c2CCCc12
Oc1ccccc1-c1nc(NCCN2CCOCC2)c2ccccc2n1
Cc1ccc2[nH]c3c(NCc4ccco4)ncnc3c2c1
CC1(C)CCCN(C1)C(=O)c1coc(=O)c(Br)c1
NC(=O)C1CCN(CC1)c1oc(nc1C#N)-c1ccc(OCc2ccc(Cl)cc2)cc1
COc1ccc2[nH]c(=O)c(cc2c1)-c1noc(n1)-c1ccccc1
c1cc(c2c(c1Cl)c3c([nH]2)C(=O)NCC3)Cl
Brc1ccc(o1)-c1nc2ccc(cc2[nH]1)N1C(=O)c2ccccc2C1=O
OP(O)(=O)c1ccccc1OCc1ccccc1
COc1ccc(cc1)-c1cnc(N)nc1-c1ccc(OC)cc1O
Cc1n[nH]c(NC=C2C(=O)CC(C)(C)CC2=O)c1-c1ccccc1 |(8.76,5.94,;7.85,4.69,;6.31,4.69,;5.84,3.23,;7.08,2.32,;7.08,.78,;5.75,.01,;5.75,-1.53,;4.41,-2.3,;3.08,-1.53,;4.41,-3.84,;5.75,-4.61,;4.98,-5.94,;6.52,-5.94,;7.08,-3.84,;7.08,-2.3,;8.41,-1.53,;8.33,3.23,;9.79,2.75,;10.11,1.25,;11.58,.77,;12.72,1.8,;12.4,3.31,;10.94,3.78,)|
Cc1n[nH]c(NC=C2C(=O)CC(C)(C)CC2=O)c1-c1ccc(Cl)cc1 |(8.76,5.94,;7.85,4.69,;6.31,4.69,;5.84,3.23,;7.08,2.32,;7.08,.78,;5.75,.01,;5.75,-1.53,;7.08,-2.3,;8.41,-1.53,;7.08,-3.84,;5.75,-4.61,;4.98,-5.94,;6.52,-5.94,;4.41,-3.84,;4.41,-2.3,;3.08,-1.53,;8.33,3.23,;9.79,2.75,;10.11,1.25,;11.58,.77,;12.72,1.8,;14.19,1.33,;12.4,3.31,;10.94,3.78,)|
O=C1Nc2ccc(NS(=O)(=O)c3cccs3)c3cccc1c23
FC(F)(F)c1cnc2Sc3ccccc3Nc2c1
CC(C)(C)c1cc(NC(=O)COC(=O)c2ccc3c(c2)nc2CCCn2c3=O)n(n1)-c1ccccc1
CCCn1c(NC(=O)c2ccc(Cl)c(c2)S(=O)(=O)N2CCCC2)nc2ccccc12
CCOC(=O)c1sc2N=C3CCCC(=O)C3C(c3cccs3)c2c1C |t:8|
Cc1ccc2c(Cl)cc(Cl)c(OCc3nnc(o3)-c3ccccc3)c2n1
C[C@H]1CCCC(=O)CCCC=Cc2cc(O)cc(O)c2C(=O)O1
COc1ccc(cc1)-c1nnc(Nc2nc3c(OC)cccc3s2)o1
[#6]C([#6])([#6])[#6](=O)-[#7]\[#6](=[#6](/Cl)Cl)P([#8])([#8])=O
CCOC(=O)c1cccc2C(N=O)c3ccccc3-c12
N#CCSc1nc(Nc2ccc3OCOc3c2)c2ccccc2n1
Cc1ccc2cc3cc(oc3nc2c1)C(=O)NCc1ccc2OCOc2c1
O=c1n(CN2CCOCC2)nc2-c3ccccc3-c3cccc1c23
O=C(Nc1ccc(cc1)-n1nncc1-c1ccco1)c1cc2ccccc2oc1=O
Fc1ccccc1CS(=O)(=O)Cc1ccc(o1)C(=O)NCCCN1CCCCCC1
O=C1Nc2ccccc2C1C=Nc1ccc2OCCOc2c1 |w:11.13|
CSc1nc2ccc3nc(NC(=O)c4cccs4)sc3c2s1
Cn1c2ccccc2c(=O)n2c1cc1ccccc1c2=O
O=C(NCCc1c[nH]c2ccccc12)C1CCN(CC1)c1nnc(s1)N1CCCC1=O
OP(O)(=O)c1ccccc1OCCCCCOc1ccccc1P(O)(O)=O
O=c1[nH]c(Nc2ccccc2)cc2ccccc12
COc1ccc(cc1OC)N=CC1C(=O)Nc2ccccc12 |w:10.10|
CN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)NCc1ccco1
O=c1oc2ccccc2n1CCn1c2ccccc2c2nc3ccccc3nc12
O=C(Nc1cccc(c1)C(=O)Nc1cccc(c1)-c1nc2ccccc2[nH]1)c1ccco1
COc1cc(cc(OC)c1O)C1Nc2ccc3ncccc3c2C2=C1C(=O)CCC2 |c:26|
CCN1CCc2c(C1)sc(N)c2C#N
Cc1cc(NC(=O)Cc2cccs2)no1
OC(=O)c1cccc(c1)S(=O)(=O)Nc1ccccc1Cl
NC(=O)c1sc2nc3CCCc3c(-c3ccco3)c2c1N
COc1cc2nc(oc(=O)c2cc1OC)-c1ccc(Br)o1
OC(=O)c1ccc(F)c(c1)S(=O)(=O)Nc1ccccc1Cl
COc1ccc(OC)c(NS(=O)(=O)Cc2ccccc2)c1
COc1ccc(cc1NC(=O)c1ccc(Br)o1)-c1cc2ccccc2oc1=O
O=C(CSc1nnc2scc(-c3ccccc3)n12)Nc1nsc(n1)-c1ccccc1
Cc1ccc(OCC(=O)Nc2ccc(cc2)-c2nc3ncccc3o2)c(C)c1
OC(=O)c1ccccc1OCCOCCOc1ccccc1C(O)=O
COC(=O)C1C(NC(=O)N=C1CSCc1ccco1)c1cc(C)ccc1C |c:9|
O=C1Cc2ccccc2C(=O)N1CCc1ccccc1
Cc1nnc2sc(nn12)-c1ccc(C)c(NC(=O)COc2ccc(Cl)c(C)c2)c1
OC(=O)c1ccc(F)c(c1)S(=O)(=O)Nc1ccccc1
CCc1ccc(OCC(=O)Nc2ccc(-c3nc4ccccc4o3)c(O)c2)cc1
CCOCCOC(=O)C1C(c2ccsc2)C2=C(CC(CC2=O)c2cccs2)N=C1C |c:30,t:16|
COC(=O)C1C(c2ccsc2)C2=C(CC(CC2=O)c2cccs2)N=C1C |c:26,t:12|
Cc1cc(C)cc(OCC(=O)Nc2ccc(cc2)N2CCCC2)c1
CCCCn1c(CN2C(=O)c3ccccc3C2=O)nc2ccccc2c1=O
Nc1ncnc2oc(-c3ccco3)c(-c3ccco3)c12
COc1cc(cc(OC)c1OC)N=CC1C(=O)Nc2ccccc12 |w:12.12|
COC(=O)Cc1ccc2c(c1)n(C)c1ccccc21
O=C(Nc1ccc2oc(nc2c1)-c1cccnc1)c1cc2ccccc2o1
CCOC(=O)c1cnn(c1N)-c1ncnc2sc(CC)cc12
CCN(CC)c1ccc2cc(-c3nc4ccccc4[nH]3)c(=O)oc2c1
Cc1c(C(N)=O)c(N)c(C(=O)c2ccccc2)n1-c1ccccc1
O=NCc1c(Nc2ccccc2)nc2ccccn2c1=O
CN(C)C=NC(=O)C(C#N)C1=Nc2ccccc2CC1 |w:4.4,t:10|
Cc1c(N2C(=O)c3ccc4CCc5ccc(C2=O)c3c45)c(=O)n(-c2ccccc2)n1C
O=C1C(C(=O)c2ccccc12)c1ccnc2ccccc12
COc1cc(cc(OC)c1O)C1Nc2ccc3ncccc3c2C2=C1C(=O)CC(C)(C)C2 |c:26|
CCOC(=O)CSc1nc(nc2ccccc12)C(C)C
CC(C)c1nc(SCC(=O)Nc2cc(C)on2)c2ccccc2n1
CN(C)CCN1CCc2ccccc12
O=C(Nc1ccc(cc1)-c1nc2ccc(NC(=O)c3cccs3)cc2[nH]1)c1cccs1
Cc1ccc2nc(oc(=O)c2c1)-c1ccc(Br)o1
Brc1ccc(o1)-c1nc2ccccc2c(=O)o1
O=C1Cc2ccccc2C(=O)N1Cc1ccccc1
Cc1oc(cc1C(=O)Nc1cccc2ccccc12)-c1ccccc1
CCOC(=O)C1=C(OC(=N)C(C#N)C1C1CCCCC1)c1ccccc1 |t:5|
CCOc1ccc(cc1)-n1c(SCc2nc(no2)-c2ccc(C)cc2)nnc1-c1ccncc1
Fc1ccc(cc1)-c1onc2ccc(C=O)cc12
Cc1ccc(cc1)-c1onc2ccc(C=O)cc12
O=Cc1ccc2noc(-c3ccccc3)c2c1
Nc1ccc-2c(c1)C(=O)C(=O)c1ccccc-21
O=C(Nc1ccc(cc1)N1CCCC1)C(c1ccccc1)c1ccccc1
c1nc2ccccc2n1-c1ccc(cc1)-c1ccnc(n1)-c1ccccc1
COc1ccc(cc1)C(=O)Nc1nc2ccc3nc(C)sc3c2s1
NC(=O)C(C#N)C1=Nc2ccccc2CC1 |t:6|
CCc1c(C)nc(SCC(=O)c2cccs2)c(C#N)c1C
COc1ccc(cc1OC)-c1nc(-c2cccs2)c([nH]1)-c1cccs1
Clc1cccc(c1)N1CCN(CC1)C(=O)CCCn1c(=S)[nH]c2ccccc2c1=O
Oc1ccc2ccccc2c1C=Nc1ccc(cc1)N1CCOCC1 |w:12.14|
Brc1ccc(o1)C(=O)Oc1ccc(cc1)-c1cnc2ccccc2n1
CCOC(=O)CNC(=O)c1sc2ncnc(N3CCc4ccccc4C3)c2c1C
O=c1cc(oc2c3ccccc3ccc12)-c1ccco1
O=C(c1coc-2c1C(=O)C(=O)c1ccccc-21)c1ccccc1
C(N1CCOCC1)c1ccc2ccc3cccc4ccc1c2c34
Cc1ccc(OC(=O)c2ccccc2P(O)(O)=O)cc1
COc1ccc(cc1)N=CC1C(=O)Nc2ccccc12 |w:8.8|
COc1ccc(cc1)-n1nc(C(=O)Nc2ccc(OC)c(OC)c2)c2c3ccccc3n(C)c2c1=O
CCOC(=O)c1ccc(NC2=CC(=O)C(=O)c3ccccc23)cc1 |t:10|
CN1C(=O)\C(=C\c2cn(CC(=O)N3CCCCC3)c3ccccc23)c2ccccc12
COC(=O)c1ccccc1NC(=O)c1c(Br)cnn1C
OP(O)(=O)c1ccccc1C(=O)Oc1ccccc1Cl
Oc1ccccc1C(=O)\N=N\c1ccc(NOC(=O)c2ccccc2)cc1
CC(=O)c1ccc(NC(=O)c2ccc3nc(-c4ccco4)c(nc3c2)-c2ccco2)cc1
CCc1n[nH]c2cccc3c(OC)ccc1c23
CC(C)(C)C(=O)Nc1nc-2c(COc3ccccc-23)s1
CC1CCN(CC1)c1ncnc2nc[nH]c12
CCN(CC)C(=O)CSc1nc(N)c2c3CCC(C)Cc3sc2n1
Cc1oc-2c(c1C(=O)c1ccccc1)C(=O)C(=O)c1ccccc-21
CC(N1C(=S)S\C(=C/C=C/c2ccco2)C1=O)C(O)=O
[H]C12CC3([H])CC([H])(C1)CC(C2)(C3)C(=O)c1sc2nc3CCN(C)Cc3cc2c1N |TLB:8:1:12:6.9.5,8:6:12:1.11.2,THB:5:6:11:3.12.2|
COc1nnc(-c2ccc(N3CCCCC3)c(NC(C)=O)c2)c2ccccc12
CN1CCN(CC1)c1ccc(N)cc1
Cc1nn2C(C3C(=O)CCCC3=Nc2c1-c1ccccc1)c1ccccc1 |c:12|
CC(=O)c1ccc(NCC(=O)N2CCN(CC2)c2ccccc2)cc1
C=CCn1c(SCC(=O)N2CCCC2)nc2scc(-c3cccs3)c2c1=O
CCN(CC)S(=O)(=O)c1cc(ccc1NNC(=O)Nc1ccccc1)[N+]([O-])=O
Clc1ccc(c(Cl)c1Cl)-c1cc(C(=O)OCC(=O)N2CCN(CC2)C(=O)c2ccco2)c2ccccc2n1
OP(=O)(c1nc2ccccc2n1CC=C)c1ccccc1
Cc1cc(N)ccc1N1CCCC1
[O-][N+](=O)c1ccccc1NC(=O)[C-]1c2[nH]c3ccccc3[n+]2CCC1=O
[O-][N+](=O)c1c[c-](C[NH+]=Nc2nccs2)ccc1=O |w:7.6|
O=C1C(=O)c2ccccc2-c2ccccc12
Cc1ccc(Cl)cc1NC1=CC(=NS(=O)(=O)c2cccs2)c2ccccc2C1=O |w:12.13,t:10|
O=C(CSc1ccc2-c3ccccc3C(=O)c3cccc1c23)Nc1cccc(c1)C#N
Cc1ccccc1NC1=CC(=NS(=O)(=O)c2cccs2)c2ccccc2C1=O |w:11.12,t:9|
Clc1ccc(cc1)C(=O)NN=c1c2cccc3cccc(c23)c1=O |w:10.10|
COc1ccccc1CNC(=O)COC(=O)c1cc(nc2ccccc12)-c1ccco1
COc1ccc(cc1)-c1ccc2c(N)c(sc2n1)C(=O)c1ccc(OC)c(OC)c1
COc1cccc(c1)\N=c1/oc2ccc(OC)cc2cc1-c1nc2ccccc2[nH]1
Cn1c(SCC(=O)Nc2ccc3nc(SCC(=O)N4CCCC4)sc3c2)nnc1-c1ccc(N)cc1
NNC(=O)C(=NNc1c(Cl)cccc1Cl)C#N |w:5.5|
Cc1ccc(cc1)-c1cc(nc2ncnc(N)c12)-c1ccc(F)cc1
Cc1ccc(cc1C)C(=O)COC(=O)c1ccc2C(=O)N(C(=O)c2c1)c1cccc2ncccc12
Clc1ccc2nc(N=NCc3ccccc3C#N)nc(-c3ccccc3)c2c1 |w:7.6|
Clc1ccc(CSc2nc(ccc2C#N)-c2cccnc2)c(Cl)c1
COc1ccc(cc1OC)C(=O)c1sc2nc(ccc2c1N)-c1ccccc1
Nc1ncnc2nc(cc(-c3ccc(F)cc3)c12)-c1ccccc1
COc1cccc(Cn2cc(O)c(c2N)-c2nc(cs2)-c2ccc(Cl)cc2)c1
O=C(NN=Cc1ccc2ccccc2c1)c1ccc(COc2ccc3CCCc3c2)o1 |w:3.2|
CCOc1ccc(NC2=NC(=O)SC2=Cc2ccc(Cl)cc2)cc1 |w:14.15,t:8|
Nc1c(sc2nc(ccc12)-c1cccs1)C(=O)Nc1nc2ccccc2s1
COc1ccc(cc1Cl)-n1nc(C(=O)NCC(=O)Nc2ccccn2)c2ccccc2c1=O
N#Cc1cnn2c1nc(N1CCCCC1)c1ccccc21
N#Cc1cnn2c1nc(N1CCOCC1)c1ccccc21
Clc1ccc2[nH]cc(-c3nnnn3-c3ccccc3)c2c1
Clc1cc(C=NNC(=O)c2cc3ccccc3o2)ccc1OCC(=O)Nc1ccccc1 |w:5.5|
[O-][N+](=O)c1ccc(N2CCCCCC2)c([CH+][N-]NC(=O)Cn2c3ccccc3c(=O)c3ccccc23)c1
Cc1n[nH]c(C)c1N=Nc1cc(Cl)ccc1Cl |w:8.9|
CCOc1cc(\C=C2\NC(=S)NC2=O)ccc1OCc1ccc(cc1)[N+]([O-])=O
O=C1CCCC2=C1C(Nc1ccc3ncccc3c21)c1cccs1 |c:5|
O=C(CSc1nc(nc2ccccc12)C1CC1)NCc1ccc2OCOc2c1
CC(C)c1nc(SCC(=O)Nc2nnc(C)s2)c2ccccc2n1
O=C(CSc1nc(nc2ccccc12)C1CC1)Nc1ccc2OCCOc2c1
CCc1nc(SCC(=O)NNC(=O)C2CCCCC2)c2ccccc2n1
O=C(CSc1nc(nc2ccccc12)C1CC1)N1CCc2ccccc2C1
Cc1ccsc1C1Nc2ccc3ncccc3c2C2=C1C(=O)CCC2 |c:21|
CCOc1ccc2nc(NC3=NC(CC(=O)N3)c3ccc(OC)cc3)nc(C)c2c1 |t:10|
COc1ccc2nc(C)cc(SCC(=O)NN=Cc3cccc4ccccc34)c2c1 |w:16.15|
Clc1c(sc2ccccc12)C(=O)Nc1cccc(c1)-c1nc2ncccc2o1
O=C(COc1ccccc1)Nc1sc2CCCCc2c1C(=O)NCc1cccnc1
Fc1ccc(C=NNC(=O)c2cc(nc3ccccc23)-c2ccco2)cc1 |w:6.6|
Brc1cc(C=NNC(=O)c2cc3ccccc3o2)ccc1OCC(=O)Nc1ccccc1 |w:5.5|
[O-][N+](=O)c1cccc(C=Cc2nc3ccc(cc3[nH]2)[N+]([O-])=O)c1 |w:9.9|
Fc1cccc(C=NNC(=O)c2cc(nc3ccccc23)-c2ccco2)c1 |w:7.7|
Cc1ccsc1C1Nc2ccc3ncccc3c2C2=C1C(=O)CC(C)(C)C2 |c:21|
CCOc1ccc(cc1)S(=O)(=O)N(CC(=O)N\N=C\c1ccc(o1)-c1ccc(cc1)[N+]([O-])=O)c1ccccc1
Cc1ccc(cc1)C(=O)NNC(=O)CSc1nnc2c(n1)[nH]c1ccc(F)cc21
Cc1cc2cc3c(N)[nH]nc3nc2cc1C
CCc1ccc2nc3n[nH]c(N)c3cc2c1
O=C1Nc2ccccc2C1=Cc1cnc[nH]1 |w:10.12|
CN(C)c1cc(N(C)C)c2C(=O)c3ccccc3C(=O)c2c1
Clc1ccc(cc1S(=O)(=O)Nc1ccccc1)C(=O)Nc1ccccc1C(=O)NCC=C
COc1ccc(cc1COc1cc(C)cc2oc(=O)cc(-c3ccccc3)c12)[N+]([O-])=O
COC(=O)c1cc(Cl)c(NC(=O)\C=C\c2ccc(Cl)cc2)cc1OC
O=C(Nc1cccc(c1)-c1cn2ccccc2n1)c1cc2ccccc2oc1=O
CCOC(=O)c1cnc2ccc(C)cc2c1Nc1ccc(cc1)N1CCOCC1
Clc1cc(NC(=O)c2cccnc2)ccc1-c1cc2ccccc2oc1=O
CC(=O)Nc1ccc(Nc2ncc(c(Nc3ccc(NC(C)=O)cc3)n2)[N+]([O-])=O)cc1
COc1ccc(cc1NC(=S)NC(=O)c1ccc2OCCOc2c1)-c1cc2ccccc2oc1=O
CCOC(=O)C1=C(OC(=N)C(C#N)C1c1cccs1)c1ccccc1 |t:5|
Cc1cc(OCC(=O)Nc2ccc(cc2)N2CCN(CC2)C(=O)c2ccco2)cc(C)c1Cl
[O-][N+](=O)c1ccc(\C=C\C=N\NC(=O)c2cccs2)cc1
COc1ccc(cc1F)-c1coc2cc3oc(=O)cc(C)c3cc12
Clc1c(sc2cc(Cl)ccc12)C(=O)Nc1cccc(c1)-c1nc2ncccc2o1
Cn1c(SCC(=O)c2ccc-3c(Cc4ccccc-34)c2)nnc1-c1ccccc1
COC(=O)c1ccc(COc2ccc(\C=C(/C#N)c3nc4ccccc4[nH]3)cc2OC)o1
COc1ccccc1-c1cccn2nc(Nc3ccc(cc3)N3CCOCC3)nc12
CS(=O)(=O)c1ccc(cc1)c2cccn3c2nc(n3)Nc4ccc(cc4)N5CCOCC5
C1CN(CCO1)c1ccc(Nc2nc3c(cccn3n2)-c2cccnc2)cc1
COc1ccc(cn1)-c1cccn2nc(Nc3ccc(cc3)N3CCOCC3)nc12
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3ccc(OCCN4CCCC4)cc3)nc12
C1CN(CCO1)c1ccc(Nc2nc3c(cccn3n2)-c2ccncc2)cc1
CS(=O)(=O)c1ccc(cc1)-c1cccc2nc(Nc3ccc(cc3)N3CCOCC3)nn12
CS(=O)(=O)c1cccc(c1)-c1cccn2nc(Nc3ccc(OCCN4CCCC4)cc3)nc12
COc1ccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)cc1
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3ccc(OCCN4CCOCC4)cc3)nc12
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3cccc(c3)N3CCOCC3)nc12
CS(=O)(=O)c1cccc(c1)-c1cccn2nc(Nc3cccc(c3)N3CCOCC3)nc12
CN1CCN(CC1)c1ccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)cc1
CN1CCN(CC1)c1cccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)c1
CS(=O)(=O)c1ccc(cc1)-c1ccc2nc(Nc3ccc(cc3)N3CCOCC3)nn2c1
CN1CCN(CC1)c1ccc(Nc2nc3ccc(cn3n2)-c2ccc(cc2)S(C)(=O)=O)cc1
COc1ccc(Nc2nc3c(Nc4ccc(cc4)S(C)(=O)=O)cccn3n2)cc1
COc1ccc(Nc2nc3c(cccn3n2)-c2cn[nH]c2)cc1
COc1cccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)c1
COc1ccc(Nc2nc3c(NC4CCN(CC4)S(C)(=O)=O)cccn3n2)cc1
COc1ccc(Nc2nc3c(cccn3n2)-c2cnn(c2)S(C)(=O)=O)cc1
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3ccc(CN4CCOCC4)cc3)nc12
CN1CCN(Cc2ccc(Nc3nc4c(cccn4n3)-c3ccc(cc3)S(C)(=O)=O)cc2)CC1
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3ccc(OS(=O)(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)F)cc3)nc12
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3cccc(CN4CCOCC4)c3)nc12
COc1ccc(Nc2nc3c(Nc4ccccc4S(C)(=O)=O)cccn3n2)cc1
CN1CCN(CC1)c1ccc(Nc2nc3c(cccn3n2)-c2ccc(CS(C)(=O)=O)cc2)cc1
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3ccc(cc3)N3CCC(CC3)N3CCOCC3)nc12
CN1CCC(CC1)c1ccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)cc1
CN1CCN(CC1)C1CCN(CC1)c1ccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)cc1
CC(C)S(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3ccc(cc3)N3CCN(C)CC3)nc12
CC(C)S(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3cccc(c3)N3CCN(C)CC3)nc12
CN(C)S(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3ccc(cc3)N3CCN(C)CC3)nc12
COc1ccccc1-c1cccn2nc(Nc3ccc(cc3)N3CCN(C)CC3)nc12
COc1ccccc1-c1cccn2nc(Nc3cccc(c3)N3CCN(C)CC3)nc12
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3cccc(c3)N3CCC(CC3)N3CCOCC3)nc12
CN1CCN(CC1)C1CCN(CC1)c1cccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)c1
CN1CCN(CC1)c1ccc(Nc2nc3c(cccn3n2)-c2cccc(c2)S(C)(=O)=O)cc1
CN1CCN(CC1)c1cccc(Nc2nc3c(cccn3n2)-c2cccc(c2)S(C)(=O)=O)c1
CN1CCC(CC1)c1cccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)c1
CN(c1ccc(cc1)-c1cccn2nc(Nc3ccc(cc3)N3CCN(C)CC3)nc12)S(C)(=O)=O
CN(c1ccc(cc1)-c1cccn2nc(Nc3cccc(c3)N3CCN(C)CC3)nc12)S(C)(=O)=O
CN1CCN(CC1)c1ccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)C(F)(F)F)cc1
CN1CCN(CC1)c1cccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)C(F)(F)F)c1
CN1CCN(CC1)c1ccc(Nc2nc3c(cccn3n2)-c2ccccc2S(C)(=O)=O)cc1
CN1CCN(CC1)c1cccc(Nc2nc3c(cccn3n2)-c2ccccc2S(C)(=O)=O)c1
CN1CCN(CC1)c1cccc(Nc2nc3c(Nc4ccccc4S(C)(=O)=O)cccn3n2)c1
CS(=O)(=O)c1ccccc1Nc1nc2c(Nc3ccccc3S(C)(=O)=O)cccn2n1
CN1CCN(CC1)c1ccc(Nc2nc3cccc(-c4ccc(CN5CCS(=O)(=O)CC5)cc4)n3n2)cc1
CN1CCN(CC1)c1cccc(Nc2nc3cccc(-c4ccc(CN5CCS(=O)(=O)CC5)cc4)n3n2)c1
CN1CCN(CC1)c1ccc(Nc2nc3c(Nc4ccccc4S(C)(=O)=O)cccn3n2)cc1
CS(=O)(=O)c1ccc(cc1)-c1cccc2nc(Nc3ccc(OCCN4CCCC4)cc3)nn12
CC(C)(C)OC(=O)N1CCN(CC1)c1ccc(Nc2nc3cccc(-c4ccc(cc4)S(C)(=O)=O)n3n2)cc1
C(CN1CCCC1)Oc1ccc(Nc2nc3cccc(-c4ccccc4)n3n2)cc1
CS(=O)(=O)c1cccc(c1)-c1cccc2nc(Nc3ccc(cc3)N3CCOCC3)nn12
CN1CCN(CC1)c1ccc(Nc2nc3cccc(-c4ccc(cc4)S(C)(=O)=O)n3n2)cc1
CN1CCN(CC1)c1ccc(Nc2nc3cccc(-c4cccc(c4)S(C)(=O)=O)n3n2)cc1
CN1CCN(CC1)c1ccc(Nc2nc3cccc(-c4cccc(NS(C)(=O)=O)c4)n3n2)cc1
CN1CCN(CC1)c1ccc(Nc2nc3cccc(-c4ccc(NS(C)(=O)=O)cc4)n3n2)cc1
CS(=O)(=O)c1ccc(cc1)-c1cccc2nc(Nc3ccc(CN4CCOCC4)cc3)nn12
CN1CCN(Cc2ccc(Nc3nc4cccc(-c5ccc(cc5)S(C)(=O)=O)n4n3)cc2)CC1
CS(=O)(=O)c1cccc(c1)-c1cccc2nc(Nc3ccc(CN4CCOCC4)cc3)nn12
CN1CCN(Cc2ccc(Nc3nc4cccc(-c5cccc(c5)S(C)(=O)=O)n4n3)cc2)CC1
CN1CCN(CC1)c1ccc(NC(=O)Nc2nc3cccc(-c4cccc(c4)S(C)(=O)=O)n3n2)cc1
CN1CCN(CC1)c1ccc(NC(=O)Nc2nc3cccc(-c4ccc(cc4)S(C)(=O)=O)n3n2)cc1
COc1ccc(Nc2nc3cccc(-c4ccc(cc4)S(C)(=O)=O)n3n2)cc1
CN1CCN(CC1)c1cccc(Nc2nc3cccc(-c4ccc(cc4)S(C)(=O)=O)n3n2)c1
CS(=O)(=O)c1ccc(Nc2nc3cccc(-c4ccc(cc4)S(C)(=O)=O)n3n2)cc1
CS(=O)(=O)c1ccc(cc1)-c1cccc2nc(Nc3cccc(c3)S(C)(=O)=O)nn12
COc1ccc(Nc2nc3cccc(-c4ccc(CN5CCS(=O)(=O)CC5)cc4)n3n2)cc1
CN1CCN(CC1)c1nc2c(NCc3cccc(c3)[N+]([O-])=O)cccn2n1
[O-][N+](=O)c1cccc(CNc2cccn3nc(nc23)N2CCOCC2)c1
NC1CCN(CC1)c1nc2c(NCc3cccnc3)cccn2n1
C(CN1CCOCC1)Nc1nc2c(NCc3cccnc3)cccn2n1
CN1CCN(CC1)c1cccc(Nc2nc3c(cc(cn3n2)C(F)(F)F)-c2ccc(cc2)S(C)(=O)=O)c1
CN1CCN(CC1)c1ccc(Nc2nc3c(cc(cn3n2)C(F)(F)F)-c2ccc(cc2)S(C)(=O)=O)cc1
CN1CCN(CC1)c1ccc(Nc2nc3c(cc(cn3n2)C(F)(F)F)-c2ccc(cc2)S(C)(=O)=O)cn1
CN1CCN(CC1)c1cccc(c1)N(c1nc2c(cc(F)cn2n1)-c1ccc(cc1)S(C)(=O)=O)c1cccc(c1)N1CCN(C)CC1
CN1CCN(CC1)c1ccc(Nc2nc3c(cc(F)cn3n2)-c2ccc(cc2)S(C)(=O)=O)cc1
CN1CCN(CC1)c1cccc(Nc2nc3cncc(-c4ccc(cc4)S(C)(=O)=O)n3n2)c1
CN1CCN(CC1)c1cncc(Nc2nc3cncc(-c4ccc(cc4)S(C)(=O)=O)n3n2)c1
CN1CCN(CC1)c1ccc(Nc2nc3c(Nc4cccc(c4)S(C)(=O)=O)cccn3n2)cc1
CN1CCN(CC1)c1cccc(Nc2nc3c(Nc4cccc(c4)S(C)(=O)=O)cccn3n2)c1
CN(c1ncccc1Nc1cccn2nc(Nc3cccc(c3)N3CCN(C)CC3)nc12)S(C)(=O)=O
CS(=O)(=O)c1ccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)cc1
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3cccc(c3)S(C)(=O)=O)nc12
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3ccc(CN4CCS(=O)(=O)CC4)cc3)nc12
CS(=O)(=O)c1ccc(cc1)-c1cccc2nc(Nc3ccc(CN4CCS(=O)(=O)CC4)cc3)nn12
CN1CCN(Cc2cccc(Nc3nc4c(cccn4n3)-c3ccc(cc3)S(C)(=O)=O)c2)CC1
CS(=O)(=O)c1ccc(cc1)-c1cccc2nc(Nc3cccc(CN4CCOCC4)c3)nn12
CN1CCN(Cc2cccc(Nc3nc4cccc(-c5ccc(cc5)S(C)(=O)=O)n4n3)c2)CC1
CN(c1ccc(cc1)-c1cccn2nc(Nc3ccc(CN4CCS(=O)(=O)CC4)cc3)nc12)S(C)(=O)=O
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3cccc(CN4CCS(=O)(=O)CC4)c3)nc12
CS(=O)(=O)c1ccc(cc1)-c1cccc2nc(Nc3cccc(CN4CCS(=O)(=O)CC4)c3)nn12
CN(c1ncccc1CNc1cccn2nc(Nc3ccc(cc3)N3CCN(C)CC3)nc12)S(C)(=O)=O
CN(c1ncccc1CNc1cccn2nc(Nc3ccc(cc3)C3CCN(C)CC3)nc12)S(C)(=O)=O
CN(c1ncccc1CNc1cccn2nc(Nc3ccc(OCCN4CCCC4)cc3)nc12)S(C)(=O)=O
CN1CCC(CC1)c1ccc(Nc2nc3c(Nc4ccccc4S(C)(=O)=O)cccn3n2)cc1
CS(=O)(=O)c1ccccc1Nc1cccn2nc(Nc3ccc(OCCN4CCCC4)cc3)nc12
CN(c1cccc(c1)-c1cccn2nc(Nc3ccc(cc3)N3CCN(C)CC3)nc12)S(C)(=O)=O
CN(c1cccc(c1)-c1cccn2nc(Nc3ccc(OCCN4CCCC4)cc3)nc12)S(C)(=O)=O
CN(c1cccc(c1)-c1cccn2nc(Nc3cccc(c3)C3CCN(C)CC3)nc12)S(C)(=O)=O
CN(c1ccccc1-c1cccn2nc(Nc3cccc(c3)C3CCN(C)CC3)nc12)S(C)(=O)=O
CN(c1ncccc1Nc1cccn2nc(Nc3ccc(cc3)N3CCN(C)CC3)nc12)S(C)(=O)=O
CN(c1ncccc1Nc1cccn2nc(Nc3ccc(OCCN4CCCC4)cc3)nc12)S(C)(=O)=O
CN(c1ncccc1Nc1cccn2nc(Nc3ccc(cc3)C3CCN(C)CC3)nc12)S(C)(=O)=O
CN(c1ncccc1CNc1cccn2nc(Nc3ccc(cc3)S(C)(=O)=O)nc12)S(C)(=O)=O
CN(c1ncccc1CNc1cccn2nc(Nc3cccc(c3)S(C)(=O)=O)nc12)S(C)(=O)=O
CN(c1ncccc1CNc1cccn2nc(Nc3cccc(c3)N3CCN(C)CC3)nc12)S(C)(=O)=O
COc1cc(ccc1Nc1nc2c(NCc3cccnc3N(C)S(C)(=O)=O)cccn2n1)N1CCN(C)CC1
CN1CCN(CC1)c1ccc(Nc2nc3c(NCc4ccccc4S(C)(=O)=O)cccn3n2)cc1
CN1CCN(CC1)c1cccc(Nc2nc3c(NCc4ccccc4S(C)(=O)=O)cccn3n2)c1
CN1CCC(CC1)c1ccc(Nc2nc3c(NCc4ccccc4S(C)(=O)=O)cccn3n2)cc1
CS(=O)(=O)c1ccccc1CNc1cccn2nc(Nc3ccc(OCCN4CCCC4)cc3)nc12
C[C@H](O)CN1CCN(CC1)c1cccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)c1 |r|
C[C@@H](O)CN1CCN(CC1)c1cccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)c1 |r|
CC(C)(O)CN1CCN(CC1)c1cccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)c1
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3ccc4CCC(CCc4c3)N3CCOCC3)nc12
CN(c1ncccc1CNc1cccn2nc(Nc3ccc4N(C)C(=O)Cc4c3)nc12)S(C)(=O)=O
CN(c1ccccc1CNc1cccn2nc(Nc3ccc(cc3)N3CCN(C)CC3)nc12)S(C)(=O)=O
CN(c1ccccc1CNc1cccn2nc(Nc3cccc(c3)N3CCN(C)CC3)nc12)S(C)(=O)=O
CN(c1ccccc1CNc1cccn2nc(Nc3ccc(cc3)C3CCN(C)CC3)nc12)S(C)(=O)=O
CN(c1ccccc1CNc1cccn2nc(Nc3ccc(OCCN4CCCC4)cc3)nc12)S(C)(=O)=O
CN1CCN(CC1)c1ccc(Nc2nc3c(NCc4cccnc4)cccn3n2)cc1
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3cccc(c3)N3CCN(CCO)CC3)nc12
CN1CCN(CC1)c1cccc(Nc2nc3c(NCc4cccnc4)cccn3n2)c1
C(CN1CCCC1)Oc1ccc(Nc2nc3c(NCc4cccnc4)cccn3n2)cc1
CN(c1ncccc1CNc1cccn2nc(Nc3ccc(cc3)N3CCN(CCO)CC3)nc12)S(C)(=O)=O
CN(Cc1ccccc1CNc1cccn2nc(Nc3ccc(cc3)N3CCN(C)CC3)nc12)S(C)(=O)=O
CN(Cc1ccccc1CNc1cccn2nc(Nc3cccc(c3)N3CCN(C)CC3)nc12)S(C)(=O)=O
CN(Cc1ccccc1CNc1cccn2nc(Nc3ccc(OCCN4CCCC4)cc3)nc12)S(C)(=O)=O
CN(Cc1ccccc1CNc1cccn2nc(Nc3ccc(cc3)C3CCN(C)CC3)nc12)S(C)(=O)=O
CN1CCN(CC1)c1ccc(Nc2nc3c(NCc4cccc(c4)S(C)(=O)=O)cccn3n2)cc1
CN1CCN(CC1)c1cccc(Nc2nc3c(NCc4cccc(c4)S(C)(=O)=O)cccn3n2)c1
CN1CCC(CC1)c1ccc(Nc2nc3c(NCc4cccc(c4)S(C)(=O)=O)cccn3n2)cc1
CN1CCN(CC1)c1ccc(Nc2nc3c(NCC4CCN(C4)C(=O)OC(C)(C)C)cccn3n2)cc1
CN1CCN(CC1)c1ccc(Nc2nc3c(Nc4ccccc4CS(C)(=O)=O)cccn3n2)cc1
CN1CCC(CC1)c1ccc(Nc2nc3c(Nc4ccccc4CS(C)(=O)=O)cccn3n2)cc1
CN(c1ncccc1CNc1cccn2nc(Nc3ccc4CN(C)Cc4c3)nc12)S(C)(=O)=O
CN(c1ccccc1CNc1cccn2nc(Nc3ccc4CN(C)Cc4c3)nc12)S(C)(=O)=O
CN1Cc2ccc(Nc3nc4c(cccn4n3)-c3ccc(cc3)S(C)(=O)=O)cc2C1
CN(c1cccc(CNc2cccn3nc(Nc4ccc(cc4)N4CCN(C)CC4)nc23)c1)S(C)(=O)=O
CN1CCN(CC1)c1ccc(Nc2nc3c(NCC4CCCN4S(C)(=O)=O)cccn3n2)cc1
CN(Cc1ccccc1Nc1cccn2nc(Nc3ccc(cc3)N3CCN(C)CC3)nc12)S(C)(=O)=O
CN(Cc1ccccc1Nc1cccn2nc(Nc3cccc(c3)N3CCN(C)CC3)nc12)S(C)(=O)=O
CN(Cc1ccccc1Nc1cccn2nc(Nc3ccc(OCCN4CCCC4)cc3)nc12)S(C)(=O)=O
CN(Cc1ccccc1Nc1cccn2nc(Nc3ccc(cc3)C3CCN(C)CC3)nc12)S(C)(=O)=O
CN(Cc1cccc(c1)-c1cccn2nc(Nc3ccc(cc3)N3CCN(C)CC3)nc12)S(C)(=O)=O
CN(Cc1cccc(c1)-c1cccn2nc(Nc3cccc(c3)N3CCN(C)CC3)nc12)S(C)(=O)=O
CN(Cc1cccc(c1)-c1cccn2nc(Nc3ccc(OCCN4CCCC4)cc3)nc12)S(C)(=O)=O
CN(Cc1cccc(c1)-c1cccn2nc(Nc3ccc(cc3)C3CCN(C)CC3)nc12)S(C)(=O)=O
CC(C)(C)OC(=O)N1CCN(CC1)c1cccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)c1
CC(C)(C)OC(=O)N1CCC(CC1)c1cccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)c1
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3cccc(c3)N3CCNCC3)nc12
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3cccc(c3)C3CCNCC3)nc12
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3cccc(c3)N3CCN(CC(N)=O)CC3)nc12
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3cccc(c3)C3CCN(CC(N)=O)CC3)nc12
CN(Cc1ccccc1N(C)S(C)(=O)=O)c1cccn2nc(Nc3ccc(cc3)N3CCN(C)CC3)nc12
CC(C)(C)OC(=O)N1CC[C@H]([C@@H](O)C1)c1cccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)c1 |r|
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3cccc(c3)N3CCN(CCCF)CC3)nc12
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3cccc(c3)[C@@H]3CCNC[C@@H]3O)nc12 |r|
CN(c1ccccc1C#Cc1cccn2nc(Nc3ccc(cc3)N3CCN(C)CC3)nc12)S(C)(=O)=O
CS(=O)(=O)CCN1CCC(CC1)c1cccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)c1
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3cccc(c3)[C@@H]3CCN(CC(N)=O)C[C@@H]3O)nc12 |r|
CN(c1ccccc1C#Cc1cccn2nc(Nc3cccc(c3)N3CCN(C)CC3)nc12)S(C)(=O)=O
CN(c1ccccc1C#Cc1cccn2nc(Nc3ccc4CN(C)Cc4c3)nc12)S(C)(=O)=O
CN(c1ccccc1CCc1cccn2nc(Nc3ccc(cc3)N3CCN(C)CC3)nc12)S(C)(=O)=O
CN(c1ccccc1COc1cccn2nc(Nc3ccc(cc3)N3CCN(C)CC3)nc12)S(C)(=O)=O
CN(c1ccccc1\C=C\c1cccn2nc(Nc3ccc(cc3)N3CCN(C)CC3)nc12)S(C)(=O)=O
CC(Nc1cccn2nc(Nc3ccc(cc3)N3CCN(C)CC3)nc12)c1ccccc1N(C)S(C)(=O)=O
CN1CCN(CC1)c1cccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)P(C)(C)=O)c1
CP(C)(=O)c1ccc(cc1)-c1cccn2nc(nc12)N(CCS(C)(=O)=O)c1cccc(c1)C1CCN(CCS(C)(=O)=O)CC1
CN(c1ccccc1CNc1cccn2nc(Nc3ccc4CCC(CCc4c3)N3CCOCC3)nc12)S(C)(=O)=O
CN(c1ccccc1CNc1cccn2nc(Nc3ccc4cnccc4c3)nc12)S(C)(=O)=O
CN(c1ccccc1CNc1cccn2nc(Nc3ccccc3)nc12)S(C)(=O)=O
CP(C)(=O)c1ccc(cc1)-c1cccn2nc(Nc3cccc(c3)C3CCN(CCS(C)(=O)=O)CC3)nc12
CN1CCN(C(=O)C1)c1cccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)c1
CCN1CCN(C(=O)C1)c1cccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)c1
CN1CCN(CC1)C1CCN(CC1)c1ccc(cc1)-c1cccn2nc(Nc3cccc(c3)N3CCN(C)CC3)nc12
CN1CCN(C(=O)C1)c1cccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)P(C)(C)=O)c1
CCN1CCN(C(=O)C1)c1cccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)P(C)(C)=O)c1
CCn1cc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)cn1
Cc1nn(C)c(C)c1Nc1nc2c(cccn2n1)-c1ccc(cc1)S(C)(=O)=O
CCn1cc(Nc2nc3c(Oc4ccc(cc4)S(C)(=O)=O)cccn3n2)cn1
CC(C)(C)OC(=O)N1CCC(CC1)n1cc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)cn1
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3cnn(c3)C3CCNCC3)nc12
CN1CCN(CC1)c1cccc(Nc2nc3c(Oc4ccc(cc4)S(C)(=O)=O)cccn3n2)c1
CCn1cc(Nc2nc3c(cccn3n2)-c2ccc(cc2)C(F)(F)F)cn1
FC(F)(F)c1ccc(cc1)-c1cccn2nc(Nc3cnn(CCN4CCCC4)c3)nc12
CS(=O)(=O)c1ccc(Oc2cccn3nc(Nc4cnn(CCN5CCCC5)c4)nc23)cc1
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(Nc3cnn(CCN4CCCC4)c3)nc12
Oc1cccn2nc(Nc3ccc(cc3)C(F)(F)F)nc12
COCc1ccccc1-c1cccc2nc(Nc3ccc4CCN(CCc4c3)C(=O)OC(C)(C)C)nn12
C1CN(c2nc3cccc(N4CCCc5ccccc45)n3n2)c2ccccc2C1
COCc1ccccc1-c1cccc2nc(Nc3ccc4CCNCCc4c3)nn12
COCc1ccccc1-c1cccc2nc(Nc3ccc4CCN(CC(=O)N(C)C)CCc4c3)nn12
COCc1ccccc1-c1cccc2nc(Nc3ccc4CCN(CCS(C)(=O)=O)CCc4c3)nn12
COc1ccc(cc1-c1cccc2nc(Nc3ccc4CCNCCc4c3)nn12)C(F)(F)F
COc1ccc(cc1-c1cccc2nc(Nc3ccc4CCN(CCSC)CCc4c3)nn12)C(F)(F)F
COc1cc(ccc1-c1cccc2nc(Nc3ccc4CCNCCc4c3)nn12)C(F)(F)F
COc1ccc(cc1-c1cccc2nc(Nc3ccc4CCN(CC(=O)N(C)C)CCc4c3)nn12)C(F)(F)F
COc1cc(ccc1-c1cccc2nc(Nc3ccc4CCN(CCS(C)(=O)=O)CCc4c3)nn12)C(F)(F)F
CCOc1ccccc1-c1cccn2nc(Nc3ccc4CCN(CCc4c3)C(=O)OC(C)(C)C)nc12
CCOc1ccccc1-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12
CC(C)(C)OC(=O)N1CCc2ccc(Nc3nc4c(cccn4n3)-c3cccc4OC(F)(F)Oc34)cc2CC1
FC1(F)Oc2cccc(c2O1)-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12
CCOc1ccccc1-c1cccn2nc(Nc3ccc4CCN(CCS(C)(=O)=O)CCc4c3)nc12
CCOc1ccccc1-c1cccn2nc(Nc3ccc4CCN(CC(=O)N(C)C)CCc4c3)nc12
CS(=O)(=O)CCN1CCc2ccc(Nc3nc4c(cccn4n3)-c3cccc4OC(F)(F)Oc34)cc2CC1
CN(C)C(=O)CN1CCc2ccc(Nc3nc4c(cccn4n3)-c3cccc4OC(F)(F)Oc34)cc2CC1
COc1ccc(cc1-c1cccn2nc(Nc3ccc(cc3)N3CCN(C)CC3)nc12)C(F)(F)F
COc1ccc(cc1-c1cccn2nc(Nc3cccc(c3)N3CCN(C)CC3)nc12)C(F)(F)F
COc1ccc(cc1-c1cccn2nc(Nc3cccc(c3)C3CCN(CC3)C(=O)OC(C)(C)C)nc12)C(F)(F)F
COc1ccc(cc1-c1cccn2nc(Nc3cccc(c3)C3CCNCC3)nc12)C(F)(F)F
COc1ccc(cc1-c1cccn2nc(Nc3ccc(OCCN4CCOCC4)cc3)nc12)C(F)(F)F
COc1ccc(cc1-c1cccn2nc(Nc3ccc(OCCN4CCCC4)cc3)nc12)C(F)(F)F
CN1CCN(CC1)c1ccc(Nc2nc3c(OCc4cccc(Cl)c4)cccn3n2)cc1
CN1CCN(CC1)c1cccc(Nc2nc3c(OCc4cccc(Cl)c4)cccn3n2)c1
CN1CCN(CC1)c1ccc(Nc2nc3c(OCc4ccccc4C#N)cccn3n2)cc1
CN1CCN(CC1)c1cccc(Nc2nc3c(OCc4ccccc4C#N)cccn3n2)c1
CN1CCN(CC1)c1ccc(Nc2nc3c(O)cccn3n2)cc1
Cc1cccn2nc(Nc3ccc(cc3)S(C)(=O)=O)nc12
CN1CCN(CC1)c1cccc(Nc2nc3c(OCc4ccccc4C(N)=O)cccn3n2)c1
CC(=O)Nc1cccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)c1
CS(=O)(=O)CCN1CCc2ccc(Nc3nc4c(cccn4n3)-c3cc(ccc3Cl)C(F)(F)F)cc2CC1
CC(C)(C)OC(=O)N1CCc2ccc(Nc3nc4c(cccn4n3)-c3cc(ccc3F)C(F)(F)F)cc2CC1
Fc1ccc(cc1-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12)C(F)(F)F
COc1ncccc1-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC3)C(=O)OC(C)(C)C)nc12
COc1ncccc1-c1cccn2nc(Nc3ccc(cc3)C3CCNCC3)nc12
COc1ncccc1-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC(=O)N(C)C)CC3)nc12
COc1ncccc1-c1cccn2nc(Nc3ccc4ncccc4c3)nc12
CN(C)C(=O)CN1CCC(CC1)c1ccc(Nc2nc3c(cccn3n2)-c2ccc[nH]c2=O)cc1
O=c1[nH]cccc1-c1cccn2nc(Nc3ccc4ncccc4c3)nc12
COc1ncc(cc1-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC3)C(=O)OC(C)(C)C)nc12)C(F)(F)F
COc1ncc(cc1-c1cccn2nc(Nc3ccc(cc3)C3CCNCC3)nc12)C(F)(F)F
COc1ncc(cc1-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC(=O)N(C)C)CC3)nc12)C(F)(F)F
CC(C)(C)OC(=O)N1CCC(CC1)c1ccc(Nc2nc3c(cccn3n2)-c2cnn(c2)-c2ccc(F)cc2)cc1
CC(=O)Nc1ccc(Sc2cccn3nc(Nc4ccc(cc4)C4CCN(CC4)C(=O)OC(C)(C)C)nc23)cc1
Fc1ccc(cc1)-n1cc(cn1)-c1cccn2nc(Nc3ccc(cc3)C3CCNCC3)nc12
CN(C)C(=O)CN1CCC(CC1)c1ccc(Nc2nc3c(cccn3n2)-c2cnn(c2)-c2ccc(F)cc2)cc1
COc1cnc(cn1)-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC3)C(=O)OC(C)(C)C)nc12
COc1cnc(cn1)-c1cccn2nc(Nc3ccc(cc3)C3CCNCC3)nc12
COc1cnc(cn1)-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC(=O)N(C)C)CC3)nc12
Cc1ccc(cc1)-n1cc(cn1)-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC3)C(=O)OC(C)(C)C)nc12
CN1CCN(CC1)c1cccc(Nc2nc3c(cccn3n2)-c2cnn(c2)-c2ccc(F)cc2)c1
Cc1ccc(cc1)-n1cc(cn1)-c1cccn2nc(Nc3ccc(cc3)C3CCNCC3)nc12
COc1ccc(cc1Nc1cccn2nc(Nc3cccc(c3)N3CCN(C)CC3)nc12)C(F)(F)F
CC(C)COc1ccccc1-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12
CC(C)COc1cccc(c1)-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12
CC(C)COc1cc(C)ccc1-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12
CC(C)Oc1ccccc1-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12
C(Oc1ccccc1-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12)C1CC1
CC(C)COc1ccc(C)cc1-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12
CCCOc1ccc(Cl)cc1-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12
CCCOc1ccc(Cl)cc1-c1cccn2nc(Nc3ccc4CCN(CC(=O)N(C)C)CCc4c3)nc12
CCOc1ccc(Cl)cc1-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12
COc1ccccc1-c1cccn2nc(Nc3ccc4CCN(CC(=O)N(C)C)CCc4c3)nc12
COc1ccccc1-c1cccn2nc(Nc3ccc4CCN(CCS(C)(=O)=O)CCc4c3)nc12
COc1ccc(cc1-c1cccn2nc(Nc3ccc4CCN(CC(=O)N(C)C)CCc4c3)nc12)C(F)(F)F
CCOc1ccc(cc1-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12)C(F)(F)F
CCOc1ccc(cc1-c1cccn2nc(Nc3ccc4CCN(CCS(C)(=O)=O)CCc4c3)nc12)C(F)(F)F
CCOc1ccc(cc1-c1cccn2nc(Nc3ccc4CCN(CC(=O)N(C)C)CCc4c3)nc12)C(F)(F)F
COc1ccc(cc1-c1cccn2nc(Nc3ccc4CCN(CCS(C)(=O)=O)CCc4c3)nc12)C(F)(F)F
COc1ccc(F)cc1-c1cccn2nc(Nc3ccc4CCN(CC(=O)N(C)C)CCc4c3)nc12
COc1cc(F)ccc1-c1cccn2nc(Nc3ccc4CCN(CC(=O)N(C)C)CCc4c3)nc12
COc1cc(Cl)ccc1-c1cccn2nc(Nc3ccc4CCN(CC(=O)N(C)C)CCc4c3)nc12
CC(C)Oc1ccc(cc1-c1cccn2nc(Nc3ccc4CCN(CC(=O)N(C)C)CCc4c3)nc12)C(F)(F)F
CN(C)C(=O)CN1CCC(CC1)c1ccc(Nc2nc3c(cccn3n2)-c2cc(ccc2OCC(F)F)C(F)(F)F)cc1
FC(F)COc1ccc(cc1-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12)C(F)(F)F
CN(C)C(=O)CN1CCc2ccc(Nc3nc4c(cccn4n3)-c3cc(ccc3OCC(F)F)C(F)(F)F)cc2CC1
COc1cc(Cl)ccc1-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC(=O)N(C)C)CC3)nc12
COc1cc(Cl)ccc1-c1cccn2nc(Nc3ccc4CN(CC(=O)N(C)C)CCc4c3)nc12
COc1cc(Cl)ccc1-c1cccn2nc(Nc3cccc(c3)C3CCN(CC(=O)N(C)C)CC3)nc12
COc1ccc(cc1-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC3)C(=O)OC(C)(C)C)nc12)C(F)(F)F
COc1ccc(cc1-c1cccn2nc(Nc3ccc(cc3)C3CCNCC3)nc12)C(F)(F)F
COc1ccc(cc1-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC(=O)N(C)C)CC3)nc12)C(F)(F)F
COc1ccc(cc1-c1cccn2nc(Nc3ccc4CN(CCc4c3)C(=O)OC(C)(C)C)nc12)C(F)(F)F
COc1ccc(cc1-c1cccn2nc(Nc3ccc4CNCCc4c3)nc12)C(F)(F)F
COc1ccc(cc1-c1cccn2nc(Nc3ccc4CN(CC(=O)N(C)C)CCc4c3)nc12)C(F)(F)F
COc1cc(ccc1-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC3)C(=O)OC(C)(C)C)nc12)C(F)F
COc1cc(ccc1-c1cccn2nc(Nc3ccc(cc3)C3CCNCC3)nc12)C(F)F
COc1cc(ccc1-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC(=O)N(C)C)CC3)nc12)C(F)F
CC(C)(C)OC(=O)N1CCC(CC1)c1ccc(Nc2nc3c(cccn3n2)-c2ccc(F)cc2)cc1
Fc1ccc(cc1)-c1cccn2nc(Nc3ccc(cc3)C3CCNCC3)nc12
COc1cccc(c1)-c1cccn2nc(Nc3ccc4CNCc4c3)nc12
CN(C)C(=O)CN1CCC(CC1)c1ccc(Nc2nc3c(cccn3n2)-c2ccc(F)cc2)cc1
COc1cccc(c1)-c1cccn2nc(Nc3ccc(cc3)C3CCNCC3)nc12
COc1cccc(c1)-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC(=O)N(C)C)CC3)nc12
COc1cccc(c1F)-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC3)C(=O)OC(C)(C)C)nc12
COc1cccc(c1F)-c1cccn2nc(Nc3ccc(cc3)C3CCNCC3)nc12
COc1cccc(c1F)-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC(=O)N(C)C)CC3)nc12
COc1cccc(c1OC)-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC3)C(=O)OC(C)(C)C)nc12
COc1cccc(c1OC)-c1cccn2nc(Nc3ccc(cc3)C3CCNCC3)nc12
COc1cccc(c1OC)-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC(=O)N(C)C)CC3)nc12
CC(C)(C)OC(=O)N1CCC(CC1)c1ccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)C#N)cc1
N#Cc1ccc(cc1)-c1cccn2nc(Nc3ccc(cc3)C3CCNCC3)nc12
CN(C)C(=O)CN1CCC(CC1)c1ccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)C#N)cc1
COc1ccc(c(F)c1)-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC3)C(=O)OC(C)(C)C)nc12
COc1ccc(c(F)c1)-c1cccn2nc(Nc3ccc(cc3)C3CCNCC3)nc12
CN(C)c1cccc(c1)-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC3)C(=O)OC(C)(C)C)nc12
COc1ccc(c(F)c1)-c1cccn2nc(Nc3ccc(cc3)C3CCN(CC(=O)N(C)C)CC3)nc12
CN(C)c1cccc(c1)-c1cccn2nc(Nc3ccc(cc3)C3CCNCC3)nc12
CN(C)C(=O)CN1CCC(CC1)c1ccc(Nc2nc3c(cccn3n2)-c2cccc(c2)N(C)C)cc1
CN1CCN(CC1)c1cccc(Nc2nc3c(cccn3n2)-c2ccc(F)cc2)c1
FC(F)COc1ccccc1-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12
CN(C)C(=O)CN1CCc2ccc(Nc3nc4c(cccn4n3)-c3ccccc3OCC(F)F)cc2CC1
CS(=O)(=O)c1ccc(c(OCC(F)F)c1)-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12
CS(=O)(=O)c1ccc(OCC(F)F)c(c1)-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12
CN(C)C(=O)CN1CCc2ccc(Nc3nc4c(cccn4n3)-c3cc(ccc3OCC(F)F)S(C)(=O)=O)cc2CC1
FC(F)(F)c1cccc(c1)-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12
FC(F)COc1ccc(Cl)cc1-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12
CN(C)C(=O)CN1CCc2ccc(Nc3nc4c(cccn4n3)-c3cc(F)ccc3OCC(F)F)cc2CC1
CC(C)COc1ccc(cc1-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12)C(F)(F)F
CC(C)COc1ccc(cc1-c1cccn2nc(Nc3ccc4CCN(CC(=O)N(C)C)CCc4c3)nc12)C(F)(F)F
CN(C)C(=O)CN1CCc2ccc(Nc3nc4c(cccn4n3)-c3cc(Cl)ccc3OCC(F)F)cc2CC1
FC(F)COc1ccc(cc1-c1cccn2nc(Nc3ccc4CCNCCc4c3)nc12)C(F)F
CN(C)C(=O)CN1CCc2ccc(Nc3nc4c(cccn4n3)-c3cc(ccc3OCC(F)F)C(F)F)cc2CC1
CN1CCN(CC1)c1cncc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)n1
COc1ccccc1CNc1cccn2nc(Nc3ccc(cc3)N3CCN(C)CC3)nc12
COc1ccccc1CNc1cccn2nc(Nc3cccc(c3)N3CCN(C)CC3)nc12
CN(c1ccccc1CNc1cccn2nc(Nc3cncc(n3)N3CCN(C)CC3)nc12)S(C)(=O)=O
COc1cccc(CNc2cccn3nc(Nc4ccc(cc4)N4CCN(C)CC4)nc23)c1
COc1ccc(CNc2cccn3nc(Nc4ccc(cc4)N4CCN(C)CC4)nc23)cc1
COc1cccc(CNc2cccn3nc(Nc4cccc(c4)N4CCN(C)CC4)nc23)c1
COc1ccc(CNc2cccn3nc(Nc4cccc(c4)N4CCN(C)CC4)nc23)cc1
COc1cccc(CNc2cccn3nc(Nc4ccc(OC)nc4)nc23)c1
CN1CCN(CC1)c1cccc(Nc2nc3c(NCc4ccccc4F)cccn3n2)c1
CN1CCN(CC1)c1cccc(Nc2nc3c(NCc4ccc(F)cc4)cccn3n2)c1
COc1cccc(CNc2cccn3nc(Nc4ccnc(C)c4)nc23)c1
COc1cccc(CNc2cccn3nc(Nc4cccnc4)nc23)c1
COc1cccc(CNc2cccn3nc(Nc4ccncc4)nc23)c1
COc1ccccc1CNc1cccn2nc(Nc3cccnc3)nc12
COc1ccccc1CNc1cccn2nc(Nc3ccncc3)nc12
COc1ccc(Nc2nc3c(NCc4ccccc4OC)cccn3n2)cn1
COc1ccccc1CNc1cccn2nc(Nc3ccc(C)nc3)nc12
COc1ccccc1CNc1cccn2nc(Nc3ccnc(C)c3)nc12
COc1cccc(CNc2cccn3nc(Nc4ccc(C)nc4)nc23)c1
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(NCCc3ccccn3)nc12
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(NCCc3cccnc3)nc12
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(NCc3cccnc3)nc12
CS(=O)(=O)c1ccc(cc1)-c1cccn2nc(NCc3ccccn3)nc12
COc1ccc(cc1-c1cccn2nc(Nc3cccc(c3)C3CCN(CC(=O)N(C)C)CC3)nc12)C(F)(F)F
CCN1CCP(=O)(CC1)c1ccc(Nc2nc3c(cccn3n2)-c2ccc(cc2)S(C)(=O)=O)cc1
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4cccc(NS(C)(=O)=O)c4)c3n2)cn1
Cc1ccc(Nc2ncc3scc(-c4cccc(NS(C)(=O)=O)c4)c3n2)cn1
CS(=O)(=O)Nc1cccc(c1)-c1csc2cnc(Nc3ccc(nc3)N3CCOCC3)nc12
CN(C)CCOc1ccc(Nc2ncc3scc(-c4cccc(NS(C)(=O)=O)c4)c3n2)cn1
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4cccc(c4)C(=O)NC4CC4)c3n2)cn1
Cc1ccc(Nc2ncc3scc(-c4cccc(c4)C(=O)NC4CC4)c3n2)cn1
O=C(NC1CC1)c1cccc(c1)-c1csc2cnc(Nc3ccc(nc3)N3CCOCC3)nc12
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4cnc5ccccc5c4)c3n2)cn1
COc1cc(ccc1Nc1ncc(c(Oc2cccc3C(C)CCc23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2cccc3C(C)CCc23)n1)C(F)(F)F
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2ccccc2)n1)C(F)(F)F
COC(=O)c1ccccc1Oc1nc(Nc2cc(F)c(cc2OC)C(=O)NC2CCN(C)CC2)ncc1C(F)(F)F
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2ccccc2C(N)=O)n1)C(F)(F)F
COc1cc(ccc1Nc1ncc(c(Oc2ccc(cc2)C(O)=O)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2ccc(cc2)C(N)=O)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2cccc(c2)C(C)=O)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2cccnc2)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COC(=O)c1ccccc1Oc1nc(Nc2ccc(cc2OC)C(=O)NC2CCN(C)CC2)ncc1C(F)(F)F
COc1cc(ccc1Nc1ncc(c(Oc2cccc(c2)C(N)=O)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2cccc(CC(N)=O)c2)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2ccc(CC(O)=O)cc2)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2cccc(Cl)c2)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2ccccc2Cl)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2ccccc2CC(N)=O)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
CNC(=O)Cc1ccccc1Oc1nc(Nc2ccc(cc2OC)C(=O)NC2CCN(C)CC2)ncc1C(F)(F)F
COc1cc(ccc1Nc1ncc(c(Oc2ccccc2CC(=O)N(C)C)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2ccc(cc2)S(C)(=O)=O)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2cccc3[nH]ccc23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2cccc3nc[nH]c23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2ccc3[nH]cnc3c2)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
CNC(=O)c1cccc(Oc2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2C(F)(F)F)c1
COc1cc(ccc1Nc1ncc(c(Oc2cccc(c2)C(=O)N(C)C)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
CNC(=O)Cc1cccc(Oc2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2C(F)(F)F)c1
COc1cc(ccc1Nc1ncc(c(Oc2cccc(CC(=O)N(C)C)c2)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2ccc(CC(N)=O)cc2)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
CNC(=O)Cc1ccc(Oc2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2C(F)(F)F)cc1
COc1cc(ccc1Nc1ncc(c(Oc2ccc(CC(=O)N(C)C)cc2)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2ccccc2C(=O)N(C)C)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
CNC(=O)c1ccc(Oc2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2C(F)(F)F)cc1
COc1cc(ccc1Nc1ncc(c(Oc2ccc(cc2)C(=O)N(C)C)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2ccccc2C(C)=O)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2cccc(F)c2C(C)=O)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2ccccc2-c2cc[nH]n2)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2ccccc2-c2csnn2)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2ccc(Br)cc2C#N)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2cc(Br)ccc2C#N)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2cccc(Cl)c2C#N)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2cccc(F)c2C#N)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1ccc(C#N)c(Oc2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2C(F)(F)F)c1
COc1cc(ccc1Nc1ncc(c(Oc2ccc(Cl)cc2C#N)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2cccc3NC(=O)Cc23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2cccc3NC(=O)Cc23)n1)C(F)(F)F
COc1cc(ccc1Nc1ncc(c(Oc2ccccc2C#N)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2ccccc2C#N)n1)C(F)(F)F
COc1cc(ccc1Nc1ncc(c(Sc2ccccc2)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Sc2ccccc2)n1)C(F)(F)F
FC(F)(F)c1cnc(Nc2ccc(cc2)C(=O)NCc2ccccc2)nc1OCCN1CCCC1=O
FC(F)(F)C(=O)NCCCOc1nc(Nc2ccc(cc2)C(=O)NCc2ccccc2)ncc1C(F)(F)F
CCCNC(=O)c1ccc(Nc2ncc(c(OCCCNC(=O)C(F)(F)F)n2)C(F)(F)F)cc1
COc1cccc(COc2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2C(F)(F)F)c1
COc1cc(ccc1Nc1ncc(c(OCCN2CCCC2=O)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(OCC2CCCO2)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(OCC2CCCCN2C)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(OC2CCCN(C)C2)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1ccc(OC)c(CCOc2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2C(F)(F)F)c1
COc1cc(ccc1Nc1ncc(c(OCc2cccc(OC)c2OC)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(OCC2CCCCO2)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(OCC2CCCCC2)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COC(=O)COc1nc(Nc2ccc(cc2OC)C(=O)NC2CCN(C)CC2)ncc1C(F)(F)F
COc1cc(ccc1Nc1ncc(c(Oc2ccccc2-c2cncs2)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1ncc(s1)-c1ccccc1Oc1nc(Nc2ccc(cc2OC)C(=O)NC2CCN(C)CC2)ncc1C(F)(F)F
COc1cc(ccc1Nc1ncc(c(Oc2ccccc2-c2ccon2)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2cc(C)ccc2C#N)n1)C(F)(F)F
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2cccc(C)c2C#N)n1)C(F)(F)F
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)N(C)c23)n1)C(F)(F)F)C(O)=O
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)N(C)c23)n1)C(F)(F)F)C(=O)NCCN(C)C
COc1cc(ccc1Nc1ncc(c(Oc2ccccc2NS(C)(=O)=O)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2cccc3NS(=O)(=O)Cc23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2ccccc2N(C)S(C)(=O)=O)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
CCN(c1ccccc1Oc1nc(Nc2ccc(cc2OC)C(=O)NC2CCN(C)CC2)ncc1C(F)(F)F)S(C)(=O)=O
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2ccccc2N(C)S(C)(=O)=O)n1)C(F)(F)F
CCN(c1ccccc1Oc1nc(Nc2cc(F)c(cc2OC)C(=O)NC2CCN(C)CC2)ncc1C(F)(F)F)S(C)(=O)=O
COc1cc(ccc1Nc1ncc(c(Oc2c(Cl)cccc2NS(C)(=O)=O)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2ccc(Cl)cc2NS(C)(=O)=O)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2cc(F)ccc2NS(C)(=O)=O)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2cc(C)ccc2NS(C)(=O)=O)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2cccc3NS(=O)(=O)Cc23)n1)C(F)(F)F
COc1cc(ccc1Nc1ncc(c(Oc2cccc(C)c2N(C)C(C)=O)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2cccc3COC(=O)c23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2cccc3COC(=O)c23)n1)C(F)(F)F
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)N[C@H]1CCN(C)C[C@H]1F |r|
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)N[C@@H]1CCN(C)C[C@@H]1F |r|
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)N[C@@H]1CCN(C)C[C@H]1F |r|
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)N[C@H]1CCN(C)C[C@@H]1F |r|
COc1cc(C(=O)N[C@@H]2CCN(C)C[C@@H]2F)c(F)cc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F |r|
COc1cc(C(=O)N[C@H]2CCN(C)C[C@H]2F)c(F)cc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F |r|
COc1cc(C(=O)N[C@@H]2CCN(C)C[C@H]2F)c(F)cc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F |r|
COc1cc(C(=O)N[C@H]2CCN(C)C[C@@H]2F)c(F)cc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F |r|
COc1cc(ccc1Nc1ncc(c(Oc2ccc(Cl)c3C(C)CC(=O)c23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2ccc(Cl)c3C(C)CC(=O)c23)n1)C(F)(F)F
COc1cc(C(=O)NC2CCN(C)CC2)c(Cl)cc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F
COc1cc(C(=O)N[C@@H]2CCN(C)C2)c(Cl)cc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F |r|
COc1cc(C(=O)N[C@H]2CCN(C)C2)c(Cl)cc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F |r|
COc1cc(C(=O)NC2CCN(C)CC2)c(Cl)cc1Nc1ncc(c(Oc2ccc(C)c3CCC(=O)c23)n1)C(F)(F)F
COc1cc(C(=O)N[C@@H]2CCN(C)C2)c(Cl)cc1Nc1ncc(c(Oc2ccc(C)c3CCC(=O)c23)n1)C(F)(F)F |r|
COc1cc(C(=O)N[C@H]2CCN(C)C2)c(Cl)cc1Nc1ncc(c(Oc2ccc(C)c3CCC(=O)c23)n1)C(F)(F)F |r|
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)NC1CCN(CC1)C1CCOCC1
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)NC(C)(C)C
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)NC1CCOCC1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)NC1CC[C@H](O)CC1 |r,wD:36.40,(1.43,-4.23,;1.43,-2.69,;.09,-1.93,;-1.24,-2.69,;-2.57,-1.93,;-2.57,-.38,;-1.24,.38,;.09,-.38,;1.43,.38,;1.43,1.93,;.09,2.69,;.09,4.23,;1.43,5,;2.76,4.23,;4.1,5,;5.43,4.23,;5.43,2.69,;6.76,1.93,;8.1,2.69,;8.1,4.23,;9.24,5.27,;8.61,6.67,;7.08,6.51,;5.75,7.28,;6.76,5,;2.76,2.69,;1.43,6.54,;.09,7.31,;2.76,7.31,;2.76,5.78,;-3.91,-2.69,;-5.24,-1.93,;-3.91,-4.23,;-5.24,-5,;-5.24,-6.54,;-6.57,-7.31,;-7.91,-6.54,;-9.24,-7.31,;-7.91,-5,;-6.57,-4.23,)|
Fc1c2CC(=O)Nc2ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F
FC(F)(F)c1cnc(Nc2ccc3NC(=O)Cc3c2)nc1Oc1cccc2CCC(=O)c12
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)-n1ccnn1
COc1cc(ccc1Nc1ncc(c(Oc2cccc3C(C)N(CCF)C(=O)c23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(c(Oc2cccc3COC(=O)c23)n1)C(F)(F)F)C(=O)NC1CCOCC1
FC(F)(F)c1cnc(Nc2ccc3NC(=O)Cc3c2)nc1Oc1cccc2COC(=O)c12
Fc1c2CC(=O)Nc2ccc1Nc1ncc(c(Oc2cccc3COC(=O)c23)n1)C(F)(F)F
COc1cc(ccc1Nc1ncc(c(Oc2cccc3[C@H](C)N(CCF)C(=O)c23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1 |r|
COc1cc(ccc1Nc1ncc(c(Oc2cccc3[C@@H](C)N(CCF)C(=O)c23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1 |r|
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2cccc3[C@H](C)N(CCF)C(=O)c23)n1)C(F)(F)F |r|
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2cccc3[C@@H](C)N(CCF)C(=O)c23)n1)C(F)(F)F |r|
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
CON1Cc2cccc(Oc3nc(Nc4ccc(cc4OC)C(=O)NC4CCN(C)CC4)ncc3C(F)(F)F)c2C1=O
COc1cc(ccc1Nc1ncc(c(Oc2ccc(C)c3CCC(=O)c23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2ccc(C)c3CCC(=O)c23)n1)C(F)(F)F
CC[C@H]1COc2cccc(Oc3nc(Nc4ccc(cc4OC)C(=O)NC4CCN(C)CC4)ncc3C(F)(F)F)c2C(=O)N1 |r|
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)NC1CCN(CC1)c1ncccn1
COc1cc(C(=O)N[C@H]2CCN(C)C[C@H]2F)c(Cl)cc1Nc1ncc(Cl)c(Oc2cccc3C(C)C(C)C(=O)c23)n1 |r|
CCc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)NC
CCc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)NOC
COc1cc(C(=O)N[C@H]2CCN(C)C[C@H]2F)c(Cl)cc1Nc1ncc(Cl)c(Oc2cccc3[C@H](C)N(C)C(=O)c23)n1 |r|
COc1cc(ccc1Nc1ncc(c(Oc2cccc3OC(C)(C)C(=O)c23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2cccc3OC(C)(C)C(=O)c23)n1)C(F)(F)F
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(O)=O
Cc1nc2ccc(Nc3ncc(c(Oc4cccc5CCC(=O)c45)n3)C(F)(F)F)cc2n1C
CCc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)N(C)C
CCc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
CCN1CCC(CC1)NC(=O)c1ccc(Nc2ncc(c(Oc3cccc4CCC(=O)c34)n2)C(F)(F)F)c(CC)c1
CCc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)NC1CCN(CC1)C(C)C
CCc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)N[C@H]1CC[C@@H](CC1)N1CCOCC1 |r,wU:33.36,wD:36.43,(4.1,-.77,;2.76,-1.54,;1.43,-.77,;.09,-1.54,;-1.24,-.77,;-1.24,.77,;.09,1.54,;1.43,.77,;2.76,1.54,;2.76,3.08,;1.43,3.85,;1.43,5.39,;2.76,6.16,;4.1,5.39,;5.43,6.16,;6.76,5.39,;6.76,3.85,;8.1,3.08,;9.43,3.85,;9.43,5.39,;10.57,6.42,;9.95,7.83,;8.42,7.67,;7.08,8.44,;8.1,6.16,;4.1,3.85,;2.76,7.7,;1.43,8.47,;4.1,8.47,;4.1,6.93,;-2.57,-1.54,;-3.91,-.77,;-2.57,-3.08,;-3.91,-3.85,;-3.91,-5.39,;-5.24,-6.16,;-6.57,-5.39,;-6.57,-3.85,;-5.24,-3.08,;-7.91,-6.16,;-9.24,-5.39,;-10.57,-6.16,;-10.57,-7.7,;-9.24,-8.47,;-7.91,-7.7,)|
CCc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)NC1CCCN(C)C1
CCN1Cc2cccc(Oc3nc(Nc4ccc(cc4OC)C(=O)NC4CCN(C)CC4)ncc3C(F)(F)F)c2C1=O
OC(=O)c1ccc(Nc2ncc(c(Oc3cccc4CCC(=O)c34)n2)C(F)(F)F)cc1
CCN1CCC(CC1)NC(=O)c1cc(OC)c(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)cc1Cl
CCN1CCC(CC1)NC(=O)c1ccc(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)c(OC)c1
COc1cc(C(=O)N[C@H]2CCN(C)C[C@H]2F)c(Cl)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F |r|
COc1cc(C(=O)N[C@@H]2CCN(C)C[C@@H]2F)c(Cl)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F |r|
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F)C(=O)N[C@@H]1CCN(C)C[C@@H]1F |r|
COc1cc(C(=O)N[C@H]2CCN(C)C[C@H]2F)c(F)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F |r|
COc1cc(C(=O)N[C@@H]2CCN(C)C[C@@H]2F)c(F)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F |r|
CCN1CCC(CC1)NC(=O)c1cc(OC)c(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)cc1F
COc1cc(C(=O)NC2CCN(C)CC2)c(Cl)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F)C(=O)N[C@H]1CCN(C)C[C@H]1F |r|
COc1cc(ccc1Nc1nccc(Oc2cccc3CCC(=O)c23)n1)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(F)c(Oc2cccc3CCC(=O)c23)n1)C(=O)NC1CCN(C)CC1
COc1ccc(Nc2ncc(F)c(Oc3cccc4CCC(=O)c34)n2)c(OC)c1
COc1ccc(Nc2ncc(F)c(Oc3cccc4CCC(=O)c34)n2)cc1
COc1ccc(Nc2nccc(Oc3cccc4CCC(=O)c34)n2)c(OC)c1
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CCN(C)C(=O)c23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(Br)c(Oc2cccc3CCC(=O)c23)n1)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(Cl)c(Oc2cccc3CN(C)C(=O)c23)n1)C(=O)NC1CCN(C)CC1
COc1ccc(Nc2nccc(Oc3cccc4CCC(=O)c34)n2)cc1
COc1cc(F)ccc1Nc1nccc(Oc2cccc3CCC(=O)c23)n1
CON1Cc2cccc(Oc3nc(Nc4cc(F)c(cc4OC)C(=O)NC4CCN(C)CC4)ncc3Cl)c2C1=O
COc1cc(ccc1Nc1ncc(C(C)C)c(Oc2cccc3CCC(=O)c23)n1)C(=O)NC1CCN(C)CC1
COc1cc(ccc1Nc1ncc(Cl)c(Oc2cccc3CCC(=O)c23)n1)N1CCN(C)CC1
COc1cc(C(=O)OCc2ccccc2)c(Cl)cc1Nc1ncc(Cl)c(Oc2cccc3CN(C)C(=O)c23)n1
COc1ccc(Nc2ncc(C(C)C)c(Oc3cccc4CCC(=O)c34)n2)c(OC)c1
COc1ccc(Nc2ncc(C(C)C)c(Oc3cccc4CCC(=O)c34)n2)cc1
COc1ccc(Nc2ncc(C(C)=O)c(Oc3cccc4CCC(=O)c34)n2)cc1
COc1cc(ccc1Nc1ncc(c(Oc2cccc3C(C)N(C)C(=O)c23)n1)C(F)(F)F)C(=O)N[C@H]1CCN(C)C[C@H]1F |r,w:20.22|
COc1cc(ccc1Nc1ncc(Cl)c(Oc2cccc3C(C)N(C)C(=O)c23)n1)N1CCN(C)CC1
COc1cc(O[C@@H]2CO[C@@H]3[C@H](O)CO[C@H]23)ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F |r|
COc1cc(C(=O)NC2CCN(C)CC2)c(Cl)cc1Nc1ncc(Cl)c(Oc2cccc3CN(C)C(=O)c23)n1
COc1cc(CN(C)C)ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F
COc1cc(CN2CCCC2)ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F
COc1cc(ccc1Nc1nccc(Oc2cccc3CCC(=O)c23)n1)N1CCN(C)CC1
COc1cc(ccc1Nc1ncc(F)c(Oc2cccc3CCC(=O)c23)n1)N1CCN(C)CC1
COc1cc(O[C@H]2CCOC2)ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F |r|
CN1Cc2cccc(Oc3nc(Nc4ccc(O[C@H]5CCOC5)cc4)ncc3C(F)(F)F)c2C1=O |r|
CN1Cc2cccc(Oc3nc(Nc4ccc(OC5CCOCC5)cc4)ncc3C(F)(F)F)c2C1=O
COc1cc(OC2CCOCC2)ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F)N1CCN(C)CC1
CN1Cc2cccc(Oc3nc(Nc4ccc(NC5CCN(C)CC5)c(F)c4)ncc3C(F)(F)F)c2C1=O
COc1cc(ccc1Nc1nccc(Oc2cccc3CN(C)C(=O)c23)n1)C(O)=O
COc1cc(ccc1Nc1ncc(c(Oc2cccc3C(C)N(C)C(=O)c23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1 |w:20.22|
COc1cc(O[C@@H]2CO[C@@H]3[C@H](O)CO[C@H]23)ccc1Nc1ncc(c(Oc2cccc3C(C)N(C)C(=O)c23)n1)C(F)(F)F |r,w:30.34|
COc1ccc(Nc2ncc(C#N)c(Oc3cccc4CCC(=O)c34)n2)cc1
COc1cc(ccc1Nc1ncc(Br)c(Oc2cccc3CN(C)C(=O)c23)n1)C(=O)OCc1ccccc1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3CN(C)C(=O)c23)n1
COc1cc(ccc1Nc1nccc(Oc2cccc3CN(C)C(=O)c23)n1)C(=O)NC1CCN(C)CC1
COc1cc(F)ccc1Nc1ncc(F)c(Oc2cccc3CCC(=O)c23)n1
COc1cc(C(=O)NC2CCN(C)CC2)c(Cl)cc1Nc1ncc(c(Oc2cccc3C(C)N(C)C(=O)c23)n1)C(F)(F)F |w:31.34|
COc1cc(ccc1Nc1ncc(C#N)c(Oc2cccc3CCC(=O)c23)n1)N1CCN(C)CC1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(C#N)c(Oc2cccc3CCC(=O)c23)n1
COc1cc(C(=O)NC2CCN(C)CC2)c(Cl)cc1Nc1ncc(C#N)c(Oc2cccc3CCC(=O)c23)n1
CON1Cc2cccc(Oc3nc(Nc4cc(F)c(cc4OC)C(=O)NC4CCN(C)CC4)ncc3C(F)(F)F)c2C1=O
CON1Cc2cccc(Oc3nc(Nc4cc(F)c(cc4OC)C(=O)N[C@@H]4CCCN(C)C4)ncc3C(F)(F)F)c2C1=O |r|
CON1Cc2cccc(Oc3nc(Nc4ccc(cc4OC)C(=O)N[C@@H]4CCCN(C)C4)ncc3C(F)(F)F)c2C1=O |r|
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2cccc3c2C(=O)N(C)C3(C)C)n1)C(F)(F)F
CO[C@H]1CN(C)CC[C@H]1NC(=O)c1cc(OC)c(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)cc1F |r|
COc1cc(C(=O)N[C@H]2CCN(C)C[C@H]2F)c(Cl)cc1Nc1ncc(c(Oc2cccc3c2C(=O)N(C)C3(C)C)n1)C(F)(F)F |r|
CO[C@H]1CN(C)CC[C@H]1NC(=O)c1cc(OC)c(Nc2ncc(c(Oc3cccc4c3C(=O)N(C)C4(C)C)n2)C(F)(F)F)cc1Cl |r|
COc1cc(C(=O)NCC(C)(C)CN(C)C)c(F)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F
COc1cc(C(=O)NC2CCOC2)c(F)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F
COc1cc(C(=O)NC[C@@H]2CCCO2)c(F)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F |r|
COc1cc(C(=O)NCCN(C)C)c(F)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F
COc1cc(C(=O)N[C@H]2CC[C@H](O)CC2)c(F)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F |r,wU:11.11,wD:8.7,(-6.62,4.23,;-6.62,2.69,;-5.29,1.92,;-5.29,.38,;-3.96,-.39,;-3.96,-1.93,;-2.62,-2.7,;-5.29,-2.7,;-5.29,-4.24,;-6.62,-5.01,;-6.62,-6.55,;-5.29,-7.32,;-5.29,-8.86,;-3.96,-6.55,;-3.96,-5.01,;-2.62,.38,;-1.29,-.39,;-2.62,1.92,;-3.96,2.69,;-3.96,4.23,;-2.62,5,;-2.62,6.54,;-1.29,7.31,;.05,6.54,;.05,5,;1.38,4.23,;1.38,2.69,;.05,1.92,;.05,.38,;1.38,-.39,;2.71,.38,;4.18,-.09,;5.08,1.15,;6.62,1.15,;4.18,2.4,;4.95,3.73,;2.71,1.92,;-1.29,4.24,;1.38,7.32,;2.71,6.55,;1.38,8.86,;1.78,5.83,)|
COc1cc(C(=O)NC2CCN(CC2)C2CC2)c(F)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F
COc1cc(C(=O)NC[C@H](O)CO)c(F)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F |r|
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3CCC(=O)c23)n1
COc1cc(C(=O)N[C@H]2CCCN(C)C2)c(Cl)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F |r|
COc1cc(C(=O)N[C@H]2CCN(C)C[C@H]2F)c(Cl)cc1Nc1ncc(Cl)c(Oc2cccc3CN(C)C(=O)c23)n1 |r|
CO[C@H]1CN(C)CC[C@H]1NC(=O)c1cc(OC)c(Nc2ncc(Cl)c(Oc3cccc4CN(C)C(=O)c34)n2)cc1Cl |r|
COc1cc(C(=O)NC2CCN(CC2)C2CCOCC2)c(Cl)cc1Nc1ncc(Cl)c(Oc2cccc3CN(C)C(=O)c23)n1
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F)N1CCN(CC2CC2)CC1
COc1cc(OC2CCN(C)C2)c(F)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F
COc1cc(C(=O)NC2CCCN(C)C2)c(C)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F
COc1cc(C(=O)N[C@@H]2CCCN(C)C2)c(C)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F |r|
COc1cc(C(=O)N[C@H]2CCCN(C)C2)c(C)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F |r|
COc1cc(C(=O)NCCN(C)C)c(C)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F
COc1cc(C(=O)N(C)C)c(C)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F
CNC(=O)c1cc(OC)c(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)cc1C
COc1cc(C(=O)NC2CCN(C)CC2)c(C)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F
COc1cc(C(=O)NC2CCN(C)CC2)c(C)cc1Nc1ncc(Cl)c(Oc2cccc3CN(C)C(=O)c23)n1
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F)C(=O)NC1CCOCC1
COc1cc(C(=O)NC2CCN(C)CC2)c(Cl)cc1Nc1ncc(Cl)c(Oc2cccc3[C@H](C)N(C)C(=O)c23)n1 |r|
COc1cc(C(=O)NC2CCN(C)CC2)c(Cl)cc1Nc1ncc(Cl)c(Oc2cccc3[C@@H](C)N(C)C(=O)c23)n1 |r|
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3[C@H](C)N(C)C(=O)c23)n1 |r|
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3[C@@H](C)N(C)C(=O)c23)n1 |r|
COc1cc(C(=O)NC2CCN(CC2)C2CCOCC2)c(C)cc1Nc1ncc(Cl)c(Oc2cccc3CN(C)C(=O)c23)n1
COc1cc(C(=O)N[C@H]2CC[C@@H](CC2)N2CCN(CC3CC3)CC2)c(C)cc1Nc1ncc(Cl)c(Oc2cccc3CN(C)C(=O)c23)n1 |r,wU:8.7,wD:11.14,(-5.85,8.37,;-5.85,6.83,;-4.52,6.06,;-4.52,4.52,;-3.19,3.75,;-3.19,2.21,;-1.85,1.44,;-4.52,1.44,;-4.52,-.1,;-3.19,-.87,;-3.19,-2.41,;-4.52,-3.18,;-5.85,-2.41,;-5.85,-.87,;-4.52,-4.72,;-5.85,-5.49,;-5.85,-7.03,;-4.52,-7.8,;-4.52,-9.34,;-5.85,-10.11,;-7.39,-10.11,;-6.62,-11.45,;-3.19,-7.03,;-3.19,-5.49,;-1.85,4.52,;-.52,3.75,;-1.85,6.06,;-3.19,6.83,;-3.19,8.37,;-1.85,9.14,;-1.85,10.68,;-.52,11.45,;.82,10.68,;2.15,11.45,;.82,9.14,;2.15,8.37,;2.15,6.83,;.82,6.06,;.82,4.52,;2.15,3.75,;3.48,4.52,;4.95,4.04,;5.85,5.29,;7.39,5.29,;4.95,6.53,;5.72,7.87,;3.48,6.06,;-.52,8.37,)|
COc1cc(C(=O)NCC2CC2)c(C)cc1Nc1ncc(Cl)c(Oc2cccc3CN(C)C(=O)c23)n1
CO[C@@H]1CN(C)CC[C@@H]1NC(=O)c1cc(OC)c(Nc2ncc(Cl)c(Oc3cccc4[C@H](C)N(C)C(=O)c34)n2)cc1Cl |r|
COc1cc(C(=O)NCC2CCCO2)c(F)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F
COc1cc(C(=O)N[C@H]2CC[C@@H](CC2)N2CCN(CC3CC3)CC2)c(F)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F |r,wU:8.7,wD:11.14,(-5.85,7.6,;-5.85,6.06,;-4.52,5.29,;-4.52,3.75,;-3.19,2.98,;-3.19,1.44,;-1.85,.67,;-4.52,.67,;-4.52,-.87,;-3.19,-1.64,;-3.19,-3.18,;-4.52,-3.95,;-5.85,-3.18,;-5.85,-1.64,;-4.52,-5.49,;-5.85,-6.26,;-5.85,-7.8,;-4.52,-8.57,;-4.52,-10.11,;-5.85,-10.88,;-6.62,-12.22,;-7.39,-10.88,;-3.19,-7.8,;-3.19,-6.26,;-1.85,3.75,;-.52,2.98,;-1.85,5.29,;-3.19,6.06,;-3.19,7.6,;-1.85,8.37,;-1.85,9.91,;-.52,10.68,;.82,9.91,;.82,8.37,;2.15,7.6,;2.15,6.06,;.82,5.29,;.82,3.75,;2.15,2.98,;3.48,3.75,;4.95,3.27,;5.85,4.52,;7.39,4.52,;4.95,5.76,;5.72,7.1,;3.48,5.29,;-.52,7.6,;2.15,10.68,;2.15,12.22,;3.48,9.91,;2.55,9.19,)|
COc1cc(C(=O)NC2CCN(CC2)C2CCOCC2)c(F)cc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F
CON1Cc2cccc(Oc3nc(Nc4cc(F)c(cc4OC)C(=O)N[C@H]4CCN(C)C[C@H]4F)ncc3Cl)c2C1=O |r|
CO[C@H]1CN(C)CC[C@H]1NC(=O)c1cc(OC)c(Nc2ncc(Cl)c(Oc3cccc4CN(OC)C(=O)c34)n2)cc1F |r|
CO[C@H]1CN(C)CC[C@H]1NC(=O)c1cc(OC)c(Nc2ncc(Cl)c(Oc3cccc4[C@@H](C)N(C)C(=O)c34)n2)cc1Cl |r|
COc1cc(C(=O)N[C@H]2CCN(C)C[C@H]2F)c(Cl)cc1Nc1ncc(Cl)c(Oc2cccc3[C@@H](C)N(C)C(=O)c23)n1 |r|
CO[C@H]1CN(C)CC[C@H]1NC(=O)c1cc(OC)c(Nc2ncc(Cl)c(Oc3cccc4[C@H](C)N(C)C(=O)c34)n2)cc1F |r|
COc1cc(C(=O)N[C@H]2CCN(C)C[C@H]2F)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3[C@@H](C)N(C)C(=O)c23)n1 |r|
CO[C@H]1CN(C)CC[C@H]1NC(=O)c1cc(OC)c(Nc2ncc(Cl)c(Oc3cccc4[C@@H](C)N(C)C(=O)c34)n2)cc1F |r|
CCN1CC[C@H](NC(=O)c2cc(OC)c(Nc3ncc(Cl)c(Oc4cccc5[C@H](C)N(C)C(=O)c45)n3)cc2F)[C@H](F)C1 |r|
COc1cc(C(=O)N[C@H]2CCN(C[C@H]2F)C(C)C)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3[C@H](C)N(C)C(=O)c23)n1 |r|
COc1cc(C(=O)N[C@H]2CCN(C)C[C@H]2F)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3[C@H](C)N(C)C(=O)c23)n1 |r|
COc1cc(C(=O)N[C@@H]2CCN(C)C[C@@H]2F)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3CN(C)C(=O)c23)n1 |r|
CO[C@H]1CN(C)CC[C@H]1NC(=O)c1cc(OC)c(Nc2ncc(Cl)c(Oc3cccc4CN(C)C(=O)c34)n2)cc1F |r|
CO[C@H]1CN(C)CC[C@H]1NC(=O)c1cc(OC)c(Nc2ncc(Cl)c(Oc3cccc4CN(C)C(=O)c34)n2)cc1C |r|
COc1cc(C(=O)N[C@H]2CCN(C)C[C@H]2F)c(C)cc1Nc1ncc(Cl)c(Oc2cccc3CN(C)C(=O)c23)n1 |r|
CON1Cc2cccc(Oc3nc(Nc4cc(F)c(cc4OC)C(=O)NC4CCOCC4)ncc3C(F)(F)F)c2C1=O
CO[C@H]1CN(C)CC[C@H]1NC(=O)c1cc(OC)c(Nc2ncc(Cl)c(Oc3cccc4c3C(=O)N(C)C4(C)C)n2)cc1C |r|
COc1cc(C(=O)N[C@H]2CCN(C)C[C@H]2F)c(C)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C3(C)C)n1 |r|
COc1cc(ccc1Nc1ncc(c(Oc2cccc3OCCN(C)C(=O)c23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2cccc3OCCN(C)C(=O)c23)n1)C(F)(F)F
COc1cc(ccc1Nc1ncc(Cl)c(Oc2cccc3OC[C@H](C)NC(=O)c23)n1)C(=O)NC1CCN(C)CC1 |r|
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3OC[C@H](C)NC(=O)c23)n1 |r|
COc1cc(ccc1Nc1ncc(c(Oc2cccc3OCC(C)(C)NC(=O)c23)n1)C(F)(F)F)C(=O)NC1CCN(C)CC1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2cccc3OCC(C)(C)NC(=O)c23)n1)C(F)(F)F
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F)C(=O)NC1CCN(CCO)CC1
CONC(=O)c1ccc(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)c(OC)c1
CN1Cc2cccc(Oc3nc(Nc4ccc(cc4C)C(=O)NC4CCN(CC4)C(C)=O)ncc3C(F)(F)F)c2C1=O
COCCNC(=O)c1ccc(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)c(C)c1
CN1Cc2cccc(Oc3nc(Nc4ccc(cc4C)C(=O)NC4CCN(CCO)CC4)ncc3C(F)(F)F)c2C1=O
CN1Cc2cccc(Oc3nc(Nc4ccc(cc4C)C(=O)NC4CCC(F)(F)CC4)ncc3C(F)(F)F)c2C1=O
COCCN1CCC(CC1)NC(=O)c1ccc(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)c(C)c1
CNC(=O)c1ccc(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)c(C)c1
CNC(=O)c1ccc(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)c(OC)c1
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F)C(=O)NC1CCCCC1
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F)C(=O)NC1CCC(F)(F)CC1
COCCN1CCC(CC1)NC(=O)c1ccc(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)c(OC)c1
CN1Cc2cccc(Oc3nc(Nc4ccc(cc4C)C(=O)NC4CCCN(C)C4)ncc3C(F)(F)F)c2C1=O
CN1Cc2cccc(Oc3nc(Nc4ccc(cc4C)C(=O)NC4CCN(C)CC4)ncc3C(F)(F)F)c2C1=O
CONC(=O)c1ccc(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)c(C)c1
COCCNC(=O)c1ccc(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)c(OC)c1
COCCCNC(=O)c1ccc(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)c(OC)c1
COc1cc(CN(C)C)ccc1Nc1ncc(Cl)c(Oc2cccc3CN(C)C(=O)c23)n1
COc1cc(C[C@@H](O)CO)ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F |r|
COc1cc(C[C@H](O)CO)ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F |r|
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F)N1CCN(CC1)C(C)C
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F)N1CCN(CC(=O)N(C)C)CC1
CON(C)C(=O)CN1CCN(CC1)c1ccc(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)c(OC)c1
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F)N1CCN(CC1)C1COC1
CO[C@@H]1CN(C)CCC1NC(=O)c1cc(OC)c(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)cc1F |r|
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F)C#CC(=O)N(C)C
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(c(Oc2ccc(C)c3CN(C)C(=O)c23)n1)C(F)(F)F
CO[C@@H]1CN(C)CCC1NC(=O)c1ccc(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)c(OC)c1 |r|
CO[C@@H]1CN(C)CCC1NC(=O)c1cc(OC)c(Nc2ncc(Cl)c(Oc3cccc4c3C(=O)N(C)C4(C)C)n2)cc1C |r|
CO[C@H]1CN(C)CC[C@@H]1NC(=O)c1cc(OC)c(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)cc1F |r|
CO[C@H]1CN(C)CC[C@@H]1NC(=O)c1ccc(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)c(OC)c1 |r|
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F)C#CCN(C)C
CO[C@@H]1CN(C)CC[C@H]1NC(=O)c1cc(OC)c(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)cc1C |r|
CO[C@H]1CN(C)CC[C@@H]1NC(=O)c1cc(OC)c(Nc2ncc(c(Oc3cccc4CN(C)C(=O)c34)n2)C(F)(F)F)cc1C |r|
COc1cc(\C=C\C(=O)N(C)C)ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CN(C)C(=O)c23)n1)C(F)(F)F)C(\C)=C\C(=O)N(C)C
NC(=O)Cc1ccccc1CCc1nc(Nc2ccc(cc2)N2CCNCC2)ncc1C(F)(F)F
CN1CCN(CC1)c1ccc(Nc2ncc(c(CCc3cccc(c3)C(N)=O)n2)C(F)(F)F)cc1
CN1CCN(CC1)c1ccc(Nc2ncc(c(CCc3ccccc3CC(N)=O)n2)C(F)(F)F)cc1
NC(=O)Cc1ccccc1CCc1nc(Nc2ccc(cc2)C2CCCNC2)ncc1C(F)(F)F
CN1CCCC(C1)c1ccc(Nc2ncc(c(CCc3ccccc3CC(N)=O)n2)C(F)(F)F)cc1
CN1CCN(CC1)c1cccc(Nc2ncc(c(CCc3cccc(c3)C(N)=O)n2)C(F)(F)F)c1
NC(=O)Cc1ccccc1CCc1nc(Nc2ccc(cc2)C2CCCCN2)ncc1C(F)(F)F
CN1CCCCC1c1ccc(Nc2ncc(c(CCc3ccccc3CC(N)=O)n2)C(F)(F)F)cc1
CCN1CCN(CC1)c1ccc(Nc2ncc(c(CCc3ccccc3CC(N)=O)n2)C(F)(F)F)cc1
NC(=O)Cc1ccccc1CCc1nc(Nc2ccc(cc2)C2CCNCC2)ncc1C(F)(F)F
CC(C(N)=O)c1ccccc1CCc1nc(Nc2ccc(cc2)C2CCNCC2)ncc1C(F)(F)F
CC(=O)N1CCN(CC1)c1ccc(Nc2ncc(c(CCc3ccccc3CC(N)=O)n2)C(F)(F)F)cc1
CNC(=O)Cc1ccccc1CCc1nc(Nc2ccc(cc2)N2CCNCC2)ncc1C(F)(F)F
CN1CCC(CC1)c1ccc(Nc2ncc(c(CCc3ccccc3CC(N)=O)n2)C(F)(F)F)cc1
CN1CCN(CC1)c1cccc(Nc2ncc(c(CCc3ccccc3CC(N)=O)n2)C(F)(F)F)c1
CNC(=O)Cc1ccccc1CCc1nc(Nc2cccc(c2)N2CCN(C)CC2)ncc1C(F)(F)F
Cc1ccc(CCc2nc(Nc3ccc(cc3)N3CCNCC3)ncc2C(F)(F)F)cc1C(N)=O
NC1CCN(CC1)c1ccc(Nc2ncc(c(CCc3ccccc3CC(N)=O)n2)C(F)(F)F)cc1
NC(=O)Cc1ccccc1CCc1nc(Nc2ccc3CNCCc3c2)ncc1C(F)(F)F
NC(=O)Cc1ccccc1CCc1nc(Nc2ccc(cc2)C2CNCCO2)ncc1C(F)(F)F
CC(=O)N1CCC(CC1)c1ccc(Nc2ncc(c(CCc3ccccc3CC(N)=O)n2)C(F)(F)F)cc1
CC(=O)C1CCN(CC1)c1ccc(Nc2ncc(c(CCc3ccccc3CC(N)=O)n2)C(F)(F)F)cc1
NC(=O)Cc1ccccc1CCc1nc(Nc2ccc(CN3CCNCC3)cc2)ncc1C(F)(F)F
NC(=O)Cc1nccnc1CCc1nc(Nc2ccc(cc2)C2CCNCC2)ncc1C(F)(F)F
CN1CCC(CC1)c1ccc(Nc2ncc(c(CCc3nccnc3CC(N)=O)n2)C(F)(F)F)cc1
CN1CCc2cc(Nc3ncc(c(CCc4ccccc4CC(N)=O)n3)C(F)(F)F)ccc2C1
NC(=O)Cc1cncnc1CCc1nc(Nc2ccc(cc2)C2CCNCC2)ncc1C(F)(F)F
CN1CCC(CC1)c1ccc(Nc2ncc(c(CCc3ncncc3CC(N)=O)n2)C(F)(F)F)cc1
CCN1CCC(CC1)c1ccc(Nc2ncc(c(CCc3ccccc3CC(N)=O)n2)C(F)(F)F)cc1
NC(=O)Cc1cccnc1CCc1nc(Nc2ccc(cc2)C2CCNCC2)ncc1C(F)(F)F
CN1CCC(CC1)c1ccc(Nc2ncc(c(CCc3ncccc3CC(N)=O)n2)C(F)(F)F)cc1
CN1CCC(CC1)c1ccc(Nc2ncc(c(CCc3cc(ccn3)C(N)=O)n2)C(F)(F)F)cc1
NC(=O)Cc1ccccc1CCc1nc(Nc2ccc(cc2)C2CCNC2)ncc1C(F)(F)F
CN1CCN(Cc2ccc(Nc3ncc(c(CCc4ccccc4CC(N)=O)n3)C(F)(F)F)cc2)CC1
NC(=O)c1cccc(CCc2nc(Nc3ccc(CN4CCNCC4)cc3)ncc2C(F)(F)F)c1
CCN1CCC(CC1)c1ccc(Nc2ncc(c(CCc3ncccc3CC(N)=O)n2)C(F)(F)F)cc1
NC(=O)Cc1cccnc1CCc1nc(Nc2ccc(cc2)C2CCCNC2)ncc1C(F)(F)F
CCN1CCCC(C1)c1ccc(Nc2ncc(c(CCc3ncccc3CC(N)=O)n2)C(F)(F)F)cc1
COc1cc(ccc1Nc1ncc(c(CCc2ccccc2CC(N)=O)n1)C(F)(F)F)N1CCNCC1
COc1cc(ccc1Nc1ncc(c(CCc2ccccc2CC(N)=O)n1)C(F)(F)F)C1CCNCC1
COc1cc(ccc1Nc1ncc(c(CCc2ccccc2CC(N)=O)n1)C(F)(F)F)C1CCN(C)CC1
CCN1CCC(CC1)c1ccc(Nc2ncc(c(CCc3ccccc3CC(N)=O)n2)C(F)(F)F)c(OC)c1
COc1cc(ccc1Nc1ncc(c(CCc2cccc(c2)C(N)=O)n1)C(F)(F)F)C1CCNCC1
COc1cc(ccc1Nc1ncc(c(CCc2cccc(c2)C(N)=O)n1)C(F)(F)F)C1CCN(C)CC1
CCN1CCC(CC1)c1ccc(Nc2ncc(c(Cc3ccccc3C(N)=O)n2)C(F)(F)F)c(OC)c1
CCc1cc(ccc1Nc1ncc(c(CCc2ccccc2CC(N)=O)n1)C(F)(F)F)C1CCNCC1
CCc1cc(ccc1Nc1ncc(c(CCc2ccccc2CC(N)=O)n1)C(F)(F)F)C1CCN(C)CC1
NC(=O)Cc1ccccc1CCc1nc(Nc2ccc(cc2OC(F)(F)F)C2CCNCC2)ncc1C(F)(F)F
CN1CCC(CC1)c1ccc(Nc2ncc(c(CCc3ccccc3CC(N)=O)n2)C(F)(F)F)c(OC(F)(F)F)c1
CN1CCC(CC1)c1ccc(Nc2ncc(c(CCc3ccccc3CC(N)=O)n2)C(F)(F)F)c(C)c1
CN1CCC(CC1)c1ccc(Nc2ncc(c(CCc3ccccc3CC(N)=O)n2)C(F)(F)F)c(F)c1
CNC(=O)c1cccc(c1)-c1csc2c(N)nc(Nc3ccc(nc3)N3CCOCC3)nc12
CNC(=O)c1cccc(c1)-c1csc2c(N)nc(Nc3ccc(cc3)N3CCC(O)CC3)nc12
CCN1CCN(CC1)c1ccc(Nc2nc(N)c3scc(-c4cccc(c4)C(=O)NC)c3n2)cc1
CNC(=O)c1cccc(c1)-c1csc2c(N)nc(Nc3ccc(cc3)N3CCC(CC3)N3CCCC3)nc12
COc1cc(Nc2nc(N)c3scc(-c4cccc(NC(=O)C5CC5)c4)c3n2)cc(OC)c1OC
CCS(=O)(=O)Nc1cccc(c1)-c1csc2c(N)nc(Nc3cc(OC)c(OC)c(OC)c3)nc12
CNS(=O)(=O)c1cccc(c1)-c1csc2c(N)nc(Nc3cc(OC)c(OC)c(OC)c3)nc12
CCN1CCN(CC1)c1ccc(Nc2nc(N)c3scc(-c4cccc(NS(C)(=O)=O)c4)c3n2)cn1
CCN1CCN(CC1)c1ccc(Nc2nc(N)c3scc(-c4cnc5ccccc5c4)c3n2)cn1
CCN1CCN(CC1)c1ccc(Nc2nc(N)c3scc(-c4cnc5ccccc5c4)c3n2)cc1
Nc1nc(Nc2ccc(nc2)N2CCOCC2)nc2c(csc12)-c1cnc2ccccc2c1
CCN1CCN(CC1)c1cccc(Nc2nc(N)c3scc(-c4cnc5ccccc5c4)c3n2)c1
C[C@H](O)CNc1nc(NCc2ccccc2)c2scc(C#C)c2n1 |r|
C[C@H](O)CNc1nc(N[C@H](C)c2ccccc2)c2scc(C#C)c2n1 |r|
C=Cc1csc2c(NCc3ccccc3)nc(NCCN3CCOCC3)nc12
C[C@@H](Nc1nc(NCCN2CCOCC2)nc2c(C=C)csc12)c1ccccc1 |r|
CCc1csc2c(NCc3ccccc3)nc(NCCN3CCOCC3)nc12
Cc5nc4c(=O)[nH]c3cnc(Nc2ccc(N1CCN(C)CC1)cc2)nc3n(C)c4s5
Cc5nc4c(=O)[nH]c3cnc(Nc2ccc(N1CCC(O)CC1)cc2)nc3n(C)c4s5
COc3cc(N2CCC(N1CCN(C)CC1)CC2)ccc3Nc6ncc5[nH]c(=O)c4nc(C)sc4n(C)c5n6
COc4cc(Nc3ncc2[nH]c(=O)c1nc(C)sc1n(C)c2n3)ccc4N5CCN(C)CC5
COc3cc(N2CCC(N1CCN(C)CC1)CC2)ccc3Nc4ncc6c(n4)n(C)c5sc(C)nc5c(=O)n6C
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCCc12
CNC(=O)c1ccc2OCOc2c1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCCc12
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2C(=O)N2CCCC2)n1)N1CCOCC1
CNS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCCc12
CCCNS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCCc12
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC2CCC2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC2CCCC2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC2CCCCC2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2NC(C)=O)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2N(C)S(C)(=O)=O)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCCc2c(NCc2ccccc2N(C)S(C)(=O)=O)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2cccc(C)n2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccc(F)c(F)c2)n1)N1CCOCC1
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2CO)N2CCOCC2)nc2NCCc12
CNC(=O)c1ccccc1Nc1nc(Nc2cccc3OCCOc23)nc2NCCc12
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCOCC3)c3OCCOc23)nc2NCCc12
CCN1c2ccc(Nc3nc4NCCc4c(Nc4ccccc4C(=O)NC)n3)c(OC)c2CCCC1=O
CNC(=O)c1ccccc1Nc1nc(Nc2cccc3ccoc23)nc2NCCc12
CNC(=O)c1ccccc1Nc1nc(Nc2cc(C)nn2C)nc2NCCc12
CNC(=O)c1ccccc1Nc1nc(Nc2cc(OC)c(OC)c(OC)c2)nc2NCCc12
CNC(=O)c1ccccc1Nc1nc(Nc2cccc3n(CCCN4CCOCC4)ccc23)nc2NCCc12
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCC(C)c12
COc1cc(ccc1Nc1nc2NCC(C)c2c(Nc2ccccc2C(=O)N2CCCC2)n1)N1CCOCC1
CNS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCC(C)c12
CCCNS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCC(C)c12
COc1cc(ccc1Nc1nc2NCC(C)c2c(Nc2ccccc2S(=O)(=O)NC2CCC2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)c2c(Nc2ccccc2S(=O)(=O)NC2CCCC2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)c2c(Nc2ccccc2S(=O)(=O)NC2CCCCC2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)c2c(Nc2ccccc2NC(C)=O)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)c2c(Nc2ccccc2N(C)S(C)(=O)=O)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)c2c(NCc2ccccc2N(C)S(C)(=O)=O)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)c2c(Nc2cccc(C)n2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)c2c(Nc2ccc(F)c(F)c2)n1)N1CCOCC1
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NC[C@@H](C)c12 |r|
COc1cc(ccc1Nc1nc2NC[C@@H](C)c2c(Nc2ccccc2S(=O)(=O)NC2CCC2)n1)N1CCOCC1 |r|
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCC(C)(C)c12
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)N(C)C)n1)N1CCOCC1
CCCCNS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCCc12
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(N)(=O)=O)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC2CC2)n1)N1CCOCC1
CCNS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCCc12
CCC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCCc12
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NCC(C)C)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)(C)C)n1)N1CCOCC1
COCCCNS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCCc12
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NCCN(C)C)n1)N1CCOCC1
COCCNS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCCc12
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)Nc2ccccc2)n1)N1CCOCC1
CC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)N2CCOCC2)nc2NCCc12
CNC(=O)c1ccc(Nc2nc3NCCc3c(Nc3ccccc3S(=O)(=O)NC(C)C)n2)cc1
CC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(CO)cc2)nc2NCCc12
CC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2F)N2CCOCC2)nc2NCCc12
COc1nc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCOCC1
CC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(nc2)N2CCOCC2)nc2NCCc12
CC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cn2)N2CCOCC2)nc2NCCc12
CCOc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCOCC1
CC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2C(F)(F)F)N2CCOCC2)nc2NCCc12
CC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(F)(F)F)nc2NCCc12
CC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N(C)C)nc2NCCc12
CC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(NC(C)=O)cc2)nc2NCCc12
CNS(=O)(=O)c1ccc(Nc2nc3NCCc3c(Nc3ccccc3S(=O)(=O)NC(C)C)n2)cc1
CC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N2CCOCC2)nc2NCCc12
CC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2C)N2CCOCC2)nc2NCCc12
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCCC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCCCC1
CC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(C)O)nc2NCCc12
COc1cc(OCCN2CCOCC2)ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1
CC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(OC(F)(F)F)cc2)nc2NCCc12
CC(C)NC(C)c1ccc(Nc2nc3NCCc3c(Nc3ccccc3S(=O)(=O)NC(C)C)n2)cc1
CC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2cccc(NS(C)(=O)=O)c2)nc2NCCc12
CNC(=O)c1cccc(Nc2nc3NCCc3c(Nc3ccccc3S(=O)(=O)NC(C)C)n2)c1
CC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2cccc(NC(C)=O)c2)nc2NCCc12
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCC(CC1)N(C)C
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)-n1ccnc1
CC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N2CCCC2)nc2NCCc12
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCC(CO)CC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCC(O)C1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCCC(O)C1
CC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(C)N2CCCCC2)nc2NCCc12
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)-n1ccccc1=O
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1C(C)COCC1C
COc1cc(NCCN2CCOCC2)ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCC(O)CC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCS(=O)(=O)CC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)-n1ncnn1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCC(C1)N(C)C
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)-n1cc(C)nc1C
CC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2nc(C)cs2)nc2NCCc12
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCC(CC1)N1CCCCC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCC(CC1)N1CCCC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)-n1cccn1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCC(CC1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCC(CC1)N1CCN(C)CC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCC(CC1)N1CCNCC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCCCC1=O
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1C(=O)CCc2ccccc12
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2S(=O)(=O)C(C)C)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)c2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCOCC1
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NC[C@H](C)c12 |r|
CNS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCC(C)(C)c12
COc1cc(ccc1Nc1nc2NCC(C)(C)c2c(Nc2ccccc2S(=O)(=O)NC2CCC2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)(C)c2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCOCC1
CCCNS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCC(C)(C)c12
COc1cc(ccc1Nc1nc2NCC(C)(C)c2c(Nc2ccccc2S(=O)(=O)NCC(C)C)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)(C)c2c(Nc2ccccc2S(=O)(=O)NC2CCCC2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)(C)c2c(Nc2ccccc2S(=O)(=O)NC2CCCCC2)n1)N1CCOCC1
CCCCNS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCC(C)(C)c12
COc1cc(ccc1Nc1nc2NCC(C)(C)c2c(Nc2ccccc2S(=O)(=O)N(C)C)n1)N1CCOCC1
CCC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCC(C)(C)c12
CCNS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCC(C)(C)c12
COCCCNS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCC(C)(C)c12
COCCNS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCC(C)(C)c12
COc1cc(ccc1Nc1nc2NCC(C)(C)c2c(Nc2ccccc2S(=O)(=O)Nc2ccccc2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)(C)c2c(Nc2ccccc2S(=O)(=O)NC(C)(C)C)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)(C)c2c(Nc2ccccc2S(=O)(=O)NCC2CC2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)(C)c2c(Nc2ccccc2S(=O)(=O)NCCO)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)(C)c2c(Nc2ccccc2S(=O)(=O)NCCN(C)C)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)(C)c2c(Nc2ccccc2C(=O)N2CCCC2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)(C)c2c(Nc2ccccc2N(C)S(C)(=O)=O)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)(C)c2c(Nc2cccc(C)n2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)(C)c2c(Nc2ccccc2NC(C)=O)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC(C)(C)c2c(Nc2ccc(F)c(F)c2)n1)N1CCOCC1
CNC(=O)c1ccc2OCOc2c1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCC(C)(C)c12
COc1cc(ccc1Nc1nc2NCC(C)(C)c2c(NC2CCCCC2N(C)S(C)(=O)=O)n1)N1CCOCC1
CNC(=O)c1ccccc1Nc1nc(Nc2cccc3OCCOc23)nc2NCC(C)(C)c12
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCOCC3)c3OCCOc23)nc2NCC(C)(C)c12
CNC(=O)c1ccccc1Nc1nc(Nc2cc(OC)c(OC)c(OC)c2)nc2NCC(C)(C)c12
CNC(=O)c1ccccc1Nc1nc(Nc2cccc3ccoc23)nc2NCC(C)(C)c12
CNC(=O)c1ccccc1Nc1nc(Nc2cc(C)nn2C)nc2NCC(C)(C)c12
CCN1c2ccc(Nc3nc4NCC(C)(C)c4c(Nc4ccccc4C(=O)NC)n3)c(OC)c2CCCC1=O
CNC(=O)c1ccccc1Nc1nc(Nc2ccc3n(CCCN4CCOCC4)ccc3c2)nc2NCC(C)(C)c12
CNS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCC3(CC3)c12
COc1cc(ccc1Nc1nc2NCC3(CC3)c2c(Nc2ccccc2S(=O)(=O)NC(C)(C)C)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC3(CC3)c2c(Nc2ccccc2S(=O)(=O)NCC(C)C)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC3(CC3)c2c(Nc2ccccc2S(=O)(=O)NC(C)C)n1)N1CCOCC1
CCNS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCC3(CC3)c12
COc1cc(ccc1Nc1nc2NCC3(CC3)c2c(Nc2ccccc2S(=O)(=O)NCC2CC2)n1)N1CCOCC1
COCCNS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCC3(CC3)c12
COc1cc(ccc1Nc1nc2NCC3(CC3)c2c(Nc2ccccc2S(=O)(=O)NCCO)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC3(CC3)c2c(Nc2ccccc2S(=O)(=O)Nc2ccccc2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC3(CC3)c2c(Nc2ccccc2S(=O)(=O)NCC=C)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC3(CC3)c2c(Nc2ccccc2S(=O)(=O)NC2CCCC2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC3(CC3)c2c(Nc2ccccc2S(=O)(=O)NC2CC2)n1)N1CCOCC1
CCC(C)NS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCC3(CC3)c12
CCCNS(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCC3(CC3)c12
COc1cc(ccc1Nc1nc2NCC3(CC3)c2c(Nc2ccccc2S(=O)(=O)NC2CCCCC2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC3(CC3)c2c(Nc2ccccc2S(=O)(=O)NC2CCC2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC3(CC3)c2c(Nc2ccccc2S(=O)(=O)N(C)C)n1)N1CCOCC1
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2NCC3(CC3)c12
COc1cc(ccc1Nc1nc2NCC3(CC3)c2c(Nc2ccc(F)c(F)c2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC3(CC3)c2c(Nc2cccc(C)n2)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC3(CC3)c2c(Nc2ccccc2NC(C)=O)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCC3(CC3)c2c(Nc2ccccc2N(C)S(C)(=O)=O)n1)N1CCOCC1
CNS(=O)(=O)c1ccccc1Nc1nc(Nc2cc(OC)c(OC)c(OC)c2)nc2NCC3(CC3)c12
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)N2CCOCC2)nc2NCCc12
CNC(=O)c1ccccc1Nc1nc(Nc2ccccc2OC)nc2NCCc12
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2C(O)=O)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2C=O)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2CCO)n1)N1CCOCC1
COc1cc(ccc1Nc1nc2NCCc2c(Nc2ccccc2P(C)(C)=O)n1)N1CCC(CC1)N1CCNCC1
COc3cc(N2CCC(N1CCN(C)CC1)CC2)ccc3Nc6ncc5[nH]c(=O)c4ncsc4n(C)c5n6
COc2cc(N1CCN(C)CC1)ccc2Nc5ncc4[nH]c(=O)c3nc(C)sc3n(C)c4n5
CCc6nc5c(=O)[nH]c4cnc(Nc3ccc(N2CCC(N1CCN(C)CC1)CC2)cc3OC)nc4n(C)c5s6
CCn6c4nc(Nc3ccc(N2CCC(N1CCN(C)CC1)CC2)cc3OC)ncc4[nH]c(=O)c5nc(C)sc56
CNC(=O)c4ccc(Nc3ncc2[nH]c(=O)c1nc(C)sc1n(C)c2n3)cc4
COc2cc(N1CCN(S(C)(=O)=O)CC1)ccc2Nc5ncc4[nH]c(=O)c3nc(C)sc3n(C)c4n5
COc2cc(N1CCNCC1)ccc2Nc3ncc5c(n3)n(C)c4sc(C)nc4c(=O)n5C
C=CC(=O)N5CCN(c4ccc(Nc1ncc3c(n1)n(C)c2sc(C)nc2c(=O)n3C)c(OC)c4)CC5
COc2cc(N1CCN(C)CC1)ccc2Nc3ncc5c(n3)n(C)c4sc(C)nc4c(=O)n5C
CCOc2cc(N1CCN(C)CC1)ccc2Nc3ncc5c(n3)n(C)c4sc(C)nc4c(=O)n5C
Cc5nc4c(=O)n(C)c3cnc(Nc2ccc(N1CCN(C)CC1)cc2OCCO)nc3n(C)c4s5
COc2cc(N1CCN(C)CC1)c(C)cc2Nc3ncc5c(n3)n(C)c4sc(C)nc4c(=O)n5C
COc2cc(C1CCN(C)CC1)ccc2Nc3ncc5c(n3)n(C)c4sc(C)nc4c(=O)n5C
COc2cc(N1CCN(CCO)CC1)ccc2Nc3ncc5c(n3)n(C)c4sc(C)nc4c(=O)n5C
CNC(=O)c4ccc(Nc1ncc3c(n1)n(C)c2sc(C)nc2c(=O)n3C)c(OC)c4
COC2C=C1CCN(C)CC1=CC2Nc3ncc5c(n3)n(C)c4sc(C)nc4c(=O)n5C
Cc5nc4c(=O)n(C)c3cnc(NC2C=C1CCC(=O)NC1=CC2)nc3n(C)c4s5
Cc5nc4c(=O)n(C)c3cnc(Nc2ccc(N1CCN(C)CC1)cn2)nc3n(C)c4s5
Cc4nc3c(=O)n(C)c2cnc(Nc1cnn(C)c1)nc2n(C)c3s4
COc3cc(C(=O)N2CCC(N1CCN(C)CC1)CC2)ccc3Nc4ncc6c(n4)n(C)c5sc(C)nc5c(=O)n6C
CCN1c2cnc(Nc3ccc(cc3OC)N3CCC(CC3)N3CCN(C)CC3)nc2N(C)c2sc(C)nc2C1=O
CCN1c2sc(C)nc2C(=O)N(C)c2cnc(Nc3ccc(cc3OC)N3CCC(CC3)N3CCN(C)CC3)nc12
COc3cc(N2CCC(N1CCN(C)CC1)CC2)ccc3Nc4ncc6c(n4)n(C)c5sc(C(F)(F)F)nc5c(=O)n6C
CN1CCN(c2ccc(Nc3ncc4c(n3)N(C)c3sc(-c5ccccc5)nc3C(=O)N4C)cc2)CC1
COc3cc(N2CCC(N1CCN(C)CC1)CC2)ccc3Nc4ncc7c(n4)n(C)c6sc(c5ccccc5)nc6c(=O)n7C
CCc6nc5c(=O)n(C)c4cnc(Nc3ccc(N2CCC(N1CCN(C)CC1)CC2)cc3OC)nc4n(C)c5s6
COC4C=C(Nc3ncc2[nH]c(=O)c1nc(C)sc1n(C)c2n3)C=CC4N6CCC(N5CCN(C)CC5)CC6
COc3cc(N2CCN(C1CCN(C)CC1)CC2)ccc3Nc4ncc6c(n4)n(C)c5sc(C)nc5c(=O)n6C
COc2cc(N1CCN(C)CC1=O)ccc2Nc3ncc5c(n3)n(C)c4sc(C)nc4c(=O)n5C
CNC(=O)c4ccc(Nc1ncc3c(n1)n(C)c2sc(C)nc2c(=O)n3C)cc4
COc2cc(N1CCN(S(C)(=O)=O)CC1)ccc2Nc3ncc5c(n3)n(C)c4sc(C)nc4c(=O)n5C
COc2cc(N1CCN(C(C)=O)CC1)ccc2Nc3ncc5c(n3)n(C)c4sc(C)nc4c(=O)n5C
COc2cc(N1CCN(CCN(C)C)CC1)ccc2Nc3ncc5c(n3)n(C)c4sc(C)nc4c(=O)n5C
Cc5nc4c(=O)n(C)c3cnc(Nc2ccc(N1CCN(C)CC1)cc2OCC(F)(F)F)nc3n(C)c4s5
CCCOc2cc(N1CCN(C)CC1)ccc2Nc3ncc5c(n3)n(C)c4sc(C)nc4c(=O)n5C
COc3cc(N2CCC(N1CCN(C)CC1)CC2)ccc3Nc4ncc6c(n4)n(C)c5sc(C(C)C)nc5c(=O)n6C
COc3cc(N2CCC(N1CCN(C)CC1)CC2)ccc3Nc4ncc6c(n4)n(CC(F)(F)F)c5sc(C)nc5c(=O)n6C
CCCn6c4nc(Nc3ccc(N2CCC(N1CCN(C)CC1)CC2)cc3OC)ncc4n(C)c(=O)c5nc(C)sc56
C[C@H]1CNC(=O)c2cnn3c2nc(cc3)N[C@@H](c4cc(ccc4O1)F)C
CCC1(OCCCOc2ccc(Nc3ncc(F)c(N[C@@H]4CCCN(C4)C(=O)C=C)n3)cc2)OCC(C)(C)CO1 |r|
Fc1cnc(Nc2ccc3OCCOCCOCCOc3c2)nc1N[C@@H]1CCCN(C1)C(=O)C=C |r|
C=CC(=O)N1CCC[C@H](C1)Nc1nc(Nc2ccc3OCCOCCOCCOc3c2)nc2[nH]cnc12 |r|
CCC(=O)N1CCC[C@H](C1)Nc1nc(Nc2ccc3OCCOCCOCCOc3c2)nc2[nH]cnc12 |r|
CCC1(OCCCOc2ccc(Nc3ncc(F)c(Nc4cccc(NC(=O)C=C)c4)n3)cc2)OCC(C)(C)CO1
Fc1cnc(Nc2ccc3OCCOCCOCCOc3c2)nc1Nc1cccc(NC(=O)C=C)c1
C=CC(=O)Nc1cccc(Nc2nc(Nc3ccc4OCCOCCOCCOc4c3)nc3[nH]cnc23)c1
CCC(=O)Nc1cccc(Nc2nc(Nc3ccc4OCCOCCOCCOc4c3)nc3[nH]cnc23)c1
CCC1(OCCCOc2ccc(Nc3ncc(F)c(Nc4ccccc4NC(=O)C=C)n3)cc2)OCC(C)(C)CO1
Fc1cnc(Nc2ccc3OCCOCCOCCOc3c2)nc1Nc1ccccc1NC(=O)C=C
C=CC(=O)Nc1ccccc1Nc1nc(Nc2ccc3OCCOCCOCCOc3c2)nc2[nH]cnc12
CCC(=O)Nc1ccccc1Nc1nc(Nc2ccc3OCCOCCOCCOc3c2)nc2[nH]cnc12
CCC(=O)Nc1ccccc1Nc1nc(Nc2ccc3OCCOCCOCCOc3c2)nc2[nH]ccc12
CCC(=O)Nc1ccccc1Nc1nc(Nc2ccc3OCCOCCOCCOc3c2)nc2[nH]ncc12
CONC(=O)c1ccccc1Nc1nc(Nc2ccc3OCCOCCOCCOc3c2)nc2[nH]ncc12
CN([C@@H]1CCCC[C@H]1Oc1nc(Nc2ccc3OCCOCCOCCOc3c2)nc2[nH]ccc12)S(C)(=O)=O |r|
CN([C@@H]1CCCC[C@H]1Oc1nc(Nc2ccc3OCCOCCOCCOc3c2)nc2[nH]ncc12)S(C)(=O)=O |r|
CN(C1CCCC1Oc1nc(Nc2ccc3OCCOCCOCCOc3c2)nc2[nH]ccc12)S(C)(=O)=O
CN([C@@H]1CCC[C@H]1Oc1nc(Nc2ccc3OCCOCCOCCOc3c2)nc2[nH]ncc12)S(C)(=O)=O |r|
CN(c1cnccc1CNc1nc(Nc2ccc3OCCOCCOCCOc3c2)nc2[nH]ccc12)S(C)(=O)=O
CN(c1cnccc1CNc1nc(Nc2ccc3OCCOCCOCCOc3c2)nc2[nH]ncc12)S(C)(=O)=O
C1COCCOc2cc(Nc3nc(Nc4cccc5[nH]ccc45)c4nc[nH]c4n3)ccc2OCCO1
C1COCCOc2cc(Nc3nc(Nc4cccc5cc[nH]c45)c4nc[nH]c4n3)ccc2OCCO1
CC(=O)Nc1cc(C)ccc1Nc1nc(Nc2ccc3OCCOCCOCCOc3c2)nc2[nH]cnc12
CC(=O)Nc1cc(F)ccc1Nc1nc(Nc2ccc3OCCOCCOCCOc3c2)nc2[nH]cnc12
CC(=O)Nc1cc(ccc1Nc1nc(Nc2ccc3OCCOCCOCCOc3c2)nc2[nH]cnc12)C(F)(F)F
Fc1cnc(Nc2ccc3OCCOCCOCCOc3c2)nc1-c1cccc(NC(=O)C=C)c1
CN([C@H]1[C@@H](Cc2ccccc12)Oc1nc(Nc2ccc3OCCOCCOCCOc3c2)nc2[nH]cnc12)S(C)(=O)=O |r|
CN([C@H]1[C@@H](Cc2ccccc12)Oc1nc(Nc2ccc3OCCOCCOCCOc3c2)ncc1C(F)(F)F)S(C)(=O)=O |r|
CN([C@@H]1CCC[C@H]1Oc1nc(Nc2ccc3OCCOCCOCCOc3c2)nc2sccc12)S(C)(=O)=O |r|
C=CC(=O)N1CCC(NC(=O)c2ccc(Nc3ncc(C(F)(F)F)c(NCc4nccnc4N(C)S(C)(=O)=O)n3)c(OC)c2)CC1
C=CC(=O)N1CCC(NC(=O)c2ccc(Nc3ncc(C(F)(F)F)c(NCc4nccnc4N(C)S(C)(=O)=O)n3)c(OC)c2)C1
C=CC(=O)N1CCCC(NC(=O)c2ccc(Nc3ncc(C(F)(F)F)c(NCc4nccnc4N(C)S(C)(=O)=O)n3)c(OC)c2)C1
C=CC(=O)N1CCC(CNC(=O)c2ccc(Nc3ncc(C(F)(F)F)c(NCc4nccnc4N(C)S(C)(=O)=O)n3)c(OC)c2)CC1
C=CC(=O)NC1CCC(CNC(=O)c2ccc(Nc3ncc(C(F)(F)F)c(NCc4nccnc4N(C)S(C)(=O)=O)n3)c(OC)c2)CC1
C=CC(=O)N1CCCC(c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(Nc5ccccc5C(=O)NC)n4)cc3)c2)C1
C=CC(=O)N1CCC(CNC(=O)c2ccc(Nc3ncc(C(F)(F)F)c(Nc4ccccc4P(C)(C)=O)n3)cc2)CC1
C=CC(=O)N1CCC(CNC(=O)c2ccc(Nc3ncc(C(F)(F)F)c(Nc4ccccc4P(C)(C)=O)n3)c(OC)c2)CC1
C=CC(=O)N1CCCC1c1ccc(NCc2ccc(Nc3ncc(C(F)(F)F)c(Nc4ccccc4C(=O)NC)n3)cc2)cc1
C=CC(=O)N1CCCC(c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(Nc5ccccc5P(C)(C)=O)n4)cc3)c2)C1
C=CC(=O)N1CCCC(c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(Nc5ccccc5C(=O)NOC)n4)cc3)c2)C1
C=CC(=O)N1CCCC(c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(Nc5ccccc5C(=O)NC)n4)c(OC)c3)c2)C1
C=CC(=O)N1CCCC(c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(Nc5cccc(F)c5C(=O)NC)n4)cc3)c2)C1
C=CC(=O)N1CCCC(c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(NCc5nccnc5N(C)S(C)(=O)=O)n4)cc3)c2)C1
C=CC(=O)N1CCCC(c2cccc(NCc3ccc(Nc4ncc(Cl)c(Nc5ccccc5C(=O)NC)n4)cc3)c2)C1
C=CC(=O)N1CCCC(c2cccc(NCc3ccc(Nc4ncc(Br)c(Nc5ccccc5C(=O)NC)n4)cc3)c2)C1
C=CC(=O)N1CCCC(c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(Nc5ccccc5C(=O)NCC)n4)cc3)c2)C1
C=CC(=O)N1CCCC(c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(Nc5ccccc5C(=O)NC(C)C)n4)cc3)c2)C1
C=CC(=O)N1CCCC(c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(Nc5ccccc5S(=O)(=O)NC(C)C)n4)cc3)c2)C1
C=CC(=O)N1CCCC(c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(Nc5cccc6c5C(=O)N(C)C6)n4)cc3)c2)C1
CC#CC(=O)N1CCCC(c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(Nc5ccccc5C(=O)NC)n4)cc3)c2)C1
C=C(C)C(=O)N1CCCC(c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(Nc5ccccc5C(=O)NC)n4)cc3)c2)C1
C=CC(=O)N1CCCC(c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(Nc5ccccc5S(=O)(=O)NC)n4)cc3)c2)C1
C#CC(=O)N1CCCC(c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(Nc5ccccc5C(=O)NC)n4)cc3)c2)C1
C/C=C/C(=O)N1CCCC(c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(Nc5ccccc5C(=O)NC)n4)cc3)c2)C1
C=C(F)C(=O)N1CCCC(c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(Nc5ccccc5C(=O)NC)n4)cc3)c2)C1
C=CC(=O)N1CCC[C@H](c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(Nc5ccccc5C(=O)NC)n4)cc3)c2)C1
C=CC(=O)N1CCC[C@@H](c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(Nc5ccccc5C(=O)NC)n4)cc3)c2)C1
C=CC(=O)N1CCC[C@H](c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(Nc5ccccc5C(=O)NOC)n4)cc3)c2)C1
C=CC(=O)N1CCC[C@@H](c2cccc(NCc3ccc(Nc4ncc(C(F)(F)F)c(Nc5ccccc5C(=O)NC)n4)cc3)c2)C1
CNC(=O)c1ccc(Nc2ncc(C(F)(F)F)c(Oc3cccc4c3C(=O)N(C)C43CC3)n2)cc1
CNC(=O)c1ccc(Nc2ncc(C(F)(F)F)c(Oc3cccc4c3C(=O)N(C)C43CC3)n2)c(OC)c1
COc1cc(C(=O)NC2CCN(C)CC2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCN(C)CC2)c(Cl)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2(C)CCN(C)CC2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2(C)CCN(C)CC2)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CC3(CCN(C)CC3)C2)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CC3(CCN(C)CC3)C2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC3(CC2)CN(C)C3)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC3(CC2)CN(C)C3)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC23CCN(C)CC3)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC23CCN(C)CC3)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC3(CC2)CCN3C)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC3(CC2)CCN3C)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2COC3(CCN(C)CC3)C2)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2COC3(CCN(C)CC3)C2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC3(CCN(C)CC3)C2)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC3(CCN(C)CC3)C2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC3(CC2)CCN(C)C3)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC3(CC2)CCN(C)C3)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC3(CC2)CCN(C)CC3)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC3(CC2)CCN(C)CC3)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC3(CCN(C)C3)C2)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC3(CCN(C)C3)C2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2COC3(CCN(C)C3)C2)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2COC3(CCN(C)C3)C2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCN3CCN(C)C3C2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCN3CCOC3C2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCN3CCN=C3C2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCn3ccnc3C2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCn3cnnc3C2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCN(C)CC2F)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCN(C)CC2OC)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCNCC2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
[2H]C([2H])([2H])N1CCC(NC(=O)c2ccc(Nc3ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)c(OC)c2)CC1
CCN1CCC(NC(=O)c2ccc(Nc3ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)c(OC)c2)CC1
COc1cc(C(=O)NC2CCN(CS(C)(=O)=O)CC2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCN(CC(N)=O)CC2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
[2H]C([2H])([2H])N1CCC(NC(=O)c2cc(OC)c(Nc3ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)cc2F)CC1
CCN1CCC(NC(=O)c2cc(OC)c(Nc3ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)cc2F)CC1
[2H]C([2H])([2H])N1CCC(C)(NC(=O)c2ccc(Nc3ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)c(OC)c2)CC1
[2H]C([2H])([2H])N1CCC(C)(NC(=O)c2cc(OC)c(Nc3ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)cc2F)CC1
COc3cc(C(=O)NC2CC1(CCNCC1)C2)ccc3Nc7ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C56CC6)n7
[2H]C([2H])([2H])N1CCC2(CC1)CC(NC(=O)c1ccc(Nc3ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)c(OC)c1)C2
CCN1CCC7(CC1)CC(NC(=O)c6ccc(Nc5ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C34CC4)n5)c(OC)c6)C7
[2H]C([2H])([2H])N1CCC2(CC1)CC(NC(=O)c1cc(OC)c(Nc3ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)cc1F)C2
CCN1CCC2(CC1)CC(NC(=O)c1cc(OC)c(Nc3ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)cc1F)C2
C=Cc2cc(C(=O)NC1CCN(C)CC1)ccc2Nc6ncc(C(F)(F)F)c(Oc3cccc4c3C(=O)N(C)C45CC5)n6
CCc2cc(C(=O)NC1CCN(C)CC1)ccc2Nc6ncc(C(F)(F)F)c(Oc3cccc4c3C(=O)N(C)C45CC5)n6
CCc2cc(C(=O)NC1CCN(C)CC1)c(F)cc2Nc6ncc(C(F)(F)F)c(Oc3cccc4c3C(=O)N(C)C45CC5)n6
CCc3cc(C(=O)NC2CC1(CCN(C)CC1)C2)ccc3Nc7ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C56CC6)n7
CN1CCC(NC(=O)c2ccc(Nc3ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)c(OC(F)(F)F)c2)CC1
COc1cc(C(=O)NC2CCN(C)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)N2CC3(CCN(C)CC3)C2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)N2CCC3(CCN(C)CC3)CC2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)N2CCC3(CCN(C)C3)C2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)N2CCC3(CCN(C)C3)C2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc3cc(C(=O)N1CCC12CCN(C)CC2)ccc3Nc7ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C56CC6)n7
COc1cc(C(=O)N2CCC3(CCN(C)CC3)C2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)N2CCC3(CCCN(C)C3)C2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC3(CCN(C)CC3)C2=O)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3(CCN(C)CC3)CC2=O)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc3cc(N2CC1(CCN(C)CC1)OC2=O)ccc3Nc7ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C56CC6)n7
COc1cc(N2CC3(CCN(C)C3)OC2=O)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3(CCC2=O)CCN(C)CC3)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3(CCN(C)C3)OCC2=O)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C2=NOC3(CCN(C)CC3)C2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
CN1C(=O)c2c(Oc3nc(Nc4ccc5c(c4)CC(=O)N5)ncc3C(F)(F)F)cccc2C12CC2
CN1C(=O)c2c(Oc3nc(Nc4ccc5c(c4)CNC5=O)ncc3C(F)(F)F)cccc2C12CC2
CN1C(=O)c2c(Oc3nc(Nc4ccc5c(c4)CCNC5=O)ncc3C(F)(F)F)cccc2C12CC2
CN1CCC(N2C(=O)Cc3cc(Nc4ncc(C(F)(F)F)c(Oc5cccc6c5C(=O)N(C)C65CC5)n4)ccc32)CC1
COc1cc(N2CCN(C)CC2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCNCC2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCN(CC(=O)N(C)C)CC2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COCCN1CCN(c2ccc(Nc3ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)c(OC)c2)CC1
COc1cc(N2CCOCC2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC(N3CCN(C)CC3)CC2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3(CCN(C)CC3)C2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(CN(C)C)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(CN2CCCC2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(CN2CCN(C)CC2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCN(C)CC2=O)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C2CCN(C)CC2)ccc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
CN1CCN(c2ccc(Nc3ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)nc2)CC1
COc1cc2c(cc1Nc1ncc(C(F)(F)F)c(Oc3cccc4c3C(=O)N(C)C43CC3)n1)CN(C)CC2
CN1CCc2c(cc(Nc3ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)cc2C2CC2)C1
CN1Cc2cc(Nc3ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)cc3c2C(CCC3)C1
CN1Cc2cc(Nc3ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)cc3c2C(CCO3)C1
COc1cc2c(cc1Nc1ncc(C(F)(F)F)c(Oc3cccc4c3C(=O)N(C)C43CC3)n1)CN(C)C(=O)C2
Cc1cc(Nc2ncc(C(F)(F)F)c(Oc3cccc4c3C(=O)N(C)C43CC3)n2)n(C(C)C)n1
CN1C(=O)c2c(Oc3nc(Nc4cc5n(n4)CCC5)ncc3C(F)(F)F)cccc2C12CC2
Cc1c(Nc2ncc(C(F)(F)F)c(Oc3cccc4c3C(=O)N(C)C43CC3)n2)nn2c1CCC2
CN1C(=O)c2c(Oc3nc(Nc4cc5n(n4)CCOC5)ncc3C(F)(F)F)cccc2C12CC2
CN1C(=O)c2c(Oc3nc(Nc4cnn5c4COCC5)ncc3C(F)(F)F)cccc2C12CC2
CN1CCn2nc(Nc3ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)cc2C1
CN1CCC(n2ccc(Nc3ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)n2)CC1
Cc1cn(C2CCN(C)CC2)nc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCN(C)CC2)ccc1Nc1ncc(C(F)(F)F)c(Cc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(C(F)(F)F)c(Cc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CC3(CCN(C)CC3)C2)ccc1Nc1ncc(C(F)(F)F)c(Cc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CC3(CCN(C)CC3)C2)c(F)cc1Nc1ncc(C(F)(F)F)c(Cc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC3(CC2)CN(C)C3)ccc1Nc1ncc(C(F)(F)F)c(Cc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC3(CCN(C)C3)C2)ccc1Nc1ncc(C(F)(F)F)c(Cc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2COC3(CCN(C)C3)C2)ccc1Nc1ncc(C(F)(F)F)c(Cc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC3(CC2)CCN(C)C3)ccc1Nc1ncc(C(F)(F)F)c(Cc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC3(CC2)CCN(C)CC3)ccc1Nc1ncc(C(F)(F)F)c(Cc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC23CCN(C)CC3)ccc1Nc1ncc(C(F)(F)F)c(Cc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCC3(CC2)CCN3C)ccc1Nc1ncc(C(F)(F)F)c(Cc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCN3CCN(C)C3C2)ccc1Nc1ncc(C(F)(F)F)c(Cc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCN(C)CC2)ccc1Nc1ncc(C(F)(F)F)c(Cc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCOCC2)ccc1Nc1ncc(C(F)(F)F)c(Cc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC(N3CCN(C)CC3)CC2)ccc1Nc1ncc(C(F)(F)F)c(Cc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCN(C)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCN(C)CC2)ccc1Nc1ncc(C)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCN(C)CC2)ccc1Nc1ncc(Br)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2(C)CCN(C)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C2CCN(C)CC2)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3(CCN(C)CC3)C2)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC(N3CCN(C)CC3)CC2)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCN(C)CC2)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COCCN1CCN(c2cc(OC)c(Nc3ncc(C(F)(F)F)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)cc2F)CC1
COc1cc(N2CCN(CC(=O)N(C)C)CC2)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3(CN(C)C3)C2)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC3(CC2)CN(C)C3)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC3(CCN(C)C3)C2)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC(N(C)C)CC2)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCN(C)CC2=O)c(F)cc1Nc1ncc(C(F)(F)F)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCN(C)CC2)ccc1Nc1ncc(C2CC2)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3(CCN(C)CC3)C2)ccc1Nc1ncc(C2CC2)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CC3(CCN(C)CC3)C2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CC3(CCN(C)CC3)C2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C2CCN(C)CC2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C2CCN(C)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C2CC3(CCN(C)CC3)C2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3(CCN(C)CC3)C2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC(N3CCN(C)CC3)CC2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC(N3CCN(C)CC3)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCN(C)CC2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCN(C)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COCCN1CCN(c2ccc(Nc3ncc(Cl)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)c(OC)c2)CC1
COCCN1CCN(c2cc(OC)c(Nc3ncc(Cl)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)cc2F)CC1
COc1cc(N2CCN(CC(=O)N(C)C)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3(CN(C)C3)C2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3(CN(C)C3)C2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC3(CCN(C)CC3)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC3(CC2)CN(C)C3)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC3(CC2)CN(C)C3)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC3(CCN(C)C3)C2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC3(CCN(C)C3)C2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC(N(C)C)CC2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(CN2CCN(C)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(CN(C)C2CCN(C)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(CNC2CCN(C)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(CN(C)C2CCN(C)CC2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC(N3CCN(C)CC3)C2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC(N3CC(N(C)C)C3)C2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC(N(C)C)C2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC(N(C)C)C2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC(N3C4CCC3CN(C)C4)C2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC(N3C4CC3CN(C)C4)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC(N3CC4CC(C3)N4C)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2C3CC2CN(C)C3)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3CC(C2)N3C)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2C3CCC2CN(C)C3)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC3C(CCN3C)C2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC3CN(C)CCC32)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3CN(C)CC3C2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3CCN(C)C3C2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3CCN(C)C3C2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC3CN(C)CC32)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC3CN(C)CC3C2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(Br)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CC3(CCN(C)CC3)C2)c(F)cc1Nc1ncc(Br)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CC3(CCN(C)CC3)C2)ccc1Nc1ncc(Br)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3(CCN(C)CC3)C2)ccc1Nc1ncc(Br)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3(CCN(C)CC3)C2)c(F)cc1Nc1ncc(Br)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C2CCN(C)CC2)ccc1Nc1ncc(Br)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C2CCN(C)CC2)c(F)cc1Nc1ncc(Br)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC(N3CCN(C)CC3)CC2)c(F)cc1Nc1ncc(Br)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC(N3CCN(C)CC3)CC2)ccc1Nc1ncc(Br)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCN(C)CC2)c(F)cc1Nc1ncc(Br)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCN(C)CC2)ccc1Nc1ncc(Br)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COCCN1CCN(c2ccc(Nc3ncc(Br)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)c(OC)c2)CC1
COCCN1CCN(c2cc(OC)c(Nc3ncc(Br)c(Oc4cccc5c4C(=O)N(C)C54CC4)n3)cc2F)CC1
COc1cc(N2CCN(CC(=O)N(C)C)CC2)ccc1Nc1ncc(Br)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3(CN(C)C3)C2)ccc1Nc1ncc(Br)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC3(CCN(C)CC3)CC2)ccc1Nc1ncc(Br)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC3(CC2)CN(C)C3)ccc1Nc1ncc(Br)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC(N(C)C)CC2)c(F)cc1Nc1ncc(Br)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCN(C)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(C#N)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CC3(CCN(C)CC3)C2)c(F)cc1Nc1ncc(C#N)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C(=O)NC2CC3(CCN(C)CC3)C2)ccc1Nc1ncc(C#N)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3(CCN(C)CC3)C2)ccc1Nc1ncc(C#N)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3(CCN(C)CC3)C2)c(F)cc1Nc1ncc(C#N)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C2CCN(C)CC2)ccc1Nc1ncc(C#N)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(C2CCN(C)CC2)c(F)cc1Nc1ncc(C#N)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC(N3CCN(C)CC3)CC2)ccc1Nc1ncc(C#N)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCN(C)CC2)c(F)cc1Nc1ncc(C#N)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CCC3(CC2)CN(C)C3)ccc1Nc1ncc(C#N)c(Oc2cccc3c2C(=O)N(C)C32CC2)n1
COc1cc(N2CC3(CCN(C)CC3)C2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CCC2)n1
COc1cc(C(=O)NC2CC3(CCN(C)CC3)C2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CCC2)n1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CCC2)n1
COc1cc(N2CC3(CCN(C)CC3)C2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CCC2)n1
COc1cc(N2CC3(CCN(C)CC3)C2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CCCC2)n1
COc1cc(C(=O)NC2CC3(CCN(C)CC3)C2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CCCC2)n1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CCCC2)n1
COc1cc(N2CC3(CCN(C)CC3)C2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CCCCC2)n1
COc1cc(N2CC3(CCN(C)CC3)C2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CCCCC2)n1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CCCCC2)n1
COc1cc(N2CC3(CCN(C)CC3)C2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CCOCC2)n1
COc1cc(N2CC3(CCN(C)CC3)C2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CCOCC2)n1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32CCOCC2)n1
COc1cc(N2CC3(CCN(C)CC3)C2)ccc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32COC2)n1
COc1cc(N2CC3(CCN(C)CC3)C2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32COC2)n1
COc1cc(C(=O)NC2CCN(C)CC2)c(F)cc1Nc1ncc(Cl)c(Oc2cccc3c2C(=O)N(C)C32COC2)n1
Cc1cc(OCCOCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)ccc1Nc1ncc(C(F)(F)F)c(NCc2cccc(N(C)S(C)(=O)=O)c2)n1
Cc1cc(Cc2ncc(C(F)(F)F)c(NCC3C=C(N(C)S(C)(=O)=O)CCC3)n2)ccc1OCCOCCOCCOc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O
Cc1cc(OCCOCCOCCOC2C=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC2)ccc1Nc1ncc(C(F)(F)F)c(NCC2=CC(P(C)(C)=O)CC=C2)n1
CN(c1nccnc1CNc1nc(Nc2ccc(C(=O)NC3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O
CN(c1nccnc1CNc1nc(Nc2ccc(C(=O)N3CCC(N4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O
CN(C1=NC=CNC1CNc1nc(Nc2ccc(CNC3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCCNC5=O)C6)CC4)CC3)cc2)ncc1CF)S(C)(=O)=O
CN(C1=NC=CNC1CNc1nc(Nc2ccc(CNC3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O
CN(C)CC[N@@](Cc1ccc(cc1)Cl)c2ccccn2
CN(C)CCN(Cc1ccc(Cl)cc1)c1ccc2ccccc2n1
[O-][N+](=O)c1cnc(\C=C/c2ccccc2Cl)n1CCOC(=O)c1cccc2OCCOc12
[O-][N+](=O)c1cnc(\C=C/c2cccc(Cl)c2)n1CCOC(=O)c1cccc2OCCOc12
[O-][N+](=O)c1cnc(\C=C/c2ccc(Cl)cc2)n1CCOC(=O)c1cccc2OCCOc12
[O-][N+](=O)c1cnc(\C=C/c2ccccc2Br)n1CCOC(=O)c1cccc2OCCOc12
[O-][N+](=O)c1cnc(\C=C/c2cccc(Br)c2)n1CCOC(=O)c1cccc2OCCOc12
[O-][N+](=O)c1cnc(\C=C/c2ccc(Br)cc2)n1CCOC(=O)c1cccc2OCCOc12
[O-][N+](=O)c1cnc(\C=C/c2ccccc2F)n1CCOC(=O)c1cccc2OCCOc12
[O-][N+](=O)c1cnc(\C=C/c2cccc(F)c2)n1CCOC(=O)c1cccc2OCCOc12
[O-][N+](=O)c1cnc(\C=C/c2ccc(F)cc2)n1CCOC(=O)c1cccc2OCCOc12
Cc1ccccc1\C=C/c1ncc(n1CCOC(=O)c1cccc2OCCOc12)[N+]([O-])=O
Cc1cccc(\C=C/c2ncc(n2CCOC(=O)c2cccc3OCCOc23)[N+]([O-])=O)c1
Cc1ccc(\C=C/c2ncc(n2CCOC(=O)c2cccc3OCCOc23)[N+]([O-])=O)cc1
COc1ccccc1\C=C/c1ncc(n1CCOC(=O)c1cccc2OCCOc12)[N+]([O-])=O
COc1cccc(\C=C/c2ncc(n2CCOC(=O)c2cccc3OCCOc23)[N+]([O-])=O)c1
COc1ccc(\C=C/c2ncc(n2CCOC(=O)c2cccc3OCCOc23)[N+]([O-])=O)cc1
[O-][N+](=O)c1cnc(\C=C/c2c(F)cccc2Cl)n1CCOC(=O)c1cccc2OCCOc12
[O-][N+](=O)c1cnc(\C=C/c2cccc3ccccc23)n1CCOC(=O)c1cccc2OCCOc12
[O-][N+](=O)c1cnc(\C=C/c2ccccc2)n1CCOC(=O)c1cccc2OCCOc12
C[C@@]12[C@@H]([C@@H](C[C@@H](O1)n3c4ccccc4c5c3c6n2c7ccccc7c6c8c5C(=O)NC8)NC)OC
C[C@H]1Oc2cc(cnc2N)-c2c(CN(C)C(=O)c3ccc(F)cc13)nn(C)c2C#N |r|
CN1CCN(CCC(=O)Nc2c(C)[nH]c(\C=C3/C(=O)Nc4ccc(F)cc34)c2C)CC1
CC(C)(C)CNC(=O)CC1CNC(=O)c2cc(cn12)-c1ccsc1
CN1CCN(C[C@@H](NC(=O)C[C@H]2CNC(=O)c3cc(cn23)-c2cccc(Cl)c2)C2CCCCC2)CC1 |r|
C[C@@]12[C@](C[C@@H](O1)n3c4ccccc4c5c3c6n2c7ccccc7c6c8c5C(=O)NC8)(CO)O
C[C@@]12[C@@H]([C@@H](C[C@@H](O1)n3c4ccccc4c5c3c6n2c7ccccc7c6c8c5C(=O)NC8)N(C)C(=O)c9ccccc9)OC
CN1CCN(CC1)CC(=O)N(C)c2ccc(cc2)N/C(=C\3/c4ccc(cc4NC3=O)C(=O)OC)/c5ccccc5
CN(c1cccc(c1)-c1ccc2cnc(Nc3ccc(cc3)C3CCN(CC(N)=O)CC3)nn12)S(C)(=O)=O
NC(=O)CN1CCC(CC1)c1ccc(Nc2ncc3ccc(-c4cccc(CO)c4)n3n2)cc1
COc1ccc(cn1)-c1ccc2cnc(Nc3ccc(cc3)C3CCN(CC(N)=O)CC3)nn12
CS(=O)(=O)Nc1cccc(c1)-c1ccc2cnc(Nc3ccc(cc3)C3CCN(CC(N)=O)CC3)nn12
CN(c1ccccc1-c1ccc2cnc(Nc3ccc(cc3)C3CCN(CC(N)=O)CC3)nn12)S(C)(=O)=O
CC(C)(C)NS(=O)(=O)c1cccc(c1)-c1ccc2cnc(Nc3ccc(cc3)C3CCN(CC(N)=O)CC3)nn12
COc1ccccc1-c1ccc2cnc(Nc3ccc(cc3)C3CCN(CC(N)=O)CC3)nn12
CN(c1ncccc1-c1ccc2cnc(Nc3ccc(cc3)C3CCN(CC(N)=O)CC3)nn12)S(C)(=O)=O
COc1cccnc1-c1ccc2cnc(Nc3ccc(cc3)C3CCN(CC(N)=O)CC3)nn12
CN(c1ccccc1-c1cc(C)c2cnc(Nc3ccc(cc3)C3CCN(CC(N)=O)CC3)nn12)S(C)(=O)=O
CS(=O)(=O)c1ccc(cc1)-c1ccc2cnc(Nc3ccc(cc3)C3CCN(CC(N)=O)CC3)nn12
CN(c1ccccc1-c1cc(Cl)c2cnc(Nc3ccc(cc3)C3CCN(CC(N)=O)CC3)nn12)S(C)(=O)=O
CS(=O)(=O)c1cccc(c1)-c1ccc2cnc(Nc3ccc(cc3)C3CCN(CC(N)=O)CC3)nn12
CCc1ccc(cc1)-c1ccc2N(C)S(=O)(=O)c3c[nH]nc3-c2c1
CN1c2ccc(NCc3ccc(cc3)C(C)(C)C)cc2-c2c(cnn2C)S1(=O)=O
CCc1ccc(cc1)-c1ccc2N(C)S(=O)(=O)c3cnn(C)c3-c2c1
CN1c2ccc(NCc3ccc(Br)cc3)cc2-c2c(cnn2C)S1(=O)=O
CN1c2ccc(NCc3ccc(F)cc3)cc2-c2c(cnn2C)S1(=O)=O
CN1c2ccc(Nc3ccc(F)cc3)cc2-c2c(cnn2C)S1(=O)=O
NC(=O)c1cc([nH]c1-c1ccccc1)-c1ccnc(N)n1
Cc1cccc(Cl)c1NC(=O)c1cnc(NC(=O)C2CC2)s1
c1cc2c(c(c1)F)c3nc(nn3c(n2)Cc4ccc5c(c4)OCO5)N
Nc1nc2c3ccc(N)cc3nc(Cc3ccc4OCOc4c3)n2n1
OCCCNc1ccc2c3ncnn3c(nc2c1)-c1ccc2OCOc2c1
c1cc2c(cc1Cc3nc4cc(ccc4c5n3nc(n5)N)NCCO)OCO2
CN1CCN(CC1)c1cc(F)c2c3nc(N)nn3c(Cc3ccc4OCOc4c3)nc2c1
c1ccc2c(c1)N3CC(=O)NN=C3CO2
Cc1cccc(c1NC(=O)c2cnc(s2)Nc3cc(nc(n3)C)N4CCN(CC4)CCO)Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(CN)cc2)nc2nccn12
COC(=O)c1ccccc1Nc1nc(Nc2ccc(CN)cc2)n2ccnc2n1
COC(=O)c1ccccc1Nc1nc(Nc2ccc(CN)cc2)nc2nccn12
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(CNC(=O)OC=C)cc2)n2ccnc2n1
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(CNC(=O)OC=C)cc2)nc2nccn12
COC(=O)c1ccccc1Nc1nc(Nc2ccc(CNC(=O)OC=C)cc2)n2ccnc2n1
COC(=O)c1ccccc1Nc1nc(Nc2ccc(CNC(=O)OC=C)cc2)nc2nccn12
CS(=O)(=O)Nc1ccccc1Nc1nc(Nc2ccc(cc2)C#N)n2ccnc2n1
CS(=O)(=O)Nc1ccccc1Nc1nc(Nc2ccc(cc2)C#N)nc2nccn12
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C#N)n2ccnc2n1
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C#N)nc2nccn12
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)n2ccnc2n1
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2nccn12
COC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)n2ccnc2n1
COC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2nccn12
CNC(=O)c1ccccc1Nc1nc(Nc2cc(OC)c(OC)c(OC)c2)n2ccnc2n1
CNC(=O)c1ccccc1Nc1nc(Nc2cc(OC)c(OC)c(OC)c2)nc2nccn12
COC(=O)c1cccc(Nc2nc(Nc3cc(OC)c(OC)c(OC)c3)n3ccnc3n2)c1
COC(=O)c1cccc(Nc2nc(Nc3cc(OC)c(OC)c(OC)c3)nc3nccn23)c1
COC(=O)c1ccccc1Nc1nc(Nc2cc(OC)c(OC)c(OC)c2)n2ccnc2n1
COC(=O)c1ccccc1Nc1nc(Nc2cc(OC)c(OC)c(OC)c2)nc2nccn12
CNC(=O)c1ccccc1Nc2c(cnc(n2)Nc3ccc(cc3OC)N4CCOCC4)Cl
COc1cc(NC2=Nc3nccn3C(Cc3ccccc3NC(C)=O)N2)cc(OC)c1OC |t:6|
COc1cc(Nc2nc(Cc3ccccc3NS(C)(=O)=O)nc3nccn23)cc(OC)c1OC
CNC(=O)c1ccccc1Cc1nc(Nc2cc(OC)c(OC)c(OC)c2)nc2nccn12
COC(=O)c1ccccc1Cc1nc(Nc2cc(OC)c(OC)c(OC)c2)nc2nccn12
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(CN)cc2)n2ccnc2n1
CNC(=O)c1ccccc1Nc2ncnc(n2)Nc3cc(c(c(c3)OC)OC)OC
c1ccc(c(c1)[C@H]2c3c[nH]nc3NC4=C2C(=O)CNC4)F
CCc1c(NC(=O)OCCn2ccnc2)cn2ncnc(Nc3ccc4n(Cc5ccccc5)ncc4c3)c12
Cc1cc(cc2c1nc([nH]2)C3=C(C=CNC3=O)NC[C@H](c4cccc(c4)Cl)O)N5CCOCC5
COc1cc2Cc3c(Nc4cccc(F)c4)[nH]nc3-c2cc1OC
CCn1nc(C#Cc2cc(ccc2C)C(=O)Nc2ccc(CN3CCN(C)CC3)c(c2)C(F)(F)F)c2c(N)ncnc12
CSc1cccc(Nc2ncc3ccn(-c4ccccn4)c3n2)c1
COc1cc(Nc2ncc3CCC(=O)N(c4ccccn4)c3n2)cc(OC)c1OC
C1CCc2c(C1)cccc2Nc1ncc2ccn(-c3ccccn3)c2n1
Cc1ccccc1Nc1ncc2ccn(-c3ccccn3)c2n1
COc1cc(Nc2ncc3ccn(-c4cccs4)c3n2)cc(OC)c1OC
C1Oc2ccc(Nc3ncc4ccn(-c5ccccn5)c4n3)cc2O1
Cc1ccc(cc1Nc1ncc2ccn(-c3ccccn3)c2n1)[N+]([O-])=O
FC(F)(F)c1ccccc1Nc1ncc2ccn(-c3ccccn3)c2n1
N(c1ccc2cc[nH]c2c1)c1ncc2ccn(-c3ccccn3)c2n1
COc1cc(Nc2ncc3CCCN(c4ccccn4)c3n2)cc(OC)c1OC
Cc1ccc(I)cc1Nc1ncc2ccn(-c3ccccn3)c2n1
Brc1ccccc1Nc1ncc2ccn(-c3ccccn3)c2n1
Cc1cc(I)ccc1Nc1ncc2ccn(-c3ccccn3)c2n1
COc1ccncc1-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
CN1CCN(CC1)c1ncc2ccn(-c3ccccn3)c2n1
COc1cc(Nc2ncc3ccn(-c4cnccc4Cl)c3n2)cc(OC)c1OC
COc1cccc(Nc2ncc3ccn(-c4ccccn4)c3n2)c1
COc1ccc(C)c(Nc2ncc3ccn(-c4ccccn4)c3n2)c1
CC(C)c1ccccc1Nc1ncc2ccn(-c3ccccn3)c2n1
COc1cc(Nc2ncc3ccn(-c4ccc(C)cn4)c3n2)cc(OC)c1OC
Cc1ccc(cc1Nc1ncc2ccn(-c3ccccn3)c2n1)-c1cnc2ccccc2n1
CCOC(=O)Cc1cnc(Nc2cc(OC)c(OC)c(OC)c2)nc1Nc1ccccn1
COc1cc(Nc2ncc3ccn(-c4ccnc(Cl)c4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4ccncc4)c3n2)cc(OC)c1OC
C(Nc1ncc2ccn(-c3ccccn3)c2n1)c1ccccc1
Cc1ccc(CO)cc1Nc1ncc2ccn(-c3ccccn3)c2n1
COc1cc(Nc2ncc3ccn(-c4nccc(Cl)n4)c3n2)cc(OC)c1OC
O=C1CCCN1CCCNc1ncc2ccn(-c3ccccn3)c2n1
CCc1ccccc1Nc1ncc2ccn(-c3ccccn3)c2n1
COc1cc(Nc2ncc3ccc(=O)n(-c4ccccn4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(Cc4cccnc4)c3n2)cc(OC)c1OC
COc1cc(CNc2ncc3ccn(-c4ccccn4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccnc4)c3n2)cc(OC)c1OC
Oc1cccc(Nc2ncc3ccn(-c4ccccn4)c3n2)c1
COc1cc(Nc2ncc3ccn(-c4nccs4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(CCc4ccncc4)c3n2)cc(OC)c1OC
FC(F)(F)c1ccc(Nc2ncc3ccn(-c4ccccn4)c3n2)cc1
Clc1ccccc1Nc1ncc2ccn(-c3ccccn3)c2n1
COc1cc(Nc2ncc3ccn(CCc4cccnc4)c3n2)cc(OC)c1OC
Cc1ccc(cc1Nc1ncc2ccn(-c3ccccn3)c2n1)C(N)=O
COc1cc(Nc2ncc3ccn(-c4ccccn4)c3n2)cc(OC)c1OC
CSc1ccccc1Nc1ncc2ccn(-c3ccccn3)c2n1
COc1cc(Nc2ncc3ccn(-c4cnccc4F)c3n2)cc(OC)c1OC
Cc1ccc(Br)cc1Nc1ncc2ccn(-c3ccccn3)c2n1
CCOC(=O)Cc1cnc(Nc2cc(OC)c(OC)c(OC)c2)nc1Cl
COc1cc(Nc2ncc(Br)c(Nc3ccccn3)n2)cc(OC)c1OC
COc1cc(Nc2ncc3CC(=O)N(c3n2)c2ccccn2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4ccnc(Cl)n4)c3n2)cc(OC)c1OC
Fc1ccccc1Nc1ncc2ccn(-c3ccccn3)c2n1
COc1cc(Nc2ncc3CCN(c3n2)c2ccccn2)cc(OC)c1OC
COc1ccccc1Nc1ncc2ccn(-c3ccccn3)c2n1
COc1cc(Nc2ncc3CCC(O)N(c4ccccn4)c3n2)cc(OC)c1OC
Cc1cccc(Nc2ncc3ccn(-c4ccccn4)c3n2)c1
C1CN(CCO1)c1ncc2ccn(-c3ccccn3)c2n1
COC(=O)CNC(=O)Cc1cccc(c1)-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
COc1cc(Nc2ncc3ccn(-c4ccc(C)cc4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(CC(=O)NCCN)c4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(c4)C(=O)NCCN4CCCC4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(CCc5nnn[nH]5)c4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(c4)C(=O)NCCNC(C)=O)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(CN)c4)c3n2)cc(OC)c1OC
COC(=O)c1ccccc1-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
CNC(=O)c1cccc(c1)-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
CNC(=O)Cc1cccc(c1)-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
COc1cc(Nc2ncc3ccn(-c4cccc(c4)C(=O)NCCN)c3n2)cc(OC)c1OC
COC(=O)CNC(=O)CCc1cccc(c1)-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
COc1cc(Nc2ncc3ccn(-c4ccc(cc4)C(O)=O)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(CCC(O)=O)c4)c3n2)cc(OC)c1OC
CCc1ccccc1-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
CCNC(=O)c1cccc(c1)-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
COc1cc(Nc2ncc3ccn(-c4cccc(c4)C(N)=O)c3n2)cc(OC)c1OC
CCCNS(=O)(=O)c1ccccc1-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
CCc1ccc(cc1)-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
COc1cc(Nc2ncc3ccn(-c4cccc(CC(=O)NC5CCCC5)c4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4ccccc4C(=O)NCCN)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(n4)C(=O)NCCC#N)c3n2)cc(OC)c1OC
CCNC(=O)Cc1cccc(c1)-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
COc1cc(Nc2ncc3ccn(-c4ccccc4C(=O)NCCCN(C)C)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(CC#N)c4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4ccccc4[N+]([O-])=O)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(CC(=O)NC5CC5)c4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4ccc(SC)cc4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(c4)C(=O)NCCCN(C)C)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(c4)C#N)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4ccccc4N)c3n2)cc(OC)c1OC
CNC(=O)c1cccc(n1)-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
COc1cc(Nc2ncc3ccn(-c4cccc(c4)C(=O)NC4CCCC4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(n4)C(=O)NCC(C)C)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4ccc(cc4)C(C)(C)C)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(c4)C(=O)NCC(C)C)c3n2)cc(OC)c1OC
COC(=O)c1cccc(c1)-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
CCNC(=O)CCc1cccc(c1)-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
COc1cc(Nc2ncc3ccn(-c4ccc(cc4)[N+]([O-])=O)c3n2)cc(OC)c1OC
CCCCc1ccc(cc1)-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
COc1cc(Nc2ncc3ccn(-c4ccccc4CO)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(n4)C(=O)NCCCN)c3n2)cc(OC)c1OC
CNS(=O)(=O)c1cccc(c1)-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
COc1cc(Nc2ncc3ccn(-c4ccccc4NC(C)=O)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(CCC(=O)NCCN(C)C)c4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(c4)C(=O)NCCN(C)C)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(CCC#N)c4)c3n2)cc(OC)c1OC
CNC(=O)c1ccccc1-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
COc1cc(Nc2ncc3ccn(-c4ccccc4C(O)=O)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(c4)C(=O)NC4CC4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4ccccc4C(N)=O)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4ccccc4C#N)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(c4)C(=O)NCCO)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(c4)C(O)=O)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(CC(O)=O)c4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(CCC(=O)NCC(C)C)c4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(c4)C(=O)NCCCO)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4ccc(cc4)C(F)(F)F)c3n2)cc(OC)c1OC
CNC(=O)CCc1cccc(c1)-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
COc1cc(Nc2ncc3ccn(-c4cccc(CC(=O)NCCCN)c4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(N)c4)c3n2)cc(OC)c1OC
COC(=O)CNC(=O)c1cccc(n1)-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
COc1cc(Nc2ncc3ccn(-c4cccc(n4)C(=O)NCCN)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(C)c4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(c4)C(=O)NCCCCN(C)C)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(CCC(O)=O)n4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(n4)C(=O)NCC#N)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3cc(C(O)=O)n(-c4ccccn4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(c4)-c4nnn[nH]4)c3n2)cc(OC)c1OC
COC(=O)c1ccc(cc1)-n1ccc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
COC(=O)c1cc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc2n1-c1ccccn1
COc1cc(Nc2ncc3ccn(-c4cccc(Cc5nnn[nH]5)c4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4ccccc4C)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(CC(=O)NCCCN(C)C)c4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(c4)C(F)(F)F)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3ccn(-c4cccc(n4)C(=O)NCCN(C)C)c3n2)cc(OC)c1OC
NC(=O)c1cnc2[nH]ccc2c1N[C@@H]1CCN(C[C@@H]1F)c1ccc(cn1)C#N |r|
COc1cc(cc(OC)c1OC)C1=C(C(=O)NC1=O)c1c[nH]c2ccccc12 |t:13|
CS(=O)(=O)c1cccc(c1)CNc2c(cnc(n2)Nc3ccc4c(c3)CCC(=O)N4)C(F)(F)F
c1c(cc(c2c1CN(C2=O)C3CCN(CC3)C4CCC(CC4)(F)F)C(=O)N)F
COc1cc(cc(OC)c1OC)C1=C(C(=O)NC1)c1cn(C)c2ccccc12 |t:13|
COc1cc(cc(OC)c1OC)C1=C(CNC1=O)c1cn(COCc2ccccc2)c2ccccc12 |t:13|
COc1cc(cc(OC)c1OC)C1=C(CNC1=O)c1cn(COc2ccccc2)c2ccccc12 |t:13|
COc1cc(cc(OC)c1OC)C1=C(CNC1=O)c1cn(COC(C)(C)C)c2ccccc12 |t:13|
COc1cc(cc(OC)c1OC)C1=C(CNC1=O)c1cn(COC(C)C)c2ccccc12 |t:13|
CCOCn1cc(C2=C(C(=O)NC2)c2cc(OC)c(OC)c(OC)c2)c2ccccc12 |t:7|
COCn1cc(C2=C(C(=O)NC2)c2cc(OC)c(OC)c(OC)c2)c2ccccc12 |t:6|
COc1cc(cc(OC)c1OC)C1=C(CNC1=O)c1c[nH]c2ccccc12 |t:13|
CN(c1cccc(CNc2nc(Nc3ccc4NC(=O)Cc4c3)ncc2C(F)(F)F)c1)S(C)(=O)=O
CS(=O)(=O)c1cccc(CNc2nc(Nc3ccc4NC(=O)Cc4c3)ncc2C(F)(F)F)c1
CS(=O)(=O)c1ccccc1CNc1nc(Nc2ccc3NC(=O)Cc3c2)ncc1C(F)(F)F
FC(F)(F)c1cnc(Nc2ccc3NC(=O)Cc3c2)nc1NCc1ccccc1S(=O)(=O)N1CCCC1
FC(F)(F)c1cnc(Nc2ccc3NC(=O)Cc3c2)nc1N[C@@H]1CCCCNC1=O |r|
CN(C)[C@@H]1CCC[C@H]1Nc1nc(Nc2ccc3NC(=O)Cc3c2)ncc1C(F)(F)F |r|
FC(F)(F)c1cnc(Nc2ccc3NC(=O)CCc3c2)nc1NCc1ccccn1
CN(c1ccccc1CNc1nc(Nc2ccc3C(=O)NCc3c2)ncc1C(F)(F)F)S(C)(=O)=O
CN(C)[C@@H]1CCC[C@H]1Nc1nc(Nc2ccc3c(CCCNC3=O)c2)ncc1C(F)(F)F |r|
CN(C)[C@@H]1CCC[C@H]1Nc1nc(Nc2ccc3c(CCS3(=O)=O)c2)ncc1C(F)(F)F |r|
CN(c1ccccc1CNc2c(cnc(n2)Nc3ccc4c(c3)CC(=O)N4)C(F)(F)F)S(=O)(=O)C
Cn1ccc2cc(Nc3ncc(c(NCc4ccccn4)n3)C(F)(F)F)ccc12
FC(F)(F)c1cnc(Nc2ccc3[nH]ncc3c2)nc1NCc1ccccn1
O=C1Cc2cc(Nc3nccc(NCc4ccccn4)n3)ccc2N1
Cc1cnc(Nc2ccc3NC(=O)Cc3c2)nc1NCc1ccccn1
Clc1cnc(Nc2ccc3NC(=O)Cc3c2)nc1NCc1ccccn1
Brc1cnc(Nc2ccc3NC(=O)Cc3c2)nc1NCc1ccccn1
O=C1Cc2cc(Nc3ncc(C#N)c(NCc4ccccn4)n3)ccc2N1
FC(F)(F)c1cnc(Nc2ccc3NC(=O)Cc3c2)nc1NCc1ccccn1
FC(F)(F)c1cnc(Nc2ccc3NC(=O)Cc3c2)nc1NCc1ccccc1
CN(C)[C@@H]1CCC[C@H]1Nc1nc(Nc2ccc3c(CN(C)S3(=O)=O)c2)ncc1C(F)(F)F |r|
CN(C)[C@@H]1CCC[C@H]1Nc1nc(Nc2ccc(cc2)S(C)(=O)=O)ncc1C(F)(F)F |r|
CN(c1ccccc1CNc1nc(Nc2ccc(cc2)S(C)(=O)=O)ncc1C(F)(F)F)S(C)(=O)=O
CNS(=O)(=O)c1ccc(Nc2ncc(c(N[C@@H]3CCC[C@H]3N(C)C)n2)C(F)(F)F)cc1 |r|
CCN(CC)C(=O)c1ccc(Nc2ncc(c(N[C@@H]3CCC[C@H]3N(C)C)n2)C(F)(F)F)cc1 |r|
CN(C)[C@@H]1CCC[C@H]1Nc1nc(Nc2cccc(c2)C(=O)N(C)C)ncc1C(F)(F)F |r|
CN(C)[C@@H]1CCC[C@H]1Nc1nc(Nc2ccc3C4CCC(N4C(C)=O)c3c2)ncc1C(F)(F)F |r,TLB:26:25:19.18:21,THB:15:16:19.18:21,22:21:19.18:16.25|
CN(C)[C@@H]1CCC[C@H]1Nc1nc(Nc2ccncc2)ncc1C(F)(F)F |r|
CN(c1ccccc1CNc1nc(Nc2ccc3NS(=O)(=O)Cc3c2)ncc1C(F)(F)F)S(C)(=O)=O
CN(C)[C@@H]1CCC[C@H]1Nc1nc(Nc2ccc3NS(=O)(=O)Cc3c2)ncc1C(F)(F)F |r|
CCS(=O)(=O)Nc1ccc2c(c1)C(C(=O)N2)/C(=N/c3ccc(cc3)CN4CCCCC4)/c5ccccc5
NC(=N)SCCCn1c(=O)c2c(n3c(cc4ccccc34)c3cccc4ccn2c34)c1=O
Nc1ncc(NC(=O)c2cc(NC(=O)c3cccc(c3)C(F)(F)F)ccc2Cl)cc1Cl
Cn1c2nc(Nc3ccc4[nH]ccc4c3)ncc2cc(c1=O)S(=O)(=O)c1ccc(F)cc1F
Oc1ccc(NC(=S)NC(=O)c2ccc(cc2)[N+]([O-])=O)cc1-c1nc2ccccc2s1
C[C@@H]1C[C@H]1C(=O)N1CCN(C[C@H]1C)c1cnc(C#N)c(n1)-c1cnn(C)c1 |r|
C[C@@H](N1c2cc(ccc2C(=O)NC1(C)C)-n1c2cccnc2[nH]c1=O)c1ccccc1 |r|
CN1CCN(CC1)c2ccc(c(c2)NC3CCOCC3)C(=O)Nc4c5cc(ccc5[nH]n4)Cc6cc(cc(c6)F)F
COc1cc(cc(OC)c1OC)-c1nc(c[nH]c1=O)-c1c[nH]c2ccccc12
[H][C@@]12C[C@@]([H])(C=C1)[C@@H]([C@@H]2Nc1nc(Nc2ccc3C[C@H](CCCc3c2OC)N2CCN(C)CC2)ncc1Cl)C(N)=O |r,c:5|
CNC(=O)c1ccccc1Nc1nc(Nc2ccc3CC(CCCc3c2OC)N2CCN(CCO)CC2)ncc1Cl
COc1c(Nc2ncc(Cl)c(Nc3ccccc3N3CCCS3(=O)=O)n2)ccc2CC(CCCc12)N1CCN(CCO)CC1
[H][C@@]12C[C@@]([H])(C=C1)[C@@H]([C@@H]2Nc1nc(Nc2ccc3C[C@@H](CCCc3c2OC)N2CCN(C)CC2)ncc1Cl)C(N)=O |r,c:5|
COc1c(Nc2ncc(Cl)c(Nc3ccccc3N(C)S(C)(=O)=O)n2)ccc2CC(CCCc12)N1CCN(CCO)CC1
COc1c(Nc2ncc(Cl)c(Nc3ccccc3-c3nccn3C)n2)ccc2CC(CCCc12)N1CCN(CCO)CC1
COc1ccccc1Nc1nc(Nc2ccc3CC(CCCc3c2OC)N2CCN(CCO)CC2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc3C[C@@H](CCCc3c2OC)N2CCN(CCO)CC2)ncc1Cl |r|
COc1c(Nc2ncc(Cl)c(N[C@@H]3[C@@H]4C[C@@H](C=C4)[C@@H]3C(N)=O)n2)ccc2CC[C@@H](CCc12)N1CCOCC1 |r,c:16|
CNC(=O)c1ccccc1Nc1nc(Nc2ccc3C[C@H](CCCc3c2OC)N2CCN(CCO)CC2)ncc1Cl |r|
COc1c(Nc2ncc(Cl)c(Nc3ccccc3N(C)S(C)(=O)=O)n2)ccc2CC(CCCc12)N1CCN(C)CC1
COc1c(Nc2ncc(Cl)c(Nc3ccccc3NS(C)(=O)=O)n2)ccc2CC(CCCc12)N1CCN(CCO)CC1
COc1c(Nc2ncc(Cl)c(Nc3ccccc3-n3cccn3)n2)ccc2CC(CCCc12)N1CCN(CCO)CC1
CS(=O)(=O)N(CC=C)c1ncccc1CNc1nc(Nc2ccc(N3CCOCC3)c(Br)c2)ncc1C(F)(F)F
CCS(=O)(=O)N1CCCCC(=O)N2CCc3cc(Nc4ncc(c(NCc5ccccc15)n4)C(F)(F)F)ccc23
CN(c1c(cccn1)CNc2c(cnc(n2)Nc3ccc4c(c3)CC(=O)N4)C(F)(F)F)S(=O)(=O)C
FC(F)(F)c1cnc2Nc3ccc4N(CCc4c3)C(=O)CCCNS(=O)(=O)c3ncccc3CNc1n2
CS(=O)(=O)N1C\C=C\c2cccc(Nc3ncc(c(NCc4cccnc14)n3)C(F)(F)F)c2 |t:6|
CN1Cc2cccnc2N(C\C=C\c2cc(Nc3ncc(c1n3)C(F)(F)F)ccc2N1CCOCC1)S(C)(=O)=O |t:12|
CN1Cc2ccncc2N(C\C=C\c2cc(Nc3ncc(c1n3)C(F)(F)F)ccc2N1CCOCC1)S(C)(=O)=O |t:12|
CN(Cc1ccncc1N(CC=C)S(C)(=O)=O)c1nc(Nc2ccc(N3CCOCC3)c(Br)c2)ncc1C(F)(F)F
CS(=O)(=O)N1CCCc2cccc(Nc3ncc(c(NCc4cccnc14)n3)C(F)(F)F)c2
CN(Cc1ccccc1N(CCCCC(O)=O)S(C)(=O)=O)c1nc(Nc2ccc3NCCc3c2)ncc1C(F)(F)F
CCS(=O)(=O)N(CCCCC(O)=O)c1ccccc1CNc1nc(Nc2ccc3NCCc3c2)ncc1C(F)(F)F
CS(=O)(=O)N1CCCCC(=O)N2CCc3c2ccc(c3)Nc4ncc(c(n4)NCc5c1nccc5)C(F)(F)F
CS(=O)(=O)N1Cc2cccc(c2)C(=O)N2CCc3cc(Nc4ncc(c(NCc5cccnc15)n4)C(F)(F)F)ccc23
CN1Cc2ccccc2N(CCCCC(=O)N2CCc3cc(Nc4ncc(c1n4)C(F)(F)F)ccc23)S(C)(=O)=O
CS(=O)(=O)N1C\C=C\c2cc(Nc3ncc(c(NCc4cccnc14)n3)C(F)(F)F)ccc2N1CCOCC1 |t:6|
CS(=O)(=O)N1CCCc2cc(Nc3ncc(c(NCc4cccnc14)n3)C(F)(F)F)ccc2N1CCOCC1
CS(=O)(=O)N1CCCCC(=O)N2CCc3cc(Nc4ncc(c(NCc5ccccc15)n4)C(F)(F)F)ccc23
CS(=O)(=O)N1CCCC(=O)N2CCc3cc(Nc4ncc(c(NCc5cccnc15)n4)C(F)(F)F)ccc23
CS(=O)(=O)N(CC=C)c1ncccc1CNc1nc(Nc2cccc(Br)c2)ncc1C(F)(F)F
CNC(=O)c1nn(C)c-2c1CCc1cnc(NC3CCN(CC3)C(=O)C3CCN(CC3)S(C)(=O)=O)nc-21
CC(=O)N1CCC(CC1)Nc1ncc2CCc3c(nn(C)c3-c2n1)C(N)=O
Cn1nc(C(N)=O)c2CCc3cnc(NC4CCN(CC4)C(=O)c4ccccc4)nc3-c12
CN1CCN(CC1)CCCOc2cc3c(cc2OC)c(c(cn3)C#N)Nc4cc(c(cc4Cl)Cl)OC
CC(C)(C)c1cc(NC(=O)Nc2ccc(cc2)-c2cn3c(n2)sc2cc(OCCN4CCOCC4)ccc32)no1
COc1cc2c(ncnc2cc1OCCCN1CCCCC1)N1CCN(CC1)C(=O)Nc1ccc(OC(C)C)cc1
CNC(=O)c1cc(ccn1)Oc2ccc(cc2)NC(=O)Nc3ccc(c(c3)C(F)(F)F)Cl
CO[C@@H]1[C@@H](C[C@H]2O[C@]1(C)n1c3ccccc3c3c4[C@H](O)NC(=O)c4c4c5ccccc5n2c4c13)N(C)C(=O)c1ccccc1 |r|
Cn1ccc2c1c(ncn2)Oc3ccc(c(c3)F)NC(=O)Nc4cccc(c4)C(F)(F)F
Cc1n[nH]c2Nc3ccc(cc3C(=Nc12)c1ccccc1Cl)[N+]([O-])=O |c:13|
Fc1ccccc1C1=Nc2cn[nH]c2Nc2ccc(cc12)C#N |t:8|
Nc1ccc2Nc3[nH]ncc3N=C(c3ccccc3Cl)c2c1 |t:12|
CC(=O)Nc1ccc2Nc3[nH]ncc3N=C(c3ccccc3Cl)c2c1 |t:15|
COc1ccc2cc([nH]c2c1)-c1n[nH]c2cccnc12
COc1ccc(CNc2ccnc3oc4ccccc4c23)cc1
CNc1cncc(n1)-c1c[nH]c(=O)c(NC(=O)c2ccc(cc2)N2CCC[C@H]2CN2CCCC2)c1 |r|
CN1CCN(CC1)c1ccc(OC(F)(F)F)c(Nc2ncc3CCc4c(nn(CCO)c4-c3n2)C(N)=O)c1
CN(C)[C@@H]1CCC[C@H]1Nc1nc(Nc2ccc(cc2)S(=O)(=O)NC2CC2)ncc1C(F)(F)F |r|
Cc1cc(O)cc2oc3cc(O)cc(O)c3c(=O)c12
Cc1c(O)c(O)cc2oc3cc(O)cc(O)c3c(=O)c12
CCN1CCN(CC1)c2ccc(cc2)Nc3cc(ncn3)N(C)C(=O)Nc4c(c(cc(c4Cl)OC)OC)Cl
CCN1CCN(Cc2ccc(NC(=O)Nc3ccc(Oc4cc(NC)ncn4)cc3)cc2C(F)(F)F)CC1
COc1cc2c(Oc3ccc4[nH]c(C)cc4c3F)ncnc2cc1OCCCN1CCCC1
CN1CCC(CC1)COc2cc3c(cc2OC)c(ncn3)Nc4ccc(cc4F)Br
CCOc1cc2ncc(C#N)c(Nc3ccc(OCc4ccccn4)c(Cl)c3)c2cc1NC(=O)\C=C\CN(C)C
Cn1cc(C2=C(C(=O)NC2=O)c2cn(C3CCN(Cc4ccccn4)CC3)c3ccccc23)c2ccccc12 |t:4|
C[C@@H]1CCN(C[C@@H]1N(C)c1ncnc2[nH]ccc12)C(=O)CC#N |r|
CN(C)C[C@@H]1CCn2cc(C3=C(C(=O)NC3=O)c3cn(CCO1)c1ccccc31)c1ccccc21 |r,t:10|
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(OCCN2CCOCC2)c2ccccc12)C(C)(C)C
CNC(=O)c1c(F)cccc1Nc1nc(Nc2cc3N(CCc3cc2OC)C(=O)CN(C)C)nc2[nH]ccc12
Cc1cnc(nc1Nc2cccc(c2)S(=O)(=O)NC(C)(C)C)Nc3ccc(cc3)OCCN4CCCC4
CC(C)S(=O)(=O)c1ccccc1Nc2c(cnc(n2)Nc3ccc(cc3OC)N4CCC(CC4)N5CCN(CC5)C)Cl
c1c[nH]c2c1c(ncn2)c3cnn(c3)[C@H](CC#N)C4CCCC4
COc1ccc(c(c1C(=O)c2cnc(nc2N)NC3CCN(CC3)S(=O)(=O)C)F)F
C[C@@H](O)COc1cn2ncnc(Oc3ccc4[nH]c(C)cc4c3F)c2c1C
CN1CC[C@@H]([C@H](O)C1)c1c(O)cc(O)c2c1oc(cc2=O)-c1ccccc1Cl |r|
CS(=O)c1ccc(cc1)-c1nc(c([nH]1)-c1ccc(F)cc1)-c1ccncc1
CN(C)C/C=C/C(=O)Nc1cc2c(cc1O[C@H]3CCOC3)ncnc2Nc4ccc(c(c4)Cl)F
Clc1cccc(Cl)c1C(=O)Nc1cn[nH]c1C(=O)NC1CCNCC1
CS(=O)(=O)CCNCc1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
Cn1c(Nc2ccc(cc2)C(F)(F)F)nc2cc(Oc3ccnc(c3)-c3ncc([nH]3)C(F)(F)F)ccc12
Nc1nc(N)c2nc(-c3cccc(O)c3)c(nc2n1)-c1cccc(O)c1
C[C@@H](Oc1cc(sc1C(N)=O)-n1cnc2ccc(CN3CCN(C)CC3)cc12)c1ccccc1C(F)(F)F |r|
CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)CC1
CCN(CCCOc1ccc2c(c1)ncnc2Nc3cc(n[nH]3)CC(=O)Nc4cccc(c4)F)CCO
COc1c(Cl)cc2c3ccncc3[nH]c2c1NC(=O)c1cccnc1C
CC[C@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2N(C)C1=O |r|
CNC(=O)c1ccccc1Sc2ccc3c(c2)[nH]nc3/C=C/c4ccccn4
CN1c2c(cnc(n2)Nc3cccc(c3)SC)C=C(C1=O)c4c(cccc4Cl)Cl
Clc1ccc(Nc2nnc(Cc3ccncc3)c3ccccc23)cc1
CN(c1ccc2c(C)n(C)nc2c1)c1ccnc(Nc2ccc(C)c(c2)S(N)(=O)=O)n1
Cc1n[nH]c2ccc(cc12)-c1cncc(OC[C@@H](N)Cc2ccccc2)c1 |r|
C[C@@H](Oc1cc(cnc1N)-c1cnn(c1)C1CCNCC1)c1c(Cl)ccc(F)c1Cl |r|
c1cc(c(c(c1)Cl)C2=C3C=CC(=NN3C=NC2=O)Sc4ccc(cc4F)F)Cl
COc1cc2c(cc1OCCCN3CCOCC3)c(ncn2)Nc4ccc(c(c4)Cl)F
CC(C)n1nc(-c2cc3cc(O)ccc3[nH]2)c2c(N)ncnc12
CC1(CNc2c1ccc(c2)NC(=O)c3cccnc3NCc4ccncc4)C
COc1cc2c(Oc3ccc(NC(=O)C4(CC4)C(=O)NC4=CCC(F)C=C4)cc3F)ccnc2cc1OCCCN1CCOCC1 |c:26,t:21|
CC(C)(C)c1cnc(o1)CSc2cnc(s2)NC(=O)C3CCNCC3
Fc1ccc(C(=O)NOCC2CC2)c(Nc2ccc(I)cc2Cl)c1F
COc1cc(Oc2ccnc3cc(OC)c(OC)cc23)ccc1NC(=O)NC(C)c1nccs1
CC1(C(=O)Nc2c(ccc(n2)Nc3c(cnc(n3)Nc4cc(c(c(c4)OC)OC)OC)F)O1)C
CN1CCN(CC1)c1ccc2nc([nH]c2c1)-c1c(N)c2c(F)cccc2[nH]c1=O
CN1CCN(CC1)c1cc(Nc2cc(C)n[nH]2)nc(Sc2ccc(NC(=O)C3CC3)cc2)n1
COCCOc1cc2c(cc1OCCOC)ncnc2Nc3cccc(c3)C#C
OC(=O)c1ccc(Nc2ncc3CN=C(c4cc(Cl)ccc4-c3n2)c2c(F)cccc2F)cc1 |c:13|
CN(C)CC(=O)N1CCC(CC1)c1ccc(NC(=O)c2ncc([nH]2)C#N)c(c1)C1=CCCCC1 |t:31|
Cc1ccc(cc1Nc2nc(cs2)c3cccnc3)NC(=O)c4ccc(cc4)CN5CCN(CC5)C
Cn1cc(cn1)-c1ccc2nnc(Sc3ccc4ncccc4c3)n2n1
Cc1[nH]c(\C=C2/C(=O)Nc3ccc(cc23)S(=O)(=O)Cc2c(Cl)cccc2Cl)c(C)c1C(=O)N1CCC[C@@H]1CN1CCCC1 |r|
C=CC(=O)Nc1cc2c(cc1OCCCN3CCOCC3)ncnc2Nc4ccc(c(c4)Cl)F
CS(=O)(=O)N1CCN(Cc2cc3nc(nc(N4CCOCC4)c3s2)-c2cccc3[nH]ncc23)CC1
CCn1c(nc2c(ncc(OC[C@H]3CCCNC3)c12)C#CC(C)(C)O)-c1nonc1N |r|
Cn1cnc2c1cc(c(c2F)Nc3ccc(cc3Cl)Br)C(=O)NOCCO
Oc1cccc(c1)-c1nc(N2CCOCC2)c2oc3ncccc3c2n1
OCCn1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
Cc1cn(cn1)-c1cc(NC(=O)c2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)cc(c1)C(F)(F)F
Cc1cnc2c(NCCN)nc3ccc(C)cc3n12
O=C(N1CCNCC1)c1ccc(\C=C\c2n[nH]c3ccccc23)cc1
COc1ccc(cc1)COc2ccc(cc2OC)Cc3cnc(nc3N)N
Cc1ccc(F)c(NC(=O)Nc2ccc(cc2)-c2cccc3[nH]nc(N)c23)c1
CC(C)C\C=C\[C@@H](C)[C@H]1CC[C@H]2[C@H](CCc3cc(O)ccc3C)[C@@H](O)CC[C@]12C |r|
CC(C)C\C=C\[C@@H](C)[C@H]1CC[C@H]2[C@H](CCc3cc(O)ccc3C)C(=O)CC[C@]12C |r|
CC(C)C(=C)CC[C@@H](C)[C@H]1CC[C@H]2[C@H](CCc3cc(O)ccc3C)C(=O)CC[C@]12C |r|
CC(C)CCC[C@@H](C)[C@H]1CC[C@H]2[C@H](CCc3cc(O)ccc3C)C(=O)CC[C@]12C |r|
CC(C)CCC[C@@H](C)[C@H]1CC[C@H]2[C@H](CCc3cc(O)ccc3C)[C@H](O)CC[C@]12C |r|
CC(C)CCC[C@@H](C)[C@H]1[C@@H](O)C[C@H]2[C@H](CCc3cc(O)ccc3C)C(=O)CC[C@]12C |r|
CC(C)C(=C)CC[C@@H](C)[C@H]1CC[C@H]2[C@H](CCc3cc(O)ccc3C)[C@H](O)CC[C@]12C |r|
CC(C)CCC[C@@H](C)[C@H]1[C@@H](O)C[C@H]2[C@H](CCc3cc(O)ccc3C)[C@H](O)CC[C@]12C |r|
CC(C)(CC(=O)NCCn1ccc2c1c(ncn2)Nc3ccc(c(c3)Cl)Oc4cccc(c4)C(F)(F)F)O
CC(C)(C)c1cc(c(s1)NC(=O)Nc2cccc(c2Cl)Cl)C(=O)N3CCC(=O)N(CC3)CCN(C)C
COc1cc(Nc2ncc3ccc(-c4ccccc4)n3n2)cc(OC)c1OC
COc1cc(ccc1Nc1ncc2ccc(-c3ccccc3OC)n2n1)C1CCN(CC(N)=O)CC1
NC(=O)CN1CCC(CC1)c1ccc(Nc2ncc3ccc(-c4ncccn4)n3n2)cc1
NC(=O)CN1CCC(CC1)c1ccc(Nc2ncc3ccc(-c4cnccn4)n3n2)cc1
NC(=O)CN1CCC(CC1)c1ccc(Nc2ncc3ccc(-c4cccc5OC(F)(F)Oc45)n3n2)cc1
CN(C)Cc1ccc(cc1)-c1ccc2cnc(Nc3ccc(cc3)C3CCN(CC(N)=O)CC3)nn12
CS(=O)(=O)N1Cc2cccc(c2C1)-c1ccc2cnc(Nc3ccc(cc3)C3CCN(CC(N)=O)CC3)nn12
NC(=O)CN1CCC(CC1)c1ccc(Nc2ncc3ccc(-c4cccc5cccnc45)n3n2)cc1
CC(=O)OC[C@H]1O[C@@H](O[C@@H]2[C@@H](COC(C)=O)O[C@H]([C@H](OC(C)=O)[C@H]2OC(C)=O)n2[se]c3ccccc3c2=O)[C@H](OC(C)=O)[C@@H](OC(C)=O)[C@H]1OC(C)=O |r|
CC(=O)OC[C@H]1O[C@@H](NC(=O)CCCn2[se]c3ccccc3c2=O)[C@H](OC(C)=O)[C@@H](OC(C)=O)[C@@H]1OC(C)=O |r|
OC[C@H]1O[C@@H](NC(=O)CCCn2[se]c3ccccc3c2=O)[C@H](O)[C@@H](O)[C@@H]1O |r|
Cn1c2c(C(C#N)C3(CCNCC3)NC2=O)c2ccc(Cl)c(Cl)c12
COc1ccc(cc1\C=C\c1ccc(Cl)cc1)C(=O)NC[C@@H](O)CO |r|
COc1ccc(cc1\C=C\c1ccc(Cl)cc1)C(=O)NC[C@H](O)CO |r|
CC(C)n1c2CCCC(=O)c2c2C(=O)c3ccccc3-c12
c1c2c-3c(c(c1O)O)OC(=O)c4c3c(c(c(c4)O)O)OC2=O
COc1cc2ncccc2cc1NC(=O)c1csc2cncnc12
Cc1c2ccc(cc2[nH]n1)Nc3nc4ccoc4c(n3)NC5CC5
CCCNC(=O)c1ccc(Nc2nc(NCC(F)(F)F)c3cc[nH]c3n2)cc1
CC1(C)OCC(=O)Nc2cc(Nc3nc(NCC(F)(F)F)c4occc4n3)ccc12
FC(F)(F)CNc1nc(Nc2ccc3cn[nH]c3c2)nc2ccoc12
FC(F)(F)CNc1nc(Nc2ccc(N3CCOCC3)c(Cl)c2)nc2ccoc12
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nnc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)N2CCOCC2)nnc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2cc(C)c(Cl)cc2OC)nnc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2cc(OC)c(OC)c(OC)c2)nnc1Cl
COc1cc(Nc2nnc(Cl)c(Nc3cccc(NS(C)(=O)=O)c3)n2)cc(OC)c1OC
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(CN)cc2)nnc1Cl
COc1ccc(cc1)N1CCN(Cn2nc(oc2=S)-c2ccc3OCCOc3c2)CC1
S=c1oc(nn1CN1CCN(CC1)C(c1ccccc1)c1ccccc1)-c1ccc2OCCOc2c1
COc1ccccc1N1CCN(Cn2nc(oc2=S)-c2ccc3OCCOc3c2)CC1
S=c1oc(nn1CN1CCN(CC1)c1ccccn1)-c1ccc2OCCOc2c1
FC(F)(F)c1cccc(c1)N1CCN(Cn2nc(oc2=S)-c2ccc3OCCOc3c2)CC1
COc1cccc(c1)N1CCN(Cn2nc(oc2=S)-c2ccc3OCCOc3c2)CC1
S=c1oc(nn1CN1CCN(Cc2ccccc2)CC1)-c1ccc2OCCOc2c1
[O-][N+](=O)c1ccc(cc1)N1CCN(Cn2nc(oc2=S)-c2ccc3OCCOc3c2)CC1
Clc1ccccc1N1CCN(Cn2nc(oc2=S)-c2ccc3OCCOc3c2)CC1
Clc1ccc(cc1Cl)N1CCN(Cn2nc(oc2=S)-c2ccc3OCCOc3c2)CC1
CC1C\C(=C/c2nc(C)c(C)nc2C)C(=O)\C(C1)=C\c1nc(C)c(C)nc1C
CC(C)N1C\C(=C/c2nc(C)c(C)nc2C)C(=O)\C(C1)=C\c1nc(C)c(C)nc1C
COc1cc(Br)c(\C=C2/CC(C)C\C(=C/c3nc(C)c(C)nc3C)C2=O)cc1OC
COc1cc(Cl)c(\C=C2/CN(C\C(=C/c3nc(C)c(C)nc3C)C2=O)C(C)C)cc1OC
[#6]-[#6]1-[#6]\[#6](=[#6]/c2nc(-[#6])c(-[#6])nc2-[#6])\[#6](=[#7]/[#8])\[#6](\[#6]-1)=[#6]\c1nc(-[#6])c(-[#6])nc1-[#6]
[#6]-[#7]1-[#6]\[#6](=[#6]/c2nc(-[#6])c(-[#6])nc2-[#6])\[#6](=[#7]/[#8])\[#6](\[#6]-1)=[#6]\c1nc(-[#6])c(-[#6])nc1-[#6]
COc1cc(Br)c(\C=C2/CC(C)C/C(=C\c3nc(C)c(C)nc3C)/C/2=N/O)cc1OC
COc1cc(Br)c(\C=C2/CN(C)C/C(=C\c3nc(C)c(C)nc3C)/C/2=N\O)cc1OC
COc1cc(Br)c(\C=C2/CN(C/C(=C\c3nc(C)c(C)nc3C)/C/2=N/O)C(C)C)cc1OC
CN1C\C(=C/c2nc(C)c(C)nc2C)C(=O)\C(C1)=C\c1nc(C)c(C)nc1C
COc1cc(Br)c(\C=C2/CN(C)C\C(=C/c3nc(C)c(C)nc3C)C2=O)cc1OC
[#6]-[#6](-[#6])-[#7]1-[#6]\[#6](=[#6]/c2nc(-[#6])c(-[#6])nc2-[#6])\[#6](=[#7]/[#8])\[#6](\[#6]-1)=[#6]\c1nc(-[#6])c(-[#6])nc1-[#6]
COc1cc2c(Nc3ncc(CC(=O)Nc4cccc(F)c4)s3)ncnc2cc1OCCCN1CCC(CO)CC1
Nc1nccn2c(nc(-c3ccc4ccc(nc4c3)-c3ccccc3)c12)[C@@H]1C[C@H](CN2CCC2)C1 |wU:26.30,28.33,(7.04,-25.52,;7.05,-27.06,;5.72,-27.83,;5.72,-29.37,;7.05,-30.15,;8.39,-29.37,;9.86,-29.85,;10.77,-28.6,;9.86,-27.34,;10.64,-26.02,;9.88,-24.69,;10.64,-23.36,;12.19,-23.36,;12.96,-22.02,;14.5,-22.04,;15.28,-23.37,;14.5,-24.71,;12.96,-24.7,;12.18,-26.03,;16.82,-23.38,;17.59,-24.72,;19.13,-24.72,;19.9,-23.38,;19.12,-22.05,;17.59,-22.05,;8.39,-27.82,;10.34,-31.32,;9.65,-32.69,;11.02,-33.38,;11.5,-34.85,;10.47,-35.99,;8.93,-36.07,;9.01,-37.61,;10.55,-37.53,;11.72,-32.01,)|
CN1CCN(CC1)c1cc(Nc2cc(C)n[nH]2)nc(C=Cc2ccccc2)n1 |w:19.20|
COc1cc(ccc1Nc1nc(NC2CCCCC2)c2cc[nH]c2n1)N1CCOCC1
Cc1cc(cc2[nH]c(nc12)-c1c(NC[C@@H](O)c2ccccc2Cl)cc[nH]c1=O)N1CCN(CCC#N)CC1 |r|
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(NS(=O)(=O)c3ccc(F)cc3)cc2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(NS(=O)(=O)c3ccc(F)cc3)c(OC)c2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(NS(=O)(=O)c3ccc(C)cc3)c(C)c2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(Oc3ccc(NS(=O)(=O)C(F)(F)F)cc3)cc2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(Oc3ccc(NS(C)(=O)=O)cc3)cc2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(NS(=O)(=O)c3ccc(OC)cc3)c(C)c2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(NS(=O)(=O)c3ccc(OC)cc3)cc2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(NS(=O)(=O)c3ccc(C)cc3)c(OC)c2)ncc1Cl
COCC(=O)NC\C=C\c1ccc2ncnc(Nc3ccc(Oc4ccc(C)nc4)c(C)c3)c2c1
CCOc1cc2c(cc1NC(=O)/C=C/CN(C)C)c(c(cn2)C#N)Nc3ccc(c(c3)Cl)F
c1cc(c(c(c1)F)C(=O)n2c(nc(n2)Nc3ccc(cc3)S(=O)(=O)N)N)F
CC[C@H](CO)Nc1nc(NCc2ccccc2)c2ncn(C(C)C)c2n1 |r|
Oc1ccc(cc1)-c1nc(c([nH]1)-c1ccc(F)cc1)-c1ccncc1
NC(=O)c1ccc(cc1)-c1nc(c([nH]1)-c1ccc2OCOc2c1)-c1ccccn1
CNc1ccn(-c2ccccc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OC)c(OC)cc23)cn1
COc1cc2nccc(Oc3ccc(NC(=O)c4c(ccn(-c5ccccc5)c4=O)N(C)C)nc3)c2cc1OC
COCCNc1ccn(-c2ccccc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OC)c(OC)cc23)cn1
COc1cc2nccc(Oc3ccc(NC(=O)c4c(NC5CCOCC5)ccn(-c5ccccc5)c4=O)nc3)c2cc1OC
COc1cc2nccc(Oc3ccc(NC(=O)c4c(ccn(-c5ccccc5)c4=O)N4CCN(C)CC4)nc3)c2cc1OC
COc1cc2nccc(Oc3ccc(NC(=O)c4c(Nc5ccccc5)ccn(-c5ccccc5)c4=O)nc3)c2cc1OC
COCCNc1ccn(-c2ccccc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OC)ccc23)cn1
CNc1ccn(Cc2ccccc2)c(=O)c1C(=O)Nc1ccc(Oc2ccnc3cc(OC)c(OC)cc23)cn1
COc1cc2nccc(Oc3ccc(NC(=O)c4cc(cn(-c5ccccc5)c4=O)-c4cccs4)nc3)c2cc1OC
COc1cc2nccc(Oc3ccc(NC(=O)c4cc(cn(-c5ccccc5)c4=O)-c4cccnc4)nc3)c2cc1OC
COc1cc2nccc(Oc3ccc(NC(=O)c4cc(Cc5ccccc5)cn(-c5ccccc5)c4=O)nc3)c2cc1OC
COc1ccc2c(Oc3ccc(NC(=O)c4cc(cn(-c5ccccc5)c4=O)-c4cccnc4)nc3)ccnc2c1
COc1ccc2c(Oc3ccc(NC(=O)c4cc(cn(-c5ccccc5)c4=O)-c4cnccn4)nc3)ccnc2c1
COc1ccc(cc1OC)C(=O)NCc1cccc(c1)C(=O)Nc1ccc2CCNCc2c1
COc1ccc(Cn2ncc(NC(=O)c3cc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)ccc3C)c2N)cc1
Nc1ncnc(Nc2ccc(OCc3ccccn3)c(Cl)c2)c1-c1nc(CNC(=O)C=C)co1
Cn1c(nc2ccccc12)-c1ccnc(Nc2ccc(cc2)N2CCOCC2)n1
Cn1c(nc2ccccc12)-c1ccnc(Nc2ccccc2)n1
Cc1ccc(Nc2nccc(n2)-c2nc3ccccc3n2C)cc1
Cn1c(nc2ccccc12)-c1ccnc(Nc2ccc(Cl)cc2)n1
CCOc1ccc(Nc2nccc(n2)-c2nc3ccccc3n2C)cc1
COc1ccc(Nc2nccc(n2)-c2nc3ccccc3n2C)cc1
Cn1c(nc2ccccc12)-c1ccnc(Nc2ccc(O)cc2)n1
Cn1c(nc2ccccc12)-c1ccnc(Nc2cccc(O)c2)n1
Cn1c(nc2ccccc12)-c1ccnc(Nc2ccc(O)c(Cl)c2)n1
COc1ccc(Nc2nccc(n2)-c2nc3ccccc3n2C)cc1O
Cn1c(nc2ccccc12)-c1ccc2c(n1)n(C)c(=O)n(C)c2=O
COc1ccc(Nc2ncc3CC(=O)Nc4ccccc4-c3n2)cc1O
CC(C)(N)C(=O)NCCn1ccc2ncnc(Nc3ccc(Oc4cccc5sncc45)c(Cl)c3)c12
CC(C)(C(=O)NCCn1ccc2ncnc(Nc3ccc(Oc4cccc(Cl)c4)c(Cl)c3)c12)S(C)(=O)=O
CC(C)Oc1cc(n[nH]1)-n1cnc2ccc(N[C@@H](C)c3ccc(F)cn3)nc12 |r|
CC(C)(C)NS(=O)(=O)c1cncc(c1)-c1ccn2nc(N)nc2c1
CC(C)NC(=O)c1cc2cccc(NC(=O)Nc3cc(nn3-c3ccc(C)cc3)C(C)(C)C)c2[nH]1
COc1ccc(-c2cc(NC(=O)Nc3cc(nn3-c3ccc(C)cc3)C(C)(C)C)[nH]n2)c(C)c1
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1cc(n[nH]1)-c1ccc2ncccc2c1)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1cc(n[nH]1)-c1ccc2nccnc2c1)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1cc(COc2cccnc2)n[nH]1)C(C)(C)C
COc1ccc(nc1)-c1cc(NC(=O)Nc2cc(nn2-c2ccc(C)cc2)C(C)(C)C)[nH]n1
CCOCCCNC(=O)c1cc2cccc(NC(=O)Nc3cc(nn3-c3ccc(C)cc3)C(C)(C)C)c2[nH]1
CN(CCc1ccccn1)C(=O)c1cc2cccc(NC(=O)Nc3cc(nn3-c3ccc(C)cc3)C(C)(C)C)c2[nH]1
CNS(=C)(=O)c1ccc(Nc2ncc(c(N[C@@H]3CCC[C@H]3N(C)C)n2)C(F)(F)F)cc1 |r|
CCNS(=C)(=O)c1ccc(Nc2ncc(c(N[C@@H]3CCC[C@H]3N(C)C)n2)C(F)(F)F)cc1 |r|
CN(c1ncccc1CNc1ncnc2[nH]c(C)cc12)S(C)(=O)=O
CN(c1ncccc1CNc1ncnc2[nH]ccc12)S(C)(=O)=O
Fc1ccccc1Nc1ncnc2n[nH]cc12
CN(c1ncccc1CNc1c(C)cnc2[nH]ccc12)S(C)(=O)=O
CN(c1ncccc1CNc1c(cnc2[nH]c(cc12)-c1ccnc(C)c1)C#N)S(C)(=O)=O
CN(c1ncccc1CNc1ccnc2[nH]c(cc12)-c1ccc(F)cc1)S(C)(=O)=O
CN(c1ncccc1CNc1ccnc2[nH]ccc12)S(C)(=O)=O
CN(c1ncccc1CNc1c(Br)cnc2nc([nH]c12)-c1ccc(F)cc1)S(C)(=O)=O
CN(c1ncccc1CNc1c(cnc2[nH]ccc12)C#N)S(C)(=O)=O
CN(c1ncccc1CNc1c(cnc2[nH]c(cc12)-c1ccc(F)cc1)C(F)(F)F)S(C)(=O)=O
CN(c1ncccc1CNc1c(cnc2[nH]c(cc12)-c1ccc(F)cc1)C#N)S(C)(=O)=O
COc1cc(ccc1-c1cc2c(Nc3ccccc3C#N)c(cnc2[nH]1)C(F)(F)F)N1CCOCC1
CN(c1c(cccn1)CNc2c3cc([nH]c3ncc2C#N)c4ccccc4)S(=O)(=O)C
CN(c1ncccc1CNc1c(C)cnc2[nH]c(cc12)-c1ccc(F)cc1)S(C)(=O)=O
CN(c1ncccc1CNc1c(cnc2nc([nH]c12)-c1ccc(Br)cc1)C(F)(F)F)S(C)(=O)=O
Fc1cc(F)cc(Nc2c(cnc3[nH]c(cc23)-c2ccc(cc2)N2CCOCC2)C(F)(F)F)c1
CNC(=O)c1ccccc1Nc1c(cnc2[nH]c(cc12)-c1ccc(F)cc1)C(F)(F)F
CCCCc1ccc(cc1)-c1cc2c(NCc3cccnc3N(C)S(C)(=O)=O)c(cnc2[nH]1)C#N
CNC(=O)c1ccccc1Nc1c(cnc2[nH]c(cc12)-c1ccc(F)cc1)C#N
CN(c1ncccc1CNc1c(cnc2[nH]c(cc12)C1CCCCC1)C#N)S(C)(=O)=O
CN1Cc2cccc(Nc3c(cnc4[nH]c(cc34)-c3ccc(F)cc3)C(F)(F)F)c2C1=O
CNC(=O)c1ccccc1Nc1c(Br)cnc2nc([nH]c12)-c1ccc(F)cc1
CN(c1ncccc1CNc1c(cnc2nc([nH]c12)-c1ccc(F)cc1)C(F)(F)F)S(C)(=O)=O
CNC(=O)c1ccccc1Nc1c(cnc2[nH]c(cc12)-c1ccc(nc1)N1CCOCC1)C(F)(F)F
CNC(=O)c1ccccc1Nc1c(cnc2[nH]c(cc12)-c1ccc(cc1)N1CCOCC1)C(F)(F)F
CNC(=O)c1ccccc1Nc1c(cnc2[nH]c(cc12)-c1cccnc1)C(F)(F)F
Fc1ccc(cc1)-c1cc2c(NCc3cc(F)ccc3F)c(cnc2[nH]1)C(F)(F)F
Clc1ccc(cc1Cl)C1=NN(C(C1)c1ccc2ccccc2c1)c1ccccc1 |t:9|
Cc1ccc(cc1)C1=NN(C(C1)c1ccc2ccccc2c1)c1ccccc1 |t:8|
COc1ccc(cc1)C1=NN(C(C1)c1cccc2ccccc12)c1ccccc1 |t:9|
NC(=S)N1N=C(CC1c1ccc2ccccc2c1)c1ccc(Cl)c(Cl)c1 |c:4|
Cc1ccc(cc1)C1=NN(C(C1)c1ccc2ccccc2c1)C(N)=S |t:8|
COc1ccc(cc1)C1=NN(C(C1)c1cccc2ccccc12)C(N)=S |t:9|
Oc1ccc(CCNC(=O)C(Cc2cc(Br)c(O)c(Oc3ccc(CCNC(=O)C(Cc4cc(Br)c(O)c(c4)-c4cc(CC(N=O)C(=O)NCCc5ccc(O)c(Br)c5)cc(Br)c4O)N=O)cc3Br)c2)N=O)cc1Br
Oc1ccc(CCNC(=O)C(Cc2cc(Br)c(O)c(c2)-c2cc(CC(N=O)C(=O)NCCc3ccc(O)c(Br)c3)cc(Br)c2O)N=O)cc1Br
Oc1c(Br)cc2CCNC(=O)C(Cc3ccc(Oc4cc(CC(N=O)C(=O)NC=Cc5ccc(Oc1c2)c(Br)c5)cc(Br)c4O)c(Br)c3)N=O |w:29.29|
Cc1c(F)c(ccc1C(=O)N1CCOc2ccc(cc2C1)-c1ccc(N)nc1)S(C)(=O)=O
CN1c2ccc(NC(=O)c3ccc(F)cc3)cc2-c2c(cnn2C)S1(=O)=O
CN1c2ccc(CNc3ccc(F)cc3)cc2-c2c(cnn2C)S1(=O)=O
CN1c2ccc(cc2-c2c(cnn2C)S1(=O)=O)C(=O)Nc1ccc(F)cc1
CCc1ccc(cc1)-c1ccc2N(C)S(=O)(=O)c3cn(C)nc3-c2c1
CCc1ccc(cc1)-c1ccc2N(C)S(=O)(=O)c3cnn(CC)c3-c2c1
CN1c2ccc(cc2-c2n[nH]cc2S1(=O)=O)-c1ccc(cc1)C(=O)N1CCC(CCO)CC1
CN1c2ccc(cc2-c2n[nH]cc2S1(=O)=O)-c1ccc(cc1)C(=O)NCCO
CN1c2ccc(cc2-c2n[nH]cc2S1(=O)=O)-c1ccc(cc1)C(N)=O
Fc1ccc(CSc2nnc(Cn3nnc4ccccc34)o2)cc1F
Clc1ccc(CSc2nnc(Cn3nnc4ccccc34)o2)cc1Cl
[O-][N+](=O)c1ccc(CSc2nnc(Cn3nnc4ccccc34)o2)cc1
COc1ccc(CSc2nnc(Cn3nnc4ccccc34)o2)cc1
Cc1ccc(CSc2nnc(Cn3nnc4ccccc34)o2)cc1
Brc1ccc(CSc2nnc(Cn3nnc4ccccc34)o2)cc1
Fc1ccc(CSc2nnc(Cn3nnc4ccccc34)o2)cc1
[O-][N+](=O)c1cccc(CSc2nnc(Cn3nnc4ccccc34)o2)c1
COc1cccc(CSc2nnc(Cn3nnc4ccccc34)o2)c1
Cc1cccc(CSc2nnc(Cn3nnc4ccccc34)o2)c1
Brc1cccc(CSc2nnc(Cn3nnc4ccccc34)o2)c1
Clc1cccc(CSc2nnc(Cn3nnc4ccccc34)o2)c1
Fc1cccc(CSc2nnc(Cn3nnc4ccccc34)o2)c1
[O-][N+](=O)c1ccccc1CSc1nnc(Cn2nnc3ccccc23)o1
COc1ccccc1CSc1nnc(Cn2nnc3ccccc23)o1
Cc1ccccc1CSc1nnc(Cn2nnc3ccccc23)o1
Brc1ccccc1CSc1nnc(Cn2nnc3ccccc23)o1
Clc1ccccc1CSc1nnc(Cn2nnc3ccccc23)o1
Fc1ccccc1CSc1nnc(Cn2nnc3ccccc23)o1
Cc1cc(C(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)nn4c3)ccc2F)n(C)n1
COc1cc(Nc2nc(Nc3ccccc3NC(C)=O)nc(n2)C(F)(F)F)cc(OC)c1OC
COc1cc(Nc2nc(C)nc(Nc3ccccc3NC(=O)N(C)C)n2)cc(OC)c1OC
COC(=O)Nc1ccccc1Nc1nc(C)nc(Nc2cc(OC)c(OC)c(OC)c2)n1
COc1cc(Nc2nc(C)nc(Nc3ccccc3NC(C)=O)n2)cc(OC)c1OC
COc1cc(Nc2nc(C)nc(Nc3ccccc3NS(C)(=O)=O)n2)cc(OC)c1OC
CNc1nc(Nc2cccc(NS(C)(=O)=O)c2)nc(Nc2cc(OC)c(OC)c(OC)c2)n1
COc1cc(Nc2ncnc(Nc3cccc(NS(C)(=O)=O)c3)n2)cc(OC)c1OC
COc1cc(Nc2nc(Cl)nc(Nc3cccc(NS(C)(=O)=O)c3)n2)cc(OC)c1OC
CNc1nc(Nc2cc(OC)c(OC)c(OC)c2)nc(Nc2ccccc2NS(C)(=O)=O)n1
COc1cc(Nc2ncnc(Nc3ccccc3NS(C)(=O)=O)n2)cc(OC)c1OC
COc1cc(Nc2nc(Cl)nc(Nc3ccccc3NS(C)(=O)=O)n2)cc(OC)c1OC
CCC(CC)NC(=O)c1ccccc1Nc1ncnc(Nc2ccc(CN)cc2)n1
CC(C)NC(=O)c1ccccc1Nc1ncnc(Nc2ccc(CN)cc2)n1
CCNC(=O)c1ccccc1Nc1ncnc(Nc2ccc(CN)cc2)n1
CNC(=O)c1ccccc1Nc1ncnc(Nc2ccc(CN)cc2)n1
CS(=O)(=O)Nc1ccccc1Nc1ncnc(Nc2ccc(CN)cc2)n1
CNC(=O)c1ccccc1Nc1ncnc(Nc2cc(CCC(N)=O)c(OC)c(OC)c2)n1
CNC(=O)c1ccccc1Nc2ncnc(n2)Nc3ccc(cc3OC)N4CCOCC4
COc1ccc(Nc2ncnc(Nc3ccccc3NC(C)=O)n2)c(OC)c1
CNC(=O)c1ccccc1Nc1ncnc(Nc2ccc(OC)cc2OC)n1
COc1ccc(Nc2ncnc(Nc3ccccc3NS(C)(=O)=O)n2)c(OC)c1
COC(=O)c1ccccc1Nc1ncnc(Nc2cc(OC)c(OC)c(OC)c2)n1
COc1cc(Nc2ncnc(Nc3ccccc3C(=O)NCCN(C)C)n2)cc(OC)c1OC
COc1cc(Nc2ncnc(Nc3ccccc3C(=O)NCCO)n2)cc(OC)c1OC
COc1cc(Nc2ncnc(Nc3ccccc3C(=O)NC3CCCC3)n2)cc(OC)c1OC
CCC(CC)NC(=O)c1ccccc1Nc1ncnc(Nc2cc(OC)c(OC)c(OC)c2)n1
COc1cc(Nc2ncnc(Nc3ccccc3C(=O)NC3CC3)n2)cc(OC)c1OC
COc1cc(Nc2ncnc(Nc3ccccc3C(=O)NC(C)C)n2)cc(OC)c1OC
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(cc1)-c1cccnc1)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(cc1)-n1cnc(Cl)c1Cl)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(cc1)-n1ccnc1)C(C)(C)C
Cc1cn(cn1)-c1ccc(NC(=O)Nc2cc(nn2-c2ccc(C)cc2)C(C)(C)C)cc1
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(cc1)-n1cnc2c(N)ncnc12)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(cc1)-c1ccc(OCc2ccccc2)nc1)C(C)(C)C
COc1ccc(cn1)-c1ccc(NC(=O)Nc2cc(nn2-c2ccc(C)cc2)C(C)(C)C)cc1
COc1cc(OC)nc(n1)-c1ccc(NC(=O)Nc2cc(nn2-c2ccc(C)cc2)C(C)(C)C)cc1
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(cc1)-c1ccncc1)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(cc1)-c1ccc(N)nc1)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(cc1)-c1nncn1C)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(cc1)-n1cnnn1)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(cc1)-c1cnco1)C(C)(C)C
Cc1nnnn1-c1ccc(NC(=O)Nc2cc(nn2-c2ccc(C)cc2)C(C)(C)C)cc1
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(cc1)-c1csnn1)C(C)(C)C
Cc1cncn1-c1ccc(NC(=O)Nc2cc(nn2-c2ccc(C)cc2)C(C)(C)C)cc1
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(cc1)-c1n[nH]c(=S)n1C)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(cc1)-n1cnnc1)C(C)(C)C
Cc1[nH]n2c(nc(C)cc2=O)c1C#N
CCOc1ccccc1NC(=O)c1ccoc1
CC(=O)Nc1sccc1C(N)=O
Cc1c([nH]c2CCCC(=O)c12)C(O)=O
C1CN(CCO1)c1ncnc2ccccc12
O=C(N1CCCC1)c1cnc2ccccc2n1
Cc1[nH]nc2cn[nH]c12
c1ncc(o1)-c1ccncc1
Brc1cncc(c1)-c1nnn[nH]1
Nc1nccc(n1)-c1cccnc1
CC(=O)Nc1ccc(Cl)cn1
CNC(=O)c1ccccc1Nc1cc(Nc2ccc(cc2OC)N2CCOCC2)ncc1C(F)(F)F
CN(C)c1ccc(Oc2cc(O)cc(O)c2-c2cc(no2)C(=O)NC2CCN(CC2)C2CCC3(CC2)OCCO3)cc1
CC(C)Nc1ccc(Oc2cc(O)cc(O)c2-c2cc(no2)C(=O)NC2CCN(C)CC2)cc1
CN(C)c1ccc(Oc2cc(O)cc(O)c2-c2cc(no2)C(=O)NC2CCN(C)CC2)cc1
CN1CCC(CC1)NC(=O)c2cc(on2)c3c(cc(cc3Oc4ccc(cc4)[N+](=O)[O-])O)O
CNS(=O)(=O)Nc1cccc(Cc2c(C)c3cc(Cl)c(OC(=O)N(C)C)cc3oc2=O)c1
c1cc(c(cc1C2=C(C(=O)c3c(cc(cc3O2)O)O)O)O)O
Cc1c(O)c(O)c2oc(cc2c1C=O)-c1c(C)c(O)c(O)c(O)c1C=O
Cc1c2COC(=O)c2c(O)c(O)c1O
COCc1c(C)c(O)c(O)c(O)c1C=O
COC1OC(=O)c2c1c(C)c(O)c(O)c2O
Cc1c(O)c(O)c2O[C@H]3O[C@H](C(=O)c4c(O)c(O)c(O)c(C)c34)c2c1C=O |r|
COC(=O)c1cc(O)c(O)c(C[C@]2(C)[C@@H](C)CC[C@]3(C)[C@H]2CCC=C3C)c1 |r,c:24|
COc1cc2nc(C)oc2c(C[C@]2(C)[C@@H](C)CC[C@]3(C)[C@H]2CCC=C3C)c1O |r,c:25|
CC(C)CC=Nc1cc(O)c(O)c(C[C@]2(C)[C@@H](C)CC[C@]3(C)[C@H]2CCC=C3C)c1O |r,w:5.5,c:26|
C[C@@H](Oc1cc(cnc1N)-c1sc(nc1C)[C@](C)(O)CO)c1cc(F)ccc1-n1nccn1 |r|
Fc1ccc(Cc2cnc(NC(=O)CCc3nc4ccccc4c(=O)[nH]3)s2)cc1F
O=c1[nH]c(CSc2nnc(NCC3CCCO3)s2)nc2sc(cc12)-c1ccccc1
Fc1ccc2nc(NC(=O)CSc3nnc(COc4ccc5CCCCc5c4)o3)sc2c1
COc1ccc2nc(NC(=O)CSc3nnc(COc4ccc5CCCCc5c4)o3)sc2c1
[O-][N+](=O)c1cnc(NC(=O)CSc2nnc(COc3ccc4CCCCc4c3)o2)s1
CCOP(=O)(CCCOc1ccc(Nc2ncc(c(Nc3ccccc3C(=O)NC)n2)[N+]([O-])=O)cc1)OCC
CCOP(=O)(Cc1ccc(Nc2ncc(c(Nc3ccccc3C(=O)NC)n2)[N+]([O-])=O)cc1)N1CCOCC1
CCOP(=O)(CCCOc1ccc(Nc2ncc(c(Nc3ccccc3C(=O)NC)n2)[N+]([O-])=O)cc1)N1CCOCC1
CCOP(=O)(CCCOc1ccc(Nc2ncc(Cl)c(Nc3ccccc3C(=O)NC)n2)cc1)OCC
CCOP(=O)(Cc1ccc(Nc2ncc(Cl)c(Nc3ccccc3C(=O)NC)n2)cc1)OCC
CCOP(=O)(Cc1ccc(Nc2ncc(c(Nc3ccccc3C(=O)NC)n2)[N+]([O-])=O)cc1)OCC
O=C(Cc1cccc(OCCCN2CCNCC2)c1)Nc1nc(cs1)-c1ccncc1
O=C(Cc1cccc(OCCCC2CCNCC2)c1)Nc1nc(cs1)-c1ccncc1
CN1CCN(CCCOc2cccc(CC(=O)Nc3nc(cs3)-c3c[nH]c4ncccc34)c2)CC1
CS(=O)(=O)Nc1cccc(CC(=O)Nc2nc(cs2)-c2c[nH]c3ncccc23)c1
O=C(Cc1cccc(OCCCC2CCNCC2)c1)Nc1nc(cs1)-c1c[nH]c2ncccc12
CCn1cc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)ncnc12
COc1cc(O)c2c(c1)c1c(C)cc(O)c(O)c1oc2=O
COc1cc(O)c2c(c1)c1c(C)cc(O)cc1oc2=O
COc1cc2c(C(=O)OC22C(C)CC(=O)C2=O)c(O)c1
COc1cc(O)c2c(c1)-c1cc(O)c(O)cc1COC2=O
Cc1cc(O)c(O)cc1-c1cc(O)cc(O)c1C(O)=O
[H][C@]12[C@@H](O)CC(=O)c3c(O)ccc(-c4ccc(O)c5C(=O)CC[C@]1(O)c45)c23 |r|
COc1cc(O)c(C(O)=O)c(c1)C1=C(C)C[C@@H](O)C1=O |r,wD:16.17,c:13,(10.48,-22.79,;11.26,-21.46,;10.49,-20.12,;11.26,-18.8,;10.49,-17.47,;11.26,-16.14,;8.97,-17.47,;8.2,-16.14,;8.96,-14.8,;6.65,-16.13,;8.21,-18.79,;8.97,-20.12,;6.66,-18.79,;5.76,-17.54,;4.98,-16.2,;4.29,-18.01,;4.29,-19.55,;3.04,-20.45,;5.75,-20.03,;6.22,-21.5,)|
Cc1cc(O)cc2oc(=O)c3c(O)cc(OS(O)(=O)=O)cc3c12
COc1cc(O)c(C(O)=O)c(c1)-c1cc(O)c(O)cc1C
Cc1cc(O)cc2oc(=O)c3c(O)cc(O)cc3c12
COc1cc(O)c2C(=O)C3=C([C@@H](O)[C@](C)(O)[C@H](O)[C@H]3O)C(=O)c2c1-c1c(O)c2C(=O)c3cc(O)c(C)cc3C(=O)c2cc1OC |r,wU:18.19,11.11,13.13,wD:16.16,t:9,(-6.62,-6.52,;-5.29,-5.75,;-3.96,-6.52,;-3.96,-8.06,;-2.63,-8.83,;-2.63,-10.37,;-1.3,-8.07,;.04,-8.83,;.05,-10.37,;1.38,-8.06,;1.38,-6.5,;2.72,-5.72,;2.71,-4.19,;4.06,-6.5,;4.82,-5.16,;5.38,-7.27,;4.07,-8.06,;5.4,-8.82,;2.72,-8.83,;2.72,-10.37,;.03,-5.73,;.02,-4.19,;-1.3,-6.52,;-2.63,-5.75,;-2.6,-3.5,;-1.27,-2.73,;.06,-3.5,;-1.26,-1.19,;.06,-.41,;1.4,-1.16,;.05,1.13,;1.37,1.91,;1.36,3.45,;2.68,4.23,;.01,4.21,;-.01,5.74,;-1.31,3.42,;-1.29,1.89,;-2.62,1.11,;-3.96,1.87,;-2.6,-.43,;-3.93,-1.19,;-3.93,-2.74,;-5.26,-3.5,;-6.59,-2.73,)|
COc1cc(O)c2C(=O)c3c(O)c(O)c(C)cc3C(=O)c2c1
COc1cc(O)c2C(=O)C3=C([C@@H](O)[C@](C)(O)[C@H](O)[C@H]3O)C(=O)c2c1 |r,t:9|
COc1cc(O)c2C(=O)c3cc(O)c(C)cc3C(=O)c2c1
Clc1ccc(CC(=O)Nc2nnc(s2)-c2ccc3OCCOc3c2)cc1
Clc1cccc(CC(=O)Nc2nnc(s2)-c2ccc3OCCOc3c2)c1
Clc1ccc(cn1)C(=O)Nc1nnc(s1)-c1ccc2OCCOc2c1
O=C(CCc1ccccc1)Nc1nnc(s1)-c1ccc2OCCOc2c1
O=C(Nc1nnc(s1)-c1ccc2OCCOc2c1)c1ccccc1
O=C(Nc1nnc(s1)-c1ccc2OCCOc2c1)\C=C\c1ccccc1
Brc1cccc(CC(=O)Nc2nnc(s2)-c2ccc3OCCOc3c2)c1
Brc1ccc(CC(=O)Nc2nnc(s2)-c2ccc3OCCOc3c2)cc1
O=C(Cc1ccccc1)Nc1nnc(s1)-c1ccc2OCCOc2c1
Fc1ccc(CC(=O)Nc2nnc(s2)-c2ccc3OCCOc3c2)cc1
Oc1ccc(Br)cc1\C=N\NC(=O)CSc1nnc(-c2ccncc2)n1-c1ccccc1
Brc1ccc(\C=N\NC(=O)CSc2nnc(-c3ccncc3)n2-c2ccccc2)cc1
O=C(CSc1nnc(-c2ccncc2)n1-c1ccccc1)N\N=C\C=C\c1ccccc1
Fc1ccc(\C=N\NC(=O)CSc2nnc(-c3ccncc3)n2-c2ccccc2)cc1
Clc1ccc(\C=N\NC(=O)CSc2nnc(-c3ccncc3)n2-c2ccccc2)cc1
Brc1cccc(CSc2nnc(-c3ccncc3)n2-c2ccccc2)c1
Fc1ccc(CSc2nnc(-c3ccncc3)n2-c2ccccc2)c(F)c1
C[C@@H]1C[C@H](N)C[C@@H](C1)c1ccncc1NC(=O)c1ccc(F)c(n1)-c1c(F)cccc1F |r,wU:6.8,3.3,1.0,(-.67,2.69,;-2,1.93,;-3.33,2.69,;-4.67,1.93,;-6,2.69,;-4.67,.38,;-3.33,-.38,;-2,.38,;-3.33,-1.93,;-4.67,-2.69,;-4.67,-4.23,;-3.33,-5,;-2,-4.23,;-2,-2.69,;-.67,-1.93,;.67,-2.69,;.67,-4.23,;2,-1.93,;3.33,-2.69,;4.67,-1.93,;4.67,-.38,;6,.38,;3.33,.38,;2,-.38,;3.33,1.93,;4.67,2.69,;6,1.93,;4.67,4.23,;3.33,5,;2,4.23,;2,2.69,;.67,1.93,)|
CC(=O)Nc1ccc(Nc2nc(Nc3ccccc3P(C)(C)=O)c3cc[nH]c3n2)cc1
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)N2CCNCC2)nc2[nH]ccc12
CCOc1cc(ccc1Nc1nc(Nc2ccccc2P(C)(C)=O)c2cc[nH]c2n1)C(=O)NC1CCNCC1
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(C(=O)NC3CCNCC3)c(F)c2)nc2[nH]ccc12
COCCn1cc(Nc2nc(Nc3ccccc3P(C)(C)=O)c3sccc3n2)cn1
COc1cc(ccc1Nc1nc(Nc2ccccc2P(C)(C)=O)c2sccc2n1)C(=O)NC1CCNCC1
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2[nH]ccc12
CNC(=O)c1ccc(Nc2nc(Nc3ccccc3P(C)(C)=O)c3cc[nH]c3n2)cc1
CNC(=O)c1ccc(Nc2nc(NCc3ccccc3N(C)S(C)(=O)=O)c3cc[nH]c3n2)cc1
COc1cc(ccc1Nc1nc(Nc2cccn(C)c2=O)c2cc[nH]c2n1)N1CCOCC1
CNC(=O)c1ccc(Nc2nc(Nc3cccn(C)c3=O)c3cc[nH]c3n2)cc1
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)NC2CCNCC2)nc2[nH]ccc12
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)NC2CCOCC2)nc2[nH]ccc12
CN1CCC(CC1)NC(=O)c1ccc(Nc2nc(Nc3ccccc3P(C)(C)=O)c3cc[nH]c3n2)cc1
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N2CCOCC2)nc2[nH]ccc12
CN1CCN(CC1)c1ccc(Nc2nc(Nc3ccccc3P(C)(C)=O)c3cc[nH]c3n2)cc1
CP(C)(=O)c1ccccc1Nc1nc(Nc2cnn(CC(F)F)c2)nc2[nH]ccc12
COCCn1cc(Nc2nc(Nc3ccccc3P(C)(C)=O)c3cc[nH]c3n2)cn1
CP(C)(=O)c1ccccc1Nc1nc(Nc2cnn(c2)C2CCNCC2)nc2[nH]ccc12
CP(C)(=O)c1ccccc1Nc1nc(Nc2cnn(CC(=O)N3CCOCC3)c2)nc2[nH]ccc12
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2F)C(=O)NC2CCNCC2)nc2[nH]ccc12
COc1cc(C(=O)NC2CCNCC2)c(F)cc1Nc1nc(Nc2ccccc2P(C)(C)=O)c2cc[nH]c2n1
COc1cc(ccc1Nc1nc(Nc2ccccc2P(C)(C)=O)c2cc[nH]c2n1)N1CCOCC1
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N2CCNCC2)nc2[nH]ccc12
CP(C)(=O)c1ccccc1Nc1nc(Nc2cnn(c2)C2CCOCC2)nc2[nH]ccc12
COc1cc(ccc1Nc1nc(Nc2ccccc2P(C)(C)=O)c2ccsc2n1)C(=O)NC1CCNCC1
COc1cc(ccc1Nc1nc(NCc2ccccc2N(C)S(C)(=O)=O)c2cc[nH]c2n1)N1CCOCC1
COP(=O)(Cc1ccc(Nc2nc(Nc3ccccc3P(C)(C)=O)c3cc[nH]c3n2)cc1)OC
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N[C@@H]2CCCNC2)nc2[nH]ccc12 |r|
Cn1cc(Nc2nc(Nc3ccccc3P(C)(C)=O)c3cc[nH]c3n2)cn1
CN(C)C(=O)Cn1cc(Nc2nc(Nc3ccccc3P(C)(C)=O)c3cc[nH]c3n2)cn1
COc1cc(ccc1Nc1nc(Nc2ccccc2P(C)(C)=O)c2cc[nH]c2n1)C(=O)NC1CCNCC1
COCCn1cc(Nc2nc(Nc3ccccc3P(C)(C)=O)c3ccsc3n2)cn1
CNC(=O)c1ccc(Nc2nc(Nc3ccccc3C(=O)NC)c3cc[nH]c3n2)cc1
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N[C@H]2CCCNC2)nc2[nH]ccc12 |r|
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2C(F)(F)F)C(=O)NC2CCNCC2)nc2[nH]ccc12
Cc1cc(Nc2nc(Nc3ccccc3P(C)(C)=O)c3cc[nH]c3n2)ccc1C(=O)NC1CCNCC1
CCNS(=O)(=O)c1ccc(Nc2nc(Nc3ccccc3P(C)(C)=O)c3cc[nH]c3n2)cc1
CC(C)Oc1cc(ccc1Nc1nc(Nc2ccccc2P(C)(C)=O)c2cc[nH]c2n1)C(=O)NC1CCNCC1
[H][C@]12C[C@@H](NCCOCCOCCOCCNC(=O)CCC3=[N+]4C(C=C3)=Cc3c(C)cc(C)n3[B-]4(F)F)[C@@H](OC)[C@](C)(O1)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r,c:24,26,t:21|
[H][C@]12C[C@H]([C@@H](OC)[C@](C)(O1)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13)N(C)CCOCCOCCOCCNC(=O)CCC1=[N+]2C(C=C1)=Cc1c(C)cc(C)n1[B-]2(F)F |r,c:63,65,t:60|
CN(c1cccc2CN(Cc12)c1nc(Nc2ccc(cc2)N2CCN(CC2)C(C)=O)ncc1C(F)(F)F)S(C)(=O)=O
COC[C@@H](C)Nc1cc(NC(=O)N2CCCc3cc(CN4CCCCOC4=O)c(C=O)nc23)ncc1C#N |r|
CN(CCc1ccc(cc1)-c1ccccc1)Cc1cn(C)c2ccc(cc12)C(=O)Nc1ccc(F)cc1
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(OCC(=O)N3CCOCC3)cc2)ncc1Cl
Clc1cnc(Nc2ccc(OCC(=O)N3CCOCC3)cc2)nc1Nc1ccccc1C(=O)NC1CC1
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(CC(=O)N3CCOCC3)cc2)ncc1Cl
CCC(Oc1ccc(Nc2ncc(Cl)c(Nc3ccccc3C(=O)NC)n2)cc1)C(=O)N1CCOCC1
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(SCC(=O)N3CCOCC3)cc2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(OC(C)C(=O)N3CCOCC3)cc2)ncc1Cl
CNC(=O)c1ccc(cc1)Nc2ncc(c(n2)NCc3c(nccn3)N(C)S(=O)(=O)C)C(F)(F)F
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N2CCN(CC2)C(=S)SCCN(C)C)ncc1Cl
CNC(=O)c1ccccc1Nc1ccnc(Nc2ccc(cc2)C(=O)N2CCN(CC2)C(=S)SCCN(C)C)n1
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N2CCN(CC2)C(=S)SCCN(C)C)ncc1C
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N2CCN(CC2)C(=S)SCCN(C)C)ncc1C(F)(F)F
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N2CCN(CC2)C(=S)SCCN(C)C)ncc1F
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N2CCN(CC2)C(=S)SCCN(C)C)ncc1OC
CN(C)c1ccc(cc1)C(=O)Nc1cccc(NC(=O)COc2ccc3c(c2)occc3=O)c1
CN(c1cccc(CNc2nc(Nc3ccc(OCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(cc4)-c4scnc4C)C(C)(C)C)cc3)ncc2C(F)(F)F)c1)S(C)(=O)=O |r|
CN(c1cccc(CNc2nc(Nc3ccc(OCCOCCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(cc4)-c4scnc4C)C(C)(C)C)cc3)ncc2C(F)(F)F)c1)S(C)(=O)=O |r|
CN(c1cccc(CNc2nc(Nc3ccc(OCCOCCOCCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(cc4)-c4scnc4C)C(C)(C)C)cc3)ncc2C(F)(F)F)c1)S(C)(=O)=O |r|
CN(c1cccc(CNc2nc(Nc3ccc(OCCCOCCC(=O)NCCOc4cccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c45)cc3)ncc2C(F)(F)F)c1)S(C)(=O)=O
CN(c1cccc(CNc2nc(Nc3ccc(OCCOCCOCCOCCOCCC(=O)NCCOc4cccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c45)cc3)ncc2C(F)(F)F)c1)S(C)(=O)=O
CN(c1cccc(CNc2nc(Nc3ccc(OCCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(cc4)-c4scnc4C)C(C)(C)C)cc3)ncc2C(F)(F)F)c1)S(C)(=O)=O |r|
CN(c1cccc(CNc2nc(Nc3ccc(OCCCOCCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(cc4)-c4scnc4C)C(C)(C)C)cc3)ncc2C(F)(F)F)c1)S(C)(=O)=O |r|
CN(c1cccc(CNc2nc(Nc3ccc(OCCOCCOCCC(=O)NCCOc4cccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c45)cc3)ncc2C(F)(F)F)c1)S(C)(=O)=O
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1ncc(Cl)c(Nc2ccccc2S(=O)(=O)C(C)C)n1
C[C@H](Oc1ccc2c(cn(-c3cc(C)[nH]n3)c2n1)C(=O)N1CCO[C@@H](C)C1)c1ccc(F)cn1 |r|
Cc1ccc(cc1)-c1nn(cc1C(=O)NOCc1ccccc1F)-c1ccccc1
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)NCCOCCOCCOCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(cc1)-c1scnc1C)C(C)(C)C |r|
COc1cc(ccc1Nc1ncc(c(Oc2cccc3CCC(=O)c23)n1)C(F)(F)F)C(=O)NCCOCCOCCOCCC(=O)Nc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12
COc1cc(ccc1Nc1ncc2N(C)C(=O)c3nc(C)sc3N(C)c2n1)N1CCC(CC1)N1CCN(C)CC1
COc1cc(ccc1Nc1ncc2NC(=O)c3ccccc3N(C)c2n1)N1CCN(C)CC1
COc1cc(ccc1Nc1ncc2NC(=O)c3nn(C)cc3N(C)c2n1)N1CCN(C)CC1
COc1cc(ccc1Nc1ncc2NC(=O)c3scnc3N(C)c2n1)N1CCN(C)CC1
COc1cc(ccc1Nc1ncc2NC(=O)c3nc(C)sc3N(C)c2n1)N1CCC(CC1)N1CCN(C)CC1
COc1cc(ccc1Nc1ncc2N(C)C(=O)c3nc(C)oc3N(C)c2n1)N1CCC(CC1)N1CCN(C)CC1
CCCN1c2sc(C)nc2C(=O)N(C)c2cnc(Nc3ccc(cc3OC)N3CCC(CC3)N3CCN(C)CC3)nc12
COc1cc(ccc1Nc1ncc2N(C)C(=O)c3nc(C)sc3N(CC(F)(F)F)c2n1)N1CCC(CC1)N1CCN(C)CC1
COc1cc(ccc1Nc1ncc2N(C)C(=O)c3nc(sc3N(C)c2n1)C(F)(F)F)N1CCC(CC1)N1CCN(C)CC1
COc1cc(ccc1Nc1ncc2N(C)C(=O)c3nc(sc3N(C)c2n1)-c1ccccc1)N1CCC(CC1)N1CCN(C)CC1
COc1cc(ccc1Nc1ncc2N(C)C(=O)c3nc(sc3N(C)c2n1)C(C)C)N1CCC(CC1)N1CCN(C)CC1
CCc1nc2c(s1)N(C)c1nc(Nc3ccc(cc3OC)N3CCC(CC3)N3CCN(C)CC3)ncc1N(C)C2=O
COc1cc(ccc1Nc1ncc2NC(=O)c3ncsc3N(C)c2n1)N1CCC(CC1)N1CCN(C)CC1
COc1cc(ccc1Nc1ncc2N(C)C(=O)c3nc(C)sc3N(C)c2n1)C(=O)N1CCC(CC1)N1CCN(C)CC1
CN1c2sc(C)nc2C(=O)N(C)c2cnc(Nc3cnn(C)c3)nc12
CN1CCN(CC1)c1ccc(Nc2ncc3N(C)C(=O)c4nc(C)sc4N(C)c3n2)nc1
COc1cc(ccc1Nc1ncc2N(C)C(=O)c3nc(C)sc3N(C)c2n1)N1CCN(CCN(C)C)CC1
COc1cc(ccc1Nc1ncc2N(C)C(=O)c3nc(C)sc3N(C)c2n1)N1CCN(CCO)CC1
COc1cc2CCN(C)Cc2cc1Nc1ncc2N(C)C(=O)c3nc(C)sc3N(C)c2n1
CN1c2sc(C)nc2C(=O)N(C)c2cnc(Nc3ccc4NC(=O)CCc4c3)nc12
CNC(=O)c1ccc(Nc2ncc3N(C)C(=O)c4nc(C)sc4N(C)c3n2)c(OC)c1
CNC(=O)c1ccc(Nc2ncc3N(C)C(=O)c4nc(C)sc4N(C)c3n2)cc1
CN1CCN(CC1)c1ccc(Nc2ncc3N(C)C(=O)c4nc(C)sc4N(C)c3n2)c(OCCO)c1
CCOc1cc(ccc1Nc1ncc2N(C)C(=O)c3nc(C)sc3N(C)c2n1)N1CCN(C)CC1
COc1cc(ccc1Nc1ncc2N(C)C(=O)c3nc(C)sc3N(C)c2n1)C1CCN(C)CC1
COc1cc(N2CCN(C)CC2)c(C)cc1Nc1ncc2N(C)C(=O)c3nc(C)sc3N(C)c2n1
COc1cc(ccc1Nc1ncc2N(C)C(=O)c3nc(C)sc3N(C)c2n1)N1CCN(CC1)C(C)=O
COc1cc(ccc1Nc1ncc2N(C)C(=O)c3nc(C)sc3N(C)c2n1)N1CCN(CC1)S(C)(=O)=O
COc1cc(ccc1Nc1ncc2N(C)C(=O)c3nc(C)sc3N(C)c2n1)N1CCN(C)CC1=O
COc1cc(ccc1Nc1ncc2N(C)C(=O)c3nc(C)sc3N(C)c2n1)N1CCNCC1
COc1cc(ccc1Nc1ncc2N(C)C(=O)c3nc(C)sc3N(C)c2n1)N1CCN(C)CC1
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(CNc3c(NCCNC(=O)C=C)c(=O)c3=O)cc2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(CNc3c(NCCNC(=O)CCl)c(=O)c3=O)cc2)ncc1Cl
CONC(=O)c1ccccc1Nc1nc(Nc2ccc(CNc3c(NCCNC(=O)C=C)c(=O)c3=O)cc2)ncc1Cl
CN(c1ccccc1CNc1nc(Nc2ccc(CNc3c(NCCNC(=O)C=C)c(=O)c3=O)cc2)ncc1Cl)S(C)(=O)=O
CN(c1cccc(CNc2nc(Nc3ccc(CNc4c(NCCNC(=O)C=C)c(=O)c4=O)cc3)ncc2Cl)c1)S(C)(=O)=O
CS(=O)(=O)c1cccc(CNc2nc(Nc3ccc(CNc4c(NCCNC(=O)C=C)c(=O)c4=O)cc3)ncc2Cl)c1
CN(c1ncccc1CNc1nc(Nc2ccc(CNc3c(NCCNC(=O)C=C)c(=O)c3=O)cc2)ncc1Cl)S(C)(=O)=O
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(CNc3c(NCCNC(=O)C=C)c(=O)c3=O)cc2)ncc1C(F)(F)F
CC\C=C(/C#N)C(=O)NCCNc1c(NCc2ccc(Nc3ncc(Cl)c(Nc4ccccc4C(=O)NC)n3)cc2)c(=O)c1=O
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(CNc3c(NCCNC(=O)C(=C\C(C)C)\C#N)c(=O)c3=O)cc2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(CNc3c(NCCNC(=O)C(=C\C4CC4)\C#N)c(=O)c3=O)cc2)ncc1Cl
COc1cc2c(c(F)c1N1C[C@H](C)N(C)[C@H](C)C1)n(C(C)C)c1[nH]c3cc(ccc3c1c2=O)C#N |r|
COc1ccccc1-c1csc2cnc(Nc3ccc(CP(=O)(OC)OC)cc3)nc12
COP(=O)(Cc1ccc(Nc2ncc3scc(-c4ccccc4C(C)=O)c3n2)cc1)OC
COP(=O)(Cc1ccc(Nc2ncc3scc(-c4cccc(c4)C(C)=O)c3n2)cc1)OC
COP(=O)(Cc1ccc(Nc2ncc3scc(-c4cccc(c4)S(C)(=O)=O)c3n2)cc1)OC
CNC(=O)c1cccc(c1)-c1csc2cnc(Nc3ccc(CP(=O)(OC)OC)cc3)nc12
COP(=O)(Cc1ccc(Nc2ncc3scc(-c4cccc(NC(C)=O)c4)c3n2)cc1)OC
COP(=O)(Cc1ccc(Nc2ncc3scc(-c4cccc(c4)N(C)S(C)(=O)=O)c3n2)cc1)OC
COc1ccc(cc1)-c1csc2cnc(Nc3ccc(CP(=O)(OC)OC)cc3)nc12
CCOP(=O)(Cc1ccc(Nc2ncc3scc(-c4ccccc4OC)c3n2)cc1)OCC
CCOP(=O)(Cc1ccc(Nc2ncc3scc(-c4ccccc4OC)c3n2)cc1)NC
CCOP(=O)(OCC)C(O)c1ccc(Nc2ncc3scc(-c4ccccc4OC)c3n2)cc1
CCOP(=O)(Cc1ccc(Nc2ncc3scc(-c4ccccc4OC)c3n2)cc1)N1CCOCC1
CNC(=O)c1ccc(Nc2ncc3scc(-c4ccccc4OC)c3n2)cc1
COc1ccccc1-c1csc2cnc(Nc3ccc(cc3)C(=O)NC3CCNCC3)nc12
COc1ccccc1-c1csc2cnc(Nc3ccc(NC(=O)C4CCNCC4)cc3)nc12
COc1ccccc1-c1csc2cnc(Nc3ccc(NC(=O)[C@H]4CCCNC4)cc3)nc12 |r|
COc1ccccc1-c1csc2cnc(Nc3ccc(NC(=O)[C@@H]4CCCNC4)cc3)nc12 |r|
COc1ccccc1-c1csc2cnc(Nc3ccc(NC(=O)CN)cc3)nc12
COc1ccccc1-c1csc2cnc(Nc3ccc(cc3F)C(=O)NC3CCNCC3)nc12
COc1ccccc1-c1csc2cnc(Nc3ccc(cc3C)C(=O)NC3CCNCC3)nc12
COc1cc(ccc1Nc1ncc2scc(-c3ccccc3OC)c2n1)C(=O)NC1CCNCC1
CCOc1cc(ccc1Nc1ncc2scc(-c3ccccc3OC)c2n1)C(=O)NC1CCNCC1
COc1ccccc1-c1csc2cnc(Nc3ccc(cc3C(F)(F)F)C(=O)NC3CCNCC3)nc12
COc1ccccc1-c1csc2cnc(Nc3ccc(C(=O)NC4CCNCC4)c(F)c3)nc12
COc1ccccc1-c1csc2cnc(Nc3ccc(C(=O)NC4CCNCC4)c(C)c3)nc12
COc1cc(C(=O)NC2CCNCC2)c(F)cc1Nc1ncc2scc(-c3ccccc3OC)c2n1
COc1ccccc1-c1csc2cnc(Nc3cc(F)c(cc3F)C(=O)NC3CCNCC3)nc12
COc1ccccc1-c1csc2cnc(Nc3ccc(C(=O)NC4CCOCC4)c(F)c3)nc12
COc1ccccc1-c1csc2cnc(Nc3ccc(C(=O)NC4CCN(C)CC4)c(F)c3)nc12
COc1ccccc1-c1csc2cnc(Nc3ccc(C(=O)N[C@H]4CCNC4)c(F)c3)nc12 |r|
COc1ccccc1-c1csc2cnc(Nc3ccc(C(=O)N[C@@H]4CCNC4)c(F)c3)nc12 |r|
COc1ccccc1-c1csc2cnc(Nc3ccc(C(=O)NCC4CCNCC4)c(F)c3)nc12
COc1ccccc1-c1csc2cnc(Nc3ccc(C(=O)NC[C@@H]4CCCNC4)c(F)c3)nc12 |r|
COc1ccccc1-c1csc2cnc(Nc3ccc(C(=O)NC[C@H]4CCCNC4)c(F)c3)nc12 |r|
C[C@@H](Nc1ccc2[nH]nc(\C=C\c3ccccn3)c2c1)c1cc(F)cc(F)c1 |r|
CCc1cc(Nc2nc(NCc3ccc(Cl)cc3OC)nc3cccc(OC)c23)n[nH]1
CONC(=O)c1ccccc1Nc1cc(Nc2cc(C)nn2C(C)C)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)N2CCOCC2)ncc1Cl
CNC(=O)c1ccc(Nc2ncc(c(NCc3cccnc3N(C)S(C)(=O)=O)n2)C(F)(F)F)cc1
CONC(=O)c1ccccc1Nc1nc(Nc2cc(C)nn2C(C)C)ncc1Cl
OC(=O)c1ccc(NC(=O)CSc2nnc(-c3ccncc3)n2CC=C)cc1
OC(=O)c1ccc(NC(=O)CSc2nnc(-c3ccncc3)n2-c2ccccc2)cc1
CC(C)n1cc(C(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O
CNC(=O)c1ccc(Nc2ncc(c(NCc3ccccc3F)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(NCc3ccccc3Cl)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(NCc3ccccc3Br)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(NCc3cccc(F)c3)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(NCc3cccc(Cl)c3)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(NCc3cccc(Br)c3)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(NCc3ccc(F)cc3)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(NCc3ccc(Cl)cc3)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(NCc3ccc(Br)cc3)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(NCc3ccccc3OC)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(NCc3ccc(OC)cc3)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(Nc3ccc(F)cc3)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(Nc3ccccc3Cl)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(Nc3ccccc3[N+]([O-])=O)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(Nc3ccc(N)cc3)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(Nc3cccc(N)c3)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(Nc3ccccc3OC)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(Nc3cccc(OC)c3)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(Nc3ccc(OC)cc3)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(Nc3ccc(OC)c(F)c3)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(Nc3ccc(OC)c(Cl)c3)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(Nc3ccc(NC(C)=O)cc3)n2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2ncc(c(Nc3ccc(NS(C)(=O)=O)cc3)n2)C(F)(F)F)cc1
Cn1c(SCCCCCC(O)=O)nnc1-c1ccncc1
CCn1c(SCCCCCC(O)=O)nnc1-c1ccncc1
OC(=O)CCCCCSc1nnc(-c2ccncc2)n1CC=C
OC(=O)CCCCCSc1nnc(-c2ccncc2)n1-c1ccccc1
Cn1c(SCCCCCC(=O)NO)nnc1-c1ccncc1
CCn1c(SCCCCCC(=O)NO)nnc1-c1ccncc1
ONC(=O)CCCCCSc1nnc(-c2ccncc2)n1CC=C
ONC(=O)CCCCCSc1nnc(-c2ccncc2)n1-c1ccccc1
Cn1c(SCCCCCC(=O)Nc2ccccc2N)nnc1-c1ccncc1
CCn1c(SCCCCCC(=O)Nc2ccccc2N)nnc1-c1ccncc1
Nc1ccccc1NC(=O)CCCCCSc1nnc(-c2ccncc2)n1CC=C
Nc1ccccc1NC(=O)CCCCCSc1nnc(-c2ccncc2)n1-c1ccccc1
Cn1c(SCc2ccc(cc2)C(=O)NO)nnc1-c1ccncc1
CCn1c(SCc2ccc(cc2)C(=O)NO)nnc1-c1ccncc1
ONC(=O)c1ccc(CSc2nnc(-c3ccncc3)n2CC=C)cc1
ONC(=O)c1ccc(CSc2nnc(-c3ccncc3)n2-c2ccccc2)cc1
Cn1c(SCc2ccc(cc2)C(=O)Nc2ccccc2N)nnc1-c1ccncc1
CCn1c(SCc2ccc(cc2)C(=O)Nc2ccccc2N)nnc1-c1ccncc1
Nc1ccccc1NC(=O)c1ccc(CSc2nnc(-c3ccncc3)n2CC=C)cc1
Nc1ccccc1NC(=O)c1ccc(CSc2nnc(-c3ccncc3)n2-c2ccccc2)cc1
CN(c1ncccc1CNc1nc(Nc2ccc3NC(=O)Cc3c2)nc2[nH]ccc12)S(C)(=O)=O
CN(c1ncccc1CNc1nc(Nc2ccc3NC(=O)Cc3c2)nc2[nH]ncc12)S(C)(=O)=O
CN(c1ncccc1CNc1nc(Nc2ccc3NC(=O)Cc3c2)nc2[nH]cc(C)c12)S(C)(=O)=O
CN(c1ncccc1CNc1nc(Nc2ccc3NC(=O)Cc3c2)nc2[nH]c(C)cc12)S(C)(=O)=O
CN(c1ncccc1CNc1nc(Nc2ccc3NC(=O)Cc3c2)nc2[nH]cc(F)c12)S(C)(=O)=O
CN(c1ncccc1CNc1nc(Nc2ccc3NC(=O)Cc3c2)nc2[nH]cc(Cl)c12)S(C)(=O)=O
CN(c1ncccc1CNc1nc(Nc2ccc3NC(=O)Cc3c2)nc2[nH]cc(C#N)c12)S(C)(=O)=O
CN(c1ncccc1CNc1nc(Nc2ccccc2)nc2[nH]cc(F)c12)S(C)(=O)=O
CN(c1ncccc1CNc1nc(Nc2ccc(F)cc2)nc2[nH]cc(F)c12)S(C)(=O)=O
CN(c1ncccc1CNc1nc(Nc2ccc(F)c(Cl)c2)nc2[nH]cc(F)c12)S(C)(=O)=O
CN(c1ncccc1CNc1nc(Nc2cccc(c2)C#N)nc2[nH]cc(F)c12)S(C)(=O)=O
COc1ccc(Nc2nc(NCc3cccnc3N(C)S(C)(=O)=O)c3c(F)c[nH]c3n2)cc1OC
COc1cc(Nc2nc(NCc3cccnc3N(C)S(C)(=O)=O)c3c(F)c[nH]c3n2)cc(OC)c1OC
COc1cccc(Nc2nc(NCc3cccnc3N(C)S(C)(=O)=O)c3c(F)c[nH]c3n2)c1C
CN(c1ncccc1CNc1nc(Nc2cccc(CN)c2)nc2[nH]cc(F)c12)S(C)(=O)=O
CN(c1ncccc1CNc1nc(Nc2cccc(CNC(C)=O)c2)nc2[nH]cc(F)c12)S(C)(=O)=O
CN(c1ncccc1CNc1nc(Nc2cccc(NC(C)=O)c2)nc2[nH]cc(F)c12)S(C)(=O)=O
CN(c1ncccc1CNc1nc(Nc2ccc(cc2)N2CCN(C)CC2)nc2[nH]cc(F)c12)S(C)(=O)=O
CN(c1ncccc1CNc1nc(Nc2ccc(cc2)N2CCOCC2)nc2[nH]cc(F)c12)S(C)(=O)=O
COc1cc(ccc1Nc1nc(NCc2cccnc2N(C)S(C)(=O)=O)c2c(F)c[nH]c2n1)N1CCOCC1
CNC(=O)c1ccccc1Nc1nc(Nc2ccc3NC(=O)Cc3c2)nc2[nH]cc(F)c12
CNC(=O)c1ccccc1Nc1nc(Nc2cccc(CNC(C)=O)c2)nc2[nH]cc(F)c12
CNC(=O)c1ccccc1Nc1nc(Nc2cccc(NC(C)=O)c2)nc2[nH]cc(F)c12
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)nc2[nH]cc(F)c12
COc1cc(Nc2ncc3scc(-c4ccccn4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3scc(-c4cccnc4)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3scc(-c4cccc(c4)C(O)=O)c3n2)cc(OC)c1OC
CNC(=O)c1ccccc1-c1csc2cnc(Nc3cc(OC)c(OC)c(OC)c3)nc12
COc1cc(Nc2ncc3scc(-c4ccccc4S(C)(=O)=O)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3scc(-c4cccc(c4)S(C)(=O)=O)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3scc(-c4ccccc4N(C)S(C)(=O)=O)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3scc(-c4cccc(c4)N(C)S(C)(=O)=O)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3scc(-c4ccccc4NS(C)(=O)=O)c3n2)cc(OC)c1OC
COc1cc(Nc2ncc3scc(-c4cccc(NS(C)(=O)=O)c4)c3n2)cc(OC)c1OC
CS(=O)(=O)Nc1cccc(c1)-c1csc2cnc(Nc3ccccc3)nc12
CN(C)c1ccc(Nc2ncc3scc(-c4cccc(NS(C)(=O)=O)c4)c3n2)cc1
CS(=O)(=O)Nc1cccc(c1)-c1csc2cnc(Nc3ccc(cc3)N3CCCCC3)nc12
CS(=O)(=O)Nc1cccc(c1)-c1csc2cnc(Nc3ccc(cc3)N3CCOCC3)nc12
CS(=O)(=O)Nc1cccc(c1)-c1csc2cnc(Nc3ccc(cc3)N3CCNCC3)nc12
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4cccc(NS(C)(=O)=O)c4)c3n2)cc1
CS(=O)(=O)Nc1cccc(c1)-c1csc2cnc(Nc3ccc(cc3)N3CCC(O)CC3)nc12
CCN1CCN(CC1)c1cccc(Nc2ncc3scc(-c4cccc(NS(C)(=O)=O)c4)c3n2)c1
CS(=O)(=O)Nc1cccc(c1)-c1csc2cnc(N)nc12
CS(=O)(=O)Nc1cccc(c1)-c1csc2cnc(NC3CC3)nc12
CS(=O)(=O)Nc1cccc(c1)-c1csc2cnc(NC3CCCCC3)nc12
CS(=O)(=O)Nc1cccc(c1)-c1csc2cnc(NCCO)nc12
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4ccccc4)c3n2)cc1
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4ccccn4)c3n2)cc1
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4cccnc4)c3n2)cc1
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4ccccc4[N+]([O-])=O)c3n2)cc1
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4cccc(c4)[N+]([O-])=O)c3n2)cc1
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4ccccc4S(C)(=O)=O)c3n2)cc1
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4cccc(c4)S(C)(=O)=O)c3n2)cc1
CCOC(=O)c1ccccc1-c1csc2cnc(Nc3ccc(cc3)N3CCN(CC)CC3)nc12
CCOC(=O)c1cccc(c1)-c1csc2cnc(Nc3ccc(cc3)N3CCN(CC)CC3)nc12
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4cccc(c4)C(O)=O)c3n2)cc1
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4cccc(c4)C(=O)NC)c3n2)cc1
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4cccc(OC)c4)c3n2)cc1
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4cccc(c4)S(=O)(=O)NC)c3n2)cc1
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4cccc(c4)N(C)S(C)(=O)=O)c3n2)cc1
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4cccc(c4)N4CCCS4(=O)=O)c3n2)cc1
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4ccc5ccccc5c4)c3n2)cc1
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4cnc5ccccc5c4)c3n2)cc1
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4ccc5cc[nH]c5c4)c3n2)cc1
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)N2CCN(CC2)C(=O)CNC(=O)C=C)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)N2CCN(CC2)C(=O)CCNC(=O)C=C)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)N2CCN(CC2)C(=O)[C@@H](C)NC(=O)C=C)ncc1Cl |r|
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)N2CCN(CC2)C(=O)CNC(=O)C=C)ncc1C(F)(F)F
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)N2CCN(CC2)C(=O)C(C)NC(=O)C=C)ncc1C(F)(F)F
CN1Cc2nn(C)c(C#N)c2-c2cnc3[nH]c(F)c(-c4cn(CCCC1=O)nc4C(F)(F)F)c3c2
CCOC(=O)C1CCN(CC1)c1ccc(Nc2ncc(Cl)c(Nc3ccccc3S(=O)(=O)C(C)C)n2)cc1
CCOC(=O)C1CCN(Cc2ccc(Nc3ncc(Cl)c(Nc4ccccc4S(=O)(=O)C(C)C)n3)cc2)CC1
CC(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(CN3CCC(CO)CC3)cc2)ncc1Cl
CC(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(CN3CCSCC3)cc2)ncc1Cl
CCOP(=O)(Cc1ccc(Nc2ncc(Cl)c(Nc3ccccc3S(=O)(=O)C(C)C)n2)cc1)OCC
CC(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(OCC(=O)N3CCOCC3)cc2)ncc1Cl
CCOC(=O)C1CCN(CC(=O)Nc2ccc(Nc3ncc(Cl)c(Nc4ccccc4S(=O)(=O)C(C)C)n3)cc2)CC1
CCOP(=O)(CC(=O)Nc1ccc(Nc2ncc(Cl)c(Nc3ccccc3S(=O)(=O)C(C)C)n2)cc1)OCC
CC(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(SCCCN3CCOCC3)cc2)ncc1Cl
CC(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)N2CCC(CC2)C(O)=O)ncc1Cl
CC(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(CN3CCC(CC3)C(O)=O)cc2)ncc1Cl
CC(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(NC(=O)CN3CCC(CC3)C(O)=O)cc2)ncc1Cl
CC(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(CN3CCC(CC3)C(=O)NCCO)cc2)ncc1Cl
CCC(C)C(CO)NC(=O)C1CCN(Cc2ccc(Nc3ncc(Cl)c(Nc4ccccc4S(=O)(=O)C(C)C)n3)cc2)CC1
COC(=O)CCCCCNC(=O)C1CCN(CC1)c1ccc(Nc2ncc(Cl)c(Nc3ccccc3S(=O)(=O)C(C)C)n2)cc1
COC(=O)CCCCCNC(=O)C1CCN(CC(=O)Nc2ccc(Nc3ncc(Cl)c(Nc4ccccc4S(=O)(=O)C(C)C)n3)cc2)CC1
CC(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)N2CCC(CC2)C(=O)NCCCCCC(=O)NO)ncc1Cl
CC(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(CN3CCC(CC3)C(=O)NCCCCCC(=O)NO)cc2)ncc1Cl
CC(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(NC(=O)CN3CCC(CC3)C(=O)NCCCCCC(=O)NO)cc2)ncc1Cl
COCC1CN(C1)C1CCN(CC1)c1cc(OC)c(Nc2ncc(Br)c(Nc3ccc4OCCOc4c3P(C)(C)=O)n2)cc1C
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CCOCCOCCNC(=O)CNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)CC2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CCCCCCCCNC(=O)CNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)CC2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CCCOCCC(=O)NCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)CC2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CCOCCOCCOCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)CC2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CCCCC(=O)Nc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)CC2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CCCCCC(=O)Nc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)CC2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CCCCCCC(=O)Nc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)CC2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CCCCCCCC(=O)Nc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)CC2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CCCCCCCCC(=O)Nc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)CC2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CCCCCCCCCC(=O)Nc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)CC2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CCCCC(=O)NCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)CC2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CCCCCC(=O)NCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)CC2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CCCCCCC(=O)NCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)CC2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CCCCCCCC(=O)NCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)CC2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CCCCCCCCCC(=O)NCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)CC2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CC2)C(=S)SCCCCCCCC(=O)Nc2cccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c23)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CC2)C(=S)SCCCCCCCCCC(=O)Nc2cccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c23)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CCCCC(=O)Nc3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)CC2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCN(CCCCC(=O)Nc3cccc4C(=O)N(Cc34)C3CCC(=O)NC3=O)CC2)ncc1Cl
Nc1cc(N)c(N)cc1N
COc1cc(ccc1Nc1nc(-n2ccc3ccccc23)c2cc[nH]c2n1)N1CCC(CC1)N1CCN(C)CC1
COc1cc(ccc1Nc1nc(-n2ccc3ccccc23)c2cc[nH]c2n1)N1CCN(C)CC1
COc1cc(ccc1Nc1nc(-n2cnc3ccccc23)c2cc[nH]c2n1)N1CCC(CC1)N1CCN(C)CC1
COc1cc(ccc1Nc1nc(-n2cnc3ccccc23)c2cc[nH]c2n1)N1CCN(C)CC1
COc1cc(ccc1Nc1nc(-c2cnn(C)c2)c2cc[nH]c2n1)N1CCN(C)CC1
COc1cc(ccc1Nc1nc(-c2cnn(C)c2)c2cc[nH]c2n1)N1CCC(CC1)N1CCN(C)CC1
COc1cc(ccc1Nc1nc(Oc2cccc3CCC(=O)c23)c2cc[nH]c2n1)N1CCN(C)CC1
CN1CCN(CC1)C1CCN(CC1)c1ccc(Nc2nc(Oc3cccc4CCC(=O)c34)c3cc[nH]c3n2)cc1
COc1cc(ccc1Nc1nc(Oc2ccc(C)c3CCC(=O)c23)c2cc[nH]c2n1)N1CCN(C)CC1
CN1CCN(CC1)C1CCN(CC1)c1ccc(Nc2nc(Oc3ccc(C)c4CCC(=O)c34)c3cc[nH]c3n2)cc1
CN1CCN(CC1)c1ccc(Nc2nc(Oc3cccc4CCC(=O)c34)c3cc[nH]c3n2)cc1
O=C1CCc2cccc(Oc3nc(Nc4ccc(cc4)N4CCOCC4)nc4[nH]ccc34)c12
COc1cc(ccc1Nc1nc(Oc2cccc3CCC(=O)c23)c2cc[nH]c2n1)N1CCOCC1
CN1CCN(CC1)c1ccc(Nc2nc(Oc3cccc4CCC(=O)c34)c3ccsc3n2)cc1
O=C1CCc2cccc(Oc3nc(Nc4ccc(cc4)N4CCOCC4)nc4sccc34)c12
COc1cc(ccc1Nc1nc(Oc2cccc3CCC(=O)c23)c2ccsc2n1)N1CCN(C)CC1
COc1cc(ccc1Nc1nc(Oc2cccc3CCC(=O)c23)c2ccsc2n1)N1CCOCC1
COc1cc(ccc1Nc1nc(Oc2cccc3CCC(=O)c23)c2ccsc2n1)N1CCC(CC1)N1CCN(C)CC1
CN1CCN(CC1)c1ccc(Nc2nc(Oc3cccc4CCC(=O)c34)c3[nH]ccc3n2)cc1
O=C1CCc2cccc(Oc3nc(Nc4ccc(cc4)N4CCOCC4)nc4cc[nH]c34)c12
COc1cc(ccc1Nc1nc(Oc2cccc3CCC(=O)c23)c2[nH]ccc2n1)N1CCN(C)CC1
COc1cc(ccc1Nc1nc(Oc2cccc3CCC(=O)c23)c2[nH]ccc2n1)N1CCOCC1
COc1cc(ccc1Nc1nc(Oc2cccc3CCC(=O)c23)c2[nH]ccc2n1)N1CCC(CC1)N1CCN(C)CC1
CN1CCN(CC1)c1ccc(Nc2nc(Oc3cccc4CCC(=O)c34)c3sccc3n2)cc1
O=C1CCc2cccc(Oc3nc(Nc4ccc(cc4)N4CCOCC4)nc4ccsc34)c12
COc1cc(ccc1Nc1nc(Oc2cccc3CCC(=O)c23)c2sccc2n1)N1CCN(C)CC1
COc1cc(ccc1Nc1nc(Oc2cccc3CCC(=O)c23)c2sccc2n1)N1CCOCC1
COc1cc(ccc1Nc1nc(Oc2cccc3CCC(=O)c23)c2sccc2n1)N1CCC(CC1)N1CCN(C)CC1
CN1CCN(CC1)c1ccc(Nc2nc(Oc3cccc4CCC(=O)c34)c3ccccc3n2)cc1
O=C1CCc2cccc(Oc3nc(Nc4ccc(cc4)N4CCOCC4)nc4ccccc34)c12
COc1cc(ccc1Nc1nc(Oc2cccc3CCC(=O)c23)c2ccccc2n1)N1CCN(C)CC1
COc1cc(ccc1Nc1nc(Oc2cccc3CCC(=O)c23)c2ccccc2n1)N1CCOCC1
COc1cc(ccc1Nc1nc(Oc2cccc3CCC(=O)c23)c2ccccc2n1)N1CCC(CC1)N1CCN(C)CC1
COc1cc(ccc1Nc1nc(Oc2cccc3CCC(=O)c23)c2cc[nH]c2n1)N1C[C@H](C)O[C@H](C)C1 |r|
[H][C@]12CN(c3ccc(Nc4nc(Oc5cccc6CCC(=O)c56)c5cc[nH]c5n4)c(OC)c3)[C@]([H])(CO1)C2 |r|
COc1cc(ccc1Nc1nc(Oc2cccc3CCC(=O)c23)c2cc[nH]c2n1)C(=O)NC1CCNCC1
COc1cc(ccc1Nc1nc(Oc2cccc3CCC(=O)c23)c2cc[nH]c2n1)C(=O)NC1CC1
CN1CCN(CC1)c1ccc(Nc2nc(Oc3cccc4CCC(=O)c34)c3cc[nH]c3n2)c(c1)C(F)(F)F
CN1CCN(CC1)c1ccc(Nc2nc(Oc3cccc4CCC(=O)c34)c3cc[nH]c3n2)c(C)c1
CN1CCN(CC1)c1ccc(Nc2nc(Oc3cccc4CCC(=O)c34)c3cc[nH]c3n2)cc1F
CN1CCN(CC1)c1ccc(Nc2nc(Oc3cccc4CCC(=O)c34)c3cc[nH]c3n2)cc1Cl
CN1CCN(CC1)c1ccc(Nc2nc(Oc3cccc4CCC(=O)c34)c3cc[nH]c3n2)cc1C#N
Cc1cc(Nc2nc(Oc3cccc4CCC(=O)c34)c3cc[nH]c3n2)ccc1N1CCN(CC2CC2)CC1
Cc1cc(Nc2nc(Oc3cccc4CCC(=O)c34)c3cc[nH]c3n2)ccc1N1CCN(CC1)C1COC1
CN(C)CCOc1ccc(Nc2nc(Oc3cccc4CCC(=O)c34)c3cc[nH]c3n2)cc1C
COc1nc(ccc1Nc1nc(Oc2cccc3CCC(=O)c23)c2cc[nH]c2n1)N1CCN(C)CC1
CC(C)n1nc(C)cc1Nc1nc(Oc2cccc3CCC(=O)c23)c2cc[nH]c2n1
O=C1CCc2cccc(Oc3nc(Nc4ccc5C(=O)NCc5c4)nc4[nH]ccc34)c12
C[C@@H]1CCN(C[C@@H]1n1ccc2cnc3[nH]ccc3c12)C(=O)CC#N |r|
C[C@@H]1CCN(C[C@@H]1n1ccc2cnc3[nH]cc(C#N)c3c12)C(=O)CC#N |r|
OC1CCCN(C1)C(=O)c1cccc(c1)-c1n[nH]c2ncc(Cc3cc(F)ccc3F)cc12
O[C@@H]1CCCN(C1)C(=O)c1cccc(c1)-c1n[nH]c2ncc(Cc3cc(F)ccc3F)cc12 |r|
O[C@H]1CCCN(C1)C(=O)c1cccc(c1)-c1n[nH]c2ncc(Cc3cc(F)ccc3F)cc12 |r|
c1ccc(nc1)-c1nnn[nH]1
c1ccc(nc1)-c1nc2ccccc2[nH]1
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(cc2OC)N2CCOCC2)ncc1C(F)(F)F
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N2CCOCC2)ncc1Cl
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N2CCNCC2)ncc1Cl
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N2CCC[C@@H](N)C2)ncc1Cl |r|
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N2CCC[C@H](N)C2)ncc1Cl |r|
CNC1CCN(CC1)C(=O)c1ccc(Nc2ncc(Cl)c(Nc3ccccc3P(C)(C)=O)n2)cc1
CN(C1CCNCC1)C(=O)c1ccc(Nc2ncc(Cl)c(Nc3ccccc3P(C)(C)=O)n2)cc1
CN(C1CCCNC1)C(=O)c1ccc(Nc2ncc(Cl)c(Nc3ccccc3P(C)(C)=O)n2)cc1
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)NC2CCNCC2)ncc1Cl
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N[C@H]2CCNC2)ncc1Cl |r|
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N[C@@H]2CCNC2)ncc1Cl |r|
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)NCC2CCNCC2)ncc1Cl
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)NC2CCOCC2)ncc1Cl
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)NC2CCC(O)CC2)ncc1Cl |(7.68,-.7,;6.59,.39,;8.08,.79,;6.59,1.93,;5.26,-.38,;5.25,-1.92,;3.92,-2.69,;2.59,-1.92,;2.58,-.38,;3.92,.39,;3.92,1.93,;2.59,2.7,;1.26,1.92,;-.08,2.7,;-1.41,1.93,;-1.41,.39,;-2.75,-.38,;-2.75,-1.93,;-1.41,-2.69,;-.08,-1.92,;-.08,-.38,;-1.41,-4.23,;-.08,-5,;-2.74,-5,;-4.08,-4.23,;-5.41,-5,;-6.75,-4.23,;-6.75,-2.69,;-8.08,-1.92,;-5.41,-1.92,;-4.08,-2.69,;-.08,4.24,;1.25,5,;2.59,4.23,;3.92,5,)|
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)N2CCC(CC2)N2CCOCC2)ncc1Cl
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2F)C(=O)NC2CCC(O)CC2)ncc1Cl |(7.68,-.7,;6.59,.39,;8.08,.79,;6.59,1.93,;5.26,-.38,;5.25,-1.92,;3.92,-2.69,;2.59,-1.92,;2.58,-.38,;3.92,.39,;3.92,1.93,;2.59,2.7,;1.26,1.92,;-.08,2.7,;-1.41,1.93,;-1.41,.39,;-.08,-.38,;-.08,-1.92,;-1.41,-2.69,;-2.75,-1.93,;-2.75,-.38,;-4.08,.39,;-1.41,-4.23,;-.08,-5,;-2.74,-5,;-4.08,-4.23,;-5.41,-5,;-6.74,-4.23,;-6.74,-2.69,;-8.08,-1.92,;-5.41,-1.92,;-4.08,-2.69,;-.08,4.24,;1.25,5,;2.59,4.23,;3.92,5,)|
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(C(=O)NC3CCC(O)CC3)c(F)c2)ncc1Cl |(5.68,2.38,;4.59,3.47,;6.08,3.87,;4.59,5.01,;3.26,2.7,;3.25,1.16,;1.92,.39,;.59,1.16,;.58,2.7,;1.92,3.47,;1.92,5.01,;.59,5.78,;-.74,5,;-2.08,5.78,;-3.41,5.01,;-3.41,3.47,;-2.08,2.7,;-2.08,1.16,;-3.41,.39,;-3.41,-1.15,;-2.08,-1.92,;-4.74,-1.92,;-4.74,-3.46,;-3.41,-4.23,;-3.41,-5.77,;-4.74,-6.54,;-4.74,-8.08,;-6.08,-5.77,;-6.08,-4.23,;-4.75,1.15,;-6.08,.38,;-4.75,2.7,;-2.08,7.32,;-.75,8.08,;.59,7.31,;1.92,8.08,)|
COc1cc(ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1)C(=O)NC1CCC(O)CC1 |(-5.41,-.38,;-4.08,.39,;-2.75,-.38,;-2.75,-1.93,;-1.41,-2.69,;-.08,-1.92,;-.08,-.38,;-1.41,.39,;-1.41,1.93,;-.08,2.7,;-.08,4.24,;1.25,5,;2.59,4.23,;3.92,5,;2.59,2.7,;3.92,1.93,;3.92,.39,;2.58,-.38,;2.59,-1.92,;3.92,-2.69,;5.25,-1.92,;5.26,-.38,;6.59,.39,;7.68,-.7,;8.08,.79,;6.59,1.93,;1.26,1.92,;-1.41,-4.23,;-.08,-5,;-2.74,-5,;-4.08,-4.23,;-5.41,-5,;-6.75,-4.23,;-6.75,-2.69,;-8.08,-1.92,;-5.41,-1.92,;-4.08,-2.69,)|
Cc1cc(ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1)C(=O)NC1CCC(O)CC1 |(-4.08,.39,;-2.75,-.38,;-2.75,-1.93,;-1.41,-2.69,;-.08,-1.92,;-.08,-.38,;-1.41,.39,;-1.41,1.93,;-.08,2.7,;-.08,4.24,;1.25,5,;2.58,4.23,;3.92,5,;2.59,2.7,;3.92,1.93,;3.92,.39,;2.58,-.38,;2.59,-1.92,;3.92,-2.69,;5.25,-1.92,;5.26,-.38,;6.59,.39,;7.68,-.7,;8.08,.79,;6.59,1.93,;1.26,1.92,;-1.41,-4.23,;-.08,-5,;-2.74,-5,;-4.08,-4.23,;-5.41,-5,;-6.74,-4.23,;-6.74,-2.69,;-8.08,-1.92,;-5.41,-1.92,;-4.08,-2.69,)|
Cc1cc(Nc2ncc(Cl)c(Nc3ccccc3P(C)(C)=O)n2)ccc1C(=O)NC1CCC(O)CC1 |(-6.08,.38,;-4.75,1.15,;-4.75,2.7,;-3.41,3.47,;-3.41,5.01,;-2.08,5.78,;-2.08,7.32,;-.75,8.08,;.59,7.31,;1.92,8.08,;.59,5.78,;1.92,5.01,;1.92,3.47,;.58,2.7,;.59,1.16,;1.92,.39,;3.26,1.16,;3.26,2.7,;4.59,3.47,;5.68,2.38,;6.08,3.87,;4.59,5.01,;-.74,5,;-2.08,2.7,;-2.08,1.16,;-3.41,.39,;-3.41,-1.15,;-2.08,-1.92,;-4.74,-1.92,;-4.74,-3.46,;-3.41,-4.23,;-3.41,-5.77,;-4.74,-6.54,;-4.74,-8.08,;-6.08,-5.77,;-6.08,-4.23,)|
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2F)C(=O)NC2CCNCC2)ncc1Cl
CP(C)(=O)c1ccccc1Nc1nc(Nc2ccc(C(=O)NC3CCNCC3)c(F)c2)ncc1Cl
COc1cc(ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1)C(=O)NC1CCNCC1
Cc1cc(ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1)C(=O)NC1CCNCC1
Cc1cc(Nc2ncc(Cl)c(Nc3ccccc3P(C)(C)=O)n2)ccc1C(=O)NC1CCNCC1
COc1c(Nc2cc(C)[nH]n2)nc(Sc2ccc(cc2F)S(=O)(=O)Cc2cccc(c2F)[N+]([O-])=O)nc1N1CCOCC1
CC(C)Nc1cc(F)cc(c1)-c1n[nH]c2ncc(cc12)-c1cccc(c1)S(C)(=O)=O
CC(=O)Nc1cc(F)cc(c1)-c1n[nH]c2ncc(cc12)-c1cccc(c1)S(C)(=O)=O
CS(=O)(=O)c1cccc(c1)-c1cnc2[nH]nc(-c3cc(F)cc(NC(=O)Nc4ccccc4)c3)c2c1
CS(=O)(=O)c1cccc(c1)-c1cnc2[nH]nc(-c3cc(F)cc(NC(=O)Nc4cccnc4)c3)c2c1
CS(=O)(=O)c1cccc(c1)-c1cnc2[nH]nc(-c3cc(F)cc(NC(=O)Nc4cncnc4)c3)c2c1
Fc1cc(NC(=O)Nc2cncnc2)cc(c1)-c1n[nH]c2ncc(cc12)-c1ccc(CN2CCOCC2)cc1
CN1CCN(Cc2ccc(cc2)-c2cnc3[nH]nc(-c4cc(F)cc(NC(=O)Nc5cncnc5)c4)c3c2)CC1
CCOc1cc(ccc1Nc1ncc2cc(-c3cccc(NC(=O)c4cccc(c4)C(F)(F)F)c3)c(=O)n(C[C@H]3CCCO3)c2n1)N1CCN(C)CC1 |r|
COc1ccc(\C=C/c2cc(OC)c(OC)c(OC)c2)cc1NC(=O)CCC(=O)N[C@@H](CCCNC(N)=N)C(O)=O |r|
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(CC(=O)OCCCCCOc3no[n+]([O-])c3S(=O)(=O)c3ccccc3)cc2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(CC(=O)OCCCCCCCOc3no[n+]([O-])c3S(=O)(=O)c3ccccc3)cc2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(CC(=O)OCCCCCCCCOc3no[n+]([O-])c3S(=O)(=O)c3ccccc3)cc2)ncc1Cl
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(CC(=O)OCC(C)COc3no[n+]([O-])c3S(=O)(=O)c3ccccc3)cc2)ncc1Cl
CN(c1ncccc1CNc1nc(Nc2ccc(N3CCN(CCCCCCC(=O)NCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(NC(=O)CCCCCCC(=O)NO)cc2)ncc1Cl
C=CC(=O)Nc1cc(Nc2nccc(-c3cnc4c(C)cccn34)n2)c(OC)cc1N(C)CCN(C)C
C[C@@H](C(F)(F)F)N(Cc1ccc(cc1)F)C(=O)CN2C(=O)[C@]3(CCc4c3ccc(c4)NC(=O)NC)OC2=O
Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1Nc1nc(-c2cccnc2)nc2nn(C)cc12
Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1Nc1nc(-c2cccnc2)nc2c1cnn2C
COc1cc2c(cc1OCCCN3CCOCC3)ncnc2Nc4ccc(cc4)NC(=O)c5ccccc5
COc1cc2nccc(Oc3ccc(NC(=O)Nc4cc(C)on4)c(Cl)c3)c2cc1OC
CCOc1cc(ccc1Nc2ncc3c(n2)N(c4ccccc4C(=O)N3C)C)N5CCC(CC5)O
C[C@@]1(O)C[C@@H](C1)c1nc(-c2ccc3ccc(nc3c2)-c2ccccc2)c2c(N)nccn12 |r,wU:1.1,4.6,wD:1.0,(18.42,-37.26,;17.1,-36.49,;16.31,-37.82,;17.79,-35.11,;16.41,-34.42,;15.72,-35.8,;15.93,-32.97,;16.83,-31.71,;15.91,-30.47,;16.38,-29.01,;15.35,-27.88,;15.81,-26.41,;17.32,-26.08,;17.78,-24.62,;19.27,-24.29,;20.31,-25.42,;19.85,-26.89,;18.35,-27.21,;17.89,-28.68,;21.81,-25.09,;22.85,-26.23,;24.35,-25.9,;24.82,-24.43,;23.77,-23.29,;22.27,-23.63,;14.45,-30.96,;13.11,-30.19,;13.11,-28.65,;11.78,-30.96,;11.78,-32.51,;13.12,-33.28,;14.46,-32.5,)|
Cc1cn(CCN2CCN(CC2)c2ccccc2-c2cc(cc(c2)C(=O)NCCCN2CCCC2)C#N)c2ccccc12
CCc1cc(Nc2nccc(n2)-c2c(nc3ccccn23)-c2ccc(OC)c(c2)C(=O)Nc2c(F)cccc2F)c(OC)cc1N1CCC(CC1)N1CCN(CC1)S(C)(=O)=O
C[C@]1(CCCN1c1nc(Nc2cc([nH]n2)C2CC2)c2cccn2n1)C(=O)Nc1ccc(F)nc1 |r|
CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3cc(nn3-c3ccc4ncccc4c3)C(C)(C)C)c(F)c2)ccn1
c1cc(c(cc1I)F)Nc2c(ccc(c2F)F)C(=O)N3CC(C3)([C@@H]4CCCCN4)O
CC1=CN2C(=O)C=C(N=C2C(=C1)[C@@H](C)Nc3ccccc3C(=O)O)N4CCOCC4
CN1CCN(CC1)C2CCN(CC2)c3ccc(c(c3)OC)Nc4ncc(c(n4)Nc5ccccc5P(=O)(C)C)Cl
CN1CCN(CC1)c2ccc(c(c2)OC)Nc3ncc(c(n3)Oc4cccc(c4)NC(=O)C=C)Cl
CCc1cccc(CC)c1NC(=O)c1nn(C)c-2c1CCc1cnc(Nc3ccc(cc3OC(F)(F)F)C(=O)NC3CCN(C)CC3)nc-21
O=C1c2ccccc2-c2n[nH]c3cccc1c23
C[C@H]1Oc2cc(cnc2N)-c2c(nn(C)c2C#N)CN(C)C(=O)C2C=CC(F)=CC21
CC[C@@H]1CN(C[C@@H]1c1cnc2cnc3[nH]ccc3n12)C(=O)NCC(F)(F)F |r|
C[C@@]12[C@@H]([C@@H](C[C@@H](O1)n3c4ccccc4c5c3c6n2c7ccccc7c6c8c5C(=O)NC8)NC)OC
CN(c1c(cccn1)CNc2ccnc(n2)Nc3ccc4c(c3)CC(=O)N4)S(=O)(=O)C
CN(c1ncccc1CNc1nc(Nc2ccccc2)ncc1C(F)(F)F)S(C)(=O)=O
CN(c1c(cccn1)CNc2c(cnc(n2)Nc3ccc4c(c3)CCC(=O)N4)C(F)(F)F)S(=O)(=O)C
c1cc(cnc1)CNc2c(cnc(n2)Nc3ccc4c(c3)CC(=O)N4)C(F)(F)F
CN(C)[C@@H]1CCC[C@H]1Nc1nc(Nc2ccc(C(=O)NC3CC3)cc2)ncc1C(F)(F)F