8484 SMILES Strings for Histone deacetylase 6

Compound Name
SMILES String
CC(C=CC(=O)NO)C=C(C)C(=O)c1ccc(cc1)N(C)C |w:8.7,2.1|
SCCCCCCC(=O)Nc1nc(cs1)-c1ccccc1
CC(C)(C)OC(=O)N[C@@H](CCCCCS)C(=O)Nc1cccc(c1)-c1ccccc1 |r|
CC(C)(C)OC(=O)N[C@@H](CCCCCS)C(=O)Nc1cnc2ccccc2c1 |r|
CC(C)(C)OC(=O)N[C@@H](CCCCCS)C(=O)NC1CCCC1 |r|
CC(C)(C)OC(=O)N[C@@H](CCCCCS)C(=O)NC1CCCCC1 |r|
CC(C)(C)OC(=O)N[C@@H](CCCCCS)C(=O)NC1CCCCCC1 |r|
CC(C)(C)NC(=O)[C@H](CCCCCS)NC(=O)OC(C)(C)C |r|
CC(C)(C)OC(=O)N[C@@H](CCCCCS)C(=O)NC12CC3CC(CC(C3)C1)C2 |r,TLB:21:22:26:20.19.25,25:20:27:24.26.23,25:24:27:20.19.21,THB:21:20:26:22.27.23|
N[C@@H](CCCCCS)C(=O)NC1CCCC1 |r|
SCCCCC[C@H](NC(=O)c1ccccc1)C(=O)NC1CCCC1 |r|
SCCCCC[C@H](NC(=O)c1ccc(Cl)cc1)C(=O)NC1CCCC1 |r|
OCC(=O)N[C@@H](CCCCCS)C(=O)NC1CCCC1 |r|
CC(C)(C)C(=O)N[C@@H](CCCCCS)C(=O)NC1CCCC1 |r|
CC(C)(C)NC(=O)N[C@@H](CCCCCS)C(=O)NC1CCCC1 |r|
CC(C)(C)NC(=S)N[C@@H](CCCCCS)C(=O)NC1CCCC1 |r|
COC(=O)N[C@@H](CCCCCS)C(=O)NC1CCCC1 |r|
SCCCCC[C@H](NC(=O)OC1CCCCC1)C(=O)NC1CCCC1 |r|
SCCCCC[C@H](NC(=O)OCc1ccccc1)C(=O)NC1CCCC1 |r|
c1ccc(cc1)NC(=O)CCCCCCC(=O)NO
C\C=C1/NC(=O)[C@H]2CSSCC\C=C\[C@H](CC(=O)N[C@H](C(C)C)C(=O)N2)OC(=O)[C@@H](NC1=O)C(C)C |r,t:12|
CC(C)[C@H]1NC(=O)[C@H]2CSSCC\C=C\[C@H](CC(=O)N[C@H](C)C(=O)N2)OC(=O)CNC1=O |r,t:13|
CC(C)[C@H]1NC(=O)C[C@@H]2OC(=O)CNC(=O)[C@H](NC(=O)[C@@H](CSSCC\C=C\2)NC1=O)C(C)C |t:26|
CC(C)[C@H]1NC(=O)[C@@H](C)NC(=O)[C@@H](C)NC(=O)C[C@@H](OC(=O)CNC1=O)\C=C\CCS |r|
CC(C)[C@H]1NC(=O)[C@H](C)NC(=O)[C@@H](C)NC(=O)C[C@@H](OC(=O)CNC1=O)\C=C\CCSC(C)=O |r|
CC1(C)NC(=O)[C@H](CCCCCC=C)NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC1=O |r|
CC1(C)NC(=O)[C@H](CCCCCC2CO2)NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC1=O |r|
CC1(C)NC(=O)[C@H](CCCCCC(=O)CBr)NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC1=O |r|
CC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC(=O)C(C)(C)NC1=O |r|
CC1(C)NC(=O)[C@H](CCCCCC(O)CO)NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC1=O |r|
CC1(C)NC(=O)[C@H](CCCCCC=O)NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC1=O |r|
CC1(C)NC(=O)[C@H](CCCCCC(=O)CO)NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC1=O |r|
OCc1ccc(cc1)[C@@H]1C[C@H](CSc2nc(c(o2)-c2ccccc2)-c2ccccc2)O[C@@H](O1)c1ccc(NC(=O)CCCCCCC(=O)NO)cc1 |r|
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)[C@H]1O[C@@H](CSc2ccncc2)C[C@H](O1)c1ccccc1 |r|
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1cn(Cc2ccccc2)nn1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1cn(Cc2ccc(F)cc2)nn1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1cn(nn1)-c1ccccc1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1cn(CC(O)c2cccc(Br)c2)nn1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(Cc2ccccc2)nn1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(Cc2ccc(F)cc2)nn1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(nn1)-c1ccccc1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(CC(O)c2cccc(Br)c2)nn1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1cnnn1Cc1ccccc1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1cnnn1Cc1ccc(F)cc1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1cnnn1-c1ccccc1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1cnnn1CC(O)c1cccc(Br)c1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cnnn1Cc1ccccc1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cnnn1Cc1ccc(F)cc1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cnnn1-c1ccccc1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cnnn1CC(O)c1cccc(Br)c1
CN(C)Cc1c(oc2ccccc12)C(=O)NCCOc1ccc(cc1)C(=O)NO
Nc1ccccc1NC(=O)c1ccc(CNc2nccc(n2)-c2cccnc2)cc1
Nc1ccccc1NC(=O)c1ccc(CNC(=O)OCc2cccnc2)cc1
COc1ccc2[nH]c(C)c(CC(=O)N[C@@H](CCCCCC(C)=O)c3nc(c[nH]3)-c3ccccc3)c2c1 |r|
CCc1nc2ccccc2n1[C@@H]1CCN(C1)C(=O)c1nc2ccc(OC)cc2[nH]1 |r|
CCC(=O)CCCCC[C@H](NC(=O)Cc1c(C)[nH]c2ccc(OC)cc12)c1nc(c[nH]1)-c1ccccc1 |r|
OCCN(CCc1c[nH]c2ccccc12)Cc1ccc(\C=C\C(=O)NO)cc1
c1ccc(cc1)NS(=O)(=O)c2cccc(c2)/C=C/C(=O)NO
CCC(C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)CC)NC(=O)[C@H]2CCCCN2C1=O |r|
FC(F)(F)C(=O)CCCCCCC(=O)Nc1cccc(c1)-c1ccccc1
CCOC(=O)c1ccc(s1)C(=O)C(F)(F)F
CCOC(=O)c1ccc(o1)C(=O)C(F)(F)F
CCNC(=O)c1ccc(s1)C(=O)C(F)(F)F
FC(F)(F)C(=O)c1ccc(s1)C(=O)NCCc1ccccc1
CN(Cc1ccccc1)C(=O)c1ccc(s1)C(=O)C(F)(F)F
C[C@@H](NC(=O)c1ccc(s1)C(=O)C(F)(F)F)c1ccccc1 |r|
C[C@H](NC(=O)c1ccc(s1)C(=O)C(F)(F)F)c1ccccc1 |r|
COc1ccc(CNC(=O)c2ccc(s2)C(=O)C(F)(F)F)cc1
FC(F)(F)C(=O)c1ccc(s1)C(=O)NCC1CCCCC1
FC(F)(F)C(=O)c1ccc(s1)C(=O)N1CCc2ccccc12
CN(Cc1ccc2nccnc2c1)C(=O)c1ccc(s1)C(=O)C(F)(F)F
FC(F)(F)C(=O)c1ccc(s1)C(=O)N1CCn2c(C1)ncc2-c1ccccc1
CN(Cc1ccccc1)C(=O)c1ccc(s1)C(O)C(F)(F)F
FC(F)(F)C1(OCCO1)c1ccc(s1)C(=O)N1CCc2ccccc12
CN(Cc1ccc2nccnc2c1)C(=O)c1ccc(s1)C(O)=O
C[C@@H](NC(=O)c1ccc(s1)C(=O)NO)c1ccccc1 |r|
C[C@@H](NC(=O)c1ccc(s1)C(C)=O)c1ccccc1 |r|
COc1ccc(CNC(=O)c2ccc(s2)C(=O)C(F)(F)C(F)(F)F)cc1
OP(O)(=O)c1ccc(s1)C(=O)N1CCc2ccccc12
FC(F)C(=O)c1ccc(s1)C(=O)N1CCc2ccccc12
OB(O)C(=O)c1ccc(s1)C(=O)N1CCc2ccccc12
CS(=O)(=O)c1ccc(s1)C(=O)N1CCc2ccccc12
CN(Cc1ccc(s1)C(=O)C(F)(F)F)Cc1ccccc1
C[C@@H](NCc1ccc(s1)C(=O)C(F)(F)F)c1ccccc1 |r|
COc1ccc(COCc2ccc(s2)C(=O)C(F)(F)F)cc1
CN(Cc1ccccc1)S(=O)(=O)c1csc(c1)C(=O)C(F)(F)F
CN(Cc1ccccc1)S(=O)(=O)c1ccc(s1)C(=O)C(F)(F)F
CN(Cc1ccccc1)C(=O)c1cc(cs1)C(=O)C(F)(F)F
FC(F)(F)C(=O)c1csc(c1)C(=O)NCC1CCCCC1
CN(Cc1ccccc1)C(=O)c1cnc(s1)C(=O)C(F)(F)F
FC(F)(F)C(=O)c1ncc(s1)C(=O)NCC1CCCCC1
FC(F)(F)C(=O)c1ccc([nH]1)C(=O)N1CCc2ccccc12
FC(F)(F)C(=O)c1cccc(c1)C(=O)NCC1CCCCC1
FC(F)(F)C(=O)c1ccc(cc1)C(=O)NCC1CCCCC1
NC(=O)c1ccc(cn1)C(=O)C(F)(F)F
Oc1cccn(CCCn2cc(nn2)-c2ccccc2)c1=S
Oc1cccn(CCCCn2cc(nn2)-c2ccccc2)c1=S
Oc1cccn(CCCCCn2cc(nn2)-c2ccccc2)c1=S
Cc1ccc(cc1)-c1cn(CCCCCn2cccc(O)c2=S)nn1
Cc1cccc(c1)-c1cn(CCCCCn2cccc(O)c2=S)nn1
Cc1ccccc1-c1cn(CCCCCn2cccc(O)c2=S)nn1
Oc1cccn(CCCCCn2cc(nn2)-c2ccc(cc2)C#N)c1=S
Oc1cccn(CCCCCn2cc(nn2)-c2cccc(c2)C#N)c1=S
CN(C)c1ccc(cc1)-c1cn(CCCCCn2cccc(O)c2=S)nn1
Oc1cccn(CCCCCn2cc(nn2)-c2ccc(C#N)c(c2)C(F)(F)F)c1=S
Oc1cccn(Cc2ccc(Cn3cc(nn3)-c3ccccc3)cc2)c1=S
CCCC(CCC)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1 |r|
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)N(c1ccccc1)c1ccccc1
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)N(c1ncccn1)c1ncccn1
COc1ccc(cc1)N(c1ccc(OC)cc1)c1ccc(cc1)C(=O)NCCCCCCC(=O)NO
CN(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)c1c(Cl)cccc1Cl
ONC(=O)CCCCCCCNC(=O)c1ccc(cc1)N(c1ncccn1)c1ncccn1
CN(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)c1ccccc1C(F)(F)F
CC(C)c1cccc(C(C)C)c1N(C)c1ccc(cc1)C(=O)NCCCCCCC(=O)NO
CN(c1ccccc1)c1ncc(cn1)C(=O)NCCCCCCC(=O)NO
CC(C)c1cccc(C(C)C)c1Nc1ccc(cc1)C(=O)NCCCCCCC(=O)NO
CC(C)c1ccccc1N(C)c1ncc(cn1)C(=O)NCCCCCCC(=O)NO
Cc1cccc(C)c1Nc1ccc(cc1)C(=O)NCCCCCCC(=O)NO
CCN(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)c1ccccc1C(F)(F)F
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)N(c1ccccc1)c1ccccc1
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)N(c1ncccn1)c1ncccn1
CCN(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)c1c(Cl)cccc1Cl
ONC(=O)CCCCCCNC(=O)c1ccc(Nc2c(Cl)cccc2Cl)cc1
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)N(c1ccccc1)c1ncccn1
CC(C)c1ccccc1N(C)c1ncc(cn1)C(=O)N(C)CCCCCCC(=O)NO
CN(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)c1c(C)cccc1Cl
CN(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)c1c(F)cccc1F
CCN(c1ccc(cc1)C(=O)N(C)CCCCCCC(=O)NO)c1ccccc1C(F)(F)F
ONC(=O)CCCCCCNC(=O)c1ccc(Nc2c(F)cccc2F)cc1
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)N(c1cccc(Cl)c1)c1cccc(Cl)c1
Cc1cccc(C)c1Nc1ncc(cn1)C(=O)NCCCCCCC(=O)NO
c1ccc(cc1)N(c2ccccc2)c3ncc(cn3)C(=O)NCCCCCCC(=O)NO
CN(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)c1cnccn1
CN(CCCCCCC(=O)NO)C(=O)c1ccc(Nc2c(C)cccc2C)cc1
CCN(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)c1cnccn1
Cn1c(Nc2ccc(cc2)C(=O)NCCCCCCC(=O)NO)nc2ccccc12
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)N(c1ccccc1)c1cncnc1
CC(=O)N(c1ccccc1)c1ccc(cc1)C(=O)NCCCCCCC(=O)NO
ONC(=O)CCCCCCNC(=O)c1ccc(Nc2nc3ccccc3o2)cc1
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)N(c1ccccc1)c1cnccn1
CN(CCCCCCC(=O)NO)C(=O)c1cnc(Nc2c(C)cccc2C)nc1
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)N(c1ccccc1)c1ccccn1
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)N(c1ccccc1)S(=O)(=O)c1ccccc1
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)N(c1ccccc1)c1cccnc1
Cc1cccnc1N(c1ccccc1)c1ccc(cc1)C(=O)NCCCCCCC(=O)NO
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)N(C)c1nc2ccccc2o1
CN(c1nc2ccccc2o1)c1ccc(cc1)C(=O)NCCCCCCC(=O)NO
CN(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)c1ccccc1C#N
ONC(=O)CCCCCCNC(=O)c1ccc(Nc2nc3ccccc3s2)cc1
CC(=O)N(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)c1c(C)cccc1C
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)N(c1ccccc1)c1cccnc1
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)N(C)c1ccccc1C#N
ONC(=O)CCCCCCNC(=O)c1ccc(Nc2ccccc2)cc1
Cc1cccc(C)c1Nc1ccc(C(=O)NCCCCCCC(=O)NO)c(F)c1
CN(c1ccc(C(=O)NCCCCCCC(=O)NO)c(F)c1)c1c(C)cccc1C
CN(CCCCCCC(=O)NO)C(=O)c1ccc(Nc2ccccc2)cc1
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1F)N(C)c1c(C)cccc1C
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)N(C(C)=O)c1ccccc1
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)N(C(C)=O)c1c(C)cccc1C
CC(C)C(=O)N(c1ccccc1)c1ccc(cc1)C(=O)N(C)CCCCCCC(=O)NO
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)N(c1ccccc1)c1ccccn1
CC(C)C(=O)N(c1ccc(cc1)C(=O)N(C)CCCCCCC(=O)NO)c1c(C)cccc1C
Cc1cccc(C)c1Nc1ccc(cc1F)C(=O)NCCCCCCC(=O)NO
CN(CCCCCCC(=O)NO)C(=O)c1ccc(Nc2nc3ccccc3s2)cc1
CC(C)CC(=O)N(c1ccc(cc1)C(=O)N(C)CCCCCCC(=O)NO)c1c(C)cccc1C
CN(CCCCCCC(=O)NO)C(=O)c1ccc(Nc2c(C)cccc2C)c(F)c1
Cc1cccc(C)c1Nc1cccc(c1)C(=O)NCCCCCCC(=O)NO
CN(CCCCCCC(=O)NO)C(=O)c1cccc(Nc2c(C)cccc2C)c1
CC(C)c1cccc(C(C)C)c1Nc1ccc(cc1)C(=O)N(C)CCCCCCC(=O)NO
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)N(c1ccccc1)c1ncccc1C
CN(CCCCCCC(=O)NO)C(=O)c1ccccc1Nc1c(C)cccc1C
CN(CCCCCCC(=O)NO)C(=O)c1ccc(Nc2c(C)cc(C)cc2C)cc1
CN(CCCCCCC(=O)NO)C(=O)c1ccc(Nc2c(C)cccc2Cl)cc1
Cc1cccc(C)c1N(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)c1ncccn1
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)N(c1ccccc1)c1ncccn1
CN(CCCCCC(=O)NO)C(=O)c1ccc(Nc2c(C)cccc2C)cc1
Cc1ccccc1N(c1ccccc1)c1ncc(cn1)C(=O)NCCCCCCC(=O)NO
CN(CCCCCCC(=O)NO)C(=O)c1cnc(Nc2c(C)cc(C)cc2C)nc1
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)N(c1ncccn1)c1c(C)cccc1C
CC(C)c1cccc(C(C)C)c1Nc1ncc(cn1)C(=O)N(C)CCCCCCC(=O)NO
CN(CCCCC(=O)NO)C(=O)c1ccc(Nc2c(C)cccc2C)cc1
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)C(O)(c1ccccc1)c1ccccc1
OCC(c1ccccc1)(c1ccccc1)c1ccc(cc1)C(=O)NCCCCCCC(=O)NO
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)C(O)(c1ccccc1)c1ccncc1
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)N(C(=O)c1ccccc1)c1ccccc1
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)N(C(=O)c1ccccc1)c1ccccc1
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)C(O)(c1ccc(F)cc1)c1ccc(F)cc1
COC(c1ccc(F)cc1)(c1ccc(F)cc1)c1ccc(cc1)C(=O)NCCCCCCC(=O)NO
COC(c1ccccc1)(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)c1cccnc1
COC(c1ccccc1)(c1ccc(cc1)C(=O)N(C)CCCCCCC(=O)NO)c1cccnc1
COC(c1ccccc1)(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)c1ccccn1
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)C(O)(c1ccccn1)c1ccccn1
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)C(O)(c1ccccn1)c1ccccn1
Cc1ccccc1N(c1ncc(cn1)C(=O)NCCCCCCC(=O)NO)c1ccccc1C
c1ccc(cc1)N(c2ccccc2Cl)c3ncc(cn3)C(=O)NCCCCCCC(=O)NO
Cc1cccc(C)c1N(c1ccccc1)c1ncc(cn1)C(=O)NCCCCCCC(=O)NO
Cc1cccc(C)c1Nc1ccc2C(=O)N(CCCCCCC(=O)NO)Cc2c1
COC(c1ccccc1)(c1ccncc1)c1ccc(cc1)C(=O)NCCCCCCC(=O)NO
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)C(O)(c1ccccc1)c1ccncc1
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)C(c1ccccc1)c1ccccc1
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)C(c1ccccc1)c1ccccc1
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)N(C(=O)c1ccccn1)c1ccccc1
CCOC(c1ccccc1)(c1ccccc1)c1ccc(cc1)C(=O)NCCCCCCC(=O)NO
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)C(O)(c1cccc(F)c1)c1cccc(F)c1
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)C(O)(c1cccc(F)c1)c1cccc(F)c1
COC(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)(c1cccc(F)c1)c1cccc(F)c1
CC(O)(c1ccc(F)cc1)c1ccc(cc1)C(=O)NCCCCCCC(=O)NO
CCOC(c1ccccc1)(c1ccccc1)c1ccc(cc1)C(=O)N(C)CCCCCCC(=O)NO
CCOC(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)(c1ccccn1)c1ccccn1
CCOC(c1ccc(cc1)C(=O)N(C)CCCCCCC(=O)NO)(c1ccccn1)c1ccccn1
COC(c1ccc(cc1)C(=O)N(C)CCCCCCC(=O)NO)(c1cccc(F)c1)c1cccc(F)c1
C[C@](O)(c1ccc(F)cc1)c1ccc(cc1)C(=O)NCCCCCCC(=O)NO |r|
C[C@@](O)(c1ccc(F)cc1)c1ccc(cc1)C(=O)NCCCCCCC(=O)NO |r|
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)C(C)(O)c1ccc(F)cc1
COC(C)(c1ccc(F)cc1)c1ccc(cc1)C(=O)NCCCCCCC(=O)NO
COC(C)(c1ccc(F)cc1)c1ccc(cc1)C(=O)N(C)CCCCCCC(=O)NO
CC(O)(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)c1ccccn1
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)C(C)(O)c1ccccn1
COC(C)(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)c1ccccn1
COC(C)(c1ccc(cc1)C(=O)N(C)CCCCCCC(=O)NO)c1ccccn1
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)C(O)(c1ccccc1F)c1ccccc1F
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)C(O)(c1ccccc1F)c1ccccc1F
COC(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)(c1ccccc1F)c1ccccc1F
COC(c1ccc(cc1)C(=O)N(C)CCCCCCC(=O)NO)(c1ccccc1F)c1ccccc1F
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)C(O)(c1ccc(F)cc1F)c1ccc(F)cc1F
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)C(O)(c1ccc(F)cc1F)c1ccc(F)cc1F
COC(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)(c1ccc(F)cc1F)c1ccc(F)cc1F
COC(c1ccc(cc1)C(=O)N(C)CCCCCCC(=O)NO)(c1ccc(F)cc1F)c1ccc(F)cc1F
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)C(O)(c1cc(F)cc(F)c1)c1cc(F)cc(F)c1
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)C(O)(c1cc(F)cc(F)c1)c1cc(F)cc(F)c1
COC(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)(c1cc(F)cc(F)c1)c1cc(F)cc(F)c1
COC(c1ccc(cc1)C(=O)N(C)CCCCCCC(=O)NO)(c1cc(F)cc(F)c1)c1cc(F)cc(F)c1
Cc1cc(F)ccc1C(O)(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)c1ccc(F)cc1C
COC(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)(c1ccc(F)cc1C)c1ccc(F)cc1C
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)C(O)(c1ccc(F)cc1)c1ccccn1
CN(CCCCCCC(=O)NO)C(=O)c1ccc(cc1)C(O)(c1ccc(F)cc1)c1ccccn1
COC(c1ccc(F)cc1)(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)c1ccccn1
COC(c1ccc(F)cc1)(c1ccc(cc1)C(=O)N(C)CCCCCCC(=O)NO)c1ccccn1
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)C(O)(c1nccs1)c1nccs1
ONC(=O)CCCCCCNC(=O)c1cccc(c1)C(O)(c1ccc(F)cc1)c1ccc(F)cc1
CN(CCCCCCC(=O)NO)C(=O)c1cccc(c1)C(O)(c1ccc(F)cc1)c1ccc(F)cc1
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)C(O)(c1ccc(F)cc1)C(F)(F)F
COC(c1ccc(F)cc1)(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)C(F)(F)F
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)C1(CCCO1)c1ccc(F)cc1
OCCN(c1ccccc1)c1ncc(cn1)C(=O)NCCCCCCC(=O)NO
ONC(=O)CCCCCCNC(=O)c1cccc(c1)C(O)(c1ccccn1)c1ccccn1
COC(c1cccc(c1)C(=O)NCCCCCCC(=O)NO)(c1ccccn1)c1ccccn1
CN(C)C(=O)c1ccc(cc1)C(O)(c1ccccc1)c1ccc(cc1)C(=O)NCCCCCCC(=O)NO
CN(C)C(=O)c1cccc(c1)C(O)(c1ccccc1)c1ccc(cc1)C(=O)NCCCCCCC(=O)NO
ONC(=O)CCCCCCNC(=O)c1cnc(nc1)N(c1ccc(F)cc1)c1ccc(F)cc1
NC(=O)CCCCCCNC(=O)c1cnc(nc1)N(c1ccccc1)c1ccccc1
COC(c1ccccc1)(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)c1ccc(cc1)C(=O)N(C)C
COC(c1ccccc1)(c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)c1cccc(c1)C(=O)N(C)C
OC(=O)CCCCCCNC(=O)c1cnc(nc1)N(c1ccccc1)c1ccccc1
ONC(=O)CCCCCCNC(=O)c1ccc(cc1)C1(OC(=O)c2ccccc12)c1ccccc1
ONC(=O)CCCCCCNC(=O)c1cnc(NC(c2ccc(F)cc2)c2ccc(F)cc2)nc1
ONC(=O)CCCCCCNC(=O)c1cnc(nc1)N1CCCc2ccccc12
ONC(=O)CCCCCCNC(=O)c1cnc(nc1)N1CCc2ccccc2C1
OCCN(CC(c1ccc(F)cc1)c1ccc(F)cc1)c1ncc(cn1)C(=O)NCCCCCCC(=O)NO
OCCN(CCc1c[nH]c2ccccc12)c1ncc(cn1)C(=O)NCCCCCCC(=O)NO
ONC(=O)CCCCCCNC(=O)c1cnc(nc1)N1CCOCC1
C[C@H]1CN(C[C@@H](C)O1)c1ncc(cn1)C(=O)NCCCCCCC(=O)NO |r|
ONC(=O)CCCCCCNC(=O)c1cnc(nc1)N1CCNCC1
ONC(=O)CCCCCCNC(=O)c1cnc(nc1)N1CCN(Cc2ccccc2)CC1
OCCN1CCN(CC1)c1ncc(cn1)C(=O)NCCCCCCC(=O)NO
COc1cc2CCN(Cc2cc1OC)c1ncc(cn1)C(=O)NCCCCCCC(=O)NO
ONC(=O)CCCCCCNC(=O)c1cnc(nc1)N1CCn2c(C1)nnc2C(F)(F)F
ONC(=O)CCCCCCNC(=O)c1cnc(nc1)N1CCN(CC1)c1ccccc1
COc1ccc(cc1)N1CCN(CC1)c1ncc(cn1)C(=O)NCCCCCCC(=O)NO
COCCN1CCN(CC1)c1ncc(cn1)C(=O)NCCCCCCC(=O)NO
ONC(=O)CCCCCCNC(=O)c1cnc(nc1)N1CCN(CC1)c1nccc(n1)C(F)(F)F
OCC1CN(CCO1)c1ncc(cn1)C(=O)NCCCCCCC(=O)NO
ONC(=O)CCCCCCNC(=O)c1cnc(nc1)N1CCC[C@@H](O)C1 |r|
NC(=O)C1CCN(CC1)c1ncc(cn1)C(=O)NCCCCCCC(=O)NO
ONC(=O)CCCCCCNC(=O)c1cnc(nc1)N1CCC(O)(CC1)c1ccccc1
ONC(=O)CCCCCCNC(=O)c1cnc(nc1)N1CCC(O)(CC1)c1ccc(Cl)cc1
CN(C)[C@@H]1CCN(C1)c1ncc(cn1)C(=O)NCCCCCCC(=O)NO |r|
OC[C@@H]1CCCN1c1ncc(cn1)C(=O)NCCCCCCC(=O)NO |r|
CN1CCN(C(C1)c1ccccc1)c1ncc(cn1)C(=O)NCCCCCCC(=O)NO
ONC(=O)CCCCCCNC(=O)c1cnc(nc1)N1CCN(CC1)c1ccc(F)cc1
ONC(=O)CCCCCCNC(=O)c1cnc(nc1)N1CCCNCC1
ONC(=O)CCCCCCNC(=O)c1cnc(nc1)N1CCCCC1
CN1CCN(CC1)c1ncc(cn1)C(=O)NCCCCCCC(=O)NO
ONC(=O)c1ccc(NC(=O)c2[nH]c(cc2-c2ccc(O)cc2)-c2ccoc2)cc1
ONC(=O)c1ccc(NC(=O)c2[nH]c(cc2-c2ccc(O)cc2)-c2ccccc2)cc1
ONC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccc(F)cc2)-c2cccs2)nc1
ONC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccc(F)cc2)-c2ccoc2)cc1
ONC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccc(O)cc2)-c2cccs2)cc1
ONC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccsc2)-c2ccc(O)cc2)cc1
ONC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccoc2)-c2ccc(O)cc2)cc1
COc1ccc(cc1)-c1cc([nH]c1C(=O)NCc1ccc(cc1)C(=O)Nc1ccccc1N)-c1ccccc1
COc1ccc(cc1)-c1cc([nH]c1C(=O)NCc1ccc(cc1)C(=O)Nc1ccccc1S)-c1ccccc1
COc1ccc(cc1)-c1cc([nH]c1C(=O)NCc1ccc(cc1)C(=O)Nc1ccccn1)-c1ccccc1
COc1ccc(cc1)-c1cc([nH]c1C(=O)NCc1ccc(cc1)C(=O)Nc1ncccn1)-c1ccccc1
COc1ccc(cc1)-c1cc(-c2ccoc2)c([nH]1)C(=O)NCc1ccc(cc1)C(=O)NO
COc1ccc(cc1)-c1cc(-c2ccsc2)c([nH]1)C(=O)NCc1ccc(cc1)C(=O)NO
Nc1ccccc1NC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccsc2)-c2ccc(O)cc2)cc1
Nc1ccccc1NC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccc(O)cc2)-c2ccoc2)cc1
Nc1ccccc1NC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccccc2)-c2ccc(O)cc2)cc1
Nc1ccccc1NC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccc(O)cc2)-c2ccsc2)cc1
Nc1ccccc1NC(=O)c1ccc(CNC(=O)c2[nH]c(cc2-c2ccoc2)-c2ccc(O)cc2)cc1
ONC(=O)CCCCCn1c2ccccc2c2ccccc12
ONC(=O)CCCCCn1c2CCCCc2c2ccccc12
CN1CCc2c(C1)n(CCCCCC(=O)NO)c1ccccc21
CN1CCc2c(C1)c1ccccc1n2CCCCCC(=O)NO
ONC(=O)c1ccc(Cn2c3ccccc3c3ccccc23)cc1
CN1CCc2c(c3ccccc3n2Cc4ccc(cc4)C(=O)NO)C1
ONC(=O)CCn1c2ccccc2c2ccccc12
ONC(=O)CCCCn1c2ccccc2c2ccccc12
ONC(=O)CCCCCCn1c2ccccc2c2ccccc12
ONC(=O)Cc1ccc(Cn2c3ccccc3c3ccccc23)cc1
ONC(=O)c1ccc(CCn2c3ccccc3c3ccccc23)cc1
ONC(=O)n1c2ccccc2c2ccccc12
[#8]-[#7]-[#6](=O)-[#6]-[#6]-[#6]-[#6]\[#6]=[#6](\c1ccccn1)-c1ccccn1
ONC(=O)CCCCCCN(c1ccccn1)c1ccccn1
ONC(=O)CCCCCCN(c1ccccn1)c1ccc2ccccc2n1
[#8]-[#7]-[#6](=O)-[#6]-[#6]-[#6]-[#6]-[#6]\[#6]=[#6](\c1ccccn1)-c1ccccn1
ONC(=O)CCCCCCN(c1ccccn1)c1cc(ccn1)-c1ccccc1
Cc1ccc(nc1)N(CCCCCCC(=O)NO)c1ccccn1
ONC(=O)CCCCCCN(c1ccccn1)c1ccc(OCc2ccccc2)cn1
COc1ccc(nc1)N(CCCCCCC(=O)NO)c1ccccn1
ONC(=O)CCCCCCN(c1ccccn1)c1cc2ccccc2cn1
ONC(=O)CCCCCCN(c1ccccn1)c1cc(OCc2ccccc2)ccn1
Oc1cccn(Cc2ccccc2)c1=S
Oc1cccn(Cc2ccc(cc2)-c2ccccc2)c1=S
Oc1cccn(Cc2ccc(cc2)-c2ccc(cc2)C#N)c1=S
Oc1cccn(Cc2ccc(cc2)-c2ccccc2[N+]#[C-])c1=S
Cc1ccc(cc1)-c1ccc(Cn2cccc(O)c2=S)cc1
Cc1cccc(c1)-c1ccc(Cn2cccc(O)c2=S)cc1
Cc1ccccc1-c1ccc(Cn2cccc(O)c2=S)cc1
CN(C)c1ccc(cn1)-c1ccc(Cn2cccc(O)c2=S)cc1
Oc1cccn(Cc2ccc(cc2)-c2ccncc2)c1=S
CN(C)c1ccc(cc1)-n1cc(Cn2cccc(O)c2=S)nn1
Oc1ccc[nH]c1=S
ONC(=O)c1cnc(Nc2ccc(Cl)c(Cl)c2)nc1
ONC(=O)c1cnc(Nc2ccc(F)cc2)nc1
ONC(=O)c1cnc(Nc2ccccc2)nc1
Cc1ccc(Nc2ncc(cn2)C(=O)NO)cc1
COc1ccc(Nc2ncc(cn2)C(=O)NO)cc1
ONC(=O)c1cnc(Nc2ccc(Cl)cc2)nc1
ONC(=O)c1cnc(Nc2ccccc2Cl)nc1
ONC(=O)c1cnc(Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)nc1
CN(c1ccc(Cl)c(Cl)c1)c1ncc(cn1)C(=O)NO
ONC(=O)c1cnc(Nc2c(F)c(F)cc(F)c2F)nc1
ONC(=O)c1cnc(Nc2cccc(Cl)c2)nc1
ONC(=O)c1cnc(Nc2cc(F)cc(F)c2)nc1
ONC(=O)c1cnc(Nc2ccc(c(c2)C(F)(F)F)[N+]([O-])=O)nc1
ONC(=O)c1cnc(Nc2cc(Cl)ccc2Cl)nc1
ONC(=O)c1cnc(Nc2c(Cl)cccc2Cl)nc1
COc1cc(Nc2ncc(cn2)C(=O)NO)cc(c1)C(F)(F)F
ONC(=O)c1cnc(Nc2cccc(c2)C(F)(F)F)nc1
Cc1cc(C)cc(Nc2ncc(cn2)C(=O)NO)c1
COc1cc(Nc2ncc(cn2)C(=O)NO)cc(OC)c1
Cc1cc(F)cc(Nc2ncc(cn2)C(=O)NO)c1
ONC(=O)c1cnc(Nc2cc(Cl)cc(c2)C(F)(F)F)nc1
ONC(=O)c1cnc(Nc2cc(F)cc(c2)C(F)(F)F)nc1
ONC(=O)c1cnc(Nc2cc(Cl)cc(OC(F)(F)F)c2)nc1
ONC(=O)c1cnc(Nc2cccc(c2)-c2ccccc2)nc1
ONC(=O)c1cnc(Nc2cccc(c2)N2CCOCC2)nc1
ONC(=O)c1cnc(Nc2cccc(c2)-c2ccncc2)nc1
Cc1cc(Nc2ncc(cn2)C(=O)NO)ccn1
CC(Nc1ncc(cn1)C(=O)NO)c1ccccc1
ONC(=O)c1cnc(NCc2ccccc2Cl)nc1
ONC(=O)c1cnc(NCc2cccc(Cl)c2)nc1
ONC(=O)c1cnc(NCc2ccccc2)nc1
ONC(=O)c1cnc(NCc2ccc(Cl)cc2)nc1
ONC(=O)c1cnc(NCc2ccc(cc2)C(F)(F)F)nc1
ONC(=O)c1cnc(NCc2ccccc2C(F)(F)F)nc1
ONC(=O)c1cnc(NCCc2ccccc2Cl)nc1
ONC(=O)c1cnc(NCc2cccc(c2)C(F)(F)F)nc1
ONC(=O)c1cnc(NCCc2ccccc2)nc1
ONC(=O)c1cnc(NCCc2cccc(Cl)c2)nc1
ONC(=O)c1cnc(NCCc2c[nH]c3ccccc23)nc1
ONC(=O)c1cnc(NCCc2ccc(Cl)cc2)nc1
COc1ccccc1CNc1ncc(cn1)C(=O)NO
ONC(=O)c1cnc(NCc2ccc3OCOc3c2)nc1
ONC(=O)c1cnc(NCc2ccccc2OC(F)(F)F)nc1
ONC(=O)c1cnc(NCc2c(Cl)cccc2Cl)nc1
COc1cc(F)ccc1CNc1ncc(cn1)C(=O)NO
CC(C)(Nc1ncc(cn1)C(=O)NO)c1ccccc1
OCc1cccc(CO)c1CNc1ncc(cn1)C(=O)NO
Cc1cc(Cl)ccc1CNc1ncc(cn1)C(=O)NO
ONC(=O)c1cnc(NCc2ccc(F)c(Cl)c2)nc1
Cc1cccc(C)c1CNc1ncc(cn1)C(=O)NO
ONC(=O)c1cnc(NCc2ccccc2-c2ccccc2)nc1
ONC(=O)c1cnc(NCc2ccc(F)cc2C(F)(F)F)nc1
ONC(=O)c1cnc(NC23CC4CC(CC(C4)C2)C3)nc1 |TLB:8:9:12:15.16.14,16:15:18:12.11.10,16:11:18:15.17.14,THB:17:15:12:18.9.10,17:9:12:15.16.14|
ONC(=O)c1cnc(NCCc2ccccc2-c2ccccc2)nc1
ONC(=O)c1cnc(NC(c2ccccc2)c2ccccc2)nc1
C[C@H](Nc1ncc(cn1)C(=O)NO)c1ccccc1 |r|
C[C@@H](Nc1ncc(cn1)C(=O)NO)c1ccccc1 |r|
ONC(=O)c1cnc(NCCc2c(Cl)cccc2Cl)nc1
CC(C)(Nc1ncc(cn1)C(=O)NO)c1ccc(F)cc1
ONC(=O)c1cnc(NCc2ccncc2)nc1
CC(C)(Nc1ncc(cn1)C(=O)NO)c1ccc(F)cc1F
CC(C)(Nc1ncc(cn1)C(=O)NO)c1ccccc1F
Cc1cc(F)ccc1C(C)(C)Nc1ncc(cn1)C(=O)NO
ONC(=O)c1cnc(NC2(CC2)c2ccccc2)nc1
CC(C)(Nc1ncc(cn1)C(=O)NO)c1ccc(cc1)C(F)(F)F
CC(C)(Nc1ncc(cn1)C(=O)NO)c1cccc(F)c1
CC(C)(Nc1ncc(cn1)C(=O)NO)c1ccc(F)c(F)c1
ONC(=O)c1cnc(NCc2cnccn2)nc1
Cc1cc(ccc1F)C(C)(C)Nc1ncc(cn1)C(=O)NO
CC(Nc1ncc(cn1)C(=O)NO)(c1ccccc1)c1ccccc1
CC(C)(Nc1ncc(cn1)C(=O)NO)c1ccc(Cl)c(Cl)c1
ONC(=O)c1cnc(NC2(CC2)c2ccc(F)cc2)nc1
ONC(=O)c1cnc(NC2(CC2)c2ccccc2F)nc1
CC(C)(Nc1ncc(cn1)C(=O)NO)c1ccc(Cl)cc1F
ONC(=O)c1cnc(NC2(CCCCC2)c2ccccc2)nc1
CC(Nc1ncc(cn1)C(=O)NO)c1ccncc1
CC(C)(Nc1ncc(cn1)C(=O)NO)c1ccc(cc1F)C(F)(F)F
ONC(=O)c1cnc(NC2(CC2)c2cccc(F)c2)nc1
ONC(=O)c1cnc(NC2(CCCC2)c2ccccc2)nc1
ONC(=O)c1cnc(NC(c2ccc(F)cc2)c2ccc(F)cc2)nc1
ONC(=O)c1cnc(NC2(CC2)c2ccccc2Cl)nc1
ONC(=O)c1cnc(NC2(CC2)c2ccccc2C(F)(F)F)nc1
CC(C)(Nc1ncc(cn1)C(=O)NO)c1cc(cc(c1)C(F)(F)F)C(F)(F)F
Cc1ccc(cc1)C1(CC1)Nc1ncc(cn1)C(=O)NO
ONC(=O)c1cnc(NC2(CC2)c2cccc(Cl)c2)nc1
ONC(=O)c1cnc(NC2(CCOCC2)c2ccccc2)nc1
CC(Nc1ncc(cn1)C(=O)NO)(c1ccc(F)cc1)c1ccc(F)cc1
OCc1ccc(cc1)C1(CC1)Nc1ncc(cn1)C(=O)NO
ONC(=O)c1cnc(NC2(CC2)c2cccs2)nc1
ONC(=O)c1cnc(NC2(CC2)c2ccco2)nc1
ONC(=O)c1cnc(NC2(CCCCC2)c2ccc(F)cc2)nc1
ONC(=O)c1cnc(NC2(CCCCC2)c2cccc(F)c2)nc1
ONC(=O)c1cnc(NC2(CC2)c2cc3ccccc3s2)nc1
ONC(=O)c1cnc(NC2CCCCC2)nc1
ONC(=O)c1cnc(NC2CCOCC2)nc1
ONC(=O)c1cnc(NCc2cccs2)nc1
ONC(=O)c1cnc(NCc2cccnc2)nc1
ONC(=O)c1cnc(NCc2ccc(cc2)-c2ccccc2)nc1
ONC(=O)c1cnc(NCc2ccccn2)nc1
ONC(=O)c1cnc(NC2(Cc3ccccc3)CC2)nc1
CC1(CCCCC1)Nc1ncc(cn1)C(=O)NO
ONC(=O)c1cnc(NC2c3ccccc3-c3ccccc23)nc1
COc1cccc(c1)C1(CC1)Nc1ncc(cn1)C(=O)NO
ONC(=O)c1cnc(NC2(CC2)c2cccc(c2)C(F)(F)F)nc1
COc1ccc(cc1)C1(CCCCC1)Nc1ncc(cn1)C(=O)NO
ONC(=O)c1cnc(NC2(CC2)c2ccc(F)cc2F)nc1
ONC(=O)c1cnc(NC2(CC2)c2c(F)cccc2F)nc1
ONC(=O)c1cnc(NC2(CC2)c2cccc(OC(F)(F)F)c2)nc1
ONC(=O)c1cnc(NC2(CC2)c2cc(ccc2F)C(F)(F)F)nc1
Cc1ccccc1C1(CC1)Nc1ncc(cn1)C(=O)NO
ONC(=O)c1cnc(NC2(CC2)c2ccc3OCOc3c2)nc1
COc1cc(OC)cc(c1)C1(CC1)Nc1ncc(cn1)C(=O)NO
ONC(=O)c1cnc(NC2(CCC2)c2ccccc2)nc1
ONC(=O)c1cnc(NC2(CC2)c2ccc(F)c(Cl)c2)nc1
ONC(=O)c1cnc(NC2(CC2)c2cc(F)cc(F)c2)nc1
COc1ccccc1C1(CC1)Nc1ncc(cn1)C(=O)NO
Cc1cccc(c1)C1(CC1)Nc1ncc(cn1)C(=O)NO
ONC(=O)c1cnc(NC2(CC2)c2ccc(cc2)C(F)(F)F)nc1
ONC(=O)c1cnc(NC2(CC2)c2ccc(Cl)cc2)nc1
ONC(=O)c1cnc(NC2(CC2)c2ccc(c(F)c2)C(F)(F)F)nc1
COc1ccc(cc1OC)C1(CC1)Nc1ncc(cn1)C(=O)NO
COc1ccc(Cl)cc1C1(CC1)Nc1ncc(cn1)C(=O)NO
ONC(=O)c1cnc(NC2(CC2)c2ccc(F)c(F)c2)nc1
ONC(=O)c1cnc(NC2(CC2)c2ccc(Cl)c(Cl)c2)nc1
Cc1cc(ccc1F)C1(CC1)Nc1ncc(cn1)C(=O)NO
ONC(=O)c1cnc(NC2(CC2)c2cccc(F)c2F)nc1
ONC(=O)c1cnc(NC2(CC2)c2ccc(F)cc2Cl)nc1
ONC(=O)c1cnc(NC2(CC2)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)nc1
ONC(=O)c1cnc(NC2(CC2)c2cc(Cl)cc(Cl)c2)nc1
Cc1cc(cc(c1)C1(CC1)Nc1ncc(cn1)C(=O)NO)C(F)(F)F
ONC(=O)c1cnc(NC2(CCCC2)c2ccc(F)cc2)nc1
ONC(=O)c1cnc(NC2(CCOCC2)c2cccc(F)c2)nc1
ONC(=O)c1cnc(NC2(CCOCC2)c2ccc(F)cc2)nc1
ONC(=O)c1cnc(NC2(CCCC2)c2cccc(F)c2)nc1
COc1ccc(cc1)C1(CCCC1)Nc1ncc(cn1)C(=O)NO
ONC(=O)c1cnc(NC2(CCCC2)c2cccc(Cl)c2)nc1
ONC(=O)c1cnc(NC2(CCCCC2)c2cccs2)nc1
ONC(=O)c1cnc(NC2(CCOCC2)c2cc(F)cc(F)c2)nc1
CCN(CC)CCSc1ccc(\C=C\C(=O)NO)cc1NCCCc1ccccc1
CCCCCNc1cc(\C=C\C(=O)NO)ccc1SCCN(CC)CC
CCCNc1cc(\C=C\C(=O)NO)ccc1SCCN(CC)CC
CCN(CC)CCSc1ccc(\C=C\C(=O)NO)cc1NC(C)=O
CCN(CC)CCSc1ccc(\C=C\C(=O)NO)cc1[N+]([O-])=O
CCN(CC)CCSc1ccc(\C=C\C(=O)NO)cc1NCc1ccccc1
CCN(CC)CCSc1ccc(\C=C\C(=O)NO)cc1NCC=C
CCN(CC)CCSc1ccc(\C=C\C(=O)NO)cc1NC
CCN(CC)CCSc1ccc(\C=C\C(=O)NO)cc1N
CCCCCNC(=O)Nc1cc(\C=C\C(=O)NO)ccc1SCCN(CC)CC
CCN(CC)CCSc1ccc(\C=C\C(=O)NO)cc1NS(=O)(=O)c1ccc(C)cc1
CCN(CC)CCSc1ccc(\C=C\C(=O)NO)cc1NCCCC=C
CCN(CC)CCSc1ccc(\C=C\C(=O)NO)cc1NC(=O)C(Cl)Cl
ONC(=O)CCCCC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1cccc2cccnc12 |r|
CC(=O)SCCCCC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1cccc2cccnc12 |r|
COCCOCC(=O)SCCCCC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1cccc2cccnc12 |r|
OCCSSCCCCC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1cccc2cccnc12 |r|
O=C(NC(CCCCCSSCCCCC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1cccc2cccnc12)C(=O)Nc1cccc2cccnc12)OCc1ccccc1 |r|
CN(C)C(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CNC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CNC(=O)Cc1ccc(cc1)-c1noc(n1)C(F)(F)F
CN(C)C(=O)Cc1ccc(cc1)-c1noc(n1)C(F)(F)F
CC(C)NC(=O)Cc1ccc(cc1)-c1noc(n1)C(F)(F)F
CCCCNC(=O)Cc1ccc(cc1)-c1noc(n1)C(F)(F)F
COCCNC(=O)Cc1ccc(cc1)-c1noc(n1)C(F)(F)F
CCOC(=O)CNC(=O)Cc1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CC(=O)N2CCOCC2)cc1
CN1CCN(CC1)C(=O)Cc1ccc(cc1)-c1noc(n1)C(F)(F)F
CON(C)C(=O)Cc1ccc(cc1)-c1noc(n1)C(F)(F)F
CCNC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
OCCNC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CCN(C)C(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CN(CCO)C(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
COCCNC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
COCCN(C)C(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CC(C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
COCCCNC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
FCCNC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)N1CCCC1
CC(C)N(C)C(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)NC1CCC1
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)NCC1CC1
CC(C)CNC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
C[C@H](CO)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)NC1CCCC1
CCC(CC)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CN(C)CCNC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)N1CCOCC1
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)N1CCCCC1
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)NC1CCCCC1
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)Nc1ccccc1
CN1CCN(CC1)C(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CN(C)CCN(C)C(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CN1CCC(CC1)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CN(C)C1CCN(CC1)C(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)NCCCn1ccnc1
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)N1CCN(CC1)c1ccccc1
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)N1CCC(Cc2ccccc2)CC1
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)NCc1ccc(CN2CCOCC2)cc1
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)NCCc1ccccc1
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)NCc1ccccc1
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)Nc1ccncc1
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)Nc1cccnc1
CN1CCC(CNC(=O)c2ccc(cc2)-c2noc(n2)C(F)(F)F)CC1
C[C@@H](CO)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
CC(CNC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F)N(C)C
CN(C)C(=O)CNC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CC(CN(C)C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
OC1CCN(C1)C(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CC(C)(C)OC(=O)N1CCN(CC1)C(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CCC(CO)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)NC1CCOCC1
CC(C)CC(CO)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CC(C)(C)OC(=O)N1CCC(CC1)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CC(C)(C)OC(=O)NC1CCCCC1NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
OC1CCCCC1NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CC(C)(C)OC(=O)N1CCCC(C1)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CNC(=O)CNC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CC(=O)N1CCC(CC1)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CN1C(C)(C)CC(CC1(C)C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CC(C)(C)OC(=O)N1CCC(C1)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
COc1cc(NC(=O)c2ccc(cc2)-c2noc(n2)C(F)(F)F)ccn1
Cc1cc(NC(=O)c2ccc(cc2)-c2noc(n2)C(F)(F)F)cc(C)n1
CC(C)(C)c1cc(NC(=O)c2ccc(cc2)-c2noc(n2)C(F)(F)F)ccn1
Fc1cc(NC(=O)c2ccc(cc2)-c2noc(n2)C(F)(F)F)ccn1
Oc1cc(NC(=O)c2ccc(cc2)-c2noc(n2)C(F)(F)F)ccn1
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)Nc1ccnc(c1)C#N
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)Nc1ccnc(c1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)Nc1ccnc(Cl)c1
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)NC1CCNCC1
NC1CCCCC1NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)NCC1CCCCN1
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)NC1CCCNC1
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)NC1CCNC1
C[C@H](CN(C)C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
C[C@@H](CN(C)C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
CC(C)[C@@H](CN(C)C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
CC(C)[C@H](CN(C)C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
CC(C)C[C@H](CN(C)C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
C[C@H](CN(C)C)NC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
CC(C)[C@H](CN(C)C)NC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
Cc1cc(NC(=O)c2ccc(cc2F)-c2noc(n2)C(F)(F)F)cc(C)n1
CC(CO)NC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F
CN(C)C[C@@H](Cc1ccccc1)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
CN(C)C[C@H](Cc1ccccc1)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
CC(CN(C)C)N(C)C(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
Fc1cc(ccc1C(=O)NC1CCNC1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(cc1)S(=O)(=O)Nc1ccccc1
FC(F)(F)c1nc(no1)-c1ccc(cc1)S(=O)(=O)NCc1ccccc1
CN(C)CCNS(=O)(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CN(C)CCN(C)S(=O)(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(cc1)S(=O)(=O)NCC1CCCCC1
FC(F)(F)c1nc(no1)-c1ccc(cc1)S(=O)(=O)N[C@@H]1CCNC1 |r|
Cc1ccccc1NS(=O)(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(cc1)S(=O)(=O)Nc1ccccc1Cl
Cc1cccc(NS(=O)(=O)c2ccc(cc2)-c2noc(n2)C(F)(F)F)c1
FC(F)(F)c1nc(no1)-c1ccc(cc1)S(=O)(=O)Nc1cccc(Cl)c1
Cc1ccc(NS(=O)(=O)c2ccc(cc2)-c2noc(n2)C(F)(F)F)cc1
Fc1ccc(NS(=O)(=O)c2ccc(cc2)-c2noc(n2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(cc1)S(=O)(=O)Nc1ccc(Cl)cc1
Fc1ccccc1NS(=O)(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CN(C)CCCN(C)S(=O)(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CN(C)CCCNS(=O)(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CN(C)S(=O)(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CN1CCC(CNS(=O)(=O)c2ccc(cc2)-c2noc(n2)C(F)(F)F)C1
OCCCNS(=O)(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CN(C)C[C@H](Cc1ccccc1)NC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
CN(C)C[C@@H](Cc1ccccc1)NC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
CN(C)CC(C)(C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CN(C)CC(C)(C)NC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F
CCN(CC)CC(C)NC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F
CC(CNC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F)N(C)C
CCN(CC)CC(C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
C[C@H](CN(C)C)NC(=O)c1c(F)cc(cc1F)-c1noc(n1)C(F)(F)F |r|
C[C@H](CN(C)C)NC(=O)c1ccc(cc1Cl)-c1noc(n1)C(F)(F)F |r|
CCN(CC)C[C@@H](C)NC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
CCN(CC)C[C@H](C)NC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
C[C@H](CN1CCCC1)NC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
C[C@H](CN1CCCCC1)NC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
C[C@H](CN1CCCC1)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
C[C@H](CN1CCCCC1)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
CCN(CC)C[C@@H](C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
CCN(CC)C[C@H](NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F)C(C)C |r|
CCN(CC)C[C@H](NC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F)C(C)C |r|
CCN(C)C[C@@H](C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
CCCN(CCC)C[C@@H](C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
C[C@H](CN(C)C(C)C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
CCCN(C)C[C@@H](C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
CCCN(CCC)C[C@@H](C)NC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
C[C@H](CN(C)C(C)C)NC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
CCCN(C)C[C@@H](C)NC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
CC(CN(C)C)N(C)C(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F
CCCN(CC)C[C@@H](C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
CCCN(CC)C[C@@H](C)NC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
C[C@H](CN1CCOCC1)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
C[C@H](CN1CCOCC1)NC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
CN1CCCC(C1)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
CCCCN(C)C[C@@H](C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
CCCCN(C)C[C@@H](C)NC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
CCN(C[C@@H](C)NC(=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F)C(C)C |r|
CN1CC[C@H](C1)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
CN1CCC[C@H](C1)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
CCN(CC)CCNC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
C[C@H](CN(C)Cc1ccccc1)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
CNCCNC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)NCCNc1ccccc1
CCCCNNC(=O)c1ccc(Br)cc1
CCCCNNC(=O)c1ccc(cc1)N(C)C
CCCCNNC(=O)c1ccc(cc1)C(C)(C)C
CCCCNNC(=O)c1ccc(C[N-][N+]#N)cc1
CCCNNC(=O)c1ccc(Br)cc1
CCCCCNNC(=O)c1ccc(Br)cc1
CCCCCCNNC(=O)c1ccc(Br)cc1
Cn1c(CCCC(O)=O)nc2cc(ccc12)N(CCCl)CCCl
CC[C@H](C)C(=O)O[C@H]1C[C@@H](C)C=C2C=C[C@H](C)[C@H](CC[C@@H]3C[C@@H](O)CC(=O)O3)[C@@H]12 |c:13,t:11|
C[C@@H]1C[C@H](OC(=O)Nc2ccc(cc2)C#C)[C@@H]2[C@@H](CC[C@@H]3C[C@H](CC(=O)O3)O[Si](C)(C)C(C)(C)C)[C@@H](C)C=CC2=C1 |c:39,42|
C[C@@H]1C[C@H](OC(=O)NCc2ccc(cc2)C#C)[C@@H]2[C@@H](CC[C@@H]3C[C@H](CC(=O)O3)O[Si](C)(C)C(C)(C)C)[C@@H](C)C=CC2=C1 |c:40,43|
C[C@@H]1C[C@H](OC(=O)Nc2ccc(cc2)-c2cn(CCCCCCC(=O)NO)nn2)[C@@H]2[C@@H](CC[C@@H]3C[C@H](CC(=O)O3)O[Si](C)(C)C(C)(C)C)[C@@H](C)C=CC2=C1 |r,c:53,56|
C[C@@H]1C[C@H](OC(=O)NCc2ccc(cc2)-c2cn(CCCCCCC(=O)NO)nn2)[C@@H]2[C@@H](CC[C@@H]3C[C@H](CC(=O)O3)O[Si](C)(C)C(C)(C)C)[C@@H](C)C=CC2=C1 |r,c:54,57|
C[C@@H]1C[C@H](OC(=O)NCCCCCCC(=O)NO)[C@@H]2[C@@H](CC[C@@H]3C[C@H](CC(=O)O3)O[Si](C)(C)C(C)(C)C)[C@@H](C)C=CC2=C1 |r,c:40,43|
Cc1c(c2ccccc2[nH]1)CCNCc3ccc(cc3)/C=C/C(=O)NO
CC(=O)Nc1ccc(cc1)C(=O)Nc1ccccc1N
CC(=O)Nc1ccc(cc1)C(=O)Nc1cc(ccc1N)-c1ccncc1
CC(=O)Nc1ccc(cc1)C(=O)Nc1ccc(F)cc1N
COc1cc2c(Oc3ccc(NC(=O)C4(CC4)C(=O)Nc4ccc(F)cc4)cc3F)ccnc2cc1OCCCC(=O)NO
COc1cc2c(Oc3ccc(NC(=O)C4(CC4)C(=O)Nc4ccc(F)cc4)cc3F)ccnc2cc1OCCCCCC(=O)NO
C[C@H](\C=C\C(=O)NO)\C=C(/C)C(=O)c1ccc(cc1)N(C)C |r|
C[C@@H](\C=C\C(=O)NO)\C=C(/C)C(=O)c1ccc(cc1)N(C)C |r|
ONC(=O)CCCCNC(=O)c1csc(n1)-c1nccs1
Cc1sc(nc1C(=O)NCCCCC(=O)NO)-c1nccs1
CCc1sc(nc1C(=O)NCCCCC(=O)NO)-c1nccs1
CC(C)c1sc(nc1C(=O)NCCCCC(=O)NO)-c1nccs1
CCCCc1sc(nc1C(=O)NCCCCC(=O)NO)-c1nccs1
CC(C)Cc1sc(nc1C(=O)NCCCCC(=O)NO)-c1nccs1
CC(C)Cc1sc(nc1C(=O)NCCCC(=O)NO)-c1nccs1
CC(C)Cc1sc(nc1C(=O)NCCCCCC(=O)NO)-c1nccs1
CC(C)Cc1sc(nc1C(=O)NCCCCCCC(=O)NO)-c1nccs1
CC(C)Cc1sc(nc1C(=O)NCCCCCCCC(=O)NO)-c1nccs1
ONC(=O)CCCCNC(=O)c1nc(sc1C=C)-c1nccs1
CC(C)\C=C\c1sc(nc1C(=O)NCCCCC(=O)NO)-c1nccs1
C\C=C\c1sc(nc1C(=O)NCCCCC(=O)NO)-c1nccs1
CC(C)(O)Cc1sc(nc1C(=O)NCCCCC(=O)NO)-c1nccs1
ONC(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
ONC(=O)CCCCNC(=O)c1nc(sc1C1CCCCC1)-c1nccs1
CC(C)C1CC1c1sc(nc1C(=O)NCCCCC(=O)NO)-c1nccs1
ONC(=O)CCCCNC(=O)c1nc(sc1-c1ccccc1)-c1nccs1
ONC(=O)CCCCNC(=O)c1nc(sc1-c1ccc(F)cc1)-c1nccs1
ONC(=O)CCCCNC(=O)c1nc(sc1-c1ccc(F)cc1Cl)-c1nccs1
ONC(=O)CCCCNC(=O)c1nc(sc1-c1ccccc1Cl)-c1nccs1
ONC(=O)CCCCNC(=O)c1nc(sc1-c1cccc(c1)[N+]([O-])=O)-c1nccs1
ONC(=O)CCCCNC(=O)c1nc(sc1-c1ccc(cc1)[N+]([O-])=O)-c1nccs1
ONC(=O)CCCCNC(=O)c1nc(sc1Cc1ccccc1)-c1nccs1
ONC(=O)CCCCNC(=O)c1nc(sc1\C=C\c1ccccc1)-c1nccs1
ONC(=O)CCCCNC(=O)c1nc(sc1CCOCc1ccccc1)-c1nccs1
ONC(=O)CCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
ONC(=O)CCCCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
ONC(=O)CCCCCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
ONC(=O)CCCCCCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
CC(C)Cc1sc(nc1C(=O)NCCCCC(=O)NO)-c1ncc(C)s1
Cc1csc(n1)-c1nc(C(=O)NCCCCC(=O)NO)c(s1)C1CC1
Cc1cnc(s1)-c1nc(C(=O)NCCCCC(=O)NO)c(s1)C1CC1
Cc1nc(sc1C)-c1nc(C(=O)NCCCCC(=O)NO)c(s1)C1CC1
ONC(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1nc2CCCCc2s1
ONC(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1nc2CCCc2s1
ONC(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1nc2CCCCCc2s1
ONC(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1nc2CCCCCCc2s1
ONC(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1ncc(s1)[N+]([O-])=O
ONC(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1nc(cs1)C1CC1
ONC(=O)CCCCCCNC(=O)c1nc(sc1C1CC1)-c1nc2CCCCc2s1
ONC(=O)c1ccc(CNC(=O)c2nc(sc2C2CC2)-c2nc3CCCCc3s2)cc1
ONC(=O)c1ccc(CNC(=O)c2nc(sc2C2CC2)-c2nccs2)cc1
CC(C)Cc1sc(nc1C(=O)Nc1ccc(cc1)C(=O)NO)-c1nccs1
CC(C)Cc1sc(nc1C(=O)Nc1cccc(\C=C\C(=O)NO)c1)-c1nccs1
CC(C)[C@H](NC(=O)c1csc(n1)-c1cscn1)C(=O)NCCCC(=O)NO |r|
CC(C)Cc1sc(nc1C(=O)NCCCCC(=O)NO)-c1cscn1
CC(C)Cc1sc(nc1C(=O)NCCCCC(=O)NO)-c1csc(C)n1
ONC(=O)CCCCNC(=O)c1csc(n1)-c1cscn1
Cc1nc(cs1)-c1nc(cs1)C(=O)NCCCCC(=O)NO
CC(C)(C)OC(=O)NCc1nc(cs1)-c1nc(cs1)C(=O)NCCCCC(=O)NO
CC(C)(C)OC(=O)NCc1nc(cs1)-c1nc(cs1)C(=O)NCCCCCC(=O)NO
CC(C)(C)OC(=O)NCc1nc(cs1)-c1nc(cs1)C(=O)NCCCCCCC(=O)NO
CC(C)Cc1sc(nc1C(=O)NCCCNC(=O)CS)-c1nccs1
CC(C)Cc1sc(nc1C(=O)NCCCCNC(=O)CS)-c1nccs1
CC(C)Cc1sc(nc1C(=O)NCCCCCNC(=O)CS)-c1nccs1
CC(C)Cc1sc(nc1C(=O)NCCCCCCNC(=O)CS)-c1nccs1
SCC(=O)NCCCNC(=O)c1nc(sc1C=C)-c1nccs1
[#6]\[#6](-[#6])=[#6]\c1sc(nc1-[#6](=O)-[#7]-[#6]-[#6]-[#6]-[#7]-[#6](=O)-[#6]-[#16])-c1nccs1
C\C=C\c1sc(nc1C(=O)NCCCNC(=O)CS)-c1nccs1
CC(C)\C=C\c1sc(nc1C(=O)NCCCNC(=O)CS)-c1nccs1
CC(C)[C@H](NC(=O)c1csc(n1)-c1cscn1)C(=O)OC\C=C\CCS |r|
CC(C)[C@H](NC(=O)c1csc(n1)-c1csc(C)n1)C(=O)OC\C=C\CCS |r|
ONC(=O)CCCCNC(=O)c1csc(n1)-c1cccs1
ONC(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1ncc(s1)-c1ccccc1
ONC(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1nc(cs1)-c1ccccc1
ONC(=O)\C=C\c1cccc(c1)S(=O)(=O)N[C@H](C(=O)Nc1cccc2ccccc12)c1ccccc1
Cc1ccc(NC(=O)[C@@H](NC(=O)c2ccc(cc2)C(=O)NO)c2c[nH]c3ccccc23)cc1 |r|
Cc1ccc(NC(=O)CCCCCC(=O)Nc2ccccc2N)cc1
C[C@H](\C=C(/C)\C=C\C(=O)NO)C(=O)c1ccc(cc1)N(C)C |r|
CC(=O)Nc1ccc(cc1)C(=O)Nc1cc(ccc1N)-c1cccs1
ONC(=O)C(c1ccccc1)c1ccccc1
ONC(=O)c1cnc(NC2(CCN(CC2)C(=O)Nc2ccccc2)c2ccccc2)nc1
ONC(=O)c1cnc(NC2(CCN(CC2)C(=O)OCc2ccccc2)c2ccccc2)nc1
CC(=O)N1CCC(CC1)(Nc1ncc(cn1)C(=O)NO)c1ccccc1
CCON1CCC(CC1)(Nc1ncc(cn1)C(=O)NO)c1ccccc1
CC(C)C1(CCN(CC1)C(C)=O)Nc1ncc(cn1)C(=O)NO
CCON1CCC(CC1)(Nc1ncc(cn1)C(=O)NO)C(C)C
CC(C)C1(CCN(CC1)C(=O)OCc1ccccc1)Nc1ncc(cn1)C(=O)NO
COc1ccc(NC(=O)N2CCC(CC2)(Nc2ncc(cn2)C(=O)NO)c2ccccc2)cc1
ONC(=O)c1cnc(NC2(CCN(CC2)c2ccccc2)c2ccccc2)nc1
ONC(=O)c1cnc(NC2(CCN(CC2)C(=O)Nc2ccccc2F)c2ccccc2)nc1
ONC(=O)c1cnc(NC2(CCN(CC2)C(=O)Nc2ccc(Cl)c(Cl)c2)c2ccccc2)nc1
CN(C(=O)N1CCC(CC1)(Nc1ncc(cn1)C(=O)NO)c1ccccc1)c1ccccc1
ONC(=O)c1cnc(NC2(CCN(CC2)C(=O)Nc2cccc(F)c2)c2ccccc2)nc1
ONC(=O)c1cnc(NC2(CCN(CC2)C(=O)Nc2ccc(F)cc2)c2ccccc2)nc1
Cc1ccc(NC(=O)N2CCC(CC2)(Nc2ncc(cn2)C(=O)NO)c2ccccc2)cc1
CNC(=O)N1CCC(CC1)(Nc1ncc(cn1)C(=O)NO)c1ccccc1
ONC(=O)c1cnc(NC2(CCN(CC2)C(=S)Nc2ccccc2)c2ccccc2)nc1
ONC(=O)c1cnc(NC2(CCN(CC2)S(=O)(=O)c2cccc(F)c2)c2ccccc2)nc1
ONC(=O)c1cnc(NC2(CCN(CC2)S(=O)(=O)c2ccc(Cl)cc2)c2ccccc2)nc1
Cc1ccccc1S(=O)(=O)N1CCC(CC1)(Nc1ncc(cn1)C(=O)NO)c1ccccc1
Cc1ccc(cc1)S(=O)(=O)N1CCC(CC1)(Nc1ncc(cn1)C(=O)NO)c1ccccc1
ONC(=O)c1cnc(NC2(CCN(CC2)S(=O)(=O)c2ccc(cc2)C(F)(F)F)c2ccccc2)nc1
ONC(=O)c1cnc(NC2(CCN(CC2)S(=O)(=O)c2ccccc2)c2ccccc2)nc1
ONC(=O)c1cnc(NC2(CCN(CC2)C(=O)Nc2c(F)cccc2F)c2ccccc2)nc1
CC(C)[C@@H](C(=O)N1CCC(CC1)(Nc1ncc(cn1)C(=O)NO)c1ccccc1)c1ccccc1 |r|
CC(C)[C@H](C(=O)N1CCC(CC1)(Nc1ncc(cn1)C(=O)NO)c1ccccc1)c1ccccc1 |r|
C[C@@H](C(=O)N1CCC(C)(CC1)Nc1ncc(cn1)C(=O)NO)c1ccccc1 |r|
ONC(=O)c1cnc(NC2(CCN(CC2)C(=O)Cc2c[nH]c3ccccc23)c2ccccc2)nc1
CC(C)C[C@H](C(=O)N1CCC(CC1)(Nc1ncc(cn1)C(=O)NO)c1ccccc1)c1ccccc1 |r|
CC(C)C[C@@H](C(=O)N1CCC(CC1)(Nc1ncc(cn1)C(=O)NO)c1ccccc1)c1ccccc1 |r|
ONC(=O)c1cnc(NC2(CCN(CC2)C(=O)Cc2cc3ccccc3[nH]2)c2ccccc2)nc1
Nc1ccc(cc1NC(=O)c1ccc(nc1)N1CCC2(CNC2=O)CC1)-c1cccs1
ONC(=O)c1ccc(cc1)-n1ccc2ccccc12
Cc1cc2ccccc2n1-c1ccc(cc1)C(=O)NO
Cc1cn(-c2ccc(cc2)C(=O)NO)c2ccccc12
Cc1c(CN)c2ccccc2n1-c1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(cc1)-n1cc(Cc2ccccc2)c2ccccc12
CN(C)CCc1cn(-c2ccc(cc2)C(=O)NO)c2ccccc12
CN1CCN(CCc2cn(-c3ccc(cc3)C(=O)NO)c3ccccc23)CC1
ONC(=O)c1ccc(cc1)-n1cnc2cncnc12
ONC(=O)c1ccc(cc1)-n1cnc2ncncc12
ONC(=O)c1ccc(cc1)-c1ccncc1
CN(C)c1ccc(cc1)-c1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(cc1)-n1cccc1
ONC(=O)c1ccc(cc1)-c1ccc[nH]1
ONC(=O)c1ccc(cc1)C(c1ccccc1)c1ccccc1
ONC(=O)c1ccc(cc1)C1CCCC1
COC[C@@H]1CCCC1c1ccc(cc1)C(=O)NO |r|
COC[C@H]1CCCC1c1ccc(cc1)C(=O)NO |r|
CCC(CC)c1ccc(cc1)C(=O)NO
CC(C)C(C(C)C)c1ccc(cc1)C(=O)NO
c1ccc2c(c1)ccn2Cc3ccc(cc3)C(=O)NO
Cc1cc2ccccc2n1Cc1ccc(cc1)C(=O)NO
Cc1cn(Cc2ccc(cc2)C(=O)NO)c2ccccc12
Cc1c(C)c2ccccc2n1Cc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(Cn2cc(Cc3ccccc3)c3ccccc23)cc1
ONC(=O)c1ccc(Cn2cnc3cncnc23)cc1
ONC(=O)c1ccc(Cn2cnc3ncncc23)cc1
CN1CCN(CCc2cn(CC3=CCC(C=C3)C(=O)NO)c3ccccc23)CC1 |c:15,t:11|
CN(C)CCc1cn(c2c1cccc2)Cc3ccc(cc3)C(=O)NO
Cc1c(CN)c2ccccc2n1Cc1ccc(cc1)C(=O)NO
NC(=O)c1ccc(Cn2ccc3ccccc23)cc1
CC(=O)c1ccc(Cn2ccc3ccccc23)cc1
ONC(=O)c1ccc(Cn2cnc3ccccc23)cc1
CS(=O)(=O)NCCc1cn(Cc2ccc(cc2)C(=O)NO)c2ccccc12
Cc1nc2ccccc2n1Cc1ccc(cc1)C(=O)NO
CC(=O)NCCCc1nc2ccccc2n1Cc1ccc(cc1)C(=O)NO
CN(C)CCc1nc2ccccc2n1Cc1ccc(cc1)C(=O)NO
CC(C)c1nc2ccccc2n1Cc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(Cn2cccc2)cc1
ONC(=O)c1ccc(Cn2cccn2)cc1
ONC(=O)c1ccc(Cc2ccncc2)cc1
CN(C)c1ccc(Cc2ccc(cc2)C(=O)NO)cc1
CN(C)c1cccc(Cc2ccc(cc2)C(=O)NO)c1
CCN(CC)Cc1ccc(cc1)C(=O)NO
CC(C)N(Cc1ccc(cc1)C(=O)NO)C(C)C
ONC(=O)c1ccc(CN(c2ccccc2)c2ccccc2)cc1
ONC(=O)c1ccc(CN2CCCC2)cc1
COC[C@@H]1CCCN1Cc1ccc(cc1)C(=O)NO |r|
COC[C@H]1CCCN1Cc1ccc(cc1)C(=O)NO |r|
Sc1cccc2cc(cnc12)C(=O)NCCc1nccs1
CC(=O)c1c(C)c2cnc(Nc3ccc(N(C)CCN(C)c4ncc(C(=O)NO)cn4)cn3)nc2n(C2CCCC2)c1=O
CC(=O)c1c(C)c2cnc(Nc3ccc(N(C)Cc4ccc(/C=C/C(=O)NO)cc4)cn3)nc2n(C2CCCC2)c1=O
CC(=O)c1c(C)c2cnc(Nc3ccc(N(C)CCN(C)c4ccc(C(=O)NO)cn4)cn3)nc2n(C2CCCC2)c1=O
CC(=O)c1c(C)c2cnc(Nc3ccc(OCCN(C)c4ccc(C(=O)NO)cn4)cn3)nc2n(C2CCCC2)c1=O
CC(=O)c1c(C)c2cnc(Nc3ccc(N(C)CCCCCCC(=O)NO)cn3)nc2n(C2CCCC2)c1=O
CC(=O)c1c(C)c2cnc(Nc3ccc(OCCN(C)c4ncc(C(=O)NO)cn4)cn3)nc2n(C2CCCC2)c1=O
CC(C)c1c(c(c(n1CC[C@H](C[C@H](CC(=O)O)O)O)c2ccc(cc2)F)c3ccccc3)C(=O)Nc4ccccc4
CCC(C)C(=O)OC1C[C@@H](C)C=C2C=C[C@H](C)[C@H](CC[C@@H](O)C[C@@H](O)CC(=O)NO)[C@@H]12 |r,c:13,t:11|
CCC(C)(C)C(=O)O[C@H]1C[C@@H](C)C=C2C=C[C@H](C)[C@H](CC[C@@H](O)C[C@@H](O)CC(=O)NO)[C@@H]12 |r,c:14,t:12|
CC(C)c1c(C(=O)Nc2ccccc2)c(c(-c2ccc(F)cc2)n1CC[C@@H](O)C[C@@H](O)CC(=O)NO)-c1ccccc1 |r|
CC(C)c1nc(nc(-c2ccc(F)cc2)c1\C=C\[C@@H](O)C[C@@H](O)CC(=O)NO)N(C)S(C)(=O)=O |r|
COc1ccccc1NC(=O)NCc1ccc(cc1)C(=O)NO
COc1ccccc1NC(=O)N(CCCN(C)C)Cc1ccc(cc1)C(=O)NO
COc1ccccc1NC(=O)N(CCCO)Cc1ccc(cc1)C(=O)NO
COc1ccccc1NC(=O)N(CCc1c[nH]c2ccccc12)Cc1ccc(cc1)C(=O)NO
COc1ccccc1NC(=O)N(CCc1ccc(O)cc1)Cc1ccc(cc1)C(=O)NO
COCCCN(Cc1ccc(cc1)C(=O)NO)C(=O)Nc1ccccc1
COCCN(Cc1ccc(cc1)C(=O)NO)C(=O)Nc1ccccc1
CCCCN(Cc1ccc(cc1)C(=O)NO)C(=O)Nc2ccccc2
ONC(=O)c1ccc(CN(CCc2ccccc2)C(=O)Nc2ccccc2)cc1
CCCCN(C(=O)NCc1ccc(cc1)C(=O)NO)c1ccccc1
COCCCN(C(=O)NCc1ccc(cc1)C(=O)NO)c1ccccc1
CCN(C(=O)NCc1ccc(cc1)C(=O)NO)c1ccccc1
COc1ccc(NC(=O)NCc2ccc(cc2)C(=O)NO)cc1
Cc1ccnc(NC(=O)NCc2ccc(cc2)C(=O)NO)c1
Cc1cc(NC(=O)NCc2ccc(cc2)C(=O)NO)no1
COc1ccccc1N1C(=O)N(Cc2ccc(cc2)C(=O)NO)C(C)(C)C1=O
CC(C)[C@H]1N(Cc2ccc(cc2)C(=O)NO)C(=O)N(C1=O)c1ccccc1 |r|
ONC(=O)c1ccc(CN2C(=O)N[C@@H](Cc3ccccc3)C2=O)cc1 |r|
CCC(CC)(c1ccc(OCC(=O)NO)c(C)c1)c1ccc(OCC(=O)ON)c(C)c1
CCC(CC)(c1ccc(OCC(CO)CO)c(C)c1)c1ccc(OCC(=O)NO)c(C)c1
CCC(CC)(c1ccc(OCC(=O)NO)c(C)c1)c1ccc(OCC(C)(C)O)c(C)c1
CCC(O)(CC)COc1ccc(cc1C)C(CC)(CC)c1ccc(OCC(=O)NO)c(C)c1
CCC(CC)(c1ccc(c(c1)C)OC[C@@H](C(C)(C)C)O)c2ccc(c(c2)C)OCC(=O)NO
CCC(CC)(c1ccc(OCCCC(=O)NO)c(C)c1)c1ccc(OC[C@H](O)C(C)(C)C)c(C)c1 |r|
CCC(CC)(c1ccc(CCC(=O)NO)c(C)c1)c1ccc(OC[C@H](O)C(C)(C)C)c(C)c1 |r|
CCC(CC)(c1cc(C)c(CCC(=O)NO)s1)c1ccc(OCC(O)C(C)(C)C)c(C)c1 |w:23.24|
CCC(CC)(c1ccc(OCC(O)CCC(=O)NO)c(C)c1)c1ccc(OCC(O)C(C)(C)C)c(C)c1 |w:28.29,11.11|
CCC(CC)(c1ccc(OCCCCCC(=O)NO)c(C)c1)c1ccc(OCC(O)C(C)(C)C)c(C)c1 |w:28.29|
CCC(CC)(c1ccc(OCCCCC(=O)NO)c(C)c1)c1ccc(OCC(O)C(C)(C)C)c(C)c1 |w:27.28|
CCC(CC)(c1ccc(OCCCCCCC(=O)NO)c(C)c1)c1ccc(OCC(O)C(C)(C)C)c(C)c1 |w:29.30|
CCC(CC)(c1ccc(OCC(O)C(C)(C)C)c(C)c1)c1ccc(C(=O)NCCCCCC(=O)NO)c(C)c1 |w:11.11|
CCC(CC)(c1ccc(OCC(O)C(C)(C)C)c(C)c1)c1ccc(C(=O)NCCCCCCC(=O)NO)c(C)c1 |w:11.11|
CCC(CC)(c1ccc(OCC(=O)NO)cc1)c1ccc(OCC(O)C(C)(C)C)c(C)c1 |w:23.24|
CCC(CC)(c1ccc(OCCCCCC(=O)NO)cc1)c1ccc(OCC(O)C(C)(C)C)c(C)c1 |w:27.28|
CCC(CC)(c1ccc(OCCCCC(=O)NO)cc1)c1ccc(OCC(O)C(C)(C)C)c(C)c1 |w:26.27|
CCC(CC)(c1ccc(OCCCCC(=O)NO)cc1)c1ccc(OCCC(C)(C)C)c(C)c1
CCC(CC)(c1ccc(cc1)C(=O)NCCCCCC(=O)NO)c1ccc(OCC(O)C(C)(C)C)c(C)c1 |w:29.30|
ONC(=O)c1cnc(NC2(CCCCC2)c2cc(F)cc(F)c2)nc1
ONC(=O)c1cnc(NC2(CCOCC2)c2cc(F)ccc2F)nc1
c1ccc(cc1)C2(CCC(CC2)(F)F)Nc3ncc(cn3)C(=O)NO
ONC(=O)c1cnc(NC2(CCC3(CC2)OCCO3)c2cccc(F)c2)nc1
CC(=O)Nc1cnc(cn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1cnc(NC(=O)c2ccc(cc2)C#N)cn1
CN(Cc1ccncc1)c1ncc(cn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1cnc(NCc2ccccc2)nc1
CN(Cc1ccnc(Cl)c1)c1ncc(cn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1cnc(NCc2ccncc2)nc1
CC(Nc1ncc(cn1)-c1noc(n1)C(F)(F)F)c1ccccc1
Cc1ccc(CNc2ncc(cn2)-c2noc(n2)C(F)(F)F)cn1
CC(Nc1ncc(cn1)-c1noc(n1)C(F)(F)F)c1ccncc1
FC(F)(F)c1nc(no1)-c1cnc(NCc2cccnc2)nc1
Cc1cccc(CNc2ncc(cn2)-c2noc(n2)C(F)(F)F)n1
C[C@@H](Nc1ncc(cn1)-c1noc(n1)C(F)(F)F)c1ccccc1 |r|
CC[C@@H](Nc1ncc(cn1)-c1noc(n1)C(F)(F)F)c1ccccc1 |r|
CN(CCc1ccncc1)c1ncc(cn1)-c1noc(n1)C(F)(F)F
CCC(Nc1ncc(cn1)-c1noc(n1)C(F)(F)F)c1ccncc1
CC(Nc1ncc(cn1)-c1noc(n1)C(F)(F)F)c1ccnc(C)c1
CN(Cc1ccnc(C)c1)c1ncc(cn1)-c1noc(n1)C(F)(F)F
C[C@H](CN(C)C)NC(=O)c1ccc(nc1)-c1noc(n1)C(F)(F)F |r|
CC(CN(C)C)NC(=O)c1ccc(nc1)-c1noc(n1)C(F)(F)F
C[C@@H](CO)NC(=O)c1ccc(nc1)-c1noc(n1)C(F)(F)F |r|
C[C@H](CN(C)Cc1ccccc1)NC(=O)c1ccc(nc1)-c1noc(n1)C(F)(F)F |r|
CCN(CC)C[C@H](NC(=O)c1ccc(nc1)-c1noc(n1)C(F)(F)F)C(C)C |r|
CCN(CC)C[C@@H](C)NC(=O)c1ccc(nc1)-c1noc(n1)C(F)(F)F |r|
C[C@H](CN(C)C)NC(=O)c1ccc(cn1)-c1noc(n1)C(F)(F)F |r|
C[C@H](CN(C)C)NC(=O)c1ncc(cc1Cl)-c1noc(n1)C(F)(F)F |r|
C[C@H](CN(C)C)NC(=O)c1cnc(nc1)-c1noc(n1)C(F)(F)F |r|
FC(F)(F)c1nc(no1)-c1ccc(NCc2ccccc2)cn1
FC(F)(F)c1nc(no1)-c1ccc(NCc2ccccc2)nc1
CC(Nc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1ccccc1
FC(F)(F)c1nc(no1)-c1ccc(NCc2cccnc2)nc1
FC(F)(F)c1nc(no1)-c1ccc(NCc2ccncc2)nc1
Cc1ccc(CNc2ccc(cn2)-c2noc(n2)C(F)(F)F)cn1
FC(F)(F)c1nc(no1)-c1cnc(NCc2ccccc2)c(Cl)c1
C[C@@H](Nc1ncc(cc1Cl)-c1noc(n1)C(F)(F)F)c1ccccc1 |r|
FC(F)(F)c1nc(no1)-c1cnc(NCc2ccncc2)c(Cl)c1
CC(Nc1ncc(cc1Cl)-c1noc(n1)C(F)(F)F)c1ccncc1
FC(F)(F)c1nc(no1)-c1cnc(NCc2cccnc2)c(Cl)c1
Cc1ccc(CNc2ncc(cc2Cl)-c2noc(n2)C(F)(F)F)cn1
FC(F)(F)c1nc(no1)-c1cnc(NCc2ccccn2)c(Cl)c1
FC(F)(F)c1nc(no1)-c1ccc(NCc2ccccc2)nn1
C[C@@H](Nc1cnc(nc1)-c1noc(n1)C(F)(F)F)c1ccccc1 |r|
C[C@H](Nc1cnc(nc1)-c1noc(n1)C(F)(F)F)c1ccccc1 |r|
FC(F)(F)c1nc(no1)-c1ncc(NCc2ccncc2)cn1
C[C@@H](Nc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1ccncc1 |r|
C[C@@H](Nc1ccc(nn1)-c1noc(n1)C(F)(F)F)c1ccncc1 |r|
C[C@H](CN(C)Cc1ccccc1)NC(=O)c1cnc(nc1)-c1noc(n1)C(F)(F)F |r|
Cc1nsc(n1)N(CCCCCCC(=O)NO)c1ccccn1
Cc1nsc(n1)N(CCCCCCC(=O)NO)c1cccnc1
Cc1noc(n1)N(CCCCCCC(=O)NO)c1ccccn1
Cc1noc(n1)N(CCCCCCCC(=O)NO)c1ccccn1
Cn1ccc(n1)N(CCCCCCC(=O)NO)c1ccccn1
Cn1ccc(n1)N(CCCCCCCC(=O)NO)c1ccccn1
ONC(=O)CCCCCCN(c1nncs1)c1ccccn1
ONC(=O)CCCCCCCN(c1nncs1)c1ccccn1
Cc1nnc(s1)N(CCCCCCC(=O)NO)c1ccccn1
Cc1nnc(s1)N(CCCCCCCC(=O)NO)c1ccccn1
ONC(=O)CCCCCCN(c1nc2ccccc2o1)c1ccccn1
ONC(=O)CCCCCCCN(c1nc2ccccc2o1)c1ccccn1
Cn1c(nc2ccccc12)N(CCCCCCC(=O)NO)c1ccccn1
Cn1c(nc2ccccc12)N(CCCCCCCC(=O)NO)c1ccccn1
ONC(=O)CCCCCCN(c1ncns1)c1ccccn1
ONC(=O)CCCCCCCN(c1ncns1)c1ccccn1
Cc1noc(n1)N(CCCCCCC(=O)NO)c1ccc(F)cn1
Cc1noc(n1)N(CCCCCCCC(=O)NO)c1ccc(F)cn1
Cn1c(nc2ccccc12)N(CCCCCCC(=O)NO)c1ccc(F)cn1
Cn1c(nc2ccccc12)N(CCCCCCC(=O)C(=O)NO)c1ccc(F)cn1
Cn1ccc(n1)N(CCCCCCC(=O)NO)c1ccc(F)cn1
Cn1ccc(n1)N(CCCCCCCC(=O)NO)c1ccc(F)cn1
ONC(=O)CCCCCCN(c1nc2ccccc2o1)c1ccc(F)cn1
ONC(=O)CCCCCCCN(c1nc2ccccc2o1)c1ccc(F)cn1
Cn1ccc(n1)N(CCCCCCC(=O)NO)c1cc(ccn1)-c1ccc(F)cc1
Cn1ccc(n1)N(CCCCCCCC(=O)NO)c1cc(ccn1)-c1ccc(F)cc1
ONC(=O)CCCCCCN(c1nc(ns1)C(F)(F)F)c1ccccn1
ONC(=O)CCCCCCCN(c1nc(ns1)C(F)(F)F)c1ccccn1
Cc1nsc(n1)N(CCCCCCC(=O)NO)c1ccc(F)cn1
Cc1nsc(n1)N(CCCCCCCC(=O)NO)c1ccc(F)cn1
Cc1nsc(n1)N(CCCCCCC(=O)NO)c1cc(ccn1)-c1ccc(F)cc1
Cc1nsc(n1)N(CCCCCCCC(=O)NO)c1cc(ccn1)-c1ccc(F)cc1
ONC(=O)CCCCCCN(c1nc(ns1)C(F)(F)F)c1ccc(F)cn1
ONC(=O)CCCCCCCN(c1nc(ns1)C(F)(F)F)c1ccc(F)cn1
ONC(=O)CCCCCCN(c1nc2ccccc2s1)c1ccccn1
ONC(=O)CCCCCCCN(c1nc2ccccc2s1)c1ccccn1
ONC(=O)CCCCCCN(c1nccs1)c1ccccn1
ONC(=O)CCCCCCCN(c1nccs1)c1ccccn1
FC(F)c1nnc(o1)-c1cnc(COc2ccc(F)cc2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cc(Cl)ccc2F)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(Cl)cc2F)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(F)cc2Cl)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(F)cc2F)nc1
FC(F)c1nnc(o1)-c1cnc(COc2ccc(F)cc2)c(F)c1
FC(F)c1nnc(o1)-c1ccc(COc2cc(F)ccc2Cl)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(Cl)cc2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(F)c(F)c2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc3cccnc23)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc3ccccc23)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(F)cc2)nc1
FC(F)c1nnc(o1)-c1ccc(nc1)C(F)(F)Oc1cccc2cccnc12
FC(F)c1nnc(o1)-c1ccc(nc1)C(F)(F)Oc1cccc2ccccc12
FC(F)c1nnc(o1)-c1ccc(nc1)C(F)(F)Oc1ccc(F)cc1
FC(F)c1nnc(o1)-c1cnc(COc2ccc(F)c(F)c2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc(c2)C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc(F)c2C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(F)c(c2)C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc3ccncc3c2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc3cnccc3c2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc3ccncc23)nc1
FC(F)c1nnc(-c2ccc(COc3ccc4cccnc4c3)nc2)o1
FC(F)c1nnc(o1)-c1ccc(COc2cccc3cnccc23)nc1
FC(F)c4nnc(c3ccc(COc2ccc1nccnc1c2)nc3)o4
FC(F)c1nnc(o1)-c1ccc(COc2cccc(c2)C#C)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccccc2C#C)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccccc2C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(CC#N)cc2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccccc2CC#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(F)cc2C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc(C#N)c2F)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(cc2F)C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2c(F)cccc2C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cc(ccc2F)C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cc(F)ccc2C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cc(F)cc(c2)C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(C#N)c(F)c2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc3nccnc23)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc3ncccc3c2)nc1
FC(F)c1nnc(-c2ccc(COc3cccc4ncccc34)nc2)o1
FC(F)c1nnc(o1)-c1cnc(COc2ccc3cccnc3c2)c(F)c1
FC(F)c1nnc(o1)-c1cnc(COc2cccc3cnccc23)c(F)c1
FC(F)c1nnc(o1)-c1cnc(COc2cccc3ccncc23)c(F)c1
FC(F)c1nnc(o1)-c1cnc(COc2ccccc2C#N)c(F)c1
FC(F)c1nnc(o1)-c1cnc(COc2cccc(c2)C#C)c(F)c1
FC(F)c1nnc(o1)-c1cnc(COc2ccc(F)c(F)c2)c(F)c1
FC(F)c1nnc(o1)-c1cnc(COc2cccc3cccnc23)c(F)c1
FC(F)c1nnc(o1)-c1cnc(COc2ccc(F)cc2F)c(F)c1
FC(F)c1nnc(o1)-c1cnc(COc2cccc3ncccc23)c(F)c1
FC(F)c1nnc(o1)-c1cnc(COc2ccc3ncccc3c2)nc1
FC(F)c1nnc(o1)-c1cnc(COc2ccc3ncccc3c2)c(F)c1
FC(F)c1nnc(o1)-c1cnc(COc2ccc3cnccc3c2)nc1
FC(F)c1nnc(o1)-c1cnc(COc2ccc3cnccc3c2)c(F)c1
FC(F)c1nnc(o1)-c1cnc(COc2ccc3ccncc3c2)nc1
FC(F)c1nnc(o1)-c1cnc(COc2ccc3ccncc3c2)c(F)c1
FC(F)c1nnc(o1)-c1cnc(COc2cccc(c2)C#N)nc1
Fc1cc(-c2nnc(C(F)F)o2)cnc1COc1cccc2ncncc12
FC(F)c1nnc(o1)-c1cnc(COc2ccc3cncnc3c2)c(F)c1
FC(F)c1nnc(o1)-c1cnc(COc2ccc3ncncc3c2)c(F)c1
FC(F)c1nnc(o1)-c1cnc(COc2ccc3ccccc3c2)c(F)c1
CNC(=O)c1cccc(OCc2ccc(-c3nnc(C(F)F)o3)cn2)c1
CC(Oc1ccc(F)cc1)c1ccc(cn1)-c1nnc(o1)C(F)F
CC(=C/[C@@H](C)C(=O)c1ccc(N(C)C)cc1)/C=C/C(=O)NO
ONC(=O)\C=C\c1ccccc1
COc1ccc(\C=C\C(=O)NO)cc1
CN(c1ccccc1)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1
CN(CCc1ccccc1)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1
CCCCc1nc2cc(\C=C\C(=O)NO)ccc2n1CCN(C)C
Cn1cc(CCNCc2ccc(\C=C\C(=O)NO)cc2)c2ccccc12
COc1ccc(cc1)Cn2ccc3c2cc(cc3)C(=O)NO
COc1ccc2Sc3ccccc3N(CCCCCC(=O)NO)C(=O)c2c1
COc1ccc2c(c1)C(=O)N(CCCCCC(=O)NO)c1ccccc1S2(=O)=O
ONC(=O)\C=C\c1ccc(CNCC23CC4CC(CC(C4)C2)C3)cc1 |TLB:16:17:21:15.20.14,20:15:22:21.19.18,20:19:22:15.16.14,THB:16:15:21:22.17.18|
CN(Cc1ccc(\C=C\C(=O)NO)cc1)CC12CC3CC(CC(C3)C1)C2 |TLB:19:20:24:18.23.17,23:18:25:24.22.21,23:22:25:18.19.17,THB:19:18:24:25.20.21|
ONC(=O)\C=C\c1cccc(CNC23CC4CC(CC(C4)C2)C3)c1 |TLB:16:17:21:15.20.14,20:15:22:21.19.18,20:19:22:15.16.14,THB:16:15:21:22.17.18|
CN(Cc1ccc2C=C(CCc2c1)C(=O)NO)CC12CC3CC(CC(C3)C1)C2 |c:7,TLB:25:20:27:26.24.23,25:24:27:20.21.19,21:22:26:20.25.19,THB:21:20:26:27.22.23|
ONC(=O)\C=C\c1ccc(CNCC2CCCCC2)cc1
CN(C)Cc1ccc(\C=C\C(=O)NO)cc1
ONC(=O)\C=C\c1ccc(CN(CCF)CC23CC4CC(CC(C4)C2)C3)cc1 |TLB:19:20:24:18.23.17,23:18:25:24.22.21,23:22:25:18.19.17,THB:19:18:24:25.20.21|
ONC(=O)\C=C\c1ccc(CNCC23CC4CC(CC(C4)C2)C3)c(F)c1 |TLB:16:17:21:15.20.14,20:15:22:21.19.18,20:19:22:15.16.14,THB:16:15:21:22.17.18|
CN(Cc1ccc(\C=C\C(=O)NO)cc1F)CC12CC3CC(CC(C3)C1)C2 |TLB:20:21:25:19.24.18,24:19:26:25.23.22,24:23:26:19.20.18,THB:20:19:25:26.21.22|
CCCCN(Cc1ccc(cc1)C(=O)NO)C(=O)Nc1ccccc1OC
ONC(=O)\C=C\c1ccc(CNCC2CCCCC2)c(F)c1
CN(CC1CCCCC1)Cc1ccc(\C=C\C(=O)NO)cc1F
COc1ccccc1NC(=O)NCc1ccc(cc1)C(N)=O
OCc1ccc(NC(=O)NCc2ccc(cc2)C(=O)NO)cc1
ONC(=O)CCCCCC(=O)Nc1ccccc1
CCCCN(Cc1ccc(cc1)C(=O)NO)C(=O)Nc1ncccn1
CCCCN(Cc1ccc(cc1)C(=O)NO)C(=O)Nc1ccc2cn[nH]c2c1
CCCCN(Cc1ccc(cc1)C(=O)NO)C(=O)Nc1cccc(c1)N(C)C
CC(F)(F)C(=O)N[C@@H]1CCCC[C@H]1N1Cc2ccc(-c3nnc(C(F)F)o3)cc2S1(=O)=O
O=C(N[C@@H]1CCCC[C@H]1N1Cc2ccc(-c3nnc(C(F)F)o3)cc2S1(=O)=O)C(F)F
O=C(N[C@@H]1CCCC[C@H]1N1Cc2ccc(-c3nnc(C(F)F)o3)cc2S1(=O)=O)C(F)(F)C(F)(F)F
O=S(=O)(N[C@@H]1CCCC[C@H]1N1Cc2ccc(-c3nnc(C(F)F)o3)cc2S1(=O)=O)C1CC1
O=C(N[C@@H]1CCCC[C@H]1N1C(=O)c2ccc(-c3nnc(C(F)F)o3)cc2S1(=O)=O)C(F)F
CC(F)(F)C(=O)N[C@H]1[C@H](N2Cc3ccc(-c4nnc(C(F)F)o4)cc3S2(=O)=O)CCCC1(F)F
CC(F)(F)C(=O)N[C@@H]1CCCC(F)(F)[C@H]1N1Cc2ccc(-c3nnc(C(F)F)o3)cc2S1(=O)=O
CC(C)(C)OC(=O)N[C@@H]1CCCC[C@H]1N1Cc2ccc(-c3nnc(C(F)F)o3)cc2S1(=O)=O
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1[C@@H]1CCCC[C@H]1O
CS(=O)(=O)N[C@@H]1CCCC[C@H]1N1Cc2ccc(-c3nnc(C(F)F)o3)cc2S1(=O)=O
CC(F)(F)C(=O)N[C@@H]1CCCC[C@H]1N1Cc2c(F)cc(-c3nnc(C(F)F)o3)cc2S1(=O)=O
O=C(N[C@@H]1CCCC[C@H]1N1Cc2c(F)cc(-c3nnc(C(F)F)o3)cc2S1(=O)=O)C(F)F
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1[C@@H]1CCOC[C@H]1O
O=C(N[C@@H]1CCCC[C@H]1N1Cc2ccc(-c3nnc(C(F)F)o3)cc2S1(=O)=O)C(F)(F)F
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1Cc1cccc(Cl)c1
O=C(N[C@H]1[C@H](N2Cc3ccc(-c4nnc(C(F)F)o4)cc3S2(=O)=O)CCCC1(F)F)C(F)F
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1C(c1ccccn1)[C@@H](O)c1ccccn1
Cn1cc(-c2ccccc2N2Cc3ccc(-c4nnc(C(F)F)o4)cc3S2(=O)=O)cn1
Cn1cc([C@H]([C@@H](O)c2ccccc2)N2Cc3ccc(-c4nnc(C(F)F)o4)cc3S2(=O)=O)cn1
Cn1cc([C@@H]([C@@H](O)c2ccccc2)N2Cc3ccc(-c4nnc(C(F)F)o4)cc3S2(=O)=O)cn1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1C(c1ccccn1)[C@H](O)c1ccccn1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1C(c1ccccn1)[C@@H](O)c1ccccn1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1C(c1ccccn1)[C@H](O)c1ccccn1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1[C@@H](c1ccccn1)[C@H](O)c1ccc(F)cn1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1[C@H](c1ccccn1)[C@@H](O)c1ccc(F)cn1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1[C@@H](c1ccccn1)[C@@H](O)c1ccc(F)cn1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1[C@H](c1ccccn1)[C@H](O)c1ccc(F)cn1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1[C@@H](c1ccc(F)cn1)[C@H](O)c1ccc(F)cn1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1[C@H](c1ccc(F)cn1)[C@@H](O)c1ccc(F)cn1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1[C@@H](c1ccc(F)cn1)[C@@H](O)c1ccc(F)cn1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1[C@H](c1ccc(F)cn1)[C@H](O)c1ccc(F)cn1
COC(=O)N[C@@H]1CCCC[C@H]1N1Cc2ccc(-c3nnc(C(F)F)o3)cc2S1(=O)=O
CN(C)C(=O)N[C@@H]1CCCC[C@H]1N1Cc2ccc(-c3nnc(C(F)F)o3)cc2S1(=O)=O
CNC(=O)N[C@@H]1CCCC[C@H]1N1Cc2ccc(-c3nnc(C(F)F)o3)cc2S1(=O)=O
Cn1cc([C@@H](O)[C@H](c2cnn(C)c2)N2Cc3ccc(-c4nnc(C(F)F)o4)cc3S2(=O)=O)cn1
Cn1cc([C@H]([C@@H](O)c2cnn(C)c2)N2Cc3ccc(-c4nnc(C(F)F)o4)cc3S2(=O)=O)cn1
Cn1cc([C@H](O)[C@H](c2cnn(C)c2)N2Cc3ccc(-c4nnc(C(F)F)o4)cc3S2(=O)=O)cn1
Cn1cc([C@@H](O)[C@@H](c2cnn(C)c2)N2Cc3ccc(-c4nnc(C(F)F)o4)cc3S2(=O)=O)cn1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1[C@@H](c1cnccn1)[C@H](O)c1cnccn1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1[C@H](c1cnccn1)[C@@H](O)c1cnccn1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1[C@@H](c1cnccn1)[C@@H](O)c1cnccn1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1[C@H](c1cnccn1)[C@H](O)c1cnccn1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1[C@@H](c1ncccn1)[C@H](O)c1ncccn1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1[C@H](c1ncccn1)[C@@H](O)c1ncccn1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1[C@@H](c1ncccn1)[C@@H](O)c1ncccn1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1[C@H](c1ncccn1)[C@H](O)c1ncccn1
O=C(NC1CC1)N[C@@H]1CCCC[C@H]1N1Cc2ccc(-c3nnc(C(F)F)o3)cc2S1(=O)=O
O=C(NCC1CC1)N[C@@H]1CCCC[C@H]1N1Cc2ccc(-c3nnc(C(F)F)o3)cc2S1(=O)=O
O=C(N[C@@H]1CCCC[C@H]1N1Cc2ccc(-c3nnc(C(F)F)o3)cc2S1(=O)=O)N1CCCC1
O=C(N[C@@H]1CCCC[C@H]1N1Cc2ccc(-c3nnc(C(F)F)o3)cc2S1(=O)=O)C1CC1
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1[C@@H]1CCCC[C@H]1NS(=O)(=O)C(F)(F)F
O=S1(=O)c2cc(-c3nnc(C(F)F)o3)ccc2CN1c1ccccc1-c1ccccn1
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)C1(C)COC1
CC1(C(=O)N2Cc3ccc(-c4nnc(C(F)F)o4)cc3OC[C@@H]2c2ccccc2)CCOCC1
CC1(C(=O)N2Cc3ccc(-c4noc(C(F)(F)F)n4)cc3OC[C@@H]2c2ccccc2)CCOCC1
CC1(C(=O)N2Cc3ccc(-c4noc(C(F)(F)F)n4)cc3OC[C@@H]2c2ccccc2)COC1
O=C(N1Cc2ccc(-c3noc(C(F)(F)F)n3)cc2OC[C@@H]1c1ccccc1)C(F)(F)F
COCC1(C(=O)N2Cc3ccc(-c4noc(C(F)(F)F)n4)cc3OC[C@@H]2c2ccccc2)COC1
CC(C)(C)OC(=O)N1Cc2ccc(-c3noc(C(F)(F)F)n3)cc2OC[C@@H]1c1ccccc1
C[C@@]1(C(=O)N2Cc3ccc(-c4noc(C(F)(F)F)n4)cc3OC[C@@H]2c2ccccc2)CCCOC1
C[C@]1(C(=O)N2Cc3ccc(-c4noc(C(F)(F)F)n4)cc3OC[C@@H]2c2ccccc2)CCCOC1
CC(C)(C)C(=O)N1Cc2c(F)cc(-c3noc(C(F)(F)F)n3)cc2OC[C@@H]1c1ccccc1
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)ccc2CN1C(=O)C1(C)CCOCC1
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)ccc2CN1C(=O)C(C)(C)C
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)C1(C)CCOCC1
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)C(C)(C)C
C[C@H]1COc2cc(-c3nnc(C(F)F)o3)ccc2CN1C(=O)C(C)(C)C
CC(C)(C)C(=O)N1Cc2ccc(-c3nnc(C(F)F)o3)cc2OC[C@@H]1c1ccccc1
CC(C)(C)C(=O)N1Cc2ccc(-c3noc(C(F)(F)F)n3)cc2OC[C@@H]1c1ccccc1
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)C(F)(F)F
CC(=O)N1Cc2c(F)cc(-c3noc(C(F)(F)F)n3)cc2OC[C@@H]1C
COC[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)ccc2CN1C(=O)C1(C)CCOCC1
COC[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)ccc2CN1C(=O)C(C)(C)C
CC1(C(=O)N2CCOc3cc(-c4noc(C(F)(F)F)n4)cc(F)c3C2)CCOCC1
CC(C)(C)C(=O)N1CCOc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2C1
COCC1(C(=O)N2Cc3c(F)cc(-c4noc(C(F)(F)F)n4)cc3OC[C@@H]2C)COC1
COCC1(C(=O)N2Cc3c(F)cc(-c4noc(C(F)(F)F)n4)cc3OC[C@@H]2C)CC1
CC1(C(=O)N2Cc3ccc(-c4noc(C(F)(F)F)n4)cc3OC[C@@H]2C2CC2)CCOCC1
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)ccc2CN1S(C)(=O)=O
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)ccc2CN1S(=O)(=O)C(C)(C)C
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)ccc2CN1C
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)ccc2CN1CC(F)(F)F
CC1(C(=O)N2CCOc3cc(-c4noc(C(F)(F)F)n4)cc(F)c3C2)COC1
CC(C)C(=O)N1Cc2c(F)cc(-c3noc(C(F)(F)F)n3)cc2OC[C@@H]1C
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)C1CCOCC1
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)CO
COCC(=O)N1Cc2c(F)cc(-c3noc(C(F)(F)F)n3)cc2OC[C@@H]1C
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)CCN(C)C
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)CN(C)C
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)c1ccccc1
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)c1cccnc1
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)Cc1ccncc1
CC1(C(=O)N2Cc3ccc(-c4noc(C(F)(F)F)n4)cc3OCC23CC3)COC1
CC(=O)N1CCC(C)(C(=O)N2Cc3c(F)cc(-c4noc(C(F)(F)F)n4)cc3OC[C@@H]2C)CC1
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)c1ccncc1
CC1Oc2cc(-c3noc(C(F)(F)F)n3)ccc2CNC1=O
FC(F)(F)c1nc(-c2ccc3c(c2)OCCN(c2nc4ccccc4[nH]2)C3)no1
CC1(C(=O)N2CCOc3cc(-c4noc(C(F)(F)F)n4)ccc3C2)COC1
CC(C)C(=O)N1CCOc2cc(-c3noc(C(F)(F)F)n3)ccc2C1
O=C(C1CCOCC1)N1CCOc2cc(-c3noc(C(F)(F)F)n3)ccc2C1
CCN1CCC(C)(C(=O)N2Cc3c(F)cc(-c4noc(C(F)(F)F)n4)cc3OC[C@@H]2C)CC1
CC(C)N1CCC(C)(C(=O)N2Cc3c(F)cc(-c4noc(C(F)(F)F)n4)cc3OC[C@@H]2C)CC1
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)C1(C)COC1
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)OC(C)(C)C
COc1ccc(CN2Cc3c(F)cc(-c4noc(C(F)(F)F)n4)cc3OC[C@@H]2C)cc1
CC(C)(C)C(=O)N1Cc2ccc(-c3noc(C(F)(F)F)n3)cc2OCC12CC2
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)Cc1ccccc1
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)cnc2CN1C(=O)C(C)(C)C
C[C@H]1COc2cc(-c3noc(C(F)(F)F)n3)cnc2CN1C(=O)C1(C)CCOCC1
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)C1(C)CCN(C)CC1
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)[C@@H]1CCNC1=O
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)CC(C)(C)O
C[C@]1(C(=O)N2Cc3ccc(-c4noc(C(F)(F)F)n4)cc3OC[C@H]2c2ccccc2)CCOC1
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)CCc1nccs1
CNC(=O)c1ccc(C(=O)N2Cc3c(F)cc(-c4noc(C(F)(F)F)n4)cc3OC[C@H]2C)cc1
C[C@@]1(C(=O)N2Cc3ccc(-c4noc(C(F)(F)F)n4)cc3OC[C@H]2c2ccccc2)CCOC1
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)C1(O)CC1
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)c1cnn2ccccc12
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)C(C)(C)N
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)CS(C)(=O)=O
CC(C)[C@@H]1Oc2cc(-c3noc(C(F)(F)F)n3)ccc2CNC1=O
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)c1ccc(N2CCOCC2)nc1
O=C1COc2cc(-c3noc(C(F)(F)F)n3)ccc2CN1
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)CC#N
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)c1ccoc1
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)C1CS(=O)(=O)C1
Cc1cc(C(=O)N2Cc3c(F)cc(-c4noc(C(F)(F)F)n4)cc3OC[C@H]2C)on1
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)C1(C#N)CC1
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)c1csnn1
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)[C@@H]1CCCO1
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)C12CCN(CC1)CC2
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)C1(C#N)CCN(C)CC1
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)C1(F)CCN(C)CC1
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)C1(C)CCNCC1
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)[C@H]1CCN(C)C1
CNC(=O)CC(=O)N1Cc2c(F)cc(-c3noc(C(F)(F)F)n3)cc2OC[C@H]1C
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)C1CN(C)C1
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)CCN
C[C@@H]1COc2cc(-c3noc(C(F)(F)F)n3)cc(F)c2CN1C(=O)[C@@H]1CCN(C)C1
C[C@@H]1COc2cc(-c3nnc(C(F)F)o3)cc(F)c2CN1C(=O)C1(C)CCOCC1
C[C@@H]1COc2cc(-c3nnc(C(F)F)o3)ccc2CN1C(=O)C1(C)CCOCC1
COc1ccccc1N1C(=O)[C@@H](C(C)C)N(Cc2ccc(cc2)C(=O)NO)C1=O |r|
ONC(=O)c1ccc(Cn2sc3ncccc3c2=O)cc1
FC(F)(F)c1nc(no1)-c1cccc(c1)C(=O)NCC1(CCOCC1)c1nc(cs1)-c1ccccc1
FC(F)(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccccc2)nc1
CC(Nc1ncc(cn1)-c1nnc(o1)C(F)(F)F)c1ccccc1
Cc1cccc(CNc2ncc(cn2)-c2nnc(o2)C(F)(F)F)n1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccccc2)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccc(F)cc2)nc1
CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccccc1
FC(F)c1nnc(o1)-c1cnc(NC(c2ccccc2)c2ccccc2)nc1
CN(c1ncc(cn1)-c1nnc(o1)C(F)F)C1(CC1)c1ccc(F)cc1
CC(C)(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccc(F)cc2F)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2c(F)cccc2F)nc1
FC(F)c1nnc(o1)-c1cnc(OC2(CC2)c2ccccc2)nc1
FC(F)c1nnc(o1)-c1cnc(NC(CC(F)(F)F)c2ccc(F)cc2)nc1
FC(F)c1nnc(o1)-c1cnc(N[C@@H](CC(F)(F)F)c2ccc(F)cc2)nc1 |r|
FC(F)c1nnc(o1)-c1cnc(N[C@H](CC(F)(F)F)c2ccc(F)cc2)nc1 |r|
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccccc2-c2ccc(F)cc2)nc1
FC(F)c1nnc(o1)-c1cnc(NC(c2ccc(F)cc2)C(F)(F)F)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccc(cc2)-c2ccc(F)cc2)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CCN(CC2)c2ccccc2)c2ccc(F)cc2)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2cccc(c2)-c2ccc(F)cc2)nc1
FC(F)c1nnc(o1)-c1cnc(NC(COc2ccccc2)c2ccc(F)cc2)nc1
CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
C[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1 |r|
C[C@@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1 |r|
COCC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
CCC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
CCCC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
CC(C)C(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccc(nc2)C#N)nc1
CC(=O)N1CCC(CC1)(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)C2CCCCC2)nc1
CC(C)C1(CC1)Nc1ncc(cn1)-c1nnc(o1)C(F)F
FC(F)c1nnc(o1)-c1cnc(NC2CCc3cc(F)ccc23)nc1
FC(F)c1nnc(o1)-c1cnc(NC(C(=O)N2CCOCC2)c2ccc(F)cc2)nc1
CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cn1
FC(F)Oc1ccc(cc1)C1(CC1)Nc1ncc(cn1)-c1nnc(o1)C(F)F
FC(F)Oc1ccc(c(F)c1)C1(CC1)Nc1ncc(cn1)-c1nnc(o1)C(F)F
FC(F)c1nnc(o1)-c1cnc(NC2CCCc3cc(F)ccc23)nc1
FC(F)c1nnc(o1)-c1cnc(NC(C(=O)Nc2ccccc2)c2ccc(F)cc2)nc1
FC(F)c1nnc(o1)-c1cnc(NC(C2CC2)c2ccc(F)cc2)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CCC(F)(F)CC2)c2ccc(F)cc2)nc1
CS(=O)(=O)NCC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
CS(=O)(=O)NC[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1 |r|
CS(=O)(=O)NC[C@@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1 |r|
FC(F)c1nnc(o1)-c1cnc(NC(CNS(=O)(=O)c2ccccc2)c2ccc(F)cc2)nc1
COc1ccccc1C1(CC1)Nc1ncc(cn1)-c1nnc(o1)C(F)(F)F
COc1cccc(c1)C1(CC1)Nc1ncc(cn1)-c1nnc(o1)C(F)(F)F
COc1ccc(cc1)C1(CC1)Nc1ncc(cn1)-c1nnc(o1)C(F)(F)F
COc1cccc(c1)C1(CC1)Nc1ncc(cn1)-c1nnc(o1)C(F)F
COc1ccc(cc1)C1(CC1)Nc1ncc(cn1)-c1nnc(o1)C(F)F
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccc(cc2)C(F)(F)F)nc1
COc1ccccc1C1(CC1)Nc1ncc(cn1)-c1nnc(o1)C(F)F
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccc(Br)cc2)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccc(cc2)C#N)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2cccc(c2)C(F)(F)F)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccc(Cl)cc2)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2cccc(Cl)c2)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccccc2Cl)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2cccc(OC(F)(F)F)c2)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccc(OC(F)(F)F)cc2)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccccc2OC(F)(F)F)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccccc2F)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2cccc(F)c2)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccccc2C(F)(F)F)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccc(F)c(F)c2)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2cccc(F)c2F)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2cc(F)ccc2F)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccc(F)cc2Cl)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccc(F)cc2C(F)(F)F)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccc(Br)nc2)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2cccnc2)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccc(Cl)cc2F)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccc(F)cn2)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccc(OCC(F)(F)F)cc2)nc1
CS(=O)(=O)NCc1ccc(cc1)C1(CC1)Nc1ncc(cn1)-c1nnc(o1)C(F)F
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccc(OC(F)(F)F)cc2F)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccc(cc2F)C(F)(F)F)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2cc(F)cc(F)c2)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2cccc(Cl)c2F)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2c(F)cc(F)cc2F)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2cc(OC(F)(F)F)ccc2F)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2cc(Cl)ccc2F)nc1
Cc1cccc(c1Cl)C1(CC1)Nc1ncc(cn1)-c1nnc(o1)C(F)F
CC(=O)NCC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
CC(=O)NC[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1 |r|
CC(=O)NCC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
FC(F)c1nnc(o1)-c1cnc(NC(CNC(=O)c2ccccc2)c2ccc(F)cc2)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2cc(F)ccc2Cl)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2cc(ccc2Cl)C(F)(F)F)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccnc(Br)c2)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccnc(c2)C#N)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2ccc(OCC(F)(F)F)cc2Cl)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2cccc(c2Cl)C(F)(F)F)nc1
FC(F)Oc1cccc(c1Cl)C1(CC1)Nc1ncc(cn1)-c1nnc(o1)C(F)F
CC(F)(F)COc1cccc(c1Cl)C1(CC1)Nc1ncc(cn1)-c1nnc(o1)C(F)F
FC(F)c1nnc(o1)-c1cnc(NC2(CCC2)c2ccc(F)cc2)nc1
FC(F)c1nnc(o1)-c1cnc(NC2(CCC2)c2ccc(OCC(F)(F)F)cc2)nc1
Cc1ccc(Cl)c(c1)C1(CC1)Nc1ncc(cn1)-c1nnc(o1)C(F)F
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2cccc(F)c2Cl)nc1
CC(O)C(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1F
NCC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
CC(C)(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1F
CC(C)(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1c(F)cccc1F
C[C@@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1F |r|
C[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1F |r|
C[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1c(F)cccc1F |r|
C[C@@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1c(F)cccc1F |r|
FC(F)c1nnc(o1)-c1cnc(N[C@@H](CC(F)(F)F)c2ccc(F)cc2F)nc1 |r|
FC(F)c1nnc(o1)-c1cnc(NC(CC(F)(F)F)c2ccc(F)cc2F)nc1
FC(F)c1nnc(o1)-c1cnc(NC(CC(F)(F)F)c2c(F)cccc2F)nc1
CS(=O)(=O)NC[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1F |r|
CS(=O)(=O)NC[C@@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1F |r|
COc1cc(F)c(c(F)c1)C1(CC1)Nc1ncc(cn1)-c1nnc(o1)C(F)F
CCS(=O)(=O)NCC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
CC(C)S(=O)(=O)NCC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
FC(F)c1nnc(o1)-c1cnc(NC(CNS(=O)(=O)C2CC2)c2ccc(F)cc2)nc1
CCCS(=O)(=O)NCC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
CC(C)CS(=O)(=O)NCC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
CN(CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1)S(C)(=O)=O
FC(F)c1nnc(o1)-c1cnc(NC(CNC(=O)C(F)(F)F)c2ccc(F)cc2)nc1
CS(=O)(=O)NC[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)F)cc1 |r|
CS(=O)(=O)NC[C@@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)F)cc1 |r|
CS(=O)(=O)NC[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)F)cc1F |r|
CS(=O)(=O)NC[C@@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)F)cc1F |r|
FC(F)c1nnc(o1)-c1cnc(NC(CNS(=O)(=O)CC(F)(F)F)c2ccc(F)cc2)nc1
FC(F)c1nnc(o1)-c1cnc(N[C@@H](CNS(=O)(=O)CC(F)(F)F)c2ccc(F)cc2)nc1 |r|
FC(F)c1nnc(o1)-c1cnc(N[C@@H](CN2CCCS2(=O)=O)c2ccc(F)cc2)nc1 |r|
FC(F)c1nnc(o1)-c1cnc(N[C@H](CN2CCCS2(=O)=O)c2ccc(F)cc2)nc1 |r|
CS(=O)(=O)NC[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)(F)F)cc1 |r|
CS(=O)(=O)NC[C@@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)(F)F)cc1 |r|
CS(=O)(=O)NC[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)C1CC1 |r|
CS(=O)(=O)NC[C@@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)C1CC1 |r|
CS(=O)(=O)NCCC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
CC(NS(C)(=O)=O)[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1 |r|
CC(NS(C)(=O)=O)[C@@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1 |r|
CS(=O)(=O)Nc1cccc(c1)C(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
CS(=O)(=O)Nc1ccc(cc1)C(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
CS(=O)(=O)Nc1ccccc1C(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
CS(=O)(=O)Nc1ccccc1CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
CS(=O)(=O)Nc1cccc(CC(Nc2ncc(cn2)-c2nnc(o2)C(F)F)c2ccc(F)cc2)c1
CS(=O)(=O)Nc1ccc(CC(Nc2ncc(cn2)-c2nnc(o2)C(F)F)c2ccc(F)cc2)cc1
FC(F)c1nnc(o1)-c1cnc(N[C@@H](COC2CC2)c2ccc(F)cc2F)nc1 |r|
FC(F)c1nnc(o1)-c1cnc(NC(COC2CC2)c2ccc(F)cc2F)nc1
CN(C[C@@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1F)S(C)(=O)=O |r|
CS(=O)(=O)N(CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1F)CC(F)(F)F
CCS(=O)(=O)NC[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1F |r|
CCS(=O)(=O)N(C)CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1F
CCS(=O)(=O)N(CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1F)CC(F)(F)F
FC(F)c1nnc(o1)-c1cnc(NC(CNS(=O)(=O)C2CC2)c2ccc(F)cc2F)nc1
CN(CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1F)S(=O)(=O)C1CC1
FC(F)c1nnc(o1)-c1cnc(NC(CN(CC(F)(F)F)S(=O)(=O)C2CC2)c2ccc(F)cc2F)nc1
CN(CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)F)cc1F)S(C)(=O)=O
CS(=O)(=O)N(CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)F)cc1F)CC(F)(F)F
CCS(=O)(=O)NCC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)F)cc1F
CCS(=O)(=O)N(C)CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)F)cc1F
CCS(=O)(=O)N(CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)F)cc1F)CC(F)(F)F
FC(F)Oc1ccc(C(CNS(=O)(=O)C2CC2)Nc2ncc(cn2)-c2nnc(o2)C(F)F)c(F)c1
CN(CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)F)cc1F)S(=O)(=O)C1CC1
FC(F)Oc1ccc(C(CN(CC(F)(F)F)S(=O)(=O)C2CC2)Nc2ncc(cn2)-c2nnc(o2)C(F)F)c(F)c1
CN(CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)(F)F)cc1F)S(=O)(=O)C1CC1
CCN(CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)(F)F)cc1)S(C)(=O)=O
CCS(=O)(=O)NCC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)(F)F)cc1
CCS(=O)(=O)N(C)CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)(F)F)cc1
CCS(=O)(=O)N(CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)(F)F)cc1)CC(F)(F)F
FC(F)c1nnc(o1)-c1cnc(NC(CNS(=O)(=O)C2CC2)c2ccc(OC(F)(F)F)cc2)nc1
CN(CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)(F)F)cc1)S(=O)(=O)C1CC1
FC(F)c1nnc(o1)-c1cnc(NC(CN(CC(F)(F)F)S(=O)(=O)C2CC2)c2ccc(OC(F)(F)F)cc2)nc1
CS(=O)(=O)C[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1 |r|
CS(=O)(=O)C[C@@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1 |r|
FC(F)c1nnc(o1)-c1cnc(N[C@H](COCC(F)(F)F)c2ccc(F)cc2)nc1 |r|
FC(F)c1nnc(o1)-c1cnc(N[C@@H](COCC(F)(F)F)c2ccc(F)cc2)nc1 |r|
FC(F)c1nnc(o1)-c1cnc(N[C@H](COCC(F)(F)F)c2ccc(F)cc2F)nc1 |r|
FC(F)c1nnc(o1)-c1cnc(N[C@H](COCC(F)(F)F)c2ccc(F)cc2F)nc1 |r|
CCS(=O)(=O)N(C[C@@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1)CC(F)(F)F |r|
CCS(=O)(=O)N(C[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1)CC(F)(F)F |r|
FC(F)c1nnc(o1)-c1cnc(N[C@H](CN(CC(F)(F)F)S(=O)(=O)C2CC2)c2ccc(F)cc2)nc1 |r|
FC(F)c1nnc(o1)-c1cnc(N[C@@H](CN(CC(F)(F)F)S(=O)(=O)C2CC2)c2ccc(F)cc2)nc1 |r|
CN(C[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1)C(C)=O |r|
CN(C[C@@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1)C(C)=O |r|
CC(=O)N(C[C@@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1)CC(F)(F)F |r|
CC(=O)N(C[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1)CC(F)(F)F |r|
FC(F)c1nnc(o1)-c1cnc(N[C@@H](CNC(=O)C2CC2)c2ccc(F)cc2)nc1 |r|
FC(F)c1nnc(o1)-c1cnc(N[C@H](CNC(=O)C2CC2)c2ccc(F)cc2)nc1 |r|
CN(C[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1)C(=O)C1CC1 |r|
CN(CC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)cc1)C(=O)C1CC1
FC(F)c1nnc(o1)-c1cnc(N[C@@H](CN(CC(F)(F)F)C(=O)C2CC2)c2ccc(F)cc2)nc1 |r|
FC(F)c1nnc(o1)-c1cnc(N[C@H](CN(CC(F)(F)F)C(=O)C2CC2)c2ccc(F)cc2)nc1 |r|
CS(=O)(=O)NCC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)c(F)c1
CS(=O)(=O)NC[C@@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)c(F)c1 |r|
CS(=O)(=O)N(C[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)c(F)c1)CC(F)(F)F |r|
CS(=O)(=O)N(C[C@@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(F)c(F)c1)CC(F)(F)F |r|
CS(=O)(=O)NC[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(Cl)cc1 |r|
CS(=O)(=O)NC[C@@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(Cl)cc1 |r|
CS(=O)(=O)N(C[C@@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(Cl)cc1)CC(F)(F)F |r|
CS(=O)(=O)N(C[C@H](Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(Cl)cc1)CC(F)(F)F |r|
FC(F)c1nnc(o1)-c1cnc(N[C@@H](Cn2cnc(c2)C(F)(F)F)c2ccc(F)cc2)nc1 |r|
FC(F)c1nnc(o1)-c1cnc(N[C@H](Cn2cnc(c2)C(F)(F)F)c2ccc(F)cc2)nc1 |r|
FC(F)c1nnc(o1)-c1cnc(N[C@@H](Cn2cc(cn2)C(F)(F)F)c2ccc(F)cc2)nc1 |r|
FC(F)c1nnc(o1)-c1cnc(N[C@H](Cn2cc(cn2)C(F)(F)F)c2ccc(F)cc2)nc1 |r|
FC(F)c1nnc(o1)-c1cnc(NC(CN2CCCC2=O)c2ccc(F)cc2)nc1
FC(F)c1nnc(o1)-c1cnc(N[C@@H](CN2CCCC2=O)c2ccc(F)cc2)nc1 |r|
ONC(=O)c1ccc(CN2CCCc3cc(Cl)ccc23)cc1
ONC(=O)c1ccc(CN2CCCc3ccccc23)cc1
ONC(=O)c1ccc(CN2CCCc3cc(Cl)ccc23)c(F)c1
CC(N1CCCc2cc(Cl)ccc12)c1ccc(cc1)C(=O)NO |w:1.0|
ONC(=O)c1ccc(CN2CCCc3cc(F)ccc23)cc1
ONC(=O)c1ccc(CN2CCCc3cc(Cl)c(Cl)cc23)cc1
ONC(=O)c1ccc(CN2CCCc3cc(F)c(Cl)cc23)cc1
ONC(=O)c1ccc(CN2CCCc3cc(Cl)c(F)cc23)cc1
CC1(C)CCc2cc(Cl)ccc2N1Cc1ccc(cc1)C(=O)NO
CC1(C)CCc2cc(F)ccc2N1Cc1ccc(cc1)C(=O)NO
CC1(C)CC(=O)N(Cc2ccc(cc2)C(=O)NO)c2ccc(Cl)cc12
CC1(C)CCN(Cc2ccc(cc2)C(=O)NO)c2ccc(Cl)cc12
CC1(C)CCN(Cc2ccc(cc2)C(=O)NO)c2ccc(F)cc12
COC(=O)c1ccc(CN2CCN(C(=O)OC(C)(C)C)c3ccccc23)cc1
ONC(=O)c1ccc(CN2CCSc3ccccc23)cc1
ONC(=O)c1ccc(CN2CCS(=O)c3ccccc23)cc1
CC(C)(C)OC(=O)N1CC(=O)N(Cc2ccc(cc2)C(=O)NO)c2ccccc12
Fc1cc(ccc1CN(c1ccccc1)S(=O)(=O)N1CCNCC1)-c1nnc(o1)C(F)(F)F
Fc1cccc(c1)N(Cc1ccc(cc1F)-c1nnc(o1)C(F)(F)F)S(=O)(=O)N1CCNCC1
FC(F)c1nnc(o1)-c1ccc(CN(c2ccc(F)c(Cl)c2)S(=O)(=O)N2CCS(=O)(=O)CC2)nc1
Fc1cc(ccc1CN(c1ccccc1)S(=O)(=O)N1CCN(CC1)C1COC1)-c1nnc(o1)C(F)(F)F
FC(F)(F)c1nnc(o1)-c1ccc(CN(c2ccccc2)S(=O)(=O)N2CCN(CC2)C2COC2)nc1
FC(F)c1nnc(o1)-c1ccc(CN(c2ccc(F)c(Cl)c2)S(=O)(=O)N2CCN(CC2)C2COC2)cc1
CN1CCN(CC1)S(=O)(=O)N(Cc1ccc(cc1)-c1nnc(o1)C(F)F)c1ccc(F)c(Cl)c1
C[C@H]1CN(C[C@@H](C)N1C(C)=O)S(=O)(=O)N(Cc1ccc(cn1)-c1nnc(o1)C(F)F)c1ccccc1 |r|
C[C@H]1CN(C[C@@H](C)N1C(C)=O)S(=O)(=O)N(Cc1ccc(cc1)-c1nnc(o1)C(F)F)c1cccnc1 |r|
CCN1[C@@H](C)CN(C[C@H]1C)S(=O)(=O)N(Cc1ccc(cn1)-c1nnc(o1)C(F)F)c1ccccc1 |r|
C[C@H]1CN(C[C@@H](C)N1C)S(=O)(=O)N(Cc1ccc(cc1)-c1nnc(o1)C(F)F)c1cccnc1 |r|
CN(CCN1CCN(C)CC1)S(=O)(=O)N(Cc1ccc(cc1)-c1nnc(o1)C(F)F)c1ccccc1
ONC(=O)c1cccc(Nc2nc3cc(Cl)c(Cl)cc3o2)c1
CC1(C)N(Cc2c1cccc2C(=O)NO)c1nc2ccc(cc2[nH]1)C(F)(F)F
Cc1cc(O)cc(C)c1-c1nc2ccc(cc2[nH]1)C(=O)NO
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccccc1C(F)(F)F
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccc(Br)cc1
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1ccccc1
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccc2OCCOc2c1
ONC(=O)c1ccc2nc([nH]c2c1)-c1cccc(Br)c1
CC(C)c1ccc(cc1)-c1nc2ccc(cc2[nH]1)C(=O)NO
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccnc2ccccc12
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)C#C
COc1cccc(-c2nc3ccc(cc3[nH]2)C(=O)NO)c1O
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccc2OCCc2c1
CC(C)Oc1ccc(cc1)-c1nc2ccc(cc2[nH]1)C(=O)NO
ONC(=O)c1ccc2nc([nH]c2c1)-c1cccs1
ONC(=O)c1ccc2nc([nH]c2c1)-c1cc(Cl)ccc1O
CCc1ccc(cc1)-c1nc2ccc(cc2[nH]1)C(=O)NO
Cn1c(cc2ccccc12)-c1nc2ccc(cc2[nH]1)C(=O)NO
COc1ccc(Oc2cccc(c2)-c2nc3ccc(cc3[nH]2)C(=O)NO)cc1
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccccc1-c1ccccc1
CCN(CC)CCOc1ccc(cc1)-c1nc2ccc(cc2[nH]1)C(=O)NO
ONC(=O)c1ccc2nc([nH]c2c1)-c1cccc(OCCOc2ccccc2)c1
CC(C)(C)c1ccc(cc1)-c1nc2ccc(cc2[nH]1)C(=O)NO
CCCCc1ccc(cc1)-c1nc2ccc(cc2[nH]1)C(=O)NO
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1ccccc1F
COc1ccc(cc1OC)-c1ccc(o1)-c1nc2ccc(cc2[nH]1)C(=O)NO
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccc(s1)-c1ccccc1F
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccc(s1)-c1cccc(Cl)c1
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccc(s1)-c1ccccc1
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccc(c(F)c1)-c1ccccc1
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1cccc(CN2CCCCC2)c1
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1ccc(CN2CCOCC2)cc1
COCCCNCc1ccc(cc1)-c1ccc(cc1)-c1nc2ccc(cc2[nH]1)C(=O)NO
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1ccc(\C=N\O)cc1
CN(C)C(=O)c1cccc(c1)-c1ccc(cc1)-c1nc2ccc(cc2[nH]1)C(=O)NO
ONC(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1ccc(CN2CCCC2)cc1
C[C@H]1CN(Cc2ccc(cc2)-c2ccc(cc2)-c2nc3ccc(cc3[nH]2)C(=O)NO)C[C@@H](C)O1 |r|
CS(=O)(=O)Nc1ccc(cc1)-c1ccc(cc1)-c1nc2ccc(cc2[nH]1)C(=O)NO
CN1CCN(Cc2ccc(cc2)-c2nc3ccc(cc3[nH]2)C(=O)NO)CC1
CC(C)c1ccc(cc1)-c1nc2cc(ccc2n1C)C(=O)NO
Cn1c(nc2cc(ccc12)C(=O)NO)-c1ccc(cc1)-c1ccccc1
COc1c(C)cc(cc1C)-c1nc2cc(ccc2n1C)C(=O)NO
CC(C)c1ccc(cc1)-c1nc2cc(ccc2o1)C(=O)NO
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(Br)cc1
CC(C)(C)c1ccc(cc1)-c1nc2cc(ccc2o1)C(=O)NO
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(F)c(F)c1
ONC(=O)c1ccc2oc(nc2c1)-c1ccccc1
ONC(=O)c1ccc2oc(nc2c1)-c1ccc2OCOc2c1
COc1ccc(cc1)-c1nc2cc(ccc2o1)C(=O)NO
ONC(=O)c1ccc2oc(nc2c1)-c1ccccc1Cl
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(nc1)N1CCOCC1
ONC(=O)c1ccc2oc(nc2c1)-c1cccc(Br)c1
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(cc1)-c1ccccc1F
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(cc1)-c1ccncc1
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(cc1)-c1cccnc1
COc1ccncc1-c1ccc(cc1)-c1nc2cc(ccc2o1)C(=O)NO
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(cc1)C1CC1
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(cc1)-c1ccc(CN2CCCCC2)cc1
CCN(CC)c1ccc(cc1)-c1nc2cc(ccc2o1)C(=O)NO
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(cc1)C#N
ONC(=O)c1ccc2oc(nc2c1)-c1ccc2[nH]nnc2c1
Cc1ncccc1-c1nc2cc(ccc2o1)C(=O)NO
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(nc1)N1CCCC1
ONC(=O)c1ccc2oc(Nc3ccccc3)nc2c1
CN(Cc1ccccc1)c1nc2cc(ccc2o1)C(=O)NO
ONC(=O)c1ccc2oc(NCCc3ccccc3)nc2c1
ONC(=O)c1ccc2oc(nc2c1)N1CCc2ccccc2C1
ONC(=O)c1ccc2oc(Nc3cccc(OCc4ccccc4)c3)nc2c1
ONC(=O)c1ccc2oc(nc2c1)N1CCC(Cc2ccccc2)CC1
CC(C)c1ccc(cc1)-c1nc2ccc(cc2o1)C(=O)NO
ONC(=O)c1ccc2nc(oc2c1)-c1ccc(F)cc1
CC(C)(C)c1ccc(cc1)-c1nc2ccc(cc2o1)C(=O)NO
COc1ccc(cc1)-c1nc2ccc(cc2o1)C(=O)NO
ONC(=O)c1ccc2nc(oc2c1)-c1ccc2[nH]nnc2c1
ONC(=O)c1ccc2nc(oc2c1)-c1ccc(nc1)-c1cccnc1
CC(C)c1ccc(cc1)-c1nc2ncc(cc2[nH]1)C(=O)NO
CC(C)c1ccc(cc1)-c1cc2cc(ccc2[nH]1)C(=O)NO
CC(C)c1ccc(cc1)-c1nc2cc(ccc2s1)C(=O)NO
ONC(=O)c1ccc2sc(nc2c1)-c1ccc(F)cc1
COc1ccc(cc1)-c1nc2cc(ccc2s1)C(=O)NO
ONC(=O)c1ccc2sc(Cc3ccc(F)cc3)nc2c1
ONC(=O)c1ccc2sc(nc2c1)-c1cncc(Br)c1
COc1cccc2cc(oc12)-c1nc2cc(ccc2s1)C(=O)NO
CCc1ccc(cc1)-c1nc2cc(ccc2s1)C(=O)NO
CC(C)c1ccc(cc1)-c1cc2cc(cnc2[nH]1)C(=O)NO
CC(C)c1ccc(cc1)-c1cc2cc(cnc2s1)C(=O)NO
CC(C)c1ccc(cc1)-c1cc2ccc(cc2s1)C(=O)NO
CC(C)c1ccc(cc1)-c1cc2cc(ccc2s1)C(=O)NO
ONC(=O)c1ccc2sc(cc2c1)-c1cccc(c1)C(F)(F)F
COc1ccc(cc1)-c1cc2cc(ccc2s1)C(=O)NO
ONC(=O)c1ccc2sc(cc2c1)-c1ccc2[nH]ccc2c1
ONC(=O)c1ccc2sc(cc2c1)-c1cccnc1
COc1ncccc1-c1cc2cc(ccc2s1)C(=O)NO
Cn1cc(cn1)-c1cc2cc(ccc2s1)C(=O)NO
Cc1noc(C)c1-c1cc2cc(ccc2s1)C(=O)NO
ONC(=O)c1ccc2sc(cc2c1)-c1ccc(OC(F)(F)F)cc1
ONC(=O)c1ccc2sc(cc2c1)-c1cc(F)ccc1O
COc1ccc(F)cc1-c1cc2cc(ccc2s1)C(=O)NO
CN(C)C(=O)c1ccc(cc1)-c1cc2cc(ccc2s1)C(=O)NO
CS(=O)(=O)Nc1ccc(cc1)-c1cc2cc(ccc2s1)C(=O)NO
CC(C)c1ccc(cc1)-c1cc2ncc(cc2s1)C(=O)NO
CC(C)c1ccc(cc1)-c1cc2ccc(cc2o1)C(=O)NO
CC(C)c1ccc(cc1)-c1cc2cc(cnc2o1)C(=O)NO
CC(C)c1ccc(cc1)-c1cc2ncc(cc2o1)C(=O)NO
CCN(CC)Cc1cc2ccc(cc2o1)C(=O)NO
OCc1cc2ccc(cc2o1)C(=O)NO
ONC(=O)c1ccc2nc(NCc3ccc(cc3)-c3ccccc3)[nH]c2c1
ONC(=O)c1ccc2nc([nH]c2c1)N1CCN(CC1)c1ccc(F)cc1
ONC(=O)c1ccc2nc(NCc3ccccc3)[nH]c2c1
ONC(=O)c1ccc2nc(Nc3cccc(OCc4ccccc4)c3)[nH]c2c1
ONC(=O)c1ccc2nc(Nc3cccc(c3)-c3ccccc3)[nH]c2c1
Cn1c(Nc2ccccc2)nc2cc(ccc12)C(=O)NO
CC(C)c1ccc(Nc2nc3cc(ccc3n2C)C(=O)NO)cc1
CN(Cc1ccccc1)c1nc2cc(ccc2n1C)C(=O)NO
Cn1c(NCCc2ccccc2)nc2cc(ccc12)C(=O)NO
Cn1c(nc2cc(ccc12)C(=O)NO)N(Cc1ccccc1)c1ccccc1
Cn1c(Nc2cccc(OCc3ccccc3)c2)nc2cc(ccc12)C(=O)NO
Cn1c(nc2cc(ccc12)C(=O)NO)N1CCC(Cc2ccccc2)CC1
Cn1c(Nc2cccc(c2)-c2ccccc2)nc2cc(ccc12)C(=O)NO
Cn1c(nc2cc(ccc12)C(=O)NO)N1CCc2ccccc2C1
ONC(=O)c1ccc2cc(sc2c1)-c1ccoc1
COc1cc(ccc1O)-c1cc2ccc(cc2s1)C(=O)NO
CC1CCN(CC1)c1ccc(cn1)-c1nc2cc(ccc2o1)C(=O)NO
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(NC2CCCCCC2)nc1
COc1ccccc1N1CCN(CC1)c1ccc(cn1)-c1nc2cc(ccc2o1)C(=O)NO
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(nc1)-c1ccccc1
ONC(=O)c1ccc2oc(COc3cccc(F)c3)cc2c1
CC(C)(C)c1ccc(OCc2cc3cc(ccc3o2)C(=O)NO)cc1
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(cc1F)-c1ccccc1
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(cc1F)-c1cccnc1
CS(=O)(=O)c1ccc(cc1)-c1ccc(cc1)-c1nc2cc(ccc2o1)C(=O)NO
Cc1noc(C)c1-c1ccc(cc1)-c1nc2cc(ccc2o1)C(=O)NO
COc1cc(ccc1-c1nc2cc(ccc2o1)C(=O)NO)-c1ccccc1F
C[C@H]1CN(Cc2cccc(c2)-c2nc3cc(ccc3o2)C(=O)NO)C[C@@H](C)O1 |r|
COCCN(C)Cc1cccc(c1)-c1nc2cc(ccc2o1)C(=O)NO
C[C@H]1CN(Cc2ccc(cc2)-c2nc3cc(ccc3o2)C(=O)NO)C[C@@H](C)O1 |r|
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(CN2CCN(CC2)c2ccncc2)cc1
CC(C)c1ccc(cc1F)-c1nc2cc(ccc2o1)C(=O)NO
ONC(=O)c1ccc2oc(nc2c1)-c1ccc2OCCOc2c1
ONC(=O)c1ccc2oc(nc2c1)-c1cccc(O)c1
Cc1[nH]c2ccccc2c1-c1nc2cc(ccc2o1)C(=O)NO
ONC(=O)c1ccc2oc(Nc3cccc(c3)-c3ccccc3)nc2c1
ONC(=O)c1ccc2oc(NC3CCCCCCC3)nc2c1
ONC(=O)c1ccc2oc(NCc3ccc(cc3)-c3ccccc3)nc2c1
ONC(=O)c1ccc2oc(nc2c1)N(Cc1ccccc1)c1ccccc1
COc1ccc(CN(CCN(C)C)c2nc3cc(ccc3o2)C(=O)NO)cc1OC
Cn1cc(CNCC2CCN(CC2)c2nc3cc(ccc3o2)C(=O)NO)c2ccccc12
ONC(=O)c1ccc2oc(NC3(CCCCC3)c3cccc(F)c3)nc2c1
Cc1ccc(Nc2nc3cc(ccc3o2)C(=O)NO)cc1
ONC(=O)c1ccc2sc(COCc3ccccc3)nc2c1
OCc1nc2cc(ccc2s1)C(=O)NO
ONC(=O)c1ccc2sc(Cc3ccc(cc3)-c3ccncc3)nc2c1
ONC(=O)c1ccc2sc(CN3CCCCC3)nc2c1
CC(C)CN(CC(C)C)Cc1nc2cc(ccc2s1)C(=O)NO
CC(C)c1ccc(NCc2nc3cc(ccc3s2)C(=O)NO)cc1
COc1ccc(cn1)-c1cc2cc(ccc2o1)C(=O)NO
OCc1ccccc1-c1cc2cc(ccc2o1)C(=O)NO
ONC(=O)c1ccc2cc(oc2c1)-c1ccccc1
CN(C)Cc1ccc(cc1)-c1cc2ccc(cc2o1)C(=O)NO
ONC(=O)c1ccc2cc(oc2c1)-c1cccc(O)c1
COc1cccc(c1)-c1cc2ccc(cc2o1)C(=O)NO
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(OC(F)(F)F)cc1
ONC(=O)c1ccc2oc(nc2c1)-c1ccc(cc1)C(F)(F)F
COc1ccc(cn1)-c1ccc(cc1)-c1nc2cc(ccc2o1)C(=O)NO
COc1ncccc1-c1ccc(cc1)-c1nc2cc(ccc2o1)C(=O)NO
CC(C)c1ccc(Nc2nc3cc(ccc3o2)C(=O)NO)cc1
ONC(=O)c1ccc2nc(sc2c1)-c1cccc2cccnc12
CC(C)(C)c1ccc(cc1)-c1nc2cc(ccc2s1)C(=O)NO
COc1ccc(cn1)-c1ccc(-c2nc3cc(ccc3o2)C(=O)NO)c(F)c1
CC(O)COC[C@H]1O[C@@H]2O[C@@H]3[C@@H](COCC(C)O)O[C@H](O[C@@H]4[C@@H](COCC(C)O)O[C@H](O[C@@H]5[C@@H](COCC(C)O)O[C@H](O[C@@H]6[C@@H](COCC(C)O)O[C@H](O[C@@H]7[C@@H](COCC(C)O)O[C@H](O[C@@H]8[C@@H](COCC(C)O)O[C@H](O[C@H]1[C@@H](O)[C@@H]2O)[C@@H](O)[C@@H]8O)[C@@H](O)[C@@H]7O)[C@@H](O)[C@@H]6O)[C@@H](O)[C@@H]5O)[C@@H](O)[C@@H]4O)[C@@H](O)[C@@H]3O
CCCCNNC(=O)c1ccc(CN=[N+]=[N-])cc1
CCCCNNC(=O)c1ccc(cc1)-c1cccc(F)c1F
CCCCNNC(=O)c1ccc(cc1)-c1cc(C)cc(F)c1
CCCCNNC(=O)c1ccc(cc1)-c1cc(ccc1F)C(=O)OCC
COc1ccc(cc1CNc1ncc(cn1)C(=O)NO)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](COCC1=O)c1ccccc1 |r|
Fc1cc(ccc1-c1noc(n1)C(F)(F)F)N1[C@@H](COCC1=O)c1ccccc1 |r|
CC(C)(C)OC(=O)N1CCN([C@H](C1)c1ccccc1)c1ccc(cn1)-c1noc(n1)C(F)(F)F |r|
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CC[NH2+]C[C@@H]1c1ccccc1 |r|
Fc1cc(cnc1N1C(CCC1=O)c1ccccc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1[C@@H](CCC1=O)c1ccccc1 |r|
CC(C)(C)OC(=O)[C@@H]1CCC(=O)N1c1cc(F)c(cc1F)-c1noc(n1)C(F)(F)F |r|
Cc1noc(n1)[C@@H]1CCC(=O)N1c1cc(F)c(cc1F)-c1noc(n1)C(F)(F)F |r|
Cc1noc(n1)[C@H]1CCCCN1c1ncc(cc1Cl)-c1noc(n1)C(F)(F)F |r|
Cc1noc(n1)[C@H]1CCCCN1c1ncc(cn1)-c1noc(n1)C(F)(F)F |r|
Cc1noc(n1)[C@@H]1CCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1F |r|
CC(C)(C)OC(=O)N1CCN([C@H](C1)c1ccccc1)c1c(F)cc(cc1F)-c1noc(n1)C(F)(F)F |r|
Fc1cc(cc(F)c1-c1noc(n1)C(F)(F)F)N1C(CCC1=O)c1ccccc1Cl
FC(F)(F)c1nc(no1)-c1ccc(cn1)N1[C@@H](COCC1=O)c1ccccc1 |r|
Fc1cc(-c2noc(n2)C(F)(F)F)c(F)cc1N1[C@@H](COC1=O)c1ccccc1 |r|
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](CCC1=O)c1nc(no1)-c1ccccn1 |r|
Cc1noc(n1)[C@H]1CCCCN1c1ccc(-c2noc(n2)C(F)(F)F)c(Cl)c1 |r|
CN(C(=O)[C@@H]1CCC(=O)N1c1cc(F)c(cc1F)-c1noc(n1)C(F)(F)F)C(C)(C)C |r|
Nc1ccccc1NC(=O)[C@@H]1CCC(=O)N1c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](CCC1=O)c1nc2ccccc2[nH]1 |r,$;;;;;;;;;;;;;;;;;;;;;;;;;;;;;HN$|
Fc1cc(ccc1N1[C@@H](CCC1=O)c1nc2ccccc2o1)-c1noc(n1)C(F)(F)F |r|
Fc1ccccc1COc1cc(ccn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](CCCC1=O)c1nc2ccccc2s1 |r|
FC(F)(F)c1nc(no1)-c1ccc(N[C@@H]2CCCC[C@H]2c2ccccc2)nc1 |r|
FC(F)(F)c1nc(no1)-c1ccc(CN(c2ccccn2)c2ccccn2)cc1
FC(F)(F)c1nc(no1)-c1ccc(Cn2c3ccccc3ccc2=O)cc1
Cc1nc2cc(F)ccc2n1Cc1ccc(cc1F)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)C2CCS(=O)(=O)CC2)c2cccc(c2)C(F)(F)F)cc1
Fc1ccccc1Cc1cnc(-c2noc(n2)C(F)(F)F)c(F)c1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)N2CCOCC2)c2cccc(c2)C(F)(F)F)cc1
CN1CCN(C(C1)c1ccccc1)c1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](COCC1=O)c1nc(no1)-c1ccccn1 |r|
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](COCC1=O)c1nc2ccccc2o1 |r|
CN1CCN(C(C1O)c1cccc(F)c1)c1ccc(cn1)-c1noc(n1)C(F)(F)F
Fc1cc(ccc1-c1noc(n1)C(F)(F)F)N1C(CCC1=O)c1ccccc1Cl
Fc1cc(F)cc(c1)[C@@H]1CNC(C2CCOCC2)C(=O)N1c1ccc(cn1)-c1noc(n1)C(F)(F)F |r|
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1C(CNCC1=O)c1ccccc1
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1C(CCCC1=O)c1ccccc1
Fc1cc(-c2noc(n2)C(F)(F)F)c(F)cc1N1C(CCC1=O)c1ccccc1
Fc1cc(ccc1N1C(CCC1=O)c1ccccc1)-c1noc(n1)C(F)(F)F
Fc1cc(ccc1-c1noc(n1)C(F)(F)F)N1C(CCC1=O)c1ccccc1
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1C(CCCC1=O)c1nc(no1)-c1ccccc1
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](COCC1=O)c1nc(no1)-c1ccncc1 |r|
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](COCC1=O)c1nc(no1)-c1cccnc1 |r|
Cc1noc(n1)[C@@H]1COCC(=O)N1c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
Cc1noc(n1)C1CCCC(=O)N1c1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)N2CCOCC2)c2cccc(c2)C(F)(F)F)nc1
FC(F)(F)c1nc(no1)-c1cnc(CN(C(=O)N2CCOCC2)c2cccc(c2)C(F)(F)F)nc1
CN1CCc2c(C1)n(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1ccccc21
FC(F)(F)c1nc(no1)-c1cccc(c1)S(=O)(=O)Nc1ccccc1
CC(C)c1ncc(cn1)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
Fc1cccc(c1)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)C(=O)C1CCS(=O)(=O)C1
Fc1cccc(c1)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)C(=O)C1CCS(=O)(=O)CC1
Cc1nccnc1C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
CCN1CCCC(C1)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
CC(C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1)c1ccn(C)n1
Cc1cc(CC(=O)N(Cc2ccc(cn2)-c2noc(n2)C(F)(F)F)c2cccc(F)c2)on1
Fc1cccc(c1)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)C(=O)C1CCOCC1
CC(C)N1CCCC(C1)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
Cc1nonc1CC(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
CC1(C)CC(CCO1)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
CC(C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1)n1cc(C)nn1
Fc1cccc(c1)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)C(=O)C1(CN2CCOCC2)CC1
CC(C(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F)n1cncn1
CC1=NN(CC(=O)N(Cc2ccc(cn2)-c2noc(n2)C(F)(F)F)c2cccc(F)c2)C(=O)C1 |t:1|
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)Cn2cncn2)c2cccc(c2)C(F)(F)F)cc1
CC(=O)N1CCN(CC(=O)N(Cc2ccc(cc2)-c2noc(n2)C(F)(F)F)c2cccc(c2)C(F)(F)F)CC1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)Cn2ncccc2=O)c2cccc(c2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)c2cncnc2)c2cccc(c2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)CCCn2cncn2)c2cccc(c2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)C2CC2c2cncnc2)c2cccc(c2)C(F)(F)F)cc1
CS(=O)(=O)CC(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
Cc1nnc(CC(=O)N(Cc2ccc(cc2)-c2noc(n2)C(F)(F)F)c2cccc(c2)C(F)(F)F)n1C
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)Cn2ccnn2)c2cccc(c2)C(F)(F)F)cc1
Cc1nc(C)n(CC(=O)N(Cc2ccc(cc2)-c2noc(n2)C(F)(F)F)c2cccc(c2)C(F)(F)F)n1
CC(=O)NCCC(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
CC(Cn1cncn1)C(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)CC2COC2)c2cccc(c2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)CN2CCS(=O)(=O)CC2)c2cccc(c2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)CC2CNCCO2)c2cccc(c2)C(F)(F)F)cc1
CN(C)CC(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)C2COCCO2)c2cccc(c2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)C2CCOCC2)c2cccc(c2)C(F)(F)F)cc1
COCCn1nc(ccc1=O)C(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
CC(C(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F)c1ncccn1
Cn1nc(ccc1=O)C(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)CCn2cncn2)c2cccc(c2)C(F)(F)F)cc1
CC(C)C(=O)N1CCC(CC1)C(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
CC(C)(C)OC(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
CC(C)(C#N)C(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
CN1CCN(CC(=O)N(Cc2ccc(cc2)-c2noc(n2)C(F)(F)F)c2cccc(c2)C(F)(F)F)CC1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)Cc2cnccn2)c2cccc(c2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)CC2COCCO2)c2cccc(c2)C(F)(F)F)cc1
Cn1ccc(CN(Cc2ccc(cc2)-c2noc(n2)C(F)(F)F)c2cccc(c2)C(F)(F)F)n1
CCC(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)Cn2cnc3ccccc23)c2cccc(c2)C(F)(F)F)cc1
Cc1nc2ccc(F)cc2n1Cc1ccc(cc1F)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccnc(OCc2cnc3ccccc3c2)c1
CN(C)c1cccc(COc2cc(ccn2)-c2noc(n2)C(F)(F)F)n1
FC(F)(F)c1nc(no1)-c1ccnc(OC2CCOCC2)c1
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](CCC1=O)c1nc2ccccc2o1 |r|
CCc1nnc(o1)[C@@H]1CCC(=O)N1c1cc(F)c(cc1F)-c1noc(n1)C(F)(F)F |r|
Fc1cc(ccc1N1[C@@H](CCC1=O)c1nc2ccccc2[nH]1)-c1noc(n1)C(F)(F)F |r|
Cn1c(nc2ccccc12)[C@@H]1CCC(=O)N1c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
Cn1c(nc2ccccc12)[C@@H]1CCC(=O)N1c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
CNc1ccccc1NC(=O)[C@@H]1CCC(=O)N1c1ccc(cc1)-c1noc(n1)C(F)(F)F |r,$;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;;$|
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](CCC1=O)C(=O)Nc1ccccc1 |r,$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;$|
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](CCC1=O)C(=O)NCCc1ccccc1 |r,$;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;$|
CC(C)(C)NC(=O)[C@@H]1CCC(=O)N1c1ccc(cc1)-c1noc(n1)C(F)(F)F |r,$;;;;HN;;;;;;;;;;;;;;;;;;;;;;;$|
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](CCC1=O)c1nc(no1)-c1cccnc1 |r|
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1[C@@H](CCC1=O)c1nc(no1)-c1ccncc1 |r|
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1C(CCC1=O)c1ccccc1
Fc1cc(ccc1N1C(CCC1=O)c1cccc(Cl)c1)-c1noc(n1)C(F)(F)F
Fc1cc(ccc1N1C(CCC1=O)c1ccccc1Cl)-c1noc(n1)C(F)(F)F
Fc1ccccc1C1CCC(=O)N1c1ccc(cc1F)-c1noc(n1)C(F)(F)F
Fc1cc(ccc1N1C(CCC1=O)c1ccc(Cl)cc1)-c1noc(n1)C(F)(F)F
Fc1cc(-c2noc(n2)C(F)(F)F)c(F)cc1N1C(CCC1=O)c1ccccc1Cl
Cc1noc(n1)[C@H]1CCCCN1c1cc(F)c(cc1F)-c1noc(n1)C(F)(F)F |r|
Cc1noc(n1)[C@@H]1CCC(=O)N1c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
Cc1noc(n1)[C@@H]1CCC(=O)N1c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
CC(C)(C)OC(=O)[C@@H]1CCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1F |r|
CC(C)(C)OC(=O)[C@@H]1CCC(=O)N1c1ccc(cc1F)-c1noc(n1)C(F)(F)F |r|
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1[C@@H](COCC1=O)c1ccccc1 |r|
CC(C)(C)OC(=O)N1C[C@H](N(C(=O)C1C1CCOCC1)c1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cc(F)cc(F)c1 |r|
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1C(CCCC1=O)c1ccccc1
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1C(CCC1=O)c1ccccc1Cl
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCOCC1c1ccccc1Cl
CN1CCN(C(C1O)c1cccc(F)c1)c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1
Fc1cccc(c1)C1N(CCNC1=O)c1ccc(cn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCOCC1c1cccnc1
CN1CCN([C@H](C1)c1ccccc1)c1ccc(cn1)-c1noc(n1)C(F)(F)F |r|
Fc1ccccc1C1COCCN1c1ccc(cn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCNCC1c1ccccc1
Fc1cccc(c1)C1COCCN1c1ccc(cn1)-c1noc(n1)C(F)(F)F
Cc1noc(n1)[C@H]1CCCCN1c1ccc(cn1)-c1noc(n1)C(F)(F)F |r|
Cc1cccc(CCOc2cc(ccn2)-c2noc(n2)C(F)(F)F)n1
Cc1noc(n1)[C@@H]1CCCCN1c1ccc(cn1)-c1noc(n1)C(F)(F)F |r|
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCOC[C@@H]1c1ccccc1 |r|
Fc1ccc(cc1)C1COCCN1c1ccc(cn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCOC[C@H]1c1ccccc1 |r|
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCOCC1c1ccccc1
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCOCC1c1cccc(c1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCCCC1c1ccccn1
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCCCC1c1ccncc1
OCC1CCC(N(C1)c1ccc(cn1)-c1noc(n1)C(F)(F)F)c1ccccc1
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCCC1c1ccncc1
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCCC1c1cccnc1
OCC1CC(N(C1)c1ccc(cn1)-c1noc(n1)C(F)(F)F)c1ccccc1
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCCC1c1ccccn1
Cc1nonc1C1CCCN1c1ccc(cn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCc2nc3ncccc3cc2C1
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1CCCCC1c1cccnc1
Cc1cc(=O)n2CCN(Cc2n1)c1ccc(cn1)-c1noc(n1)C(F)(F)F
CCOC(=O)N1CCN(C(C1)c1ccccc1)c1ccc(cn1)-c1noc(n1)C(F)(F)F
Fc1cc(-c2noc(n2)C(F)(F)F)c(F)cc1N1[C@@H](COCC1=O)c1ccccc1 |r|
Fc1cc(ccc1N1[C@@H](COCC1=O)c1ccccc1)-c1noc(n1)C(F)(F)F |r|
CN1CC(N(C(=O)C1)c1ccc(cc1)-c1noc(n1)C(F)(F)F)c1ccccc1
CC(C)(C)OC(=O)N1C[C@H](N(C(=O)C1)c1ccc(cc1)-c1noc(n1)C(F)(F)F)c1ccccc1 |r|
FC(F)(F)c1nc(no1)-c1cnc(cn1)N1[C@@H](COCC1=O)c1ccccc1 |r|
FC(F)(F)c1nc(no1)-c1ccc(nn1)N1[C@@H](COCC1=O)c1ccccc1 |r|
FC(F)(F)c1nc(no1)-c1ncc(cn1)N1[C@@H](COCC1=O)c1ccccc1 |r|
FC(F)(F)c1nc(no1)-c1ccnc(OCCc2cccc3cn[nH]c23)c1
Fc1cc(ccc1COc1ccccc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CC(C(=O)N2CCS(=O)(=O)CC2)c2cccc(c2)C(F)(F)F)nc1
FC(F)(F)c1nc(no1)-c1ccc(C[C@@H](C(=O)N2CCS(=O)(=O)CC2)c2cccc(c2)C(F)(F)F)nc1 |r|
Fc1cc(COc2ccccc2)ccc1-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)C2CCS(=O)(=O)CC2)c2cccc(c2)C(F)(F)F)nn1
NC(=O)c1ccccc1NCc1ccc(cn1)-c1noc(n1)C(F)(F)F
NC(=O)c1cccc(NCc2ccc(cc2)-c2noc(n2)C(F)(F)F)c1
FC(F)(F)C(=O)NC(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
CC(=O)NC(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
CS(=O)(=O)NC(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F |$;;;;HN;;;;;;;;;;;;;;;;;;;;;;;;;;;$|
CCNC(=O)NC(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F |$;;HN;;;HN;;;;;;;;;;;;;;;;;;;;;;;;;;;$|
COC(=O)NC(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F |$;;;;HN;;;;;;;;;;;;;;;;;;;;;;;;;;;$|
COC(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
CCNC(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
CS(=O)(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
Cc1nc(Cl)cnc1COc1ccc(cn1)-c1noc(n1)C(F)(F)F
Cc1ncc(OCc2ccc(cn2)-c2noc(n2)C(F)(F)F)cn1
Cc1cc(C)nc(COc2nccc(-c3noc(n3)C(F)(F)F)c2Cl)n1
Fc1c(OCc2nc(no2)C2CC2)nccc1-c1noc(n1)C(F)(F)F
OC[C@@H]1CCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1 |r|
Fc1cc(ccc1-c1noc(n1)C(F)(F)F)N1[C@H](CN2CCOCC2)CCC1=O |r|
FC(F)(F)c1nc(no1)-c1ccnc(OCC(=O)N2CCOCC2)c1
FC(F)(F)c1nc(no1)-c1ccc(CNC(=O)C2CCCC2)cc1
CC(C)NC(=O)OCc1ccc(cn1)-c1noc(n1)C(F)(F)F |$;;;HN;;;;;;;;;;;;;;;;;;;$|
Fc1ccc2NC(=O)C(Cc3ccc(cc3)-c3noc(n3)C(F)(F)F)c2c1
CNC(=O)OCc1ccc(cn1)-c1noc(n1)C(F)(F)F |$;HN;;;;;;;;;;;;;;;;;;;$|
FC(F)(F)c1nc(no1)-c1ccc(COC(=O)NC2CCOCC2)nc1 |$;;;;;;;;;;;;;;;;;HN;;;;;;;;$|
CN(C(=O)[C@@H]1COCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1)C(C)(C)C |r|
Fc1cc(ccc1-c1noc(n1)C(F)(F)F)N1[C@@H](CCC1=O)C(=O)OCCOCCCl |r|
COC(=O)N1CCC(CC1)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CC(C(=O)N2CCS(=O)CC2)c2cccc(c2)C(F)(F)F)nc1
FC(F)(F)c1nc(no1)-c1ccnc(OCc2nc3ccccc3[nH]2)c1 |$;;;;;;;;;;;;;;;;;;;;;;;;HN;$|
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)C2CCS(=O)(=O)CC2)c2ccccc2C(F)(F)F)nc1
Cc1ccncc1COc1ccc(cn1)-c1noc(n1)C(F)(F)F
CC(Oc1cc(ccn1)-c1noc(n1)C(F)(F)F)c1nc2ccccc2[nH]1
FC(F)(F)c1nc(no1)-c1ccc(CNC(=O)c2cc(ccn2)N2CCOCC2)cc1
Oc1cccc(c1)C(=O)NCc1ccc(cc1)-c1noc(n1)C(F)(F)F
CCn1cc(COc2cc(ccn2)-c2noc(n2)C(F)(F)F)c(C)n1
FC(F)(F)c1nc(no1)-c1ccnc(OCc2ccno2)c1
FC(F)(F)c1nc(no1)-c1ccnc(OCc2c(Cl)nc3sccn23)c1
FC(F)(F)c1nc(no1)-c1ccnc(OCc2cnn3CCCOc23)c1
FC(F)(F)c1nc(no1)-c1ccnc(OCc2cc3OCCCn3n2)c1
Cc1cc(C)nc(COc2cc(ccn2)-c2noc(n2)C(F)(F)F)c1
FC(F)(F)c1nc(no1)-c1ccnc(OCc2ccnn2-c2cccnc2)c1
Cc1cnc(COc2cc(ccn2)-c2noc(n2)C(F)(F)F)cn1
FC(F)(F)c1nc(no1)-c1ccnc(OCc2cnc(Cl)cn2)c1
FC(F)(F)c1nc(no1)-c1ccnc(OCc2cncc(Cl)n2)c1
FC(F)(F)c1nc(no1)-c1ccnc(OCc2cncc(n2)N2CCNCC2)c1
FC(F)(F)c1nc(no1)-c1ccnc(OCc2ncccc2Cl)c1
FC(F)Cn1nc(COc2cc(ccn2)-c2noc(n2)C(F)(F)F)cc1C1CC1
FC(F)(F)Cn1nc(COc2cc(ccn2)-c2noc(n2)C(F)(F)F)cc1C1CC1
Cc1cc(COc2cc(ccn2)-c2noc(n2)C(F)(F)F)nn1CC(F)F
Cn1nccc1COc1cc(ccn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccnc(OCc2ccn(n2)C2CC2)c1
CC(C)n1ccc(COc2cc(ccn2)-c2noc(n2)C(F)(F)F)n1
Cn1nc(COc2cc(ccn2)-c2noc(n2)C(F)(F)F)cc1C(C)(C)C
Cc1nc(COc2cc(ccn2)-c2noc(n2)C(F)(F)F)no1
FC(F)(F)c1nc(no1)-c1ccnc(OC2CCCc3ccc(Cl)nc23)c1
Fc1cc(COc2cccc3[nH]nnc23)ccc1-c1noc(n1)C(F)(F)F
Fc1cc(COc2nncc3ccccc23)ccc1-c1noc(n1)C(F)(F)F
Cn1nccc1OCc1ccc(-c2noc(n2)C(F)(F)F)c(F)c1
Fc1cnc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)nc1
Fc1cc(COc2cccc3C(=O)NCCc23)ccc1-c1noc(n1)C(F)(F)F
Fc1cc(COc2cc[nH]n2)ccc1-c1noc(n1)C(F)(F)F
Cn1cccc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)c1=O
Fc1cc(COc2ccc3cnccc3n2)ccc1-c1noc(n1)C(F)(F)F
Cn1c(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)nc2ccccc12
Fc1cc(COc2cncnc2)ccc1-c1noc(n1)C(F)(F)F
Cc1cc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)cc(C)n1
Cn1c(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)nc2cccnc12
COc1cnnc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)c1
Fc1cc(COc2ccc3ncnn3c2)ccc1-c1noc(n1)C(F)(F)F
Cc1nccc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)n1
FC(F)c1cc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)ncn1
COc1ccc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)nc1
Cc1cncnc1OCc1ccc(-c2noc(n2)C(F)(F)F)c(F)c1
Fc1cc(COc2cnc3COCc3c2)ccc1-c1noc(n1)C(F)(F)F
COc1ncccc1OCc1ccc(-c2noc(n2)C(F)(F)F)c(F)c1
Fc1cc(COc2nc[nH]n2)ccc1-c1noc(n1)C(F)(F)F
Cc1nc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)c2cnn(C)c2n1
Fc1cc(COc2[nH]nc3CCOCc23)ccc1-c1noc(n1)C(F)(F)F
Fc1ccccc1OCc1cc(ccn1)-c1noc(n1)C(F)(F)F
Fc1ccccc1OCc1ccc(cn1)-c1noc(n1)C(F)(F)F
Nc1cccnc1COCc1ccc(-c2noc(n2)C(F)(F)F)c(F)c1
Cc1ccc(NCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)cn1
Fc1cc(CNc2ccc3ccncc3c2)ccc1-c1noc(n1)C(F)(F)F
Cn1cnc2cc(COc3nccc(-c4noc(n4)C(F)(F)F)c3Cl)ccc12
CC(Oc1nccc(-c2noc(n2)C(F)(F)F)c1Cl)c1cccnc1
Fc1cc(COc2cccnn2)ccc1-c1noc(n1)C(F)(F)F
COc1cncc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)c1
Fc1cc(COc2cnc3[nH]ccc3c2)ccc1-c1noc(n1)C(F)(F)F
Fc1ccc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)cn1
Fc1ccc2ccc(OCc3ccc(-c4noc(n4)C(F)(F)F)c(F)c3)nc2n1
Fc1cc(COc2nnnc3ccccc23)ccc1-c1noc(n1)C(F)(F)F
Cc1ccc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)nn1
NC(=O)c1cccc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)c1
Fc1cc(COc2cccc3CCNCc23)ccc1-c1noc(n1)C(F)(F)F
Cc1ccnnc1OCc1ccc(-c2noc(n2)C(F)(F)F)c(F)c1
NCc1cccc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)c1
Fc1cc(COc2nccc3nccn23)ccc1-c1noc(n1)C(F)(F)F
Cc1cncc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)c1
NCc1ccccc1OCc1ccc(-c2noc(n2)C(F)(F)F)c(F)c1
Fc1cc(COc2cccc3[nH]ncc23)ccc1-c1noc(n1)C(F)(F)F
Fc1cc(COc2nc3cccnc3n2C2CC2)ccc1-c1noc(n1)C(F)(F)F
Cn1c(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)nc2ncccc12
Cc1ncc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)cn1
COc1ccc2cc(OCc3ccc(-c4noc(n4)C(F)(F)F)c(F)c3)nnc2c1
Fc1cc(COc2cnc(nc2)C2CC2)ccc1-c1noc(n1)C(F)(F)F
Fc1cc(COc2nc3ncccc3n2CC(F)(F)F)ccc1-c1noc(n1)C(F)(F)F
Fc1cc(COc2nc3cccnc3n2CC(F)(F)F)ccc1-c1noc(n1)C(F)(F)F
COc1ncc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)cn1
Fc1cc(COc2nnc(o2)C2CC2)ccc1-c1noc(n1)C(F)(F)F
Cc1csc(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)n1
Fc1cc(COc2ccc3cccc(F)c3n2)ccc1-c1noc(n1)C(F)(F)F
Fc1cc(F)c(OCc2ccc(-c3noc(n3)C(F)(F)F)c(F)c2)cn1
CNC(=O)c1ccccc1OCc1ccc(-c2noc(n2)C(F)(F)F)c(F)c1
Fc1cc(COc2ccc3cncnc3c2)ccc1-c1noc(n1)C(F)(F)F
Fc1cc(COc2cccc(Cl)n2)ccc1-c1noc(n1)C(F)(F)F
Fc1cc(COc2cncc(Cl)c2)ccc1-c1noc(n1)C(F)(F)F
Fc1cc(COc2ccc(Cl)nc2)ccc1-c1noc(n1)C(F)(F)F
Cn1ccc(COc2nccc(-c3noc(n3)C(F)(F)F)c2Cl)n1
Cc1cnc(COc2nccc(-c3noc(n3)C(F)(F)F)c2Cl)cn1
Fc1cccnc1COc1nccc(-c2noc(n2)C(F)(F)F)c1Cl
Cc1ncc(COc2nccc(-c3noc(n3)C(F)(F)F)c2Cl)c(C)n1
Cn1cc(COc2nccc(-c3noc(n3)C(F)(F)F)c2Cl)nn1
FC(F)(F)c1nc(no1)-c1ccnc(OCc2nccnc2Cl)c1Cl
FC(F)(F)c1nc(no1)-c1ccnc(OCc2ncccc2Cl)c1Cl
FC(F)(F)c1nc(no1)-c1ccc(COc2nc(no2)C2CC2)nc1
FC(F)(F)c1nc(no1)-c1ccc(COc2cccc3[nH]nnc23)nc1
FC(F)(F)c1nc(no1)-c1ccc(COc2nncc3ccccc23)nc1
FC(F)(F)c1nc(no1)-c1ccc(COc2cccc3C(=O)NCCc23)nc1
Cn1cccc(OCc2ccc(cn2)-c2noc(n2)C(F)(F)F)c1=O
FC(F)(F)c1nc(no1)-c1ccc(Cn2c3ccncc3ccc2=O)nc1
Cn1c(OCc2ccc(cn2)-c2noc(n2)C(F)(F)F)nc2ccccc12
FC(F)(F)c1nc(no1)-c1ccc(COc2nccc3nccn23)nc1
Cn1c(OCc2ccc(cn2)-c2noc(n2)C(F)(F)F)nc2cccnc12
FC(F)(F)c1nc(no1)-c1ccc(COc2ccc3ncnn3c2)nc1
FC(F)c1cc(OCc2ccc(cn2)-c2noc(n2)C(F)(F)F)ncn1
Cc1cncnc1OCc1ccc(cn1)-c1noc(n1)C(F)(F)F
COc1ncccc1OCc1ccc(cn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(COc2cc(Cl)ncn2)nc1
FC(F)(F)c1nc(no1)-c1ccc(COc2ccc(Cl)nc2)nc1
FC(F)(F)c1nc(no1)-c1ccc(COc2ccc3cnccc3n2)nc1
CC1(C)CC(N(C1=O)c1ccc(cc1F)-c1noc(n1)C(F)(F)F)c1ccccc1
Fc1cc(ccc1N1C(CCC1=O)c1c(F)cccc1F)-c1noc(n1)C(F)(F)F
COc1ccccc1C1CCC(=O)N1c1ccc(cc1F)-c1noc(n1)C(F)(F)F
Fc1ccc2N(Cc3ccc(cc3)-c3noc(n3)C(F)(F)F)C(=O)CCc2c1
Fc1ccc2N(Cc3ccc(cn3)-c3noc(n3)C(F)(F)F)C(=O)CCc2c1
Fc1ccc2CCC(=O)N(Cc3ccc(cc3)-c3noc(n3)C(F)(F)F)c2c1
FC(F)(F)c1nc(no1)-c1ccc(CN2C(=O)CCc3ccc(Br)cc23)cc1
Fc1ccccc1N1C(CCC1=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(Cn2c3cc(Br)ccc3ccc2=O)cc1
Fc1ccc2ccc(=O)n(Cc3ccc(cc3)-c3noc(n3)C(F)(F)F)c2c1
Fc1ccc2CCC(=O)N(Cc3ccc(cn3)-c3noc(n3)C(F)(F)F)c2c1
FC(F)(F)c1nc(no1)-c1ccc(CN2C(=O)CCc3ccccc23)nc1
Fc1cccc(c1)N1C(CCC1=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F
Fc1ccc2ccc(OCc3ccc(cn3)-c3noc(n3)C(F)(F)F)nc2c1
Fc1ccc2CCN(Cc3ccc(cn3)-c3noc(n3)C(F)(F)F)C(=O)c2c1
FC(F)(F)c1nc(no1)-c1ccc(CN2C(=O)CCc3ncccc23)nc1
FC(F)(F)c1nc(no1)-c1ccc(CN2C(=O)CCc3cccnc23)nc1
CC(C)(C)OC(=O)[C@@H]1CCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1 |r|
Fc1cc(ccc1-c1noc(n1)C(F)(F)F)N1[C@@H](COC1=O)c1ccccc1 |r|
Cc1noc(n1)[C@@H]1CCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1 |r|
Fc1cc(-c2noc(n2)C(F)(F)F)c(F)cc1N1[C@@H](CCC1=O)C(=O)N1CCCc2ccccc12 |r|
Fc1cc(-c2noc(n2)C(F)(F)F)c(F)cc1N1[C@@H](CCC1=O)C(=O)N1CCc2ccccc2C1 |r|
Fc1cc(-c2noc(n2)C(F)(F)F)c(F)cc1N1[C@@H](CCC1=O)C(=O)N1CCCC1 |r|
FC(F)(F)c1nc(no1)-c1ccc(nc1)N1C(CNC1=O)c1ccccc1
CC1(C)CCCN1C(=O)[C@@H]1CCC(=O)N1c1cc(F)c(cc1F)-c1noc(n1)C(F)(F)F |r|
CN(C(=O)[C@@H]1CCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1)C(C)(C)C |r|
Fc1cc(-c2noc(n2)C(F)(F)F)c(F)cc1N1[C@@H](CCC1=O)C(=O)N1CCC1 |r|
CC1(C)CCCN1C(=O)[C@@H]1CCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1 |r|
CC1(C)CCCCN1C(=O)[C@@H]1CCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1 |r|
CC1(C)COCCN1C(=O)[C@@H]1CCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1 |r|
CC1(C)N(CCNC1=O)C(=O)[C@@H]1CCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1 |r|
CC1(Cc2ccc(cc2)-c2noc(n2)C(F)(F)F)C(=O)Nc2ccc(F)cc12
Fc1ccc2OCCN(Cc3ccc(cn3)-c3noc(n3)C(F)(F)F)c2c1
Cc1cccc(c1)N1CCC(CC1)NCc1ccc(cc1)-c1noc(n1)C(F)(F)F
Cc1nc2CCC(Cc2c(=O)[nH]1)NCc1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CNC2CCc3ncccc3C2)cc1
Cc1ccc2c3CC(CCc3nn2c1)NCc1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CNC2CCc3[nH]nc(c3C2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(CNC2CCN(C2)c2ncccn2)cc1
CN1Cc2ccc(NCc3ccc(cn3)-c3noc(n3)C(F)(F)F)cc2C1=O
FC(F)(F)c1nc(no1)-c1ccc(CNc2ccc3nccn3c2)nc1
Cn1ccc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)cc1=O
Cc1ccc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)cn1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cccc(c2)-c2cnco2)nc1
OCc1cc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)ccc1F
Cc1ccc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)nn1
COc1ccc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)cn1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cccc(c2)-n2cncn2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cc3ccccn3n2)nc1
Cn1ncc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)n1
OCc1ccnc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)c1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cnccn2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cncnc2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2ccc3ccncc3c2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNC2CCc3ncccc3C2)nc1
Cc1n[nH]c2CCC(Cc12)NCc1ccc(cn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CNC2c3ccccc3CCNC2=O)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNC2CCC(=O)Nc3ccccc23)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNC2Cc3ccccc3NC2=O)nc1
FC(F)(F)c1nc(no1)-c1ccc(CN[C@H]2CC[C@]3(CC2)NC(=O)NC3=O)nc1 |r,wU:15.15,18.22,(10.1,-.49,;8.61,-.89,;8.21,-2.37,;9.7,-1.97,;7.52,.2,;6.06,-.27,;5.15,.97,;6.06,2.22,;7.52,1.74,;3.61,.97,;2.84,-.36,;1.3,-.36,;.53,.97,;-1.01,.97,;-1.78,-.36,;-3.32,-.36,;-4.09,-1.69,;-5.63,-1.69,;-6.4,-.36,;-5.63,.97,;-4.09,.97,;-7.3,-1.61,;-8.77,-1.13,;-10.1,-1.9,;-8.77,.41,;-7.3,.89,;-6.9,2.37,;1.3,2.31,;2.84,2.31,)|
FC(F)(F)c1nc(no1)-c1ccc(CNC2CCCCNC2=O)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNC2Cc3ccccc3C2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNC2CCN(CC2)c2ccccn2)nc1
Cc1cc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)on1
FC(F)(F)c1nc(no1)-c1ccc(CNc2ccccn2)cc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cccnc2)cc1
Fc1ccccc1NCc1ccc(cc1)-c1noc(n1)C(F)(F)F
Fc1ccc(NCc2ccc(cc2)-c2noc(n2)C(F)(F)F)cc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2ncccn2)cc1
Cn1nccc1CCOc1cc(ccn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(Cn2c3cc(ccc3ccc2=O)C(F)(F)F)nc1
CC(C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1)n1cccn1
CC(C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1)n1ccnc1C
CC(C)(C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1)n1cccn1
CC(C)(C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1)n1cncn1
Cc1n[nH]c(CC(=O)N(Cc2ccc(cn2)-c2noc(n2)C(F)(F)F)c2cccc(F)c2)n1
Cc1ncc(CC(=O)N(Cc2ccc(cn2)-c2noc(n2)C(F)(F)F)c2cccc(F)c2)s1
Cc1nnc(CC(=O)N(Cc2ccc(cn2)-c2noc(n2)C(F)(F)F)c2cccc(F)c2)s1
Cc1noc(CC(=O)N(Cc2ccc(cn2)-c2noc(n2)C(F)(F)F)c2cccc(F)c2)n1
Fc1cccc(c1)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)C(=O)Cc1[nH]nc2ccccc12
Fc1cccc(c1)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)C(=O)CC1CCS(=O)(=O)C1
CC(C)c1ncncc1C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
Cc1ccc(nn1)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
Cc1ncc(cn1)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
CN1CC(CCC1=O)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
CN1CCC(C1)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
CS(=O)(=O)N1CC(C1)C(=O)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(F)c1
Fc1cccc(c1)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)C(=O)C1CCCS(=O)(=O)C1
Fc1cccc(c1)N(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)C(=O)C1CCN(CC1)C1CC1
COc1cccc(NCc2ccc(cc2)-c2noc(n2)C(F)(F)F)c1
NC(=O)c1ccc(NCc2ccc(cc2)-c2noc(n2)C(F)(F)F)cc1
NC(=O)c1ccccc1NCc1ccc(cc1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CNc2ccc(cc2)C#N)cc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2ccc3c[nH]nc3c2)cc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cccc(c2)C#N)cc1
OCc1cccc(NCc2ccc(cc2)-c2noc(n2)C(F)(F)F)c1
Fc1cccc(NCc2ccc(cc2)-c2noc(n2)C(F)(F)F)c1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cccc3[nH]ncc23)cc1
OCCn1cc2cc(NCc3ccc(cc3)-c3noc(n3)C(F)(F)F)ccc2n1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cnccn2)cc1
OCc1ccnc(NCc2ccc(cc2)-c2noc(n2)C(F)(F)F)n1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cncnc2)cc1
COCc1cc(=O)n(Cc2ccc(cn2)-c2noc(n2)C(F)(F)F)c2ccccc12
COCc1cc(OCc2ccc(cn2)-c2noc(n2)C(F)(F)F)nc2ccccc12
FC(F)(F)c1nc(no1)-c1ccc(cc1)N1C(CN(CC2CCOCC2)C1=O)c1ccccc1
FC(F)(F)c1nc(no1)-c1ccnc(OC[C@@H]2C[C@@H]2c2ncccn2)c1 |r|
CCn1cc(CCCOc2cc(ccn2)-c2noc(n2)C(F)(F)F)cn1
Cn1cc(CCCOc2cc(ccn2)-c2noc(n2)C(F)(F)F)cn1
FC(COc1cc(ccn1)-c1noc(n1)C(F)(F)F)CN1CCOCC1
COCCN1Cc2ccccc2N(Cc2ccc(cn2)-c2noc(n2)C(F)(F)F)C1=O
FC(F)(F)c1nc(no1)-c1ccc(CNc2[nH]nc3ccccc23)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2c[nH]nn2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cc[nH]n2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cnsc2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cnoc2)nc1
CC(C)N1CCC(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)C1=O
C[Si]1(C)CCC(CC1)NCc1ccc(cn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CNC2CCNC(=O)C2)nc1
CN(C)C(=O)c1cccc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)c1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cccc(c2)C(=O)N2CCCC2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cccc(c2)C(=O)Nc2ccccc2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2cccc(c2)C(=O)NCc2ccccn2)nc1
NC(=O)c1ccnc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)c1
CC(C)NC(=O)c1ccccc1NCc1ccc(cn1)-c1noc(n1)C(F)(F)F
CNC(=O)c1ccccc1NCc1ccc(cn1)-c1noc(n1)C(F)(F)F
NC(=O)c1ncccc1NCc1ccc(cn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CNc2ccccc2C(=O)NC2CC2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2ccccc2C(=O)Nc2ccccc2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNc2ccccc2C(=O)NCc2ccccc2)nc1
NC(=O)c1cccc(NCc2ccc(cn2)-c2noc(n2)C(F)(F)F)c1
FC(F)(F)c1nc(no1)-c1ccc(CNC[C@@H]2COCC(=O)N2)nc1 |r|
FC(F)(F)c1nc(no1)-c1ccc(CNC[C@H]2COCC(=O)N2)nc1 |r|
CN1CCOC(CNCc2ccc(cn2)-c2noc(n2)C(F)(F)F)C1
FC(F)(F)c1nc(no1)-c1ccc(CNCC2CN(Cc3ccccc3)CCO2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CNCC2CN(CCO2)c2ccccc2)nc1
CC(=O)N1CCC(CNCc2ccc(cn2)-c2noc(n2)C(F)(F)F)CC1
FC(F)(F)c1nc(no1)-c1ccc(CN(C(=O)C2CCS(=O)(=O)CC2)c2cccc(c2)C(F)(F)F)nc1
FC(F)(F)c1nc(no1)-c1ccc(COc2ncccn2)cc1
FC(F)(F)c1nc(no1)-c1ccc(CNC2CCCNC2=O)nc1
NC(=O)c1cccc(CCOc2cc(ccn2)-c2noc(n2)C(F)(F)F)c1
FC(F)(F)c1nc(no1)-c1ccc(Cn2c3ccccc3ccc2=O)nc1
FC(F)(F)c1nc(no1)-c1ccc(COc2ccc3ccccc3n2)nc1
FC(F)(F)c1nc(no1)-c1ccc(CN2C(=O)COc3ccccc23)nc1
FC(F)(F)c1nc(no1)-c1ccc(CN2C(=O)CSc3ccccc23)nc1
FC(F)(F)c1nc(no1)-c1ccc(CN2C(=O)CCc3cc(ccc23)C(F)(F)F)nc1
Cc1nc2ccc(F)cc2n1Cc1ccc(cn1)-c1noc(n1)C(F)(F)F
Cc1nc2cc(F)ccc2n1Cc1ccc(cn1)-c1noc(n1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(Cn2c3ccccc3ncc2=O)nc1
CC(C)(C)OC(=O)C1COCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1
FC(F)(F)c1nc(no1)-c1ccc(Cn2c3ccccc3[nH]c(=O)c2=O)nc1
FC(F)(F)c1nc(no1)-c1cnc(CN(C(=O)C2CCS(=O)(=O)CC2)c2cccc(c2)C(F)(F)F)cn1
CC(C)(C)OC(=O)[C@@H]1COCC(=O)N1c1ccc(-c2noc(n2)C(F)(F)F)c(F)c1 |r|
COC(=O)N1CC(=O)N(Cc2ccc(cn2)-c2noc(n2)C(F)(F)F)c2ccccc12
FC(F)(F)c1nc(no1)-c1cnc(COc2ccc3ccccc3n2)nc1
FC(F)(F)c1nc(no1)-c1cnc(Cn2c3ccccc3ccc2=O)nc1
FC(F)(F)c1nc(no1)-c1ccc(CN2C(=O)CCc3cccc(c23)C(F)(F)F)nc1
COCc1cccc(CCOc2cc(ccn2)-c2noc(n2)C(F)(F)F)c1
FC(F)(F)c1nc(no1)-c1ccc(CC(NC(=O)C2CCS(=O)(=O)CC2)c2cccc(c2)C(F)(F)F)nc1
CC(C)C(=O)NC(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
CCCC(=O)NC(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
COCC(=O)NC(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
CC(C)(C)CC(=O)NC(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
CC1(COC1)C(=O)NC(Cc1ccc(cn1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CC(NC(=O)C2CCOCC2)c2cccc(c2)C(F)(F)F)nc1
FC(F)(F)c1nc(no1)-c1ccc(CC(NC(=O)c2ncccn2)c2cccc(c2)C(F)(F)F)nc1
FC(F)(F)c1nc(no1)-c1ccc(CC(NC(=O)CN2CCOCC2)c2cccc(c2)C(F)(F)F)nc1
FC(F)(F)c1nc(no1)-c1ccc(CC(NC(=O)c2ccccc2)c2cccc(c2)C(F)(F)F)nc1
FC(F)(F)c1nc(no1)-c1ccc(CC(NC(=O)c2cccnc2)c2cccc(c2)C(F)(F)F)nc1
FC(F)(F)c1nc(no1)-c1ccc(CC(NC(=O)c2ccccn2)c2cccc(c2)C(F)(F)F)nc1
Fc1cc(CN(C(=O)C2CCS(=O)(=O)CC2)c2cccc(c2)C(F)(F)F)ccc1-c1noc(n1)C(F)(F)F
Fc1cc(ccc1CN(C(=O)C1CCS(=O)(=O)CC1)c1cccc(c1)C(F)(F)F)-c1noc(n1)C(F)(F)F
CCS(=O)(=O)N(Cc1ccc(cc1)-c1noc(n1)C(F)(F)F)c1cccc(c1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1ccc(CN(c2cccc(c2)C(F)(F)F)S(=O)(=O)C2CCS(=O)(=O)C2)cc1
Cc1nc2c(F)cc(-c3nc(Nc4ccc(CN5CCN(CCCCCCC(=O)NO)CC5)cn4)ncc3F)cc2n1C(C)C
Cc1nc2c(F)cc(-c3nc(Nc4ccc(N(C)CCN(C)c5ncc(C(=O)NO)cn5)cn4)ncc3F)cc2n1C(C)C
Cc1nc2c(F)cc(-c3nc(Nc4ccc(N(C)CCCCCCC(=O)NO)cn4)ncc3F)cc2n1C(C)C
Cc1nc2c(F)cc(-c3nc(Nc4ccc(C(=O)NO)cn4)ncc3F)cc2n1C(C)C
Cc1nc2c(F)cc(-c3nc(Nc4ccc(/C=C/C(=O)NO)cn4)ncc3F)cc2n1C(C)C
Cc1nc2c(F)cc(-c3nc(Nc4ccc(N(C)Cc5ccc(/C=C/C(=O)NO)cc5)cn4)ncc3F)cc2n1C(C)C
Cc1nc2c(F)cc(-c3nc(Nc4ccc(N(C)Cc5ccc(/C=C/C(=O)NO)cc5)cn4)ncc3F)cc2n1C(C)C
Cc1nc2c(F)cc(-c3nc(Nc4ccc(N5CCN(Cc6ccc(C(=O)NO)cc6)CC5)cn4)ncc3F)cc2n1C(C)C
Cc1nc2c(F)cc(-c3nc(Nc4ccc(N5CCN(CCCCCCC(=O)NO)CC5)cn4)ncc3F)cc2n1C(C)C
Cc1nc2c(F)cc(-c3nc(Nc4ccc(N5CCN(C(=O)CCCCCCC(=O)NO)CC5)cn4)ncc3F)cc2n1C(C)C
Cc1nc2c(F)cc(-c3nc(Nc4ccc(C(=O)NO)nc4)ncc3F)cc2n1C(C)C
Cc1nc2c(F)cc(-c3nc(Nc4cc(C(=O)NO)ccn4)ncc3F)cc2n1C(C)C
Cc1nc2c(F)cc(-c3nc(Nc4ccc(N5CCN(CCCCC(=O)NO)CC5)cn4)ncc3F)cc2n1C(C)C
Cc1nc2c(F)cc(-c3nc(Nc4ccc(N5CCN(CCC(=O)NO)CC5)cn4)ncc3F)cc2n1C(C)C
Cc1nc2c(F)cc(-c3nc(Nc4ccc(N5CCC(C(=O)NO)CC5)cn4)ncc3F)cc2n1C(C)C
Cc1nc2c(F)cc(-c3nc(Nc4ccc(-c5ccc(C(=O)NO)cn5)cn4)ncc3F)cc2n1C(C)C
ONC(=O)c1ccc(CN2CCN(CC2)c2ccc(Nc3nc(cn4ccnc34)-c3ccc4cn[nH]c4c3)cc2)cc1
ONC(=O)CCCCCCC(=O)N1CCN(CC1)c1ccc(Nc2nc(cn3ccnc23)-c2ccc3cn[nH]c3c2)cc1
CN(Cc1ccc(cc1F)C(=O)NO)CC23CC4CC(C2)CC(C4)C3
CN(c1ncc(cn1)C(=O)NO)C12CC3CC(CC(C3)C1)C2 |TLB:21:12:19:15.16.17,1:12:15:18.19.17,THB:21:16:19:20.13.12,20:18:15:21.13.12,20:12:15:18.19.17|
ONC(=O)c1ccc(CNCC23CC4CC(CC(C4)C2)C3)cc1F |TLB:20:11:18:14.15.16,THB:20:15:18:11.19.12,19:11:14:18.17.16,19:17:14:11.20.12,10:11:18:14.15.16|
ONC(=O)c1cc(F)c(CNCC23CC4CC(CC(C4)C2)C3)c(F)c1 |TLB:21:12:19:15.16.17,THB:21:16:19:12.20.13,20:12:15:19.18.17,20:18:15:12.21.13,11:12:19:15.16.17|
ONC(=O)c1ccc(CNCC23CC4CC(CC(C4)C2)C3)c(c1)C(F)(F)F |TLB:20:11:18:14.15.16,THB:20:15:18:11.19.12,19:11:14:18.17.16,19:17:14:11.20.12,10:11:18:14.15.16|
Cc1cc(ccc1CNCC12CC3CC(CC(C3)C1)C2)C(=O)NO |TLB:19:10:17:13.14.15,THB:19:14:17:10.18.11,18:10:13:17.16.15,18:16:13:10.19.11,9:10:17:13.14.15|
CN(Cc1ccc(cc1)C(=O)NO)CC12CC3CC(CC(C3)C1)C2 |TLB:23:14:21:17.18.19,THB:23:18:21:14.22.15,22:14:17:21.20.19,22:20:17:14.23.15,13:14:21:17.18.19|
ONC(=O)c1ccc(CNCC23CC4CC(CC(C4)C2)C3)nc1 |TLB:20:11:18:14.15.16,THB:20:15:18:11.19.12,19:11:14:18.17.16,19:17:14:11.20.12,10:11:18:14.15.16|
ONC(=O)c1ccc(CNCC23CC4CC(CC(C4)C2)C3)c(Cl)c1 |TLB:20:11:18:14.15.16,THB:20:15:18:11.19.12,19:11:14:18.17.16,19:17:14:11.20.12,10:11:18:14.15.16|
ONC(=O)c1ccc(CNCC23CC4CC(CC(C4)C2)C3)c(Br)c1 |TLB:20:11:18:14.15.16,THB:20:15:18:11.19.12,19:11:14:18.17.16,19:17:14:11.20.12,10:11:18:14.15.16|
ONC(=O)c1ccc(CNCC23CC4CC(CC(C4)C2)C3)c(F)c1 |TLB:20:11:18:14.15.16,THB:20:15:18:11.19.12,19:11:14:18.17.16,19:17:14:11.20.12,10:11:18:14.15.16|
ONC(=O)c1ccc(CNCC23CC4CC(CC(C4)C2)C3)cc1 |TLB:20:11:18:14.15.16,THB:20:15:18:11.19.12,19:11:14:18.17.16,19:17:14:11.20.12,10:11:18:14.15.16|
ONC(=O)c1ccc(CNC23CC4CC(CC(C4)C2)C3)cc1 |TLB:9:10:13:17.16.15,9:10:17:13.14.15,19:10:17:13.14.15,THB:18:10:13:17.16.15,18:16:13:10.19.11,19:14:17:10.18.11|
CC(NCc1ccc(cc1)C(=O)NO)C12CC3CC(CC(C3)C1)C2 |TLB:23:14:21:17.18.19,THB:23:18:21:14.22.15,22:14:17:21.20.19,22:20:17:14.23.15,1:14:21:17.18.19|
CC(N(C)Cc1ccc(cc1)C(=O)NO)C12CC3CC(CC(C3)C1)C2 |TLB:24:15:22:18.19.20,THB:24:19:22:15.23.16,23:15:18:22.21.20,23:21:18:15.24.16,1:15:22:18.19.20|
CCC(NCc1ccc(cc1)C(=O)NO)C12CC3CC(CC(C3)C1)C2 |TLB:24:15:22:18.19.20,THB:24:19:22:15.23.16,23:15:18:22.21.20,23:21:18:15.24.16,2:15:22:18.19.20|
CCC(N(C)Cc1ccc(cc1)C(=O)NO)C12CC3CC(CC(C3)C1)C2 |TLB:25:16:23:19.20.21,THB:25:20:23:16.24.17,24:16:19:23.22.21,24:22:19:16.25.17,2:16:23:19.20.21|
CC1(C)C2CC1C(CNCc1ccc(cc1)C(=O)NO)CC2
CCCCCN(CC1CCC2CC1C2(C)C)Cc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(CNCC2CCCCC2)cc1
CC(=O)c1c(C)c2cnc(Nc3ccc(cn3)N3CCN(CC3)C(=O)CCCCCCC(=O)NO)nc2n(C2CCCC2)c1=O
CC(=O)c1c(C)c2cnc(Nc3ccc(cn3)N3CCN(CCCCCCC(=O)NO)CC3)nc2n(C2CCCC2)c1=O
CC(=O)c1c(C)c2cnc(Nc3ccc(cn3)N3CCN(CCCCCCCC(=O)NO)CC3)nc2n(C2CCCC2)c1=O
CC(=O)c1c(C)c2cnc(Nc3ccc(cn3)N3CCN(Cc4ccc(cc4)C(=O)NO)CC3)nc2n(C2CCCC2)c1=O
CC(=O)c1c(C)c2cnc(Nc3ccc(cn3)C(=O)NO)nc2n(C2CCCC2)c1=O
CC(=O)c1c(C)c2cnc(Nc3ccc(cn3)C(=O)NCCCCCCC(=O)NO)nc2n(C2CCCC2)c1=O
ONC(=O)c1ccc(Nc2nc3ccccc3n2CC2CCCCC2)cc1
ONC(=O)c1ccc(Nc2nc3ccccc3n2C2CCCCC2)cc1
ONC(=O)c1ccc(Nc2nc3ccccc3n2C2CCCCCC2)cc1
CN1CCN(CC1)c1ccc(cn1)C(=O)Nc1nc(ccc1N)-c1ccc(F)cc1
Nc1ccc(nc1NC(=O)c1ccc(nc1)N1CCNCC1)-c1ccc(F)cc1
NC1CCN(CC1)c1ccc(cn1)C(=O)Nc1nc(ccc1N)-c1ccc(F)cc1
CN1CCN(CC1)c1ccc(cn1)C(=O)Nc1nc(ccc1N)-c1cccs1
ONC(=O)\C=C\c1ccc(CNC2CC2c2ccc(cc2)-c2ccc(Cl)cc2)cc1
ONC(=O)\C=C\c1ccc(CNC2CC2c2ccc(cc2)-c2cncnc2)cc1
ONC(=O)c1cnc(nc1)N1CCC(CNC2CC2c2ccc(F)cc2)CC1
ONC(=O)c1cnc(nc1)N1CCC(CC1)NC1CC1c1ccc(OCc2ccc(F)cc2)cc1
ONC(=O)c1cnc(nc1)N1CCC(CNC2CC2c2ccc(cc2)-c2ccc(F)cc2)CC1
ONC(=O)c1cnc(nc1)N1CCC(CNC2CC2c2ccc(cc2)-c2cncnc2)CC1
ONC(=O)c1cnc(nc1)N1CCC(CN[C@@H]2C[C@H]2c2ccc(F)cc2)CC1 |r|
ONC(=O)c1cnc(nc1)N1CCC(CN[C@H]2C[C@@H]2c2ccc(F)cc2)CC1 |r|
ONC(=O)c1ccc(cc1)N1CCC(CNC2CC2c2ccc(F)cc2)CC1
ONC(=O)c1cnc(nc1)N1CCn2cc(CNC3CC3c3ccccc3)nc2C1
ONC(=O)c1cccc(CNC2CC2c2ccccc2)c1
ONC(=O)c1ccc(CNC2CC2c2ccccc2)cc1
ONC(=O)CCCCCNC1CC1c1ccccc1
ONC(=O)c1ccc(CCCNC2CC2c2ccc(F)cc2)cc1
ONC(=O)C1CCC(CC1)NC1CC1c1ccccc1 |(7.44,1.93,;6.1,1.15,;4.77,1.93,;4.77,3.47,;3.44,1.15,;3.44,-.38,;2.1,-1.15,;.77,-.38,;.77,1.15,;2.1,1.93,;-.56,-1.15,;-1.9,-.38,;-2.67,.95,;-3.44,-.38,;-4.77,-1.15,;-6.1,-.38,;-7.44,-1.15,;-7.44,-2.69,;-6.1,-3.47,;-4.77,-2.69,)|
CC(NC1CC1c1ccccc1)[C@H]1CC[C@@H](CC1)C(=O)NO |r,wU:15.20,wD:12.13,(.1,3.08,;.1,1.54,;-1.23,.77,;-2.56,1.54,;-3.33,2.87,;-4.1,1.54,;-5.44,.77,;-6.77,1.54,;-8.11,.77,;-8.11,-.77,;-6.77,-1.54,;-5.44,-.77,;1.44,.77,;1.44,-.77,;2.77,-1.54,;4.1,-.77,;4.1,.77,;2.77,1.54,;5.44,-1.54,;5.44,-3.08,;6.77,-.77,;8.11,-1.54,)|
Cn1cc(ccc1=O)-c1ccc(cc1)C1CC1NCC1CCN(Cc2ccc(cc2)C(=O)NO)CC1
ONC(=O)c1ccc(CN2CCC(CNC3CC3c3ccccc3)CC2)cc1
Cc1noc(C)c1-c1ccc(cc1)C1CC1NCC1CCN(Cc2ccc(cc2)C(=O)NO)CC1
ONC(=O)c1ccc(CN2CCC(CNC3CC3c3ccc(cc3)-c3cncnc3)CC2)cc1
Cc1noc(C)c1-c1ccc(cc1)C1CC1NCC1CCN(Cc2ccc(cn2)C(=O)NO)CC1
ONC(=O)c1ccc(Cn2cc(CNC3CC3c3ccccc3)cn2)cc1
ONC(=O)c1ccc(Cn2cc(CNC3CC3c3ccccc3)nn2)cc1
ONC(=O)c1ccc(CCN2CCC(CNC3CC3c3ccccc3)CC2)cc1
ONC(=O)c1ccc(CCCN2CCC(CNC3CC3c3ccccc3)CC2)cc1
ONC(=O)c1ccc(CCCN2CCC(CC2)NC2CC2c2ccccc2)cc1
ONC(=O)c1ccc(CCCN2CC3(CC(C3)NC3CC3c3ccccc3)C2)cc1
ONC(=O)c1ccc(CCCN2CCC(CNC3CC3c3ccc(F)cc3)CC2)cc1
ONC(=O)c1ccc(CCCN2CC(CNC3CC3c3ccc(F)cc3)C2)cc1
ONC(=O)c1ccc(CCCN2CCC(CNC3CC3c3ccc(F)c(F)c3)CC2)cc1
COc1ccc(cc1)C1CC1NCC1CCN(CCCc2ccc(cc2)C(=O)NO)CC1
ONC(=O)c1ccc(CCCN2CCC(CNC3CC3c3ccc(OCc4ccc(F)cc4)cc3)CC2)cc1
ONC(=O)c1ccc(CCCN2CCC(CNC3CC3c3ccc(cc3)C(=O)N3CCOCC3)CC2)cc1
ONC(=O)c1ccc(CCCN2CCC(CNC3CC3c3ccc(cc3)C(=O)N3CCCCC3)CC2)cc1
CN(C)CCNC(=O)c1ccc(cc1)C1CC1NCC1CCN(CCCc2ccc(cc2)C(=O)NO)CC1
ONC(=O)c1ccc(CCCN2CCC(CNC3CC3c3ccc(cc3)-c3ccc(Cl)cc3)CC2)cc1
ONC(=O)c1ccc(CCCN2CCC(CNC3CC3c3ccc(cc3)-c3ccc(F)cc3)CC2)cc1
ONC(=O)c1ccc(CCCN2CC(CNC3CC3c3ccc(cc3)-c3ccc(F)cc3)C2)cc1
ONC(=O)c1ccc(CCCN2CCC(CNC3CC3c3ccc(cc3)-c3ccc(cc3)C#N)CC2)cc1
Cn1ccc(cc1=O)-c1ccc(cc1)C1CC1NCC1CCN(CCCc2ccc(cc2)C(=O)NO)CC1
ONC(=O)c1ccc(CCCN2CCC(CNC3CC3c3ccc(cc3)-c3cncnc3)CC2)cc1
Cn1cc(cn1)-c1ccc(cc1)C1CC1NCC1CCN(CCCc2ccc(cc2)C(=O)NO)CC1
Cn1cc(cn1)-c1ccc(cc1)C1CC1NCC1CN(CCCc2ccc(cc2)C(=O)NO)C1
Cc1noc(C)c1-c1ccc(cc1)C1CC1NCC1CN(CCCc2ccc(cc2)C(=O)NO)C1
Cc1noc(C)c1-c1ccc(cc1)C1CC1NCC1CN(CCCc2cccc(c2)C(=O)NO)C1
ONC(=O)c1ccc(CCCN2CCC(CNC3CC3c3ccc(cc3)-c3ccc(nc3)C(F)(F)F)CC2)cc1
CC(C)n1cc(cn1)C1CC1NCC1CCN(CCCc2ccc(cc2)C(=O)NO)CC1
ONC(=O)c1ccc(CCCN2CCC(CNC3CC3c3cnn(c3)-c3ccccc3)CC2)cc1
COc1ccc(cc1)C1CC1NCc1cn2CCN(CCCc3ccc(cc3)C(=O)NO)Cc2n1
ONC(=O)c1ccc(CCCN2CCn3cc(CNC4CC4c4ccc(F)cc4)nc3C2)cc1
ONC(=O)c1ccc(CCCn2cnc(CNC3CC3c3ccc(F)c(F)c3)c2)cc1
ONC(=O)c1ccc(CCCn2cncc2CNC2CC2c2ccccc2)cc1
ONC(=O)c1ccc(CCCn2cnc(CNC3CC3c3ccccc3)c2)cc1
ONC(=O)c1ccc(CCCn2cc(CNC3CC3c3ccccc3)cn2)cc1
ONC(=O)c1ccc(CCCn2cc(CNC3CC3c3ccccc3)nn2)cc1
ONC(=O)c1ccc(CCCN2CCc3cc(CNC4CC4c4ccc(F)cc4)ccc3C2)cc1
ONC(=O)c1ccc(CN2CCc3ccc(CNC4CC4c4ccc(F)cc4)cc3C2)cc1
ONC(=O)c1ccc(CN2CCn3cc(CNC4CC4c4ccc(F)cc4)nc3C2)cc1
CN1C(=O)C(C)(C)c2cc(ccc12)C1CC1NCC1CCN(CCCc2ccc(cc2)C(=O)NO)CC1
ONC(=O)c1ccc(CCC(=O)N2CCC(CNC3CC3c3ccccc3)CC2)cc1
ONC(=O)c1ccc(CCC(=O)N2CCC(CC2)NC2CC2c2ccccc2)cc1
ONC(=O)c1ccc(CC(=O)N2CCC(CNC3CC3c3ccccc3)CC2)cc1
ONC(=O)c1ccc(CC(=O)N2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 |r|
ONC(=O)c1ccc(CC(=O)N2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 |r|
ONC(=O)c1ccc(cc1)S(=O)(=O)N1CCC(CNC2CC2c2ccccc2)CC1
ONC(=O)c1ccc(CS(=O)(=O)NCCN2CCC(CNC3CC3c3ccccc3)CC2)cc1
ONC(=O)c1ccc(cc1)S(=O)(=O)NCCN1CCC(CNC2CC2c2ccc(F)cc2)CC1
ONC(=O)c1ccc(CCS(=O)(=O)N2CCC(CNC3CC3c3ccccc3)CC2)cc1
ONC(=O)c1ccc(cc1)C(=O)NCCN1CCC(CNC2CC2c2ccccc2)CC1
ONC(=O)c1ccc(cc1)C(=O)NCCN1CCC(CNC2CC2c2ccc(F)c(F)c2)CC1
ONC(=O)c1ccc(CN2CCN(CC2)C(=O)CNC2CC2c2ccccc2)cc1
ONC(=O)c1ccc(CCC(=O)N2CCN(CC2)C(=O)CNC2CC2c2ccccc2)cc1
ONC(=O)c1ccc(CCCC2CCN(CC2)C(=O)CNC2CC2c2ccccc2)cc1
ONC(=O)c1ccc(OCCNC2CC2c2ccccc2)cc1
ONC(=O)c1ccc(OCCN2CCC(CNC3CC3c3ccc(F)cc3)CC2)nc1
ONC(=O)c1ccc(OCCN2CCC(CNC3CC3c3ccccc3)CC2)nc1
ONC(=O)c1ccc(OCCN2CCC(CNC3CC3c3ccc(cc3)-c3ccc(F)cc3)CC2)nc1
ONC(=O)c1ccc(OCCN2CCC(CNC3CC3c3ccccc3)CC2)cc1
ONC(=O)c1ccc(OCCCNC2CC2c2ccccc2)cc1
ONC(=O)c1cnc(NCCN2CCC(CNC3CC3c3ccc(F)cc3)CC2)nc1
ONC(=O)c1cc2CN(CCc2s1)C(=O)CNC1CC1c1ccc(F)cc1
ONC(=O)c1cc2CN(CCc2s1)C(=O)CN[C@@H]1C[C@H]1c1ccc(F)cc1 |r|
ONC(=O)c1cc2CN(CCc2s1)C(=O)CN[C@H]1C[C@@H]1c1ccc(F)cc1 |r|
ONC(=O)c1ccc2CCN(Cc2c1)C(=O)CNC1CC1c1ccc(F)cc1
ONC(=O)c1ccc2CCN(Cc2c1)C(=O)CN[C@H]1C[C@@H]1c1ccc(F)cc1 |r|
ONC(=O)c1ccc2CCN(Cc2c1)C(=O)CN[C@@H]1C[C@H]1c1ccc(F)cc1 |r|
ONC(=O)c1cc2CN(CCc2s1)C(=O)CCCNC1CC1c1ccc(F)cc1
ONC(=O)c1cc2CN(CCc2s1)C(=O)CCCN1CCC(CNC2CC2c2ccc(F)cc2)CC1
ONC(=O)c1ccc2CCN(Cc2c1)C(=O)CCCNC1CC1c1ccc(F)cc1
ONC(=O)c1ccc2CN(Cc2c1)C(=O)CCCNC1CC1c1ccc(F)cc1
ONC(=O)c1ccc2CN(Cc2c1)C(=O)CCCN1CCC(CNC2CC2c2ccccc2)CC1
ONC(=O)c1c[nH]c(CCCN2CCC(CNC3CC3c3ccccc3)CC2)n1
ONC(=O)c1csc(CCCN2CCC(CNC3CC3c3ccc(cc3)-c3ccc(F)cc3)CC2)n1
ONC(=O)c1cnc(CCCN2CCC(CNC3CC3c3ccccc3)CC2)s1
ONC(=O)c1csc(CCCN2CCC(CNC3CC3c3ccccc3)CC2)n1
ONC(=O)c1ccc(\C=C\C(=O)N2CCC(CNC3CC3c3ccccc3)CC2)cc1
ONC(=O)c1ccc(\C=C\C(=O)N2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 |r|
ONC(=O)c1ccc(\C=C\C(=O)N2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 |r|
ONC(=O)c1ccc(\C=C\C(=O)N2CCC(CN[C@H]3C[C@@H]3c3ccc(F)cc3)CC2)cc1 |r|
ONC(=O)c1ccc(\C=C\C(=O)N2CCC(CN[C@@H]3C[C@H]3c3ccc(F)cc3)CC2)cc1 |r|
Cc1noc(C)c1-c1ccc(cc1)C1CC1NCC1CCN(CC1)C(=O)\C=C\c1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(\C=C\C(=O)N2CCC(CNC3CC3c3ccc(cc3)-c3cncnc3)CC2)cc1
ONC(=O)c1ccc(\C=C\C(=O)N2CC(CNC3CC3c3ccc(F)cc3)C2)cc1
Cn1cc(cn1)-c1ccc(cc1)C1CC1NCC1CN(C1)C(=O)\C=C\c1ccc(cc1)C(=O)NO
Nc1ccccc1NC(=O)c1ccc(CCCN2CC3(CC(C3)NC3CC3c3ccccc3)C2)cc1
CC(C)n1cc(cn1)C1CC1NCC1CCN(CCCc2ccc(cc2)C(=O)Nc2ccccc2N)CC1
Nc1ccccc1NC(=O)c1ccc(CCCN2CCC(CNC3CC3c3cnn(c3)-c3ccccc3)CC2)cc1
Nc1ccc(F)cc1NC(=O)c1ccc(CCCN2CCC(CNC3CC3c3ccc(F)cc3)CC2)cc1
Nc1ccccc1NC(=O)c1ccc(CCC(=O)N2CCC(CC2)NC2CC2c2ccccc2)cc1
Nc1ccccc1NC(=O)c1ccc(CCC(=O)N2CCC(CNC3CC3c3ccccc3)CC2)cc1
Nc1ccccc1NC(=O)c1ccc(CCCn2cnc(CNC3CC3c3ccc(F)c(F)c3)c2)cc1
Nc1ccccc1NC(=O)c1ccc(CCCn2cnc(CNC3CC3c3ccccc3)c2)cc1
Nc1ccccc1NC(=O)c1ccc(CCCn2cc(CNC3CC3c3ccccc3)nn2)cc1
Nc1ccccc1NC(=O)c1ccc(CCCn2cc(CNC3CC3c3ccccc3)cn2)cc1
Nc1ccccc1NC(=O)c1ccc(CCN2CCC(CNC3CC3c3ccccc3)CC2)cc1
Nc1ccccc1NC(=O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 |r|
Cn1cc(ccc1=O)-c1ccc(cc1)C1CC1NCC1CCN(Cc2ccc(cc2)C(=O)Nc2ccccc2N)CC1
Cn1cc(cn1)-c1ccc(cc1)C1CC1NCC1CCN(Cc2ccc(cc2)C(=O)Nc2ccccc2N)CC1
Cc1noc(C)c1-c1ccc(cc1)C1CC1NCC1CCN(Cc2ccc(cc2)C(=O)Nc2ccccc2N)CC1
Nc1ccccc1NC(=O)c1ccc(CN2CCC(CNC3CC3c3ccc(cc3)-c3cncnc3)CC2)cc1
Nc1ccccc1NC(=O)c1ccc(Cn2cc(CNC3CC3c3ccccc3)cn2)cc1
Nc1ccccc1NC(=O)c1ccc(Cn2cc(CNC3CC3c3ccccc3)nn2)cc1
Nc1ccccc1NC(=O)c1ccc(CC(=O)N2CCC(CNC3CC3c3ccc(F)cc3)CC2)cc1
Nc1ccccc1NC(=O)c1ccc(OCCNC2CC2c2ccc(F)cc2)cc1
Nc1ccccc1NC(=O)c1ccc(OCCN2CCC(CNC3CC3c3ccc(F)cc3)CC2)nc1
Nc1ccccc1NC(=O)c1cnc(NCCN2CCC(CNC3CC3c3ccc(F)cc3)CC2)nc1
Nc1ccccc1NC(=O)c1cc2CN(CCc2s1)C(=O)CNC1CC1c1ccc(F)cc1
Nc1ccccc1NC(=O)c1ccc2CCN(Cc2c1)C(=O)CNC1CC1c1ccc(F)cc1
Nc1ccccc1NC(=O)c1coc(CCCN2CCC(CNC3CC3c3ccccc3)CC2)n1
Nc1ccccc1NC(=O)c1cnc(CCCN2CCC(CNC3CC3c3ccccc3)CC2)s1
Nc1ccccc1NC(=O)c1ccc(CNC(=O)CNC2CC2c2ccc(F)cc2)cc1
Nc1ccccc1NC(=O)c1ccc(\C=C\C(=O)N2CCC(CNC3CC3c3ccc(F)cc3)CC2)cc1
Nc1ccccc1NC(=O)c1ccc(\C=C\C(=O)N2CC(CNC3CC3c3ccc(F)cc3)C2)cc1
Nc1ccccc1NC(=O)c1ccc(CNC(=O)N2CCC(CNC3CC3c3ccc(F)cc3)CC2)cc1
Nc1ccccc1NC(=O)c1ccc(cc1)S(=O)(=O)N1CCC(CNC2CC2c2ccccc2)CC1
COc1ccc(\C=C\C(=O)NO)c(c1)-c1ccc(Br)cc1
COc1ccc(\C=C\C(=O)NO)c(c1)-c1ccc(cc1)-c1ccccc1
ONC(=O)c1ccc(Cn2c3cc(F)ccc3c(=O)n(CCc3ccccc3)c2=O)cc1
COc1ccc2c(c1)n(Cc1ccc(cc1)C(=O)NO)c(=O)n(CCc1ccccc1)c2=O
ONC(=O)c1ccc(Cn2c3cc(ccc3c(=O)n(CCc3ccccc3)c2=O)C#N)cc1
ONC(=O)c1ccc(Cn2c3cc(O)ccc3c(=O)n(CCc3ccccc3)c2=O)cc1
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3ccccc3)c2=O)cc1
ONC(=O)c1cccc(Cn2c3ccccc3c(=O)n(CCc3ccccc3)c2=O)c1
ONC(=O)c1cccc(Cn2c3cc(ccc3c(=O)n(CCc3ccccc3)c2=O)C#N)c1
ONC(=O)c1ccc(Cn2c3cc(Cl)ccc3c(=O)n(CCc3ccccc3)c2=O)cc1
ONC(=O)c1ccc(Cn2c3ccc(Cl)cc3c(=O)n(CCc3ccccc3)c2=O)cc1
Cn1c(=O)n(Cc2ccc(cc2)C(=O)NO)c2cc(Cl)ccc2c1=O
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(Cc3ccccc3)c2=O)cc1
ONC(=O)c1ccc(Cn2c3ncccc3c(=O)n(CCc3ccccc3)c2=O)cc1
ONC(=O)c1ccc(Cn2c3cc(ccc3c(=O)n(CCc3ccccc3)c2=O)C(F)(F)F)cc1
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3ccc(F)cc3)c2=O)cc1
COc1ccccc1CCn1c(=O)n(Cc2ccc(cc2)C(=O)NO)c2ccccc2c1=O
ONC(=O)c1ccc(Cn2c3ccc(F)cc3c(=O)n(CCc3ccccc3)c2=O)cc1
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3ccccc3O)c2=O)cc1
ONC(=O)c1ccc(Cn2c3sccc3c(=O)n(CCc3ccccc3)c2=O)cc1
Cc1ccc2c(c1)n(Cc1ccc(cc1)C(=O)NO)c(=O)n(CCc1ccccc1)c2=O
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3cccs3)c2=O)cc1
ONC(=O)c1cc(Cn2c3ccccc3c(=O)n(CCc3ccccc3)c2=O)cs1
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3cccc(F)c3)c2=O)cc1
ONC(=O)c1ccc(Cn2c3cc(ccc3c(=O)n(CCc3ccccc3)c2=O)C2CC2)cc1
CNc1ccc(CCn2c(=O)n(Cc3ccc(cc3)C(=O)NO)c3ccccc3c2=O)cc1
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3ccc(cc3)N3CCOCC3)c2=O)cc1
CC1(C)N(Cc2c1cccc2C(=O)NO)c1cnc(cn1)C(F)(F)F
COC(=O)c1cccc2c1CN(c1cnc(cn1)C(F)(F)F)C2(C)C
ONC(=O)c1ccc2CCN(Cc2c1)c1nc2ccccc2[nH]1
ONC(=O)c1cccc2CN(CCc12)c1nc2ccccc2[nH]1
ONC(=O)c1ccc2CN(CCc2c1)c1nc2ccccc2[nH]1
ONC(=O)c1cccc2CCN(Cc12)c1nc2ccccc2[nH]1
ONC(=O)c1cccc2CN(Cc12)c1nc2ccccc2[nH]1
ONC(=O)c1cccc2CCN(CCc12)c1nc2ccccc2[nH]1
Cn1ncc2c(SCC(=O)c3ccc(CNC(=O)C4CC4)s3)ccnc21
O=C(CSc1nc(C(F)(F)F)nc2nn(C3CC3)cc12)c1ccc(CNC(=O)C2CC2(F)F)s1
O=C(CSc1nc(C(F)(F)F)nc2nn(C3CC3)cc12)c1ccc(CNC(=O)C(F)(F)C(F)(F)F)s1
COc1ccc2nc(C)nc(SCC(=O)c3ccc(CNC(=O)CO)s3)c2c1
Cn1cc2c(SCC(=O)c3ccc(CNC(=O)CO)s3)nc(C(F)(F)F)nc2n1
Cc1nc(SCC(=O)c2ccc(CNC(=O)CO)s2)c2cccnc2n1
Cn1cc2c(SCC(=O)c3ccc(CNC(=O)CO)s3)nc(C(F)F)nc2n1
O=C(CO)NCc1ccc(C(=O)CSc2nc3cc(C(F)(F)F)ncc3o2)s1
O=C(CO)NCc1ccc(C(=O)CSc2nc3nc(C(F)(F)F)ccc3o2)s1
Cc1nc(SCC(=O)c2ccc(CNC(=O)CO)s2)c2cc(Cl)c(F)cc2n1
Cn1ncc2c(SCC(=O)c3ccc(CNC(=O)CO)s3)nc(C(F)(F)F)nc21
COc1cc2c(SCC(=O)c3ccc(CNC(=O)CO)s3)nc(C)nc2cc1F
Cc1nc(SCC(=O)c2ccc(CNC(=O)CO)s2)c2cc(C(F)(F)F)ccc2n1
O=C(CO)NCc1ccc(C(=O)CSc2nc(C(F)(F)F)nc3nn(C4CC4)cc23)s1
Cc1nc(SCC(=O)c2ccc(CNC(=O)CO)s2)c2cc(N3CCN(C)CC3)ccc2n1
COc1cc(F)c2nc(C)nc(SCC(=O)c3ccc(CNC(=O)CO)s3)c2c1
COc1ccc2nc(C)nc(SCC(=O)c3ccc(CN(C)C(=O)CO)s3)c2c1
O=C(CO)NCc1ccc(C(=O)CSc2nc(C(F)(F)F)nc3ncccc23)s1
O=C(CSc1nc(C(F)(F)F)nc2ncccc12)c1ccc(CNC(=O)C2CC2(F)F)s1
CN(Cc1ccc(C(=O)CSc2nc(C(F)(F)F)nc3nn(C)cc23)s1)C(=O)CO
O=C(CO)NCc1ccc(C(=O)CSc2nc3ccc(C(F)(F)F)nc3o2)s1
O=C(CO)NCc1ccc(C(=O)CSc2nc3ncc(C(F)(F)F)cc3o2)s1
Cc1nc(SCC(=O)c2ccc(CNC(=O)CO)s2)c2cc(C(F)(F)F)cnc2n1
Cc1nc(SCC(=O)c2ccc(CNC(=O)CO)s2)c2cc(F)cnc2n1
COCCn1ncc2c(SCC(=O)c3ccc(CNC(=O)CO)s3)nc(C(F)(F)F)nc21
Cc1nc(SCC(=O)c2ccc(CNC(=O)CO)s2)c2cc(OC(F)(F)F)ccc2n1
COCCn1cc2c(SCC(=O)c3ccc(CNC(=O)CO)s3)nc(C(F)(F)F)nc2n1
O=C(CO)NCc1ccc(C(=O)CSc2nc(C(F)(F)F)nc3c2cnn3C2CC2)s1
CCn1cc2c(SCC(=O)c3ccc(CNC(=O)CO)s3)nc(C(F)(F)F)nc2n1
O=C(CSc1nc(C(F)(F)F)nc2ncccc12)c1ccc(CN2CCOCC2=O)s1
COc1cnc2nc(C)nc(SCC(=O)c3ccc(CNC(=O)CO)s3)c2c1
Cc1nc(SCC(=O)c2ccc(CNC(=O)CO)s2)c2cc(Cl)cc(F)c2n1
Cc1nc(SCC(=O)c2ccc(CNC(=O)CO)s2)c2cc(N3CC4CCC3CO4)ccc2n1
COc1cc(C(F)(F)F)cc2c(SCC(=O)c3ccc(CNC(=O)CO)s3)nc(C)nc12
O=C(CO)NCc1ccc(C(=O)CSc2nc(C(F)(F)F)nc3cccnc23)s1
Cc1nc(SCC(=O)c2ccc(CNC(=O)CO)s2)c2ncccc2n1
COc1cc2c(SCC(=O)c3ccc(CNC(=O)CO)s3)nc(C(F)(F)F)nc2cn1
COc1ccc2nc(C)nc(SCC(=O)c3ccc(CNC(=O)CO)s3)c2c1F
COc1cc2c(SCC(=O)c3ccc(CN(C)C(=O)CO)s3)nc(C(F)(F)F)nc2cn1
CCOc1cnc2nc(C)nc(SCC(=O)c3ccc(CNC(=O)CO)s3)c2c1
COCC(=O)NCc1ccc(C(=O)CSc2nc(C)nc3ncc(OC)cc23)s1
COc1cnc2nc(C(F)F)nc(SCC(=O)c3ccc(CNC(=O)CO)s3)c2c1
CC(C)c1nc(SCC(=O)c2ccc(CNC(=O)C(C)(C)C)s2)c2ccccc2n1
CC(C)(C)C(=O)NCc1ccc(C(=O)CSc2nc(C3CC3)nc3ccccc23)s1
Cc1nc(SCC(=O)c2ccc(CNC(=O)C(C)(C)C)s2)c2ccccc2n1
COCc1nc(SCC(=O)c2ccc(CNC(=O)C(C)(C)C)s2)c2ccccc2n1
Cc1nc(SCC(=O)c2ccc(CNC(=O)C(C)(C)C)s2)c2cnn(C)c2n1
Cn1ncc2c(SCC(=O)c3ccc(CNC(=O)C(C)(C)C)s3)nc(C3CC3)nc21
Cc1nc(SCC(=O)c2ccc(CNC(=O)C(C)(C)C)s2)c2cccnc2n1
Cc1nc(SCC(=O)c2ccc(CNC(=O)C(C)(C)C)s2)c2ccc(Cl)cc2n1
Cc1nc(SCC(=O)c2ccc(CNC(=O)C(C)(C)C)s2)c2cc(F)ccc2n1
Cc1nc(SCC(=O)c2ccc(CNC(=O)C(C)(C)C)s2)c2ccc(F)cc2n1
Cc1ccc2c(SCC(=O)c3ccc(CNC(=O)C(C)(C)C)s3)nc(C)nc2c1
COc1ccc2c(SCC(=O)c3ccc(CNC(=O)C(C)(C)C)s3)nc(C)nc2c1
Cc1nc(SCC(=O)c2ccc(CNC(=O)C(C)(C)C)s2)c2cccc(F)c2n1
CN(C)c1nc(SCC(=O)c2ccc(CNC(=O)C(C)(C)C)s2)c2ccccc2n1
CC(C)(C)C(=O)NCc1ccc(C(=O)CSc2nc(C(F)F)nc3ccccc23)s1
Cn1ncc2c(SCC(=O)c3ccc(CNC(=O)C(C)(C)C)s3)nc(C(F)(F)F)nc21
Cn1ncc2c(SCC(=O)c3ccc(CNC(=O)C(C)(C)C)s3)nc(C(F)F)nc21
Cc1ccc2oc(SCC(=O)c3ccc(CNC(=O)C(C)(C)C)s3)nc2n1
CC1CCN(Cc2ccc(C(=O)CSc3ncnc4c3cnn4C)s2)C1=O
Cn1ncc2c(SCC(=O)c3ccc(CN4CCCC4=O)s3)ncnc21
O=C(CSc1nc(C(F)(F)F)nc2ccccc12)c1ccc(CCN2CCCC2=O)s1
Cn1ncc2c(SCC(=O)c3cc(F)c(CNC(=O)C(C)(C)C)s3)ncnc21
CC(C)(C)C(=O)NCCc1ccc(C(=O)CSc2nc(C(F)(F)F)nc3ccccc23)s1
Cn1ncc2c(SCC(=O)c3ccc(CNC(=O)c4ccccc4)s3)ncnc21
Cn1ncc2c(SCC(=O)c3ccc(CNC(=O)Cc4ccccc4)s3)ncnc21
CN(Cc1ccc(C(=O)CSc2ncnc3c2cnn3C)s1)C(=O)C(C)(C)C
CN(Cc1ccc(C(=O)CSc2ncnc3c2cnn3C)s1)C(=O)C1CC1
Cc1nc(SCC(=O)c2ccc(CNC(=O)C3CC3)s2)c2ccccc2n1
O=C(CSc1nc(C(F)(F)F)nc2ccccc12)c1ccc(CCNC(=O)C2CC2)s1
O=C(NCCc1ccc(C(=O)CSc2nc(C(F)(F)F)nc3ccccc23)s1)c1ccccc1
CC(C)(C)C(=O)NCc1ccc(C(=O)CSc2nc(C(F)(F)F)nc3ccccc23)s1
Cn1ncc2c(SCC(=O)c3ccc(CNC(=O)Cc4ccccn4)s3)ncnc21
Cn1ncc2c(SCC(=O)c3ccc(CNC(=O)Cc4cccnc4)s3)ncnc21
Cn1ncc2c(SCC(=O)c3ccc(CNC(=O)Cc4ccncc4)s3)ncnc21
COCC(=O)NCc1ccc(C(=O)CSc2ncnc3c2cnn3C)s1
Cn1ncc2c(SCC(=O)c3ccc(CNC(=O)CO)s3)ncnc21
Cn1ncc2c(SCC(=O)c3ccc(CNS(C)(=O)=O)s3)ncnc21
Cn1ncc2c(SCC(=O)c3ccc(CNS(=O)(=O)Cc4ccccc4)s3)ncnc21
CN(Cc1ccc(C(=O)CSc2ncnc3c2cnn3C)s1)S(=O)(=O)C1CC1
CN(Cc1ccc(C(=O)CSc2ncnc3c2cnn3C)s1)S(=O)(=O)Cc1ccncc1
Cc1nc(SCC(=O)c2ccc(CNS(=O)(=O)CC3CC3)s2)c2ccccc2n1
Cc1nc(SCC(=O)c2ccc(CCNS(C)(=O)=O)s2)c2ccccc2n1
CS(=O)(=O)N1CCC(c2ccc(C(=O)CSc3nc(C(F)(F)F)nc4ccccc34)s2)C1
Cc1nc(SCC(=O)c2ccc(CNS(C)(=O)=O)s2)c2ccccc2n1
CS(=O)(=O)NCCc1ccc(C(=O)CSc2nc(C(F)(F)F)nc3ccccc23)s1
CC(C)(C)C(=O)NCc1ccc(C(=O)CSc2nc(C(F)(F)F)cc3ccccc23)s1
Cn1ncc2c(SCC(=O)c3nnc(CNC(=O)C(C)(C)C)s3)ncnc21
CC(C)(C)C(=O)NCc1ccc(C(=O)CSc2nncc3ccccc23)s1
Cc1nnc(SCC(=O)c2ccc(CNC(=O)C(C)(C)C)s2)c2ccccc12
CC(C)(C)C(=O)NCc1ccc(C(=O)CSc2nnc(C(F)(F)F)c3ccccc23)s1
CC1(C)Oc2cccnc2N(Cc2ncc(s2)-c2nnc(o2)C(F)F)C1=O
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccc(Cl)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccc(Cl)c1
FC(F)c1nnc(o1)-c1cnc(CN(c2cccc(Cl)c2)S(=O)(=O)C2CC2)s1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(F)c(F)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccnc1
FC(F)c1nnc(o1)-c1cnc(CNc2cccc(c2)C(F)(F)F)s1
FC(F)c1nnc(o1)-c1cnc(CN(C(=O)c2cccnc2)c2cccc(c2)C(F)(F)F)s1
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccccc1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccccc1
FC(F)(F)c1nc(no1)-c1cnc(CN(c2cccc(Cl)c2)S(=O)(=O)C2CC2)s1
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(F)c(Cl)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(F)c(Cl)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc2cnn(C)c2c1
CN(C)S(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccc(Cl)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)C1CC1
FC(F)c1nnc(o1)-c1cnc(NC2(CC2)c2c(F)cccc2F)s1
FC(F)c1nnc(o1)-c1cnc(NCCc2ccccc2)s1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)C1(CC1)c1ccccc1
CN(C)C(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccnc1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(nc1)N1CCN(C)CC1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(nc1)N1CCOCC1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccc(c1)C(=O)OC
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(cc1)C(=O)OC(C)(C)C
COC(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccnc1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncnc1
FC(F)c1nnc(o1)-c1cnc(CNc2cccnc2)s1
CN(Cc1ccccc1)S(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(F)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(F)nc1
CC(C)S(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccnc1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(=O)n(C)c1
FC(F)c1nnc(o1)-c1cnc(CN(c2ccc(F)c(Cl)c2)S(=O)(=O)N2CCOCC2)s1
FC(F)c1nnc(o1)-c1cnc(CN(c2cccc(Cl)c2)S(=O)(=O)N2CCS(=O)(=O)CC2)s1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(cc1)-n1ccnc1
FC(F)c1nnc(o1)-c1cnc(CN(c2cccc(Cl)c2)S(=O)(=O)N2CCOCC2)s1
CN(C)S(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(F)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(F)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(cc1)-n1cccn1
FC(F)c1nnc(o1)-c1cnc(CN(c2cccnc2)S(=O)(=O)N2CCOCC2)s1
FC(F)c1nnc(o1)-c1cnc(s1)N1[C@@H](COC1=O)c1ccccc1 |r|
FC(F)c1nnc(o1)-c1cnc(s1)N1[C@H](COC1=O)c1ccccc1 |r|
CN(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccnc1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cnn(CC2CC2)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cnn(c1)C1CC1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cnn(c1)C(F)F
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cnn(CCOC)c1
FC(F)c1nnc(o1)-c1cnc(CN(c2cccnc2)S(=O)(=O)C2CC2)s1
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccnc1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(c1)C#N
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(nc1)C(C)(C)C#N
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1nc2cc(F)ccc2o1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1nc2ccc(F)cc2o1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(OC(F)F)nc1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cc(C)n(C)n1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(c1)C1CC1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(c1)C(F)(F)F
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(c1)C(F)F
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(nc1)C(C)C
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccc(n1)C(F)F
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1nc(C)cc(C)n1
CCn1cc(cn1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(=O)(=O)CC
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cnn(C)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(nc1)C#N
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(cn1)C#N
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(C)n1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cc(C)cc(C)n1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccc(n1)C(F)(F)F
FC(F)c1nnc(o1)-c1cnc(COc2cccc(Cl)c2)s1
CN(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccc(Cl)c1
FC(F)c1nnc(o1)-c1cnc(CNc2cccc(Cl)c2)s1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(nc1)C1CC1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cnccn1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccnnc1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cnc(nc1)C(F)(F)F
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(nc1)C(F)(F)F
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(C)nc1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(F)cn1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ncc(F)cn1
CCC(=O)N(Cc1nc(cs1)-c1nnc(o1)C(F)F)c1cccc(Cl)c1
FC(F)c1nnc(o1)-c1csc(CN(c2cccc(Cl)c2)S(=O)(=O)C2CC2)n1
FC(F)c1nnc(o1)-c1csc(CN(C(=O)C2CC2)c2cccc(Cl)c2)n1
CCS(=O)(=O)N(Cc1nc(cs1)-c1nnc(o1)C(F)F)c1cccc(Cl)c1
FC(F)c1nnc(o1)-c1coc(CN(c2cccc(Cl)c2)S(=O)(=O)C2CC2)n1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccnc(c1)C1CC1
FC(F)Oc1ccc(cn1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(=O)(=O)C1CC1
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(c1)C(F)(F)F
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cnccn1
FC(F)c1nnc(o1)-c1cnc(CN(c2cnccn2)S(=O)(=O)C2CC2)s1
FC(F)c1nnc(o1)-c1cnc(CN(c2cncc(F)c2)S(=O)(=O)C2CC2)s1
Cc1cncc(c1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(C)(=O)=O
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(F)c1
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(Cl)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(OC(F)F)c1
FC(F)c1nnc(o1)-c1cnc(CN(c2ccc(nc2)C#N)S(=O)(=O)C2CC2)s1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccnc(c1)C(F)(F)F
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(Cl)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(nc1)C(F)F
FC(F)c1nnc(o1)-c1cnc(s1)N1C(CCC1=O)c1ccccc1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(cn1)C(C)(C)O
CC1(CC1)S(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccnc1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(COC)nc1
CCCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(F)cn1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(nc1)C(C)(C)O
COCCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccnc1
CCOc1cncc(c1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(=O)(=O)CC
CCCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(Cl)c1
CCCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(F)c1
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(c1)C#N
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(c1)C(C)(F)F
CCCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(c1)C#N
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)c1ccccc1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)c1cncc(F)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(nc1)C(C)(F)F
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)c1cncc(Cl)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)c1cnccn1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)c1cccnc1
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)c1cncc(c1)C#N
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)c1cccc(F)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)c1ccccc1
Cn1cc(cn1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(C)(=O)=O
CN(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(c1)C#N
CCCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccnc1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cnn(CCOC(F)(F)F)c1
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(F)cn1
CCCn1cc(cn1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(=O)(=O)C(F)F
CCCn1cc(cn1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(C)(=O)=O
Cn1cc(cn1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(=O)(=O)C1CC1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(C)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(OCC(F)F)c1
FC(F)c1nnc(o1)-c1cnc(CN(c2ccc(F)cn2)S(=O)(=O)C(F)F)s1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cnn(c1)C(C)(C)C#N
CCN(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccc(Cl)c1
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(c1)C1CC1
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccc(n1)C(F)F
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cnn(c1)C(C)C
CC(C)n1cc(cn1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(C)(=O)=O
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccc(n1)C(F)(F)F
FC(F)c1nnc(o1)-c1cnc(CN(c2cccnc2)S(=O)(=O)C(F)F)s1
COCCN(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccc(Cl)c1
FC(F)c1nnc(o1)-c1cnc(CN(c2cncc(c2)C#N)S(=O)(=O)C2CC2)s1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cnn(C)c1C
CC(C)S(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(OC(F)F)c1
CCc1cncc(c1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(=O)(=O)CC
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(OC(F)F)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(OC)c1
CC(C)S(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(c1)C#N
CC(F)(F)c1cncc(c1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(C)(=O)=O
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(Cl)cn1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(OC(C)C)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(C)cn1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cc(C)ccn1
FC(F)c1nnc(o1)-c1cnc(CN(c2cncc(Cl)c2)S(=O)(=O)CCN2CCOCC2)s1
CC(C)CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(OC(F)F)c1
FC(F)c1nnc(o1)-c1cnc(CN(c2cncc(Cl)c2)S(=O)(=O)CCC#N)s1
COCCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(c1)C(C)(F)F
CCCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(C)c1
COCCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(Cl)c1
CCCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(OC(F)F)c1
CC(C)CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccnc1
FC(F)c1nnc(o1)-c1cnc(CN(c2cccnc2)S(=O)(=O)CCN2CCOCC2)s1
COCCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(OC(F)F)c1
COCCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(C)c1
CCCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccc(Cl)cn1
CC(C)CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(c1)C#N
CCCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccc(C)n1
CCCCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccnc1
FC(F)c1nnc(o1)-c1cnc(CN2C(=O)CCc3ccncc23)s1
FC(F)c1nnc(o1)-c1cnc(CN2C(=O)COc3ccncc23)s1
FC(F)c1nnc(o1)-c1cnc(CN(c2cccnc2)S(=O)(=O)CCN2CC3COCC3C2)s1
FC(F)c1nnc(o1)-c1cnc(CN(C(=O)CCN2CCOCC2)c2cncc(F)c2)s1
FC(F)c1nnc(o1)-c1cnc(CN2C(=O)COc3cnccc23)s1
CCC(C)S(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(OC(F)F)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)Cc1cccnc1
FC(F)c1nnc(o1)-c1cnc(CN(c2cccnc2)S(=O)(=O)CCN2C3CC2COC3)s1
FC(F)c1nnc(o1)-c1cnc(CN(c2cncc(F)c2)S(=O)(=O)CCN2CC3COCC3C2)s1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)Cc1ccc(F)cn1
FC(F)c1nnc(o1)-c1cnc(CN(c2cncc(F)c2)S(=O)(=O)CCN2C3CC2COC3)s1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)Cc1ccccn1
FC(F)c1nnc(o1)-c1cnc(CN(c2cccnc2)S(=O)(=O)CCN2CC3CC(C2)O3)s1
FC(F)c1nnc(o1)-c1cnc(CN(C(=O)CCN2CCOCC2)c2cccnc2)s1
FC(F)c1nnc(o1)-c1cnc(CN(c2cncc(F)c2)S(=O)(=O)CCN2CCCOCC2)s1
FC(F)c1nnc(o1)-c1cnc(CN(c2cccnc2)S(=O)(=O)CCN2C[C@@H]3C[C@H]2CO3)s1 |r|
FC(F)c1nnc(o1)-c1cnc(CN(c2cncc(F)c2)S(=O)(=O)CCN2C[C@H]3C[C@@H]2CO3)s1 |r|
C[C@H]1CN(CCS(=O)(=O)N(Cc2ncc(s2)-c2nnc(o2)C(F)F)c2cccnc2)CCO1 |r|
FC(F)c1nnc(o1)-c1cnc(CN(c2cncc(Cl)c2)S(=O)(=O)CCN2C3CC2COC3)s1
FC(F)c1nnc(o1)-c1cnc(CN(c2cncc(Cl)c2)S(=O)(=O)CCN2CC3CC(C2)O3)s1
FC(F)c1nnc(o1)-c1cnc(CN(c2cncc(F)c2)S(=O)(=O)CCN2CC3CC(C2)O3)s1
FC(F)c1nnc(o1)-c1cnc(CN(c2cccnc2)S(=O)(=O)CCN2CCCOCC2)s1
C[C@@H]1CN(CCS(=O)(=O)N(Cc2ncc(s2)-c2nnc(o2)C(F)F)c2cccnc2)CCO1 |r|
FC(F)c1nnc(o1)-c1cnc(CN(C(=O)CCN2CCOCC2)c2cncc(Cl)c2)s1
FC(F)c1nnc(o1)-c1cnc(CN(c2cccnc2)S(=O)(=O)CCN2C[C@H]3C[C@@H]2CO3)s1 |r|
C[C@@H]1CN(CCS(=O)(=O)N(Cc2ncc(s2)-c2nnc(o2)C(F)F)c2cncc(Cl)c2)CCO1 |r|
CCC(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(Cl)c1
CCC(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccnc1
FC(F)c1nnc(o1)-c1cnc(CN2c3ccncc3CCCC2=O)s1
FC(F)c1nnc(o1)-c1cnc(CN(c2cncc(F)c2)S(=O)(=O)CCN2C[C@@H]3C[C@H]2CO3)s1 |r|
C[C@H]1CN(CCS(=O)(=O)N(Cc2ncc(s2)-c2nnc(o2)C(F)F)c2cncc(Cl)c2)CCO1 |r|
C[C@H]1CN(CCS(=O)(=O)N(Cc2ncc(s2)-c2nnc(o2)C(F)F)c2cncc(F)c2)CCO1 |r|
C[C@@H]1CN(CCS(=O)(=O)N(Cc2ncc(s2)-c2nnc(o2)C(F)F)c2cncc(F)c2)CCO1 |r|
FC(F)c1nnc(o1)-c1cnc(CN(c2cncc(Cl)c2)S(=O)(=O)CCN2C[C@H]3C[C@@H]2CO3)s1 |r|
FC(F)c1nnc(o1)-c1cnc(CN(c2cncc(Cl)c2)S(=O)(=O)CCN2C[C@@H]3C[C@H]2CO3)s1 |r|
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(c1)[C@H](C)F |r|
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(c1)[C@@H](C)F |r|
CCC(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(F)c1
FC(F)c1nnc(o1)-c1cnc(CN2C(=O)CCc3cnccc23)s1
CC[C@@H](C)S(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccnc1 |r|
CC[C@H](C)S(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccnc1 |r|
FC(F)c1nnc(o1)-c1cnc(CN(c2cncc(c2)C#N)S(=O)(=O)CCN2CCOCC2)s1
FC(F)c1nnc(o1)-c1cnc(CN(c2cncc(F)c2)S(=O)(=O)CCN2CCOCC2)s1
CCC(C)S(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccnc1
C[C@H](F)c1cncc(c1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(C)(=O)=O |r|
C[C@@H](F)c1cncc(c1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(C)(=O)=O |r|
CC(F)c1cncc(c1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(C)(=O)=O
Cc1cncc(c1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(=O)(=O)CCC#N
FC(F)Oc1cncc(c1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(=O)(=O)CCN1CCOCC1
CCc1ccc(cn1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(=O)(=O)CC
CC(C)(F)c1cncc(c1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(C)(=O)=O
CC(C)CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(F)c1
CC(F)(F)COc1cncc(c1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(C)(=O)=O
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(OCC(C)(F)F)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(c1)C(C)(C)F
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(c1)C(C)F
CCc1ccc(cn1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(C)(=O)=O
CCc1cncc(c1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(C)(=O)=O
CCc1cncc(c1)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(=O)(=O)CCOC
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cc2COCCn2n1
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)c1cncc(OC(F)F)c1
CCCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)c1cncc(OC(F)F)c1
CCCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)c1cncc(c1)C#N
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)c1cnc[nH]1
Cc1cccc(c1)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)S(C)(=O)=O
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)c1cncc(c1)C(F)(F)F
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)c1cncc(c1)C1CC1
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)c1cncc(Cl)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(CCOC)c1
CCCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)c1cccc(F)c1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)c1cncc(c1)C#N
CCCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)c1cncc(Cl)c1
C[C@@H]1CCc2ccncc2N(Cc2ncc(s2)-c2nnc(o2)C(F)F)C1=O |r|
C[C@H]1CCc2ccncc2N(Cc2ncc(s2)-c2nnc(o2)C(F)F)C1=O |r|
FC(F)c1nnc(o1)-c1cnc(CN2C(=O)C3(CC3)c3ccncc23)s1
C[C@H]1CC(=O)N(Cc2ncc(s2)-c2nnc(o2)C(F)F)c2cnccc12 |r|
C[C@@H]1CC(=O)N(Cc2ncc(s2)-c2nnc(o2)C(F)F)c2cnccc12 |r|
C[C@@H]1Cc2ccncc2N(Cc2ncc(s2)-c2nnc(o2)C(F)F)C1=O |r|
C[C@H]1Cc2ccncc2N(Cc2ncc(s2)-c2nnc(o2)C(F)F)C1=O |r|
CC1CCc2ccncc2N(Cc2ncc(s2)-c2nnc(o2)C(F)F)C1=O
CC1(C)CCc2ccncc2N(Cc2ncc(s2)-c2nnc(o2)C(F)F)C1=O
CC1(C)C(=O)N(Cc2ncc(s2)-c2nnc(o2)C(F)F)c2cnccc12
CC1Cc2ccncc2N(Cc2ncc(s2)-c2nnc(o2)C(F)F)C1=O
CC1CC(=O)N(Cc2ncc(s2)-c2nnc(o2)C(F)F)c2cnccc12
Oc1[nH]c2cnccc2c1Cc1ncc(s1)-c1nnc(o1)C(F)F
CCS(=O)(=O)N(Cc1cnc(s1)-c1nnc(o1)C(F)F)c1cncc(Cl)c1
CCS(=O)(=O)N(Cc1cnc(s1)-c1nnc(o1)C(F)F)c1cccnc1
CCS(=O)(=O)N(Cc1cnc(s1)-c1nnc(o1)C(F)F)c1cccc(Cl)c1
CS(=O)(=O)N(Cc1cnc(s1)-c1nnc(o1)C(F)F)c1cncc(F)c1
CCS(=O)(=O)N(Cc1cnc(s1)-c1nnc(o1)C(F)F)c1cncc(F)c1
CS(=O)(=O)N(Cc1ccc(s1)-c1nnc(o1)C(F)F)c1cncc(OC(F)(F)F)c1
FC(F)c1nnc(o1)-c1cnc(CN(c2cccnc2)S(=O)(=O)CCC#N)s1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(OC(F)(F)F)c1
NC(=O)CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccnc1
FC(F)c1nnc(o1)-c1cnc(CN2c3cnccc3CCCC2=O)s1
FC(F)c1nnc(o1)-c1cnc(CN2CCCc3ccccc23)s1
FC(F)c1nnc(o1)-c1ccn(CC(=O)N2CCOCC2)c(=O)c1
FC(F)c1nnc(o1)-c1ccn(CC(=O)N2CCCC2)c(=O)c1
Cn1ccc(cc1=O)-c1nnc(o1)C(F)F
FC(F)c1nnc(o1)-c1ccn(Cc2ccccc2)c(=O)c1
FC(F)c1nnc(o1)-c1ccn(CCc2ccccc2)c(=O)c1
FC(F)(F)c1nnc(o1)-c1cc[nH]c(=O)c1
CC(C)(C)OC(=O)Cn1ccc(cc1=O)-c1nnc(o1)C(F)(F)F
Cn1ccc(cc1=O)-c1nnc(o1)C(F)(F)F
FC(F)(F)c1nnc(o1)-c1ccn(CCc2ccccc2)c(=O)c1
OC(=O)Cn1ccc(cc1=O)-c1nnc(o1)C(F)F
CC(C)(C)OC(=O)Cn1ccc(cc1=O)-c1nnc(o1)C(F)F
FC(F)c1nnc(o1)-c1cc[nH]c(=O)c1
Cc1ccc(OCCn2ccc(cc2=O)-c2nnc(o2)C(F)F)cn1
FC(F)c1nnc(o1)-c1ccn(CCOc2cc(F)cc(F)c2)c(=O)c1
FC(F)c1nnc(o1)-c1ccn(Cc2ccnc(c2)C2CC2)c(=O)c1
FC(F)c1nnc(o1)-c1ccn(CCOc2cccc(F)c2)c(=O)c1
FC(F)c1nnc(o1)-c1cnn(CCOc2cccc(F)c2)c(=O)c1
FC(F)c1nnc(o1)-c1ccn(CC(=O)Nc2ccccc2)c(=O)c1
FC(F)c1nnc(o1)-c1ccn(C[C@@H]2C[C@H]2c2ccccc2)c(=O)c1 |r|
CN(Cc1cc(no1)-c1nnc(o1)C(F)F)c1cccc(Cl)c1
CCS(=O)(=O)N(Cc1cc(no1)-c1nnc(o1)C(F)F)c1cccnc1
CCS(=O)(=O)N(Cc1cc(no1)-c1nnc(o1)C(F)F)c1cccc(Cl)c1
FC(F)c1nnc(o1)-c1cc(CN(c2cccc(Cl)c2)S(=O)(=O)C2CC2)on1
CCS(=O)(=O)N(Cc1cc(on1)-c1nnc(o1)C(F)F)c1cccc(Cl)c1
CN(Cc1cc(on1)-c1nnc(o1)C(F)F)c1cccc(Cl)c1
FC(F)c1nnc(o1)-c1cc(CNc2cccc(Cl)c2)no1
FC(F)c1nnc(o1)-c1cnc2cc(Cc3ccccc3)nn2c1
Nc1nc2ccc(cc2s1)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)nn1
CC(C)(C)OC(=O)N1CCC2(CC1)C(=O)Nc1ccc(cc21)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
Oc1ccc(cc1NC(=O)N1CCOCC1)-c1nnn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)n1
[#6]-[#7](-[#6])-[#6](=[#7]/c1ccc(cc1)-c1cn(-[#6]-c2ccc(cc2)-c2nnc(o2)-[#6](F)F)nn1)\[#7](-[#6])-[#6]
Nc1nc2cc(ccc2s1)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)nn1
Nc1ccc(cn1)-c1nnc(Cc2ccc(cc2)-c2nnc(o2)C(F)F)o1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc3CNC(=O)c3c2)nc1
CC(C)(c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1)c1ccncc1
Nc1ccc(cn1)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccco2)cc1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2cccc(NC(=O)N3CCOCC3)c2)nc1
Nc1ccc(cn1)-c1cn(nn1)C(Cc1ccccc1)c1ccc(cc1)-c1nnc(o1)C(F)F
Nc1nc2cc(ccc2o1)-c1nnn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3cn[nH]c3c2)cc1
Nc1nc2cc(ccc2[nH]1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
NC(=O)c1cccc(c1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)cn1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3nc(Cl)[nH]c3c2)nc1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc(N3CCNCC3)c(F)c2)cc1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc(NC3=NCCN3)cc2)cc1 |t:25|
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc3oc(=O)[nH]c3c2)cc1
Cn1c(N)nc2cc(ccc12)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
NC(=O)c1cccc(c1)-c1noc(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Nc1ccc(cn1)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)cn1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(cn2)-c2cccc(NC(=O)N3CCOCC3)c2)cc1
Nc1ccc(cn1)-c1cnn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)c1
FC(F)c1nnc(o1)-c1ccc(Cc2noc(n2)-c2cccc(NC(=O)N3CCOCC3)c2)cc1
Nc1nc2ccc(cc2s1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
CC(c1ccc(cc1)-c1nnc(o1)C(F)F)n1nnc(n1)-c1ccc2CCN(C)C(=O)c2c1
Nc1ccc(cn1)-c1cn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc(cc2)C(=O)N2CCOCC2)cc1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2cccc(NC(=O)N3CCOCC3)c2)cc1F
Nc1ccc(cn1)-c1cn(nn1)C(Cc1ccc(Cl)cc1)c1ccc(cc1)-c1nnc(o1)C(F)F
Cn1c(N)nc2cc(ccc12)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)nn1
CN1CCC(CC1)NC(=O)c1ccc(cc1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
CCNc1nc2ccc(cc2[nH]1)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)nn1
COc1ccccc1-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3NC(=O)C4(CCNCC4)c3c2)nc1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccccc2)cc1
FC(F)c1nnc(o1)-c1ccc(Cn2cnc(c2)-c2ccc(NC3=NCCN3)cc2)nc1 |t:25|
CCCCC(c1ccc(cc1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1ccc(N)nc1
Nc1ccc(cn1)-c1cn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2F)nn1
Nc1ccc(cn1)-c1cn(nn1)C(COc1ccccc1)c1ccc(cc1)-c1nnc(o1)C(F)F
FC(F)c1nnc(o1)-c1ccc(Cn2cnc(c2)-c2ccc(NC3=NCCN3)cc2)cc1 |t:25|
CN1Cc2ccc(cc2NC(=O)C1)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
Cn1c(N)nc2cc(ccc12)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cc2nnc(s2)-c2ccccc2)cc1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc(NC3=NCCN3)cc2)nc1 |t:25|
FC(F)c1nnc(o1)-c1cc(F)c(Cn2cc(nn2)-c2ccc(cc2)C(=O)N2CCCC(C2)C(=O)NCC2CC2)c(F)c1
Oc1ccc(cc1NC(=O)N1CCOCC1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
CC(C)(C)OC(=O)N1CCn2ncc(c2C1)-c1cccc(c1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3NC(=O)C4(CCCC4)c3c2)nc1
Cc1nc(F)ccc1-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc3NC(=O)C4(CCCC4)Nc3c2)nc1
Nc1ccc(cn1)-c1cn(nn1)C(CC1CCC1)c1ccc(cc1)-c1nnc(o1)C(F)F
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3NC(=O)C4(CCNC4)c3c2)nc1
Nc1ccc(cn1)-c1noc(n1)C(F)(F)c1ccc(cc1)-c1nnc(o1)C(F)F
NC(=O)c1cccc(c1)-c1nnn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)n1
CCCCC(c1ccc(cc1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1cccc(NC(=O)N2CCOCC2)c1
Nc1nc2ccc(cc2[nH]1)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)nn1
CC1(C)NC(=O)c2cc(ccc12)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
CN(C)C(=O)Nc1cc(ccc1O)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccc(c2)-c2ccccc2)cc1
C[C@H](c1ccc(cn1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1ccc(N)nc1
Nc1ccc(cn1)-c1nc(Cc2ccc(cc2)-c2nnc(o2)C(F)F)no1
NCc1ccc(cc1)-c1nnn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2cccc(F)c2)cc1
CNc1ccc2cc(ccc2n1)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)nn1
CN(C)c1nc2cc(ccc2o1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Nc1cc(ccc1O)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
CCC[C@@H](c1ccc(cc1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1ccc(N)nc1 |r|
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3NC(=O)C4(CCNCC4)Nc3c2)nc1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(Cc3ccccn3)n2)cc1
CC(=O)Nc1cccc(c1)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)nn1
Cn1c(N)nc2cc(ccc12)-c1nnn(Cc2ncc(cn2)-c2nnc(o2)C(F)F)n1
Nc1ncc(s1)-c1cccc(c1)-c1nnn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccc(c2)-c2cnc(s2)N2CCOCC2)cc1
Nc1ccc(cn1)-c1cn(Cc2cc(F)c(cc2F)-c2nnc(o2)C(F)F)nn1
CN(Cc1ccncc1)Cc1ccc(cc1)-c1nc(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)no1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc3CNC(=O)c3c2)c(F)c1
C[C@@H](c1ccc(cc1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1ccc(N)nc1 |r|
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3NC4(CCNCC4)C(=O)Nc3c2)nc1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)C2(CC2)c2ccccc2)cc1
Nc1ccc(cn1)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
CC(=O)N1CCC(CC1)c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
NCc1ccc(cc1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc(Sc3ccccc3)c(NC(=O)N3CCOCC3)c2)cc1
NCc1ccc(cc1)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
CN(Cc1ccc(cc1)-c1nc(Cc2ccc(cc2)-c2nnc(o2)C(F)F)no1)C(=O)C(F)F
Nc1ccc(cn1)-c1nnn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)n1
OC(=O)c1cccc(c1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3NC(=O)C4(CCNCC4)c3c2)cc1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccs2)cc1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2cccc(NC(=O)N3CCOCC3)c2)c(F)c1
NC(=O)c1cccc(c1)-c1nc(Cc2ccc(cc2)-c2nnc(o2)C(F)F)no1
Nc1ccc(cn1)-c1cn(Cc2ccc(cc2F)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc(Cl)cc2Cl)cc1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3NC(=O)C4(CCNC4)c3c2)cc1
FC(F)c1nnc(o1)-c1ccc(Cn2cnc(c2)-c2cccc(NC(=O)N3CCOCC3)c2)nc1
NC(=O)c1cccc(c1)-c1nnn(Cc2ccc(cc2F)-c2nnc(o2)C(F)F)n1
CC(C)(C)OC(=O)N1CCC2(C1)C(=O)Nc1ccc(cc21)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)nn1
CN1CCN(CC1)C(=O)Nc1cccc(c1)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)nn1
Nc1ccc(cn1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2cnc(c2)-c2cccc(NC(=O)N3CCOCC3)c2)cc1
COc1ncccc1-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)nn1
CC(C)(C)OC(=O)N1CCC2(CC1)Nc1cc(ccc1NC2=O)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
NC(=O)c1cccc(c1)-c1nnn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(cn2)-c2ccc(NC3=NCCN3)cc2)cc1 |t:25|
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc3CNC(=O)c3c2)cc1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(cn2)-c2ccc(NC3=NCCN3)cc2)nc1 |t:25|
Oc1ccc(cc1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3NC(=O)C4(CCNCC4)Nc3c2)cc1
FC(F)c1nnc(o1)-c1cc(F)c(Cn2nnc(n2)-c2ccc3CNC(=O)c3c2)c(F)c1
CC(C)(C)OC(=O)N1CCc2[nH]c(nc2C1)-c1cccc(c1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
CN1CCN(CC1)c1cccc(c1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3NC(=O)[C@]4(CCNC4)c3c2)nc1 |r|
CC(c1ccc(cn1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1ccc(N)nc1
CCNc1nc2ccc(cc2[nH]1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
OC(=O)c1cccc(c1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3NC(=O)C4(CCCC4)c3c2)cc1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccc(c2)-c2nc3CNCCc3[nH]2)nc1
CS(=O)(=O)NCCC(c1ccc(cc1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1ccc(N)nc1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3NC4(CCNCC4)C(=O)Nc3c2)cc1
CN1CCN(CC1)C(=O)Nc1cccc(c1)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
Nc1ncc2cc(ccc2n1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Nc1ccc(cn1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
CC(C)(C)OC(=O)N1CCC2(CC1)Nc1ccc(cc1NC2=O)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
Cc1ncc(cc1N)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2cnc3cccnn23)cc1
CC(c1ccc(cn1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1cccc(NC(=O)N2CCOCC2)c1
CN(C)c1ccc(cc1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1cc(F)c(Cn2cc(nn2)-c2cnc3cccnn23)c(F)c1
CN(Cc1ccncc1)Cc1ccc(cc1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
FC(F)C(=O)Nc1ccc(cn1)-c1nnn(Cc2ncc(cn2)-c2nnc(o2)C(F)F)n1
CCN(Cc1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1)C(=O)Nc1cccnc1OC
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccc(c2)C(=O)N2CCOCC2)nc1
Cn1c(Sc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nnc1-c1ccc(N)nc1
CC(=O)Nc1cccc(c1)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
Cn1c(Sc2ccc(cc2)-c2nnc(o2)C(F)F)nnc1-c1ccc(N)nc1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccc(NC(=O)N3CCOCC3)c2)cc1
COc1ncc(NCc2ccc(cc2)-n2cc(Cc3ccc(cc3)-c3nnc(o3)C(F)F)nn2)cc1C(N)=O
NC(=O)c1cc(ccc1N)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2nnnc2-c2ncccn2)cc1
Nc1cncc(c1)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnnc2-c2csc3ccccc23)cc1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2cnc3cccnn23)nc1
FC(F)c1nnc(o1)-c1ccc(Cn2nnnc2-c2cccc(c2)-n2cccn2)cc1
NC(=O)c1cccc(c1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Nc1ccc(cn1)-c1nnnn1Cc1ncc(cn1)-c1nnc(o1)C(F)F
NC(=O)c1cc(cnc1N)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Cn1c(N)nc2cc(ccc12)-c1nnnn1Cc1ncc(cn1)-c1nnc(o1)C(F)F
Nc1ccc(cn1)-c1nnn(Cc2ncc(cn2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2cnc(c2)-c2ccc3CNC(=O)c3c2)nc1
FC(F)c1nnc(o1)-c1cc(F)c(Cn2cc(nn2)-c2cccc(NC(=O)N3CCOCC3)c2)c(F)c1
CS(=O)(=O)NCCC(c1ccc(cn1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1ccc(N)nc1
Nc1ncc(cn1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2cnc(c2)-c2ccc3CNC(=O)c3c2)cc1
CN1CCC(CC1)NC(=O)c1cccc(c1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Nc1ccc(cn1)-c1cn(nn1)C(CCNC(=O)C(F)F)c1ccc(cn1)-c1nnc(o1)C(F)F
CN(C)C(=O)c1cccc(c1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Nc1ccc(cc1)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cncc(Br)c2)cc1
Nc1cccc(c1)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc3CCNC(=O)c3c2)cc1
FC(F)c1nnc(o1)-c1cnc(Cn2nnnc2-c2ccc3CNC(=O)c3c2)nc1
Nc1ncnc2cc(ccc12)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1cnc(Cn2nnnc2-c2cccs2)nc1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2cccs2)nc1
Nc1nc2cc(ccc2s1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)cn1
CN1CC(C1)C(=O)Nc1cccc(c1)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
Nc1ccc(cn1)-c1cn(nn1)C(CN1CCCC1)c1ccc(cn1)-c1nnc(o1)C(F)F
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc(CN3CCCCC3)cc2)cc1
CS(=O)(=O)NCC(c1ccc(cc1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1ccc(N)nc1
FC(F)C(=O)Nc1ccc(cn1)-c1cn(Cc2ncc(cn2)-c2nnc(o2)C(F)F)nn1
Nc1ccc(cn1)-c1cn(nn1)C(CCCN1CCCCC1)c1ccc(cc1)-c1nnc(o1)C(F)F
NC(=O)c1cccc(c1)-c1nnn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2)n1
Nc1ccc(cn1)-c1cn(Cc2ncc(cc2F)-c2nnc(o2)C(F)F)nn1
Nc1cncc(c1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
NC(=O)c1cccc(c1)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)cn1
CCNC(=O)c1cccc(c1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Nc1nc2ccc(cc2s1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)cn1
CC1(C)CN(C1=O)c1cccc(c1)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
Nc1nc2ccc(cc2s1)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)cn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccc(c2)C(=O)N2CCOCC2)c(F)c1
Nc1nc2cc(ccc2o1)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)cn1
Nc1ccc(cn1)-c1cn(nn1)C(CO)c1ccc(cc1)-c1nnc(o1)C(F)F
Nc1nc2cc(ccc2o1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)cn1
Oc1ccc(cc1NC(=O)N1CCOCC1)-c1nnn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)n1
CS(=O)(=O)NCC[C@@H](c1ccc(cc1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1ccc(N)nc1 |r|
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccc(c2)C(=O)NCc2ccco2)cc1
CS(=O)(=O)NCC[C@H](c1ccc(cc1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1ccc(N)nc1 |r|
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc3CNC(=O)c3c2)cc1F
Nc1ccc(cn1)-c1cn(nn1)[C@@H](CN1CCCC1)c1ccc(cc1)-c1nnc(o1)C(F)F |r|
FC(F)c1nnc(o1)-c1cc(F)c(Cn2nnc(n2)-c2cccc(NC(=O)N3CCOCC3)c2)c(F)c1
Nc1ccc(cn1)-c1cn(nn1)[C@H](CN1CCCC1)c1ccc(cc1)-c1nnc(o1)C(F)F |r|
CCNc1ccc(cn1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Nc1ccc(cn1)-c1cn(nn1)[C@@H](CO)c1ccc(cc1)-c1nnc(o1)C(F)F |r|
NCc1ccc(cc1)-c1nc(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)no1
Nc1ccc(cc1)-n1cc(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
NCc1ccc(cn1)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cc2cn(nn2)-c2ccc(NC3=NCCN3)cc2)cc1 |t:25|
FC(F)C(=O)Nc1ccc(cn1)-c1nnc(Cc2ccc(cn2)-c2nnc(o2)C(F)F)s1
Nc1ncnc2cc(ccc12)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc(cc2)N2CCNCC2)cc1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(cn2)-c2ccc3CNC(=O)c3c2)nc1
C[C@@H](c1ccc(cc1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1cccc(NC(=O)N2CCOCC2)c1 |r|
FC(F)c1nnc(o1)-c1ccc(Cn2cc(cn2)-c2ccc3CNC(=O)c3c2)cc1
Cc1ncccc1-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
Cn1c(N)nc2cc(ccc12)-c1cnn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)c1
C[C@H](c1ccc(cc1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1ccc(N)nc1 |r|
Cn1c(N)nc2cc(ccc12)-c1cnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)c1
FC(F)c1nnc(o1)-c1cnc(Cn2nnc(n2)-c2ccc3CNC(=O)c3c2)nc1
Nc1nc2cc(ccc2s1)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)cn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccc(c2)-c2nc3CNCCc3[nH]2)cc1
Nc1ccc(cn1)-c1cn(nn1)C(CCN1CCCC1)c1ccc(cc1)-c1nnc(o1)C(F)F
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3CNC(=O)c3c2)cc1
CC1(C)C(=O)Nc2ccc(cc12)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc3NC(=O)C4(CCCC4)Nc3c2)cc1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3NC(=O)Cc3c2)nc1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc(cc2)-c2cnn3CCNCc23)cc1
Nc1nc2ccc(cc2s1)-c1cnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)c1
FC(F)c1nnc(o1)-c1cc(F)c(Cn2nnc(n2)-c2cccc(c2)C(=O)N2CCOCC2)c(F)c1
Nc1nc2ccc(cc2s1)-c1cnn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)c1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc3ccccc3n2)cc1
Cn1c(N)nc2cc(ccc12)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)cn1
CCNc1cccc(c1)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
Cn1c(N)nc2cc(ccc12)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)cn1
Cc1ncccc1-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)nn1
Nc1ccc(cc1)-c1ncc(Cc2ccc(cc2)-c2nnc(o2)C(F)F)o1
NC(=O)c1ccc(cc1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Nc1nc2cc(ccc2[nH]1)-c1cnn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)c1
CC(c1ccc(cc1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1ccc(N)nc1
Nc1nc2cc(ccc2[nH]1)-c1cnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)c1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cncc3ccccc23)cc1
NC(=O)c1cccc(c1)-c1cnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)c1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(cn2)-c2cccc(NC(=O)N3CCOCC3)c2)nc1
NC(=O)c1cccc(c1)-c1cnn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)c1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccc(c2)C(=O)N2CCOCC2)cc1
Nc1ccc(cn1)-c1cn(nn1)C(CCCO)c1ccc(cc1)-c1nnc(o1)C(F)F
Nc1ccc(cc1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1cnc(Cn2cc(nn2)-c2cccc(NC(=O)N3CCOCC3)c2)c(F)c1
FC(F)c1nnc(o1)-c1cc(F)c(Cn2cc(nn2)-c2cccs2)c(F)c1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2cccc(NC(=O)N3CCOCC3)c2)c(Cl)c1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3c(NC(=O)C33CCCC3)c2)nc1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2cccc(NC(=O)N3CCOCC3)c2)c(F)c1F
Nc1ccc(cn1)-c1cn(nn1)C(CN1CCCC1)c1ccc(cc1)-c1nnc(o1)C(F)F
Nc1nc2ccc(cc2s1)-c1cn(Cc2ccc(cc2F)-c2nnc(o2)C(F)F)nn1
Nc1ccc(cn1)-c1cn(Cc2ncc(cn2)-c2nnc(o2)C(F)F)nn1
Nc1nc2ccc(cc2s1)-c1cn(Cc2ccc(cc2Cl)-c2nnc(o2)C(F)F)nn1
FC(F)C(=O)Nc1ccc(cn1)-c1cn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)cn1
Nc1nc2ccc(cc2s1)-c1cn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc3ccncc3c2)cc1
Nc1nc2ccc(cc2s1)-c1cn(Cc2ncc(cc2F)-c2nnc(o2)C(F)F)nn1
COc1ccc(cc1OC)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Nc1nc2ccc(cc2s1)-c1cn(Cc2cc(F)c(cc2F)-c2nnc(o2)C(F)F)nn1
Nc1cccc(c1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Cn1c(N)nc2cc(ccc12)-c1cn(Cc2ccc(cc2Cl)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccc(c2)-c2cnc(s2)N2CCOCC2)nc1
Cn1c(N)nc2cc(ccc12)-c1cn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2F)nn1
COc1ncccc1-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
Cn1c(N)nc2cc(ccc12)-c1cn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2)nn1
Nc1nc2cc(ccc2s1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
Nc1nc2ccc(cc2s1)-c1cn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2)nn1
CC(=O)Nc1cc(cnc1C)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Cn1c(N)nc2cc(ccc12)-c1nnn(Cc2ccc(cc2F)-c2nnc(o2)C(F)F)n1
Nc1ccc(cn1)-c1cn(Cc2ccc(cc2Cl)-c2nnc(o2)C(F)F)nn1
Cn1c(N)nc2cc(ccc12)-c1cn(Cc2ncc(cc2F)-c2nnc(o2)C(F)F)nn1
Nc1ccc(cn1)-c1noc(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Cn1c(N)nc2cc(ccc12)-c1cn(Cc2cc(F)c(cc2F)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3nc(Cl)[nH]c3c2)cc1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccc(c2)C(=O)N2CCOCC2)cc1F
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2cccc(NC(=O)N3CCOCC3)c2)cc1
COc1ncc(NCc2ccc(cc2)-c2cn(Cc3ccc(cc3)-c3nnc(o3)C(F)F)nn2)cc1C(N)=O
FC(F)c1nnc(o1)-c1cnc(Cn2nnc(n2)-c2cccc(c2)-c2nc3CNCCc3[nH]2)c(F)c1
CC(=O)Nc1cccc(c1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccc(c2)-c2nc3CNCCc3[nH]2)c(F)c1
CC(=O)c1cccc(c1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccc(c2)-c2nc3CNCCc3[nH]2)c(F)c1F
Nc1ccc(cn1)-c1nc(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)no1
CNc1ccc2cc(ccc2n1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2cnc(c2)-c2ccc(NC3=NCCN3)cc2)c(F)c1 |t:25|
CCC[C@H](c1ccc(cc1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1ccc(N)nc1 |r|
FC(F)c1nnc(o1)-c1ccc(Cn2cnc(c2)-c2ccc(NC3=NCCN3)cc2)c(Cl)c1 |t:25|
NCC(=O)Nc1cccc(c1)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2cnc(c2)-c2ccc(NC3=NCCN3)cc2)c(F)c1F |t:25|
FC(F)c1nnc(o1)-c1cc(F)c(Cc2noc(n2)-c2cccc(NC(=O)N3CCOCC3)c2)c(F)c1
FC(F)c1nnc(o1)-c1ccc(Cn2cnc(c2)-c2ccc(NC3=NCCN3)cc2)cc1F |t:25|
CN1CCN(CC1)C(=O)Nc1cccc(c1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1cc(F)c(Cn2cnc(c2)-c2ccc(NC3=NCCN3)cc2)cc1F |t:26|
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)C2(CC2)c2ccccn2)cc1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc(nc2)N2CCNCC2)cc1
FC(F)c1nnc(o1)-c1cc(F)c(Cn2cc(nn2)-c2cccc(NC(=O)N3CCOCC3)c2)cc1F
CN1CC(C1)C(=O)Nc1cccc(c1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccc(c2)-c2nc3CCNCc3[nH]2)cc1F
[O-][N+](=O)c1ccccc1-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccc(c2)-c2nc3CCNCc3[nH]2)c(Cl)c1
Nc1ccc(cn1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)cn1
Nc1nc2ccc(cc2s1)-c1cc(Cc2ccc(cc2)-c2nnc(o2)C(F)F)on1
Nc1nc2cc(ccc2o1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1cc(F)c(Cn2nnc(n2)-c2cccc(c2)-c2nc3CNCCc3[nH]2)cc1F
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccc3cnccc23)cc1
COc1ncc(NCc2ccc(cc2)-c2cn(Cc3c(F)cc(cc3F)-c3nnc(o3)C(F)F)nn2)cc1C(N)=O
NCc1ccc(cn1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
Cn1c(N)nc2cc(ccc12)-c1nnn(Cc2ncc(cc2F)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccc(NC(=O)c3ccccc3)c2)cc1
Cn1c(N)nc2cc(ccc12)-c1nnn(Cc2ncc(-c3nnc(o3)C(F)F)c(F)c2F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc3NC(=O)C4(CCCCC4)Nc3c2)cc1
Cn1c(N)nc2cc(ccc12)-c1nnn(Cc2cc(F)c(cc2F)-c2nnc(o2)C(F)F)n1
Nc1ccc(cn1)-c1cn(nn1)C(CC(F)(F)F)c1ccc(cc1)-c1nnc(o1)C(F)F
Cn1c(N)nc2cc(ccc12)-c1nnn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2)n1
C[C@@H]1CN(CCN1)c1ccc(cn1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1 |r|
Cn1c(N)nc2cc(ccc12)-c1nnn(Cc2ccc(cc2Cl)-c2nnc(o2)C(F)F)n1
Nc1cc(ccc1OC(=O)N1CCOCC1)-c1nnn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)n1
Nc1ccc(cc1)-c1noc(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3c(NC(=O)C33CCNCC3)c2)cc1
Cn1c2ccc(cc2n(C)c1=N)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
Nc1nc2ccc(cc2s1)-n1cc(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
CN(C)S(=O)(=O)c1ccc(F)c(c1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Cn1c(N)nc2cc(ccc12)-c1cn(Cc2ccc(cc2F)-c2nnc(o2)C(F)F)nn1
CNc1ccc(cc1N)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cc2nc(no2)-c2ccc(NC3=NCCN3)cc2)cc1 |t:25|
CC(c1ccc(cc1F)-c1nnc(o1)C(F)F)n1cc(nn1)-c1cccc(NC(=O)N2CCOCC2)c1
FCc1nnc(o1)-c1ccc(Cc2nc(no2)-c2ccc(NC3=NCCN3)cc2)cc1 |t:24|
Cn1c(N)nc2ccc(cc12)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc3C(=O)NCc3c2)cc1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc3[nH]c(=O)[nH]c3c2)cc1
FC(F)c1nnc(o1)-c1ccc(Cc2nc(no2)-c2ccc(NC3=NCCN3)cc2)cc1F |t:25|
CCS(=O)(=O)N1CCN(Cc2ccc(cc2)-c2cn(Cc3c(F)cc(cc3F)-c3nnc(o3)C(F)F)nn2)CC1
Nc1ccc(cc1)-c1noc(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2)n1
CNC(=O)Nc1ccc(cn1)-c1nnc(Cc2ccc(cc2)-c2nnc(o2)C(F)F)o1
Nc1ccc(cc1)-c1noc(Cc2ccc(cc2F)-c2nnc(o2)C(F)F)n1
C[C@@H](c1ccc(cn1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1ccc(N)nc1
FC(F)c1nnc(o1)-c1ccc(Cc2nc(no2)-c2ccc(NC3=NCCN3)cc2)c(F)c1 |t:25|
CC(C)(C)OC(=O)NCC(=O)Nc1cccc(c1)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
Nc1ncnc2sc(cc12)-c1cn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2F)nn1
CN1CCc2ccc(cc2C1=O)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3nc([nH]c3c2)N2CCOCC2)cc1
Nc1ncnc2sc(cc12)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
NC(=S)Nc1cccc(c1)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
Nc1ncnc2cc(ccc12)-c1cn(Cc2ccc(cc2F)-c2nnc(o2)C(F)F)nn1
CNc1ccc(cc1NC(=O)N1CCOCC1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
CNc1ccc2cc(ccc2n1)-c1nnn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)n1
CC(C)(C)OC(=O)N1CCC2(C1)C(=O)Nc1ccc(cc21)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
CNc1ncc2cc(ccc2n1)-c1cn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2F)nn1
Nc1ncnc2sc(cc12)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
CNc1ncc2cc(ccc2n1)-c1cn(Cc2ccc(cc2F)-c2nnc(o2)C(F)F)nn1
CN(Cc1ccncc1)Cc1ccc(cc1)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
CNc1ncc2cc(ccc2n1)-c1cn(Cc2cc(F)c(cc2F)-c2nnc(o2)C(F)F)nn1
CCNc1cccc(c1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
CNc1ncc2cc(ccc2n1)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccccc2F)cc1
CNc1ncc2cc(ccc2n1)-c1cn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2)nn1
C[C@H]1CN(CCN1)c1ccc(cn1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1 |r|
CCNc1ncc2cc(ccc2n1)-c1cn(Cc2cc(F)c(cc2F)-c2nnc(o2)C(F)F)nn1
CC(=O)N(Cc1ccco1)c1cccc(c1)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
CCNc1ncc2cc(ccc2n1)-c1cn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2)nn1
CC[C@H](c1ccc(cc1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1cccc(NC(=O)N2CCOCC2)c1 |r|
Nc1nccc2cc(ccc12)-c1nnn(Cc2cc(F)c(cc2F)-c2nnc(o2)C(F)F)n1
CC(c1ccc(cc1F)-c1nnc(o1)C(F)F)n1cc(nn1)-c1ccc(N)nc1
Nc1nccc2cc(ccc12)-c1nnn(Cc2ccc(cc2F)-c2nnc(o2)C(F)F)n1
CC(c1ccc(-c2nnc(o2)C(F)F)c(F)c1)n1cc(nn1)-c1ccc(N)nc1
Nc1cnc2ccc(cc2c1)-c1nnn(Cc2cc(F)c(cc2F)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1cnc(Cn2nnc(n2)-c2cccs2)nc1
CN(C)c1ccc2cc(ccc2n1)-c1cn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccc(c2)-n2cccn2)cc1
Nc1cnc2ccc(cc2c1)-c1nnn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2)n1
CC(c1ccc(-c2nnc(o2)C(F)F)c(F)c1)n1cc(nn1)-c1cccc(NC(=O)N2CCOCC2)c1
CNc1ccc2cc(ccc2n1)-c1nnn(Cc2ccc(cc2F)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc3nc([nH]c3c2)N2CCCC2)cc1
CNc1ccc2cc(ccc2n1)-c1nnn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2)n1
NCc1ccc(cc1)-c1nc(Cc2ccc(cc2)-c2nnc(o2)C(F)F)no1
Nc1cc2cc(ccc2cn1)-c1cn(Cc2ccc(cc2Cl)-c2nnc(o2)C(F)F)nn1
Nc1cccc(c1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
Nc1cc2cc(ccc2cn1)-c1cn(Cc2ccc(cc2F)-c2nnc(o2)C(F)F)nn1
Nc1cc2cc(ccc2cn1)-c1cn(Cc2cc(F)c(cc2F)-c2nnc(o2)C(F)F)nn1
CC[C@H](c1ccc(cc1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1ccc(N)nc1 |r|
CNc1ccc2cc(ccc2n1)-c1nnn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc3NC4(CCCC4)C(=O)Nc3c2)cc1
CCNc1ccc2cc(ccc2n1)-c1nnn(Cc2cc(F)c(cc2F)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1cc(F)c(Cn2nnc(n2)-c2ccc(OC(=O)N3CCOCC3)c(NC(=O)N3CCOCC3)c2)c(F)c1
CCNc1ccc2cc(ccc2n1)-c1nnn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2)n1
Nc1cccc(c1)-c1cn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)cn1
Nc1ccc(cn1)-n1cc(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
Nc1ccc(cn1)-c1cn(Cc2ccc(nn2)-c2nnc(o2)C(F)F)nn1
Cn1c(N)nc2cc(ccc12)-n1cc(Cc2ccc(cc2)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cncc(NC(=O)N3CCOCC3)c2)cc1
Nc1ncnc2sc(cc12)-c1cn(Cc2cc(F)c(cc2F)-c2nnc(o2)C(F)F)nn1
Nc1ncc(s1)-c1cccc(c1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Nc1ncnc2sc(cc12)-c1cn(Cc2ccc(cc2F)-c2nnc(o2)C(F)F)nn1
CN(Cc1ccncc1)Cc1ccc(cc1)-c1nnn(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)n1
Nc1ncnc2sc(cc12)-c1cn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2)nn1
Nc1ccc(cn1)-c1cc(Cc2ccc(cc2)-c2nnc(o2)C(F)F)on1
Nc1ncnc2cc(ccc12)-c1cn(Cc2ccc(-c3nnc(o3)C(F)F)c(F)c2)nn1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc3CCC(=O)c3c2)cc1
Nc1nccc2cc(ccc12)-c1nnn(Cc2ccc(cc2Cl)-c2nnc(o2)C(F)F)n1
COc1ccc(cc1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Nc1ncc2cc(ccc2n1)-c1nnn(Cc2cc(F)c(cc2F)-c2nnc(o2)C(F)F)n1
CCC[C@@H](c1ccc(cc1)-c1nnc(o1)C(F)F)n1cc(nn1)-c1cccc(NC(=O)N2CCOCC2)c1 |r|
Nc1ncc2cc(ccc2n1)-c1nnn(Cc2ccc(cc2F)-c2nnc(o2)C(F)F)n1
CN(Cc1ccc(cc1)-c1nc(Cc2c(F)cc(cc2F)-c2nnc(o2)C(F)F)no1)C(=O)C(F)F
Nc1ncc2cc(ccc2n1)-c1nnn(Cc2ccc(cc2Cl)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2csc3ccccc23)cc1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc3cnccc3c2)c(Cl)c1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2cccc3C(=O)CCc23)cc1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc3cnccc3c2)c(F)c1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccc3NC4(CCCCC4)C(=O)Nc3c2)cc1
FC(F)c1nnc(o1)-c1cc(F)c(Cn2nnc(n2)-c2ccc3cnccc3c2)cc1F
Cn1c2ccc(cc2[nH]c1=O)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Nc1cc2cc(ccc2cn1)-c1nnn(Cc2ccc(cc2Cl)-c2nnc(o2)C(F)F)n1
Nc1ccc(cn1)-c1cnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)c1
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2nccc3ccccc23)c(F)c1
CN1CCN(CC1)c1ccc(cn1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Nc1ncnc2cc(ccc12)-c1cn(Cc2cc(F)c(cc2F)-c2nnc(o2)C(F)F)nn1
CN1CCN(CC1)c1ccc(cc1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
Nc1ncnc2cc(ccc12)-c1cn(Cc2ccc(cc2Cl)-c2nnc(o2)C(F)F)nn1
FC(F)c1nnc(o1)-c1cc(F)c(Cn2cc(nn2)-c2ccc(CN3CC(C3)C(F)(F)F)cc2)c(F)c1
CNc1ccc2cc(ccc2n1)-c1nnn(Cc2cc(F)c(cc2F)-c2nnc(o2)C(F)F)n1
CN(Cc1ccncc1)Cc1ccc(cc1)-c1nnn(Cc2ccc(cc2)-c2nnc(o2)C(F)F)n1
CC1(C)N(Cc2ccc(cc2F)-c2nnc(o2)C(F)F)C(=O)N(C1=O)c1ccccc1
CC1(C)N(Cc2ccc(cc2F)-c2nnc(o2)C(F)(F)F)C(=O)N(C1=O)c1ccccc1
FC(F)c1nnc(o1)-c1ccc(CN2C(=O)CN(C2=O)c2ccccc2)c(F)c1
FC(F)c1nnc(o1)-c1ccc(CN2C(=O)CN(C2=O)c2ccccc2)nc1
CC(C)(C)OC(=O)N1CCC2(CC1)N(C(=O)N(Cc1ccc(cn1)-c1nnc(o1)C(F)F)C2=O)c1cccc(F)c1
CN1CCC2(CC1)N(C(=O)N(Cc1ccc(cn1)-c1nnc(o1)C(F)F)C2=O)c1cccc(F)c1
FC(F)c1nnc(o1)-c1ccc(CN2C(=O)N(c3cccc(F)c3)C3(CCN(CC3)C3COC3)C2=O)nc1
CC(C)N1CCC2(CC1)N(C(=O)N(Cc1ccc(cn1)-c1nnc(o1)C(F)F)C2=O)c1cccc(F)c1
CC1(C)N(C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C1=O)c1cccc(F)c1
CC1(C)N(C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C1=O)c1cccc(Br)c1
CC1(C)N(C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C1=O)c1ccc(F)cc1
CC1(C)N(C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C1=O)c1c(F)cccc1F
CC1(C)N(C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C1=O)c1ccc(F)cc1F
CC1(C)N(C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C1=O)c1cccc(F)c1F
CC1(C)N(C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C1=O)c1ccc(F)c(F)c1
CC1(C)N(C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C1=O)c1cc(F)cc(F)c1
CC1(C)N(C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C1=O)c1ccccc1
CN1CCC(=CC1)c1cccc(c1)N1C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C(=O)C1(C)C |c:4|
CN1CCC(CC1)c1cccc(c1)N1C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C(=O)C1(C)C
CN1CC2(C1)N(C(=O)N(Cc1ccc(cn1)-c1nnc(o1)C(F)F)C2=O)c1ccccc1
CC(C)N1CC2(C1)N(C(=O)N(Cc1ccc(cn1)-c1nnc(o1)C(F)F)C2=O)c1ccccc1
CC(=O)N1CC2(C1)N(C(=O)N(Cc1ccc(cn1)-c1nnc(o1)C(F)F)C2=O)c1ccccc1
FC(F)c1nnc(o1)-c1ccc(CN2C(=O)N(c3ccccc3)C3(CCC3)C2=O)nc1
CC1(C)N(C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C1=O)c1ccc(cc1)-c1ccoc1
CC1(C)N(C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C1=O)c1ccc(cc1)-c1ccncc1
CC1(C)N(C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C1=O)c1ccc(cc1)-c1cccnc1
CC1(C)N(C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C1=O)c1ccc(cc1)-c1cccc(F)c1
CC1(C)N(C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C1=O)c1ccc(cc1)-c1ccccc1F
CC(C)(C)OC(=O)n1ccc2c(cccc12)N1C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C(=O)C1(C)C
CC(C)(C)OC(=O)N1CCc2c1cccc2N1C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C(=O)C1(C)C
CC1(C)N(C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C1=O)c1cccc2[nH]ccc12
CC1(C)N(C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C1=O)c1cccc2NCCc12
CC1(C)N(C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C1=O)c1cccc(c1)[N+]([O-])=O
CC1(C)N(C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C1=O)c1cccc(N)c1
CC(=O)Nc1cccc(c1)N1C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C(=O)C1(C)C
CC(=O)N1CCc2c1cccc2N1C(=O)N(Cc2ccc(cn2)-c2nnc(o2)C(F)F)C(=O)C1(C)C
FC(F)c1nnc(o1)-c1ccc(COc2ccccn2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccnc2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccncc2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cncc(F)c2)nc1
FC(F)c1nnc(o1)-c1ccc(COCC23CC4CC(CC(C4)O2)C3)nc1 |TLB:24:15:22:20.19.18,14:15:20:22.17.18,THB:16:15:20:22.17.18,16:17:20:15.24.23,24:19:22:15.16.23|
FC(F)c1nnc(o1)-c1ccc(COCC2CC3CCC(C2)N3)nc1
CN1C[C@@]2(COCc3ccc(cn3)-c3nnc(o3)C(F)F)C[C@@H]1CO2 |r|
FC(F)c1nnc(o1)-c1ccc(COc2cccc(CC#N)c2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc3ocnc23)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc3nccnc3c2)nc1
Cn1ncc2cc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)ccc12
Cc1nc2ccc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)cc2o1
FC(F)c1nnc(o1)-c1ccc(COc2ccc3ocnc3c2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc3CCCCc3c2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc3cncnc23)nc1
Cn1cnc2cc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)ccc12
Cn1ncc2c(OCc3ccc(cn3)-c3nnc(o3)C(F)F)cccc12
Cc1noc2cc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)ccc12
Cc1noc2cccc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)c12
Cc1nc2cc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)ccc2o1
FC(F)c1nnc(o1)-c1ccc(COc2cncc3ncccc23)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccon2)nc1
Cn1cc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)cn1
Cn1ccc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)n1
Cn1nccc1OCc1ccc(cn1)-c1nnc(o1)C(F)F
FC(F)c1nnc(o1)-c1ccc(COc2cnccn2)nc1
CCn1ccc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)n1
Cc1ccc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)cn1
Cc1ccnc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)c1
Cc1cccc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)n1
Cc1cccnc1OCc1ccc(cn1)-c1nnc(o1)C(F)F
Cc1cc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)ccn1
Cc1cnccc1OCc1ccc(cn1)-c1nnc(o1)C(F)F
FC(F)c1nnc(o1)-c1ccc(COc2ccc(F)cn2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ncccc2F)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ncccn2)nc1
CC(C)n1ccc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)n1
Cc1nc(Cl)cc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)n1
Cc1ncc(F)c(OCc2ccc(cn2)-c2nnc(o2)C(F)F)n1
FC(F)c1nnc(o1)-c1ccc(COc2cccn3ccnc23)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(nn2)C2CC2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(cn2)C2CC2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2nccn3ccnc23)nc1
FC(F)c1nnc(o1)-c1ccc(COc2nnc3ccccn23)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cncc3ccccc23)nc1
Cc1ccc2nnc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)n2c1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(nc2)C(F)(F)F)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc(n2)C(F)(F)F)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cncc(c2)C(F)(F)F)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(cn2)C(F)(F)F)nc1
Cc1ccc2ncnc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)c2c1
Cc1cccc2c(OCc3ccc(cn3)-c3nnc(o3)C(F)F)ncnc12
Cc1nc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)c2ccccc2n1
FC(F)c1nnc(o1)-c1ccc(COc2ncnc3cc(Cl)ccc23)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccnc(n2)N2CCOCC2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ncco2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cncnc2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccnn2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccncn2)nc1
Cn1ccnc1OCc1ccc(cn1)-c1nnc(o1)C(F)F
FC(F)c1nnc(o1)-c1ccc(COc2ncc(F)cn2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ncncc2F)nc1
FC(F)c1nnc(o1)-c1ccc(COC2CC3CCC(C2)O3)nc1
FC(F)c1nnc(o1)-c1ccc(CO[C@H]2C[C@@H]3CC[C@H](C2)O3)nc1 |r|
CN1[C@H]2CC[C@@H]1C[C@H](C2)OCc1ccc(cn1)-c1nnc(o1)C(F)F |r,TLB:0:1:4.3:7.6.8|
FC(F)c1nnc(o1)-c1ccc(COc2ccc(cc2)C#N)nc1
FC(F)c1nnc(o1)-c1ccc(COCc2ccc(s2)C#N)nc1
CN1CCc2cc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)ccc2C1
NC(=O)c1ccc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)cc1
FC(F)c1nnc(o1)-c1cnc(COc2cccn3ccnc23)c(F)c1
Cc1noc2cccc(OCc3ncc(cn3)-c3nnc(o3)C(F)F)c12
Cc1noc2cc(OCc3ncc(cn3)-c3nnc(o3)C(F)F)ccc12
Cc1noc2cc(OCc3ncc(cc3F)-c3nnc(o3)C(F)F)ccc12
Cn1ncc2cc(OCc3ncc(cn3)-c3nnc(o3)C(F)F)ccc12
Cn1ncc2cc(OCc3ncc(cc3F)-c3nnc(o3)C(F)F)ccc12
Cc1nc2cc(OCc3ncc(cn3)-c3nnc(o3)C(F)F)ccc2o1
Cc1nc2cc(OCc3ncc(cc3F)-c3nnc(o3)C(F)F)ccc2o1
FC(F)c1nnc(o1)-c1cnc(COc2ccc3ocnc3c2)nc1
FC(F)c1nnc(o1)-c1cnc(COc2cccc3ocnc23)nc1
Cn1cnc2cc(OCc3ncc(cn3)-c3nnc(o3)C(F)F)ccc12
Cn1cnc2cc(OCc3ncc(cc3F)-c3nnc(o3)C(F)F)ccc12
FC(F)c1nnc(o1)-c1cnc(COc2ccc3nccnc3c2)nc1
FC(F)c1nnc(o1)-c1cnc(COc2ccc3nccnc3c2)c(F)c1
FC(F)c1nnc(o1)-c1cnc(COc2cccc3nccnc23)nc1
FC(F)c1nnc(o1)-c1cnc(COc2cccc3nccnc23)c(F)c1
FC(F)c1nnc(o1)-c1cnc(COc2cccc3cncnc23)nc1
FC(F)c1nnc(o1)-c1cnc(COc2cccc3cncnc23)c(F)c1
FC(F)c1nnc(o1)-c1cnc(COc2cccnc2)nc1
FC(F)c1nnc(o1)-c1cnc(COc2ccc(cc2)C#N)nc1
FC(F)c1nnc(o1)-c1cnc(COc2ccc(cc2)C#N)c(F)c1
FC(F)c1nnc(o1)-c1cnc(COc2cccc(c2)C#N)c(F)c1
FC(F)c1nnc(o1)-c1cnc(COc2ccccc2C#C)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc3CNCCc3c2)nc1
Cn1cc2cc(OCc3ncc(cc3F)-c3nnc(o3)C(F)F)ccc2n1
FC(F)c1nnc(o1)-c1ccc(COc2cnc3ccnn3c2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccn3cnnc3c2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(cc2)-c2ccccc2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccnc(c2)-c2ccccc2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccccc2-c2ccccc2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc(c2)-c2ccccc2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccnc(Cl)c2)nc1
CN1CCc2c(OCc3ccc(cn3)-c3nnc(o3)C(F)F)noc2C1
CN1CCc2onc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)c2C1
Cc1c[nH]c(n1)-c1cc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)ccn1
Cn1c(nc2ccccc12)-c1ccc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)cc1
Cn1c(nc2ccccc12)-c1cccc(OCc2ccc(cn2)-c2nnc(o2)C(F)F)c1
CCn1cnc2ccc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)cc12
CC(C)n1cnc2ccc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)cc12
Cn1nc(ccc1=O)-c1nc2ccc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)cc2o1
FC(F)c1nnc(o1)-c1ccc(COc2cnc(nc2)C(F)(F)F)nc1
FC(F)c1nnc(o1)-c1ccc(COc2cccc(c2)-c2nc3ccccc3[nH]2)nc1
FC(F)c1nnc(o1)-c1ccc(COc2ccc(cc2)-c2nc3ccccc3[nH]2)nc1
Cn1cnc2c(OCc3ccc(cn3)-c3nnc(o3)C(F)F)cccc12
FC(F)c1nnc(o1)-c1ccc(COc2ccc3n(CCN4CCCC4)cnc3c2)nc1
CN(C)CCn1cnc2cc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)ccc12
CCn1cnc2cc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)ccc12
CC(C)n1cnc2cc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)ccc12
Cn1cnc2ccc(OCc3ccc(cn3)-c3nnc(o3)C(F)F)cc12
FC(F)c1nnc(o1)-c1ccc(COc2ccc(cc2)-c2nn[nH]n2)nc1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(C)F)c1ccc2cnn(C)c2c1
CCN\C=C(/C=N)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)S(=O)(=O)CC
CCS(=O)(=O)N(Cc1ncc(s1)C(=N)OC(=N)C(F)F)c1cc2COCCn2n1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cnc[nH]1
CCS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cccc(C)n1
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)(F)F)c1cccc(F)c1
CCS(=O)(=O)N(Cc1cnc(s1)-c1nnc(o1)C(F)F)c1cncc(OC(F)F)c1
CS(=O)(=O)N(Cc1cnc(s1)-c1nnc(o1)C(F)F)c1cncc(Cl)c1
CS(=O)(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1cncc(OC(F)(F)F)c1
ONC(=O)c1cncc(F)c1
Cc1ncc(cc1F)C(=O)NO
ONC(=O)c1cnc(NC2(CC2)c2ccccc2)c(F)c1
ONC(=O)c1cnc(CNC2(CC2)c2ccccc2)c(F)c1
ONC(=O)c1cnc(NCC2(CC2)c2ccccc2)c(F)c1
ONC(=O)c1cnc(NC2Cc3ccccc3C2)c(F)c1
C[C@@H](Nc1ncc(cc1F)C(=O)NO)c1ccccc1 |r|
C[C@H](Nc1ncc(cc1F)C(=O)NO)c1ccccc1 |r|
Nc1ncc(cc1F)C(=O)NO
ONC(=O)c1cnc(NS(=O)(=O)c2ccccc2)c(F)c1
COc1ncc(cc1F)C(=O)NO
COc1ccccc1N1CCN(CC1)c1ncc(cc1F)C(=O)NO
ONC(=O)c1cnc(N2CCc3ccccc3C2)c(F)c1
ONC(=O)c1cnc(N[C@H](C2CC2)c2ccccn2)c(F)c1 |r|
ONC(=O)c1cnc(N[C@@H](C2CC2)c2ccccn2)c(F)c1 |r|
ONC(=O)c1cnc(N2CCC(CC2)c2ccccc2)c(F)c1
CC(C)(Nc1ncc(cc1F)C(=O)NO)c1ccccn1
ONC(=O)c1cnc(NC2(CC2)c2c(F)cccc2F)c(F)c1
ONC(=O)c1cnc(NC2(CC2)c2ccccn2)c(F)c1
CN(C)c1ncc(cc1F)C(=O)NO
ONC(=O)c1cnc(N[C@@H](C2CC2)c2ccccc2)c(F)c1 |r|
CN(Cc1ncc(cc1F)C(=O)NO)C1(CC1)c1ccccc1
ONC(=O)c1cnc(CN(CC2COC2)C2(CC2)c2ccccc2)c(F)c1
ONC(=O)c1cnc(NC(c2ccccc2)c2ccccc2)c(F)c1
Cc1nc2ccccc2n1Cc1ncc(cc1F)C(=O)NO
ONC(=O)c1cnc(N2CCc3ncccc3C2)c(F)c1
CN(c1ncc(cc1F)C(=O)NO)C1(CC1)c1ccccc1
ONC(=O)c1cnc(C2CC2)c(F)c1
ONC(=O)c1cnc(OC2(CC2)c2ccccc2)c(F)c1
ONC(=O)c1cnc(N2CCS(=O)(=O)CC2)c(F)c1
CC[C@H](Nc1ncc(cc1F)C(=O)NO)c1ccccc1 |r|
CN1CCC2C(C1)c1ccccc1N2Cc1ncc(cc1F)C(=O)NO
ONC(=O)c1cnc(CN2Cc3ccccc3OC2=O)c(F)c1
CN1CCN(CC1)c1ncc(cc1F)C(=O)NO
ONC(=O)c1cnc(CN2CCc3ccccc3C2)c(F)c1
ONC(=O)c1cnc(NC(C2CC2)C2CC2)c(F)c1
ONC(=O)c1cnc(N[C@H](C2CC2)c2ccccc2)c(F)c1 |r|
ONC(=O)c1cnc(Cn2ccc3cccnc23)c(F)c1
C[C@H](Nc1ncc(cc1F)C(=O)NO)C1CC1 |r|
C[C@@H](Nc1ncc(cc1F)C(=O)NO)C1CC1 |r|
ONC(=O)c1cnc(Cn2c(nc3ccccc23)C(F)F)c(F)c1
ONC(=O)c1cnc(NC2(COC2)c2ccccc2)c(F)c1
CC[C@@H](Nc1ncc(cc1F)C(=O)NO)c1ccccc1 |r|
ONC(=O)c1cnc(CN2C3COCCC3c3ccccc23)c(F)c1
C[C@@H](Nc1ncc(cc1F)C(=O)NO)C1CCCCC1 |r|
C[C@H](Nc1ncc(cc1F)C(=O)NO)C1CCCCC1 |r|
ONC(=O)c1cnc(NC2(CC2)C(F)(F)F)c(F)c1
ONC(=O)c1cnc(NC2CC(F)(F)C2)c(F)c1
CNC(=O)C(C)(C)Nc1ncc(cc1F)C(=O)NO
CC1(C)Oc2cccnc2N(Cc2ncc(cc2F)C(=O)NO)C1=O
CN1CCCC(Nc2ncc(cc2F)C(=O)NO)C1=O
CO[C@@H]1CCC[C@@H]1Nc1ncc(cc1F)C(=O)NO |r|
CC(CC12CC3CC(CC(C3)C1)C2)NCc1ccc(cc1)C(=O)NO |TLB:12:3:10:6.7.8,2:3:6:10.9.8,2:3:10:6.7.8,THB:12:7:10:11.4.3,11:9:6:12.4.3,11:3:6:10.9.8|
CC(CC12CC3CC(CC(C3)C1)C2)N(C)Cc1ccc(cc1)C(=O)NO |TLB:12:3:10:6.7.8,2:3:6:10.9.8,2:3:10:6.7.8,THB:12:7:10:11.4.3,11:9:6:12.4.3,11:3:6:10.9.8|
C[C@@H](c1ccc(cc1)C(=O)Nc1ccc(F)cc1N)n1nc(ccc1=O)-c1ccc(CN(C)C)cc1 |r|
CC(c1ccc(cc1)C(=O)Nc1ccc(F)cc1N)n1nc(ccc1=O)-c1ccc(CN(C)C)cc1
C[C@H](c1ccc(cc1)C(=O)Nc1ccc(F)cc1N)n1nc(ccc1=O)-c1ccc(CN(C)C)cc1 |r|
C[C@@H](c1ccc(cc1)C(=O)Nc1ccccc1N)n1nc(ccc1=O)-c1ccc(CN(C)C)cc1 |r|
CC(c1ccc(cc1)C(=O)Nc1ccccc1N)n1nc(ccc1=O)-c1ccc(CN(C)C)cc1
C[C@H](c1ccc(cc1)C(=O)Nc1ccccc1N)n1nc(ccc1=O)-c1ccc(CN(C)C)cc1 |r|
C[C@@H](c1ccc(cc1)C(=O)Nc1ccccc1N)n1nc(ccc1=O)-c1cccc(Cl)c1 |r|
CC(c1ccc(cc1)C(=O)Nc1ccccc1N)n1nc(ccc1=O)-c1cccc(Cl)c1
COc1cccc(c1)-c1ccc(=O)n(n1)[C@@H](C)c1ccc(cc1)C(=O)Nc1ccccc1N |r|
COc1cccc(c1)-c1ccc(=O)n(n1)C(C)c1ccc(cc1)C(=O)Nc1ccccc1N
C[C@@H](c1ccc(cc1)C(=O)Nc1ccccc1N)n1nc(ccc1=O)-c1cnn(C)c1 |r|
C[C@@H](c1ccc(cc1)C(=O)Nc1ccccc1N)n1nc(ccc1=O)-c1ccncc1 |r|
C[C@@H](c1ccc(cc1)C(=O)Nc1cc(F)c(F)cc1N)n1nc(ccc1=O)-c1ccc(CN(C)C)cc1 |r|
COc1ccc(NC(=O)c2ccc(cc2)[C@H](C)n2nc(ccc2=O)-c2ccc(CN(C)C)cc2)c(N)c1 |r|
C[C@@H](c1ccc(cc1)C(=O)Nc1cccc(F)c1N)n1nc(ccc1=O)-c1ccc(CN(C)C)cc1 |r|
C[C@@H](c1ccc(cc1)C(=O)Nc1ccccc1N)n1nc(ccc1=O)-c1ccccc1 |r|
C[C@H](c1ccc(cc1)C(=O)Nc1ccccc1N)n1nc(ccc1=O)-c1ccccc1 |r|
COc1ccc(N)c(NC(=O)c2ccc(cc2)[C@H](C)n2nc(ccc2=O)-c2ccc(CN(C)C)cc2)c1 |r|
C[C@@H](c1ccc(cc1)C(=O)Nc1cc(F)ccc1N)n1nc(ccc1=O)-c1ccc(CN(C)C)cc1 |r|
C[C@@H](c1ccc(cc1)C(=O)Nc1cc(C)ccc1N)n1nc(ccc1=O)-c1ccc(CN(C)C)cc1 |r|
Nc1ccc(F)cc1NC(=O)c1ccc(CNC(=O)\C=C\c2cccnc2)cc1
FC(F)c1nnc(o1)-c1ccc(CN(C(=S)N2CCOCC2)c2ccccc2)c(F)c1
FC(F)c1nnc(o1)-c1ccc(CN(C(=S)N2CCOCC2)c2ccccc2)nc1
FC(F)c1nnc(o1)-c1ccc(CN(C(=S)N2CCOCC2)c2ccccc2)cc1
CN1CCN(CC1)C(=S)N(Cc1ccc(cc1)-c1nnc(o1)C(F)F)c1ccccc1
FC(F)c1nnc(o1)-c1ccc(CN(C(=S)N2CCN(CC2)C2COC2)c2ccccc2)cc1
FC(F)c1nnc(o1)-c1ccc(CN(C(=S)N2CCS(=O)(=O)CC2)c2ccccc2)nc1
CN1CCN(CC1)C(=S)N(Cc1ccc(cc1F)-c1nnc(o1)C(F)F)c1ccccc1
CN1CCC2(CC(C2)C(=S)N(Cc2ccc(cc2F)-c2nnc(o2)C(F)F)c2ccccc2)CC1
FC(F)c1nnc(o1)-c1ccc(CN(C(=S)c2ccncc2)c2ccccc2)c(F)c1
CN1CC2(C1)CN(C2)C(=S)N(Cc1ccc(cc1F)-c1nnc(o1)C(F)F)c1ccccc1
FC(F)c1nnc(o1)-c1ccc(CN(C(=S)N2CC3(CN(C3)C3COC3)C2)c2ccccc2)c(F)c1
CN1CC2(C1)CN(C2)C(=S)N(Cc1ccc(cc1F)-c1nnc(o1)C(F)F)c1ccc(F)cc1F
CN1CC2(C1)CN(C2)C(=S)N(Cc1ccc(cc1F)-c1nnc(o1)C(F)F)c1ccc(F)c(F)c1
CN1CC2(C1)CN(C2)C(=S)N(Cc1ccc(cc1)-c1nnc(o1)C(F)F)c1cccc(F)c1
FC(F)c1nnc(o1)-c1ccc(CN(C(=S)N2CC3(CN(C3)C3COC3)C2)c2cccc(F)c2)cc1
CC(C)N1CC2(C1)CN(C2)C(=S)N(Cc1ccc(cc1)-c1nnc(o1)C(F)F)c1cccc(F)c1
CN1CC2(C1)CN(C2)C(=S)N(Cc1ccc(cc1F)-c1nnc(o1)C(F)F)c1ccc(F)cc1
CC(C)N1CC2(C1)CN(C2)C(=S)N(Cc1ccc(cc1F)-c1nnc(o1)C(F)F)c1ccc(F)cc1
FC(F)c1nnc(o1)-c1ccc(CN(C(=S)N2CC3(CN(C3)C3COC3)C2)c2ccc(F)cc2)c(F)c1
CN1CC2(C1)CN(C2)C(=S)N(Cc1ccc(cc1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
CC(C)N1CC2(C1)CN(C2)C(=S)N(Cc1ccc(cc1)-c1nnc(o1)C(F)F)c1ccc(F)cc1
FC(F)c1nnc(o1)-c1ccc(CN(C(=S)N2CC3(CN(C3)C3COC3)C2)c2ccc(F)cc2)cc1
CN1CC2(C1)CN(C2)C(=S)N(Cc1ccc(cc1F)-c1nnc(o1)C(F)F)c1ccc(Cl)c(Cl)c1
FC(F)c1nnc(o1)-c1ccc(CN(C(=S)N2CC3(CN(C3)C3COC3)C2)c2ccc(Cl)c(Cl)c2)c(F)c1
CN1CC2(C1)CN(C2)C(=S)N(Cc1ccc(cc1F)-c1nnc(o1)C(F)F)c1ccc(F)c(Cl)c1
CN1CC2(C1)CN(C2)C(=S)N(Cc1ccc(cc1)-c1nnc(o1)C(F)F)c1ccc(F)c(Cl)c1
FC(F)c1nnc(o1)-c1ccc(CN(C(=S)N2CC3(CN(C3)C3COC3)C2)c2ccc(F)c(Cl)c2)cc1
CC(C)N1CC2(C1)CN(C2)C(=S)N(Cc1ccc(cc1F)-c1nnc(o1)C(F)F)c1ccc(F)c(Cl)c1
CC(C)N1CC2(C1)CN(C2)C(=S)N(Cc1ccc(cc1)-c1nnc(o1)C(F)F)c1ccc(F)c(Cl)c1
CN1CC2(C1)CN(C2)C(=S)N(Cc1ccc(cc1)-c1nnc(o1)C(F)F)c1ccc(F)c(F)c1
CC(C)N1CC2(C1)CN(C2)C(=S)N(Cc1ccc(cc1)-c1nnc(o1)C(F)F)c1ccc(F)c(F)c1
FC(F)c1nnc(o1)-c1ccc(CN(C(=S)N2CC3(CN(C3)C3COC3)C2)c2ccc(F)c(F)c2)cc1
CC(=O)N1CC2(C1)CN(C2)C(=S)N(Cc1ccc(cc1F)-c1nnc(o1)C(F)F)c1ccc(F)c(F)c1
FC(F)c1nnc(o1)-c1ccc(CN(C(=S)N2CC3(CN(C3)C3COC3)C2)c2ccc(F)c(F)c2)c(F)c1
FC(F)c1nnc(o1)-c1ccc(CN(C(=S)N2CC3(COC3)C2)c2ccc(F)c(F)c2)c(F)c1
CN1CC2(C1)CN(C2)C(=S)N(Cc1ccc(cc1F)-c1nnc(o1)C(F)F)c1cccc(F)c1
CC(C)N1CC2(C1)CN(C2)C(=S)N(Cc1ccc(cc1F)-c1nnc(o1)C(F)F)c1cccc(F)c1
FC(F)c1nnc(o1)-c1ccc(CN(C(=S)N2CC3(CN(C3)C3COC3)C2)c2cccc(F)c2)c(F)c1
CN1C[C@@H]2C[C@H]1CN2C(=S)N(Cc1ccc(cc1F)-c1nnc(o1)C(F)F)c1ccc(F)cc1 |r|
CC(C)N1C[C@@H]2C[C@H]1CN2C(=S)N(Cc1ccc(cc1F)-c1nnc(o1)C(F)F)c1ccc(F)cc1 |r|
FC(F)c1nnc(o1)-c1ccc(CN(C(=S)N2C[C@@H]3C[C@H]2CN3C2COC2)c2ccc(F)cc2)c(F)c1 |r|
CN1C[C@@H]2C[C@H]1CN2C(=S)N(Cc1ccc(cc1F)-c1nnc(o1)C(F)F)c1ccc(F)c(F)c1 |r|
FC(F)c1nnc(o1)-c1ccc(CN(C(=S)N2C[C@@H]3C[C@H]2CN3C2COC2)c2ccc(F)c(F)c2)c(F)c1 |r|
CN1CC2(C1)CCN(CC2)C(=S)N(Cc1ccc(cc1F)-c1nnc(o1)C(F)F)c1ccc(F)c(F)c1
FC(F)c1nnc(o1)-c1ccc(CN(C(=S)N2CCC3(CN(C3)C3COC3)CC2)c2ccc(F)c(F)c2)c(F)c1
CN1CCC2(CN(C2)C(=S)N(Cc2ccc(cc2F)-c2nnc(o2)C(F)F)c2ccc(F)c(F)c2)CC1
CN(C)C(=O)N(Cc1ncc(s1)-c1nnc(o1)C(F)F)c1ccccn1
CC(C)S(=O)(=O)N(Cc1cnc(s1)-c1nnc(o1)C(F)F)c1cccnc1
FC(F)c1nnc(-c2ccc(Cn3ccc4ccccc43)cc2)o1
FC(F)c1nnc(-c2ccc(Cn3ccc4ncccc43)cc2)o1
FC(F)c1nnc(-c2ccc(Cn3ccc4cnccc43)cc2)o1
FC(F)c1nnc(-c2ccc(Cn3ccc4cccnc43)cc2)o1
O=C(c1cn(Cc2ccc(-c3nnc(C(F)F)o3)cc2)c2ccccc12)C(F)F
FC(F)c1nnc(-c2ccc(Cn3ncc4ccccc43)cc2)o1
FC(F)c1nnc(-c2ccc(Cn3cc4ccccc4n3)cc2)o1
FC(F)c1nnc(-c2ccc(Cn3cnc4ccccc43)cc2)o1
O=C(c1nc2cc(Cl)c(Cl)cc2n1Cc1ccc(-c2nnc(C(F)F)o2)cc1)C(F)F
FC(F)c1nnc(-c2ccc(Cn3cnc4cc(Cl)c(Cl)cc43)cc2)o1
FC(F)c1nnc(-c2ccc(Cn3nnc4ccccc43)cc2)o1
Cc3cccc4nnn(Cc2ccc(c1nnc(C(F)F)o1)cc2)c34
FC(F)c1nnc(-c2ccc(Cn3nnc4ccc(Cl)cc43)cc2)o1
O=c1ccc2ccccc2n1Cc1ccc(-c2nnc(C(F)F)o2)cc1
CC1(C)C(=O)N(Cc2ccc(-c3nnc(C(F)F)o3)cc2)c2ccccc21
O=C1c2ccccc2C(=O)N1Cc1ccc(-c2nnc(C(F)F)o2)cc1
FC(F)c1nnc(-c2ccc(Cn3nnnc3-c3ccccc3)cc2)o1
O=c1n(-c2ccccc2)cnn1Cc1ccc(-c2nnc(C(F)F)o2)cc1
O=C1N(Cc2ccc(-c3nnc(C(F)F)o3)cc2)c2ccccc2C12CCOCC2
CC(c1ccc(-c2nnc(C(F)F)o2)cc1)n1cnc2ccccc21
FC(F)c1nnc(-c2ccc(Cn3nnc4ccccc43)nc2)o1
FC(F)c1nnc(-c2ccc(Cn3cnc4cc(Cl)c(Cl)cc43)nc2)o1
FC(F)c1nnc(-c2ccc(Cn3nnc4cccnc43)nc2)o1
FC(F)c1nnc(-c2ccc(Cn3nnc4cc(Cl)c(Cl)cc43)nc2)o1
FC(F)c1nnc(-c2ccc(Cn3nc4cc(Cl)c(Cl)cc4n3)nc2)o1
FC(F)c1nnc(-c2ccc(Cn3cnc(-c4ccccc4)c3)nc2)o1
COC(=O)c1cn(Cc2ccc(-c3nnc(C(F)F)o3)cc2)nn1
FC(F)c1nnc(-c2ccc(Cn3cc(-c4ccc(Cl)cc4)nn3)cc2)o1
FC(F)c4nnc(c3ccc(Cn2cc(c1ccc(C(F)(F)F)cc1)nn2)cc3)o4
CC(C)(C)c1cn(Cc2ccc(-c3nnc(C(F)F)o3)cc2)nn1
FC(F)c1nnc(-c2ccc(Cn3cc(C4CCCCC4)nn3)cc2)o1
Cc1nnn(Cc2ccc(-c3nnc(C(F)F)o3)cc2)c1-c1ccccc1
Fc1ccccc1-c1nnn(Cc2ccc(-c3nnc(C(F)F)o3)cn2)c1Cl
FC(F)c1nnc(-c2ccc(Cn3cc(-c4ccncc4)nn3)cc2)o1
FC(F)c1nnc(-c2ccc(Cn3cc(-c4cccnc4)nn3)cc2)o1
FC(F)c1nnc(-c2ccc(Cn3cc(-c4ccsc4)nn3)cc2)o1
FC(F)c1nnc(-c2ccc(Cn3cc(-c4cccs4)nn3)cc2)o1
CC(c1ccc(-c2nnc(C(F)F)o2)cc1)n1cc(-c2ccccc2)nn1
FC(F)c1nnc(-c2ccc(Cn3nnc(-c4ccccc4)c3-c3ccccc3)cc2)o1
Cc1c(-c2ccccc2)nnn1Cc1ccc(-c2nnc(C(F)F)o2)cc1
FC(F)c1nnc(-c2ccc(Cn3cc(-c4ccccc4)nn3)nc2)o1
FC(F)c1nnc(-c2ccc(Cn3cc(-c4ccccc4)nn3)cn2)o1
FC(F)c1nnc(-c2ccc(Cn3cc(-c4ccc(Cl)cc4)nn3)nc2)o1
FC(F)c1nnc(-c2ccc(Cn3cc(-c4ccccc4Cl)nn3)nc2)o1
FC(F)c1nnc(-c2ccc(Cn3cc(-c4cccc(Cl)c4)nn3)nc2)o1
FC(F)c1nnc(-c2ccc(Cn3cc(-c4ccc(Cl)c(Cl)c4)nn3)nc2)o1
FC(F)c1nnc(-c2ccc(Cn3cc(-c4cc(Cl)cc(Cl)c4)nn3)nc2)o1
Fc1ccccc1-c1cn(Cc2ccc(-c3nnc(C(F)F)o3)cn2)nn1
Fc1cccc(F)c1-c1cn(Cc2ccc(-c3nnc(C(F)F)o3)cn2)nn1
COc4cccc(c3cn(Cc2ccc(c1nnc(C(F)F)o1)cn2)nn3)c4
FC(F)c1nnc(-c2ccc(Cn3nnc(-c4ccccc4)c3Cl)cc2)o1
FC(F)c1nnc(-c2ccc(Cn3nnc(-c4ccccc4)c3Cl)nc2)o1
FC(F)c1nnc(-c2ccc(Cn3nnc(-c4ccccc4Cl)c3Cl)nc2)o1
FC(F)c1nnc(-c2ccc(Cn3nnc(-c4cccc(Cl)c4)c3Cl)nc2)o1
FC(F)c1nnc(-c2ccc(C(Cl)n3cc(-c4ccccc4)nn3)nc2)o1
Fc1cc(F)cc(-c2cn(Cc3ccc(-c4nnc(C(F)F)o4)cn3)nn2)c1
Fc1cc(-c2cn(Cc3ccc(-c4nnc(C(F)F)o4)cn3)nn2)cc(F)c1F
FC(F)c1nnc(-c2ccc(Cn3c(C(F)(F)F)nc4cc(Cl)c(Cl)cc43)nc2)o1
Cc1cc2nnn(Cc3ccc(-c4nnc(C(F)F)o4)cn3)c2cc1C
Cc1nc2cc(Cl)c(Cl)cc2n1Cc1ccc(-c2nnc(C(F)F)o2)cn1
Cc1cc2ncn(Cc3ccc(-c4nnc(C(F)F)o4)cn3)c2cc1C
FC(F)c1nnc(-c2ccc(Cn3cnc4ccc(Br)cc43)nc2)o1
FC(F)c1nnc(-c2ccc(Cn3cnc4cc(Br)ccc43)nc2)o1
FC(F)c1nnc(-c2ccc(Cn3nnc4cc(Br)ccc43)nc2)o1
FC(F)c1nnc(-c2ccc(Cn3nnc4ccc(Br)cc43)nc2)o1
FC(F)c1nnc(-c2ccc(Cn3nc4ccc(Br)cc4n3)nc2)o1
COc1cc2c(Oc3ccc(NC(=O)C4(C(=O)Nc5ccc(F)cc5)CC4)cc3F)ccnc2cc1OCCCCCCSC(C)=O
COc1cc2c(Oc3ccc(NC(=O)C4(C(=O)Nc5ccc(F)cc5)CC4)cc3F)ccnc2cc1OCCCCCCS
COc1cc2c(Oc3ccc(NC(=O)C4(C(=O)Nc5ccc(F)cc5)CC4)cc3F)ccnc2cc1OCCCCCCCSC(C)=O
COc1cc2c(Oc3ccc(NC(=O)C4(C(=O)Nc5ccc(F)cc5)CC4)cc3F)ccnc2cc1OCCCCCCCS
COc1cc2c(Oc3ccc(NC(=O)C4(C(=O)Nc5ccc(F)cc5)CC4)cc3F)ccnc2cc1OC/C=C/CCCCS
COc1cc2c(Oc3ccc(NC(=O)C4(C(=O)Nc5ccc(F)cc5)CC4)cc3F)ccnc2cc1OC/C=C/CCSC(C)=O
COc1cc2c(Oc3ccc(NC(=O)C4(C(=O)Nc5ccc(F)cc5)CC4)cc3F)ccnc2cc1OC/C=C/CCS
COc1cc2nccc(Oc3ccc(NC(=O)C4(CC4)C(=O)Nc4ccc(F)cc4)cc3)c2cc1OC
COc1cc2c(Oc3ccc(NC(=O)C4(C(=O)Nc5ccc(F)cc5)CC4)cc3F)ccnc2cc1OCCCCCNC(=O)CSC(C)=O
COc1cc2c(Oc3ccc(NC(=O)C4(C(=O)Nc5ccc(F)cc5)CC4)cc3F)ccnc2cc1OCCCCCNC(=O)CS
COc1cc2c(Oc3ccc(NC(=O)C4(C(=O)Nc5ccc(F)cc5)CC4)cc3F)ccnc2cc1OCCCCNC(=O)CSC(C)=O
COc1cc2c(Oc3ccc(NC(=O)C4(C(=O)Nc5ccc(F)cc5)CC4)cc3F)ccnc2cc1OCCCCNC(=O)CS
COc1cc2c(Oc3ccc(NC(=O)C4(C(=O)Nc5ccc(F)cc5)CC4)cc3F)ccnc2cc1OCCCCCCNC(=O)CSC(C)=O
COc1cc2c(Oc3ccc(NC(=O)C4(C(=O)Nc5ccc(F)cc5)CC4)cc3F)ccnc2cc1OCCCCCCNC(=O)CS
CC(=O)SCC(=O)NCCCCCOc1cc2nccc(Oc3ccc(NC(=O)NC4CC4)c(Cl)c3)c2cc1C(N)=O
CC(=O)SCC(=O)NCCCCCOc1cc2nccc(Oc3ccc(NC(=O)C4(C(=O)Nc5ccc(F)cc5)CC4)cc3F)c2cc1C(N)=O
O=C(NO)c1ccc(Cn2cc(CN[C@@H]3C[C@H]3c3ccccc3)cn2)cc1
O=C(NO)c1ccc(Cn2cc(CN[C@H]3CC3c3ccccc3)cn2)cc1
O=C(NO)c1ccc(CCCN2CCC(CN[C@@H]3C[C@H]3c3cnn(-c4ccccc4)c3)CC2)cc1
O=C(NO)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3cnn(-c4ccccc4)c3)CC2)cc1
O=C(NO)c1ccc(/C=C/C(=O)N2CC(CN[C@@H]3C[C@H]3c3ccc(F)cc3)C2)cc1
O=C(NO)c1ccc(/C=C/C(=O)N2CC(CN[C@H]3C[C@@H]3c3ccc(F)cc3)C2)cc1
O=C(NO)c1ccc(CCCN2CCC(CN[C@@H]3C[C@H]3c3ccc(-c4cncnc4)cc3)CC2)cc1
O=C(NO)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccc(-c4cncnc4)cc3)CC2)cc1
CN1C(=O)C(C)(C)c2cc([C@@H]3C[C@H]3NCC3CCN(CCCc4ccc(C(=O)NO)cc4)CC3)ccc21
CN1C(=O)C(C)(C)c2cc([C@H]3C[C@@H]3NCC3CCN(CCCc4ccc(C(=O)NO)cc4)CC3)ccc21
ONC(=O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 |r|
ONC(=O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 |r|
ONC(=O)c1ccc(CCCN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 |r|
ONC(=O)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 |r|
Nc1ccccc1NC(=O)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccc(F)c(F)c3)CC2)cc1
Nc1ccccc1NC(=O)c1ccc(Cn2cc(CN[C@@H]3C[C@H]3c3ccccc3)cn2)cc1
O=C(NO)c1cnc2c(c1)CCN(CC13CC4CC(CC(C4)O1)C3)C2
O=C(NO)c1cnc2c(c1)CCN(C1CC3(CCCCC3)C1)C2
O=C(NO)c1cnc2c(c1)CCN(C1CC3(CCOCC3)C1)C2
O=C(NO)c4cnc3CN(C2CC1(CCCC1)C2)CCc3c4
O=C(NO)c4cnc3CN(C2CC1(CCOC1)C2)CCc3c4
O=C(NO)c4cnc3CN(C2CC1(CCOC1)C2)CCc3c4
O=C(NO)c1cnc2c(c1)CCN(C1CCC3(CCC3)CC1)C2
O=C(NO)c4cnc3CN([C@@H]2CCCC1(CCC1)C2)CCc3c4
O=C(NO)c1cnc2c(c1)CCN([C@H]1CCCC3(CCC3)C1)C2
O=C(NO)c4cnc3CN(C2CC1(CCNCC1)C2)CCc3c4
CN1CCC2(CC1)CC(N1CCc3cc(C(=O)NO)cnc3C1)C2
CC(=O)N1CCC2(CC1)CC(N1CCc3cc(C(=O)NO)cnc3C1)C2
O=C(NO)c1cnc2c(c1)CCN(C1CC3(CNC3)C1)C2
O=C(NO)c1cnc2c(c1)CCN(C1CC3(CCCNC3)C1)C2
O=C(NO)c1cnc2c(c1)CCN(C1CC3(CCCNC3)C1)C2
CN1CCC[C@]2(C1)C[C@@H](N1CCc3cc(C(=O)NO)cnc3C1)C2
CN1CCC[C@]2(C1)C[C@H](N1CCc3cc(C(=O)NO)cnc3C1)C2
O=C(NO)c4cnc3CN([C@H]2CCC1(CCC1)C2)CCc3c4
O=C(NO)c4cnc3CN([C@@H]2CCC1(CCC1)C2)CCc3c4
CN1CCC2(CCC(N3CCc4cc(C(=O)NO)cnc4C3)C2)CC1
O=C(NO)c1cc2c(cn1)CN(C1CC3(CCCCC3)C1)CC2
O=C(NO)c1ccc2c(n1)CCN(C1CC3(CCCCC3)C1)C2
O=C(NO)c1cnc2c(c1)CCN(C1CC3(CCNCC3)C1)C2
CN1CC(C(=O)N[C@@H](CCCCCC(=O)c2ncco2)c2nc(-c3ccc(F)cc3)c[nH]2)C1
O=C(CCCCC[C@H](NC(=O)c1cncs1)c1nc(-c2ccc(F)cc2)c[nH]1)c1ncco1
CN1CCC(C(=O)N[C@@H](CCCCCC(=O)c2ncco2)c2nc(-c3ccc(F)cc3)c[nH]2)CC1
O=C(CCCCC[C@H](NC(=O)[C@H]1CC12CCOCC2)c1nc(-c2ccc(F)cc2)c[nH]1)c1ncco1
CN1CCC(C(=O)N[C@@H](CCCCCC(=O)c2nccs2)c2nc(-c3ccc(F)cc3)c[nH]2)CC1
O=C(N[C@@H](CCCCCC(=O)c1nccs1)c1nc(-c2ccc(F)cc2)c[nH]1)c1cncs1
Cc1coc(C(=O)CCCCC[C@H](NC(=O)C2CCN(C)CC2)c2nc(-c3ccc(F)cc3)c[nH]2)n1
Cc1ccc2c(n1)=CCC(C1=CNC([C@@H](N)CCCCCC(=O)C3NC=CO3)N1)C=2
CCn1ccc2c(c1=O)=CCC(C1=CNC([C@@H](N)CCCCCC(=O)C3NC=CO3)N1)C=2
COc1nc(C)ccc1-c1c[nH]c([C@@H](N)CCCCCC(=O)c2ncco2)n1
COc1cc2nc(C)ccc2cc1-c1c[nH]c([C@@H](N)CCCCCC(=O)c2ncco2)n1
COc1nc2cnccc2cc1-c1c[nH]c([C@@H](N)CCCCCC(=O)c2ncco2)n1
N[C@@H](CCCCCC(=O)c1ncco1)c1nc(-c2ccc3nn(C4CC4)cc3c2)c[nH]1
COc1nc2ccccc2cc1-c1c[nH]c([C@@H](N)CCCCCC(=O)c2ncco2)n1
N[C@@H](CCCCCC(=O)C1NC=CO1)C1NC=C(C2C=c3cccnc3=CC2)N1
CC(C)n1ccc2cc(-c3cnc([C@@H](N)CCCCCC(=O)c4ncco4)[nH]3)ccc2c1=O
CN(C)c1ccc2cc(-c3cnc([C@@H](N)CCCCCC(=O)c4ncco4)[nH]3)ccc2n1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2ccc3nc(N4CCCC4)ccc3c2)[nH]1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2ccc(-c3cnccn3)cc2)[nH]1
COc1cc2c(ccc(=O)n2C)cc1-c1cnc([C@@H](N)CCCCCC(=O)c2ncco2)[nH]1
Cc1ccc2cc(-c3cnc([C@@H](N)CCCCCC(=O)c4ncco4)[nH]3)c(Cl)cc2n1
COC1C=c2ncccc2=CC1C1=CNC([C@@H](N)CCCCCC(=O)C2NC=CO2)N1
COC1=NC(C2CC2)=CCC1C1=CNC([C@@H](N)CCCCCC(=O)C2NC=CO2)N1
N[C@@H](CCCCCC(=O)C1NC=CO1)c1[nH]c(-c2ccc(F)cc2)nc1Cl
Cc1ccc2c(n1)=CCC(C1=CNC(C(N)CCCCCC(=O)C3NC=CO3)O1)C=2
COC1C=c2nc(C)ccc2=CC1C1=CNC([C@@H](N)CCCCCC(=O)C2NC=CO2)O1
COC1=NC=CCC1C1=CNC([C@@H](N)CCCCCC(=O)C2NC=CO2)O1
Cc1ccc2c(n1)=CCC(C1=CN(C)C([C@@H](N)CCCCCC(=O)C3NC=CO3)N1)C=2
CCn1cc(-c2ccc3nc(C)ccc3c2)nc1[C@@H](N)CCCCCC(=O)c1ncco1
COC1C=c2nc(C)ccc2=CC1C1=CNC([C@@H](N)CCCCCC(=O)c2ccon2)N1
Cn1c(=O)ccc2cc(-c3c[nH]c([C@@H](N)CCCCCC(=O)c4ccon4)n3)ccc21
COC1=NC=CCC1C1=CNC([C@@H](N)CCCCCC(=O)c2ccon2)N1
COC1C=c2ncccc2=CC1C1=CNC([C@@H](N)CCCCCC(=O)c2ccon2)N1
COc1cc2c(ccc(=O)n2C)cc1-c1cnc([C@@H](N)CCCCCC(=O)c2ccon2)[nH]1
N[C@@H](CCCCCC(=O)C1COC=N1)C1NC=C(c2ccccc2F)N1
N[C@@H](CCCCCC(=O)c1ccon1)C1NC=C(c2ccccc2F)N1
CN1CC(C1)C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1ncc([nH]1)-c1ccccc1F |r|
CN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1nc(-c2ccccc2F)c[nH]1
COc1nc2ccccc2cc1-c1c[nH]c([C@H](CCCCCC(=O)c2ccon2)NC(=O)C2CCN(C)CC2)n1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)CN(C)C)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2cncs2)[nH]1
Cc1ccc2cc(-c3c[nH]c([C@H](CCCCCC(=O)c4ccon4)NC(=O)C4CN(C)C4)n3)ccc2n1
Cc1ccc2cc(-c3c[nH]c([C@H](CCCCCC(=O)c4ccon4)NC(=O)[C@H]4CC45CCN(C)CC5)n3)ccc2n1
Cc1cc(C(=O)CCCCC[C@H](N)c2nc(-c3ccccc3F)c[nH]2)no1
CN(C)CC(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2ccc3c(ccc(=O)n3C)c2)[nH]1
CN(C)CC(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1nc(-c2ccccc2F)c[nH]1
Cc1cc(C(=O)CCCCC[C@H](NC(=O)CN(C)C)c2nc(-c3ccccc3F)c[nH]2)no1
O=C(CCCCC[C@H](NC(=O)C(F)(F)F)c1nc(-c2ccccc2F)c[nH]1)c1ccon1
CCN(CC)CC(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cc3ccccc3nc2OC)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)CN2CCC2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)CN2CCCC2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)CN2CCCCC2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)CN2CCOCC2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)CCCN(C)C)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2cc(C)on2)NC(=O)CN(C)C)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2cc(C)on2)NC(=O)C2CN(C)C2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2cc(C)on2)NC(=O)C2CC23CCN(C)CC3)[nH]1
Cc1cc(C(=O)CCCCC[C@H](NC(=O)C2CN(C)C2)c2nc(-c3ccccc3F)c[nH]2)no1
CN1CCC1C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1ncc(-c2ccccc2F)[nH]1
CC(C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1ncc(-c2ccccc2F)[nH]1)N(C)C
CN(C)C1(C(=O)N[C@@H](CCCCCC(=O)c2ccon2)c2ncc(-c3ccccc3F)[nH]2)CC1
CN(C)C1(C(=O)N[C@@H](CCCCCC(=O)c2ccon2)c2ncc(-c3ccccc3F)[nH]2)CCC1
CN(C)C1(C(=O)N[C@@H](CCCCCC(=O)c2ccon2)c2ncc(-c3ccccc3F)[nH]2)CCCC1
O=C1CC[C@](CCCCCC(=O)C2NC=CO2)(c2ncc(-c3ccc(F)cc3)[nH]2)N1
O=C1NC(CCCCCC(=O)C2NC=CO2)(C2=NC(c3ccc(F)cc3)CN2)CO1
O=C1CC[C@@](CCCCCC(=O)c2ccon2)(C2=NC(c3ccc(C4NC=CO4)cc3F)CN2)N1
O=C1CC[C@@](CCCCCC(=O)c2ccon2)(C2=NC(c3ccc(C4CC4)cc3F)CN2)N1
O=C1CC[C@@](CCCCCC(=O)c2ccon2)(C2=NC(c3ccccc3F)CN2)N1
COC1C=c2nc(C)ccc2=CC1C1=CNC([C@@]2(CCCCCC(=O)c3ccon3)CCC(=O)N2)N1
COC1=NC=CCC1C1=CNC([C@]2(CCCCCC(=O)c3ccon3)CCCC(=O)N2)N1
O=C1CCCC[C@@](CCCCCC(=O)c2ccon2)(C2=NC(c3ccccc3F)CN2)N1
COc1nc2ccccc2cc1-c1cnc(CCCCCCC(=O)C2NC=CO2)[nH]1
CCN[C@@H](CCCCCC(=O)C1NC=CO1)C1NC=C(C2C=c3ccc(C)nc3=CC2)N1
CN[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2ccc3nc(C)ccc3c2)[nH]1
CN[C@@H](CCCCCC(=O)C1NC=CO1)c1ncc(-c2cc3ccc(=O)n(C)c3cc2OC)[nH]1
CCN[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cc3ccc(=O)n(C)c3cc2OC)[nH]1
Cc1ccc2c(n1)=CCC(C1=CNC([C@H](CCCCCC(=O)C3NC=CO3)NC3CCN(C)CC3)N1)C=2
Cc1ccc2cc(-c3cnc([C@H](CCCCCC(=O)C4NC=CO4)NC4CCOCC4)[nH]3)ccc2n1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC2CCOCC2)[nH]1
Cc1ccc2c(n1)=CCC(C1=CNC([C@H](CCCCCC(=O)C3NC=CO3)NCc3ccccc3)N1)C=2
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NCc2ccccc2)[nH]1
Cc1ccc2cc(-c3cnc([C@H](CCCCCC(=O)C4NC=CO4)N4CCOCC4)[nH]3)ccc2n1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)C2NC=CO2)NC2CC(OC)C2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)C2NC=CO2)Nc2ncccn2)[nH]1
COC(=O)N[C@@H](CCCCCC(=O)C1NC=CO1)c1ncc(-c2cc3ccc(C)nc3cc2OC)[nH]1
COC(=O)N[C@@H](CCCCCC(=O)C1NC=CO1)c1ncc(-c2cc3ccc(C)nc3cc2OC)[nH]1
O=C(N[C@@H](CCCCCC(=O)C1NC=CO1)C1NC(c2ccc(F)cc2)=NC1Cl)c1cncs1
COC1C=c2nc(C)ccc2=CC1C1=CNC([C@H](CCCCCC(=O)C2NC=CO2)NC(=O)CN(C)C)N1
CN(C)CC(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1[nH]c(-c2ccc(F)cc2)nc1Cl
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ccon2)NC(=O)CN(C)C)[nH]1
COc1cc2c(ccc(=O)n2C)cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)CN(C)C)[nH]1
COc1cc2c(ccc(=O)n2C)cc1-c1cnc([C@H](CCCCCC(=O)c2ccon2)NC(=O)CN(C)C)[nH]1
CCn1ccc2c(c1=O)=CC(OC)C(C1=CNC([C@H](CCCCCC(=O)c3ccon3)NC(=O)CN(C)C)N1)C=2
CN(C)CC(=O)N[C@@H](CCCCCC(=O)C1NC=CO1)C1NC=C(C2C=c3nccnc3=CC2)N1
CCn1ccc2cc(-c3cnc([C@H](CCCCCC(=O)c4ncco4)NC(=O)CN(C)C)[nH]3)c(OC)cc2c1=O
CCN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)C1NC=CO1)C1NC(c2ccc(F)cc2)=NC1Cl
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)C2NC=CO2)NC(=O)C2CCN(C)CC2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)C2NC=CO2)NC(=O)C2CN(C)C2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)C2NC=CO2)NC(=O)C2CN(C)C2)o1
CC(C)(C)OC(=O)N1CC(C(=O)N[C@@H](CCCCCC(=O)c2ncco2)c2[nH]c(-c3ccc(F)cc3)nc2Cl)C1
COc1cc2c(ccc(=O)n2C)cc1-c1cnc([C@H](CCCCCC(=O)c2ccon2)NC(=O)C2CN(C)C2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ccon2)NC(=O)C2CN(C)C2)[nH]1
COc1ncccc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2CN(C)C2)o1
CN1CC(C(=O)N[C@@H](CCCCCC(=O)c2ccon2)C2NC(c3ccccc3F)=NC2Cl)C1
CN1CC(C1)C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1nnc(o1)-c1ccccc1F |r|
CN1CC(C(=O)NC(CCCCCC(=O)c2ccon2)c2ncc(-c3ccccc3F)o2)C1
COC1C=c2nc(C)ccc2=CC1C1=CNC([C@H](CCCCCC(=O)c2ccon2)NC(=O)C2CN(C)C2)O1
Cc1ccc2c(n1)=CCC(C1=CNC([C@H](CCCCCC(=O)C3NC=CO3)NC(=O)[C@H]3CC34CCN(C)CC4)O1)C=2
COC1C=c2nc(C)ccc2=CC1C1=CNC([C@H](CCCCCC(=O)c2ccon2)NC(=O)[C@H]2CC23CCN(C)CC3)N1
Cc1ccc2cc(-c3cnc(C(CCCCCC(=O)c4ncco4)NC(=O)[C@H]4CC45CCN(C)CC5)o3)ccc2n1
CN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1[nH]c(-c2ccccc2F)nc1Cl
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)[C@H]2CC23CCN(C)CC3)o1
COc1ncccc1-c1cnc(C(CCCCCC(=O)C2NC=CO2)NC(=O)[C@H]2CC23CCN(C)CC3)o1
COc1nc(C2CC2)ccc1-c1c[nH]c([C@H](CCCCCC(=O)c2ncco2)NC(=O)[C@H]2CC23CCN(C)CC3)n1
Cc1ccc2c(n1)=CCC(C1=CNC([C@H](CCCCCC(=O)C3NC=CO3)NC(=O)C3=NOC4(CCN(C)CC4)C3)O1)C=2
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)C2NC=CO2)NC(=O)C2CCC3(CC2)CN(C)C3)[nH]1
N[C@@H](CCCCCC(=O)c1ccon1)c1cc(-c2ccc(F)cc2)on1
N[C@H](CCCCCC(=O)c1ccon1)c1cc(-c2ccc(F)cc2)on1
N[C@@H](CCCCCC(=O)c1ccon1)c1ccn(n1)-c1ccc(F)cc1 |r|
NC(CCCCCC(=O)c1ccon1)c1cnn(-c2ccc(F)cc2)c1
NC(CCCCCC(=O)c1ccon1)c1cnn(-c2ccc(F)cc2)n1
N[C@@H](CCCCCC(=O)c1ccon1)c1cc(on1)-c1ccccc1F |r|
Cn1cc2cc(-c3cc([C@@H](N)CCCCCC(=O)c4ccon4)no3)ccc2n1
Cn1cc2cc(-n3ccc([C@@H](N)CCCCCC(=O)c4ncco4)n3)ccc2n1
COc1cc(C2=CNC([C@@H](N)CCCCCC(=O)C3NC=CO3)N2)c(F)cn1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cc(OC3CCC3)ccc2F)[nH]1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cnc(C3CC3)cn2)[nH]1
N#Cc1cnc(-c2cnc([C@@H](N)CCCCCC(=O)c3ncco3)[nH]2)cn1
N#Cc1cncc(-c2cnc([C@@H](N)CCCCCC(=O)c3ncco3)[nH]2)n1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cc(F)ccc2F)[nH]1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cccc(F)c2F)[nH]1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cc(C(F)(F)F)ccc2F)[nH]1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cccc(C(F)(F)F)c2F)[nH]1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2ccc(C(F)(F)F)cc2F)[nH]1
COc1ccc(-c2cnc([C@@H](N)CCCCCC(=O)c3ncco3)[nH]2)c(F)c1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2ccc(OC(F)(F)F)cc2F)[nH]1
N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cc(OC(F)(F)F)ccc2F)[nH]1
CS(=O)(=O)c1ccc(-c2cnc([C@@H](N)CCCCCC(=O)c3ncco3)[nH]2)c(F)c1
COc1cc(O[C@H]2C[C@H](OC)C2)cc(-c2cnc([C@@H](N)CCCCCC(=O)c3ncco3)[nH]2)c1F
CCN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1cc(C2C=c3ccc(C)nc3=CC2OC)on1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2ccc(OC(F)F)nc2)[nH]1
COCC(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cc3ccccc3nc2OC)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C(C)(F)F)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2ccncn2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)Cn2cccc2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2(c3ccncc3)CC2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2COCCO2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2nc3ccccc3o2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2cc3n(n2)CCCC3)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2(c3cnccn3)CC2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)[C@H]2CCC(=O)N2)[nH]1
COc1nc2ccccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)[C@@H]2CCC(=O)N2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)CN2CCOCC2=O)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)CN2CCNCC2=O)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)Cn2cccn2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2cc3ncccn3n2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)Cn2cccc2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2cc3n(n2)CCCO3)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2cc3n(n2)CCCC3)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2cc3n(n2)CCS(=O)(=O)C3)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)Cn2ccc(C)n2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)c2cc3ccccn3n2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2CCCCO2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2CCCO2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2(C)CCCCO2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2COc3ccccc3O2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2COC(c3ccccc3)CO2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2COCCO2)[nH]1
COc1cc2nc(C)ccc2cc1-c1cnc([C@H](CCCCCC(=O)c2ncco2)NC(=O)C2COCCO2)[nH]1
CCN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1cc(-c2ccccc2F)on1
CCN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1cc(-c2ccc3nn(C)cc3c2)on1
CN1CCC2(CC1)CC(C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1cc(-c3ccc4nn(C)cc4c3)on1)=NO2
COc1cc(-c2cnc([C@H](CCCCCC(=O)c3ncco3)NC(=O)C3CN(C)C3)[nH]2)c(F)cn1
CCN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cc(OC)ncc2F)[nH]1
CCN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1ccn(-c2ccc3nn(C)cc3c2)n1
CN1CC(C(=O)N[C@@H](CCCCCC(=O)c2ncco2)c2ncc(-c3cc(OC4CCC4)ccc3F)[nH]2)C1
CCN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1ncc(-c2cc(OC3CCC3)ccc2F)[nH]1
CCN1CCC2(CC1)C[C@@H]2C(=O)NC(C)(CCCCCC(=O)c1ccon1)c1ncc(-c2ccccc2F)[nH]1
CN1CC(C(=O)NC(C)(CCCCCC(=O)c2ccon2)c2ncc(-c3ccccc3F)[nH]2)C1
N#Cc1nc(-c2ccc(F)cc2)[nH]c1[C@@H](N)CCCCCC(=O)C1NC=CO1
CN(C)CC(=O)N[C@@H](CCCCCC(=O)C1NC=CO1)C1NC(c2ccc(F)cc2)=NC1C#N
CN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1[nH]c(-c2ccc(F)cc2)nc1C#N
N#Cc1nc(-c2ccc(F)cc2)[nH]c1[C@H](CCCCCC(=O)c1ncco1)NC(=O)c1nccs1
N#Cc1nc(-c2ccc(F)cc2)oc1[C@@H](N)CCCCCC(=O)C1NC=CO1
CN(C)CC(=O)N[C@@H](CCCCCC(=O)C1NC=CO1)C1NC(c2ccc(F)cc2)=NC1C#N
CN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1oc(-c2ccc(F)cc2)nc1C#N
N#Cc1nc(-c2ccc(F)cc2)oc1[C@H](CCCCCC(=O)c1ncco1)NC(=O)c1nccs1
N[C@@H](CCCCCC(=O)c1ccon1)C1NC(Cl)=C(c2ccc(F)cc2)N1
CN(C)CC(=O)N[C@@H](CCCCCC(=O)c1ccon1)C1=NC(Cl)C(c2ccc(F)cc2)N1
CN1CCC2(CC1)C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1nc(Cl)c(-c2ccc(F)cc2)[nH]1
CN1CC(C(=O)N[C@@H](CCCCCC(=O)c2ccon2)c2nc(Cl)c(-c3ccc(F)cc3)[nH]2)C1
O=C(NO)c1ccc2cn(Cc3ccccc3)nc2c1
COc1ccc(Cn2cc3ccc(C(=O)NO)cc3n2)cc1
Cc1ccc(Cn2cc3ccc(C(=O)NO)cc3n2)cc1
O=C(NO)c1ccc2cn(Cc3ccc(F)cc3)nc2c1
O=C(NO)c1ccc2cn(Cc3ccc(Cl)cc3)nc2c1
O=C(NO)c1ccc2cn(Cc3ccc(Br)cc3)nc2c1
C/C=C(C=C(/C)OC(F)(F)F)Cn1cc2ccc(C(=O)NO)cc2n1
O=C(NO)c1ccc2cn(Cc3ccc(OC(F)(F)F)cc3)nc2c1
O=C(NO)c1ccc2cn(Cc3ccc4ccccc4c3)nc2c1
O=C(NO)c1ccc2cn(CCc3ccccc3)nc2c1
COc1ccc(CCn2cc3ccc(C(=O)NO)cc3n2)cc1
O=C(NO)c1ccc2cn(Cc3cc(F)cc(F)c3)nc2c1
O=C(NO)c1ccc2cn(Cc3ccc(OC(F)F)cc3)nc2c1
O=C(NO)c1ccc2cn(Cc3ccc(-c4ccccc4)cc3)nc2c1
CC(C)c1ccc(Cn2cc3ccc(C(=O)NO)cc3n2)cc1
O=C(NO)c1ccc2cn(CCc3ccc(F)cc3)nc2c1
C/C=C(C=C(/C)F)Cn1cc2ccc(C(=O)NO)cc2n1
O=C(NO)c1ccc2cn(Cc3cccc(Cl)c3)nc2c1
C/C=C(C=C(/C)C(F)(F)F)Cn1cc2ccc(C(=O)NO)cc2n1
O=C(NO)c1ccc2cn(Cc3ccc(C(F)(F)F)cc3)nc2c1
C/C=C(C=C(/C)OC)Cn1cc2ccc(C(=O)NO)cc2n1
C/C=C(C=C(/C)OBr)Cn1cc2ccc(C(=O)NO)cc2n1
COc1cc(Cn2cc3ccc(C(=O)NO)cc3n2)cc(OC)c1
C/C=C(C=C(/C)Oc1ccccc1)Cn1cc2ccc(C(=O)NO)cc2n1
O=C(NO)c1cc2nn(Cc3ccccc3)cc2cc1F
O=C(NO)c1cc2nn(Cc3cccc(Cl)c3)cc2cc1F
COc1cccc(Cn2cc3cc(F)c(C(=O)NO)cc3n2)c1
ONC(=O)c1cccc(\C=C\c2ccnc(c2)-c2cc(F)ccc2O)c1
ONC(=O)c1ccc(\C=C\c2ccnc(c2)-c2ccccc2O)cc1
Cc1ccc(c(F)c1)-c1cc(\C=C\c2ccc(cc2)C(=O)NO)ccn1
Nc1ncnc2n(nc(-c3ccc(Cl)cc3)c12)-c1cccc(c1)-c1cnnn1CCCCCC(=O)NO
ONC(=O)\C=C\c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccccc2)cc1 |r|
ONC(=O)\C=C\c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)Cc2ccccc2)cc1 |r|
ONC(=O)\C=C\c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(Cl)cc2)cc1 |r|
ONC(=O)\C=C\c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(F)cc2)cc1 |r|
COc1ccc(cc1)C(=O)N[C@H](COc1ccc(\C=C\C(=O)NO)cc1)Cc1c[nH]c2ccccc12 |r|
Cl.ONC(=O)\C=C\c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NCc2ccc(Cl)cc2)cc1 |r|
ONC(=O)\C=C\c1cccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(Cl)cc2)c1 |r|
COc1ccc(cc1)-c1ccc(\C=C\C(=O)NO)cc1
ONC(=O)\C=C\c1ccc(c(Cl)c1)-c1ccc(CC#N)c(c1)C12CC3CC(CC(C3)C1)C2 |TLB:25:26:24.23.29:30,THB:25:24:26.31.27:30,27:26:23:29.28.30,27:28:25.26.31:23|
ONC(=O)\C=C\c1ccc(cc1)-c1ccc(O)cc1
COc1ccc(cc1C12CC3CC(CC(C3)C1)C2)-c1ccc(\C=C\C=C\C(=O)NO)cc1 |TLB:11:12:10.9.15:16,THB:11:10:12.17.13:16,13:12:9:15.14.16,13:14:11.12.17:9|
ONC(=O)\C=C\c1ccc(cc1)-c1ccc(O)c(c1)C12CC3CC(CC(C3)C1)C2 |TLB:22:23:21.20.26:27,THB:22:21:23.28.24:27,24:23:20:26.25.27,24:25:22.23.28:20|
COc1ccc(cc1)-c1ccc(\C=C\C=C\C(=O)NO)cc1
CC(C)c1cc(C(=O)N2CCc3onc(C(=O)NCCCCCCC(=O)NO)c3C2)c(O)cc1O
CC(C)c1cc(c(O)cc1O)-n1nnc(C(=O)NCCCCCCC(=O)NO)c1-c1ccc(CN2CCOCC2)cc1
ONC(=O)\C=C\c1cccc(c1)S(=O)(=O)n1ccc2ccncc12
ONC(=O)\C=C\c1cccc(c1)S(=O)(=O)n1ccc2cccnc12
Nc1ccc(cc1NC(=O)c1ccc(nc1)N1CCC2(CNC(=O)O2)CC1)-c1cccs1
Fc1cccc(c1)-c1csc(NC(=O)CCCCCCS)n1
Cc1ccc(cc1F)-c1csc(NC(=O)CCCCCCS)n1
Fc1ccc(cc1)-c1csc(NC(=O)CCCCCCS)n1
CCCCCCCC(=O)SCC\C=C\[C@@H]1CC(=O)NCc2nc(cs2)C2=N[C@@](C)(CS2)C(=O)N[C@@H](C(C)C)C(=O)O1 |r,t:26|
[H][C@]1(CC(=O)NCc2nc(cs2)C2=N[C@@](C)(CS2)C(=O)N[C@H](C(C)C)C(=O)O1)\C=C\CCS |r,t:13|
CCCCCCCC(=O)SCC\C=C\[C@@H]1CC(=O)NCc2nc(cs2)-c2nc(cs2)C(=O)N[C@@H](C(C)C)C(=O)O1 |r|
CC(C)[C@@H]1NC(=O)c2csc(n2)-c2csc(CNC(=O)C[C@H](OC1=O)\C=C\CCS)n2 |r|
[#6]\[#6](-[#6])=[#6]/c1sc(nc1-[#6](=O)-[#7]-[#6]-[#6]-[#6]-[#6]-[#6](=O)-[#7]-[#8])-c1nccs1
C[C@@H]1NC(=O)C(C)(C)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C1=O
C[C@@H]1NC(=O)[C@]2(CCc3ccccc23)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C1=O
CC1(C)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C(=O)[C@H](CO)NC1=O
C[C@@H]1NC(=O)[C@@]2(CCc3ccccc23)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C1=O
CC1(C)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C(=O)[C@H](COCc2ccccc2)NC1=O
C[C@@H]1NC(=O)C2(Cc3ccccc3C2)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C1=O
CC1(C)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C(=O)[C@H](CCCc2ccccc2)NC1=O
CC1(C)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC1=O
CC1(C)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C(=O)[C@H](CCc2ccccc2)NC1=O
CC1(C)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C(=O)[C@@H](NC1=O)c1ccccc1
C[C@H]1CN2Cc3ccccc3C[C@@H]2C(=O)N[C@@H](CCCCCSSc2ccccn2)C(=O)NC(C)(C)C(=O)N1
C[C@@H]1NC(=O)[C@](C)(Cc2ccccc2)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C1=O
C[C@@H]1NC(=O)[C@@](C)(Cc2ccccc2)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C1=O
ONC(=O)CCCCCNC(=O)NC(=O)c1ccc(Br)cc1
ONC(=O)CCCCc1ccn(Cc2cccc(c2)-c2ccccc2)n1
ONC(=O)CCCCc1ccn(n1)-c1ccccc1
ONC(=O)CCCCc1ccn(Cc2ccc(cc2)-n2ccc3ccccc23)n1
ONC(=O)CCCCc1ccn(Cc2ccc(Nc3ccccc3)cc2)n1
ONC(=O)CCCCc1ccn(Cc2ccc(cc2)-c2ccccc2)n1
COc1cc(OC)cc(\C=C\c2ccc(OC)c(NC(=O)CCCCCCC(=O)NO)c2)c1
COc1cc(OC)cc(\C=C/c2ccc(OC)c(NC(=O)CCCCCCC(=O)NO)c2)c1
SCCCCCCC(=O)Nc1ccccc1
SCCCCCC(=O)Nc1ccccc1
SCCCCCCCC(=O)Nc1ccccc1
SCCCCC[C@H](NC(=O)[C@@H]1CCCC(=O)N1)C(=O)Nc1ccccc1 |r|
SCCCCC[C@H](NC(=O)[C@H]1CCCC(=O)N1)C(=O)Nc1ccccc1 |r|
SCCCCC[C@@H](NC(=O)[C@@H]1CCCC(=O)N1)C(=O)Nc1ccccc1 |r|
CN1[C@@H](CCCC1=O)C(=O)N[C@@H](CCCCCS)C(=O)Nc1ccccc1 |r|
SCCCCC[C@H](NC(=O)[C@@H]1CCCNC1=O)C(=O)Nc1ccccc1 |r|
SCCCCC[C@H](NC(=O)[C@H]1CCCNC1=O)C(=O)Nc1ccccc1 |r|
Cc1cccc(NC(=O)[C@H](CCCCCS)NC(=O)[C@@H]2CCCC(=O)N2)c1 |r|
Cc1ccc(NC(=O)[C@H](CCCCCS)NC(=O)[C@@H]2CCCC(=O)N2)cc1 |r|
SCCCCC[C@H](NC(=O)[C@@H]1CCC(=O)N1)C(=O)Nc1ccccc1 |r|
SCCCCC[C@@H](NC(=O)[C@@H]1CCC(=O)N1)C(=O)Nc1ccccc1 |r|
SCCCCC[C@@H](NC(=O)[C@H]1CCC(=O)N1)C(=O)Nc1ccccc1 |r|
CN1[C@H](CCC1=O)C(=O)N[C@@H](CCCCCS)C(=O)Nc1ccccc1 |r|
Cc1cccc(NC(=O)[C@H](CCCCCS)NC(=O)[C@@H]2CCC(=O)N2)c1 |r|
Cc1cccc(NC(=O)[C@H](CCCCCS)NC(=O)[C@H]2CCC(=O)N2)c1 |r|
CN1[C@H](CCC1=O)C(=O)N[C@@H](CCCCCS)C(=O)Nc1cccc(C)c1 |r|
FC(F)(F)c1cccc(NC(=O)[C@H](CCCCCS)NC(=O)[C@H]2CCC(=O)N2)c1 |r|
SCCCCC[C@H](NC(=O)[C@H]1[C@@H](CNC1=O)c1ccccc1)C(=O)Nc1ccccc1 |r|
SCCCCC[C@H](NC(=O)[C@@H]1[C@H](CNC1=O)c1ccccc1)C(=O)Nc1ccccc1 |r|
SCCCCC[C@H](NC(=O)[C@H]1[C@H](CNC1=O)c1ccccc1)C(=O)Nc1ccccc1 |r|
SCCCCC[C@H](NC(=O)[C@@H]1[C@@H](CNC1=O)c1ccccc1)C(=O)Nc1ccccc1 |r|
SCCCCC[C@H](NC(=O)[C@@H]1CC(=O)N1)C(=O)Nc1ccccc1 |r|
SCCCCCCC(=O)NC1CCCC1
SCCCCC[C@H](NC(=O)[C@@H]1CCCC(=O)N1)C(=O)NC1CCCC1 |r|
FC(F)(F)c1ccc(CNC(=O)CCCCCCS)cc1
FC(F)(F)c1ccc(CNC(=O)[C@H](CCCCCS)NC(=O)[C@@H]2CCCC(=O)N2)cc1 |r|
SCCCCCCC(=O)NCc1cccc(OCc2ccccc2)c1
SCCCCC[C@H](NC(=O)[C@@H]1CCCC(=O)N1)C(=O)NCc1cccc(OCc2ccccc2)c1 |r|
Cc1cccc(CCNC(=O)CCCCCCS)c1
Cc1cccc(CCNC(=O)[C@H](CCCCCS)NC(=O)[C@@H]2CCCC(=O)N2)c1 |r|
SCCCCC[C@H](NC(=O)[C@@H]1CCCC(=O)N1)C(=O)N1CCc2ccccc2C1 |r|
ONC(=O)c1ccc2CCC(Cc2c1)NS(=O)(=O)c1cccc(Cl)c1
ONC(=O)c1ccc2CC[C@@H](Cc2c1)Nc1nccc(n1)-c1cccnc1 |r|
ONC(=O)c1ccc2CC[C@H](Cc2c1)Nc1nccc(n1)-c1cccnc1 |r|
ONC(=O)c1ccc2CCN(Cc3ccc(o3)-c3cccc(c3)[N+]([O-])=O)Cc2c1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1ccc(F)cc1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1ccc(C#N)c(Cl)c1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1ccccn1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1ncccn1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1ccccc1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1ccc(Cl)cc1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1cccc(Cl)c1
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1ccccc1Cl
ONC(=O)c1ccc2CCC(Cc2c1)Nc1nccc(n1)-c1cccnc1
CN(C1CCc2ccc(cc2C1)C(=O)NO)c1nccc(n1)-c1cccnc1
ONC(=O)c1ccc2CCC(Cc2c1)NS(=O)(=O)c1cccc(F)c1
CC(C)[C@H]1NC(=O)C[C@H](NC(=O)[C@@H](Cc2ccc(O)cc2)NC(=O)[C@@H](C)NC1=O)\C=C\CCCC(O)=O |r|
CC(C)[C@H]1NC(=O)C[C@H](NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@@H](C)NC1=O)\C=C\CCCC(O)=O |r|
CC(C)[C@H]1NC(=O)C[C@@H](CCCCCC(O)=O)NC(=O)[C@@H](Cc2ccc(O)cc2)NC(=O)[C@@H](C)NC1=O |r|
CC(C)[C@H]1NC(=O)C[C@@H](CCCCCC(O)=O)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@@H](C)NC1=O |r|
CC(C)[C@H]1NC(=O)C[C@@H](C\C=C/CCC(O)=O)NC(=O)[C@@H](Cc2ccc(O)cc2)NC(=O)[C@@H](C)NC1=O |r|
Cn1cccc1C(=O)N1CCn2cc(nc2C1)C(=O)NO
Cn1c(cc2ccccc12)C(=O)N1CCn2nc(cc2C1)C(=O)NO
COc1ccc(cc1)C(=O)N1CCn2nc(cc2C1)C(=O)NO
Cn1cccc1C(=O)N1CCn2nc(cc2C1)C(=O)NO
ONC(=O)c1cc2CN(CCn2c1)C(=O)c1ccc(cc1)-c1ccccc1
Cn1ccc2cc(ccc12)C(=O)N1CCn2cc(cc2C1)C(=O)NO
Cn1cc(C(=O)N2CCn3cc(cc3C2)C(=O)NO)c2ccccc12
ONC(=O)c1cc2CN(CCn2c1)C(=O)c1cc2ccccc2[nH]1
ONC(=O)c1cc2CN(CCn2c1)C(=O)C1CCCCC1
COc1ccc(cc1)C(=O)N1CCn2cc(cc2C1)C(=O)NO
ONC(=O)c1cc2CN(CCn2c1)C(=O)c1cc2ccccc2s1
ONC(=O)c1cc2CN(CCn2c1)C(=O)c1cccs1
Cn1c(Cl)c(Cl)cc1C(=O)N1CCn2cc(cc2C1)C(=O)NO
Cn1cccc1C(=O)N1CCn2cc(cc2C1)C(=O)NO
ONC(=O)c1cn2CCN(Cc2n1)C(=O)c1cc2ccccc2s1
ONC(=O)c1cn2CCN(Cc2n1)C(=O)c1ccc(cc1)-c1ccccc1
Cn1cccc1C(=O)NCc1ccc(cc1)C(=O)NO
Cn1cccc1C(=O)N1CCc2cc(ccc2C1)C(=O)NO
Oc1ccc(\C=C2/Oc3ccccc3C2=O)cc1
Oc1ccc(\C=C2/Oc3ccccc3C2=O)cc1O
ON(CCCCCC(C(=O)Nc1cnc2ccccc2c1)C(=O)Nc1cnc2ccccc2c1)C=O
COC(=O)N(O)CCCCCCC(=O)Nc1ccccc1
ON(CCCCCNC(=O)c1ccccc1)C=O
Oc1cccc(\C=C2/Oc3ccccc3C2=O)c1O
CC(=O)N(O)CCCCCC(=O)Nc1ccccc1
ON(CCCCCNC(=O)c1ccc2ccccc2c1)C=O
Oc1cc2O\C(=C/c3ccc(O)c(O)c3)C(=O)c2c(O)c1
ON(CCCCCCCC(=O)Nc1ccccc1)C=O
ON(CCCCCC(=O)Nc1ccccc1)C=O
ON(CCCCCNC(=O)CCc1ccccc1)C=O
ON(CCCCCCCC(=O)Nc1ccc2ccccc2c1)C=O
ON(CCCCCC(C(=O)Nc1ccc2ncccc2c1)C(=O)Nc1ccc2ncccc2c1)C=O
CC(=O)N(O)CCCCCCCC(=O)Nc1ccccc1
ON(CCCCCCCC(=O)Nc1cccc2ccccc12)C=O
COc1ccccc1C(=O)N[C@H](COc1cccc(\C=C\C(=O)NO)c1)Cc1c[nH]c2ccccc12 |r|
COc1ccc(cc1)C(=O)N[C@H](COc1cccc(\C=C\C(=O)NO)c1)Cc1c[nH]c2ccccc12 |r|
SCCCCC[C@H](NC(=O)[C@H]1CCC(=O)N1)C(=O)Nc1ccccc1 |r|
Cc1cccc(NC(=O)[C@H](CCCCCC(=O)NO)NC(=O)[C@H]2CCC(=O)N2)c1 |r|
ONC(=O)CCCCC[C@H](NC(=O)[C@H]1CCC(=O)N1)C(=O)Nc1cccc(c1)C(F)(F)F |r|
ONC(=O)CCCCC[C@H](NC(=O)[C@@H]1CCC(=O)N1)C(=O)Nc1ccccc1 |r|
ONC(=O)CCCCC[C@H](NC(=O)[C@@H]1CC(=O)N1)C(=O)Nc1ccccc1 |r|
ONC(=O)CCCCCCC(=O)Nc1ccc2[nH]c(=O)ccc2c1
ONC(=O)CCCCCCC(=O)Nc1ccc2NC(=O)CCc2c1
CC1(C)CC(=O)Nc2ccc(NC(=O)CCCCCCC(=O)NO)cc12
ONC(=O)CCCCCCNC(=O)c1ccc2[nH]c(=O)ccc2c1
ONC(=O)CCCCCCNC(=O)c1ccc2NC(=O)CCc2c1
CC1(C)CC(=O)Nc2ccc(cc12)C(=O)NCCCCCCC(=O)NO
Cn1c2ccc(cc2ccc1=O)C(=O)NCCCCCCC(=O)NO
CN1C(=O)CC(C)(C)c2cc(ccc12)C(=O)NCCCCCCC(=O)NO
COc1ccc2cc(ccc2n1)C(=O)NCCCCCCC(=O)NO
CC1(C)CC(=O)Nc2ccc(cc12)C(=O)NCc1cccc(\C=C\C(=O)NO)c1
CC1(C)CC(=O)Nc2ccc(cc12)C(=O)NCc1ccc(\C=C\C(=O)NO)cc1
CC1(C)CC(=O)Nc2ccc(cc12)C(=O)NC[C@H]1CC[C@@H](CC1)\C=C\C(=O)NO |r,wU:17.18,wD:20.25,(21.24,-20.14,;22.02,-21.48,;22.78,-20.14,;23.36,-22.25,;23.36,-23.79,;24.69,-24.56,;22.02,-24.56,;20.69,-23.79,;19.36,-24.56,;18.02,-23.79,;18.02,-22.25,;19.36,-21.48,;20.69,-22.25,;16.7,-21.48,;16.7,-19.94,;15.36,-22.25,;14.02,-21.48,;12.69,-22.25,;12.69,-23.8,;11.35,-24.56,;10.01,-23.79,;10.02,-22.25,;11.35,-21.48,;8.67,-24.55,;7.34,-23.78,;6.01,-24.54,;6,-26.08,;4.68,-23.76,;3.34,-24.53,)|
CC1(C)CC(=O)Nc2ccc(cc12)C(=O)NC[C@H]1CC[C@H](CCC(=O)NO)CC1 |r,wU:17.18,wD:20.22,(21.54,-26.71,;22.32,-28.05,;23.08,-26.71,;23.66,-28.82,;23.66,-30.36,;24.99,-31.13,;22.32,-31.13,;20.98,-30.36,;19.66,-31.13,;18.32,-30.36,;18.32,-28.82,;19.66,-28.05,;20.98,-28.82,;16.99,-28.05,;16.99,-26.51,;15.65,-28.82,;14.32,-28.05,;12.98,-28.82,;12.99,-30.37,;11.64,-31.14,;10.31,-30.36,;8.97,-31.12,;7.64,-30.35,;6.3,-31.11,;6.3,-32.65,;4.97,-30.34,;3.64,-31.1,;10.32,-28.82,;11.65,-28.05,)|
CC1(C)CC(=O)Nc2ccc(cc12)C(=O)NC[C@H]1CC[C@H](CC1)\C=C\C(=O)NO |r,wU:17.18,20.25,(21.18,-34.58,;21.96,-35.93,;22.72,-34.58,;23.3,-36.7,;23.3,-38.24,;24.63,-39.01,;21.96,-39.01,;20.62,-38.24,;19.3,-39.01,;17.96,-38.24,;17.96,-36.7,;19.3,-35.93,;20.62,-36.7,;16.63,-35.93,;16.63,-34.39,;15.3,-36.7,;13.96,-35.93,;12.62,-36.7,;12.63,-38.24,;11.28,-39.01,;9.95,-38.24,;9.96,-36.69,;11.29,-35.93,;8.61,-39,;7.28,-38.22,;5.94,-38.99,;5.94,-40.53,;4.61,-38.21,;3.28,-38.97,)|
CC1(C)CC(=O)Nc2ccc(cc12)C(=O)NC[C@@H]1CC[C@H](CCC(=O)NO)CC1 |r,wU:17.18,20.22,(45.27,-32.85,;46.06,-34.2,;46.81,-32.85,;47.39,-34.97,;47.39,-36.51,;48.73,-37.28,;46.06,-37.28,;44.72,-36.51,;43.39,-37.28,;42.06,-36.51,;42.06,-34.97,;43.39,-34.2,;44.72,-34.97,;40.73,-34.2,;40.73,-32.66,;39.39,-34.97,;38.06,-34.2,;36.72,-34.97,;35.39,-34.2,;34.05,-34.96,;34.04,-36.5,;32.71,-37.27,;31.38,-36.49,;30.04,-37.26,;30.03,-38.8,;28.71,-36.48,;27.37,-37.24,;35.38,-37.28,;36.72,-36.51,)|
Nc1ccccc1NC(=O)c1ccc(cc1)-c1nnc(Cc2cccc3ccccc23)o1
Nc1ccccc1NC(=O)c1ccc(Cc2nnc(Cc3cccc4ccccc34)o2)cc1
ONC(=O)\C=C\c1ccc(cc1)-c1nnc(Cc2cccc3ccccc23)o1
ONC(=O)\C=C\c1ccc(cc1)-c1nnc(Cc2c[nH]c3ccccc23)o1
ONC(=O)\C=C\c1ccc(Cc2nnc(Cc3cccc4ccccc34)o2)cc1
ONC(=O)c1ccc(cc1)-c1nnc(Cc2cccc3ccccc23)o1
ONC(=O)c1ccc(Cc2nnc(Cc3cccc4ccccc34)o2)cc1
Nc1ccccc1NC(=O)\C=C\c1ccc(cc1)-c1nnc(Cc2cccc3ccccc23)o1
Nc1ccccc1NC(=O)\C=C\c1ccc(cc1)-c1nnc(Cc2ccc3ccccc3c2)o1
Nc1ccccc1NC(=O)\C=C\c1ccc(cc1)-c1nnc(Cc2c[nH]c3ccccc23)o1
Nc1ccccc1NC(=O)\C=C\c1ccc(Cc2nnc(Cc3cccc4ccccc34)o2)cc1
[H][C@]12CCCN1C(=O)[C@H](C)NC(=O)[C@@]1([H])CCCCCSSCCCCC[C@]([H])(NC2=O)C(=O)N1 |r|
[H][C@]12CCCN1C(=O)[C@@H](NC(=O)[C@@]1([H])CCCCCSSCCCCC[C@]([H])(NC2=O)C(=O)N1)C(C)C |r|
[H][C@]12CCCN1C(=O)[C@H](Cc1ccccc1)NC(=O)[C@@]1([H])CCCCCSSCCCCC[C@]([H])(NC2=O)C(=O)N1 |r|
[H][C@]12CCCN1C(=O)[C@H](C)NC(=O)[C@@]1([H])CCOCCSSCCCCC[C@]([H])(NC2=O)C(=O)N1 |r|
[H][C@]12CCCN1C(=O)[C@@H](NC(=O)[C@]1([H])CCCCCSSCCCCC[C@]([H])(NC2=O)C(=O)N1)C(C)C |r|
[H][C@]12Cc3ccccc3CN1C(=O)[C@]1([H])CCCCCSSCCCCC[C@@]([H])(NC(=O)[C@@H](NC2=O)C(C)C)C(=O)N1 |r|
[H][C@@]12CC(=O)N[C@H](C(C)C)C(=O)N[C@]([H])(CSSCC\C=C\1)C(=O)N\C(=C/C)C(=O)N[C@@H](C(C)C)C(=O)O2 |r,t:20|
[H][C@]12CCCN1C(=O)[C@@]([H])(NC(=O)[C@@H](Cc1ccc(OC)cc1)NC(=O)[C@H](CCCCCC(=O)NO)NC2=O)[C@@H](C)CC |r|
ONC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCN2C(=O)[C@@H]2CCCCCCCCCC[C@@H](NC1=O)C(=O)N2 |r|
CCCCC[C@H]1NC(=O)[C@H](CCCCCC(=O)NO)NC(=O)[C@H]2CCCN2C(=O)[C@H](CCCCC)NC1=O |r|
[H][C@]12CCCN1C(=O)[C@]1([H])CCOCCCCOCC[C@@]([H])(NC(=O)[C@H](CCCCCC(=O)NO)NC2=O)C(=O)N1 |r|
[H][C@]12CCCN1C(=O)[C@]1([H])CCCCCCCCCC[C@]([H])(NC(=O)[C@H](CCCCCC(=O)NO)NC2=O)C(=O)N1 |r|
[H][C@]12CCCN1C(=O)[C@H](CCCCCC(=O)NO)NC(=O)[C@@]1([H])CCCCCCCCCC[C@]([H])(NC2=O)C(=O)N1 |r|
[H][C@]12CCCN1C(=O)[C@H](CCCCC)NC(=O)[C@H](CCCCC)NC(=O)[C@H](CCCCCC(=O)NO)NC2=O |r|
[H][C@]12CCCN1C(=O)[C@H](CCCCCC(=O)NO)NC(=O)[C@@H](CCCCC)NC(=O)[C@H](CCCCC)NC2=O |r|
COc1ccc2cc(C(=O)\C=C\C=C\c3ccc(OC)c(OC)c3)c(=O)oc2c1
COc1cc2ncnc(Nc3ccc(Cl)cc3Cl)c2cc1OCCCCCC(=O)NO
ONC(=O)\C=C\c1ccc2C(=O)N(Cc3ccccc3)C(=O)c2c1
ONC(=O)c1ccc2NCC(Cc2c1)Nc1nccc(n1)-c1cccnc1
ONC(=O)c1ccc(NC2CCN(C2=O)c2ccccc2)cc1
CN(C1CCN(C1=O)c1ccccc1)c1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(OC2CCN(C2=O)c2ccccc2)cc1
CNc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(NC2CN(C(=O)C2)c2ccccc2)cc1
ONC(=O)c1ccc(NC2CCN(Cc3ccccc3)C2=O)cc1
ONC(=O)c1ccc(NC2CCN(CCc3ccccc3)C2=O)cc1
ONC(=O)c1ccc(NC2CCN(C2=O)c2ccc(Cl)cc2)cc1
ONC(=O)c1ccc(NC2CCN(C2=O)c2cccc(Cl)c2)cc1
ONC(=O)c1ccc(NC2CCN(C2=O)c2ccccc2Cl)cc1
ONC(=O)c1ccc(NC2CCN(C2=O)c2ccc(cc2)C(F)(F)F)cc1
ONC(=O)c1ccc(NC2CCN(C2=O)c2ccc(Cl)c(Cl)c2)cc1
CS(=O)(=O)c1ccc(cc1)N1CCC(Nc2ccc(cc2)C(=O)NO)C1=O
ONC(=O)c1ccc(NC2CCN(C2=O)c2ccc(cc2)C#N)cc1
ONC(=O)c1ccc(NC2CCN(C2=O)c2ccc(Cl)cc2)c(Cl)c1
ONC(=O)c1ccc(NC2CCN(C2)c2ccc(Cl)cc2)cc1
CC1(CCN(C1=O)c1ccccc1)Nc1ccc(cc1)C(=O)NO
CC1(CCN(C1=O)c1ccc(Cl)cc1)Nc1ccc(cc1)C(=O)NO
CC1(CCN(C1=O)c1ccc2ncccc2c1)Nc1ccc(cc1)C(=O)NO
C[C@@]1(CCN(C1=O)c1ccc(Cl)cc1)Nc1ccc(cc1)C(=O)NO |r|
C[C@]1(CCN(C1=O)c1ccc(Cl)cc1)Nc1ccc(cc1)C(=O)NO |r|
CN(C)CCOc1cccc(c1)N1CCC(Nc2ccc(cc2)C(=O)NO)C1=O
ONC(=O)c1ccc(NC2CCN(C2=O)c2ccc3ccccc3c2)cc1
ONC(=O)c1ccc(NC2CCN(C2=O)c2ccc(Cl)cc2)cc1F
Nc1nc2ncc(CNc3ccc(cc3)C(=O)N[C@@H](CCC(=O)NCCCCCCCCC(=O)NO)C(O)=O)nc2c(=O)[nH]1 |r|
Nc1nc2ncc(CNc3ccc(cc3)C(=O)N[C@@H](CCC(=O)NCCCCCCCC(=O)NO)C(O)=O)nc2c(=O)[nH]1 |r|
Nc1nc2ncc(CNc3ccc(cc3)C(=O)N[C@@H](CCC(=O)NCCCCCCC(=O)NO)C(O)=O)nc2c(=O)[nH]1 |r|
Nc1nc2ncc(CNc3ccc(cc3)C(=O)N[C@@H](CCC(=O)NCCCC(=O)NO)C(O)=O)nc2c(=O)[nH]1 |r|
Nc1nc2ncc(CNc3ccc(cc3)C(=O)NCCCCCCCCCC(=O)NO)nc2c(=O)[nH]1
Nc1nc2ncc(CNc3ccc(cc3)C(=O)NCCCCCCCCC(=O)NO)nc2c(=O)[nH]1
Nc1nc2ncc(CNc3ccc(cc3)C(=O)NCCCCCCCC(=O)NO)nc2c(=O)[nH]1
Nc1nc2ncc(CNc3ccc(cc3)C(=O)NCCCCCCC(=O)NO)nc2c(=O)[nH]1
Nc1nc2ncc(CNc3ccc(cc3)C(=O)NCCCCCC(=O)NO)nc2c(=O)[nH]1
Nc1nc2ncc(CNc3ccc(cc3)C(=O)NCCCCC(=O)NO)nc2c(=O)[nH]1
Nc1nc2ncc(CNc3ccc(cc3)C(=O)NCCCC(=O)NO)nc2c(=O)[nH]1
Nc1nc2ncc(CNc3ccc(cc3)C(=O)NO)nc2c(=O)[nH]1
ONC(=O)\C=C\c1ccc(NC(=O)C(Cc2ccccc2)c2ccccc2)cn1
ONC(=O)CCCCSc1nc(cc(=O)[nH]1)-c1ccc(cc1)-c1ccccc1
ONC(=O)CCCCCOc1no[n+]([O-])c1S(=O)(=O)c1ccccc1
NC(=O)C1CCCc2c1[nH]nc2-c1ccc(Cl)c(Cl)c1
CN1C2N(CCc3c2[nH]c2ccc(O)cc32)C(=O)c2cc(NCc3ccc(cc3)-c3noc(CCCCCCC(=O)NO)n3)ccc12
CC1=C(C)C(=O)C(CONC(=O)CCCCCCC(=O)Nc2ccccc2)=C(C)C1=O |c:1,t:27|
O=C(CCCCCCC(=O)Nc1ccccc1)NOCc1ccccc1
COC(=O)CCCCCCC(=O)Nc1ccc(OS(=O)(=O)C2CC3OC2C(=C3c2ccc(O)cc2)c2ccc(O)cc2)cc1 |c:27|
OC(=O)CCCCCCC(=O)Nc1ccc(OS(=O)(=O)C2CC3OC2C(=C3c2ccc(O)cc2)c2ccc(O)cc2)cc1 |c:26|
ONC(=O)CCCCCCC(=O)Nc1ccc(OS(=O)(=O)C2CC3OC2C(=C3c2ccc(O)cc2)c2ccc(O)cc2)cc1 |c:27|
COc1ccc(OS(=O)(=O)C2CC3OC2C(=C3c2ccc(O)cc2)c2ccc(NC(=O)CCCCCCC(O)=O)cc2)cc1 |c:16|
Cc1ccccc1OS(=O)(=O)C1CC2OC1C(=C2c1ccc(O)cc1)c1ccc(NC(=O)CCCCCCC(O)=O)cc1 |c:18|
OC(=O)CCCCCCC(=O)Nc1ccc(cc1)C1=C(C2CC(C1O2)S(=O)(=O)Oc1cccc(O)c1)c1ccc(O)cc1 |t:19|
OC(=O)CCCCCCC(=O)Nc1ccc(cc1)C1=C(C2CC(C1O2)S(=O)(=O)Oc1ccc(Cl)cc1)c1ccc(O)cc1 |t:19|
OC(=O)CCCCCCC(=O)Nc1ccc(cc1)C1=C(C2CC(C1O2)S(=O)(=O)Oc1ccc(cc1)C(F)(F)F)c1ccc(O)cc1 |t:19|
OC(=O)CCCCCCC(=O)Nc1ccc(cc1)C1=C(C2CC(C1O2)S(=O)(=O)Oc1ccc2ccccc2c1)c1ccc(O)cc1 |t:19|
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)C1=C(C2CC(C1O2)S(=O)(=O)Oc1ccc(Br)cc1)c1ccc(O)cc1 |t:20|
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)C1=C(C2CC(C1O2)S(=O)(=O)Oc1cccc2ccccc12)c1ccc(O)cc1 |t:20|
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)C1=C(C2CC(C1O2)S(=O)(=O)Oc1ccc2ccccc2c1)c1ccc(O)cc1 |t:20|
ONC(=O)c1ccc(NC(=O)CCN2C(=O)C3(OCCCO3)c3cc(Br)ccc23)cc1
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C[C@H](OC1=O)\C=C\CCS)n2 |r,c:11|
CC(C)[C@H]1C(=O)N[C@@H](CC(=O)NCc2nc(cs2)C3=N[C@@](CS3)(C(=O)N1)C)/C=C/CCS
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2cccc(CNC(=O)C[C@H](OC1=O)\C=C\CCS)n2 |r,c:11|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2ccnc(CNC(=O)C[C@H](OC1=O)\C=C\CCS)c2 |r,c:11|
CC(C)[C@H]1C(=O)N[C@@H](CC(=O)NCc2cc(ccn2)C3=N[C@@](CS3)(C(=O)N1)C)/C=C/CCS
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C[C@H](OC1=O)\C=C\CCSSC[C@H](NC(=O)OC(C)(C)C)C(=O)OC(C)(C)C)n2 |r,c:11|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C[C@H](OC1=O)\C=C\CCSSCC\C=C\[C@@H]1CC(=O)NCc3nc(cs3)C3=N[C@@](C)(CS3)C(=O)N[C@@H](C(C)C)C(=O)O1)n2 |r,c:11,t:50|
ONC(=O)CCCCC(=O)Nc1cc2c(Nc3ccc(F)c(Cl)c3)ncnc2s1
ONC(=O)CCCCCCC(=O)Nc1cc2c(Nc3ccc(F)c(Cl)c3)ncnc2s1
ONC(=O)CCCCCC(=O)Nc1cc2c(Nc3ccc(F)c(Cl)c3)ncnc2s1
ONC(=O)CCCCCC(=O)Nc1cc2c(Nc3ccc(Cl)c(c3)C(F)(F)F)ncnc2s1
ONC(=O)CCCCCCC(=O)Nc1cc2c(Nc3ccc(Cl)c(c3)C(F)(F)F)ncnc2s1
ONC(=O)CCCCCCC(=O)Nc1cc2c(Nc3ccc(Cl)cc3F)ncnc2s1
ONC(=O)CCCCCCC(=O)Nc1cc2c(Nc3ccc(F)cc3F)ncnc2s1
ONC(=O)CCCCCCC(=O)Nc1cc2c(Nc3ccc(I)cc3F)ncnc2s1
ONC(=O)CCCCCCC(=O)Nc1cc2c(Nc3ccc(Br)cc3F)ncnc2s1
ONC(=O)CCCCCCC(=O)Nc1cc2c(Nc3cccc(Cl)c3)ncnc2s1
ONC(=O)CCCCCCC(=O)Nc1cc2c(Nc3cccc(Cl)c3F)ncnc2s1
ONC(=O)CCCCCCC(=O)Nc1cc2c(Nc3ccccc3)ncnc2s1
ONC(=O)CCCCCC(=O)Nc1cc2c(Nc3ccccc3)ncnc2s1
Cc1ccc(Nc2ncnc3sc(NC(=O)CCCCCC(=O)NO)cc23)cc1
Cc1ccc(Nc2ncnc3sc(NC(=O)CCCCCC(=O)NO)cc23)cc1C
Cc1ccc(Nc2ncnc3sc(NC(=O)CCCCCCC(=O)NO)cc23)cc1
CCN(CC)c1ccc(Nc2ncnc3sc(NC(=O)CCCCCCC(=O)NO)cc23)cc1
Cc1ccc(Nc2ncnc3sc(NC(=O)CCCCCCC(=O)NO)cc23)cc1C
CN(C)c1ccc(Nc2ncnc3sc(NC(=O)CCCCCCC(=O)NO)cc23)cc1F
CCN(CC)c1ccc(Nc2ncnc3sc(NC(=O)CCCCCCC(=O)NO)cc23)cc1F
ONC(=O)CCCCCCC(=O)Nc1cc2c(Nc3ccc(N4CCCCC4)c(F)c3)ncnc2s1
ONC(=O)CCCCCCC(=O)Nc1cc2c(Nc3ccc(O[C@H]4CCOC4)c(Cl)c3)ncnc2s1 |r|
ONC(=O)CCCCCCC(=O)Nc1cc2c(Nc3ccc(cc3)N3CCCC3)ncnc2s1
ONC(=O)CCCCCCC(=O)Nc1cc2c(Nc3ccc(N4CCCC4)c(F)c3)ncnc2s1
ONC(=O)CCCCCCC(=O)Nc1cc2c(Cl)ncnc2s1
C[C@@]12Nc3ccccc3[C@]1(O)CCN2Cc1ccc(\C=C\C(N)=O)cc1 |r|
Cc1[nH]c2cc(O)ccc2c1CCNCc1ccc(\C=C\C(N)=O)cc1
C[C@@]12Nc3ccccc3[C@]1(O)CCN2Cc1ccc(\C=C\C(=O)NO)cc1 |r|
Cc1[nH]c2ccccc2c1CCNCc1ccc(\C=C\C(N)=O)cc1
ONC(=O)c1ccc(cc1)-c1cccc2ccccc12
c1ccc2c(c1)cccc2C(=O)NO
ONC(=O)c1cccc(c1)-c1ccccc1
ONC(=O)\C=C\c1cccc2ccccc12
ONC(=O)\C=C\C#Cc1ccc(NS(=O)(=O)c2ccccc2)cc1
Cn1cc(c2c1cccc2)CNCC3CCN(CC3)c4ncc(cn4)C(=O)NO
CCCCc1nc2cc(\C=C\C(=O)NO)ccc2n1CCN(CC)CC
CCN(CC)Cc1ccc2cc(ccc2c1)COC(=O)Nc3ccc(cc3)C(=O)NO
CN(C)c1ccc(cc1)C(=O)NCCCNC(=O)CS
CN(C)c1ccc(cc1)C(=O)NCCCCNC(=O)CS
SCC(=O)NCCCCCCNC(=O)Nc1ccccc1
ONC(=O)CCCCCNC(=O)NC12CC3CC(CC(C3)C1)C2 |THB:18:17:14:20.19.21,18:19:16.17.22:14,21:19:16:22.13.14,21:13:16:20.18.19,12:13:16:20.18.19|
SCC(=O)NCCCCCC(=O)Nc1cccc2cccnc12
CN(C)c1ccc(cc1)C(=O)NCCCCCCNC(=O)CS
N[C@@H](Cc1ccccc1)C(=O)Nc1ccccc1-c1ccc(NC(=O)CCCCCCC(=O)NO)cc1
CN(C)c1ccc(cc1)C(=O)NCCCCCNC(=O)CS
N[C@@H](Cc1ccc(O)cc1)C(=O)Nc1ccccc1-c1ccc(NC(=O)CCCCCCC(=O)NO)cc1
ONC(=O)CCCCCCC(=O)Nc1nc(cs1)-c1cccc(c1)[N+]([O-])=O
CN(C)c1ccc(NC(=O)NCCCCCCC(=O)NO)cc1
N[C@@H](Cc1c[nH]c2ccccc12)C(=O)Nc1ccccc1-c1ccc(NC(=O)CCCCCCC(=O)NO)cc1
CN(C)c1ccc(CNC(=O)NCCC(=O)NO)cc1
Cc1ccc(Nc2nccc3ccc(NC(=O)CCCCCCC(=O)NO)cc23)c(Cl)c1
Cc1ccc(Nc2nccc3ccc(NC(=O)CCCCCCC(=O)NO)cc23)c(Br)c1
ONC(=O)CCCCCCC(=O)Nc1ccc2ccnc(Nc3ccccc3F)c2c1
CC(C)CCn1ccc2ccc(NC(=O)CCCCCCC(=O)NO)cc2c1=O
COCCN(CCOC)c1nccc2ccc(NC(=O)CCCCCCC(=O)NO)cc12
COc1ccc(Cn2ccc3ccc(NC(=O)CCCCCCC(=O)NO)cc3c2=O)c(OC)c1
ONC(=O)CCCCCCC(=O)Nc1ccc2ccnc(N3CCOCC3)c2c1
ONC(=O)c1ccc(OCC(=O)Nc2ccc3ccnc(Nc4ccc5ccccc5c4)c3c2)cc1
CC(C)N1CCN(CC1)c1nccc2ccc(NC(=O)CCCCCCC(=O)NO)cc12
Cc1ccc(Nc2nccc3ccc(NCc4ccc(cc4)C(=O)NO)cc23)cc1
COCCCNc1nccc2ccc(NC(=O)CCCCCCC(=O)NO)cc12
Cc1ccc(Nc2nccc3ccc(NCc4ccc(\C=C\C(=O)NO)cc4)cc23)cc1
CCCCn1ccc2ccc(NC(=O)CCCCCCC(=O)NO)cc2c1=O
Cc1ccc(Nc2nccc3ccc(NCc4ccc(\C=C\C(=O)NO)cc4)cc23)c(Cl)c1
CCN(CC)CCn1ccc2ccc(NC(=O)CCCCCCC(=O)NO)cc2c1=O
Cc1ccc(Nc2nccc3ccc(NCc4ccc(\C=C\C(=O)NO)cc4)cc23)c(Br)c1
ONC(=O)CCCCCCC(=O)Nc1ccc2ccnc(Nc3ccc4ccccc4c3)c2c1
Cc1ccc(Nc2nccc3ccc(NC(=O)CCCCCCC(=O)NO)cc23)c(F)c1
ONC(=O)CCCCCCC(=O)Nc1ccc2ccnc(Nc3ccc(Br)cc3F)c2c1
ONC(=O)CCCCCCC(=O)Nc1ccc2ccnc(Nc3cccc(Cl)c3F)c2c1
Cc1ccc(Nc2nccc3ccc(NC(=O)CCCCCCC(=O)NO)cc23)cc1
Nc1ccccc1NC(=O)c1ccc(cc1)C(C(=O)Nc1ccccc1)C(=O)Nc1ccccc1
ONC(=O)\C=C\c1ccc2CN(Cc3ccc(cc3)-c3ccncc3)C(=O)c2c1
ONC(=O)\C=C\c1ccc2CN(Cc3ccc(cc3)-c3ccccc3)C(=O)c2c1
ONC(=O)\C=C\c1ccc2CN(Cc3ccccc3)C(=O)c2c1
CC(C)(C)c1ccc(CN2Cc3ccc(\C=C\C(=O)NO)cc3C2=O)cc1
ONC(=O)\C=C\c1ccc2CN(Cc3ccc(cc3)-c3cccnc3)C(=O)c2c1
C[C@H]1CN(CCN1C(=O)OCc1ccccc1)c1ccc(cn1)C(=O)Nc1ccccc1N |r|
Nc1ccccc1NC(=O)c1ccc(CNC2=N[C@H]([C@@H](O2)c2ccccc2)c2ccccc2)cc1 |r,t:17|
CC[C@H](C)[C@@H]1NC(=O)C(C)(C)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C1=O
CCCC[C@@H]1NC(=O)C(C)(C)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C1=O
CC(C)C[C@@H]1NC(=O)C(C)(C)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C1=O
O=C1N[C@@H](CCCCCSSc2ccccn2)C(=O)N[C@@H]2CCCCCCCCCCCC[C@H](NC2=O)C(=O)N2CCC[C@H]12
CCOC(=O)NCc1ccc(cc1)C(=O)Nc1cc(ccc1N)-c1cccs1
COC(=O)NCc1ccc(cc1)C(=O)Nc1cc(ccc1N)-c1ccccc1
Nc1ccc(cc1NC(=O)c1ccc(CNC(=O)OCc2cccnc2)cc1)-c1ccccc1
Nc1ccc(cc1NC(=O)c1ccc(CNC(=O)OCc2cccnc2)cc1)-c1cccs1
COC(=O)NCc1ccc(cc1)C(=O)Nc1cc(ccc1N)-c1cccs1
Oc1ccc(cc1NC(=O)c1cccs1)-c1ccccc1
C1=CC(=S)N(C(=C1)C(=O)O)O
OC(=O)[C@H](NC(=O)c1cccc(=S)n1O)c1ccccc1 |r|
C[C@@H](NC(=O)c1cccc(=S)n1O)C(O)=O |r|
Nc1ccccc1NC(=O)c1ccc(s1)-c1cn(CCc2cccc(c2)[N+]([O-])=O)nn1
Nc1ccccc1NC(=O)c1ccc(cc1)-c1cn(CCc2ccsc2)nn1
CCSC(=S)SCC(=O)c1ccc(NC(=O)Nc2ccccc2)cc1
CCSC(=S)SCC(=O)c1ccc(cc1)C(=O)NCCOc1ccccc1
CCSC(=S)SCC(=O)c1cccc(c1)C(=O)NCCOc1ccccc1
CCSC(=S)SCC(=O)c1ccc(CNC(=O)c2ccccc2)cc1
CCSC(=S)SCC(=O)c1ccc(cc1)C(=O)NCc1ccccc1
CCSC(=S)SCC(=O)c1cccc(c1)C(=O)NCc1ccccc1
CCSC(=S)SCC(=O)c1cccc(NC(=O)c2cnc3ccccc3c2)c1
CCSC(=S)SCC(=O)c1ccc(NC(=O)c2cccnc2)cc1
CCSC(=S)SCC(=O)c1cccc(NC(=O)c2cccnc2)c1
CCSC(=S)SCC(=O)c1ccc(Nc2ncnc3ccccc23)cc1
CCSC(=S)SCC(=O)c1ccc(NS(=O)(=O)c2ccccc2)cc1
CCSC(=S)SCC(=O)c1cccc(NS(=O)(=O)c2ccccc2)c1
CCSC(=S)SCC(=O)c1ccc(NC(=O)c2ccccc2)cc1
CCSC(=S)SCC(=O)c1cccc(NC(=O)c2ccccc2)c1
CCSC(=S)SCC(=O)c1ccc(cc1)C(=O)Nc1ccccc1
CCSC(=S)SCC(=O)c1cccc(c1)C(=O)Nc1ccccc1
CCSC(=S)SCC(=O)c1ccc(CCNC(C)=O)cc1
CCSC(=S)SCC(=O)c1ccc(CN(C)C(C)=O)cc1
CCSC(=S)SCC(=O)c1ccc(NS(C)(=O)=O)cc1
CCSC(=S)SCC(=O)c1ccc(CNC(C)=O)cc1
CCSC(=S)SCC(=O)c1cccc(CNC(C)=O)c1
CCSC(=S)SCC(=O)c1cccc(NC(C)=O)c1
CCNC(=S)SCC(=O)c1ccc(NC(C)=O)cc1
CCOC(=S)SCC(=O)c1ccc(NC(C)=O)cc1
CCCC(=S)SCC(=O)c1ccc(NC(C)=O)cc1
CCSC(=S)SCC(=O)c1ccc(NC(C)=O)cc1
CCSC(=S)SCC(=O)c1ccc(C)cc1
CCSC(=S)SCC(=O)c1ccc(NC(=O)c2cnc3ccccc3c2)cc1
CCSC(=S)SCC(=O)c1ccc(OC)cc1
COCCSC(=S)SCC(=O)c1ccc(OC)cc1
COc1ccc(cc1)C(=O)CSC(=S)SCCNC(C)=O
COc1ccc(cc1)C(=O)CSC(=S)SCCOc1ccccc1
CCNC(=O)SCC(=O)c1ccc(OC)cc1
CCOC(=O)SCC(=O)c1ccc(OC)cc1
CCNC(=S)SCC(=O)c1ccc(OC)cc1
CCOC(=S)SCC(=O)c1ccc(OC)cc1
CCCC(=S)SCC(=O)c1ccc(OC)cc1
CCSC(=S)SCC(=O)c1ccn(c1)S(=O)(=O)c1ccccc1
CCSC(=S)SCC(=O)c1ccc(s1)-c1ccc(N)cn1
CCSC(=S)SCC(=O)c1ccc(s1)-c1ccc(CNc2cnc3ccccc3c2)cn1
CCSC(=S)SCC(=O)c1ccc(CC(=O)NCCOc2ccccc2)s1
CCSC(=S)SCC(=O)c1ccc(CC(=O)Nc2ccc(OC)cc2)s1
CCSC(=S)SCC(=O)c1ccc(CC(=O)NCc2ccc(OC)cc2)s1
CCSC(=S)SCC(=O)c1ccc(CC(=O)NCc2ccccc2)s1
CCSC(=S)SCC(=O)c1ccc(s1)C(=O)Nc1ccccc1
CCSC(=S)SCC(=O)c1ccc(s1)C(=O)NCc1cc(C)cc(C)c1
CCCSC(=S)SCC(=O)c1ccc(s1)C(=O)N[C@H](C)c1ccccc1 |r|
CCSC(=S)SCC(=O)c1ccc(s1)C(=O)N[C@@H](C)c1ccccc1 |r|
CCSC(=S)SCC(=O)c1ccc(s1)C(=O)NCc1ccccc1
CCSC(=S)SCC(=O)c1cccc(c1)S(=O)(=O)Nc1ccc2OCOc2c1
CCSC(=S)SCC(=O)c1cccc(c1)S(=O)(=O)Nc1cccc(c1)C(N)=O
CCSC(=S)SCC(=O)c1cccc(c1)S(=O)(=O)N(C)c1ccc(OC)cc1
CCSC(=S)SCC(=O)c1cccc(c1)S(=O)(=O)Nc1ccc(OC)cc1
CCSC(=S)SCC(=O)c1ccc(cc1)S(=O)(=O)Nc1ccc(OC)cc1
CCSC(=S)SCC(=O)c1cccc(NS(=O)(=O)c2ccc(Cl)cc2)c1
CCSC(=S)SCC(=O)c1ccc(NS(=O)(=O)c2ccc(Cl)cc2)cc1
CCSC(=S)SCC(=O)c1ccc(cc1)S(=O)(=O)Nc1ccc(Cl)cc1
CCSC(=S)SCC(=O)c1ccc(cc1)C(=O)Nc1ccc(Cl)cc1
C\C=C1/NC(=O)[C@@H](CS)NC(=O)[C@H](CC(=O)C[C@H](OC(=O)[C@@H](NC1=O)C(C)C)\C=C\CCS)C(C)C |r|
C\C=C1/NC(=O)[C@H](CS)NC(=O)[C@H](NC(=O)C[C@H](OC(=O)[C@@H](NC1=O)C(C)C)\C=C\CCS)C(C)C |r|
C\C=C1/NC(=O)c2csc(n2)[C@H](NC(=O)C[C@H](OC(=O)[C@@H](NC1=O)C(C)C)\C=C\CCS)C(C)C |r|
CCCCCCCC(=O)SCC\C=C\[C@@H]1CC(=O)N[C@H](C(C)C)c2nc(cs2)C(=O)N\C(=C/C)C(=O)N[C@@H](C(C)C)C(=O)O1 |r|
C\C=C1/NC(=O)c2csc(CNC(=O)C[C@H](OC(=O)[C@@H](NC1=O)C(C)C)\C=C\CCS)n2 |r|
CCCCCCCC(=O)SCC\C=C\[C@@H]1CC(=O)NCc2nc(cs2)C(=O)N\C(=C/C)C(=O)N[C@@H](C(C)C)C(=O)O1 |r|
C\C=C1/NC(=O)c2csc(CNC(=O)C[C@H](OC(=O)[C@@H](NC1=O)C(C)C)\C=C\CCSC(C)=O)n2 |r|
ONC(=O)N\C=C\c1ccc(cc1)-c1ccccc1
ONC(=O)CCCCOCc1cc(on1)-c1ccccc1
CC(=O)Nc1ccc(cc1)-c1cc(no1)C(=O)NCCCCCCC(=O)NO
Nc1ccc(cc1)-c1cc(no1)C(=O)NCCCCC(=O)NO
Nc1ccc(cc1)-c1cc(no1)C(=O)NCCCCCCC(=O)NO
CC(C)(C)OC(=O)Nc1ccc(cc1)-c1cc(no1)C(=O)NCCCCC(=O)NO
CC(C)(C)OC(=O)Nc1ccc(cc1)-c1cc(no1)C(=O)NCCCCCCC(=O)NO
Nc1cccc(c1)-c1cc(no1)C(=O)NCCCCC(=O)NO
Nc1cccc(c1)-c1cc(no1)C(=O)NCCCCCCC(=O)NO
CC(C)(C)OC(=O)Nc1cccc(c1)-c1cc(no1)C(=O)NCCCCC(=O)NO
ONC(=O)CCCCNC(=O)c1cc(on1)-c1ccccc1
C\C(\C=C\c1ccccc1)=C/C(=O)NCCCCCC(=O)NO
ONC(=O)CCCCCNC(=O)\C=C\c1ccc2cccnc2c1
[#8]-[#7]-[#6](=O)-[#6]-[#6]-[#6]-[#6]-[#6]-[#7]-[#6](=O)\[#6]=[#6]-1\c2ccccc2-c2ccccc-12
ONC(=O)CCCCCNC(=O)\C=C\c1ccc(Cl)cc1F
CCCCCCCC(=O)SCC\C=C\[C@@H]1CC(=O)N[C@H](C(C)C)C(=O)N[C@H](C)C(=O)N[C@H](C(C)C)C(=O)NCC(=O)O1 |r|
CCCCCCCCSSCC\C=C\[C@@H]1CC(=O)N[C@H](C(C)C)C(=O)N[C@H](C)C(=O)N[C@H](C(C)C)C(=O)NCC(=O)O1 |r|
CC(C)[C@H]1NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](NC(=O)C[C@H](OC(=O)Cn2cc1nn2)\C=C\CCSC(C)=O)C(C)C |r|
CC(C)[C@H]1NC(=O)[C@@H](Cc2cn(C)cn2)NC(=O)[C@H](NC(=O)C[C@H](OC(=O)Cn2cc1nn2)\C=C\CCSC(C)=O)C(C)C |r|
CS(=O)(=O)Cc1noc(n1)-c1ccc(s1)C(=O)C(F)(F)F
CCCS(=O)(=O)Cc1noc(n1)-c1ccc(s1)C(=O)C(F)(F)F
FC(F)(F)C(=O)c1ccc(s1)-c1nnc(o1)-c1cccs1
FC(F)(F)C(=O)c1ccc(s1)-c1nc(Cc2cccs2)no1
Fc1ccc(cc1)-c1noc(n1)-c1ccc(s1)C(=O)C(F)(F)F
FC(F)(F)C(=O)c1ccc(s1)-c1nnc(o1)-c1ccccc1
FC(F)(F)C(=O)c1ccc(s1)C(=O)NCc1ccccc1
FC(F)(F)C(=O)c1ccc(s1)-c1nc(CN2C(=O)COc3ccccc23)no1
FC(F)(F)C(=O)c1ccc(s1)-c1nc(no1)-c1ccccn1
FC(F)(F)C(=O)c1ccc(s1)-c1nc(CS(=O)(=O)c2cccs2)no1
FC(F)(F)C(=O)c1ccc(s1)-c1nc(no1)-c1ccncc1
FC(F)(F)C(=O)c1ccc(s1)-c1nc(no1)-c1ccccc1
Fc1ccc(-c2noc(n2)-c2ccc(s2)C(=O)C(F)(F)F)c(F)c1
Cc1ccc(cc1)-c1nnc(o1)-c1ccc(s1)C(=O)C(F)(F)F
Cc1noc(n1)-c1ccc(s1)C(=O)C(F)(F)F
FC(F)(F)C(=O)c1ccc(s1)-c1nc(no1)-c1cccs1
Cc1cccc(c1)-c1noc(n1)-c1ccc(s1)C(=O)C(F)(F)F
Fc1ccc(CS(=O)(=O)Cc2noc(n2)-c2ccc(s2)C(=O)C(F)(F)F)cc1
FC(F)(F)C(=O)c1ccc(s1)-c1nc(CC(=O)N2CCCC2)no1
FC(F)(F)C(=O)c1ccc(s1)-c1nc(COc2ccc(cc2)-c2nnco2)no1
FC(F)(F)C(=O)c1ccc(s1)-c1nc(no1)-c1cccnc1
Cc1ccc(cc1)-c1noc(n1)-c1ccc(s1)C(=O)C(F)(F)F
FC(F)(F)C(=O)c1ccc(s1)-c1ncc(s1)-c1ccccc1
FC(F)(F)C(=O)c1ccc(s1)-c1nc(no1)-c1cccc(c1)C(F)(F)F
FC(F)(F)C(=O)c1ccc(s1)-c1nc(no1)-c1ccc(Cl)cc1Cl
CC(C)(C)c1ccc(cc1)-c1noc(n1)-c1ccc(s1)C(=O)C(F)(F)F
FC(F)(F)C(=O)c1ccc(s1)-c1nc(no1)-c1ccc(cc1)C(F)(F)F
Oc1ccc(cc1NC(=O)c1ccccc1)-c1ccccc1
FC(F)(F)C(=O)c1ccc(nc1)C(=O)NCC1CCCCC1
FC(F)(F)C(=O)c1cnc(s1)C(=O)N1CCc2ccccc12
FC(F)(F)C(=O)c1ccc(s1)C(=O)NCc1ccccc1Cl
FC(F)(F)C(=O)c1ccc(s1)C(=O)N1CCC(CC1)c1nnc(o1)-c1ccccc1
CC(NC(=O)c1ccc(s1)C(=O)C(F)(F)F)c1ccncc1
CC(NC(=O)c1ccc(s1)C(=O)C(F)(F)F)c1cccc2ccccc12
COc1ccc(Cl)cc1N1CCN(CC1)C(=O)c1ccc(s1)C(=O)C(F)(F)F
COc1cccc(c1)N1CCN(CC1)C(=O)c1ccc(s1)C(=O)C(F)(F)F
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1ccccc1
Nc1ccccc1NC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1ccccc1
NS(=O)(=O)NCCCCC(=O)Nc1cccc(c1)-c1ccccc1
NS(=O)(=O)NCCCCCC(=O)Nc1cccc(c1)-c1ccccc1
NS(=O)(=O)NCCCCCCC(=O)Nc1cccc(c1)-c1ccccc1
CNS(=O)(=O)NCCCCCC(=O)Nc1cccc(c1)-c1ccccc1
CN(C)S(=O)(=O)NCCCCCC(=O)Nc1cccc(c1)-c1ccccc1
CN(CCCCCC(=O)Nc1cccc(c1)-c1ccccc1)S(N)(=O)=O
NS(=O)(=O)OCCCCCC(=O)Nc1cccc(c1)-c1ccccc1
NS(=O)(=O)NC(=O)CCCCCC(=O)Nc1cccc(c1)-c1ccccc1
CC(=O)NS(=O)(=O)NCCCCCC(=O)Nc1cccc(c1)-c1ccccc1
NS(=O)(=O)NCCCCCC(=O)Nc1ccccc1
NS(=O)(=O)NCCCCCC(=O)Nc1cccc2cccnc12
NS(=O)(=O)NCCCCCC(=O)Nc1ccc2ncccc2c1
NS(=O)(=O)NCCCCCC(=O)Nc1cnc2ccccc2c1
COc1cc(NC(=O)CCCCCNS(N)(=O)=O)c2ncccc2c1
NS(=O)(=O)NCCCCCC(=O)Nc1nc(cs1)-c1ccccc1
NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1nc(cs1)-c1ccccc1 |r|
COc1cc(NC(=O)[C@H](CCCCNS(N)(=O)=O)NC(=O)OCc2ccccc2)c2ncccc2c1 |r|
ONC(=O)c1ccc(CN2CC(=O)Nc3ccccc23)cc1
ONC(=O)c1ccc(CN2[C@H](Cc3ccccc3)C(=O)Nc3ccccc23)cc1 |r|
ONC(=O)c1ccc(CN2[C@@H](Cc3ccccc3)C(=O)Nc3ccccc23)cc1 |r|
ONC(=O)c1ccc(CN2[C@H](Cc3cccs3)C(=O)Nc3ccccc23)cc1 |r|
ONC(=O)c1ccc(CN2[C@@H](Cc3cccs3)C(=O)Nc3ccccc23)cc1 |r|
ONC(=O)c1ccc(CN2[C@H](Cc3ccc(F)c(F)c3)C(=O)Nc3ccccc23)cc1 |r|
ONC(=O)c1ccc(CN2[C@H](Cc3ccc(O)cc3)C(=O)Nc3ccccc23)cc1 |r|
ONC(=O)c1ccc(CN2[C@H](CCc3ccccc3)C(=O)Nc3ccccc23)cc1 |r|
CC(C)(C)OC(=O)NCCCC[C@H]1N(Cc2ccc(cc2)C(=O)NO)c2ccccc2NC1=O |r|
CC(C)(C)Oc1ccc(C[C@H]2N(Cc3ccc(cc3)C(=O)NO)c3ccccc3NC2=O)cc1 |r|
ONC(=O)c1ccc(CN2[C@H](Cc3ccccc3)C(=O)NCC2=O)cc1 |r|
ONC(=O)c1ccc(CN2[C@H](Cc3c[nH]c4ccccc34)C(=O)NCC2=O)cc1 |r|
ONC(=O)c1ccc(CN2[C@H](Cc3cccs3)C(=O)NCC2=O)cc1 |r|
Nc1ccccc1NC(=O)c1ccc(CNc2nccc(n2)-c2cc[nH]n2)cc1
ONC(=O)\C=C\c1ccc2n(CCN3CCCC3)c(CCc3ccccc3)nc2c1
CCOP(=O)(CNCc1ccc(cc1)C(=O)Nc1cc(ccc1N)-c1cccs1)OCC
CCOC(=O)c1csc(NC(=O)[C@H](CCCCNS(N)(=O)=O)NC(=O)OCc2ccccc2)n1 |r|
CC(C)(C)c1csc(NC(=O)[C@H](CCCCNS(N)(=O)=O)NC(=O)OCc2ccccc2)n1 |r|
NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1nc2ccccc2s1 |r|
NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1nccs1 |r|
Cn1nc(nc1-c1ccccc1)[C@H](CCCCNS(N)(=O)=O)NC(=O)OCc1ccccc1 |r|
NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)c1nnc([nH]1)-c1ccccc1 |r|
NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)c1cnc([nH]1)-c1ccccc1 |r|
NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)c1nc2cc(ccc2[nH]1)-c1cccs1 |r|
NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)c1nc2ccccc2[nH]1 |r|
NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)c1nc(no1)-c1ccc(F)cc1 |r|
NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)c1nnc(o1)-c1ccccc1 |r|
CN(C)CCOc1ccc(cc1)-c1nc(cs1)[C@H](CCCCNS(N)(=O)=O)NC(=O)OCc1ccccc1 |r|
COc1ccc(cc1)-c1nc(cs1)[C@H](CCCCNS(N)(=O)=O)NC(=O)OCc1ccccc1 |r|
NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)c1csc(n1)-c1ccccc1 |r|
NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)c1nc(cs1)-c1ccccc1 |r|
COc1ccc2[nH]c(C)c(CC(=O)N[C@@H](CCCCNS(N)(=O)=O)C(=O)Nc3nc(cs3)-c3ccccc3)c2c1 |r|
NS(=O)(=O)NCCCC[C@H](NS(=O)(=O)Cc1ccccc1)C(=O)Nc1nc(cs1)-c1ccccc1 |r|
NS(=O)(=O)NCCCC[C@H](NC(=O)NCc1ccc(F)cc1)C(=O)Nc1nc(cs1)-c1ccccc1 |r|
NS(=O)(=O)NCCCC[C@H](NC(=O)Nc1ccccc1)C(=O)Nc1nc(cs1)-c1ccccc1 |r|
NS(=O)(=O)NCCCC[C@H](NC(=O)Cc1ccccc1)C(=O)Nc1nc(cs1)-c1ccccc1 |r|
CCOC(=O)N[C@@H](CCCCNS(N)(=O)=O)C(=O)Nc1nc(cs1)-c1ccccc1 |r|
NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1cccnc1)C(=O)Nc1nc(cs1)-c1ccccc1 |r|
NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1cccc(Cl)c1)C(=O)Nc1nc(cs1)-c1ccccc1 |r|
NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)Nc1nc(cs1)-c1ccccc1 |r|
N[C@@H](CCCCNS(N)(=O)=O)C(=O)Nc1nc(cs1)-c1ccccc1 |r|
CC(C)c1ccc(cc1)-c1csc(NC(=O)[C@H](CCCCNS(N)(=O)=O)NC(=O)OCc2ccccc2)n1 |r|
NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1nc(cs1)-c1ccc(Cl)cc1 |r|
COc1cccc(c1)-c1csc(NC(=O)[C@H](CCCCNS(N)(=O)=O)NC(=O)OCc2ccccc2)n1 |r|
COc1ccc(cc1)-c1csc(NC(=O)[C@H](CCCCNS(N)(=O)=O)NC(=O)OCc2ccccc2)n1 |r|
NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1nc(c(s1)-c1ccccc1)-c1ccccc1 |r|
ONC(=O)\C=C\c1ccc(\C=N\OCc2ccc(cc2)[N+]([O-])=O)cc1
COC(=O)c1ccc(CO\N=C\c2ccc(\C=C\C(=O)NO)cc2)cc1
ONC(=O)\C=C\c1ccc(\C=N\OCCN2CCOCC2)cc1
ONC(=O)\C=C\c1ccc(cc1)-c1cc(CN2CCOCC2)on1
ONC(=O)\C=C\c1ccc(\C=N\OCc2c(F)c(F)c(F)c(F)c2F)cc1
Cc1ccc(NC(=O)c2ccc(cc2)C(=O)Nc2ccccc2N)cc1Nc1ncc(s1)-c1cccnc1
Cc1ccc(NCc2ccc(\C=C\C(=O)NO)cc2)cc1Nc1nccc(n1)-c1cccnc1
Cc1ccc(NC(=O)c2ccc(\C=C\C(=O)NO)s2)cc1Nc1ncc(s1)-c1cccnc1
Cc1ccc(NC(=O)c2ccc(\C=C\C(=O)NO)cc2)cc1Nc1ncc(s1)-c1cccnc1
ONC(=O)\C=C\c1ccc(s1)C(=O)Nc1cccc(Nc2ncc(s2)-c2cccnc2)c1
ONC(=O)\C=C\c1ccc(cc1)C(=O)Nc1cccc(Nc2ncc(s2)-c2cccnc2)c1
Cc1ccc(NC(=O)c2ccc(cc2)C(=O)NO)cc1Nc1ncc(s1)-c1cccnc1
ONC(=O)c1ccc(cc1)C(=O)Nc1cccc(Nc2ncc(s2)-c2cccnc2)c1
CN(C(=O)c1ccc(cc1)C(=O)Nc1ccccc1N)c1cccc(Nc2nccc(n2)-c2cccnc2)c1
CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)CC1
Nc1ccccc1NC(=O)c1ccc(CNCOC(=O)c2cccnc2)cc1
Cc1ccc(NC(=O)c2ccc(cc2)C(=O)Nc2ccccc2N)cc1Nc1ncc(cn1)-c1cccnc1
Cc1ccc(NC(=O)c2ccc(nc2)C(=O)Nc2ccccc2N)cc1Nc1ncc(cn1)-c1cccnc1
Cc1ccc(NC(=O)c2ccc(s2)C(=O)Nc2ccccc2N)cc1Nc1ncc(cn1)-c1cccnc1
Nc1ccccc1NC(=O)c1ccc(cn1)C(=O)Nc1cccc(Nc2ncc(s2)-c2cccnc2)c1
Cc1ccc(NC(=O)c2ccc(nc2)C(=O)Nc2ccccc2N)cc1Nc1ncc(s1)-c1cccnc1
Nc1ccccc1NC(=O)c1ccc(s1)C(=O)Nc1cccc(Nc2ncc(s2)-c2cccnc2)c1
Cc1ccc(NC(=O)c2ccc(s2)C(=O)Nc2ccccc2N)cc1Nc1ncc(s1)-c1cccnc1
Nc1ccccc1NC(=O)c1ccc(cc1)C(=O)Nc1cccc(Nc2ncc(s2)-c2cccnc2)c1
ONC(=O)\C=C\c1ccc(cc1)C(F)(F)F
ONC(=O)C=Cc1ccc2OC3(CCN(CCc4ccccc4)CC3)CC(=O)c2c1 |w:5.5|
ONC(=O)C=Cc1ccc2OC3(CCN(Cc4ccc(F)cc4)CC3)CC(=O)c2c1 |w:5.5|
ONC(=O)\C=C\c1ccc2OC3(CCN(Cc4ccccc4)C3)CC(=O)c2c1
ONC(=O)\C=C\c1ccc2OC3(CC(=O)c2c1)CCCN(Cc1ccccc1)CC3
COc1ccc2[nH]c(C)c(CC(=O)N[C@@H](CCCCCC(N)=O)c3nc(c[nH]3)-c3ccc4ccccc4c3)c2c1 |r|
OB(O)CCCCC[C@H](NC(=O)c1ccccc1)C(=O)Nc1cccc(c1)-c1ccccc1 |r|
OB(O)CCCCC[C@H](NC(=O)c1cccnc1)C(=O)Nc1cccc(c1)-c1ccccc1 |r|
OB(O)CCCCC[C@H](NC(=O)c1cncs1)C(=O)Nc1cccc(c1)-c1ccccc1 |r|
OB(O)CCCCC[C@@H](NC(=O)c1ccccc1)C(=O)Nc1cccc(c1)-c1ccccc1 |r|
OB(O)CCCCC[C@@H](NC(=O)c1cccnc1)C(=O)Nc1cccc(c1)-c1ccccc1 |r|
OB(O)CCCCC[C@@H](NC(=O)c1cncs1)C(=O)Nc1cccc(c1)-c1ccccc1 |r|
Nc1cccc(c1)-c1csc(NC(=O)CCCCCCC(=O)NO)n1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1ccccc1
ONC(=O)c1cc(CCCCC(=O)Nc2nc(cs2)-c2ccccc2)on1
Nc1cccc(c1)-c1csc(NC(=O)CCCCc2cc(no2)C(=O)NO)n1
OCc1cc(CCCCC(=O)Nc2nc(cs2)-c2ccccc2)on1
OC(=O)c1cc(CCCCC(=O)Nc2nc(cs2)-c2ccccc2)on1
NC(=O)c1cc(CCCCC(=O)Nc2nc(cs2)-c2ccccc2)on1
ONC(=O)c1cc(CCCCC(=O)Nc2cnc3ccccc3c2)on1
ONC(=O)c1cc(CCCCC(=O)Nc2ccc(cc2)-c2ccccc2)on1
ONC(=O)c1cc(CCCCC(=O)NC2CCCC2)on1
ONC(=O)c1cc(CCCCC(=O)NC2CCCCC2)on1
CC(C)(C)OC(=O)Nc1ccc(cc1)-c1cc(no1)C(=O)NCC(=O)Nc1ccc(cc1)-c1cc(no1)C(=O)NO
ONC(=O)CCCCCCC(=O)Nc1nc(cs1)-c1ccccc1
CCC(=O)CCCCC[C@H](NC(=O)C1CN(C)C1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
COc1cc2ncnc(Nc3ccc(Br)cc3)c2cc1OCCCCCCC(=O)NO
ONC(=O)\C=C\c1ccc(\C=C(\CNC2CC2)c2ccc(F)cc2)cc1
Fc1ccc(cc1)-c1cc(nn1Cc1ccccc1)C(=O)NCCCCCCS
OC(=O)Cn1nc(cc1-c1ccc(F)cc1)C(=O)NCCCCCCS
OC(=O)CCn1nc(cc1-c1ccc(F)cc1)C(=O)NCCCCCCS
OC(=O)CCCn1nc(cc1-c1ccc(F)cc1)C(=O)NCCCCCCS
OCCn1nc(cc1-c1ccc(F)cc1)C(=O)NCCCCCCS
OCCCn1nc(cc1-c1ccc(F)cc1)C(=O)NCCCCCCS
OCCCCn1nc(cc1-c1ccc(F)cc1)C(=O)NCCCCCCS
Cn1nc(cc1-c1ccc(F)cc1)C(=O)NCCCCCCS
CCn1nc(cc1-c1ccc(F)cc1)C(=O)NCCCCCCS
CCCn1nc(cc1-c1ccc(F)cc1)C(=O)NCCCCCCS
CC(C)n1nc(cc1-c1ccc(F)cc1)C(=O)NCCCCCCS
CCCCn1nc(cc1-c1ccc(F)cc1)C(=O)NCCCCCCS
CCC(C)n1nc(cc1-c1ccc(F)cc1)C(=O)NCCCCCCS
Cc1c(n[nH]c1C(=O)NCCCCCCS)-c1ccc(F)cc1
Cc1c(nn(C)c1C(=O)NCCCCCCS)-c1ccc(F)cc1
Cc1c(nn(CCCO)c1C(=O)NCCCCCCS)-c1ccc(F)cc1
Fc1ccc(cc1)-c1cc(no1)C(=O)NCCS
Fc1ccc(cc1)-c1cc(no1)C(=O)NCCCS
Fc1ccc(cc1)-c1cc(no1)C(=O)NCCCCS
Fc1ccc(cc1)-c1cc(no1)C(=O)NCCCCCS
Fc1ccc(cc1)-c1cc(no1)C(=O)NCCCCCCS
Fc1ccc(cc1)-c1cc(n[nH]1)C(=O)NCCCCCS
CC(=O)SCCCCCCNC(=O)c1cc(nn1C)-c1ccc(F)cc1
Fc1ccc(cc1)-c1cc([nH]n1)C(=O)NCCCCCCS
Fc1ccc(cc1)-c1cc(n[nH]1)C(=O)NCCNC(=O)CS
Fc1ccc(cc1)-c1cc(n[nH]1)C(=O)NCCCNC(=O)CS
Fc1ccc(cc1)-c1cc(n[nH]1)C(=O)NCCCCNC(=O)CS
Fc1ccc(cc1)-c1cc(n[nH]1)C(=O)NCCNC(=O)CCS
Fc1ccc(cc1)-c1cc(n[nH]1)C(=O)NCCCNC(=O)CCS
Fc1ccc(cc1)-c1cc(n[nH]1)C(=O)NCCCCNC(=O)CCS
Cn1nc(cc1C(=O)NCCCCCCS)-c1ccc(F)cc1
CCn1nc(cc1C(=O)NCCCCCCS)-c1ccc(F)cc1
CCCn1nc(cc1C(=O)NCCCCCCS)-c1ccc(F)cc1
CC(C)n1nc(cc1C(=O)NCCCCCCS)-c1ccc(F)cc1
CCCCn1nc(cc1C(=O)NCCCCCCS)-c1ccc(F)cc1
CCC(C)n1nc(cc1C(=O)NCCCCCCS)-c1ccc(F)cc1
Fc1ccc(cc1)-c1cc(C(=O)NCCCCCCS)n(Cc2ccccc2)n1
OC(=O)Cn1nc(cc1C(=O)NCCCCCCS)-c1ccc(F)cc1
OC(=O)CCn1nc(cc1C(=O)NCCCCCCS)-c1ccc(F)cc1
OC(=O)CCCn1nc(cc1C(=O)NCCCCCCS)-c1ccc(F)cc1
OCCn1nc(cc1C(=O)NCCCCCCS)-c1ccc(F)cc1
OCCCn1nc(cc1C(=O)NCCCCCCS)-c1ccc(F)cc1
OCCCCn1nc(cc1C(=O)NCCCCCCS)-c1ccc(F)cc1
ONC(=O)CCCCCC(=O)N\N=C\c1ccc(cc1)-c1ccccc1
ONC(=O)CCCCCC(=O)N\N=C\c1ccc(cc1)-c1cccnc1
SCCCCCCNC(=O)c1ccn[nH]1
SCCCCCCNC(=O)c1cc(n[nH]1)C1CCCCC1
SCCCCCCNC(=O)c1cc(n[nH]1)-c1ccccc1
COc1ccc(cc1)-c1cc([nH]n1)C(=O)NCCCCCCS
COc1ccc(cc1OC)-c1cc([nH]n1)C(=O)NCCCCCCS
COc1cc(cc(OC)c1OC)-c1cc([nH]n1)C(=O)NCCCCCCS
SCCCCCCNC(=O)c1cc(n[nH]1)-c1ccc(cc1)-c1ccccc1
SCCCCCCNC(=O)c1cc(n[nH]1)-c1cccc2ccccc12
SCCCCCCNC(=O)c1cc(n[nH]1)-c1ccc2ccccc2c1
SCCCCCCNC(=O)c1cc(n[nH]1)-c1ccncc1
SCCCCCCNC(=O)c1cc(n[nH]1)-c1cccnc1
SCCCCCCNC(=O)c1cc(n[nH]1)-c1ccccn1
SCCCCCCNC(=O)c1cc(n[nH]1)-c1cnccn1
SCCCCCCNC(=O)c1cc(n[nH]1)-c1c[nH]c2ccccc12
CN(C)c1ccc(cc1)C(=O)N\N=C\c1cccc(c1)C(=O)NO
CN(C)c1ccc(cc1)C(=O)N(C)\N=C\c1cccc(c1)C(=O)NO
CN(C)c1ccc(cc1)C(=O)N\N=C\c1ccc(cc1)C(=O)NO
CN(C)c1ccc(cc1)C(=O)N(C)\N=C\c1ccc(cc1)C(=O)NO
CN(C)c1ccc(cc1)C(=O)N\N=C(/C)c1ccc(cc1)C(=O)NO
CN(C)c1ccc(cc1)C(=O)N(C)\N=C(/C)c1ccc(cc1)C(=O)NO
ONC(=O)c1csc(n1)-c1cccnc1
ONC(=O)c1csc(n1)-c1cnccn1
ONC(=O)c1csc(n1)-c1ccc(Br)cc1
ONC(=O)c1csc(Cc2ccccc2)n1
ONC(=O)c1csc(n1)C(c1ccccc1)c1ccccc1
ONC(=O)c1csc(n1)-c1ccccc1
ONC(=O)c1coc(n1)-c1ccccc1
ONC(=O)c1coc(n1)-c1ccc(Br)cc1
ONC(=O)c1coc(n1)-c1ccc(cc1)-c1ccccc1
ONC(=O)c1coc(n1)C(c1ccccc1)c1ccccc1
ONC(=O)c1coc(n1)-c1cccs1
ONC(=O)c1coc(n1)-c1ccccc1Br
ONC(=O)c1coc(n1)-c1ccc(Cl)cc1
ONC(=O)c1coc(n1)-c1ccc(F)cc1
COc1ccc(cc1)-c1nc(co1)C(=O)NO
ONC(=O)c1coc(n1)-c1ccc2ccccc2c1
COc1ccc2cc(ccc2c1)-c1nc(co1)C(=O)NO
Cc1ccc(cc1)-c1nc(co1)C(=O)NO
ONC(=O)c1coc(n1)-c1cccc(c1)-c1ccccc1
ONC(=O)c1noc(n1)-c1ccccc1
ONC(=O)c1noc(n1)-c1ccc(Br)cc1
ONC(=O)c1noc(n1)-c1ccc(cc1)-c1ccccc1
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2ccc(CNC(=O)C[C@H](OC1=O)\C=C\CCSC(C)=O)cc2 |r,wU:22.27,wD:3.2,7.7,c:11,(-2.44,-5.97,;-3.02,-4.88,;-4.25,-4.85,;-2.21,-3.56,;-3.34,-2.53,;-4.03,-1.15,;-5.22,-1.48,;-4.17,.39,;-3.28,-.46,;-2.34,.31,;-1.66,1.69,;-2.82,3.1,;-3.75,1.87,;-1.51,3.91,;-.42,1.95,;1.1,1.67,;2.82,3.1,;3.75,1.87,;4.17,.39,;4.03,-1.15,;5.22,-1.48,;3.34,-2.53,;2.21,-3.56,;.77,-4.12,;-.77,-4.12,;-1,-5.33,;3.02,-4.88,;4.56,-4.83,;5.38,-6.14,;6.92,-6.09,;7.73,-7.4,;9.27,-7.35,;9.85,-6.26,;9.92,-8.39,;1.51,3.91,;,4.19,)|
[H][C@]12CCCN1C(=O)[C@]1([H])CCCN1C(=O)C[C@@H](NC(=O)[C@@H](NC2=O)C(C)C)C(=O)NCCCC(=O)NO |r|
[H][C@@]12CCCN1C(=O)[C@@]1([H])CCCN1C(=O)C[C@H](NC(=O)[C@@H](NC2=O)C(C)C)C(=O)NCCCC(=O)NO |r|
COc1ccc(Nc2nc(C)nc3ccccc23)cc1OCCCC(=O)NO
CN(c1ccc(OCC(=O)NO)cc1)c1ncnc2ccccc12
CN(c1ccc(OCCCC(=O)NO)cc1)c1ncnc2ccccc12
CN(c1ccc(OCCCCC(=O)NO)cc1)c1ncnc2ccccc12
CN(c1ccc(OCCCCCC(=O)NO)cc1)c1ncnc2ccccc12
CN(c1ccc(OCC(=O)NO)cc1)c1nc(C)nc2CCCc12
CN(c1ccc(OCCCC(=O)NO)cc1)c1nc(C)nc2CCCc12
CN(c1ccc(OCCCCC(=O)NO)cc1)c1nc(C)nc2CCCc12
CN(c1ccc(OCCCCCC(=O)NO)cc1)c1nc(C)nc2CCCc12
CN(c1cccc(OCC(=O)NO)c1)c1nc(C)nc2ccccc12
CN(c1cccc(OCCCC(=O)NO)c1)c1nc(C)nc2ccccc12
CN(c1cccc(OCCCCC(=O)NO)c1)c1nc(C)nc2ccccc12
CN(c1cccc(OCCCCCC(=O)NO)c1)c1nc(C)nc2ccccc12
COc1ccc(cc1OCC(=O)NO)N(C)c1nc(C)nc2ccccc12
COc1ccc(cc1OCCCC(=O)NO)N(C)c1nc(C)nc2ccccc12
COc1ccc(cc1OCCCCC(=O)NO)N(C)c1nc(C)nc2ccccc12
COc1ccc(cc1OCCCCCC(=O)NO)N(C)c1nc(C)nc2ccccc12
CN(c1ccc(OCC(=O)NO)cc1)c1nc(C)nc2ccccc12
CN(c1ccc(OCCCC(=O)NO)cc1)c1nc(C)nc2ccccc12
CN(c1ccc(OCCCCC(=O)NO)cc1)c1nc(C)nc2ccccc12
CN(c1ccc(OCCCCCC(=O)NO)cc1)c1nc(C)nc2ccccc12
FC(F)(F)C(=O)CCCCNC(=O)c1nc(sc1Cc1ccccc1)-c1nccs1
Cc1cnc(s1)-c1nc(C(=O)NCCCCC(=O)C(F)(F)F)c(s1)C1CC1
FC(F)(F)C(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1nc2CCCCc2s1
CC(C)Cc1sc(nc1C(=O)NCCCCC(=O)C(F)(F)F)-c1nccs1
FC(F)(F)C(=O)CCCCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
FC(F)(F)C(=O)CCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
FC(F)(F)C(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
OC(CCCCNC(=O)c1nc(sc1C1CC1)-c1nccs1)C(F)(F)F
FC(F)(F)c1nc(no1)-c1cccc(c1)C(=O)NCCCCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
ONC(=O)NCCCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
Nc1ccccc1NC(=O)CCCCNC(=O)c1nc(sc1C1CC1)-c1nccs1
ONC(=O)CCCc1csc(\C=C\c2ccccc2)n1
Cc1[nH]c2ccccc2c1\C=C\c1ccccc1-c1ccc(\C=C\C(=O)NO)cc1
ONC(=O)c1cccc(c1)N(Cc1ccccc1)Cc1ccccc1
ONC(=O)c1cccc(NC(=O)c2ccccc2)c1
Cc1ccc(cc1NC(=O)c2ccccc2)C(=O)NO
COc1ccc(cc1NC(=O)c2ccccc2)C(=O)NO
ONC(=O)c1ccc(F)c(NC(=O)c2ccccc2)c1
c1ccc(cc1)C(=O)Nc2cc(ccc2Cl)C(=O)NO
ONC(=O)c1ccc(Br)c(NC(=O)c2ccccc2)c1
ONC(=O)c1ccc(c(NC(=O)c2ccccc2)c1)C(F)(F)F
CCOc1ccc(cc1NC(=O)c1ccccc1)C(=O)NO
CC(C)Oc1ccc(cc1NC(=O)c1ccccc1)C(=O)NO
Cc1ccc(cc1NC(=O)c1ccc2ccccc2n1)C(=O)NO
COc1ccc(cc1NC(=O)c2ccc(cc2)c3ccccc3)C(=O)NO
COc1ccc(cc1)C(=O)Nc1cc(ccc1OC)C(=O)NO
COc1ccc(cc1NC(=O)c1ccc(Cl)cc1)C(=O)NO
COc1ccc(cc1NC(=O)c1ccccc1Cl)C(=O)NO
COc1ccc(cc1NC(=O)c2ccc(cc2Cl)Cl)C(=O)NO
CCOc1ccc(cc1)C(=O)Nc1cc(ccc1OC)C(=O)NO
COc1ccc(cc1NC(=O)Cc2ccccc2)C(=O)NO
COc1ccc(cc1)C(=O)Nc1cc(ccc1Cl)C(=O)NO
ONC(=O)c1ccc(Cl)c(NC(=O)c2cccc(OCc3ccccc3)c2)c1
ONC(=O)c1ccc(Cl)c(NC(=O)c2cccc(Oc3ccccc3)c2)c1
ONC(=O)c1ccc(Cl)c(NC(=O)c2ccc(Oc3ccccc3)cc2)c1
ONC(=O)c1ccc(Cl)c(NC(=O)c2ccc(Cl)cc2)c1
c1cc(c(cc1C(=O)NO)NC(=O)c2ccc(cc2Cl)Cl)Cl
CCOc1ccc(cc1NC(=O)c1ccc(cc1)-c1ccccc1)C(=O)NO
COc1ccc(cc1OCc1ccccc1)C(=O)NO
COc1ccc(cc1S(=O)(=O)Nc1ccc(C)cc1)C(=O)NO
C[C@@H]1C(=O)Nc2cc(ccc2S1)C(=O)NO
ONC(=O)c1ccc2SCCC(=O)Nc2c1
COc1ccc(cc1)-c1nc(N2CCOCC2)c2nc(CN(C)c3ncc(cn3)C(=O)NO)n(C)c2n1
CN(Cc1nc2c(nc(nc2n1C)-c1ccc(N)cc1)N1CCOCC1)c1ncc(cn1)C(=O)NO
CN(Cc1nc2c(nc(nc2n1C)-c1cnc(N)nc1)N1CCOCC1)c1ncc(cn1)C(=O)NO
COc1ccc(cn1)-c1nc(N2CCOCC2)c2nc(CN(C)c3ncc(cn3)C(=O)NO)n(C)c2n1
CN(Cc1nc2c(nc(nc2n1C)-c1ccncc1)N1CCOCC1)c1ncc(cn1)C(=O)NO
COc1ccc(cn1)-c1nc(N2CCOCC2)c2sc(CN(C)c3ncc(cn3)C(=O)NO)cc2n1
[H][C@]12CC[C@]([H])(C[C@H](C1)C(=O)Nc1cc(ccc1N)-c1ccc(F)cc1)O2 |r|
ONC(=O)CCCCCC(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12
COc1cccc2c(c[nH]c12)C(CCCCCC(=O)NO)c1c[nH]c2c(OC)cccc12
ONC(=O)CCCCCC(c1c[nH]c2ccc(cc12)[N+]([O-])=O)c1c[nH]c2ccc(cc12)[N+]([O-])=O
ONC(=O)\C=C\c1ccc(cc1)C(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12
CCOc1ccc(CC2CC(C2)C(=O)NO)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1 |(44.14,-3.5,;44.14,-5.04,;45.47,-5.81,;45.47,-7.35,;44.14,-8.12,;44.14,-9.66,;45.49,-10.43,;45.49,-11.97,;46.83,-12.74,;47.23,-14.22,;48.71,-13.81,;48.31,-12.33,;50.05,-14.58,;50.06,-16.12,;51.38,-13.8,;52.72,-14.56,;46.81,-9.66,;46.81,-8.12,;48.14,-7.35,;49.47,-8.11,;50.8,-7.34,;52.25,-7.82,;52.73,-9.28,;54.24,-9.6,;53.16,-6.58,;52.25,-5.34,;52.73,-3.87,;50.8,-5.81,;49.47,-5.03,;49.47,-3.49,;48.14,-5.81,)|
CCOc1ccc(cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1)C1CCC(CC(=O)NO)CC1 |(31.8,-34.85,;31.8,-36.39,;33.13,-37.16,;33.14,-38.7,;31.8,-39.47,;31.81,-41.01,;33.15,-41.78,;34.48,-41,;34.47,-39.47,;35.8,-38.7,;37.13,-39.46,;38.46,-38.69,;39.92,-39.16,;40.39,-40.63,;41.9,-40.95,;40.82,-37.92,;39.92,-36.68,;40.39,-35.22,;38.46,-37.16,;37.13,-36.38,;37.13,-34.84,;35.8,-37.16,;33.16,-43.32,;31.82,-44.08,;31.83,-45.62,;33.16,-46.39,;33.16,-47.93,;34.5,-48.7,;34.5,-50.24,;35.83,-47.92,;37.16,-48.69,;34.49,-45.61,;34.49,-44.07,)|
CCOc1ccc(CN2CCC(CC2)C(=O)NO)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)N1CCC2(C1)CCN(CC2)c1ncc(cn1)C(=O)NO
CCOc1ccc(CC2CCC(C2)C(=O)NO)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
CCOc1ccc(Oc2ccc(cc2)C(=O)NO)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
CCOc1ccc(CC2CC2C(=O)NO)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
CCOc1ccc(cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1)-c1ccc(cn1)C(=O)NO
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(NC2CCN(CC2)c2ccc(cc2)C(=O)NO)ccc1OCC
CCOc1ccc(CCC(=O)NO)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
CCOc1ccc(C[C@H]2C[C@@H](C2)C(=O)NO)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1 |r,wU:8.7,wD:10.12,(2.61,-17.39,;2.61,-18.93,;3.94,-19.7,;3.95,-21.24,;2.61,-22.01,;2.61,-23.56,;3.96,-24.32,;3.97,-25.86,;5.3,-26.63,;6.78,-26.22,;7.19,-27.71,;5.7,-28.11,;8.52,-28.47,;8.53,-30.01,;9.85,-27.69,;11.19,-28.46,;5.29,-23.55,;5.28,-22.01,;6.61,-21.24,;7.94,-22,;9.27,-21.23,;10.73,-21.71,;11.2,-23.17,;12.71,-23.49,;11.63,-20.47,;10.73,-19.23,;11.2,-17.76,;9.27,-19.7,;7.94,-18.92,;7.94,-17.38,;6.61,-19.7,)|
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)S(=O)(=O)N1CCN(CCCC(=O)NO)CC1
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)S(=O)(=O)N1CCN(Cc2ccc(\C=C\C(=O)NO)cc2)CC1
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(NCCC(=O)NO)ccc1OCC
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(NC2CCC(CC2)C(=O)NO)ccc1OCC |(28.99,-46.19,;28.51,-44.73,;27.01,-44.41,;26.53,-42.94,;27.43,-41.7,;26.53,-40.46,;27.01,-39,;25.07,-40.94,;25.07,-42.47,;23.75,-43.24,;22.42,-42.48,;22.42,-40.94,;23.75,-40.16,;23.75,-38.62,;21.09,-43.25,;21.09,-44.78,;19.76,-45.56,;19.77,-47.1,;21.11,-47.86,;21.1,-49.4,;22.43,-50.16,;23.77,-49.39,;23.76,-47.85,;22.43,-47.08,;25.1,-50.16,;25.11,-51.7,;26.44,-49.39,;27.77,-50.16,;18.42,-44.79,;18.42,-43.25,;19.75,-42.48,;19.75,-40.94,;18.42,-40.17,;18.41,-38.63,)|
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(NCC2CCN(CC2)c2ncc(cn2)C(=O)NO)ccc1OCC
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)N(C)C1CCN(CC1)c1ncc(cn1)C(=O)NO
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)N1CCC(CCC(=O)NO)CC1
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)N1CCC2(CCC(C2)C(=O)NO)CC1
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)N1CCCC2(CCC(CC2)C(=O)NO)C1 |(31.95,-30.68,;31.47,-29.21,;29.96,-28.89,;29.49,-27.43,;30.39,-26.19,;29.49,-24.94,;29.96,-23.48,;28.03,-25.42,;28.03,-26.95,;26.7,-27.72,;25.37,-26.96,;25.37,-25.42,;26.7,-24.64,;26.7,-23.1,;24.04,-27.73,;24.05,-29.26,;22.72,-30.04,;21.38,-29.27,;21.37,-27.73,;22.71,-26.96,;22.7,-25.42,;21.37,-24.65,;21.37,-23.11,;22.73,-31.58,;21.39,-32.35,;21.39,-33.88,;22.73,-34.65,;24.06,-33.88,;24.06,-35.42,;25.39,-36.19,;26.73,-35.42,;26.73,-33.88,;25.39,-33.1,;28.06,-36.19,;28.05,-37.73,;29.39,-35.43,;30.72,-36.2,;24.06,-32.33,)|
CCOc1ccc(OC2CCC(CC2)C(=O)NO)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1 |(53.45,-22.36,;53.45,-23.9,;54.78,-24.67,;54.78,-26.21,;53.45,-26.98,;53.45,-28.53,;54.8,-29.29,;54.8,-30.83,;56.14,-31.6,;56.14,-33.14,;57.47,-33.9,;58.8,-33.13,;58.8,-31.59,;57.46,-30.82,;60.14,-33.9,;60.14,-35.44,;61.47,-33.13,;62.8,-33.89,;56.12,-28.52,;56.12,-26.98,;57.45,-26.21,;58.78,-26.97,;60.11,-26.21,;61.57,-26.68,;62.04,-28.14,;63.55,-28.46,;62.47,-25.44,;61.57,-24.2,;62.04,-22.73,;60.11,-24.67,;58.78,-23.89,;58.78,-22.35,;57.45,-24.67,)|
CCOc1ccc(cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1)C(=O)NO
CCOc1ccc(Cc2ccc(CCC(=O)NO)cc2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
CCOc1ccc(CC2CCN(CC2)c2ncc(cn2)C(=O)NO)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
CCOc1ccc(CC2CCN(CC2)c2ccc(cn2)C(=O)NO)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
CCOc1ccc(CC2CCN(CC2)c2ccc(cc2)C(=O)NO)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
CCOc1ccc(CC2CCC(CC(=O)NO)CC2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1 |(50.87,-36.7,;50.87,-38.24,;52.21,-39.01,;52.21,-40.55,;50.88,-41.32,;50.88,-42.86,;52.22,-43.63,;52.23,-45.17,;53.57,-45.93,;53.56,-47.47,;54.89,-48.23,;56.23,-47.46,;57.56,-48.23,;58.89,-47.46,;58.89,-45.92,;60.22,-48.23,;61.56,-47.46,;56.22,-45.92,;54.89,-45.15,;53.55,-42.85,;53.54,-41.32,;54.87,-40.55,;56.2,-41.31,;57.53,-40.54,;58.99,-41.01,;59.47,-42.48,;60.97,-42.8,;59.89,-39.77,;58.99,-38.53,;59.47,-37.07,;57.53,-39.01,;56.2,-38.23,;56.2,-36.69,;54.87,-39.01,)|
CCOc1ccc(C[C@H]2CC[C@@H](CC2)C(=O)NO)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1 |r,wU:8.7,wD:11.14,(2.03,-1.64,;2.03,-3.18,;3.37,-3.95,;3.37,-5.49,;2.04,-6.26,;2.04,-7.81,;3.38,-8.57,;3.39,-10.11,;4.73,-10.88,;6.05,-10.09,;7.38,-10.87,;7.39,-12.41,;6.05,-13.18,;4.72,-12.42,;8.72,-13.18,;8.72,-14.72,;10.05,-12.41,;11.38,-13.18,;4.71,-7.8,;4.7,-6.26,;6.04,-5.49,;7.36,-6.25,;8.69,-5.48,;10.15,-5.96,;10.63,-7.42,;12.13,-7.74,;11.05,-4.72,;10.15,-3.48,;10.63,-2.01,;8.69,-3.95,;7.36,-3.17,;7.36,-1.63,;6.04,-3.95,)|
CCOc1ccc(C[C@H]2C[C@H](C2)C(=O)NO)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1 |r,wU:8.7,10.12,(57.87,-3.32,;57.87,-4.86,;59.21,-5.63,;59.21,-7.17,;57.88,-7.94,;57.88,-9.48,;59.22,-10.25,;59.23,-11.79,;60.57,-12.55,;62.04,-12.14,;62.45,-13.63,;60.96,-14.03,;63.79,-14.39,;63.79,-15.93,;65.12,-13.61,;66.45,-14.38,;60.55,-9.47,;60.54,-7.94,;61.87,-7.16,;63.2,-7.93,;64.53,-7.16,;65.99,-7.63,;66.47,-9.1,;67.97,-9.42,;66.89,-6.39,;65.99,-5.15,;66.47,-3.69,;64.53,-5.62,;63.2,-4.85,;63.2,-3.31,;61.87,-5.62,)|
CCOc1ccc(cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1)C1CC1C(=O)NO
CCOc1ccc(cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1)-c1ccc(nc1)C(=O)NO
CCOc1ccc(cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1)-c1ccc(o1)C(=O)NO
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)S(=O)(=O)N1CCC(CCC(=O)NO)CC1
CCOc1ccc(C[C@H]2CC[C@H](CC2)C(=O)NO)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1 |r,wU:8.7,11.14,(15.87,-1.64,;15.87,-3.18,;17.21,-3.95,;17.21,-5.49,;15.87,-6.26,;15.88,-7.81,;17.22,-8.57,;17.23,-10.11,;18.57,-10.88,;19.88,-10.09,;21.22,-10.87,;21.23,-12.41,;19.89,-13.18,;18.56,-12.42,;22.55,-13.18,;22.55,-14.72,;23.89,-12.41,;25.22,-13.18,;18.55,-7.8,;18.54,-6.26,;19.87,-5.49,;21.2,-6.25,;22.53,-5.48,;23.99,-5.96,;24.47,-7.42,;25.97,-7.74,;24.89,-4.72,;23.99,-3.48,;24.47,-2.01,;22.53,-3.95,;21.2,-3.17,;21.2,-1.63,;19.87,-3.95,)|
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)S(=O)(=O)Nc1ccc(\C=C\C(=O)NO)cc1
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)S(=O)(=O)N1CCN(CCC(=O)NO)CC1
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)S(=O)(=O)NC1CCN(CC1)c1ncc(cn1)C(=O)NO
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(NC2CCN(CC2)c2ncc(cn2)C(=O)NO)ccc1OCC
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)N1CCC(CC(=O)NO)CC1
CCOc1ccc(CC(=O)NO)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
CCOc1ccc(Cc2ccc(\C=C\C(=O)NO)cc2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
CCOc1ccc(CC2CCN(CCC(=O)NO)CC2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
CCOc1ccc(CN2CC(C2)C(=O)NO)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
CCOc1ccc(OC2CCN(CC2)c2ncc(cn2)C(=O)NO)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
CCOc1ccc(cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1)C1CC(C1)C(=O)NO |(3.28,-32.96,;3.28,-34.5,;4.61,-35.27,;4.61,-36.81,;3.28,-37.58,;3.28,-39.12,;4.63,-39.89,;5.95,-39.11,;5.95,-37.58,;7.28,-36.81,;8.61,-37.57,;9.94,-36.8,;11.4,-37.27,;11.87,-38.74,;13.38,-39.06,;12.3,-36.03,;11.4,-34.79,;11.87,-33.33,;9.94,-35.27,;8.61,-34.49,;8.61,-32.95,;7.28,-35.27,;4.64,-41.43,;3.55,-42.52,;4.65,-43.6,;5.73,-42.51,;4.66,-45.14,;3.33,-45.92,;5.99,-45.91,;7.32,-45.13,)|
CCOc1ccc(CN2CCN(CC2)c2ncc(cn2)C(=O)NO)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)S(=O)(=O)N1CCN(CC1)c1ncc(cn1)C(=O)NO
ONC(=O)CCCCCc1ccc2OCOc2c1
CC1(C)N(C(=S)N(C1=O)c1ccc(C#N)c(c1)C(F)(F)F)c1ccc(C(=O)NCCOCCC(=O)NO)c(F)c1
CC1(C)N(C(=S)N(C1=O)c1ccc(C#N)c(c1)C(F)(F)F)c1ccc(C(=O)NCCCCCCn2cccc(O)c2=S)c(F)c1
CC1(C)N(C(=S)N(C1=O)c1ccc(C#N)c(c1)C(F)(F)F)c1ccc(Cn2ccc3cc(\C=C\C(=O)NO)ccc23)c(F)c1
CC1(C)N(C(=S)N(C1=O)c1ccc(C#N)c(c1)C(F)(F)F)c1ccc(C(=O)Nc2ccccc2N)c(F)c1
CC1(C)N(C(=S)N(C1=O)c1ccc(C#N)c(c1)C(F)(F)F)c1ccc(C(=O)NCCCCCC(=O)NO)c(F)c1
CC1(C)N(C(=S)N(C1=O)c1ccc(C#N)c(c1)C(F)(F)F)c1ccc(C(=O)NCCCNS(N)(=O)=O)c(F)c1
CC1(C)N(C(=S)N(C1=O)c1ccc(C#N)c(c1)C(F)(F)F)c1ccc(C(=O)NCCCCCCNS(N)(=O)=O)c(F)c1
CC1(C)N(C(=S)N(C1=O)c1ccc(C#N)c(c1)C(F)(F)F)c1ccc(C(=O)NCCCn2cccc(O)c2=O)c(F)c1
CC1(C)N(C(=S)N(C1=O)c1ccc(C#N)c(c1)C(F)(F)F)c1ccc(C(=O)NCCCCCCC(=O)Nc2ccccc2N)c(F)c1
COC(=O)CCCCCCCc1ccc(cc1F)N1C(=S)N(C(=O)C1(C)C)c1ccc(C#N)c(c1)C(F)(F)F
CC1(C)N(C(=S)N(C1=O)c1ccc(C#N)c(c1)C(F)(F)F)c1ccc(\C=C\C(=O)Nc2ccccc2N)c(F)c1
CC1(C)N(C(=S)N(C1=O)c1ccc(C#N)c(c1)C(F)(F)F)c1ccc(C(=O)OCCCCCC(=O)NO)c(F)c1
CC1(C)N(C(=S)N(C1=O)c1ccc(C#N)c(c1)C(F)(F)F)c1ccc(C(=O)NCCCCCCn2cccc(O)c2=O)c(F)c1
CC1(C)N(C(=S)N(C1=O)c1ccc(C#N)c(c1)C(F)(F)F)c1ccc(C(=O)NCCCCCCc2ccc(s2)C(=O)C(F)(F)F)c(F)c1
ONC(=O)\C=C\c1cccc(c1)S(=O)(=O)c1ccc2ccccc2n1
ONC(=O)\C=C\c1cccc(c1)S(=O)(=O)c1ccc2cccc(F)c2n1
FC(F)(F)C(=O)c1cc(cs1)-c1ccccc1
COc1cccc(c1)-c1ccc(s1)C(=O)C(F)(F)F
COc1ccccc1-c1ccc(s1)C(=O)C(F)(F)F
COc1ccc(cc1)-c1ccc(s1)C(=O)C(F)(F)F
FC(F)(F)C(=O)c1ccc(s1)-c1ccccn1
FC(F)(F)C(=O)c1ccc(s1)-c1ccc2[nH]ccc2c1
OC(=O)c1cccc(c1)-c1ccc(s1)C(=O)C(F)(F)F
FC(F)(F)C(=O)c1ccc(s1)-c1ccccc1
FC(F)(F)C(=O)c1cnc(s1)-c1ccccc1
FC(F)(F)C(=O)c1ccc(s1)-c1ccc2nccnc2c1
OC(=O)c1ccc(cc1)-c1ccc(s1)C(=O)C(F)(F)F
CC(=O)c1ccc(cc1)-c1ccc(s1)C(=O)C(F)(F)F
FC(F)(F)C(=O)c1ccc(s1)-c1ccc2OCCOc2c1
FC(F)(F)C(=O)c1ccc(s1)-c1ccc(cc1)C#N
ONC(=O)CCCCCCn1cc(nn1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
Cc1ccc(Oc2ccc(Nc3ncnc4ccc(cc34)-c3cn(CCCCCCC(=O)NO)nn3)cc2C)cn1
ONC(=O)CCCCCn1cc(nn1)-c1ccc2ncnc(Nc3cccc(Cl)c3F)c2c1
ONC(=O)CCCCCn1cc(nn1)-c1ccc2ncnc(Nc3ccc(OCc4nccs4)c(Cl)c3)c2c1
ONC(=O)CCCCCCn1cc(nn1)-c1ccc2ncnc(Nc3ccc(OCc4nccs4)c(Cl)c3)c2c1
ONC(=O)CCCCCn1cc(nn1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
ONC(=O)CCCCCn1cc(nn1)-c1ccc2ncnc(Nc3ccc(F)c(Cl)c3)c2c1
ONC(=O)CCCCCCn1cc(nn1)-c1ccc2ncnc(Nc3cccc(Cl)c3F)c2c1
ONC(=O)CCCCCCn1cc(nn1)-c1ccc2ncnc(Nc3ccc(F)c(Cl)c3)c2c1
Cc1ccc(Oc2ccc(Nc3ncnc4ccc(cc34)-c3cn(CCCCCC(=O)NO)nn3)cc2C)cn1
COc1cc(Nc2ncnc3ccc(cc23)-c2cn(CCCCCCC(=O)NO)nn2)ccc1Oc1ccccc1
COc1cc(Nc2ncnc3ccc(cc23)-c2cn(CCCCCC(=O)NO)nn2)ccc1Oc1ccccc1
ONC(=O)c1cnc(nc1)N1CCN(CC1)S(=O)(=O)c1ccc2ccccc2c1
OCC(\C=C\c1ccc(F)cc1)N1CCN(CC1)c1ncc(cn1)C(=O)NO
COc1ccc2n(C(=O)c3ccc(Cl)cc3)c(C)c(CC(=O)NCCCCCCC(=O)NO)c2c1
COC(=O)Cc1c(C)n(Cc2ccc(cc2)-c2cn(CCCCCCC(=O)NO)nn2)c2ccc(OC)cc12
Cc1ccc(cc1)-c1cc(nn1-c1ccc(cc1)S(N)(=O)=O)C(=O)NCCCCCCCC(=O)NO
Cc1ccc(cc1)-c1cc(nn1-c1ccc(cc1)S(=O)(=O)NCCCCCCC(=O)NO)C(F)(F)F
Cc1ccc(cc1)-c1cc(nn1-c1ccc(cc1)S(N)(=O)=O)C(=O)NCCCCCCC(=O)NO
Cc1ccc(cc1)-c1cc(nn1-c1ccc(cc1)S(=O)(=O)NCCCCCC(=O)NO)C(F)(F)F
COC(=O)Cc1c(C)n(Cc2ccc(cc2)-c2cn(CCCCCCCC(=O)NO)nn2)c2ccc(OC)cc12
Cc1ccc(cc1)-c1cc(nn1-c1ccc(cc1)S(=O)(=O)NCCCCCCCC(=O)NO)C(F)(F)F
Cc1ccc(cc1)-c1cc(nn1-c1ccc(cc1)S(N)(=O)=O)C(=O)NCCCCCC(=O)NO
COc1ccc2n(C(=O)c3ccc(Cl)cc3)c(C)c(CC(=O)NCCCCCC(=O)NO)c2c1
COC(=O)Cc1c(C)n(Cc2ccc(cc2)-c2cn(CCCCCC(=O)NO)nn2)c2ccc(OC)cc12
COc1ccc2n(C(=O)c3ccc(Cl)cc3)c(C)c(CC(=O)NCCCCCCCC(=O)NO)c2c1
COc1ccc2n(Cc3ccc(cc3)-c3cn(CCCCCCC(=O)NO)nn3)c(C)c(CC(O)=O)c2c1
Cc1ccc(cc1)-c1cc(nn1-c1ccc(cc1)S(C)(=O)=O)C(=O)NCCCCCCC(=O)NO
COc1cc2ncnc(Nc3cccc(c3)C#C)c2cc1OCCCCCCC(=O)NO
OC(=O)c1cccc(NCCOc2ccc3Nc4nccc(n4)-c4cccc(COC\C=C\COCc2c3)c4)c1 |t:32|
OC(=O)CCCCCOc1ccc2Nc3nccc(n3)-c3cccc(COC\C=C\COCc1c2)c3 |t:29|
OC(=O)CCCCCCCOc1ccc2Nc3nccc(n3)-c3cccc(COC\C=C\COCc1c2)c3 |t:31|
ONC(=O)CCCCCCC(=O)Nc1ccc(NCCOc2ccc3Nc4nccc(n4)-c4cccc(COC\C=C\COCc2c3)c4)cc1 |t:41|
OC(=O)c1ccc(NCCOc2ccc3Nc4nccc(n4)-c4cccc(COC\C=C\COCc2c3)c4)cc1 |t:31|
ONC(=O)CCCOc1ccc2Nc3nccc(n3)-c3cccc(COC\C=C\COCc1c2)c3 |t:28|
ONC(=O)c1ccc(OCCOc2ccc3Nc4nccc(n4)-c4cccc(COC\C=C\COCc2c3)c4)cc1 |t:32|
ONC(=O)c1ccc(NCCOc2ccc3Nc4nccc(n4)-c4cccc(COC\C=C\COCc2c3)c4)cc1 |t:32|
ONC(=O)C1CCN(CCOc2ccc3Nc4nccc(n4)-c4cccc(COC\C=C\COCc2c3)c4)CC1 |t:31|
OC(=O)CCCCCCOc1ccc2Nc3nccc(n3)-c3cccc(COC\C=C\COCc1c2)c3 |t:30|
OC(=O)C1CCN(CCOc2ccc3Nc4nccc(n4)-c4cccc(COC\C=C\COCc2c3)c4)CC1 |t:30|
OC(=O)c1ccc(OCCOc2ccc3Nc4nccc(n4)-c4cccc(COC\C=C\COCc2c3)c4)cc1 |t:31|
OC(=O)CCCCCCC(=O)Nc1ccc(NCCOc2ccc3Nc4nccc(n4)-c4cccc(COC\C=C\COCc2c3)c4)cc1 |t:40|
ONC(=O)c1cccc(NCCOc2ccc3Nc4nccc(n4)-c4cccc(COC\C=C\COCc2c3)c4)c1 |t:33|
ONC(=O)CCCCCOc1ccc2Nc3nccc(n3)-c3cccc(COC\C=C\COCc1c2)c3 |t:30|
ONC(=O)CCCCOc1ccc2Nc3nccc(n3)-c3cccc(COC\C=C\COCc1c2)c3 |t:29|
ONC(=O)CCCCCCCOc1ccc2Nc3nccc(n3)-c3cccc(COC\C=C\COCc1c2)c3 |t:32|
ONC(=O)CCCCCCOc1ccc2Nc3nccc(n3)-c3cccc(COC\C=C\COCc1c2)c3 |t:31|
ONC(=O)CCCCCC(=O)Nc1ccc(NCCOc2ccc3Nc4nccc(n4)-c4cccc(COC\C=C\COCc2c3)c4)cc1 |t:40|
CCCCCCC(CCCCCC(=O)Nc1ccccc1)C(=O)NO
ONC(=O)C(CCCCCC(=O)Nc1ccccc1)Cc1ccccc1
CCCCCC(CCCCCC(=O)Nc1ccccc1)C(=O)NO
ONC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCN2C(=O)[C@@H]2CCCCCCCCC[C@@H](NC1=O)C(=O)N2 |r|
ONC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCN2C(=O)[C@@H]2CCCCCCCCCCC[C@@H](NC1=O)C(=O)N2 |r|
ONC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCN2C(=O)[C@@H]2CCCCCCCCCCCC[C@@H](NC1=O)C(=O)N2 |r|
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(nn1)-c1cc(F)cc(F)c1
Nc1ccc(cc1)-n1cc(nn1)-c1cccc(NC(=O)CCCCCCC(=O)NO)c1
COc1cc(ccc1F)-n1cc(nn1)-c1cccc(NC(=O)CCCCCCC(=O)NO)c1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(Cc2ccc(O)cc2)nn1
Nc1ccccc1NC(=O)CCCCCCC(=O)Nc1cccc(c1)-n1cc(nn1)-c1ccccc1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(nn1)-c1ccc(cc1)C(F)(F)F
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(nn1)C1CCCCC1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-n1cc(nn1)-c1ccccc1
OCc1cc(CO)cc(c1)-n1cc(nn1)-c1cccc(NC(=O)CCCCCCC(=O)NO)c1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(nn1)-c1ccc(I)cc1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-n1cc(nn1)C1CCCCC1
ONC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(nn1)-c1ccc(F)cc1
CC(C)(C)c1[nH]c2ccccc2c1[C@H]1CCCN(Cc2ccc(\C=C\C(=O)NO)cc2F)C1 |r|
CC(C)(C)c1[nH]c2ccccc2c1[C@@H]1CCCN(Cc2ccc(\C=C\C(=O)NO)cc2F)C1 |r|
C[C@H](O)C(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
OC(=O)CCC=CC[C@@H]1NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r,w:6.6|
ONC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
ONC(=O)CCCCC[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
ONC(=O)CCCCCNC(=O)NC(=O)c1ccccc1
Nc1ccc(cc1NC(=O)c1ccc(cc1)\N=C\C=N)-c1cccs1
COc1ccc(cc1)C(=O)Nc1cc(ccc1N)-c1cccs1
CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCC(=O)NO)nn2)[C@@](C)(C[C@@H](C)C2=NCCN3[C@H]([C@H]2C)[C@]1(C)OC3=O)OC |r,t:53|
CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCC(=O)NO)nn2)[C@@](C)(C[C@@H](C)C2=NCCN3[C@H]([C@H]2C)[C@]1(C)OC3=O)OC |r,t:54|
CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCCC(=O)NO)nn2)[C@@](C)(C[C@@H](C)C2=NCCN3[C@H]([C@H]2C)[C@]1(C)OC3=O)OC |r,t:55|
CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCCCC(=O)NO)nn2)[C@@](C)(C[C@@H](C)C2=NCCN3[C@H]([C@H]2C)[C@]1(C)OC3=O)OC |r,t:56|
CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCCCCC(=O)NO)nn2)[C@@](C)(C[C@@H](C)C2=NCCN3[C@H]([C@H]2C)[C@]1(C)OC3=O)OC |r,t:57|
ONC(=O)c1cc(CCCCC(=O)Nc2ccccc2)on1
ONC(=O)C1=NOC(CCCCC(=O)Nc2ccccc2)C1 |t:4|
ONC(=O)CCCCCN1C(=O)c2cccc3cccc(C1=O)c23
[#6]-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#6](=O)-[#7]-c1ccccc1-[#7])-[#6@H]1-[#6]-[#6]-[#6@H]2\[#6](-[#6]-[#6]-[#6][C@]12[#6])=[#6]\[#6]=[#6]-1/[#6]-[#6@@H](-[#8])-[#6]-[#6@H](-[#8])-[#6]-1 |r|
CC(C)(C)OC(=O)N[C@@H](CCCCCO)C(=O)NC1CCCC1 |r|
CC(C)(C)OC(=O)N[C@@H](CCCCCC(=O)NO)C(=O)NC1CCCC1 |r|
ONC(=O)CCCCC[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)Nc1cccc2cccnc12 |r|
CN(C)c1ccc(cc1)C(=O)N[C@@H](CCCCCC(=O)NO)C(=O)Nc1cccc2cccnc12 |r|
Nc1ccccc1NC(=O)c1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
Nc1ccccc1NC(=O)c1ccc(s1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
Nc1ccccc1NC(=O)\C=C\c1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
Nc1ccccc1NC(=O)\C=C\c1cccc(c1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
Nc1ccccc1NC(=O)\C=C\c1ccc(cc1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
Nc1ccccc1NC(=O)CCc1ccc(cc1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
CS(=O)(=O)CCNCc1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
ONC(=O)\C=C\c1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
ONC(=O)\C=C\c1ccc(s1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
ONC(=O)\C=C\c1cccc(c1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
ONC(=O)\C=C\c1ccc(cc1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
ONC(=O)c1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
ONC(=O)c1ccc(s1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
COc1ccc(COC(CCCCCC(=O)NO)C(=O)Nc2ccccc2)cc1 |w:8.8|
ONC(=O)CCCCCC1OCCCCCOc2ccccc2NC1=O
ONC(=O)CCCCCC1OCCCCCCOc2ccccc2NC1=O
ONC(=O)CCCCCC1OCCCCCCCOc2ccccc2NC1=O
COc1cc2COc3ccccc3NC(=O)C(CCCCCC(=O)NO)OC\C=C/c(c2)c1 |c:29|
COc1cc2COc3ccccc3NC(=O)[C@H](CCCCCC(=O)NO)OC\C=C/c(c2)c1 |r,c:29|
COc1cc2COc3ccccc3NC(=O)[C@@H](CCCCCC(=O)NO)OC\C=C/c(c2)c1 |r,c:29|
COc1cc2CCCOC(CCCCCC(=O)NO)C(=O)Nc3ccccc3OCc(c2)c1
COc1cc2CCCO[C@@H](CCCCCC(=O)NO)C(=O)Nc3ccccc3OCc(c2)c1 |r|
COc1cc2CCCO[C@H](CCCCCC(=O)NO)C(=O)Nc3ccccc3OCc(c2)c1 |r|
ONC(=O)CCC1=CCN(CCCc2ccc3ccccc3c2)C1=O |t:6|
CNC(=O)C(CCCCCCC(=O)Nc1ccccc1)N=O
CNC(=O)C(CCCCCCC(=O)Nc1ccc2ccccc2c1)N=O
CNC(=O)C(CCCCCCC(=O)Nc1cnc2ccccc2c1)N=O
CNC(=O)C(CCCCCCC(=O)NC1c2ccccc2-c2ccccc12)N=O
CNC(=O)C(CCCCCCC(=O)Nc1ccc(cc1)N(C)C)N=O
CNC(=O)C(CCCCCCC(=O)Nc1ccc(cc1)-c1ccccc1)N=O
CNC(=O)C(CCCCCCC(=O)Nc1cccc(Br)c1)N=O
CNC(=O)C(CCCCCCC(=O)Nc1cccc(c1)-c1ccccc1)N=O
CNC(=O)C(CCCCCCC(=O)Nc1cccc(c1)-c1ccc(cc1)C(O)=O)N=O
CNC(=O)C(CCCCCCC(=O)Nc1cccc(c1)-c1cccnc1)N=O
CNC(=O)C(CCCCCCC(=O)Nc1cccc(c1)-c1ccc(Cl)nc1)N=O
CNC(=O)C(CCCCCCC(=O)Nc1cccc(c1)-c1cncc2cc(Cl)ccc12)N=O
CNC(=O)C(CCCCCCNC(=O)c1cc(on1)-c1cccc(NC(=O)OC(C)(C)C)c1)N=O
CNC(=O)C(CCCCCCNC(=O)c1cc(on1)-c1ccc(NC(=O)OC(C)(C)C)cc1)N=O
CNC(=O)C(CCCCCCNC(=O)c1cc(on1)-c1cccc(N)c1)N=O
CNC(=O)C(CCCCCCNC(=O)c1cc(on1)-c1ccc(N)cc1)N=O
CNC(=O)C(CCCCC[C@H](N(Cc1ccc(OC)cc1)C(=O)OC(C)(C)C)C(=O)Nc1ccccc1)N=O |r|
CNC(=O)C(CCCCC[C@H](NCc1ccc(OC)cc1)C(=O)Nc1ccccc1)N=O |r|
CNC(=O)C(CCCCC[C@H](N(Cc1ccccc1)Cc1ccccc1)C(=O)Nc1ccccc1)N=O |r|
CC[C@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1 |r|
CC[C@H](C)[C@@H](CN1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1)NC(=O)OC(C)(C)C |r|
CC[C@H](C)[C@H](NC(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1 |r|
CC[C@H](C)[C@@H](CN1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1)NC(=O)CC(C)(C)C |r|
CC[C@H](C)[C@H](NC(=O)[C@@H](N)C(C)C)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1 |r|
CC[C@H](C)[C@H](NC(=O)C1CCN(CC1)C(=O)OC(C)(C)C)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1 |r|
CC[C@H](C)[C@H](NC(=O)C1CCNCC1)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1 |r|
CC[C@H](C)[C@H](NC(=O)[C@@H]1CCCN1)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1 |r|
ONC(=O)c1cnc(nc1)N1C[C@H]2[C@@H](C1)[C@@H]2NCc1ccc2cc(F)ccc2n1 |r|
ONC(=O)c1cnc(nc1)N1C[C@H]2[C@@H](C1)[C@@H]2NCc1ccc(Cl)cc1 |r|
CC(=O)Nc1ccc(cc1)C(=O)CSc1nc(C)cc(=O)[nH]1
CC(=O)Nc1ccc(cc1)C(=O)CSc1nccc(C)n1
COc1cc(C)nc(SCC(=O)c2ccc(NC(C)=O)cc2)n1
CC(=O)Nc1ccc(cc1)C(=O)CSc1nc(C)cc(C)n1
CC(=O)Nc1ccc(cc1)C(=O)CSc1cccc(O)c1
CC(=O)Nc1ccc(cc1)C(=O)COc1nc(C)cc(=O)[nH]1
CC(=O)Nc1ccc(cc1)C(=O)COc1cc(C)cc(=O)[nH]1
CC(=O)Nc1ccc(CSc2nc(C)cc(=O)[nH]2)cc1
CC(=O)Nc1ccc(cc1)C(O)CSc1nc(C)cc(=O)[nH]1
Cc1cc(=O)[nH]c(SCC(=O)c2ccccc2)n1
CN(C(C)=O)c1ccc(cc1)C(=O)CSc1nc(C)cc(=O)[nH]1
Cc1cc(=O)[nH]c(SCC(=O)c2ccc(NC(=O)c3ccccc3)cc2)n1
COc1ccc(cc1)C(=O)CSc1nc(C)cc(=O)[nH]1
Cc1cc(=O)[nH]c(SCC(=O)c2ccc(cc2)C(C)(C)C)n1
Cc1cc(=O)[nH]c(SCC(=O)c2ccc(Cl)cc2)n1
Cc1cc(=O)[nH]c(SCC(=O)c2ccc(O)cc2)n1
Cc1cc(=O)[nH]c(SCC(=O)c2ccc(O)c(O)c2)n1
Cc1cc(=O)[nH]c(SCC(=O)c2ccc3OCCOc3c2)n1
Cc1cc(=O)[nH]c(SCC(=O)c2ccc3CC(=O)Nc3c2)n1
Cc1cc(=O)[nH]c(SCC(=O)c2cccs2)n1
COC(=O)CSc1nc(C)cc(=O)[nH]1
CC(=O)CSc1nc(C)cc(=O)[nH]1
Cc1cc(=O)[nH]c(SCC(=O)C(C)(C)C)n1
CCOC(=O)CC(=O)CSc1nc(C)cc(=O)[nH]1
Cc1cc(=O)[nH]c(SCC(=O)NCCCCc2ccccc2)n1
Cc1cc(=O)[nH]c(SCC(=O)NCCc2ccccc2)n1
Cc1cc(=O)[nH]c(SCC(=O)NCCCCCCc2ccccc2)n1
ONC(=O)\C=C\C=C\c1ccc2OCOc2c1
ONC(=O)\C=C\C=C\CC\C=C\c1ccc2OCOc2c1
ONC(=O)\C=C\C=C\CCCCc1ccc2OCOc2c1
c1cc(cc(c1)Cl)C[C@H](C(=O)N2CCN(CC2)C(=O)c3cc(ccc3F)F)N
c1ccc2c(c1)CN(C2)C(=O)[C@@H](Cc3ccc(cc3Cl)Cl)N
CC(C)CCc1c(O)c(CCC(=O)NO)ccc1OCCCCCCC(=O)NO
CC(C)CCc1c(O)c(CCC(=O)NO)ccc1OCCCCCCCC(=O)NO
CC(C)CCc1c(OCCCCCCC(=O)NO)ccc2ccc(=O)oc12
CC(C)CCc1c(OCCCCCCC(=O)NO)ccc2CCC(=O)Oc12
CN(C)CC(C)(C)Cn1c(CCc2ccccc2)nc2cc(\C=C\C(=O)NO)ccc12
ONC(=O)\C=C\c1ccc2n(CCN3CCCCC3)c(CCc3ccccc3)nc2c1
CCCCc1nc2cc(C=CC(=O)NO)ccc2n1CCN(CC)CC
CCCCc1nc2cc(\C=C\C(=O)NO)ccc2n1CCNC(C)C
CN(C)CC(C)(C)Cn1c(CC(C)(C)C)nc2cc(\C=C\C(=O)NO)ccc12
CCCCCCc1nc2cc(\C=C\C(=O)NO)ccc2n1CCNCC
CCCCCCc1nc2cc(\C=C\C(=O)NO)ccc2n1CCNC(C)C
CCCCCCc1nc2cc(\C=C\C(=O)NO)ccc2n1CCN(C)C
CCNCCn1c(CC\C=C/CC)nc2cc(\C=C\C(=O)NO)ccc12
CCCCCc1nc2cc(\C=C\C(=O)NO)ccc2n1CCNC(C)C
CC[C@H](C)[C@H](NC(=O)CC(C)(C)C)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1 |r|
CCCC[C@H]1NC(=O)C[C@@H]2OC(=O)C[C@H](O)[C@H](NC(=O)[C@@H](CSSCC\C=C\2)NC1=O)[C@@H](C)CC |r,t:26|
CCCC[C@H]1NC(=O)C[C@H](OC(=O)C[C@H](O)[C@H](NC(=O)[C@@H](CS)NC1=O)[C@@H](C)CC)\C=C\CCS |r|
C\C=C1\NC(=O)[C@@H](CS)NC(=O)[C@H](NC(=O)C[C@H](OC(=O)[C@@H](NC1=O)C(C)C)\C=C\CCS)C(C)C |r|
CC[C@H](C)[C@H]1NC(=O)[C@H]2CSSCC\C=C\[C@H](CC(=O)N[C@H](CCSC)C(=O)N2)OC(=O)C[C@@H]1O |r,t:14|
CC[C@H](C)[C@H]1NC(=O)[C@@H](CS)NC(=O)[C@@H](CCSC)NC(=O)C[C@H](OC(=O)C[C@@H]1O)\C=C\CCS |r|
CCC(CCCCC(=O)Nc1ccccc1)CC(=O)NO
CN1CCc2c(C1)c1ccccc1n2S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1
CN1CCc2c(C1)c1ccccc1n2Cc1ccc(\C=C\C(=O)NO)cc1
CN(C)Cc1c(C)n(Cc2ccc(cc2)C(=O)NO)c2ccccc12
CN(C)Cc1c(C)n(c2ccccc12)S(=O)(=O)c1ccc(\C=C\C(=O)NO)cc1
CN(C)Cc1c(C)n(Cc2ccc(\C=C\C(=O)NO)cc2)c2ccccc12
CN(C)Cc1cn(c2ccccc12)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1
CN(C)Cc1cn(c2ccccc12)S(=O)(=O)c1ccc(\C=C\C(=O)NO)cc1
CN(C)Cc1cn(Cc2ccc(\C=C\C(=O)NO)cc2)c2ccccc12
CN(C)C(=O)c1cn(c2ccccc12)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1
CN(C)C(=O)c1cn(c2ccccc12)S(=O)(=O)c1ccc(\C=C\C(=O)NO)cc1
CN(C)C(=O)c1cn(Cc2ccc(\C=C\C(=O)NO)cc2)c2ccccc12
CN(C)Cc1c(C)n(c2ccccc12)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1
CN(C)Cc1cn(c2c1cccc2)Cc3ccc(cc3)C(=O)NO
CN(C)C(=O)c1cn(Cc2ccc(cc2)C(=O)NO)c2ccccc12
CC(C)(C)OC(=O)CC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:10|
CC(C)(C)OC(=O)CC[C@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:10|
Cc1c2OC(C)(C)Cc2c(C)c(c1C)S(=O)(=O)NC(=N)NCCC[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:27|
Cc1c2OC(C)(C)Cc2c(C)c(c1C)S(=O)(=O)NC(=N)NCCC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:27|
ONC(=O)CCCNC(=O)CC[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:13|
NC(=O)CC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:6|
CC(C)(C)OC(=O)C[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:9|
OC(=O)CC[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:6|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](C)C1=O)c1ccccc1 |r,c:16|
C[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:2|
CC(C)(C)OC(=O)NCCCC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:13|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](CC(=O)OC(C)(C)C)C1=O)c1ccccc1 |r,c:16|
C[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |t:2|
CC(C)C[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:5|
CC(C)(C)OC(=O)CC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:10|
CSCC[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:5|
ONC(=O)CC[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:7|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](CC(=O)NO)C1=O)c1ccccc1 |r,c:16|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2cc3ccccc3n2C(=O)OC(C)(C)C)C1=O)c1ccccc1 |r,c:16|
COC(=O)CCCCN1c2ccccc2C(=N[C@H](CSC(C)(C)C)C1=O)c1ccccc1 |r,c:16|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCC(=O)OC(C)(C)C)C1=O)c1ccccc1 |r,c:16|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](CC(=O)NC(c2ccccc2)(c2ccccc2)c2ccccc2)C1=O)c1ccccc1 |r,c:16|
CC(C)(C)OC(=O)NCCCC[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:13|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2ccc(O)cc2)C1=O)c1ccccc1 |r,c:16|
CC(C)(C)Oc1ccc(C[C@@H]2N=C(c3ccccc3)c3ccccc3NC2=O)cc1 |r,t:11|
OC(=O)CCCCN1c2ccccc2C(=NCC1=O)c1ccccc1 |c:15|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCC(O)=O)C1=O)c1ccccc1 |r,c:16|
[H][C@]1(N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O)[C@@H](C)O |r,t:2|
O=C1CN=C(c2ccccc2)c2ccccc2N1 |t:3|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2ccccc2)C1=O)c1ccccc1 |r,c:16|
Cc1c2OC(C)(C)Cc2c(C)c(c1C)S(=O)(=O)NC(=N)NCCC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:27|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2cc3ccccc3[nH]2)C1=O)c1ccccc1 |r,c:16|
CC(C)(C)OC(=O)C[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:9|
NCCCC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:6|
O=C(C[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O)NC(c1ccccc1)(c1ccccc1)c1ccccc1 |r,t:4|
ONC(=O)CCCCN1c2ccccc2C(=NCC1=O)c1ccccc1 |c:16|
[H][C@]1(N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O)[C@H](C)OCc1ccccc1 |r,t:2|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](CC(=O)NC(c2ccccc2)(c2ccccc2)c2ccccc2)C1=O)c1ccccc1 |r,c:16|
CC(C)(C)OC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:7|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2cncn2C(c2ccccc2)(c2ccccc2)c2ccccc2)C1=O)c1ccccc1 |r,c:16|
CC(C)C[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:5|
CC(C)(C)Oc1ccc(C[C@@H]2N=C(c3ccccc3)c3ccccc3N(CCCCC(=O)NO)C2=O)cc1 |r,t:11|
O=C(CC[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O)NC(c1ccccc1)(c1ccccc1)c1ccccc1 |r,t:5|
ONC(=O)C[C@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:6|
CC(C)(C)OC(=O)n1cc(C[C@@H]2N=C(c3ccccc3)c3ccccc3NC2=O)c2ccccc12 |r,t:12|
CSCC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:5|
OC(=O)C[C@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:5|
OC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2cncn2C(c2ccccc2)(c2ccccc2)c2ccccc2)C1=O)c1ccccc1 |r,c:15|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](CC(C)C)C1=O)c1ccccc1 |r,c:16|
CC(C)(C)OC(=O)n1c(C[C@@H]2N=C(c3ccccc3)c3ccccc3N(CCCCC(O)=O)C2=O)cc2ccccc12 |r,t:11|
C[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:2|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2cncn2C(c2ccccc2)(c2ccccc2)c2ccccc2)C1=O)c1ccccc1 |r,c:16|
OC(=O)C[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:5|
OC(=O)CCCCN1c2ccccc2C(=N[C@@H](CC(=O)NC(c2ccccc2)(c2ccccc2)c2ccccc2)C1=O)c1ccccc1 |r,c:15|
CC(C)(C)OC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:7|
CC(C)C[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:5|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCSC)C1=O)c1ccccc1 |r,c:16|
[H][C@]1(N=C(c2ccccc2)c2ccccc2NC1=O)[C@H](C)OCc1ccccc1 |r,t:2|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2ccccc2)C1=O)c1ccccc1 |r,c:16|
CC(C)[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:4|
NC(=O)C[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:5|
COC(=O)CCCCN1c2ccccc2C(=NCC1=O)c1ccccc1 |c:16|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2cnc[nH]2)C1=O)c1ccccc1 |r,c:16|
CC(C)(C)SC[C@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:7|
NC(=N)NCCC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:8|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCC(=O)NC(c2ccccc2)(c2ccccc2)c2ccccc2)C1=O)c1ccccc1 |r,c:16|
CC(C)(C)Oc1ccc(C[C@@H]2N=C(c3ccccc3)c3ccccc3N(CCCCC(O)=O)C2=O)cc1 |r,t:11|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCCCNC(=O)OC(C)(C)C)C1=O)c1ccccc1 |r,c:16|
OC(=O)CCCCN1c2ccccc2C(=N[C@@H](CC(O)=O)C1=O)c1ccccc1 |r,c:15|
CC(C)(C)SC[C@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:7|
[H][C@]1(N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O)[C@@H](C)OCc1ccccc1 |r,t:2|
OC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O |r,t:3|
OC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2ccccc2)C1=O)c1ccccc1 |r,c:15|
[H][C@]1(N=C(c2ccccc2)c2ccccc2NC1=O)[C@@H](C)CC |r,t:2|
CC(C)(C)OC(=O)NCCCC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:13|
O=C1Nc2ccccc2C(=N[C@H]1Cc1cn(cn1)C(c1ccccc1)(c1ccccc1)c1ccccc1)c1ccccc1 |r,c:10|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](CC(O)=O)C1=O)c1ccccc1 |r,c:16|
CC(C)(C)OC(=O)C[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:9|
OC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCC(=O)NC(c2ccccc2)(c2ccccc2)c2ccccc2)C1=O)c1ccccc1 |r,c:15|
OC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCC(O)=O)C1=O)c1ccccc1 |r,c:15|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCC(=O)NC(c2ccccc2)(c2ccccc2)c2ccccc2)C1=O)c1ccccc1 |r,c:16|
CC(C)(C)OC[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:7|
CC(C)[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:4|
CC(C)(C)OC(=O)n1c(C[C@@H]2N=C(c3ccccc3)c3ccccc3N(CCCCC(=O)NO)C2=O)cc2ccccc12 |r,t:11|
ONC(=O)CCCCN1c2ccccc2C(=N[C@H](CS)C1=O)c1ccccc1 |r,c:16|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCCNC(=N)NS(=O)(=O)c2c(C)c3CC(C)(C)Oc3c(C)c2C)C1=O)c1ccccc1 |r,c:16|
ONC(=O)CCCCN1c2ccccc2C(=N[C@@H](CCC(=O)NO)C1=O)c1ccccc1 |r,c:16|
CSCC[C@@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:5|
[H][C@]1(N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)OC)C1=O)[C@@H](C)OCc1ccccc1 |r,t:2|
CC(C)(C)SC[C@H]1N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O |r,t:7|
[H][C@]1(N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)NO)C1=O)[C@H](C)CC |r,t:2|
CC(C)(C)OC(=O)CC[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:10|
CC(C)[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:4|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](C(C)C)C1=O)c1ccccc1 |r,c:16|
[H][C@]1(N=C(c2ccccc2)c2ccccc2N(CCCCC(O)=O)C1=O)[C@@H](C)CC |r,t:2|
[H][C@]1(N=C(c2ccccc2)c2ccccc2N(CCCCC(=O)OC)C1=O)[C@@H](C)CC |r,t:2|
ONC(=O)CCCNC(=O)C[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:12|
OC(=O)CC[C@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:6|
CC(C)(C)OC(=O)C[C@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:9|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](Cc2ccc(OC(C)(C)C)cc2)C1=O)c1ccccc1 |r,c:16|
COC(=O)CCCCN1c2ccccc2C(=N[C@@H](COC(C)(C)C)C1=O)c1ccccc1 |r,c:16|
ONC(=O)CC[C@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:7|
O=C1Nc2ccccc2C(=N[C@H]1Cc1ccccc1)c1ccccc1 |r,c:10|
ONC(=O)C[C@@H]1N=C(c2ccccc2)c2ccccc2NC1=O |r,t:6|
SCC(=O)NCCCCCCn1ccc2cc(Cl)c(Cl)cc12
SCC(=O)NCCCCCCn1cc(Cl)c2cc(Cl)c(Cl)cc12
Fc1cc2ccn(CCCCCCNC(=O)CS)c2cc1Cl
c1cn(c2c1cc(c(c2)Cl)Cl)CCCCCNC(=O)CS
SCC(=O)NCCCCCNc1c(Cl)cc(Cl)c2cccnc12
SCC(=O)NCCCCCOc1c(Cl)cc(Cl)c2cccnc12
SCC(=O)NCC(S)CCCn1ccc2cc(Cl)c(Cl)cc12
CC(C)c1cn(CCCCCCNC(=O)CS)c2cc(Cl)c(Cl)cc12
SCC(=O)NCCCCNc1c(Cl)cc(Cl)c2cccnc12
ONC(=O)CCCCCCNC(=O)c1cc(on1)-c1ccc(NC(=O)c2cc(CN=[N+]=[N-])cc(c2)N=[N+]=[N-])cc1
ONC(=O)CCCCCCC(=O)Nc1cnn(Cc2cc(CN=[N+]=[N-])cc(c2)N=[N+]=[N-])c1
ONC(=O)CCCCCCC(=O)Nc1ccc(F)cc1
c1ccc(cc1)NC(=O)C(C(C(C(C(C(C(=O)NO)(F)F)(F)F)(F)F)(F)F)(F)F)(F)F
Cc1ccc(NC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)NO)cc1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc(Cl)cc1
CC(=O)Nc1ccc(NC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)NO)cc1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc(cc1)C#N
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc(I)cc1
Cc1ccc(NC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)NO)cc1C
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc(cc1)-c1ccccc1
CCc1cccc(NC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)NO)c1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc(cc1)-c1cn(nn1)-c1ccccc1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc2ccc3cccc4ccc1c2c34
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1nc(cs1)-c1ccccc1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc(cc1)-c1cnnn1-c1ccccc1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1cccc2ccccc12
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1cccc(c1)-c1ccccc1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc2ccccc2c1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccccc1-c1ccccc1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc2cc3ccccc3cc2c1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1cc2ccccc2c2ccccc12
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1cccc2cc3ccccc3cc12
FC(F)(C(=O)Nc1ccccc1)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccccc1
ONC(=O)C=Cc1ccc2OC3(CCN(Cc4ccccc4)CC3)CC(=O)c2c1 |w:5.5|
CCN(CC)CCNC(=O)c1ccc(cc1)-c1cn(CCCCCCC(=O)NO)nn1
CCN(CC)CCNC(=O)c1ccc(cc1)-c1cn(CCCCCCCC(=O)NO)nn1
CCN(CC)CCNC(=O)c1ccc(cn1)-c1cn(CCCCCCC(=O)NO)nn1
CCN(CC)CCNC(=O)c1ccc(cn1)-c1cn(CCCCCC(=O)NO)nn1
Cc1ccccc1Nc1ncnc2cc(NC(=O)CCCCCCC(=O)NO)sc12
Cc1cc(F)ccc1Nc1ncnc2cc(NC(=O)CCCCCCC(=O)NO)sc12
ONC(=O)CCCCCCC(=O)Nc1cc2ncnc(Nc3ccc(F)cc3F)c2s1
Cc1ccc(F)c(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)c1
COc1ccc(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)c(C)c1
ONC(=O)CCCCCCC(=O)Nc1cc2ncnc(Nc3cccc(Cl)c3)c2s1
ONC(=O)CCCCCCC(=O)Nc1cc2ncnc(Nc3cccc(Br)c3)c2s1
CCc1cccc(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)c1
CC(C)(C)c1cccc(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)c1
ONC(=O)CCCCCCC(=O)Nc1cc2ncnc(Nc3cccc(c3)C#C)c2s1
ONC(=O)CCCCCCC(=O)Nc1cc2ncnc(Nc3cccc(c3)C#N)c2s1
CCc1ccc(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)cc1
CC(C)c1ccc(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)cc1
ONC(=O)CCCCCCC(=O)Nc1cc2ncnc(Nc3ccc(Cl)cc3F)c2s1
ONC(=O)CCCCCCC(=O)Nc1cc2ncnc(Nc3cccc(F)c3)c2s1
CC(C)c1cccc(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)c1
COc1cccc(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)c1
COc1ccc(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)cc1
CN(C)c1ccc(NC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)NO)cc1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccccc1Cl
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1cccc(Cl)c1
Cc1cccc(NC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)NO)c1
COc1ccc(NC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)NO)cc1
ONC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)Nc1ccc(F)cc1
Cc1ccccc1NC(=O)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(=O)NO
CC[C@@H](C)[C@@H]1NC(=O)[C@@H](Cc2ccc(OC)cc2)NC(=O)[C@H](CCCCCC(=O)NO)NC(=O)[C@H]2CCCN2C1=O
CC[C@@H](C)[C@@H]1NC(=O)[C@@H](Cc2ccc(OC)cc2)NC(=O)[C@H](CCCCCN(O)C=O)NC(=O)[C@H]2CCCN2C1=O
CC[C@@H](C)[C@@H]1NC(=O)[C@@H](Cc2ccc(OC)cc2)NC(=O)[C@H](CCCCCN(O)C=O)NC(=O)[C@@H]2CCCN2C1=O
CC[C@@H](C)[C@@H]1NC(=O)[C@@H](Cc2ccc(OC)cc2)NC(=O)[C@H](CCCCCN(O)C=O)NC(=O)[C@H]2CCCCN2C1=O
CCC(C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)CC)NC(=O)C2CCCCN2C1=O |r|
Cc1cc(C)cc(c1)C(=O)N(CCCCCC(=O)NO)CC(=O)NC1CCCCC1
CN(C)c1ccc(cc1)C(=O)N(CCCCCC(=O)NO)CC(=O)Nc1ccc(C)cc1
Cc1cc(C)cc(c1)C(=O)N(CCCCCC(=O)NO)CC(=O)NCc1ccccc1
CN(C)c1ccc(cc1)C(=O)N(CCCCCC(=O)NO)CC(=O)NCc1ccccc1
ONC(=O)CCCCCONC(=O)Nc1cnc2ccccc2c1
COc1cc(NC(=O)NOCCCCCC(=O)NO)c2ncccc2c1
COc1cc(NC(=O)NOCCCCCC(=O)NO)c2nccc(C)c2c1
COc1cc(NC(=O)NOCCCCCC(=O)NO)c2nc(OC)cc(C)c2c1
COc1ccc(cc1)C(=O)N[C@H](COc1ccc(\C=C\C(=O)NO)cc1OC)Cc1c[nH]c2ccccc12 |r|
CCCC(CCC)C(=O)N[C@H](COc1ccc(\C=C\C(=O)NO)cc1OC)Cc1c[nH]c2ccccc12 |r|
Nc1ccccc1NC(=O)c1ccc(Cn2cc(nn2)-c2ccc(cc2)C(=O)NCc2cccnc2)cc1
Nc1ccccc1NC(=O)c1ccc(COc2ccc(F)cc2)cc1
Cn1ccc2c(CCNS(=O)(=O)c3ccc(\C=C\C(=O)NO)cc3)cccc12
ONC(=O)\C=C\c1ccc(cc1)S(=O)(=O)NCCc1cccc2[nH]ccc12
Cc1[nH]c2ccccc2c1CCNCc1cccc(C=CC(=O)NO)c1
COc1ccc(cc1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCCCCCC(=O)Nc1cc(ccc1N)-c1cccs1 |r|
COc1ccc(cc1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCCCCCC(=O)Nc1ccc(F)cc1N |r|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C[C@H](OC1=O)\C=C\CCC(=O)NO)n2 |r,c:11|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C[C@H](OC1=O)\C=C\CCSCCS)n2 |r,c:11|
Cn1ccnc1COc1nc2ccccc2nc1CCC(O)=O
OC(=O)CCc1nc2ccccc2nc1OCCOc1ccccn1
Cc1cccc(OCCOc2nc3ccccc3nc2CCC(O)=O)c1
c1cc(cnc1)C2=NN(C(=O)C=C2)CCC(=O)O
c1cc2c(cc1Cl)nc(s2)CCC(=O)O
OC(=O)CCc1nc2ccccc2nc1Sc1ccccc1
c1ccc2c(c1)nc(c(n2)OCc3ccccn3)CCC(=O)O
CN1c2ccccc2N=C(C1=O)CCC(=O)O
CCCNNC(=O)c1ccc(CNC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(OC)cc2)cc1 |r|
CCCCNNC(=O)c1ccc(CNC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(OC)cc2)cc1 |r|
CCCCCNNC(=O)c1ccc(CNC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(OC)cc2)cc1 |r|
COc1ccc(cc1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCc1ccc(cc1)C(=O)NNC1CCCC1 |r|
COc1ccc(cc1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCc1ccc(cc1)C(=O)NNc1ccccc1 |r|
COc1ccc(cc1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCc1ccc(cc1)C(=O)Nc1ccccc1N |r|
CCCNNC(=O)CCCCCNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)c1ccc(OC)cc1 |r|
CCCNNC(=O)CCCCCCNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)c1ccc(OC)cc1 |r|
CCCNNC(=O)CCCCCCCNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)c1ccc(OC)cc1 |r|
CCCNNC(=O)c1ccc(NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(OC)cc2)cc1 |r|
CCCNNC(=O)\C=C\c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(OC)cc2)cc1 |r|
CCNNC(=O)c1ccc(CNC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(OC)cc2)cc1 |r|
COc1ccc(cc1NCc1ccccc1)C(=O)NO
Cc1ccc(cc1NCc1ccc(Cl)cc1Cl)C(=O)NO
ONC(=O)c1ccc(F)c(NCc2ccccc2)c1
COc1ccc(cc1NCCc1ccccc1)C(=O)NO
Cc1ccc(cc1NCCCc1ccccc1)C(=O)NO
COc1ccc(cc1OCc1ccc(Cl)cc1)C(=O)NO
Cc1ccc(cc1NCc2ccccc2)C(=O)NO
ONC(=O)c1ccc(Cl)c(NCc2ccccc2)c1
c1ccc(cc1)NC(=O)c2cccc(c2)C(=O)NO
ONC(=O)c1ccc(CNc2cccc3ncccc23)cc1
ONC(=O)c1ccc(CNc2ccnc3ccccc23)cc1
ONC(=O)c1ccc(CNc2cnc3ccccc3c2)cc1
ONC(=O)c1ccc(CNc2cccc3CCCc23)cc1
ONC(=O)c1ccc(CNc2cccc3CCCCc23)cc1
ONC(=O)c1ccc(CNc2cccc3nccnc23)cc1
ONC(=O)c1ccc(CNc2cncc3ccccc23)cc1
ONC(=O)c1ccc(CNc2cccc3ccncc23)cc1
Cc1ccc2cccc(NCc3ccc(cc3)C(=O)NO)c2n1
ONC(=O)c1cccc(CNc2cccc3cccnc23)c1
ONC(=O)c1ccc(NCc2cccc3cccnc23)cc1
ONC(=O)c1ccc(CCc2cccc3cccnc23)cc1
ONC(=O)c1ccc(CSc2cccc3cccnc23)cc1
ONC(=O)c1ccc(cc1)C(=O)Nc1cccc2cccnc12
ONC(=O)c1ccc(cc1)C(=O)Nc1cccc2ncccc12
ONC(=O)\C=C\c1ccc(CNc2cccc3ncccc23)cc1
ONC(=O)c1ccc(CNc2cccc3cccnc23)cc1
ONC(=O)c1ccc(CNc2ccc3cccnc3c2)cc1
ONC(=O)c1ccc(CNc2ccc3ncccc3c2)cc1
ONC(=O)c1ccc(CNc2ccc3ccccc3n2)cc1
ONC(=O)c1ccc(CNc2cccc3cnccc23)cc1
ONC(=O)c1ccc(Nc2cccc3cccnc23)cc1
ONC(=O)c1ccc(COc2cccc3cccnc23)cc1
ONC(=O)\C=C\c1ccc(CNc2cccc3cccnc23)cc1
ONC(=O)c1ccc(CNc2cccc3cn[nH]c23)cc1
CC#CCOc1ccc(cc1)C(=O)N[C@H](C(=O)NO)C(C)(C)N
ONC(=O)CCCn1cc(cn1)-c1ncnc2[nH]ccc12
ONC(=O)\C=C\c1ccc(NCCCn2cc(cn2)-c2ncnc3[nH]ccc23)cc1
ONC(=O)CCCCCCC(=O)Nc1ccc(NCCCn2cc(cn2)-c2ncnc3[nH]ccc23)cc1
ONC(=O)CCCCCCC(=O)Nc1ccc(NC(=O)CCCn2cc(cn2)-c2ncnc3[nH]ccc23)cc1
ONC(=O)CCCCCCCCCCn1cc(cn1)-c1ncnc2[nH]ccc12
ONC(=O)CCCCCCCn1cc(cn1)-c1ncnc2[nH]ccc12
ONC(=O)CCCCCn1cc(cn1)-c1ncnc2[nH]ccc12
ONC(=O)CCCCn1cc(cn1)-c1ncnc2[nH]ccc12
CC(CCCCCC(=O)NO)n1cc(cn1)-c1ncnc2[nH]ccc12
ONC(=O)CCCCCCC(=O)Nc1ccc(CCCn2cc(cn2)-c2ncnc3[nH]ccc23)cc1
ONC(=O)CCCCCCn1cc(cn1)-c1ncnc2[nH]ccc12
ONC(=O)\C=C\c1ccc(CNCc2ccc3cccc(Cl)c3n2)cc1
ONC(=O)\C=C\c1ccc(CNCc2ccc3ccccc3n2)cc1
COc1ccc(Cl)cc1C(=O)NCCc1ccc(\C=C\C(=O)NO)cc1
COc1ccc(Cl)cc1C(=O)NCCc1cccc(\C=C\C(=O)NO)c1
COc1cc(ccc1O)C(=O)NCCc1ccc(\C=C\C(=O)NO)cc1
ONC(=O)\C=C\c1ccc(CCNC(=O)c2ccc3OCOc3c2)cc1
ONC(=O)\C=C\c1ccc(CCNC(=O)c2cncc(F)c2)cc1
ONC(=O)\C=C\c1ccc(CCNC(=O)c2ccc3ncccc3c2)cc1
ONC(=O)\C=C\c1ccc(CCNC(=O)c2ccc3[nH]cnc3c2)cc1
COc1ccc(Cl)cc1C(=O)NCCc1ccc(CCC(=O)NO)cc1
ONC(=O)\C=C\c1ccc(CCNC(=O)c2cc(ccc2Cl)C(F)(F)F)cc1
ONC(=O)\C=C\c1ccc(CCNC(=O)c2ccc3OCCOc3c2)cc1
ONC(=O)\C=C\c1ccc(CCNC(=O)c2c[nH]c3ncccc23)cc1
ONC(=O)c1ccc(Cn2cc(nn2)-c2ccc(CN3CCCC3)cc2)cc1
c1ccc(cc1)N(CCO)C(=O)Cc2ccc(cc2)C(=O)NO
c1ccc(cc1)CC(=O)N(CCO)Cc2ccc(cc2)C(=O)NO
ONC(=O)c1ccc(NCc2csc3ccc(Br)cc23)cc1
ONC(=O)c1ccc(Cn2c3CCS(=O)(=O)c3c3ccccc23)cc1
[H][C@]12CCCC[C@@]1([H])N(Cc1ccc(cc1)C(=O)NO)c1ccccc1S(=O)(=O)C2 |r|
ONC(=O)c1cccc(c1)-c1csc(CSc2ccccc2)n1
CN1C(=O)C2CN(Cc3c2c2ccccc2n3Cc2ccc(cc2)C(=O)NO)C1=O
ONC(=O)c1ccc(CC(=O)NC2=CC(=O)c3ccccc3C2=O)cc1 |t:12|
Cc1nc2ccccc2n1Cc1ccc(cc1F)C(=O)NO
Nc1ccccc1NC(=O)CCCCCCC(=O)Nc1cccc(c1)-c1cn(nn1)-c1ccccc1
C\C=C1/NC(=O)[C@H](CS)NC(=O)[C@H](NC(=O)C[C@H](OC(=O)[C@@H](NC1=O)C(C)C)\C=C\CS)C(C)C |r|
C[C@@H]1NC(=O)[C@H](CCCCCC(=O)NO)NC(=O)[C@H]2CCCN2C(=O)[C@H](C)NC1=O
C[C@@H]1NC(=O)[C@H](CCCCCC(=O)C2CO2)NC(=O)[C@H]2CCCN2C(=O)[C@H](C)NC1=O
O=C(CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2ccccc2)NC1=O)C1CO1
C\C=C1/NC(=O)[C@@H](CS)NC(=O)[C@H](NC(=O)C[C@H](OC(=O)[C@@H](NC1=O)C(C)C)\C=C\CCS)C(C)C
CCC(C)[C@@H]1NC(=O)[C@@H](Cc2ccc(OC)cc2)NC(=O)[C@H](CCCCCC(=O)C(F)(F)C(F)(F)F)NC(=O)[C@H]2CCCN2C1=O
CCC(C)[C@@H]1NC(=O)[C@@H](Cc2ccc(OC)cc2)NC(=O)[C@H](CCCCSCC(=O)C(F)(F)F)NC(=O)[C@H]2CCCN2C1=O
CCC(C)[C@@H]1NC(=O)[C@@H](Cc2ccc(OC)cc2)NC(=O)[C@H](CCCCCC(=O)C(F)(F)F)NC(=O)[C@H]2CCCN2C1=O
COc1ccc2c(cn(c2c1)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1)C(=O)c1cc(OC)c(OC)c(OC)c1
COc1ccc2c(cn(Cc3ccc(cc3)C(=O)NO)c2c1)C(=O)c1cc(OC)c(OC)c(OC)c1
COc1ccc2c(cn(Cc3ccc(\C=C\C(=O)NO)cc3)c2c1)C(=O)c1cc(OC)c(OC)c(OC)c1
COc1cc(cc(OC)c1OC)C(=O)c1cn(c2ccccc12)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1
COc1ccc(cc1)C(=O)c1cn(Cc2ccc(cc2)C(=O)NO)c2cc(OC)ccc12
COc1ccc2c(cn(c2c1)S(=O)(=O)c1ccc(\C=C\C(=O)NO)cc1)C(=O)c1cc(OC)c(OC)c(OC)c1
COc1cc(cc(OC)c1OC)C(=O)c1cn(Cc2ccc(\C=C\C(=O)NO)cc2)c2ccccc12
COc1ccc2[nH]c(C)c(CC(=O)N[C@@H](CCCCCC(=O)NO)C(=O)NCCc3c([nH]c4ccccc34)-c3ccccc3)c2c1
CN1CCCCC1C(=O)N[C@@H](CCCCCC(C)=O)C(=O)Nc1nc(cs1)-c1ccccc1 |r|
ONC(=O)CCCCCCNc1ncnc2ccc(Cl)cc12
ONC(=O)CCCCCCNc1ncnc2ccc(F)cc12
CN1CCCCC1N[C@@H](CCCCCC(C)=O)C(=O)Nc1nc(cs1)-c1ccccc1 |w:6.7|
CC(C)[C@H]1NC(=O)[C@@H](C)[C@@H](CC=CCCC(O)=O)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@@H](C)NC1=O |w:11.10|
OCCN(CCc1cc2ccccc2[nH]1)Cc1ccc(\C=C\C(=O)NO)cc1
C[C@H]1CN(CCN1C(=O)OCc1ccccc1)c1ccc(cn1)C(=O)Nc1cc(ccc1N)-c1ccccc1
Nc1ccccc1NC(=O)c1cccnc1
Nc1ccc(cc1NC(=O)c1ccccc1)-c1ccccc1
Nc1ccc(cc1NC(=O)c1cccnc1)-c1ccccc1
Nc1ccc(cc1NC(=O)c1ccccc1)-c1cccs1
Nc1ccccc1NC(=O)c1ccccc1
Nc1ccc(cc1NC(=O)c1cccnc1)-c1cccs1
COC(=O)[C@H](Cc1ccc(cc1)-c1ccc(cc1)-c1ccccc1)NC(=O)CCCCCCC(=O)NO
COC(=O)[C@H](Cc1ccc(cc1)-c1ccoc1)NC(=O)CCCCCCCC(=O)NO
COC(=O)[C@H](Cc1ccc(cc1)-c1ccoc1)NC(=O)CCCCCCC(=O)NO
COC(=O)[C@H](Cc1ccc(cc1)-c1ccco1)NC(=O)CCCCCCCC(=O)NO
COC(=O)[C@H](Cc1ccc(cc1)-c1ccco1)NC(=O)CCCCCCC(=O)NO
COC(=O)[C@H](Cc1ccc(cc1)-c1ccsc1)NC(=O)CCCCCCCC(=O)NO
COC(=O)[C@H](Cc1ccc(cc1)-c1ccsc1)NC(=O)CCCCCCC(=O)NO
COC(=O)[C@H](Cc1ccc(cc1)-c1cccs1)NC(=O)CCCCCCCC(=O)NO
COC(=O)[C@H](Cc1ccc(cc1)-c1cccs1)NC(=O)CCCCCCC(=O)NO
COC(=O)[C@H](Cc1ccc(cc1)-c1ccccc1)NC(=O)CCCCCCCC(=O)NO
CC1(C)NC(=O)[C@H](CCCCCC(=O)NO)NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC1=O
COC(=O)[C@H](Cc1ccc(cc1)-c1ccccc1)NC(=O)CCCCCCC(=O)NO
CN(C)c1ccc(cc1)C(=O)NCCCCCCC(=O)NO
COC(=O)[C@H](Cc1ccc(Br)cc1)NC(=O)CCCCCCC(=O)NO |r|
COC(=O)[C@H](Cc1ccc(cc1)-c1ccc2ccccc2c1)NC(=O)CCCCCCCC(=O)NO
COC(=O)[C@H](Cc1ccc(cc1)-c1ccc2ccccc2c1)NC(=O)CCCCCCC(=O)NO
COC(=O)[C@H](Cc1ccc(Br)cc1)NC(=O)CCCCCCCC(=O)NO
COC(=O)[C@H](Cc1ccc(cc1)-c1ccc(cc1)-c1ccccc1)NC(=O)CCCCCCCC(=O)NO
[H][C@]12CN(Cc3c1c1ccccc1n3Cc1ccc(cc1)C(=O)NO)C(=O)N(C)C2=O |r|
CN1C(=O)C2CN(Cc3c2c2ccccc2n3Cc2ccc(\C=C\C(=O)NO)cc2)C1=O
CN1C(=O)C2CN(Cc3c2c2ccccc2n3Cc2cccc(\C=C\C(=O)NO)c2)C1=O
CN1C(=O)C2CN(Cc3c2c2ccccc2n3Cc2ccc(cc2)C(O)=O)C1=O
ONC(=O)\C=C\c1ccc(Cn2c3C4CCCC(=O)N4CCc3c3ccccc23)cc1
CN1C(=O)C2CN(Cc3c2c2ccc4ccccc4c2n3Cc2ccc(cc2)C(=O)NO)C1=O
CN1C(=O)C2N(CCc3c2c2ccccc2n3Cc2ccc(cc2)C(=O)NO)C1=O
COc1ccc2n(Cc3ccc(cc3)C(=O)NO)c3CN4CC(c3c2c1)C(=O)N(C)C4=O
CN1C(=O)C2CN(Cc3c2c2ccccc2n3Cc2ccc(cc2)C(=O)NO)C1=S
COc1ccc2n(Cc3ccc(cc3)C(=O)NO)c3CN4CC(c3c2c1)C(=O)N(C)C4
CN1CN2CC(c3c(C2)n(Cc2ccc(cc2)C(=O)NO)c2ccccc32)C1=O
COc1ccc2c3C4CN(Cc3n(Cc3ccc(cc3)C(=O)NO)c2c1)C(=O)N(C)C4=O
CN1C(=O)C2CN(Cc3c2c2cc(OCCN4CCOCC4)ccc2n3Cc2ccc(cc2)C(=O)NO)C1=O
CN1C(=O)C2CN(Cc3c2c2cc(OCc4ccccc4)ccc2n3Cc2ccc(cc2)C(=O)NO)C1=O
CN1C(=O)C2CN(Cc3c2c2cc(O)ccc2n3Cc2ccc(cc2)C(=O)NO)C1=O
CN1C(=O)N2CC(c3c(C2)n(Cc2ccc(cc2)C(=O)NO)c2ccccc32)C1=S
CN1CC2CN(Cc3c2c2ccccc2n3Cc2ccc(cc2)C(=O)NO)C1=O
ONC(=O)c1ccc(Cn2c3CN4CCC(C4)c3c3ccccc23)cc1
[H][C@@]12CN(Cc3c1c1ccccc1n3Cc1ccc(cc1)C(=O)NO)C(=O)N(C)C2=O |r|
ONC(=O)c1ccc(Cn2c3C4CCCC(=O)N4CCc3c3ccccc23)cc1
C[C@H]1NC(=O)[C@@H](C)[C@@H](CC=CCCC(N)=O)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@@H](C)NC1=O |w:9.8|
CC(C)[C@H]1NC(=O)[C@@H](C)[C@@H](CC=CCCC(O)=O)NC(=O)[C@@H](Cc2ccc(O)cc2)NC(=O)[C@@H](C)NC1=O |w:11.10|
CC(C)[C@H]1NC(=O)[C@@H](C)[C@@H](CC=CCCC(N)=O)NC(=O)[C@@H](Cc2ccc(O)cc2)NC(=O)[C@@H](C)NC1=O |w:11.10|
CC(C)[C@H]1NC(=O)[C@@H](C)[C@@H](CC=CCCC(N)=O)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@@H](C)NC1=O |w:11.10|
ONC(=O)CCCCCCNC(=O)c1ccc(NCc2cn(CCCNC(=S)Nc3ccc(c(c3)C(O)=O)-c3c4ccccc4oc4cc(=O)ccc34)nn2)cc1 |(33.95,-8.48,;32.41,-8.48,;31.64,-7.15,;32.4,-5.81,;30.1,-7.15,;29.32,-5.82,;27.78,-5.82,;27.01,-4.48,;25.47,-4.48,;24.7,-3.15,;23.16,-3.15,;22.39,-1.81,;23.16,-.48,;20.85,-1.81,;20.08,-3.15,;18.54,-3.15,;17.79,-1.81,;16.25,-1.81,;15.48,-.47,;13.94,-.47,;12.9,.67,;11.5,.03,;10.17,.8,;8.83,.02,;7.5,.79,;6.17,.02,;4.83,.78,;4.83,2.32,;3.5,.01,;3.5,-1.53,;2.18,-2.3,;2.17,-3.85,;3.51,-4.62,;4.84,-3.85,;4.84,-2.3,;6.18,-4.61,;6.18,-6.15,;7.51,-3.84,;3.48,-7.08,;4.8,-7.85,;6.13,-7.07,;7.46,-7.83,;7.47,-9.38,;6.13,-10.16,;4.79,-9.38,;3.47,-10.15,;2.14,-9.37,;.82,-10.14,;-.51,-9.37,;-1.84,-10.14,;-.51,-7.84,;.82,-7.08,;2.14,-7.84,;11.66,-1.49,;13.17,-1.81,;18.54,-.48,;20.08,-.48,)|
NCCCn1cc(CNc2ccc(cc2)C(=O)NCCCCCCC(=O)NO)nn1
O=C1CCc2c(O1)ccc1ccccc21
CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)CC)NC(=O)[C@H]2CCCCN2C1=O |r|
CN1CCC(CC1)C(=O)N[C@@H](CCCCCC(C)=O)c1nc(c[nH]1)-c1ccc2ccccc2c1 |r|
CCC(=O)CCCCC[C@H](NC(=O)C1CCN(C)CC1)c1nc(c[nH]1)-c1ccc2ccccc2c1 |r|
CCCC(=O)CCCCC[C@H](NC(=O)C1CCN(C)CC1)c1nc(c[nH]1)-c1ccc2ccccc2c1 |r|
CCCCC(=O)CCCCC[C@H](NC(=O)C1CCN(C)CC1)c1nc(c[nH]1)-c1ccc2ccccc2c1 |r|
Cc1cc(S)c2ncccc2c1
Cc1ccc(S)c2ncccc12
Cc1ccnc2c(S)cccc12
Sc1cccc2cccnc12
Cc1cnc2c(S)cccc2c1
ONC(=O)\C=C\c1ccc(CN2CCN(CC2)C(=O)c2cc(Cc3n[nH]c(=O)c4ccccc34)ccc2F)cc1
ONC(=O)Cc1ccc(CN2CCN(CC2)C(=O)c2cc(Cc3n[nH]c(=O)c4ccccc34)ccc2F)cc1
ONC(=O)\C=C\c1ccc(CCNC(=O)c2cc(Cc3n[nH]c(=O)c4ccccc34)ccc2F)cc1
ONC(=O)c1ccc(CN2CCN(CC2)C(=O)c2cc(Cc3n[nH]c(=O)c4ccccc34)ccc2F)cc1
CCCCC(CCCC(=O)NO)CCC(=O)Nc1ccccc1
CCCCCCC(CCCC(=O)NO)CCC(=O)Nc1ccccc1
ONC(=O)CCCC(CCC(=O)Nc1ccccc1)Cc1ccccc1
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](C)NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2cccc3ccccc23)NC1=O |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@@H](C)n2nncc2[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
CC(C)C[C@H]1CC(=O)N[C@@H](C)C(=O)N[C@@H](CCCCCC(=O)NO)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1 |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](CCCCNC(C)=O)NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
CC(C)C[C@H]1CC(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H](CCCCCC(=O)NO)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1 |r|
CC(C)C[C@H]1CC(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCC(O)=O)C(=O)N[C@@H](Cc2cccc3ccccc23)C(=O)N1 |r|
CC(C)C[C@H]1CC(=O)N[C@@H](C)C(=O)N[C@@H](CCCCCC(O)=O)C(=O)N[C@@H](Cc2cccc3ccccc23)C(=O)N1 |r|
CC(C)C[C@H]1CC(=O)N[C@@H](C)C(=O)N[C@@H](CCCCCC(=O)C(F)(F)F)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1 |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@@H]2CCCN2C(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
[#6]-[#6](-[#6])-[#6@H](-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#6]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#7]-[#6](=O)-[#6@@H]-1-[#6]-[#6]-[#6]-[#7]-1-[#6](=O)-[#6]-[#7]-[#6](=O)-[#6]-[#7]-[#6](=O)-[#6]-[#6]-[#6]-c1cn(nn1)-c1ccc(cc1)-c1cn(-[#6]-[#6]-[#6]-[#6]-[#6]-[#6](=O)-[#7]-[#8])nn1)-[#6](=O)-[#7]-[#6]-[#6](=O)-[#7]-[#6]-[#6](-[#7])=O |r|
[#6]-[#6](-[#6])-[#6@H](-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#6]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#7]-[#6](=O)-[#6@@H]-1-[#6]-[#6]-[#6]-[#7]-1-[#6](=O)-[#6]-[#7]-[#6](=O)-[#6]-[#7]-[#6](=O)-[#6]-[#6]-[#6]-c1cn(nn1)-c1ccc(cc1)-c1cn(-[#6]-[#6]-[#6]-[#6]-[#6]-[#6]-[#6](=O)-[#7]-[#8])nn1)-[#6](=O)-[#7]-[#6]-[#6](=O)-[#7]-[#6]-[#6](-[#7])=O |r|
[#6]-[#6](-[#6])-[#6@H](-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#6]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#7]-[#6](=O)-[#6@@H]-1-[#6]-[#6]-[#6]-[#7]-1-[#6](=O)-[#6]-[#7]-[#6](=O)-[#6]-[#7]-[#6](=O)-[#6]-[#6]-[#6]-c1cn(nn1)-c1ccc(cc1)-c1cn(-[#6]-[#6]-[#6]-[#6]-[#6]-[#6]-[#6]-[#6](=O)-[#7]-[#8])nn1)-[#6](=O)-[#7]-[#6]-[#6](=O)-[#7]-[#6]-[#6](-[#7])=O |r|
CCC(=O)CCCCC[C@@H]1NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCCC(=O)CC)NC1=O |r|
[#6]-[#6](-[#6])-[#6]-[#6@H]-1-[#6]-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]-[#6]-[#6]-[#6](-[#8])=O)-[#6](=O)-[#7]-[#6@@H](-[#6]-c2cccc3ccccc23)-[#6](=O)-[#7]-1 |r|
[#7]\[#6](-[#7])=[#7]\[#6]-[#6]-[#6]-[#6@@H]-1-[#7]-[#6](=O)-[#6]-[#6@H](-[#6]-[#8])-[#7]-[#6](=O)-[#6@H](-[#6]-c2cccc3ccccc23)-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#6]-[#6](-[#8])=O)-[#7]-[#6]-1=O |r|
[#7]\[#6](-[#7])=[#7]\[#6]-[#6]-[#6]-[#6@@H]-1-[#7]-[#6](=O)-[#6]-[#6@H](-[#6]-c2ccc(-[#8])cc2)-[#7]-[#6](=O)-[#6@H](-[#6]-c2cccc3ccccc23)-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#6]-[#6](-[#8])=O)-[#7]-[#6]-1=O |r|
CC(=O)NCCCC[C@@H]1NC(=O)C[C@H](Cc2ccc(O)cc2)NC(=O)[C@H](Cc2cccc3ccccc23)NC(=O)[C@H](CCCCCC(O)=O)NC1=O |r|
OC(=O)CCCCC[C@@H]1NC(=O)[C@H](Cc2c(F)c(F)c(F)c(F)c2F)NC(=O)C[C@H](Cc2ccc(O)cc2)NC(=O)[C@H](Cc2cccc3ccccc23)NC1=O |r|
[#7]\[#6](-[#7])=[#7]\[#6]-[#6]-[#6]-[#6@@H]-1-[#7]-[#6](=O)-[#6]-[#6@H](-[#6]-c2ccc(-[#8])cc2)-[#7]-[#6](=O)-[#6@H](-[#6]-[#6](-[#8])=O)-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#6]-[#6](-[#8])=O)-[#7]-[#6]-1=O |r|
[#7]\[#6](-[#7])=[#7]\[#6]-[#6]-[#6]-[#6@@H]-1-[#7]-[#6](=O)-[#6]-[#6@H](-[#6]-c2ccc(-[#8])cc2)-[#7]-[#6](=O)-[#6@H](-[#6]-[#6](-[#8])=O)-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#6]-[#6](=O)-[#7]-[#8])-[#7]-[#6]-1=O |r|
CC(C)C[C@H]1CC(=O)N[C@@H](CCCCNC(C)=O)C(=O)N[C@@H](CCCCCC(O)=O)C(=O)N[C@@H](Cc2cccc3ccccc23)C(=O)N1 |r|
CC(C)C[C@H]1CC(=O)N[C@@H](C)C(=O)N[C@@H](CCCCCC(O)=O)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1 |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](C)NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
CCC(=O)CCCSC[C@@H]1NC(=O)[C@H](C)NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
CCC(=O)CCSC[C@@H]1NC(=O)[C@H](C)NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
CC(C)C[C@H]1CC(=O)N[C@@H](C)C(=O)N[C@@H](CSCCC(O)=O)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1 |r|
CC(C)C[C@H]1CC(=O)N[C@@H](C)C(=O)N[C@@H](CSCC(O)=O)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1 |r|
CC(C)C[C@H]1CC(=O)N[C@@H](CCCCCNC(C)=O)C(=O)N[C@@H](CCCCCC(O)=O)C(=O)N[C@@H](Cc2cccc3ccccc23)C(=O)N1 |r|
OC(=O)CCCCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)C[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2cccc3ccccc23)NC1=O |r|
CC(C)C[C@H]1CC(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H](CCCCCC(O)=O)C(=O)N[C@@H](Cc2cccc3ccccc23)C(=O)N1 |r|
CC1(C)NC(=O)C[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2cccc3ccccc23)NC(=O)[C@H](CCCCCC(O)=O)NC1=O |r|
CC(C)C[C@H]1CC(=O)NC(C)(C)C(=O)N[C@@H](CCCCCC(O)=O)C(=O)N[C@@H](Cc2cccc3ccccc23)C(=O)N1 |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
CC(C)C[C@H]1CC(=O)N[C@@H](CCCCNC(C)=O)C(=O)N[C@@H](CSCCC(O)=O)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1 |r|
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2[nH]1
Cn1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1
CC(C)n1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1C1CCCCC1
CN(C)CCn1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1
CCN(CC)CCn1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1
CC(C)N(CCn1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1)C(C)C
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1CCN1CCOCC1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1CC1CCNCC1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1CCN1CCCCC1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1CCN1CCCC1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1-c1ccccc1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1-c1ccc(Cl)cc1
COc1ccc(cc1)-n1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1CCc1ccccc1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1CCCc1ccccc1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1Cc1ccccc1
C[C@H](c1ccccc1)n1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1 |r|
C[C@@H](c1ccccc1)n1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1 |r|
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1C1CCCNC1
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1[C@@H]1CCCNC1 |r|
ONC(=O)\C=C\c1cccc(c1)-c1nc2ccccc2n1[C@H]1CCCNC1 |r|
CN1CCC[C@@H](C1)n1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1 |r|
CN1CCC[C@H](C1)n1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1 |r|
CCN1CCCC(C1)n1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1
CCN1CCC[C@H](C1)n1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1 |r|
CCN1CCC[C@@H](C1)n1c(nc2ccccc12)-c1cccc(\C=C\C(=O)NO)c1 |r|
Cc1c(nc(-c2cccc(\C=C\C(=O)NO)c2)n1CCN1CCOCC1)-c1ccccc1
Cc1c(nc(-c2cccc(\C=C\C(=O)NO)c2)n1CCc1ccccc1)-c1ccccc1
CN1CCC[C@H](C1)n1c(C)c(nc1-c1cccc(\C=C\C(=O)NO)c1)-c1ccccc1 |r|
CCN1CCC[C@H](C1)n1c(C)c(nc1-c1cccc(\C=C\C(=O)NO)c1)-c1ccccc1 |r|
CC(C)N1CCC[C@H](C1)n1c(C)c(nc1-c1cccc(\C=C\C(=O)NO)c1)-c1ccccc1 |r|
Cc1nc(-c2cccc(\C=C\C(=O)NO)c2)n(CCN2CCOCC2)c1-c1ccccc1
Cc1nc(-c2cccc(\C=C\C(=O)NO)c2)n(CCc2ccccc2)c1-c1ccccc1
CN1CCC[C@H](C1)n1c(nc(C)c1-c1ccccc1)-c1cccc(\C=C\C(=O)NO)c1 |r|
CCN1CCC[C@H](C1)n1c(nc(C)c1-c1ccccc1)-c1cccc(\C=C\C(=O)NO)c1 |r|
CC(C)N1CCC[C@H](C1)n1c(nc(C)c1-c1ccccc1)-c1cccc(\C=C\C(=O)NO)c1 |r|
Cc1c(Cc2ccccc2)nc(-c2cccc(\C=C\C(=O)NO)c2)n1CCN1CCOCC1
Cc1c(Cc2ccccc2)nc(-c2cccc(\C=C\C(=O)NO)c2)n1CCc1ccccc1
CN1CCC[C@H](C1)n1c(C)c(Cc2ccccc2)nc1-c1cccc(\C=C\C(=O)NO)c1 |r|
CCN1CCC[C@H](C1)n1c(C)c(Cc2ccccc2)nc1-c1cccc(\C=C\C(=O)NO)c1 |r|
Cc1nc(-c2cccc(\C=C\C(=O)NO)c2)n(CCN2CCOCC2)c1Cc1ccccc1
Cc1nc(-c2cccc(\C=C\C(=O)NO)c2)n(CCc2ccccc2)c1Cc1ccccc1
Cc1nc(-c2cccc(\C=C\C(=O)NO)c2)n(CCN2CCOCC2)c1C
Cc1nc(-c2cccc(\C=C\C(=O)NO)c2)n(CCc2ccccc2)c1C
CCN1CCC[C@H](C1)n1c(C)c(C)nc1-c1cccc(\C=C\C(=O)NO)c1 |r|
Cc1nc(C)n(CCc2ccccc2)c1-c1cccc(\C=C\C(=O)NO)c1
CCN1CCC[C@H](C1)n1c(C)nc(C)c1-c1cccc(\C=C\C(=O)NO)c1 |r|
Cc1nc(-c2ccccc2)n(CCc2ccccc2)c1-c1cccc(\C=C\C(=O)NO)c1
CCN1CCC[C@H](C1)n1c(nc(C)c1-c1cccc(\C=C\C(=O)NO)c1)-c1ccccc1 |r|
Cc1nc(Cc2ccccc2)n(CCc2ccccc2)c1-c1cccc(\C=C\C(=O)NO)c1
CCN1CCC[C@H](C1)n1c(Cc2ccccc2)nc(C)c1-c1cccc(\C=C\C(=O)NO)c1 |r|
C[C@H](\C=C(/C)\C=C\C(=O)NO)[C@H]1CC[C@H]2\C(CCC[C@]12C)=C\C=C1/C[C@@H](O)C[C@@H](O)C1 |r|
[#6]-[#6@H](-[#6]-[#6]-[#6]-[#6](=O)-[#7]-[#8])-[#6@H]1-[#6]-[#6]-[#6@H]2\[#6](-[#6]-[#6]-[#6][C@]12[#6])=[#6]\[#6]=[#6]-1/[#6]-[#6@@H](-[#8])-[#6]-[#6@H](-[#8])-[#6]-1 |r|
[#6]-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#6](=O)-[#7]-[#8])-[#6@H]1-[#6]-[#6]-[#6@H]2\[#6](-[#6]-[#6]-[#6][C@]12[#6])=[#6]\[#6]=[#6]-1/[#6]-[#6@@H](-[#8])-[#6]-[#6@H](-[#8])-[#6]-1 |r|
[#6]-[#6@H](-[#6]-[#6]-[#6]-[#6](=O)-[#7]-c1ccccc1-[#7])-[#6@H]1-[#6]-[#6]-[#6@H]2\[#6](-[#6]-[#6]-[#6][C@]12[#6])=[#6]\[#6]=[#6]-1/[#6]-[#6@@H](-[#8])-[#6]-[#6@H](-[#8])-[#6]-1 |r|
[#6]-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7]-[#6](=O)-[#6]-[#16])-[#6@H]1-[#6]-[#6]-[#6@H]2\[#6](-[#6]-[#6]-[#6][C@]12[#6])=[#6]\[#6]=[#6]-1/[#6]-[#6@@H](-[#8])-[#6]-[#6@H](-[#8])-[#6]-1 |r|
[#6]-[#6@H](-[#6]-[#6]-[#6]-[#7]S([#6])(=O)=O)-[#6@H]1-[#6]-[#6]-[#6@H]2\[#6](-[#6]-[#6]-[#6][C@]12[#6])=[#6]\[#6]=[#6]-1/[#6]-[#6@@H](-[#8])-[#6]-[#6@H](-[#8])-[#6]-1 |r|
[#6]-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7]S([#6])(=O)=O)-[#6@H]1-[#6]-[#6]-[#6@H]2\[#6](-[#6]-[#6]-[#6][C@]12[#6])=[#6]\[#6]=[#6]-1/[#6]-[#6@@H](-[#8])-[#6]-[#6@H](-[#8])-[#6]-1 |r|
[#6]-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7]S(=O)(=O)C(F)(F)F)-[#6@H]1-[#6]-[#6]-[#6@H]2\[#6](-[#6]-[#6]-[#6][C@]12[#6])=[#6]\[#6]=[#6]-1/[#6]-[#6@@H](-[#8])-[#6]-[#6@H](-[#8])-[#6]-1 |r|
[#6]-[#6]-[#6]-[#6]S(=O)(=O)[#7]-[#6]-[#6]-[#6]-[#6]-[#6@@H](-[#6])-[#6@H]1-[#6]-[#6]-[#6@H]2\[#6](-[#6]-[#6]-[#6][C@]12[#6])=[#6]\[#6]=[#6]-1/[#6]-[#6@@H](-[#8])-[#6]-[#6@H](-[#8])-[#6]-1 |r|
[#6]-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7]S(=O)(=O)c1ccccc1)-[#6@H]1-[#6]-[#6]-[#6@H]2\[#6](-[#6]-[#6]-[#6][C@]12[#6])=[#6]\[#6]=[#6]-1/[#6]-[#6@@H](-[#8])-[#6]-[#6@H](-[#8])-[#6]-1 |r|
[#6]-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7]S([#7])(=O)=O)-[#6@H]1-[#6]-[#6]-[#6@H]2\[#6](-[#6]-[#6]-[#6][C@]12[#6])=[#6]\[#6]=[#6]-1/[#6]-[#6@@H](-[#8])-[#6]-[#6@H](-[#8])-[#6]-1 |r|
[#6]-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#6]-[#7]S([#7])(=O)=O)-[#6@H]1-[#6]-[#6]-[#6@H]2\[#6](-[#6]-[#6]-[#6][C@]12[#6])=[#6]\[#6]=[#6]-1/[#6]-[#6@@H](-[#8])-[#6]-[#6@H](-[#8])-[#6]-1 |r|
[#6]-[#7]-[#6](=O)-[#6](=O)-[#6]-[#6]-[#6]-[#6]-[#6@@H](-[#6])-[#6@H]1-[#6]-[#6]-[#6@H]2\[#6](-[#6]-[#6]-[#6][C@]12[#6])=[#6]\[#6]=[#6]-1/[#6]-[#6@@H](-[#8])-[#6]-[#6@H](-[#8])-[#6]-1 |r|
CCCC(=O)O
CCCC(=O)NO
[O-]C(=O)CCCc1ccccc1
c1ccc(cc1)CCCC(=O)NO
CCCC(CCC)C(=O)O
CCCC(CCC)C(=O)NO
CC(C)C[C@H]1CC(=O)N[C@@H](C)C(=O)N[C@@H](CCCCCC(N)=O)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1 |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](C)N(C)C(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCCCC(=O)CC)NC(=O)[C@@H](C)n2cc1nn2 |r|
ONC(=O)c1ccc(Cn2c3CCN(CC=C)Cc3c3ccccc23)cc1
ONC(=O)c1ccc(Cn2c3CN(Cc4ccccc4)CCc3c3ccccc23)cc1
CN1CCc2c(C1)n(Cc1ccc(cc1)C(=O)NO)c1ccccc21
ONC(=O)c1ccc(Cn2c3CNCCc3c3ccccc23)cc1
NC(=O)CCCN1CCc2c(C1)c1ccccc1n2Cc1ccc(cc1)C(=O)NO
NC(=O)CN1CCc2c(C1)c1ccccc1n2Cc1ccc(cc1)C(=O)NO
NC(=O)CCN1CCc2c(C1)c1ccccc1n2Cc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(Cn2c3CCN(Cc4ccncc4)Cc3c3ccccc23)cc1
COc1ccc(CN2CCc3c(C2)c2ccccc2n3Cc2ccc(cc2)C(=O)NO)cc1
COc1cccc(CN2CCc3c(C2)c2ccccc2n3Cc2ccc(cc2)C(=O)NO)c1
ONC(=O)c1ccc(Cn2c3CCN(Cc4ccccc4)Cc3c3ccccc23)cc1
CC(C)N1CCc2c(C1)c1ccccc1n2Cc1ccc(cc1)C(=O)NO
CCN1CCc2c(C1)c1ccccc1n2Cc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(Cn2c3CCNCc3c3ccccc23)cc1
CC(C)(C)OC(=O)N1CCc2c(C1)c1ccccc1n2Cc1ccc(cc1)C(=O)NO
CN1CCc2c(C1)c1cc(Br)ccc1n2Cc1ccc(cc1)C(=O)NO
CN1CCc2c(C1)c1cc(Cl)ccc1n2Cc1ccc(cc1)C(=O)NO
COc1ccc2n(Cc3ccc(cc3)C(=O)NO)c3CCN(C)Cc3c2c1
CN1CCc2c(C1)c1cc(ccc1n2Cc1ccc(cc1)C(=O)NO)C(C)(C)C
CN1CCc2c(C1)c1c(C)cc(C)cc1n2Cc1ccc(cc1)C(=O)NO
CN1CCc2c(C1)c1cc(C)ccc1n2Cc1ccc(cc1)C(=O)NO
CN1CCc2c(C1)c1ccc(C)cc1n2Cc1ccc(cc1)C(=O)NO
CN1CCc2c(C1)c1cccc(C)c1n2Cc1ccc(cc1)C(=O)NO
COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](O[C@H]5C[C@H](NCc6ccc(cc6)-c6cn(CCCCCCCC(=O)NO)nn6)[C@H](O)[C@H](C)O5)c4c(O)c3C(=O)c12)C(C)=O |r|
COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](O[C@H]5C[C@H](NCc6ccc(cc6)-c6cn(CCCCCCC(=O)NO)nn6)[C@H](O)[C@H](C)O5)c4c(O)c3C(=O)c12)C(C)=O |r|
COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](O[C@H]5C[C@H](NCc6ccc(cc6)-c6cn(CCCCCC(=O)NO)nn6)[C@H](O)[C@H](C)O5)c4c(O)c3C(=O)c12)C(C)=O |r|
COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](O[C@H]5C[C@H](NCc6ccc(cc6)-c6cn(CCCCC(=O)NO)nn6)[C@H](O)[C@H](C)O5)c4c(O)c3C(=O)c12)C(C)=O |r|
COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](O[C@H]5C[C@H](NCc6ccc(NC(=O)CCCCCCC(=O)NO)cc6)[C@H](O)[C@H](C)O5)c4c(O)c3C(=O)c12)C(C)=O |r|
CSCCNC(=O)C(Cc1ccc(O)c(Br)c1)=NN |w:17.18|
COc1cc(CC(N=O)C(=O)NCCS)ccc1SC
SCCNC(=O)C(Cc1ccccc1)N=O
Oc1ccc(CC(N=O)C(=O)NCCS)cc1
Fc1ccc(CC(N=O)C(=O)NCCS)cc1
CSc1ccc(CC(N=O)C(=O)NCCS)cc1
COc1ccc(CC(N=O)C(=O)NCCS)cc1I
Fc1ccc(CC(N=O)C(=O)NCCS)cc1Br
CSc1ccc(CC(N=O)C(=O)NCCS)cc1Br
COc1cc(CC(N=O)C(=O)NCCS)cc(I)c1OC
COc1cc(CC(N=O)C(=O)NCCS)cc(Br)c1OC
COc1ccc(CC(N=O)C(=O)NCCS)cc1OC
[O-][N+](=O)c1cccc(CC(N=O)C(=O)NCCS)c1
[O-][N+](=O)c1cc(Br)cc(CC(N=O)C(=O)NCCS)c1
Oc1c(Br)cc(CC(N=O)C(=O)NCCS)cc1Br
CN(C)c1ccc(CC(N=O)C(=O)NCCS)cc1
CN(C)c1ccc(CC(N=O)C(=O)NCCS)cc1Br
CSCCNC(=O)C(Cc1ccc(O)c(Br)c1)N=O
COc1ccc(CC(N=O)C(=O)NCCSC)cc1Br
Oc1ccc(CC(N=O)C(=O)NCCSSCCNC(=O)C(Cc2ccc(O)c(Br)c2)N=O)cc1Br
COc1ccc(CC(N=O)C(=O)NCCSSCCNC(=O)C(Cc2ccc(OC)c(Br)c2)N=O)cc1Br
Oc1ccc(CC(N=O)C(=O)NCCS)cc1Br
COc1ccc(CC(N=O)C(=O)NCCS)cc1Br
CO\N=C(/Cc1ccc(O)c(Br)c1)C(=O)NCCSC
CO\N=C(/Cc1ccc(OC)c(Br)c1)C(=O)NCCSC
CO\N=C(/Cc1ccc(O)c(Br)c1)C(=O)NCCSSCCNC(=O)C(\Cc1ccc(O)c(Br)c1)=N\OC
CO\N=C(/Cc1ccc(OC)c(Br)c1)C(=O)NCCSSCCNC(=O)C(\Cc1ccc(OC)c(Br)c1)=N\OC
CO\N=C(/Cc1ccc(O)c(Br)c1)C(=O)NCCS
CO\N=C(/Cc1ccc(OC)c(Br)c1)C(=O)NCCS
CSCCNC(=O)C(=O)Cc1ccc(O)c(Br)c1
COc1ccc(CC(=O)C(=O)NCCSC)cc1Br
Oc1ccc(CC(=O)C(=O)NCCSSCCNC(=O)C(=O)Cc2ccc(O)c(Br)c2)cc1Br
COc1ccc(CC(=O)C(=O)NCCSSCCNC(=O)C(=O)Cc2ccc(OC)c(Br)c2)cc1Br
Oc1ccc(CC(=O)C(=O)NCCS)cc1Br
COc1ccc(CC(=O)C(=O)NCCS)cc1Br
COc1ccc(CC(=NN)C(=O)NCCSC)cc1Br |w:8.8|
NN=C(Cc1ccc(O)c(Br)c1)C(=O)NCCSSCCNC(=O)C(Cc1ccc(O)c(Br)c1)=NN |w:1.0,34.36|
COc1ccc(CC(=NN)C(=O)NCCSSCCNC(=O)C(Cc2ccc(OC)c(Br)c2)=NN)cc1Br |w:8.8,33.34|
NN=C(Cc1ccc(O)c(Br)c1)C(=O)NCCS |w:1.0|
COc1ccc(CC(=NN)C(=O)NCCS)cc1Br |w:8.8|
Oc1ccc(CC(=C)C(=O)NCCSSCCNC(=O)C(=C)Cc2ccc(O)c(Br)c2)cc1Br
Oc1ccc(CC(=C)C(=O)NCCS)cc1Br
ONC(=O)CCNC(=O)C(Cc1ccc(O)c(Br)c1)N=O
ONC(=O)CCCNC(=O)C(Cc1ccc(O)c(Br)c1)N=O
C(CP(CCC(=O)O)CCC(=O)O)C(=O)O
ONC(=O)\C=C\c1ccc2n(ccc2c1)S(=O)(=O)c1ccccc1
COc1ccc(cc1)S(=O)(=O)n1ccc2cc(\C=C\C(=O)NO)ccc12
COc1ccc(cc1OC)S(=O)(=O)n1ccc2cc(\C=C\C(=O)NO)ccc12
ONC(=O)\C=C\c1ccc2n(ccc2c1)S(=O)(=O)c1ccc(F)cc1
ONC(=O)\C=C\c1ccc2n(ccc2c1)S(=O)(=O)c1ccc(cc1)[N+]([O-])=O
ONC(=O)\C=C\c1ccc2n(Cc3ccccc3)ccc2c1
CC1(C)N(Cc2c1cccc2C(N)=O)c1cnc(cn1)C(F)(F)F
ONC(=O)c1nc2CCN(CCCNC(=O)CCC=C)Cc2s1
ONC(=O)c1nc2CCN(Cc2s1)C(=O)c1ccc(NC(=O)CCC=C)cc1
COc1ccc(\C=C\C(=O)Nc2ccc(cc2)C(=O)N2CCc3nc(sc3C2)C(=O)NO)cc1
ONC(=O)c1nc2CCN(Cc2s1)C(=O)c1ccc(NC(=O)c2ccc(s2)-c2ccccc2)cc1
ONC(=O)c1nc2CCN(CCCNC(=O)\C=C\c3ccccc3)Cc2s1
COc1ccc(\C=C\C(=O)NCCCN2CCc3nc(sc3C2)C(=O)NO)cc1
ONC(=O)c1nc2CCN(CCCNC(=O)c3ccc(s3)-c3ccccc3)Cc2s1
ONC(=O)c1nc2CCN(CCCCNC(=O)CCC=C)Cc2s1
ONC(=O)c1nc2CCN(CCCCNC(=O)\C=C\c3ccccc3)Cc2s1
COc1ccc(\C=C\C(=O)NCCCCN2CCc3nc(sc3C2)C(=O)NO)cc1
ONC(=O)c1nc2CCN(CCCCNC(=O)c3ccc(s3)-c3ccccc3)Cc2s1
CC(N1CCc2nc(sc2C1)C(=O)NO)c1ccc(NC(=O)CCC=C)nc1
CC(N1CCc2nc(sc2C1)C(=O)NO)c1ccc(NC(=O)\C=C\c2ccccc2)nc1
COc1ccc(\C=C\C(=O)Nc2ccc(cn2)C(C)N2CCc3nc(sc3C2)C(=O)NO)cc1
CC(N1CCc2nc(sc2C1)C(=O)NO)c1ccc(NC(=O)c2ccc(s2)-c2ccccc2)nc1
CC(C)N(C(=O)\C=C\c1ccccc1)c1cccc(CN2CCc3nc(sc3C2)C(=O)NO)c1
CCC[C@@H]1NC(=O)[C@H](C)NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2cn(CN(C)C)c3ccccc23)NC1=O |r|
CCC[C@@H]1NC(=O)[C@H](C)NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O |r|
CCCCCCC(=O)Nc1ccc(cc1)-c1cc(no1)C(=O)NCc1ccc(cc1)C(=O)NO
CC(C)(C)OC(=O)Nc1ccc(cc1)-c1cc(no1)C(=O)NCc1ccc(cc1)C(=O)NO
CC(C)(C)OC(=O)Nc1cccc(c1)-c1cc(no1)C(=O)NCc1ccc(cc1)C(=O)NO
CCCCCCC(=O)Nc1cccc(c1)-c1cc(no1)C(=O)NCc1ccc(cc1)C(=O)NO
c1ccc(cc1)CCOc2cccc(c2)Nc3ccccc3C(=O)N
CC(=O)SCCCCC[C@@H]1NC(=O)[C@H]2CCCN2C(=O)[C@H](CCOCCSC(C)=O)NC(=O)C(C)(C)NC1=O |r|
CC(=O)SCCCCC[C@@H]1NC(=O)[C@H]2CCCN2C(=O)[C@H](CCCCCSC(C)=O)NC(=O)C(C)(C)NC1=O |r|
O=C1N[C@H]2CCCCCSSCCOCC[C@@H](NC2=O)C(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCC[C@H]12 |r|
CC(=O)SCCCCC[C@@H]1NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](CCOCCSC(C)=O)NC1=O |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](CCCN=C(N)N)NC(=O)CCN(CC=C(C)C)C(=O)CN(CCc2c[nH]c3ccccc23)C1=O |r,wU:13.13,9.8,(56.09,-30.64,;54.73,-29.9,;53.42,-30.71,;53.46,-32.24,;52.07,-29.97,;50.75,-30.77,;49.4,-30.04,;48.09,-30.84,;46.73,-30.11,;45.52,-31.06,;44.06,-30.63,;43.65,-29.12,;44.6,-27.91,;41.81,-29.09,;40.95,-27.82,;39.42,-27.75,;38.63,-26.44,;37.11,-26.47,;36.31,-25.15,;37.06,-23.76,;34.83,-25.16,;41.35,-30.56,;39.92,-31.09,;38.65,-30.21,;39.92,-32.61,;41.35,-33.06,;41.36,-34.54,;40.03,-35.31,;38.69,-34.53,;37.36,-35.3,;36.03,-34.53,;37.36,-36.84,;42.79,-35.04,;42.82,-36.58,;44,-34.54,;43.97,-33.06,;44.73,-34.39,;44.72,-35.93,;46.05,-36.7,;47.45,-36.09,;48.48,-37.24,;47.7,-38.57,;48.16,-40.02,;47.14,-41.16,;45.63,-40.83,;45.17,-39.37,;46.2,-38.24,;45.59,-32.74,;46.92,-33.78,)|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](CCCCNC(C)=O)NC(=O)CCN(CC(C)C)C(=O)CN(CCc2c[nH]c3ccccc23)C1=O |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](CCCN=C(N)N)NC(=O)CCN(CC(C)C)C(=O)CN(CCc2c[nH]c3ccccc23)C1=O |r,wU:13.13,9.8,(44.46,-8.52,;43.11,-7.79,;41.79,-8.59,;41.83,-10.13,;40.44,-7.86,;39.13,-8.66,;37.77,-7.92,;36.46,-8.73,;35.11,-7.99,;33.89,-8.94,;32.43,-8.52,;32.02,-7.01,;32.97,-5.79,;30.18,-6.98,;29.32,-5.7,;27.79,-5.64,;27,-4.32,;25.48,-4.36,;24.68,-3.04,;25.43,-1.64,;23.2,-3.05,;29.72,-8.45,;28.29,-8.98,;27.03,-8.09,;28.29,-10.5,;29.73,-10.95,;29.73,-12.43,;28.4,-13.19,;27.07,-12.42,;25.73,-13.19,;27.07,-10.88,;31.17,-12.93,;31.19,-14.47,;32.37,-12.43,;32.35,-10.95,;33.1,-12.27,;33.1,-13.81,;34.43,-14.59,;35.82,-13.97,;36.85,-15.12,;36.07,-16.46,;36.54,-17.91,;35.51,-19.04,;34,-18.72,;33.54,-17.25,;34.57,-16.12,;33.96,-10.62,;35.29,-11.66,)|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](C)N(C)C(=O)CCN(CC(C)C)C(=O)CN(CCc2c[nH]c3ccccc23)C1=O |r|
CN1C[C@H]([C@@H](C1)c1ccc(\C=C\C(=O)Nc2ccccc2N)cc1)C(=O)Nc1ccc(Cl)cc1 |r|
CN1C[C@@H]([C@H](C1)c1ccc(\C=C\C(=O)Nc2ccccc2N)cc1F)C(=O)Nc1ccc(Cl)cc1 |r|
CN1C[C@@H]([C@H](C1)c1ccc(\C=C\C(=O)Nc2ccccc2N)cc1)C(=O)Nc1ccc(Cl)cc1 |r|
CNC(=O)c1ccc(Nc2c[nH]c3ccccc23)cc1
CNC(=O)c1ccc(Nc2csc3ccccc23)cc1
c1ccc(cc1)SCn2cc(nn2)c3cccc(c3)C(=O)NO
ONC(=O)c1cccc(c1)-c1cn(CCc2ccsc2)nn1
ONC(=O)c1cccc(c1)-c1cn(CCc2ccccc2)nn1
ONC(=O)c1cccc(c1)-c1cn(Cc2ccccc2)nn1
CC(C)(C)C(CCCCC(=O)NO)CC(=O)Nc1ccccc1
CCCCN(C(=O)Nc1cccc(c1)N(C)C)c1ccc(cc1)C(=O)NO
CCCCN(Cc1ccc(cc1)C(=O)NO)C(=O)Nc1cc(C)ccn1
OCCCCN(Cc1ccc(cc1)C(=O)NO)C(=O)Nc1ccccc1
CC(C)OC(=O)N(CCc1ccccc1)Cc1ccc(cc1)C(=O)NO
CCCCN(Cc1ccc(cc1)C(=O)NO)C(=O)NCCN1CCCC1
CC(C)CN(Cc1ccc(cc1)C(=O)NO)C(=O)Nc1ccccc1
CCCCN(Cc1ccc(cc1)N(O)C=O)C(=O)Nc1ccccc1
COc1ccc(cn1)-c1nc(N2CCOCC2)c2sc(CN(C)c3ccc(cc3)C(=O)NO)cc2n1
COc1ncc(cc1F)-c1cc(OCCCCCCC(=O)NO)c2ncnc(C)c2c1
ONC(=O)c1cccc(Cn2cncn2)c1
ONC(=O)c1ccc(Cn2cncn2)cc1
ONC(=O)c1ccc(Cn2cnc(Br)n2)cc1
ONC(=O)c1ccc(Cn2cnc(n2)-c2ccccc2)cc1
ONC(=O)c1ccc(Cn2cnc(n2)-c2ccccc2F)cc1
ONC(=O)c1ccc(Cn2cnc(n2)-c2cccc(F)c2)cc1
ONC(=O)c1ccc(Cn2cnc(n2)-c2ccc(F)cc2)cc1
ONC(=O)c1ccc(Cn2cnc(n2)-c2c(F)cccc2F)cc1
ONC(=O)c1ccc(Cn2cnc(n2)-c2cc(F)cc(F)c2)cc1
ONC(=O)c1ccc(Cn2cnc(n2)-c2cccc(Cl)c2)cc1
Cc1cccc(c1)-c1ncn(Cc2ccc(cc2)C(=O)NO)n1
ONC(=O)c1ccc(Cn2cnc(n2)-c2cccc(c2)C(F)(F)F)cc1
ONC(=O)c1ccc(Cn2cnc(n2)-c2cccc(OC(F)(F)F)c2)cc1
COc1cccc(c1)-c1ncn(Cc2ccc(cc2)C(=O)NO)n1
ONC(=O)c1ccc(Cn2cnc(n2)-c2cccc(O)c2)cc1
ONC(=O)c1ccc(Cn2cnc(n2)-c2cccc(c2)-c2ccccc2)cc1
ONC(=O)c1ccc(Cn2cnc(n2)-c2cccnc2)cc1
ONC(=O)c1ccc(Cn2cnc(n2)-c2cccs2)cc1
ONC(=O)c1ccc(Cn2cnc(n2)-c2ccccc2)c(F)c1
ONC(=O)c1ccc(Cn2cnc(n2)-c2ccccc2)nc1
ONC(=O)c1ccc(Cn2cnc(n2)-c2ccccc2F)c(F)c1
ONC(=O)c1cccc(Cn2cnc(n2)-c2ccccc2)c1
ONC(=O)c1cccc(Cn2ncnc2-c2ccccc2)c1
ONC(=O)c1ccc(Cn2ncnc2-c2ccccc2)cc1
ONC(=O)c1ccc(Cn2ncnc2-c2ccccc2F)cc1
ONC(=O)c1ccc(Cn2ncnc2-c2cccs2)cc1
ONC(=O)c1ccc(CCN2C(=O)c3cccc4c(ccc(C2=O)c34)N2CCOCC2)cc1
ONC(=O)c1ccc(CN2C(=O)c3cccc4c(ccc(C2=O)c34)N2CCOCC2)cc1
ONC(=O)CCCCCN1C(=O)c2cccc3c(ccc(C1=O)c23)N1CCOCC1
CN(C)c1ccc(NC(=O)NCCCCNC(=O)CS)cc1
NCC(=O)Nc1ccccc1-c1ccc(NC(=O)CCCCCNC(=O)CS)cc1
N[C@@H](Cc1ccccc1)C(=O)Nc1ccccc1-c1ccc(NC(=O)CCCCCNC(=O)CS)cc1 |r|
SCC(=O)NCCCCCC(=O)Nc1ccc(cc1)-c1ccccc1NC(=O)[C@@H]1CCCN1 |r|
N[C@@H](Cc1c[nH]c2ccccc12)C(=O)Nc1ccccc1-c1ccc(NC(=O)CCCCCNC(=O)CS)cc1 |r|
Cc1onc(c1C(=O)NCCCCCNC(=O)CS)-c1ccccc1
CC(S)C(=O)NCCCCCNC(=O)c1c(C)onc1-c1ccccc1
C[C@@H](S)C(=O)NCCCCCNC(=O)c1c(C)onc1-c1ccccc1 |r|
C[C@H](S)C(=O)NCCCCCNC(=O)c1c(C)onc1-c1ccccc1 |r|
Cc1onc(c1C(=O)NCCCCCNC(=O)C(C)(C)S)-c1ccccc1
CC(S)C(=O)NCCCCCOCc1c(C)onc1-c1ccccc1
C[C@@H](S)C(=O)NCCCCCOCc1c(C)onc1-c1ccccc1 |r|
C[C@H](S)C(=O)NCCCCCOCc1c(C)onc1-c1ccccc1 |r|
Cc1onc(c1C=CCCCCCNC(=O)CS)-c1ccccc1
Cc1onc(c1\C=C/CCCCCNC(=O)CS)-c1ccccc1
Cc1onc(c1\C=C\CCCCCNC(=O)CS)-c1ccccc1
CC(S)C(=O)NCCCCCC=Cc1c(C)onc1-c1ccccc1
Cc1onc(c1C=CCCCCCNC(=O)C(C)(C)S)-c1ccccc1
CC(S)C(=O)NCc1ccc(\C=C\c2c(C)onc2-c2ccccc2)cc1
Cc1onc(c1\C=C\c1ccc(CNC(=O)C(C)(C)S)cc1)-c1ccccc1
CC(S)C(=O)NCCCCCC#Cc1c(C)noc1-c1ccccc1
CC(S)C(=O)NCCCCCC#Cc1c(C)noc1-c1cccc(F)c1
Cc1noc(c1C#CCCCCCNC(=O)C(C)(C)S)-c1ccccc1
Cc1noc(c1C#CCCCCNC(=O)C(C)(C)S)-c1ccccc1
c1ccc(c(c1)/C=C/C(=O)NO)Cl
COc1cc2ccn(CCOc3cccc(NC(=O)CCCCCCC(=O)NO)c3)c2c(OC)c1OC
COc1cc2ccn(CCCCOc3cccc(NC(=O)CCCCCCC(=O)NO)c3)c2c(OC)c1OC
COc1ccc2n(CCOc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)ccc2c1
COc1cc2ccn(CCOc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)c2cc1OC
NCCCCNCCCCNCCCn1c(=O)c2ccc3c4c(ccc(c24)c1=O)c(=O)n(CCCCCC(=O)NO)c3=O
ONC(=O)CCCCCCN(Cc1ccc(F)cc1)c1ncc(s1)C(=O)NCCCn1ccnc1
CC(C)CCN(CCCCCCC(=O)NO)c1ncc(s1)C(=O)NCCCn1ccnc1
CN1CCC2(CC1)C(N(Cc1ccc(cc1)C(=O)NO)c1ccccc21)c1ccccc1
CN1CCC2(CC1)C(N(Cc1ccc(cc1)C(=O)NO)c1ccccc21)c1ccc(Cl)cc1
CN1CCC2(CC1)C(N(Cc1ccc(cc1)C(=O)NO)c1ccccc21)c1cccc(Cl)c1
CN1CCC2(CC1)C(N(Cc1ccc(cc1)C(=O)NO)c1ccccc21)c1ccccc1F
CN1CCC2(CC1)C(N(Cc1ccc(cc1)C(=O)NO)c1ccccc21)c1ccc(F)cc1
CN1CCC2(CC1)C(N(Cc1ccc(cc1)C(=O)NO)c1ccccc21)c1cccnc1
CC1(C)C(N(Cc2ccc(cc2)C(=O)NO)c2ccccc12)c1ccccc1
CC1(C)C(N(Cc2ccc(cc2)C(=O)NO)c2ccccc12)c1cccnc1
CC1(C)[C@@H](N(Cc2ccc(cc2)C(=O)NO)c2ccccc12)c1cccnc1 |r|
CC1(c2ccccc2N([C@@H]1c3cccnc3)Cc4ccc(cc4)C(=O)NO)C
COc1ccc2N(Cc3ccc(cc3)C(=O)NO)C(c3cccnc3)C(C)(C)c2c1
CC1(C)C(N(Cc2ccc(s2)C(=O)NO)c2ccccc12)c1cccnc1
CC1(C)C(N(Cc2ccc(OCCCC(=O)NO)cc2)c2ccccc12)c1cccnc1
CC1(C)C(N(Cc2ccc(cc2)C(=O)NO)c2ccccc12)c1ccncc1
CC(C)(C)OC(=O)N1CCC2(CC1)C(N(Cc1ccc(cc1)C(=O)NO)c1ccccc21)c1cccnc1
COc1cccc(c1)-n1nc(nc1-c1cc(OC)c(OC)c(OC)c1)C(=O)NCCCCCC(=O)NO
COc1cccc(c1)-n1nc(nc1-c1cc(OC)c(OC)c(OC)c1)C(=O)NCC(=O)NO
ONC(=O)CCCCCCN1C(=O)NC2(CCCc3ccccc23)C1=O
Cc1cc(C)cc(c1)C(=O)NOCCCCCC(=O)NO
Cc1ccc(cc1C)C(=O)NOCCCCCC(=O)NO
Cc1cccc(c1)C(=O)NOCCCCCC(=O)NO
CC(C)[C@H]1NC(=O)[C@H]2CSSCC\C=C\[C@H](CC(=O)N[C@H](C(C)C)C(=O)N2)OC(=O)C[C@@H]1O |r,t:13|
CC[C@H](C)[C@H]1NC(=O)[C@H]2CSSCC\C=C\[C@H](CC(=O)N[C@H](CCS(C)=O)C(=O)N2)OC(=O)C[C@@H]1O |r,t:14|
C1CC=C(C1)C(=O)NO
C1CCC(CC1)C(=O)NO
C1CCC(=CC1)C(=O)NO
ONC(=O)CCc1ccccc1
ONC(=O)Cc1ccccc1
c1ccc(cc1)C(=O)NO
CNC(=O)c1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(cc1)C(=O)Nc1ccccc1
ONC(=O)c1ccc(cc1)C(=O)NCc1ccccc1
ONC(=O)c1ccc(cc1)C(=O)NCCc1ccccc1
ONC(=O)c1ccc(cc1)C(=O)NCCc1ccncc1
CN1CCN(CCNC(=O)c2ccc(cc2)C(=O)NO)CC1
Oc1cccn(Cc2ccc(cc2C#N)-c2ccccc2)c1=S
ONC(=O)c1cccc(c1)S(=O)(=O)NCc1ccccc1
CC(C)[C@H](NS(=O)(=O)c1cccc(c1)C(=O)NO)C(=O)Nc1ccccc1 |r|
ONC(=O)c1cccc(c1)S(=O)(=O)Nc1ccccc1
ONC(=O)c1cccc(c1)S(=O)(=O)NCC(=O)Nc1ccccc1
C[C@H](NS(=O)(=O)c1cccc(c1)C(=O)NO)C(=O)Nc1ccccc1 |r|
ONC(=O)c1cccc(c1)S(=O)(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCc1ccccc1 |r|
ONC(=O)c1cccc(c1)S(=O)(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)Nc1ccccc1 |r|
ONC(=O)c1cccc(c1)S(=O)(=O)N[C@H](C(=O)Nc1ccccc1)c1ccccc1 |r|
ONC(=O)c1cccc(c1)S(=O)(=O)NCCc1ccccc1
ONC(=O)c1cccc(c1)S(=O)(=O)N[C@H](C(=O)NCc1ccccc1)c1ccccc1 |r|
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(Cc2ccc(s2)C(=O)NO)ccc1OCC
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(Cc2ccc(cc2OC)C(=O)NO)ccc1OCC
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)C(OC)c1ccc(cc1)C(=O)NO
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)-c1ccc(cc1)C(=O)NO
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)C1=CCC(CC(=O)NO)CC1 |t:26|
CCCc1nc(C)c2n1nc([nH]c2=O)-c1cc(Cc2ccc(s2)C(=O)NO)ccc1OCC
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)C(O)c1ccc(cc1)C(=O)NO
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)-c1ccc(CC(=O)NO)cc1
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)C1CCC(CC1)C(=O)NO |(28.33,-20.2,;27.93,-18.71,;26.43,-18.39,;25.95,-16.92,;26.86,-15.68,;25.95,-14.43,;26.43,-12.97,;24.49,-14.91,;24.49,-16.45,;23.15,-17.22,;21.82,-16.45,;21.82,-14.91,;23.15,-14.14,;23.15,-12.6,;20.49,-17.22,;20.49,-18.76,;19.15,-19.53,;17.82,-18.76,;17.82,-17.22,;19.15,-16.45,;19.15,-14.91,;17.82,-14.14,;17.82,-12.6,;19.15,-21.07,;20.49,-21.84,;20.49,-23.38,;19.15,-24.15,;17.82,-23.38,;17.82,-21.84,;19.15,-25.69,;20.49,-26.46,;17.82,-26.46,;16.48,-25.69,)|
CC[C@H](C)C(=O)O[C@H]1C[C@@H](C)C=C2C=C[C@H](C)[C@H](CC[C@@H](O)C[C@@H](O)CC(=O)NO)[C@@H]12 |r,c:13,t:11|
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(Cc2ccc(cc2)C(=O)NO)ccc1OCC
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(Cc2ccc(CC(=O)NO)cc2)ccc1OCC
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(Cc2ccc(C(=O)NO)c(OC)c2)ccc1OCC
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(Cc2ccc(C(=O)NO)c(F)c2)ccc1OCC
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(Cc2ccc(cc2F)C(=O)NO)ccc1OCC
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(OCc2ccc(cc2)C(=O)NO)ccc1OCC
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(Cc2ccc(o2)C(=O)NO)ccc1OCC
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)C(=O)c1ccc(s1)C(=O)NO
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)-c1ccc(s1)C(=O)NO
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)C1=CCC(CC1)C(=O)NO |t:26|
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)[C@@H]1CC[C@@H](CC1)C(=O)NO |r,wD:26.32,23.25,(29.43,-23.41,;29.03,-21.92,;27.53,-21.6,;27.05,-20.14,;27.96,-18.89,;27.05,-17.64,;27.53,-16.18,;25.59,-18.12,;25.59,-19.66,;24.25,-20.43,;22.92,-19.66,;22.92,-18.12,;24.25,-17.35,;24.25,-15.81,;21.58,-20.43,;21.58,-21.97,;20.25,-22.74,;18.92,-21.97,;18.92,-20.43,;20.25,-19.66,;20.25,-18.12,;18.92,-17.35,;18.92,-15.81,;20.25,-24.28,;21.58,-25.05,;21.58,-26.59,;20.25,-27.36,;18.92,-26.59,;18.92,-25.05,;20.25,-28.9,;21.58,-29.67,;18.92,-29.67,;17.58,-28.9,)|
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)[C@H]1CC[C@@H](CC1)C(=O)NO |r,wU:26.32,wD:23.25,(29.43,-23.41,;29.03,-21.92,;27.53,-21.6,;27.05,-20.14,;27.96,-18.89,;27.05,-17.64,;27.53,-16.18,;25.59,-18.12,;25.59,-19.66,;24.25,-20.43,;22.92,-19.66,;22.92,-18.12,;24.25,-17.35,;24.25,-15.81,;21.58,-20.43,;21.58,-21.97,;20.25,-22.74,;18.92,-21.97,;18.92,-20.43,;20.25,-19.66,;20.25,-18.12,;18.92,-17.35,;18.92,-15.81,;20.25,-24.28,;18.92,-25.05,;18.92,-26.59,;20.25,-27.36,;21.58,-26.59,;21.58,-25.05,;20.25,-28.9,;21.58,-29.67,;18.92,-29.67,;17.58,-28.9,)|
CCCc1nc(C)c2n1nc([nH]c2=O)-c1cc(Cc2ccc(cc2)C(=O)NO)ccc1OCC
CCCc1nc(C)c2n1nc([nH]c2=O)-c1cc(ccc1OCC)-c1ccc(cc1)C(=O)NO
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(ccc1OCC)N1CCC(CC1)C(=O)NO
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(Nc2ccc(cc2)C(=O)NO)ccc1OCC
CCCc1nc(C)c2n1nc([nH]c2=O)-c1cc(CC2CC(C2)C(=O)NO)ccc1OCC |(23.21,-13.66,;22.75,-12.19,;21.24,-11.86,;20.77,-10.39,;21.69,-9.15,;20.79,-7.9,;21.28,-6.44,;19.32,-8.37,;19.31,-9.91,;17.99,-10.68,;16.66,-9.91,;16.65,-8.37,;17.99,-7.6,;17.99,-6.06,;15.32,-10.68,;15.33,-12.23,;13.99,-13,;13.99,-14.54,;15.32,-15.31,;15.72,-16.79,;17.21,-16.4,;16.81,-14.91,;18.53,-17.17,;19.87,-16.4,;18.53,-18.71,;17.2,-19.47,;12.66,-12.23,;12.66,-10.69,;13.99,-9.92,;13.98,-8.38,;12.65,-7.61,;12.64,-6.07,)|
COc1cc(cc(OC)c1OC)C(=O)c1ccc2n(ccc2c1)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1
COc1ccc(cc1OC)C(=O)c1ccc2n(Cc3ccc(cc3)C(=O)NO)ccc2c1
COc1cc(cc(OC)c1OC)C(=O)c1ccc2n(Cc3ccc(cc3)C(=O)NO)ccc2c1
Cc1ccc(cc1)C(=O)c1ccc2n(Cc3ccc(cc3)C(=O)NO)ccc2c1
COc1ccc(cc1OC)C(=O)c1ccc2n(ccc2c1)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1
Cc1ccc(cc1)C(=O)c1ccc2n(ccc2c1)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1
COc1cc(cc(OC)c1OC)C(=O)c1ccc2n(ccc2c1)S(=O)(=O)c1ccc(\C=C\C(=O)NO)cc1
COc1cc(cc(OC)c1OC)C(=O)c1ccc2n(Cc3ccc(\C=C\C(=O)NO)cc3)ccc2c1
ONC(=O)c1ccc(Cn2ccc3cc(ccc23)C(=O)c2ccc(F)cc2)cc1
COc1ccc(cc1)C(=O)c1ccc2n(Cc3ccc(cc3)C(=O)NO)ccc2c1
ONC(=O)\C=C\c1cccc(c1)S(=O)(=O)n1ccc2cc(ccc12)C(=O)c1ccc(F)cc1
ONC(=O)c1ccc(Cn2ccc3cc(ccc23)C(=O)c2ccc(Cl)cc2)cc1
COc1ccc(cc1)C(=O)c1ccc2n(ccc2c1)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1
COc1ccc(cc1)C(=O)c1ccc2n(Cc3ccc(\C=C\C(=O)NO)cc3)ccc2c1
COc1cccc(c1)C(=O)c1ccc2n(Cc3ccc(cc3)C(=O)NO)ccc2c1
COc1cccc(c1)C(=O)c1ccc2n(ccc2c1)S(=O)(=O)c1cccc(\C=C\C(=O)NO)c1
COc1ccc(cc1)C(=O)c1ccc2n(ccc2c1)S(=O)(=O)c1ccc(\C=C\C(=O)NO)cc1
ONC(=O)CCCCCn1cc(nn1)-c1ccc2ncnc(Nc3ccc(Br)cc3F)c2c1
CC(=O)Nc1ccc(cc1)-c1ccnc(NCc2ccc(OCCCCCC(=O)NO)cc2)n1
CS(=O)(=O)Nc1ccc(cc1)-c1ccnc(Nc2ccc(cc2)N2CCC(CCc3ccc(\C=C\CC(=O)NO)cc3)CC2)n1
CN(C)C1=NC2C(N1CCCCCC(=O)NO)C(Br)=C(Br)C(Br)=C2Br |c:23,t:3,19|
COc1c(OCCCCCC(=O)NO)ccc2C3=NCCN3C(NC(=O)c3ccccc3)=Nc12 |c:33,t:17|
CSCC[C@@H]1NC(=O)C[C@@H]2OC(=O)C[C@@H](O)[C@@H](NC(=O)[C@@H](CSSCC\C=C\2)NC1=O)C(C)C |r,t:26|
CSCC[C@H]1NC(=O)C[C@@H]2OC(=O)C[C@H](O)[C@H](NC(=O)[C@@H](CSSCC\C=C\2)NC1=O)C(C)C |r,t:26|
CS(=O)(=O)Nc1ccc(cc1)-c1ccnc(Nc2ccc(cc2)N2CCC(CC2)C(=O)NCCCCCCCC(=O)NO)n1
CS(=O)(=O)Nc1ccc(cc1)-c1ccnc(Nc2ccc(cc2)N2CCC(CC2)C(=O)Nc2ccc(\C=C\C(=O)NO)cc2)n1
ONC(=O)c1ccc(cc1)-c1ccnc(Nc2ccc(cc2)N2CCOCC2)n1
Cc1ccc(cc1)NC(=O)CN(Cc2ccc(cc2)C(=O)NO)C(=O)c3ccc(cc3)N(C)C
Cc1cc(cc(c1)C(=O)N(Cc2ccc(cc2)C(=O)NO)CC(=O)NC3CCCCC3)C
CN(C)c1ccc(cc1)C(=O)N(Cc2ccc(cc2)C(=O)NO)CC(=O)NCc3ccccc3
CCOc1cc(ccc1C1=NC(C(N1C(=O)N1CCN(CCCCCCC(=O)NO)CC1)c1ccc(Cl)cc1)c1ccc(Cl)cc1)C(C)(C)C |t:10|
c1cc2ccsc2c(c1)C(=O)Nc3cc(ccc3Cl)C(=O)NO
C[C@@H](C(=O)NCc1ccccc1)NC(=O)[C@H](CC(=O)NCC(C)(C)C)NC(=O)c2ccc(cc2)C(=O)NO
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)N(CCCl)CCCl
c1ccc2c(c1)c(c(s2)C(=O)NO)Cl
COc1cccc(c1)-c1ccc2c(NC(=O)c3ccc(cc3)C(=O)NO)n[nH]c2c1
ONC(=O)c1ccc(cc1)C(=O)Nc1n[nH]c2cc(ccc12)-c1ccc(cc1)C(F)(F)F
COc1cc(OC)cc(c1)-c1ccc2c(NC(=O)c3ccc(cc3)C(=O)NO)n[nH]c2c1
ONC(=O)c1ccc(cc1)C(=O)Nc1n[nH]c2cc(ccc12)-c1cccc(Cl)c1Cl
ONC(=O)c1ccc(cc1)C(=O)Nc1n[nH]c2cc(ccc12)-c1ccccc1F
COc1cccc(-c2ccc3c(NC(=O)c4ccc(cc4)C(=O)NO)n[nH]c3c2)c1F
CCOc1cccc(c1)-c1ccc2c(NC(=O)c3ccc(cc3)C(=O)NO)n[nH]c2c1
COc1ccccc1-c1ccc2c(NC(=O)c3ccc(cc3)C(=O)NO)n[nH]c2c1
ONC(=O)c1ccc(cc1)C(=O)Nc1n[nH]c2cc(ccc12)-c1cccc(OC(F)(F)F)c1
COc1ccc(cc1OC)-c1ccc2c(NC(=O)c3ccc(cc3)C(=O)NO)n[nH]c2c1
ONC(=O)c1ccc(cc1)C(=O)Nc1n[nH]c2cc(ccc12)-c1ccccc1
ONC(=O)c1ccc(cc1)C(=O)Nc1n[nH]c2cc(ccc12)-c1ccc(Cl)c(F)c1
ONC(=O)c1ccc(cc1)C(=O)Nc1n[nH]c2cc(ccc12)-c1cc(Cl)cc(Cl)c1
ONC(=O)c1ccc(cc1)C(=O)Nc1n[nH]c2cc(ccc12)-c1cc(Cl)ccc1Cl
COc1ccc(F)cc1-c1ccc2c(NC(=O)c3ccc(cc3)C(=O)NO)n[nH]c2c1
ONC(=O)c1ccc(cc1)C(=O)Nc1n[nH]c2cc(ccc12)-c1c(Cl)cccc1Cl
ONC(=O)c1ccc(cc1)C(=O)Nc1n[nH]c2cc(ccc12)-c1cccc(Cl)c1
Cc1cc(C)cc(c1)-c1ccc2c(NC(=O)c3ccc(cc3)C(=O)NO)n[nH]c2c1
ONC(=O)c1ccc(cc1)C(=O)Nc1n[nH]c2cc(ccc12)-c1ccc(Cl)cc1
CCCOc1cccc(c1)-c1ccc2c(NC(=O)c3ccc(cc3)C(=O)NO)n[nH]c2c1
CC(C)Oc1cccc(c1)-c1ccc2c(NC(=O)c3ccc(cc3)C(=O)NO)n[nH]c2c1
COc1ccc(cc1)-c1ccc2c(NC(=O)c3ccc(cc3)C(=O)NO)n[nH]c2c1
ONC(=O)c1ccc(cc1)C(=O)Nc1n[nH]c2cc(ccc12)-c1ccc(Cl)c(Cl)c1
ONC(=O)c1ccc(cc1)C(=O)Nc1n[nH]c2cc(ccc12)-c1ccccc1Cl
c1ccc2c(c1)C(=O)N(C=N2)CC(=O)O
COc1c(nc2ccccc2n1)CCC(=O)O
CN1C(=Nc2ccccc2C1=O)CCC(=O)O
c1ccc2c(c1)nc(s2)CCC(=O)O
OC(=O)Cn1nc(O)c2ccccc2c1=O
OC(=O)Cn1cnc2c(C#N)c3CCCCn3c2c1=O
Cc1cc(C)c2c(n1)sc1c2ncn(CC(O)=O)c1=O
COc1cc2ncn(CC(O)=O)c(=O)c2cc1OC
OC(=O)CCn1nnc2ccccc2c1=O
c1ccc2c(c1)nc(s2)CC(=O)O
NC(=O)c1cc(cs1)-n1c(CCC(O)=O)nc2ccccc12
c1ccc(cc1)CC2=NN3C(=Nc4ccccc4C3=NC2=O)CCC(=O)O
OC(=O)CCc1nc(O)c2ccccc2n1
COc1cc2ncn(CCC(O)=O)c(=O)c2cc1OC
Cn1c(CCC(O)=O)nc2ccccc12
c1ccc2c(c1)ccc(n2)CCC(=O)O
c1c2c(cc3c1nc(s3)CCC(=O)O)sc(n2)CCC(=O)O
OC(=O)Cn1cnc2ccc(Br)cc2c1=O
OC(=O)Cn1cnc2c3ccccc3oc2c1=O
OC(=O)CCc1nc2cc(Cl)ccc2n(Cc2ccccc2)c1=O
CN(c1ccc2c(C)n(C)nc2c1)c1ccnc(Nc2ccc(cc2)C(=O)NCCCCCCC(=O)NO)n1
CN(c1ccc2c(C)n(C)nc2c1)c1ccnc(Nc2ccc(\C=C\C(=O)NO)cc2)n1
Cc1cc(-c2ccc(F)cc2)n(Cc2ccc(cc2)C(=O)NO)n1
Cc1ccc(cc1)-c1cc(nn1-c1ccc(cc1)C(=O)NO)C(F)(F)F
Cc1cc(nn1Cc1ccc(cc1)C(=O)NO)-c1ccc2OCOc2c1
Cc1ccc(cc1)-c1cc(nn1Cc1ccc(cc1)C(=O)NO)C(F)(F)F
ONC(=O)CCCCCNC(=O)c1cc([nH]n1)-c1ccc(F)cc1
Cc1ccc(cc1)-c1cc(nn1-c1ccc(cc1)S(N)(=O)=O)C(F)(F)F
Cc1ccc(cc1)-c1cc(nn1CCc1ccc(cc1)C(=O)NO)C(F)(F)F
Cc1ccc(cc1)-c1cc(n(CCc2ccc(cc2)C(=O)NO)n1)C(F)(F)F
Cc1cc(-c2ccc(C)cc2)n(Cc2ccc(cc2)C(=O)NO)n1
Cc1cc(nn1Cc1ccc(cc1)C(=O)NO)-c1ccc(F)cc1
CCc1cc(-c2ccc(F)cc2)n(Cc2ccc(cc2)C(=O)NO)n1
CCCc1cc(-c2ccc(F)cc2)n(Cc2ccc(cc2)C(=O)NO)n1
CCCc1cc(nn1Cc1ccc(cc1)C(=O)NO)-c1ccc(F)cc1
ONC(=O)c1ccc(Cn2nc(Cc3ccccc3)cc2-c2ccc(F)cc2)cc1
ONC(=O)c1ccc(CNC(=O)c2cc([nH]n2)-c2ccc(F)cc2)cc1
ONC(=O)CCNC(=O)c1cc([nH]n1)-c1ccc(F)cc1
ONC(=O)CCCCNC(=O)c1cc([nH]n1)-c1ccc(F)cc1
ONC(=O)CCCCCCNC(=O)c1cc([nH]n1)-c1ccc(F)cc1
Cc1ccc(cc1)-c1cc(n(Cc2ccc(cc2)C(=O)NO)n1)C(F)(F)F
ONC(=O)c1ccc(Cn2nc(cc2Cc2ccccc2)-c2ccc(F)cc2)cc1
CCc1cc(nn1Cc1ccc(cc1)C(=O)NO)-c1ccc(F)cc1
Cc1cc(-c2ccc3OCOc3c2)n(Cc2ccc(cc2)C(=O)NO)n1
Cc1cc(nn1Cc1ccc(cc1)C(=O)NO)-c1ccc(C)cc1
ONC(=O)CCCNC(=O)c1cc([nH]n1)-c1ccc(F)cc1
ONC(=O)c1ccc(\C=C\C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)Nc2cccc(Cl)c2)cc1 |r|
Cc1ccc(NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(cc2)C(=O)NO)cc1 |r|
ONC(=O)c1ccc(\C=C\C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)Nc2ccc(Cl)cc2)cc1 |r|
ONC(=O)c1ccc(\C=C\C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)Nc2ccc(Br)cc2)cc1 |r|
Cc1cn([C@@H]2C[C@@H]([C@@H](CO[Si](C)(C)C(C)(C)C)O2)C2(SCCCS2)c2ccc(NC(=O)CCCCCC(=O)NO)cc2)c(=O)[nH]c1=O |r|
COc1ccc(cc1OC)C1(SCCCS1)[C@H]1C[C@@H](O[C@@H]1CO[Si](C)(C)C(C)(C)C)n1cc(C)c(=O)[nH]c1=O |r|
Cc1cn([C@@H]2C[C@@H]([C@@H](CO[Si](C)(C)C(C)(C)C)O2)C2(SCCCS2)c2ccc(NC(=O)CCCCCCC(=O)NO)cc2)c(=O)[nH]c1=O |r|
Cc1cn([C@H]2C[C@@H]([C@@H](CO[Si](C)(C)C(C)(C)C)O2)C2(SCCCS2)c2ccc(NC(=O)CCCCCC(=O)NO)cc2)c(=O)[nH]c1=O |r|
Cc1cn([C@@H]2C[C@@H]([C@@H](CO[Si](C)(C)C(C)(C)C)O2)C2(SCCCS2)c2ccc(NC(=O)CCCCC(=O)NO)cc2)c(=O)[nH]c1=O |r|
Cc1cn([C@H]2C[C@@H]([C@@H](CO[Si](C)(C)C(C)(C)C)O2)C2(SCCCS2)c2ccc(NC(=O)CCCCC(=O)NO)cc2)c(=O)[nH]c1=O |r|
Cc1cn([C@H]2C[C@@H]([C@@H](CO[Si](C)(C)C(C)(C)C)O2)C2(SCCCS2)c2ccc(NC(=O)CCCCCCC(=O)NO)cc2)c(=O)[nH]c1=O |r|
CCNC(=O)c1cc2c(nc(N)nc2s1)-c1cc(OCCCCCCn2cc(cn2)-c2nc(Nc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)nc3[nH]ccc23)c(Cl)cc1Cl
CCNC(=O)c1cc2c(nc(N)nc2s1)-c1cc(OCCCCCCn2cc(cn2)-c2nc(Nc3ccc(NC(=O)CCCCCCC(O)=O)cc3)nc3[nH]ccc23)c(Cl)cc1Cl
CCNC(=O)c1cc2c(nc(N)nc2s1)-c1cccc(OCCCCCCOc2ccc(Nc3nc(-c4cnn(CCCCCCC(=O)NO)c4)c4cc[nH]c4n3)cc2)c1
CC(C)c1cc(C(=O)N2CCc3cc(NC(=O)CCC(=O)NO)ccc23)c(O)cc1O
CC(C)c1cc(C(=O)N2CCc3cc(NCc4ccc(cc4)C(=O)NO)ccc23)c(O)cc1O
CC(C)c1cc(C(=O)N2CCc3cc(NC(=O)CCCC(=O)NO)ccc23)c(O)cc1O
CC(C)c1cc(C(=O)N2CCc3cc(NC(=O)CCCCC(=O)NO)ccc23)c(O)cc1O
CC(C)c1cc(C(=O)N2CCc3cc(NC(=O)CCCCCC(=O)NO)ccc23)c(O)cc1O
CC(C)c1cc(C(=O)N2CCc3cc(NC(=O)CCCCCCCCC(=O)NO)ccc23)c(O)cc1O
CC(C)c1cc(C(=O)N2CCc3cc(NC(=O)CCCCCCC(=O)NO)ccc23)c(O)cc1O
CC(C)c1cc(C(=O)N2CCc3cc(NC(=O)CCCCCCCC(=O)NO)ccc23)c(O)cc1O
ONC(=O)CCCCCCC(=O)Nc1ccc(Nc2nc(-c3cnn(CCCCCOc4ccccc4)c3)c3cc[nH]c3n2)cc1
ONC(=O)CCCCCCC(=O)Nc1ccc(Nc2nc(-c3cnn(CC4CCCC4)c3)c3cc[nH]c3n2)cc1
ONC(=O)CCCCCCC(=O)Nc1ccc(Nc2nc(-c3cnn(CCCCCCOc4ccccc4)c3)c3cc[nH]c3n2)cc1
ONC(=O)CCCCCCC(=O)Nc1ccc(Nc2nc(-c3cn[nH]c3)c3cc[nH]c3n2)cc1
CS(=O)(=O)CCn1cc(cn1)-c1nc(Nc2ccc(NC(=O)CCCCCCC(=O)NO)cc2)nc2[nH]ccc12
ONC(=O)CCCCCCC(=O)Nc1ccc(Nc2nc(-c3cnn(CCCCOc4ccccc4)c3)c3cc[nH]c3n2)cc1
COCCn1cc(cn1)-c1nc(Nc2ccc(NC(=O)CCCCCCC(=O)NO)cc2)nc2[nH]ccc12
CCCn1cc(cn1)-c1nc(Nc2ccc(NC(=O)CCCCCCC(=O)NO)cc2)nc2[nH]ccc12
ONC(=O)CCCCCCC(=O)Nc1ccc(Nc2nc(-c3cnn(CCC#N)c3)c3cc[nH]c3n2)cc1
ONC(=O)CCCCCCC(=O)Nc1ccc(Nc2nc(-c3cnn(CCC=C)c3)c3cc[nH]c3n2)cc1
COc1ccc2nc3cc(Cl)ccc3c(Nc3ccc(cc3)-c3cn(CCCCCC(=O)NO)nn3)c2c1
ONC(=O)CCc1ccc(Nc2c3ccccc3nc3ccccc23)cc1
ONC(=O)CCCCCn1cc(nn1)-c1cccc(Nc2c3ccccc3nc3ccccc23)c1
COc1ccc2nc3cc(Cl)ccc3c(Nc3ccc(CCC(=O)NO)cc3)c2c1
ONC(=O)CCCCCCn1cc(nn1)-c1cccc(Nc2c3ccccc3nc3ccccc23)c1
ONC(=O)CCCCCCn1cc(nn1)-c1ccc(Nc2c3ccccc3nc3ccccc23)cc1
ONC(=O)CCCCCn1cc(nn1)-c1ccc(Nc2c3ccccc3nc3ccccc23)cc1
COc1ccc2nc3cc(Cl)ccc3c(Nc3cccc(c3)-c3cn(CCCCCC(=O)NO)nn3)c2c1
CC\C(=C(/c1ccc(O)cc1)c1ccc(OCCN(C)C)cc1)c1ccc(CCC(=O)NO)cc1
CC\C(=C(/c1ccc(O)cc1)c1ccc(OCCN(C)C)cc1)c1ccc(cc1)C(=O)NO
CC\C(=C(/c1ccc(O)cc1)c1ccc(OCCN(C)C)cc1)c1ccc(\C=C\C(=O)NO)cc1
CC\C(=C(/c1ccc(O)cc1)c1ccc(OCCN(C)C)cc1)c1ccc(CCCCC(=O)NO)cc1
CC\C(=C(/c1ccc(O)cc1)c1ccc(OCCN(C)C)cc1)c1ccc(OCCCCC(=O)NO)cc1
CCc1c2Cn3c(cc4c(COC(=O)[C@@]4(CC)OC(=O)CCCCCCCCCCC(=O)NO)c3=O)-c2nc2ccc(O)cc12 |r|
CCc1c2Cn3c(cc4c(COC(=O)[C@@]4(CC)OC(=O)CCCCCCCCC(=O)NO)c3=O)-c2nc2ccc(O)cc12 |r|
CCc1c2Cn3c(cc4c(COC(=O)[C@@]4(CC)OC(=O)CNC(=O)CCCCCCC(O)=O)c3=O)-c2nc2ccc(O)cc12 |r|
CCc1c2Cn3c(cc4c(COC(=O)[C@]4(O)CC)c3=O)-c2nc2ccc(OC(=O)N3CCN(CC3)C(=O)CCCCCCC(=O)NO)cc12 |r|
CCc1c2Cn3c(cc4c(COC(=O)[C@]4(O)CC)c3=O)-c2nc2ccc(OC(=O)N3CCN(CC3)C(=O)CCCCCCCCCC(=O)NO)cc12 |r|
CCc1c2Cn3c(cc4c(COC(=O)[C@@]4(CC)OC(=O)CCCCCC(=O)NO)c3=O)-c2nc2ccc(O)cc12 |r|
CCc1c2Cn3c(cc4c(COC(=O)[C@@]4(CC)OC(=O)CCCCCCCC(=O)NO)c3=O)-c2nc2ccc(O)cc12 |r|
CCc1c2Cn3c(cc4c(COC(=O)[C@@]4(CC)OC(=O)CCCCCCCCCC(=O)NO)c3=O)-c2nc2ccc(O)cc12 |r|
CCc1c2Cn3c(cc4c(COC(=O)[C@@]4(CC)OC(=O)CNC(=O)CCCCCCC(=O)NO)c3=O)-c2nc2ccc(O)cc12 |r|
CCc1c2Cn3c(cc4c(COC(=O)[C@]4(O)CC)c3=O)-c2nc2ccc(OC(=O)N3CCN(CC3)C(=O)CCCCCCCC(=O)NO)cc12 |r|
CCc1c2Cn3c(cc4c(COC(=O)[C@]4(O)CC)c3=O)-c2nc2ccc(OC(=O)N3CCN(CC3)C(=O)CCCCCCCCCCC(=O)NO)cc12 |r|
CCc1c2Cn3c(cc4c(COC(=O)[C@]4(O)CC)c3=O)-c2nc2ccc(OC(=O)N3CCN(CC3)C(=O)CCCCCCCCC(=O)NO)cc12 |r|
CCc1c2Cn3c(cc4c(COC(=O)[C@@]4(CC)OC(=O)CCCCCCC(=O)NO)c3=O)-c2nc2ccc(O)cc12 |r|
CCc1c2Cn3c(cc4c(COC(=O)[C@@]4(CC)OC(=O)CCCCCCC(O)=O)c3=O)-c2nc2ccc(O)cc12 |r|
COc1ccc(Nc2c(NCCCCCC(=O)NO)c(=O)c2=O)cc1
CC(C)(CCCCC(=O)NO)Nc1c(Nc2ccc(cc2)C(F)(F)F)c(=O)c1=O
CC(Nc1c(NCCCCCC(=O)NO)c(=O)c1=O)C12CC3CC(CC(C3)C1)C2 |THB:24:23:20:26.25.27,24:25:22.23.28:20,27:25:22:28.19.20,27:19:22:26.24.25|
ONC(=O)CCC(CCCC(=O)Nc1ccccc1)Cc1ccccc1
CCC(CCCC(=O)Nc1ccccc1)CCC(=O)NO
CCCCC(CCCC(=O)Nc1ccccc1)CCC(=O)NO
CCCCCCC(CCCC(=O)Nc1ccccc1)CCC(=O)NO
ONC(=O)CC[C@H](CCCC(=O)Nc1ccccc1)Cc1ccccc1 |r|
ONC(=O)CCC(CCCC(=O)Nc1ccccc1)c1ccccc1
ONC(=O)CC[C@@H](CCCC(=O)Nc1ccccc1)Cc1ccccc1 |r|
CC[C@@]1(O)C(=O)OCc2c1cc1-c3nc4ccccc4c(\C=N\OCCCCCC(=O)NCCSSCCNC(=O)C(\Cc4ccc(O)c(Br)c4)=N/O)c3Cn1c2=O |r|
CC[C@@]1(O)C(=O)OCc2c1cc1-c3nc4ccc(O)cc4c(\C=N\OCCCCCC(=O)NCCSSCCNC(=O)C(\Cc4ccc(O)c(Br)c4)=N/O)c3Cn1c2=O |r|
Nc1ccccc1NC(=O)c1ccc(CSC(=S)N2CCc3ccccc3C2)cc1
Nc1ccccc1NC(=O)c1ccc(CSC(=S)N2CCN(CC2)c2ccncc2)cc1
CCN(Cc1ccncc1)C(=S)SCc1ccc(cc1)C(=O)Nc1ccccc1N
Cc1ccc(cc1)-c1nc(NCc2ccc(cc2)C(=O)NO)cc2c3ccccc3[nH]c12
COc1cc(cc(OC)c1OC)-c1nc(NCc2ccc(cc2)C(=O)NO)cc2c3ccccc3[nH]c12
COc1cccc(c1)-c1nc(NCc2ccc(cc2)C(=O)NO)cc2c3ccccc3[nH]c12
CC1(C)OB(OC1(C)C)c1ccc(CONC(=O)\C=C\c2cccc(c2)S(=O)(=O)Nc2ccccc2)cc1
Nc1ccccc1NC(=O)c1ccc(cc1)C(=O)NCCNc1nonc1\C(Nc1ccc(F)c(Br)c1)=N\O
ONC(=O)CCCCCn1[se]c2ccccc2c1=O
ONC(=O)\C=C\c1ccc(cc1)-n1[se]c2ccccc2c1=O
ONC(=O)c1ccc(Cn2[se]c3ccc(F)cc3c2=O)cc1
ONC(=O)c1ccc(Cn2[se]c3ccc(cc3c2=O)C(F)(F)F)cc1
ONC(=O)c1cnc(nc1)N1CCC(Cn2[se]c3ccccc3c2=O)CC1
ONC(=O)c1cnc(nc1)N1CCC(CC1)n1[se]c2ccccc2c1=O
ONC(=O)CCCCCOc1ccc(cc1)-n1[se]c2ccccc2c1=O
ONC(=O)CCCOc1ccc(cc1)-n1[se]c2ccccc2c1=O
ONC(=O)c1ccc(Cn2[se]c3ccccc3c2=O)cc1
ONC(=O)CCCCCCn1[se]c2ccccc2c1=O
ONC(=O)CCCCn1[se]c2ccccc2c1=O
O=c1n([se]c2ccccc12)-c1ccccc1
ONC(=O)CCCCCCOc1ccc(cc1)-n1[se]c2ccccc2c1=O
ONC(=O)CCc1ccc(cc1)-n1[se]c2ccccc2c1=O
ONC(=O)c1ccc(cc1)-n1[se]c2ccccc2c1=O
ONC(=O)c1ccc(Cn2[se]c3ccc(O)cc3c2=O)cc1
CC(c1ccc(cc1)C(=O)NO)n1[se]c2ccccc2c1=O
CN1CCN(CC(=O)Nc2ccc(cc2)-c2ccnc(Nc3cccc(OCCCCCCC(=O)NO)c3)n2)CC1
CC(=O)Nc1ccc(cc1)-c1ccnc(Nc2ccc(NC(=O)CCCCCCC(=O)NO)cc2)n1
CC(=O)Nc1ccc(cc1)-c1ccnc(Nc2cccc(OCCCCCCCC(=O)NO)c2)n1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1ccnc(Nc2ccc(cc2)N2CCCCC2)n1
CC(=O)Nc1ccc(cc1)-c1ccnc(Nc2cccc(NC(=O)CCCCC(=O)NO)c2)n1
CC(=O)Nc1ccc(cc1)-c1nc(Nc2cccc(OCCCCCCC(=O)NO)c2)ncc1C
CC(=O)Nc1ccc(cc1)-c1ccnc(Nc2ccc(OCCCCCCC(=O)NO)cc2)n1
Cc1cnc(Nc2ccc(cc2)N2CCOCC2)nc1-c1ccc(NC(=O)CCCCCCC(=O)NO)cc1
CC(=O)Nc1ccc(cc1)-c1ccnc(Nc2ccc(OCCCCCC(=O)NO)cc2)n1
CC(=O)Nc1ccc(cc1)-c1nc(Nc2cccc(OCCCCCCCC(=O)NO)c2)ncc1C
CN1CCN(CC(=O)Nc2ccc(cc2)-c2ccnc(Nc3ccc(OCCCCCCC(=O)NO)cc3)n2)CC1
COC(=O)CCCCCCOc1ccc(Nc2nccc(n2)-c2ccc(NC(C)=O)cc2)cc1
CC(=O)Nc1ccc(cc1)-c1ccnc(Nc2ccc(NC(=O)CCCCC(=O)NO)cc2)n1
CC(=O)Nc1ccc(cc1)-c1ccnc(Nc2cccc(OCCCCCC(=O)NO)c2)n1
CC(=O)Nc1ccc(cc1)-c1ccnc(Nc2cccc(OCCCCCCC(=O)NO)c2)n1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1ccnc(Nc2ccccc2)n1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1ccnc(Nc2ccc(cc2)N2CCOCC2)n1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1ccnc(Nc2cccc(c2)N2CCCCC2)n1
CN1CCN(CC1)c1ccc(Nc2nccc(n2)-c2ccc(NC(=O)CCCCCCC(=O)NO)cc2)cc1
CN1CCN(CC1)c1ccc(Nc2ncc(C)c(n2)-c2ccc(NC(=O)CCCCCCC(=O)NO)cc2)cc1
CC(=O)Nc1ccc(cc1)-c1ccnc(Nc2ccc(OCCCCCCCC(=O)NO)cc2)n1
CC(=O)Nc1ccc(cc1)-c1ccnc(Nc2cccc(NC(=O)CCCCCCC(=O)NO)c2)n1
CC(=O)Nc1ccc(cc1)-c1nc(Nc2ccc(OCCCCCC(=O)NO)cc2)ncc1C
CCCCNC(=O)CN(Cc1ccc(cc1)C(=O)NO)C(=O)c1ccc(cc1)N(C)C
CC(C)c1ccc(cc1)C(=O)N(CC(=O)NC1CCCCC1)Cc1ccc(cc1)C(=O)NO
Cc1ccc(cc1C)C(=O)N(CC(=O)NC1CCCCC1)Cc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(CN(CC(=O)NC2CCCCC2)C(=O)c2cccc3ccccc23)cc1
Cc1ccc(cc1C)C(=O)N(CC(=O)NC(C)(C)C)Cc1ccc(cc1)C(=O)NO
CCCN1CC(=O)N2Cc3c(CC2C1=O)c1ccccc1n3Cc1ccc(cc1)C(=O)NO
CCN1C(=O)C2Cc3c(CN2C1=O)n(Cc1ccc(cc1)C(=O)NO)c1ccccc31
CCCN1C(=O)C2Cc3c(CN2C1=O)n(Cc1ccc(cc1)C(=O)NO)c1ccccc31
CN1CC(=O)N2Cc3c(CC2C1=O)c1ccccc1n3Cc1ccc(cc1)C(=O)NO
CCCCN1CC(=O)N2Cc3c(CC2C1=O)c1ccccc1n3Cc1ccc(cc1)C(=O)NO
CC(C)CN1CC(=O)N2Cc3c(CC2C1=O)c1ccccc1n3Cc1ccc(cc1)C(=O)NO
CCCN1CC(=O)N2Cc3c(CC2C1=O)c1cc(OC)ccc1n3Cc1ccc(cc1)C(=O)NO
[H][C@]12Cc3c([C@H](C)N1C(=O)CN(CCC)C2=O)n(Cc1ccc(cc1)C(=O)NO)c1ccccc31 |r|
[H][C@]12Cc3c([C@@H](C)N1C(=O)CN(CCC)C2=O)n(Cc1ccc(cc1)C(=O)NO)c1ccccc31 |r|
CCCN1CC(=O)N2Cc3c(CC2C1=O)c1cc(O)ccc1n3Cc1ccc(cc1)C(=O)NO
CCCN1CC(=O)N2Cc3c(CC2C1=O)c1cc(OCc2ccccc2)ccc1n3Cc1ccc(cc1)C(=O)NO
CCN1CC(=O)N2Cc3c(CC2C1=O)c1ccccc1n3Cc1ccc(cc1)C(=O)NO
CN1C(=O)C2Cc3c(CN2C1=O)n(Cc1ccc(cc1)C(=O)NO)c1ccccc31
CCCCN1C(=O)C2Cc3c(CN2C1=O)n(Cc1ccc(cc1)C(=O)NO)c1ccccc31
CC(C)CCN1CC(=O)N2Cc3c(CC2C1=O)c1ccccc1n3Cc1ccc(cc1)C(=O)NO
[H][C@@]12Cc3c([C@@H](C)N1C(=O)CN(CCC)C2=O)n(Cc1ccc(cc1)C(=O)NO)c1ccccc31 |r|
[H][C@@]12Cc3c([C@H](C)N1C(=O)CN(CCC)C2=O)n(Cc1ccc(cc1)C(=O)NO)c1ccccc31 |r|
CN1CCC2(CN(Cc3ccc(cc3)C(=O)NO)c3ccccc23)CC1
ONC(=O)c1ccc(CN2CC3(CCCCC3)c3ccccc23)cc1
CC(=O)N1CCC2(CN(Cc3ccc(cc3)C(=O)NO)c3ccccc23)CC1
CC(C)(C)C(=O)N1CCC2(CN(Cc3ccc(cc3)C(=O)NO)c3ccccc23)CC1
CN1CCC2(CN(Cc3ccc(s3)C(=O)NO)c3ccccc23)CC1
CC(C)(C)OC(=O)N1CCC2(CN(Cc3ccc(cc3)C(=O)NO)c3ccccc23)CC1
CC(C)(C)OC(=O)N1CCC2(CN(Cc3ccc(s3)C(=O)NO)c3ccccc23)CC1
ONC(=O)c1ccc2CCN(Cc2c1)C(=O)C(=C\c1ccc(F)cc1F)\c1ccc(F)cc1
COc1cc(\C=C(\C(=O)N2CCc3ccc(cc3C2)C(=O)NO)c2ccc(F)cc2)ccc1F
ONC(=O)c1ccc2CCN(Cc2c1)C(=O)C(=C\c1ccccc1)\c1cccc(Cl)c1
COc1ccc(\C=C(\C(=O)N2CCc3ccc(cc3C2)C(=O)NO)c2ccccc2)cc1
Cc1ccc(cc1)C(=C/c1ccc(F)cc1)\C(=O)N1CCc2ccc(cc2C1)C(=O)NO
Cc1ccc(cc1)C(=C/c1ccccc1)\C(=O)N1CCc2ccc(cc2C1)C(=O)NO
ONC(=O)c1ccc2CCN(Cc2c1)C(=O)C(=C\c1ccccc1)\c1ccccc1
COc1ccc(\C=C(\C(=O)N2CCc3ccc(cc3C2)C(=O)NO)c2ccccc2F)cc1OC
ONC(=O)c1ccc2CCN(Cc2c1)C(=O)C(=C\c1cccs1)\c1ccc(F)cc1
COc1ccc(\C=C(\C(=O)N2CCc3ccc(cc3C2)C(=O)NO)c2ccc(F)cc2)c(OC)c1
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1CCC(C1)c1ccccc1
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1CC(C1)c1ccccc1
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1CCc2ccccc2C1
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1Cc2ccccc2C1
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1CCC(CC1)N1CCCC1
OC(=O)CCC(=O)c1ccc(cc1)S(=O)(=O)N1CCC(CC1)N1CCCC1
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1CCC(CC1)c1ccccc1
OC(=O)CCC(=O)c1ccc(cc1)S(=O)(=O)N1CCC(CC1)c1ccccc1
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1CCC(CC1)c1ccc(F)c(F)c1
c1cc(ccc1C(=O)CCC(=O)O)S(=O)(=O)N2CCC(CC2)c3ccc(c(c3)F)F
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1CCCC(CC1)c1ccccc1
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1CCN(CC1)c1ccccc1
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1CCC(=CC1)c1ccccc1 |c:20|
CC1CN(CCC1c1ccccc1)S(=O)(=O)c1ccc(cc1)C(=O)NCC(O)=O
CC1CC(CCN1S(=O)(=O)c1ccc(cc1)C(=O)NCC(O)=O)c1ccccc1
[H][C@]12CC[C@]([H])(C[C@@H](C1)c1ccccc1)N2S(=O)(=O)c1ccc(cc1)C(=O)NCC(O)=O |r|
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1CCC(CC1)Oc1ccccc1
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1CCC(CC1)N1C(=O)Cc2ccccc12
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1CCC2(CC1)OCc1ccccc21
CN(C)C1CCN(CC1)S(=O)(=O)c1ccc(cc1)C(=O)NCC(O)=O
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1CCC(CC1)C1CCCC1
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1CCC(CC1)N1CCOCC1
CN1CCN(CC1)C1CCN(CC1)S(=O)(=O)c1ccc(cc1)C(=O)NCC(O)=O
CN1CCC(CC1)NS(=O)(=O)c1ccc(cc1)C(=O)NCC(O)=O
CN1CCC2(CC1)CCN(CC2)S(=O)(=O)c1ccc(cc1)C(=O)NCC(O)=O
Cc1ccc(cc1)C1CCN(CC1)S(=O)(=O)c1ccc(cc1)C(=O)NCC(O)=O
COc1ccc(cc1)C1CCN(CC1)S(=O)(=O)c1ccc(cc1)C(=O)NCC(O)=O
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1CCC(CC1)c1ccc(F)cc1
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1CCC(CC1)c1ccc(Cl)cc1
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1CCC(CC1)c1ccc(Br)cc1
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1CCC(CC1)c1cccc(c1)C(F)(F)F
COc1cccc(c1)C1CCN(CC1)S(=O)(=O)c1ccc(cc1)C(=O)NCC(O)=O
OC(=O)CNC(=O)c1ccc(cc1)S(=O)(=O)N1CCC(CC1)c1cccc(F)c1
OC(=O)CNC(=O)c1cccc(c1)S(=O)(=O)N1CCC(CC1)c1ccccc1
OC(=O)CNC(=O)c1ccc(c(F)c1)S(=O)(=O)N1CCC(CC1)c1ccccc1
OC(=O)CNC(=O)c1ccc(c(Cl)c1)S(=O)(=O)N1CCC(CC1)c1ccccc1
Cc1cc(ccc1S(=O)(=O)N1CCC(CC1)c1ccccc1)C(=O)NCC(O)=O
c1ccc(cc1)C2CCN(CC2)S(=O)(=O)c3ccc(c(c3)F)C(=O)NCC(=O)O
OC(=O)CNC(=O)c1ccc(cc1Cl)S(=O)(=O)N1CCC(CC1)c1ccccc1
Cc1cc(ccc1C(=O)NCC(O)=O)S(=O)(=O)N1CCC(CC1)c1ccccc1
OC(=O)CNC(=O)c1ccc(cn1)S(=O)(=O)N1CCC(CC1)c1ccccc1
OC(=O)CNC(=O)c1ccc(s1)S(=O)(=O)N1CCC(CC1)c1ccccc1
Cc1cc(sc1C(=O)NCC(O)=O)S(=O)(=O)N1CCC(CC1)c1ccccc1
OC(=O)CNC(=O)c1cc(cs1)S(=O)(=O)N1CCC(CC1)c1ccccc1
OC(=O)CNC(=O)c1csc(c1)S(=O)(=O)N1CCC(CC1)c1ccccc1
OC(=O)CNC(=O)c1ccc(o1)S(=O)(=O)N1CCC(CC1)c1ccccc1
Cn1cc(cc1C(=O)NCC(O)=O)S(=O)(=O)N1CCC(CC1)c1ccccc1
OC(=O)CNC(=O)c1ccc(cc1F)S(=O)(=O)N1CCC(CC1)c1ccc(Cl)cc1
OC(=O)CNC(=O)c1ccc(cc1F)S(=O)(=O)N1CCC(CC1)c1ccc(Br)cc1
OC(=O)CNC(=O)c1ccc(cc1F)S(=O)(=O)N1CCC(CC1)N1CCCC1
c1cc(ccc1C2CCN(CC2)S(=O)(=O)c3ccc(nc3)C(=O)NCC(=O)O)Cl
[O-]C(=O)CNC(=O)c1ccc(cn1)S(=O)(=O)N1CCC(CC1)c1ccc(Cl)cc1
CCc1c2Cn3c(cc4c(COC(=O)[C@]4(O)CC)c3=O)-c2nc2ccc(OCc3cn(CCCCCCC(=O)NO)nn3)cc12 |r|
CCc1c2Cn3c(cc4c(COC(=O)[C@]4(O)CC)c3=O)-c2nc2ccc(OCc3cn(CCCCCC(=O)NO)nn3)cc12 |r|
CCc1c2Cn3c(cc4c(COC(=O)[C@]4(O)CC)c3=O)-c2nc2ccc(OCc3cn(CCCC(=O)NO)nn3)cc12 |r|
CC[C@@]1(O)C(=O)OCc2c1cc1-c3nc4ccc(OCc5cn(CCCCCCC(=O)NO)nn5)cc4cc3Cn1c2=O |r|
CC[C@@]1(O)C(=O)OCc2c1cc1-c3nc4ccc(OCc5cn(CCCCC(=O)NO)nn5)cc4cc3Cn1c2=O |r|
CCc1c2Cn3c(cc4c(COC(=O)[C@]4(O)CC)c3=O)-c2nc2ccc(OCc3cn(CCCCCCCC(=O)NO)nn3)cc12 |r|
CC\C(=C(/c1ccccc1)c1ccc(OCCN(C)Cc2ccc(cc2)-c2cn(CCCCCC(=O)NO)nn2)cc1)c1ccccc1
[H][C@@]12CC[C@@](O)(c3cn(CCCCCC(=O)NO)nn3)[C@@]1(C)CC[C@]1([H])c3ccc(O)cc3CC[C@@]21[H] |r|
[H][C@@]12CC[C@@](O)(c3cn(CCCCC(=O)NO)nn3)[C@@]1(C)CC[C@]1([H])c3ccc(O)cc3CC[C@@]21[H] |r|
[H][C@@]12CC[C@@](O)(c3cn(CCCCCCCC(=O)NO)nn3)[C@@]1(C)CC[C@]1([H])c3ccc(O)cc3CC[C@@]21[H] |r|
CC\C(=C(/c1ccccc1)c1ccc(OCCN(C)Cc2ccc(NC(=O)CCCCCCC(=O)NO)cc2)cc1)c1ccccc1
[H][C@@]12CC[C@@](O)(c3cn(CCCCCCC(=O)NO)nn3)[C@@]1(C)CC[C@]1([H])c3ccc(O)cc3CC[C@@]21[H] |r|
[H][C@@]12CC[C@@](O)(c3cn(CCCC(=O)NO)nn3)[C@@]1(C)CC[C@]1([H])c3ccc(O)cc3CC[C@@]21[H] |r|
Oc1cccc(cc1=O)C1CCCC1
COc1ccc(OC)c(c1)-c1cccc(O)c(=O)c1
Oc1cccc(cc1=O)-c1ccccc1
COc1ccc(c(OC)c1OC)-c1ccccc(O)c1=O
Oc1ccccc(-c2ccc3ccccc3c2)c1=O
Oc1ccccc(-c2ccccc2)c1=O
CCC(C)c1cccc(O)c(=O)c1
COc1cccc(cc1=O)C(C)C
CC(C)(C)c1cccc(O)c(=O)c1
COc1ccc(cc1)-c1cccc(O)c(=O)c1
CC(C)C1=CC=CC(=O)C(=C1)O
COc1ccc(cc1)-c1ccccc(O)c1=O
COc1ccc(OC)c(c1)-c1ccccc(O)c1=O
CN1c2ccc(cc2C(=NC(N)C1=O)c1ccccc1)C#CCCCC(=O)NO |c:9|
CN1c2ccccc2C(=NC(NC(=O)CCCCC(=O)NO)C1=O)c1ccccc1 |c:9|
CN1c2ccccc2C(=NC(NC(=O)CCCCCCCC(=O)NO)C1=O)c1ccccc1 |c:9|
CN1c2ccc(cc2C(=NCC1=O)c1ccccc1)C#C\C=C\C(=O)NO |c:9|
C[C@@H]1N=C(c2ccccc2)c2cc(ccc2NC1=O)C#CCCCC(=O)NO |r,t:2|
CN1c2ccc(cc2C(=NCC1=O)c1ccccc1)C#CCCCC(=O)NO |c:9|
ONC(=O)CCCCCCC(=O)N1CCN=C(c2ccccc2)c2ccccc12 |t:15|
CN1c2ccc(cc2C(=NCC1=O)c1ccccc1)C#CCCC(=O)NO |c:9|
CN1c2ccccc2C(=NC(NC(=O)CCCCCC(=O)NO)C1=O)c1ccccc1 |c:9|
CN1c2ccc(cc2C(=N[C@H](O)C1=O)c1ccccc1)C#CCCCC(=O)NO |r,c:9|
CN1c2ccccc2C(=N[C@@H](NC(=O)CCCCCCC(=O)NO)C1=O)c1ccccc1 |r,c:9|
CN1c2ccccc2C(=N[C@H](NC(=O)CCCCCCC(=O)NO)C1=O)c1ccccc1 |r,c:9|
CN1c2ccc(cc2C(=NCC1=O)c1ccccc1)C#CCCCCC(=O)NO |c:9|
CN1c2ccc(cc2C(=N[C@@H](O)C1=O)c1ccccc1)C#CCCCC(=O)NO |r,c:9|
Cc1ccc(OCCN(CCc2ccc3OCOc3c2)Cc2ccc(\C=C\C(=O)NO)o2)cc1
Cc1ccc(OCCN(Cc2ccc(\C=C\C(=O)NO)o2)Cc2ccc(cc2)-c2ccccc2)cc1
Cc1ccc(OCCCN(Cc2ccc(\C=C\C(=O)NO)o2)Cc2ccccc2)cc1
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[H][C@]1(C[C@](C)(OC)[C@@](O)(CN(C)Cc2ccc(cc2)-c2cn(CCCC(=O)NO)nn2)[C@@H](C)O1)O[C@H]1[C@@H](C)[C@@H](O[C@@]2([H])O[C@@H](C)C[C@H]([C@@H]2O)N(C)C)[C@@](C)(C[C@@H](C)C(=O)[C@H](C)[C@H](O)[C@](C)(O)[C@@H](CC)OC(=O)[C@@H]1C)OC |r|
[H][C@]1(C[C@](C)(OC)[C@@](O)(CN(C)Cc2ccc(cc2)-c2cn(CCCCCC(=O)NO)nn2)[C@@H](C)O1)O[C@@H]1[C@@H](C)C(=O)O[C@@H](CC)[C@@](C)(O)[C@H](O)[C@@H](C)N(C)C[C@H](C)C[C@@](C)(O)[C@]([H])(O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@@H]1C |r|
[H][C@@]1(C[C@@](C)(OC)[C@](O)(CN(C)Cc2ccc(cc2)-c2cn(CCC(=O)NO)nn2)[C@H](C)O1)O[C@@H]1[C@@H](C)C(=O)O[C@@H](CC)[C@@](C)(O)[C@H](O)[C@@H](C)N(C)C[C@H](C)C[C@@](C)(O)[C@]([H])(O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@@H]1C |r|
[H][C@@]1(C[C@@](C)(OC)[C@](O)(CN(C)Cc2ccc(cc2)-c2cn(CCCCC(=O)NO)nn2)[C@H](C)O1)O[C@@H]1[C@H](C)[C@H](O[C@]2([H])O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@](C)(C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@](C)(O)[C@H](CC)OC(=O)[C@H]1C)OC |r|
[H][C@@]1(C[C@@](C)(OC)[C@@H](O)[C@H](C)O1)O[C@@H]1[C@H](C)[C@H](O[C@]2([H])O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCC(=O)NO)nn2)[C@](C)(C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@](C)(O)[C@H](CC)OC(=O)[C@H]1C)OC |r|
[H][C@]1(C[C@](C)(OC)[C@@](O)(CN(C)C)[C@@H](C)O1)O[C@@H]1[C@H](C)[C@H](O[C@]2([H])O[C@H](C)C[C@@H]([C@H]2O)N(C)Cc2ccc(cc2)-c2cn(CCCCCCC(=O)NO)nn2)[C@](C)(C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@](C)(O)[C@H](CC)OC(=O)[C@H]1C)OC |r|
[H][C@]1(C[C@](C)(OC)[C@H](O)[C@@H](C)O1)O[C@@H]1[C@@H](C)C(=O)O[C@H](CC)[C@@](C)(O)[C@H](O)[C@H](C)N(Cc2ccc(cc2)-c2cn(CC(=O)NO)nn2)C[C@H](C)C[C@](C)(O)[C@]([H])(O[C@@H]2O[C@H](C)C[C@@H]([C@H]2O)N(C)C)[C@H]1C |r|
[H][C@@]12CC[C@H](O)[C@@]1(C)CC[C@]1([H])c3ccc(O)cc3C[C@@H](CCCCCCCCCCC(=O)Nc3ccccc3N)[C@@]21[H] |r|
[H][C@@]12CC[C@H](O)[C@@]1(C)CC[C@]1([H])c3ccc(O)cc3C[C@@H](CCCCCCCCCCC(=O)N(O)CCCC)[C@@]21[H] |r|
[H][C@@]12CC[C@H](O)[C@@]1(C)CC[C@]1([H])c3ccc(O)cc3C[C@@H](SCCCCCC(=O)Nc3cccc(c3)C(=O)N(O)CCCC)[C@@]21[H] |r|
[H][C@@]12CC[C@H](O)[C@@]1(C)CC[C@]1([H])c3ccc(O)cc3C[C@@H](CCCCCCCCCCC(=O)NO)[C@@]21[H] |r|
ONC(=O)CCCCCCC(=O)NO
CC(C)(C)OC(=O)ON(C(=O)CCCCCCC(=O)N(OC(=O)OC(C)(C)C)C(=O)OC(C)(C)C)C(=O)OC(C)(C)C
CC(C)(C)OC(=O)ON(C(=O)CC\C=C\CCC(=O)N(OC(=O)OC(C)(C)C)C(=O)OC(C)(C)C)C(=O)OC(C)(C)C
COc1ccc(cc1)-c1nc(NC(=O)NCCCC(=O)NO)cc2c3ccccc3[nH]c12
COc1ccc(cc1)-c1nc(NC(=O)NCCCCC(=O)NO)cc2c3ccccc3[nH]c12
COc1ccc(cc1)-c1nc(NC(=O)NCCC(=O)NO)cc2c3ccccc3[nH]c12
COc1ccc(cc1)-c1nc(cc2c3ccccc3[nH]c12)C(=O)NCCCC(=O)NO
COc1ccc(cc1)-c1nc(NC(=O)NCCCC(=O)NO)cc2c3ccccc3n(C)c12
Cc1ccc(CN2C(CCC(=O)NCc3ccc(cc3)C(=O)NO)C(=O)N(C3CCCCC3)C2=O)cc1
ONC(=O)c1ccc(NC(=O)CCC2N(Cc3ccccc3)C(=O)N(C2=O)c2ccc(Cl)cc2)cc1
CCCN1C(CCC(=O)Nc2ccc(cc2)C(=O)NO)C(=O)N(C2CCCCC2)C1=O
CN1C(CCC(=O)NCc2ccc(cc2)C(=O)NO)C(=O)N(C1=O)c1ccc(Cl)cc1
CN1C(CCC(=O)Nc2ccc(cc2)C(=O)NO)C(=O)N(C1=O)c1ccc(Cl)cc1
ONC(=O)c1ccc(CNC(=O)CCC2N(Cc3ccccc3)C(=O)N(C2=O)c2ccc(Cl)cc2)cc1
ONC(=O)c1cccc(NC(=O)CCC2N(Cc3ccccc3)C(=O)N(C2=O)c2ccc(Cl)cc2)c1
Cc1ccc(CN2C(CCC(=O)Nc3cccc(c3)C(=O)NO)C(=O)N(C2=O)c2ccc(Cl)cc2)cc1
ONC(=O)c1ccc(CNC(=O)CCC2N(Cc3ccc(Br)cc3)C(=O)N(C2=O)c2ccc(Cl)cc2)cc1
ONC(=O)c1ccc(NC(=O)CCC2N(Cc3ccc(Br)cc3)C(=O)N(C2=O)c2ccc(Cl)cc2)cc1
Cc1ccc(CN2C(CCC(=O)NCc3ccc(cc3)C(=O)NO)C(=O)N(C2=O)c2ccc(Cl)cc2)cc1
ONC(=O)c1ccc(NC(=O)CCC2N(Cc3ccc(Br)cc3)C(=O)N(Cc3ccccc3)C2=O)cc1
Cc1ccc(CN2C(CCC(=O)Nc3ccc(cc3)C(=O)NO)C(=O)N(C3CCCCC3)C2=O)cc1
CCCN1C(CCC(=O)Nc2ccc(cc2)C(=O)NO)C(=O)N(C1=O)c1ccc(Cl)cc1
Cc1ccc(CN2C(CCC(=O)Nc3ccc(cc3)C(=O)NO)C(=O)N(C2=O)c2ccc(Cl)cc2)cc1
ONC(=O)c1ccc(CNC(=O)CCC2N(Cc3ccc(Br)cc3)C(=O)N(C2=O)c2ccccc2)cc1
ONC(=O)C(c1ccc(cc1)-c1ncc(cn1)C(F)(F)F)c1ccccc1F
Cc1ncc(cn1)-c1ccc(cc1)C(C(=O)NO)c1ccccc1F
ONC(=O)C1c2ccccc2-c2ccccc12
COc1ccc(cn1)-c1cc(OCCN(C)c2ncc(cn2)C(=O)NO)c2ncnc(C)c2c1
CCCCN(Cc1ccc(cc1)C(=O)NO)C(=O)Nc1ccc(OCCCCCn2cc(CNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)nn2)cc1
COc1cc2nc(nc(NC3CCN(Cc4ccccc4)CC3)c2cc1OC)N1CCN(CC1)C(=O)CCCCCCC(=O)NO
ONC(=O)CCCCCCC(=O)Nc1ccc(Nc2nc(NC3CCN(Cc4ccccc4)CC3)c3sccc3n2)cc1
COc1cc2nc(Nc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)nc(NC3CCN(Cc4ccc(F)cc4)CC3)c2cc1OC
COc1cc2nc(Nc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)nc(NC3CCN(Cc4ccccc4)CC3)c2cc1OC
COc1cc2nc(Nc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)nc(NC3CCN(Cc4ccccc4Cl)CC3)c2cc1OC
COc1ccc(CN2CCC(CC2)Nc2nc(Nc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)nc3cc(OC)c(OC)cc23)cc1
[H][C@]12CC(=O)N[C@H](C)C(=O)N[C@]([H])(CSSCC\C=C\1)C(=O)N[C@H](C(C)C)[C@@H](O)CC(=O)O2 |r,t:18|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)C(=O)NCc1cccc(c1)C(=O)NO |r|
c1cc(c(nc1)C(F)(F)F)C(=O)NCc2ccc(cc2)C(=O)NO
C[C@@H](C(=O)NCc1ccc(cc1)C(=O)NO)NC(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2
ONC(=O)c1ccc(CNC(=O)CNC(=O)CNC(=O)OCc2ccccc2)cc1
CN(C)Cc1ccc(cc1)S(=O)(=O)n2ccc(c2)/C=C/C(=O)NO
CC1([C@@H]2CC[C@H]([C@H]1C2)CNCc3ccc(cc3)C(=O)NO)C
COc1ccc(cc1\C=C\C(=O)NO)C(=C)c1cc(OC)c(OC)c(OC)c1
COc1cc(cc(OC)c1OC)C(=C)c1ccc2n(C)c(\C=C\C(=O)NO)cc2c1
COc1cc(cc(OC)c1OC)C(=C)c1ccc2n(C)cc(\C=C\C(=O)NO)c2c1
COc1ccc(C(=C)c2cc(OC)c(OC)c(OC)c2)c(\C=C\C(=O)NO)c1
ONC(=O)CCCCCSc1nc(cc(=O)[nH]1)-c1ccc(cc1)-c1ccccc1
ONC(=O)CCCCCSc1nc(cc(=O)[nH]1)-c1ccc2ccccc2c1
ONC(=O)c1ccc(NC(=O)Cc2ccccc2)cn1
ONC(=O)CCCCSc1nc(cc(=O)[nH]1)-c1ccc2ccccc2c1
ONC(=O)\C=C\c1ccc(NC(=O)Cc2cccc3ccccc23)cn1
ONC(=O)c1ccc(NC(=O)Cc2cccc3ccccc23)cn1
Nc1ccccc1NC(=O)CCCCCN1C(=O)c2cccc3c(ccc(C1=O)c23)N1CCOCC1
Nc1ccccc1NC(=O)CCCCCN1C(=O)c2cccc3cccc(C1=O)c23
CN(Cc1ccccc1)c1ccc2C(=O)N(CCCCCC(=O)NO)C(=O)c3cccc1c23
CCCNc1ccc2C(=O)N(CCCCCC(=O)NO)C(=O)c3cccc1c23
ONC(=O)CCCCCN1C(=O)c2cccc3c(Nc4ccccc4)ccc(C1=O)c23
ONC(=O)c1ccc(CNC(=O)c2cc(Cn3c4ccccc4c4ccccc34)on2)cc1
ONC(=O)CCCCCN1C(=O)c2cccc3c(NCc4ccccc4)ccc(C1=O)c23
ONC(=O)CCCCCN1C(=O)c2cccc3c(ccc(C1=O)c23)[N+]([O-])=O
ONC(=O)CCCCCN1C(=O)c2cccc3c(Nc4cccc(F)c4)ccc(C1=O)c23
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3ccc(O)cc3)c2=O)cc1
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3cccc(c3)C(F)(F)F)c2=O)cc1
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3ccccc3)c2=O)s1
COc1ccc(CCn2c(=O)n(Cc3ccc(cc3)C(=O)NO)c3ccccc3c2=O)cc1
CC1(C)CCC(CN2CCN(CC2)c2ccc(C(=O)NS(=O)(=O)c3ccc(NCCCCCC(=O)NO)c(c3)[N+]([O-])=O)c(Oc3cnc4[nH]ccc4c3)c2)=C(C1)c1ccc(Cl)cc1 |c:58|
CC1(C)CCC(CN2CCN(CC2)c2ccc(C(=O)NS(=O)(=O)c3ccc(NCCCCC(=O)NO)c(c3)[N+]([O-])=O)c(Oc3cnc4[nH]ccc4c3)c2)=C(C1)c1ccc(Cl)cc1 |c:57|
CC1(C)CCC(CN2CCN(CC2)c2ccc(C(=O)NS(=O)(=O)c3ccc(NCCCC(=O)NO)c(c3)[N+]([O-])=O)c(Oc3cnc4[nH]ccc4c3)c2)=C(C1)c1ccc(Cl)cc1 |c:56|
CC1(C)CCC(CN2CCN(CC2)c2ccc(C(=O)NS(=O)(=O)c3ccc(NCC(=O)NO)c(c3)[N+]([O-])=O)c(Oc3cnc4[nH]ccc4c3)c2)=C(C1)c1ccc(Cl)cc1 |c:54|
CC1(C)CCC(CN2CCN(CC2)c2ccc(C(=O)NS(=O)(=O)c3ccc(NCCCCCCCC(=O)NO)c(c3)[N+]([O-])=O)c(Oc3cnc4[nH]ccc4c3)c2)=C(C1)c1ccc(Cl)cc1 |c:60|
CC1(C)CCC(CN2CCN(CC2)c2ccc(C(=O)NS(=O)(=O)c3ccc(NCCC(=O)NO)c(c3)[N+]([O-])=O)c(Oc3cnc4[nH]ccc4c3)c2)=C(C1)c1ccc(Cl)cc1 |c:55|
CC1(C)CCC(CN2CCN(CC2)c2ccc(C(=O)NS(=O)(=O)c3ccc(NCCCCCCC(=O)NO)c(c3)[N+]([O-])=O)c(Oc3cnc4[nH]ccc4c3)c2)=C(C1)c1ccc(Cl)cc1 |c:59|
Nc1ccccc1NC(=O)CCCCCN(CC(=O)NC1CCCCC1)C(=O)c1ccccc1
Cc1ccc(CNC(=O)CN(CCCCCC(=O)Nc2ccccc2N)C(=O)c2cc(C)cc(C)c2)cc1
CN(C)c1ccc(cc1)C(=O)N(CCCCCC(=O)Nc1ccccc1N)CC(=O)NCc1ccccc1
Cc1cc(C)cc(c1)C(=O)N(CCCCCC(=O)Nc1ccccc1N)CC(=O)NCc1ccccc1
Nc1ccccc1NC(=O)CCCCCN(CC(=O)NCc1ccccc1)C(=O)c1cccc2ccccc12
CN(C)c1ccc(cc1)C(=O)N(CCCCCC(=O)Nc1cc(F)ccc1N)CC(=O)NCc1ccccc1
COc1ccc(CNC(=O)CN(CCCCCC(=O)Nc2ccccc2N)C(=O)c2cc(C)cc(C)c2)cc1
CN(C)c1ccc(cc1)C(=O)N(CC(=O)NCc1ccccc1)Cc1ccc(cc1)C(=O)Nc1ccccc1N
Cc1cc(C)cc(c1)C(=O)N(CC(=O)NCc1ccccc1)Cc1ccc(cc1)C(=O)Nc1ccccc1N
Cc1cc(C)cc(c1)C(=O)N(CC(=O)NCc1ccccc1)Cc1ccc(cc1)C(=O)Nc1cc(F)ccc1N
Cc1cc(C)cc(c1)C(=O)N(CCCCCC(=O)Nc1cc(ccc1N)-c1ccccc1)CC(=O)NCc1ccccc1
CN(C)c1ccc(cc1)C(=O)N(CC(=O)NCc1ccccc1)Cc1ccc(cc1)C(=O)Nc1cc(ccc1N)-c1ccccc1
Cc1cc(C)cc(c1)C(=O)N(CCCCCC(=O)Nc1ccccc1N)CC(=O)NC1CCCCC1
Nc1ccccc1NC(=O)CCCCCN(CC(=O)NC1CCCCC1)C(=O)c1cccc2ccccc12
Cc1cc(C)cc(CNC(=O)CN(CCCCCC(=O)Nc2ccccc2N)C(=O)c2cc(C)cc(C)c2)c1
Cc1cc(C)cc(c1)C(=O)N(CC(=O)NCc1ccccc1)Cc1ccc(cc1)C(=O)Nc1cc(ccc1N)-c1ccccc1
Nc1ccccc1NC(=O)c1ccc(CN(CC(=O)NCc2ccccc2)C(=O)c2cccnc2)cc1
COc1cccc(c1)-c1nc(NCc2cccc(\C=C\C(=O)NO)c2)cc2c3ccccc3[nH]c12
COc1cc(cc(OC)c1OC)-c1nc(NCc2ccc(\C=C\C(=O)NO)cc2)cc2c3ccccc3[nH]c12
COc1cccc(c1)-c1nc(NCc2ccc(\C=C\C(=O)NO)cc2)cc2c3ccccc3[nH]c12
COc1cc(cc(OC)c1OC)-c1nc(NCc2cccc(\C=C\C(=O)NO)c2)cc2c3ccccc3[nH]c12
COc1ccc2[nH]cc(Cn3cc(COc4ccc(\C=C\C(=O)NO)cc4OC)nn3)c2c1
CN1CCc2c(C1)sc1nc([nH]c(=O)c21)-c1cc(C)c(OCc2ccc(cc2)C(=O)NO)c(C)c1
Cc1noc(C)c1-c1nc2sc3CN(CCCCCC(=O)Nc4ccccc4N)CCc3c2c(=O)[nH]1
Cc1cc(cc(C)c1O)-c1nc2sc3CN(CCCCCC(=O)NO)CCc3c2c(=O)[nH]1
CN1CCc2c(C1)sc1nc([nH]c(=O)c21)-c1cc(C)c(OCc2cccc(c2)C(=O)Nc2ccccc2N)c(C)c1
CN1CCc2c(C1)sc1nc([nH]c(=O)c21)-c1cc(C)c(OCc2cccc(c2)C(=O)NO)c(C)c1
CN1CCc2c(C1)sc1nc([nH]c(=O)c21)-c1cc(C)c(OCCCCCC(=O)NO)c(C)c1
CN1CCc2c(C1)sc1nc([nH]c(=O)c21)-c1cc(C)c(OCCCC(=O)NO)c(C)c1
CN1CCc2c(C1)sc1nc([nH]c(=O)c21)-c1cc(C)c(OCCOCc2ccc(\C=C\C(=O)NO)cc2)c(C)c1
Cc1noc(C)c1-c1nc2sc3CN(CC(=O)NO)CCc3c2c(=O)[nH]1
Cc1noc(C)c1-c1nc2sc3CN(CC(=O)Nc4ccccc4N)CCc3c2c(=O)[nH]1
CN1CCc2c(C1)sc1nc([nH]c(=O)c21)-c1cc(C)c(OCCCCCC(=O)Nc2ccccc2N)c(C)c1
Cc1noc(C)c1-c1nc2sc3CN(CCCCCC(=O)NO)CCc3c2c(=O)[nH]1
CN1CCc2c(C1)sc1nc([nH]c(=O)c21)-c1cc(C)c(OCc2ccc(cc2)C(=O)Nc2ccccc2N)c(C)c1
CN1CCc2c(C1)sc1nc([nH]c(=O)c21)-c1cc(C)c(OCc2ccc(\C=C\C(=O)NO)cc2)c(C)c1
Cc1noc(C)c1-c1nc2sc3CN(CCCC(=O)NO)CCc3c2c(=O)[nH]1
[H][C@@]12C[C@@]([H])([C@@]3([H])OB(O[C@@]3(C)C1)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc(cc1)C(=O)Nc1ccccc1N)C2(C)C |r|
[H][C@@]12C[C@@]([H])([C@@]3([H])OB(O[C@@]3(C)C1)[C@H](CC(C)C)NC(=O)CNC(=O)c1cccc(\C=C\C(=O)NO)c1)C2(C)C |r|
CCCNNC(=O)c1cccc(CNCCc2c(C)[nH]c3ccccc23)c1
CN(C)NC(=O)C=Cc1ccc(CNCCc2c(C)[nH]c3ccccc23)cc1
CCCNNC(=O)c1ccc(NC(=O)c2ccccc2)cc1
COC(=O)CCNNC(=O)C=Cc1ccc(CNCCc2c(C)[nH]c3ccccc23)cc1
Cc1[nH]c2ccccc2c1CCNCc1ccc(C=CC(=O)NN2CCCCC2)cc1
CCCN(CC)NC(=O)C=Cc1ccc(CNCCc2c(C)[nH]c3ccccc23)cc1
CCCCCN(CCC)NC(=O)C=Cc1ccc(CNCCc2c(C)[nH]c3ccccc23)cc1
CCCCCCN(CCC)NC(=O)C=Cc1ccc(CNCCc2c(C)[nH]c3ccccc23)cc1
Cc1[nH]c2ccccc2c1CCNCc1ccc(C=CC(=O)NN(CCCO)CCCO)cc1
CCCNNC(=O)c1ccc(CN(CCc2c(C)[nH]c3ccccc23)C(=O)OC(C)(C)C)cc1
CCCNNC(=O)c1ccc(CNCCc2c(C)[nH]c3ccccc23)cc1
CCCNNC(=O)c1cccc(CN(CCc2c(C)[nH]c3ccccc23)C(=O)OC(C)(C)C)c1
CCCNNC(=O)c1ccc(NCc2ccccc2)cc1
Cc1[nH]c2ccccc2c1CCNCc1ccc(C=CC(=O)NNCCN)cc1
CCCNNC(=O)C=Cc1ccc(CNCCc2c(C)[nH]c3ccccc23)cc1
CCCNNC(=O)c1ccc(CNCc2ccccc2)cc1
CCCNNC(=O)c1ccc(OCc2ccccc2)cc1
Cc1[nH]c2ccccc2c1CCNCc1ccc(C=CC(=O)NN2CCCC2)cc1
CCCN(CCC)NC(=O)C=Cc1ccc(CNCCc2c(C)[nH]c3ccccc23)cc1
CCCNNC(=O)c1ccc(CN(Cc2ccccc2)C(=O)OC(C)(C)C)cc1
CCCCN(CCC)NC(=O)C=Cc1ccc(CNCCc2c(C)[nH]c3ccccc23)cc1
CCCNNC(=O)\C=C\c1ccc(CN(CCc2c(C)[nH]c3ccccc23)C(=O)OC(C)(C)C)cc1
Cc1[nH]c2ccccc2c1CCNCc1ccc(C=CC(=O)NNCCC#N)cc1
CN(Cc1ccc(cc1)-n1cnn(CCCCc2ccc(cc2)C(=O)NO)c1=O)CC(O)(Cn1cncn1)c1ccc(F)cc1F
CN(Cc1ccc(OCCCOc2ccc(CC(=O)NO)cc2)cc1)CC(O)(Cn1cncn1)c1ccc(F)cc1F
ONC(=O)CCCCCCn1cc(Nc2ncc(Cl)c(Nc3cccc(Cl)c3)n2)cn1
CNc1nc(Nc2cnn(CCCCCCC(=O)NO)c2)ncc1Cl
ONC(=O)CCCCCCCn1cc(Nc2ncc(Cl)c(Nc3ccc(F)cc3)n2)cn1
ONC(=O)c1ccc(Cn2cc(Nc3ncc(Cl)c(Nc4ccc(F)cc4)n3)cn2)cc1
ONC(=O)\C=C\c1ccc(Cn2cc(Nc3ncc(Cl)c(Nc4ccc(F)cc4)n3)cn2)cc1
c1c[nH]c2c1c(ncn2)c3cnn(c3)[C@H](CC#N)C4CCCC4
ONC(=O)CCCCn1cc(Nc2ncc(Cl)c(Nc3ccc(F)cc3)n2)cn1
ONC(=O)CCCCCn1cc(Nc2ncc(Cl)c(Nc3ccc(Cl)cc3)n2)cn1
Cc1ccc2n(c(CCN3C(=O)c4cccc5cccc(C3=O)c45)nc2c1)-c1ccncc1
ONC(=O)c1ccc(CNCc2csc3ccccc23)cc1
ONC(=O)c1ccc(CN2c3ccccc3Sc3cccnc23)cc1
CC(C)(C)OC(=O)Nc1ccc(cc1)-c1cc(no1)C(=O)NCCc1cc(no1)C(=O)NO
ONC(=O)c1cc(CCC(=O)Nc2nc(cs2)-c2ccccc2)on1
ONC(=O)c1cc(CCNC(=O)c2ccccc2)on1
ONC(=O)c1cc(CCNC(=O)c2ccc3ccccc3c2)on1
ONC(=O)c1cc(CCNC(=O)c2cccc(c2)-c2ccccc2)on1
ONC(=O)c1cc(CCCCN2CCCc3cc(Cl)ccc23)on1
ONC(=O)c1cc(CCCCN2c3ccc(Cl)cc3CCc3cc(Cl)ccc23)on1
c1cc(c(cc1C(=O)NCCc2cc(no2)C(=O)NO)Cl)Cl
ONC(=O)c1cc(CCCCn2ccc3cc(Cl)c(Cl)cc23)on1
ONC(=O)c1cc(CCCOc2ccc(Cl)c(Cl)c2)on1
ONC(=O)c1ccc(CNC(=O)c2ccc(Cl)c(Cl)c2)cc1
CC1(C)CCN(CCCCc2cc(no2)C(=O)NO)c2ccc(Cl)cc12
ONC(=O)c1cc(CCCCc2ccc(Cl)c(Cl)c2)on1
C[C@H](NC(=O)c1nc(sc1C1CC1)-c1ncc(s1)-c1ccc(F)cc1)c1ccc(cc1)C(=O)NO |r|
ONC(=O)c1ccc(cc1)C1(CC1)NC(=O)c1nc(sc1C1CC1)-c1nccs1
C[C@H](NC(=O)c1nc(sc1C1CC1)-c1nccs1)c1ccc(cc1)C(=O)NO |r|
C[C@@H](NC(=O)c1nc(sc1C1CC1)-c1nccs1)c1ccc(cc1)C(=O)NO |r|
CC(C)[C@H](NC(=O)c1nc(sc1C1CC1)-c1nccs1)c1ccc(cc1)C(=O)NO |r|
C[C@H](NC(=O)c1nc(sc1C1CC1)-c1ncc(C)s1)c1ccc(cc1)C(=O)NO |r|
C[C@H](NC(=O)c1nc(sc1C1CC1)-c1nc(C)cs1)c1ccc(cc1)C(=O)NO |r|
C[C@H](NC(=O)c1nc(sc1C1CC1)-c1ncc(s1)-c1ccccc1)c1ccc(cc1)C(=O)NO |r|
COc1ccc(cc1)-c1cnc(s1)-c1nc(C(=O)N[C@@H](C)c2ccc(cc2)C(=O)NO)c(s1)C1CC1 |r|
CC(C)Cc1sc(nc1C(=O)Nc1ccc(\C=C\C(=O)NO)cc1)-c1nccs1
C[C@H](NC(=O)c1nc(sc1C1CC1)-c1nc2CCCCc2s1)c1ccc(cc1)C(=O)NO |r|
CC(NC(=O)c1nc(sc1C1CC1)-c1nccs1)c1ccc(cc1)C(=O)NO
CC(C)(NC(=O)c1nc(sc1C1CC1)-c1nccs1)c1ccc(cc1)C(=O)NO
Cc1cc(-c2ccc(\C=C3/C(=O)N(N=C3C3CC3)c3ccc(cc3)C(O)=O)s2)c(cc1C)C(F)(F)F |c:13|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C[C@H](NC1=O)C(\F)=C\CCS)n2 |r,c:11|
CCCCCCCC(=O)SCC\C=C(/F)[C@@H]1CC(=O)NCc2nc(cs2)C2=N[C@@](C)(CS2)C(=O)N[C@@H](C(C)C)C(=O)O1 |r,t:27|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C[C@H](OC1=O)C(\F)=C\CCS)n2 |r,c:11|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C[C@H](OC1=O)\C=C(/F)CCS)n2 |r,c:11|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C[C@H](OC1=O)\C=C\C(F)(F)CS)n2 |r,c:11|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C[C@@H](OC1=O)C(\F)=C\CCS)n2 |r,c:11|
CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(CNC(=O)C(F)(F)[C@H](NC1=O)\C=C\CCS)n2 |r,c:11|
CN(Cc1nc(no1)C1CCN(Cc2ccc(C)cc2)CC1)c1ncc(cn1)C(=O)NO
CN1CCC(CNC(=O)c2cccc(c2)-c2noc(n2)C(F)(F)F)(CC1)c1nc(cs1)-c1ccccc1
CN1CCC(CNC(=O)c2cccc(c2)C(=O)NO)(CC1)c1nc(cs1)-c1ccccc1
CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(cc1)C(=O)NC(CCP(O)(O)=O)P(O)(O)=O
ONC(=O)c1ccc(CN2N=CC=C3Sc4ccccc4N=C23)cc1 |c:10,t:12,22|
COc1ccc2Sc3ccccc3N(Cc3ccc(cc3)C(=O)NO)c2c1
ONC(=O)c1ccc(CN2c3ccccc3Sc3ccccc23)cc1
ONC(=O)c1ccc(CN2c3ccccc3S(=O)(=O)c3ccccc23)cc1
ONC(=O)c1ccc(CN2c3ccccc3Sc3cccc(Cl)c23)cc1
ONC(=O)c1ccc(CN2c3ccccc3[S+]([O-])c3ccccc23)cc1
CCSc1ccc2Sc3ccccc3N(Cc3ccc(cc3)C(=O)NO)c2c1
ONC(=O)c1ccc(CN2c3ccccc3Sc3ccncc23)cc1
ONC(=O)c1ccc(CN2c3ccccc3Sc3nccnc23)cc1
ONC(=O)c1ccc(CN2c3cccnc3Sc3cccnc23)cc1
ONC(=O)c1ccc(CN2c3ccncc3Sc3ncccc23)cc1
Cc1nc2N(Cc3ccc(cc3)C(=O)NO)c3ccccc3Sc2s1
CN1CCC2=C(C1)N(Cc1ccc(cc1)C(=O)NO)c1ccccc1S2 |c:4|
ONC(=O)c1ccc(cc1)N1c2ccccc2Sc2ccccc12
ONC(=O)c1ccc(CN2c3ccccc3Sc3cc(Cl)nnc23)cc1
ONC(=O)c1ccc(CCN2c3ccccc3Sc3ccccc23)cc1
ONC(=O)c1ccc(CN2c3ccccc3Sc3ccc(Cl)cc23)cc1
ONC(=O)c1ccc(CN2c3ccccc3Sc3ccc(cc23)C(F)(F)F)cc1
ONC(=O)c1ccc(CN2c3ccncc3Sc3ccncc23)cc1
ONC(=O)c1ccc(CN2N=C(Cl)C=C3Sc4ccccc4N=C23)cc1 |t:10,13,23|
ONC(=O)c1ccc(CN2c3ccccc3Sc3ccnnc23)cc1
CC(C)c1cc(C(=O)N(C)c2ccc(NC(=O)CCCCCCCC(=O)NO)cc2)c(O)cc1O
CC(C)c1cc(C(=O)N(C)c2ccc(NC(=O)CCCCCCC(=O)NO)cc2)c(O)cc1O
CC(C)(C)c1ccc(CNc2ccc(cc2)C(=O)NO)cc1
CN(C(=O)CN(Cc1c(F)c(F)c(F)c(F)c1F)S(=O)(=O)c1ccc(F)cc1)c1ccc(cc1)C(=O)NO
CN(CC(=O)N(Cc1ccc(cc1)C(C)(C)C)c1ccc(cc1)C(=O)NO)S(=O)(=O)c1ccc(F)cc1
CC(C)(C)c1ccc(CN(C(=O)CNS(=O)(=O)c2ccc(F)cc2)c2ccc(cc2)C(=O)NO)cc1
CN(CC(=O)N(C)c1ccc(cc1)C(=O)NO)S(=O)(=O)c1ccc(F)cc1
CC(C)(C)OC(=O)N(Cc1ccc(cc1)C(C)(C)C)c1ccc(cc1)C(=O)NO
CC(C)(C)c1ccc(cc1)C(=O)Nc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(cc1)N(Cc1ccccc1)C(=O)CN(Cc1c(F)c(F)c(F)c(F)c1F)S(=O)(=O)c1ccc(F)cc1
CC(C)(C)c1ccc(CN(C(=O)CN(Cc2c(F)c(F)c(F)c(F)c2F)S(=O)(=O)c2ccc(F)cc2)c2ccc(cc2)C(=O)NO)cc1
CC(C)(C)c1ccc(CN(C(=O)CN(Cc2c(F)c(F)c(F)c(F)c2F)S(C)(=O)=O)c2ccc(cc2)C(=O)NO)cc1
CC(=O)N(Cc1ccc(cc1)C(C)(C)C)c1ccc(cc1)C(=O)NO
COc1ccc(cc1)-c1nc(NCCOc2ccc(\C=C\C(=O)NO)cc2OC)cc2c3ccccc3[nH]c12
COc1ccc(cc1)-c1nc(NCCCOc2ccc(\C=C\C(=O)NO)cc2OC)cc2c3ccccc3[nH]c12
COc1ccc(cc1)S(=O)(=O)N1CCc2cccc(NCc3ccc(cc3)C(=O)Nc3ccccc3N)c12
CN(C)Cc1nn(Cc2ccc(cc2)C(=O)NO)c2ccccc12
ONC(=O)c1ccc(Cn2c3CCOCc3c3ccccc23)cc1
ONC(=O)c1ccc(Cn2c3CCCCc3c3ccccc23)cc1
CC(=O)N1CCc2c(C1)c1ccccc1n2Cc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(Cn2cc(CN3CCCC3)c3ccccc23)cc1
CC(C)(C)OC(=O)NCc1cn(Cc2ccc(cc2)C(=O)NO)c2ccccc12
c1ccc2c(c1)c(cn2Cc3ccc(cc3)C(=O)NO)CCO
CC(C)(C)c1cc2ccccc2n1Cc1ccc(cc1)C(=O)NO
COCCc1cn(Cc2ccc(cc2)C(=O)NO)c2ccccc12
CN1CCCC1c1cn(Cc2ccc(cc2)C(=O)NO)c2ccccc12
ONC(=O)c1ccc(Cn2c3CCSCc3c3ccccc23)cc1
Cn1cncc1-c1cn(Cc2ccc(cc2)C(=O)NO)c2ccccc12
ONC(=O)CCc1csc(CCc2cccs2)n1
COc1cc(CCc2nc(CCC(=O)NO)cs2)cc(OC)c1OC
ONC(=O)CCc1csc(CCc2ccc(O)c(O)c2)n1
ONC(=O)CCc1csc(CCc2ccc(cc2)C#N)n1
ONC(=O)CCCc1csc(Cc2ccccc2)n1
ONC(=O)CCc1csc(CCc2ccc(F)cc2)n1
ONC(=O)CCc1csc(CCc2ccc(F)c(F)c2)n1
ONC(=O)CCc1csc(\C=C\c2ccc(Cl)cc2)n1
ONC(=O)CCc1csc(CCc2cc(O)c(O)c(O)c2)n1
ONC(=O)CCc1csc(CCc2c[nH]c3ccccc23)n1
COc1ccc(CCc2nc(CCC(=O)NO)cs2)cc1OC
ONC(=O)CCc1csc(Cc2ccccc2)n1
ONC(=O)CCc1csc(\C=C\c2ccc(Br)cc2)n1
ONC(=O)CCc1csc(CCc2cccc(F)c2)n1
COc1ccc(CCc2nc(CCC(=O)NO)cs2)cc1
ONC(=O)CCc1csc(\C=C\c2ccc(F)cc2)n1
ONC(=O)CCc1csc(CCc2ccc(cc2)[N+]([O-])=O)n1
ONC(=O)CCc1csc(\C=C\c2c[nH]c3ccccc23)n1
ONC(=O)CCc1csc(CCc2ccc(O)cc2)n1
ONC(=O)CCc1csc(CCc2ccc(cc2)C(F)(F)F)n1
ONC(=O)CCc1csc(\C=C\c2ccccc2)n1
ONC(=O)CCCc1csc(CCc2ccccc2)n1
ONC(=O)CCc1csc(CCc2ccc(Br)cc2)n1
ONC(=O)CCc1csc(CCc2ccccc2)n1
ONC(=O)CCc1csc(CCc2ccco2)n1
ONC(=O)CCc1csc(CCc2ccc(Cl)cc2)n1
Nc1ccc(CCc2nc(CCC(=O)NO)cs2)cc1
COc1ccc2c(c1)nc(SCc1ccc(cc1)C(=O)Nc1ccccc1N)n(-c1ccccc1Cl)c2=O |(54.36,-40.98,;55.7,-40.21,;57.03,-40.98,;57.03,-42.53,;58.36,-43.3,;59.7,-42.52,;59.7,-40.97,;58.36,-40.21,;61.03,-40.19,;62.37,-40.96,;63.7,-40.19,;65.04,-40.96,;66.37,-40.18,;67.7,-40.95,;69.03,-40.18,;69.03,-38.64,;67.68,-37.87,;66.36,-38.65,;70.36,-37.86,;70.35,-36.32,;71.7,-38.63,;73.03,-37.85,;73.01,-36.32,;74.34,-35.54,;75.68,-36.3,;75.69,-37.84,;74.36,-38.62,;74.36,-40.16,;62.38,-42.51,;63.71,-43.28,;65.03,-42.5,;66.37,-43.26,;66.37,-44.81,;65.04,-45.58,;63.71,-44.82,;62.37,-45.59,;61.04,-43.28,;61.04,-44.82,)|
Cn1c(SCc2ccc(cc2)C(=O)Nc2ccccc2N)nc2cc(Br)ccc2c1=O
CCn1c(SCc2ccc(\C=C\C(=O)Nc3ccccc3N)cc2)nc2cc(OC)ccc2c1=O
COc1ccc2c(c1)nc(SCc1ccc(cc1)C(=O)Nc1ccccc1N)n(C)c2=O
COc1ccc(\C=C(/C)C(=O)c2cc(OC)c(OC)c(OC)c2)cc1OCCCC(=O)NO
COc1ccc(\C=C(/C)C(=O)c2cc(OC)c(OC)c(OC)c2)cc1OCCCCCCCC(=O)NO
COc1ccc(\C=C\C(=O)c2cc(OC)c(OC)c(OC)c2)cc1OCCCCCCC(=O)NO
Cc1cc(C)cc(SCc2ccc(cc2)C(=O)Nc2ccccc2N)c1
CCc1ccc(SCc2ccc(cc2)C(=O)Nc2ccccc2N)cc1
COc1ccc(SCc2ccc(cc2)C(=O)Nc2ccccc2N)cc1
Nc1ccccc1NC(=O)c1ccc(CSc2nccc(n2)C(F)(F)F)cc1
COC(=O)c1ccc2ccccc2c1OCCCCCCCC(=O)NO
C[C@@H](/C=C(\C)/C=C/C(=O)NO)C(=O)c1ccc(cc1)N(C)C
CN(C)c1cccc2c(cccc12)S(=O)(=O)N(CC(=O)NCc1ccccc1)Cc1ccc(cc1)C(=O)Nc1ccccc1N
CN(C)c1cccc2c(cccc12)S(=O)(=O)N(CC(=O)NCc1ccccc1)Cc1ccc(cc1)C(=O)NO
CN(C)c1cccc2c(cccc12)S(=O)(=O)N(CCCCCC(=O)NO)CC(=O)NCc1ccccc1
ONC(=O)\C=C\c1ccc(CONC(=O)c2ccc3ccccc3n2)cc1
COc1ccc(NC(=O)NOCc2ccc(\C=C\C(=O)NO)cc2)cc1
CC(=O)Nc1cccc(c1)-c1csc(NC(=O)CCCCCC(=O)Nc2ccccc2N)n1
Nc1ccccc1NC(=O)c1cnccn1
CC(C)(C)OC(=O)Nc1cccc(c1)-c1csc(NC(=O)CCCCCC(=O)Nc2ccccc2N)n1
CCOC(=O)Nc1cccc(c1)-c1csc(NC(=O)CCCCCC(=O)Nc2ccccc2N)n1
CC(C)(C)OC(=O)Nc1cccc(c1)-c1csc(NC(=O)CCCCCC(=O)NO)n1
CCOC(=O)Nc1cccc(c1)-c1csc(NC(=O)CCCCCC(=O)NO)n1
Nc1ccccc1NC(=O)c1ccc(CN2CC(=C)c3ccccc3C2=O)cc1
Nc1cccc(c1)-c1csc(NC(=O)CCCCCC(=O)NO)n1
Nc1cccc(c1)-c1csc(NC(=O)CCCCCC(=O)Nc2ccccc2N)n1
CC(C)(C)c1ccc(CN(C(=O)CN(Cc2ccccc2C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)c2ccc(cc2)C(=O)NO)cc1
ONC(=O)c1ccc(cc1)N(Cc1ccc(cc1)C(F)(F)F)C(=O)CN(Cc1ccccc1C(F)(F)F)S(=O)(=O)c1ccc(F)cc1F
ONC(=O)c1ccc(cc1)N(Cc1ccc(cc1)C(F)(F)F)C(=O)CN(Cc1ccccc1C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
ONC(=O)c1ccc(cc1)N(Cc1ccc(cc1)C(F)(F)F)C(=O)CN(Cc1c(F)c(F)c(F)c(F)c1F)S(=O)(=O)c1ccc(F)cc1
ONC(=O)c1ccc(cc1)N(Cc1ccc(cc1)C(F)(F)F)C(=O)CN(Cc1ccccc1C(F)(F)F)S(=O)(=O)c1ccc(F)c(F)c1
CC(C)(C)c1ccc(CN(C(=O)CN(Cc2ccccc2C(F)(F)F)S(=O)(=O)c2ccc(F)cc2F)c2ccc(cc2)C(=O)NO)cc1
CC(C)(C)c1ccc(CN(C(=O)CN(Cc2ccccc2C(F)(F)F)S(=O)(=O)c2ccc(F)c(F)c2)c2ccc(cc2)C(=O)NO)cc1
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(NCc3ccc(C(=O)NO)c(C)c3)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc(N)c1C#N)c1nc2cccc(NCc3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
C[C@H](Nc1nc(N)nc(C)c1C#N)c1nc2cccc(NCc3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc(CCCCC(=O)NO)c2ccccc2n1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(CNc3ncc(cn3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
C[C@H](Nc1nc(N)nc(N)c1C#N)c1nc2cccc(CNC(=O)c3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
C[C@H](Nc1nc(N)nc(N)c1C#N)c1nc2cccc(CNc3ncc(cn3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc(NCCCC(=O)NO)c2ccccc2n1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(CCc3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(-c3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(NCc3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(NCc3ccc(cn3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1nc(N)nc(C)c1C#N)c1nc2cccc(CCCCCC(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1nc(N)ncc1C)c1nc2cccc(CCCCCC(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1nc(N)nc(N)c1C#N)c1nc2cccc(CCc3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1cc(C)nc(N)n1)c1nc2cccc(NCc3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc(N)c1Cl)c1nc2cccc(NCc3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1nc(N)nc(C)c1Cl)c1nc2cccc(NCc3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1nc(C)nc(N)c1C#N)c1nc2cccc(NCc3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1nc(N)nc(c1C#N)C(F)(F)F)c1nc2cccc(NCc3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1nc(N)nc(C(F)F)c1C#N)c1nc2cccc(NCc3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
C[C@H](Nc1nc(N)nc(N)c1C#N)c1nc2cccc(NCc3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(CNC(=O)c3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc(CCCCCC(=O)NO)c2ccccc2n1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(NCCCC(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1nc(N)nc(N)c1C#N)c1nc2cccc(CCCCCC(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1nc(N)nc(N)c1C#N)c1nc2cccc(NCc3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc(N)c1Cl)c1nc2cccc(NCc3ccc(cn3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1nc(N)nc(C2CC2)c1C#N)c1nc2cccc(NCc3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(CCCCCC(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1nc(N)nc(C)c1C#N)c1nc2cccc(NCCCCC(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(CCCCC(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1nc(N)nc(C)c1C#N)c1nc2cccc(NCc3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1nc(N)nc(N)c1Cl)c1nc2cccc(NCc3ccc(cc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(NCc3ccc(nc3)C(=O)NO)c2c(=O)n1-c1ccccc1 |r|
Brc1cccc2SC(=S)N3CCCN=C3c12 |c:13|
Clc1ccc2SC(=S)N3CCN=C3c2c1 |c:11|
S=C1Sc2cc(ccc2C2=NCCCN12)C#N |t:10|
Fc1cc(Br)cc2SC(=S)N3CCN=C3c12 |c:13|
S=C1Sc2cc(ccc2C2=NCCN12)C#N |t:10|
Brc1ccc2SC(=S)N3CCN=C3c2c1 |c:11|
Clc1cccc2SC(=S)N3CCN=C3c12 |c:12|
Ic1ccc2SC(=S)N3CCN=C3c2c1 |c:11|
Cc1ccc2SC(=S)N3CCN=C3c2c1 |c:11|
Clc1ccc2C3=NCCN3C(=S)Sc2c1 |t:5|
Ic1cccc2SC(=S)N3CCN=C3c12 |c:12|
Clc1cccc2C3=NCCN3C(=S)Sc12 |t:6|
COc1ccc2SC(=S)N3CCN=C3c2c1 |c:12|
Fc1cccc2SC(=S)N3CCN=C3c12 |c:12|
Cc1ccc2C3=NCCN3C(=S)Sc2c1 |t:5|
Cc1ccc2SC(=S)N3CCCN=C3c2c1 |c:12|
Ic1cccc2SC(=S)N3CCCN=C3c12 |c:13|
Cc1cccc2SC(=S)N3CCCN=C3c12 |c:13|
Clc1ccc2SC(=S)N3CCCN=C3c2c1 |c:12|
FC(F)(F)c1ccc2SC(=S)N3CCCN=C3c2c1 |c:15|
Fc1ccc2C3=NCCCN3C(=S)Sc2c1 |t:5|
Brc1ccc2SC(=S)N3CCCN=C3c2c1 |c:12|
Fc1cccc2SC(=S)N3CCCN=C3c12 |c:13|
Clc1ccc2C3=NCCCN3C(=S)Sc2c1 |t:5|
Fc1cccc2C3=NCCCN3C(=S)Sc12 |t:6|
Cc1cccc2C3=NCCCN3C(=S)Sc12 |t:6|
S=C1Sc2ccccc2C2=NCCCN12 |t:10|
Fc1ccc2SC(=S)N3CCN=C3c2c1 |c:11|
Fc1cccc2C3=NCCN3C(=S)Sc12 |t:6|
Cc1ccc2C3=NCCCN3C(=S)Sc2c1 |t:5|
CN(C)c1ccc2C3=NCCCN3C(=S)Sc2c1 |t:7|
Brc1cccc2SC(=S)N3CCN=C3c12 |c:12|
COc1ccc2C3=NCCN3C(=S)Sc2c1 |t:6|
Brc1ccc2C3=NCCCN3C(=S)Sc2c1 |t:5|
O=C1Sc2ccccc2C2=NCCCN12 |t:10|
Brc1ccc2C3=NCCN3C(=S)Sc2c1 |t:5|
Cc1cccc2SC(=S)N3CCN=C3c12 |c:12|
CN(C)c1ccc2C3=NCCN3C(=S)Sc2c1 |t:7|
S=C1Sc2ccccc2C2=NCCN12 |t:10|
Clc1cccc2SC(=S)N3CCCN=C3c12 |c:13|
Ic1ccc2SC(=S)N3CCCN=C3c2c1 |c:12|
Fc1ccc2SC(=S)N3CCCN=C3c2c1 |c:12|
Clc1cccc2C3=NCCCN3C(=S)Sc12 |t:6|
Cc1cccc2C3=NCCN3C(=S)Sc12 |t:6|
Nc1ccc(cc1)-c1nc(N2CCOCC2)c2cnn(CCCCCCC(=O)NO)c2n1
C[C@@H]1CN(CCO1)C(=O)Nc1ccc(cc1)-c1nc(N2CCOCC2)c2cnn(CCCCCCC(=O)NO)c2n1 |r|
Nc1ccc(cc1)-c1nnn(Cc2c(F)cc(cc2F)C(=O)NO)n1
ONC(=O)c1cc(F)c(Cn2nnc(n2)-c2ccco2)c(F)c1
Cc1nnc([nH]1)-c1ccc(cc1)C(=O)NO
NCc1ccc(cc1)-c1nnn(Cc2ccc(cc2)C(=O)NO)n1
ONC(=O)c1ccc(cc1)-c1nnc(o1)-c1ccccc1
COc1ccccc1-n1nc(nc1Cc1ccc(cc1)C(=O)NO)-c1cccs1
Cc1csc(Nc2ccc(cc2)C(=O)NO)n1
ONC(=O)c1ccc(Cn2nnc(n2)-c2ncccn2)cc1
Cc1cc(nn1C)-c1nnc(Sc2c(F)c(F)c(C(=O)NO)c(F)c2F)n1C
Cn1c(Sc2c(F)cc(cc2F)C(=O)NO)nnc1-c1cccnn1
ONC(=O)c1ccc(Cc2nnc([nH]2)-c2ccccc2)cc1
ONC(=O)c1ccc(Sc2nnc(o2)-c2ccccc2)cc1
COc1ccc(CC(=O)N[C@@H](Cc2cscn2)C(=O)Nc2ccc(cc2)C(=O)NO)cc1OC |r|
c1cc(ccc1CN)C(=O)NO
ONC(=O)c1ccc(Cc2nnc[nH]2)cc1
ONC(=O)c1ccc(Cc2nnc(o2)-c2ccccc2)cc1
ONC(=O)c1ccc(Cn2nnc(n2)-c2ccccc2)cc1
ONC(=O)c1ccc(Cc2nnc(s2)-c2ccccc2)cc1
ONC(=O)c1ccc(Cn2nnnc2-c2ccccc2)cc1
Cn1c(Cc2ccc(cc2)C(=O)NO)nnc1-c1ccccc1
ONC(=O)c1ccc(Sc2nnc(-c3ccccc3)n2-c2ccccc2)cc1
Cc1cc(nn1C)-c1nnc(Sc2ccc(cc2)C(=O)NO)n1C
CCN(CC)S(=O)(=O)c1cccc(c1)-c1nnc(Sc2ccc(cc2)C(=O)NO)n1N
ONC(=O)c1ccc(Cc2nc(nn2Cc2ccccc2)-c2ccc(Cl)cc2)cc1
ONC(=O)c1ccc(Sc2ncc(s2)-c2ccccc2)cc1
ONC(=O)c1ccc(Cn2nnc(n2)-c2cccc(c2)S(F)(F)(F)(F)F)cc1
Nc1ccc(cc1)-c1nnn(Cc2ccc(cc2)C(=O)NO)n1
ONC(=O)c1ccc(Cn2nnc(n2)-c2ccccn2)cc1
ONC(=O)c1ccc(Cn2nnc(n2)-c2ccc3ccccc3n2)cc1
ONC(=O)c1ccc(Cn2nnc(n2)-c2nccc3ccccc23)cc1
ONC(=O)c1ccc(Cn2nnc(Cc3ccccn3)n2)cc1
NCc1ccc(cc1)-c1nnn(Cc2c(F)cc(cc2F)C(=O)NO)n1
ONC(=O)c1cc(F)c(Cn2nnc(n2)-c2nccc3ccccc23)c(F)c1
Cc1cc(nn1C)-c1nnc(Sc2c(F)cc(cc2F)C(=O)NO)n1C
Cc1cc(nn1C)-c1nnc(Sc2ccc(C(=O)NO)c(F)c2)n1C
Cn1c(Sc2c(F)cc(cc2F)C(=O)NO)nnc1-c1cccs1
ONC(=O)c1cc(F)c(Cc2nnc(s2)-c2ccncc2)c(F)c1
Cn1c(Sc2c(F)cc(cc2F)C(=O)NO)nnc1-c1cccc(CN2CCCCCC2)c1
ONC(=O)c1ccc(Cn2nnc(Cc3ccccc3)n2)cc1
ONC(=O)c1ccc(Cc2noc(n2)-c2ccccc2)cc1
ONC(=O)c1ccc(Nc2nnc(s2)-c2ccccc2)cc1
Cn1c(Sc2ccc(cc2)C(=O)NO)nnc1-c1cccs1
ONC(=O)c1ccc(Cn2nnc(n2)-c2ccc(cc2)S(F)(F)(F)(F)F)cc1
ONC(=O)c1ccc(Cn2nnc(n2)-c2cccc(c2)C(O)=O)cc1
ONC(=O)c1cc(F)c(Cn2nnc(n2)-c2ncccn2)c(F)c1
ONC(=O)c1cc(F)c(Cn2nnc(n2)-c2ccc3ccccc3n2)c(F)c1
ONC(=O)c1ccc(Cn2nnnc2-c2cccs2)cc1
Cn1c(Sc2c(F)cc(cc2F)C(=O)NO)nnc1-c1ncccc1F
ONC(=O)c1ccc(Sc2nnc(s2)-c2ccccc2)cc1
ONC(=O)c1cc(F)c(Cn2nnc(n2)-c2ccccn2)c(F)c1
ONC(=O)c1ccc(Nc2nnc(o2)-c2ccccc2)cc1
ONC(=O)c1ccc(Cn2nnc(n2)-c2ccc(cc2)C(F)(F)F)cc1
Cn1c(Sc2c(F)cc(cc2F)C(=O)NO)nnc1-c1ccc(CN2CCCCC2)cc1
ONC(=O)c1ccc(Sc2nc(C3CC3)n(n2)-c2ccccc2)cc1
Nc1ccc(cc1)C(=O)NO
CC(=O)Nc1ccc(cc1)C(=O)NO
[H][C@@]12CCCC[C@@]1([H])N(Cc1ccc(cc1)C(=O)NO)c1cc(ccc1CCC2)C(F)(F)F |r|
[H][C@]12CCCN1C(=O)[C@H](Cc1ccccc1)NC(=O)C1(CCCCC1C)NC(=O)[C@H](CCCCCC(=O)NO)NC2=O |r|
ONC(=O)c1ccc2CCC3(CCN(Cc4ccncc4)C3=O)Cc2c1
COc1cc(\C=C\C(=O)NO)ccc1OCCCCN(C)C(=O)c1ccccc1O
ONC(=O)\C=C\c1ccc(cc1)C(=O)NCCCOc1no[n+]([O-])c1S(=O)(=O)c1ccccc1
CCN(CC)c1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(Cn2c3CCSCc3c3cc(F)ccc23)cc1
ONC(=O)c1ccc(Cn2c3CCS(=O)(=O)Cc3c3ccccc23)cc1
ONC(=O)c1ccc(CN2C3CCS(=O)(=O)C3c3ccccc23)cc1
[H][C@]12Cc3ccccc3N(Cc3ccc(cc3)C(=O)NO)[C@]1([H])CCCCC2 |r|
[H][C@@]12CCCC[C@@]1([H])N(Cc1ccc(cc1)C(=O)NO)c1ccccc1CCC2 |r|
CC(C)CCc1c(OCCOc2cccc(\C=C\C(=O)NO)c2)ccc2CCC(=O)Oc12
CC(C)CCc1c(OCCCOc2cccc(\C=C\C(=O)NO)c2)ccc2CCC(=O)Oc12
CC(C)CCc1c(OCCCCOc2ccc(\C=C\C(=O)NO)cc2)ccc2CCC(=O)Oc12
CCn1cnc(c1-c1ccc(\C=C\C(=O)NO)cc1)-c1ccccc1
CCn1cnc(c1-c1ccc(\C=C\C(=O)NO)cc1)-c1ccc(OC)cc1
CC(C)N1CCC2(CCc3ccc(cc3C2)C(=O)NO)C1=O
ONC(=O)c1ccc2CCC3(CCN(Cc4cc(Cl)ccc4Cl)C3=O)Cc2c1
[H][C@]12CCCN1C(=O)[C@]1([H])CCCCCCCCCCC[C@@]([H])(NC(=O)[C@H](CCCCCB(O)O)NC2=O)C(=O)N1 |r|
[H][C@]12CCCN1C(=O)[C@H](Cc1ccccc1)NC(=O)C1(CCCC(C)C1)NC(=O)[C@H](CCCCCC(=O)NO)NC2=O |r|
CC(CNC(=O)c1ccc(\C=C\C(=O)NO)cc1)Oc1no[n+]([O-])c1S(=O)(=O)c1ccccc1
CNCCOc1no[n+]([O-])c1S(=O)(=O)c1ccccc1
COc1cc(\C=C\C(=O)NO)ccc1OCCCCNC(=O)c1ccccc1O
COc1cc(\C=C\C(=O)NO)ccc1OCCN(C)C(=O)c1ccccc1O
COc1cc(\C=C\C(=O)NO)ccc1OCCCN(C)C(=O)c1ccccc1O
OCCSSCCCCCC(NC(=O)OCc1ccccc1)C(=O)Nc1cccc2cccnc12
O=C(NC(CCCCCSSCCCCCC(NC(=O)OCc1ccccc1)C(=O)Nc1cccc2cccnc12)C(=O)Nc1cccc2cccnc12)OCc1ccccc1
[H][C@]12CCCCN1C(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCCCC(=O)[C@@H]1CO1)NC(=O)C2 |r|
[H][C@]12CCC(C)=C(CC[C@]3(C)CCC=C(C)[C@@]3([H])C1)C2(C)C |r,t:5,13|
[H][C@]12CCCN1C(=O)[C@]1([H])CCCCCCCCCCC[C@@]([H])(NC(=O)[C@H](CCCCCC(=O)COC)NC2=O)C(=O)N1 |r|
CC(=O)SCCCCCC(NC(=O)OCc1ccccc1)C(=O)Nc1cccc2cccnc12
ONC(=O)c1ccc(cc1)N1CCCC1
ONC(=O)c1ccc(Cn2c3CCS(=O)(=O)Cc3c3cc(F)ccc23)cc1
[H][C@@]12CCCC[C@@]1([H])N(Cc1ccc(cc1)C(=O)NO)c1ccccc1CC2 |r|
Nc1ccccc1NC(=O)CCCCCCC(=O)Nc1ccc(cc1)-c1cn(Cc2ccccc2)nn1
[H][C@]12CCCN1C(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCCCC(=O)[C@@H]1CO1)NC(=O)C2 |r|
ONC(=O)c1ccc(Cn2c3CC[S+]([O-])Cc3c3cc(F)ccc23)cc1
ONC(=O)\C=C\c1cccn(CCc2ccc3ccccc3c2)c1=O
ONC(=O)c1ccc2CCC3(CCN(Cc4ccccc4OC(F)(F)F)C3=O)Cc2c1
COc1cc(\C=C\C(=O)NO)ccc1OCCCNC(=O)c1ccccc1O
COCCOCC(=O)SCCCCCC(NC(=O)OCc1ccccc1)C(=O)Nc1cccc2cccnc12
ONC(=O)\C=C\c1cccn(CCCc2ccc3ccccc3c2)c1=O
CN(C)Cc1c(C)n(-c2ccc(cc2)C(=O)NO)c2ccccc12
[H][C@@]12CCCC[C@@]1([H])N(Cc1ccc(cc1)C(=O)NO)c1ccccc1C2 |r|
Nc1cccc(c1)-c1csc(NC(=O)CCCCCCC(=O)Nc2ccccc2N)n1
ONC(=O)\C=C\c1ccc(cc1)C(=O)NCCOc1no[n+]([O-])c1S(=O)(=O)c1ccccc1
CC(C)CCc1c(OCCOc2ccc(\C=C\C(=O)NO)cc2)ccc2CCC(=O)Oc12
ONC(=O)c1ccc2C(=O)c3ccccc3C(=O)c2c1
ONC(=O)\C=C\c1ccc2C(=O)c3ccccc3C(=O)c2c1
ONC(=O)[C@H](Cc1ccccc1)n1nnc(c1C#Cc1ccccc1)-c1ccccc1 |r|
ONC(=O)[C@H](Cc1ccccc1)n1nnc(c1C#CC1CC1)-c1ccccc1 |r|
ONC(=O)CCCCNC(=S)Nc1ccc2C(=O)NC(=O)c2c1
ONC(=O)CCNC(=S)Nc1ccc2C(=O)NC(=O)c2c1
ONC(=O)CCCCCNC(=S)Nc1ccc2C(=O)NC(=O)c2c1
ONC(=O)CCCNC(=S)Nc1ccc2C(=O)NC(=O)c2c1
COc1cccc(CCCCCCCC(=O)NO)c1
COC(=O)c1c(CCCCCCCC(=O)NO)cccc1OC
ONC(=O)\C=C\c1ccc(cc1)C(=O)NC(Cc1c[nH]c2ccccc12)C(=O)Nc1ccc(I)cc1
ONC(=O)\C=C\c1ccc(cc1)C(=O)NC(Cc1c[nH]c2ccccc12)C(=O)Nc1cccc(Br)c1
ONC(=O)\C=C\c1ccc(cc1)C(=O)NC(Cc1c[nH]c2ccccc12)C(=O)Nc1ccc2ccccc2c1
ONC(=O)\C=C\c1ccc(cc1)C(=O)NC(Cc1c[nH]c2ccccc12)C(=O)Nc1ccc(Cl)cc1
ONC(=O)\C=C\c1ccc(cc1)C(=O)NC(Cc1c[nH]c2ccccc12)C(=O)Nc1ccc(Br)cc1
ONC(=O)CCC(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
ONC(=O)CCCC(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
ONC(=O)CCCCC(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
ONC(=O)CCCCCC(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
ONC(=O)CCCCCCC(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
ONC(=O)CCCCCCCC(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
ONC(=O)CCCCCCCCC(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
ONC(=O)c1ccc(CNCCCN2c3ccccc3CCc3ccc(Cl)cc23)cc1
ONC(=O)c1ccc(cc1)C(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
ONC(=O)\C=C\c1ccc(CNCCCN2c3ccccc3CCc3ccc(Cl)cc23)cc1
ONC(=O)\C=C\c1cccc(c1)S(=O)(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
ONC(=O)\C=C\c1ccc(cc1)S(=O)(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc12
ONC(=O)c1ccc(NCc2csc3ccccc23)cc1
CC(C)[C@H](NC(=O)C1Cc2ccccc2O1)C#Cc1ccc(cc1)C(=O)NO |r|
COc1cc(cc(OC)c1OC)C(=O)NOCCCCCC(=O)NO
CC(C)(C)c1cc(cc(c1)C(C)(C)C)C(=O)NOCCCCCC(=O)NO
ONC(=O)CCCCCONC(=O)c1cc(F)cc(F)c1
COc1cc(OC)cc(c1)C(=O)NOCCCCCC(=O)NO
ONC(=O)CCCCCONC(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F
ONC(=O)CCCCCONC(=O)c1cc(Br)cc(Br)c1
ONC(=O)CCCCCONC(=O)c1cc(I)cc(I)c1I
ONC(=O)CCCCCONC(=O)c1c(Cl)cncc1Cl
Cc1cc(C)cc(c1)C(=O)NOCCCCC(=O)NO
COc1ccc(cc1)-c1ccc2nc(\C=C\C(=O)NO)ccc2c1
ONC(=O)\C=C\c1ccc2cc(Oc3ccc(cc3)[N+]([O-])=O)ccc2n1
COc1cc(Oc2ccc3nc(\C=C\C(=O)NO)ccc3c2)cc(OC)c1OC
COc1ccc(Oc2ccc3nc(\C=C\C(=O)NO)ccc3c2)cc1
c1cc2c(cc1C(=O)O)nc(c3c2cncc3)NCCCCCCCC(=O)NO
ONC(=O)c1ccc(CN2CCc3ccc(F)cc23)cc1
Cc1cc(C(=O)NCc2c(C)cc(C)[nH]c2=O)c(C)n1-c1cccc(NC(=O)CCCCCCC(=O)NO)c1
Cc1c(cnn1-c1cccc(NC(=O)CCCCCCC(=O)NO)c1)C(=O)NCc1c(C)cc(C)[nH]c1=O
CC(=O)Nc1ccc2CN(Cc2c1)C(=O)[C@H](N)Cc1ccc(Cl)cc1Cl
CCCCC[C@H](CC(=O)NO)C(=O)N[C@@H](C(C)C)C(=O)N1CCC[C@H]1CO
ONC(=O)C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1c1nc(no1)-c1ccccc1 |r|
ONC(=O)C[C@@H](CC1CCCC1)C(=O)N1CC2(CC2)C[C@H]1c1nc(no1)-c1ccc(F)cc1C(F)(F)F |r|
CC(C)(C)c1cccc(c1)C(=O)Nc1ccc(cc1)C(=O)NO
CCN(C(=O)c1cccc(c1)C(C)(C)C)c1ccc(cc1)C(=O)NO
CCN(c1ccc(cc1)C(=O)NO)S(=O)(=O)c1cccc(c1)C(C)(C)C
CCN(C(=O)c1cccc(c1)C(F)(F)F)c1ccc(cc1)C(=O)NO
CCN(c1ccc(cc1)C(=O)NO)S(=O)(=O)c1cccc(c1)C(F)(F)F
CCN(c1ccc(cc1)C(=O)NO)S(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F
CCN(C(=O)c1cc(cc(c1)C(C)(C)C)C(C)(C)C)c1ccc(cc1)C(=O)NO
CC(C)(C)c1cc(CN(C(=O)c2cccc(c2)C(F)(F)F)c2ccc(cc2)C(=O)NO)cc(c1)C(C)(C)C
ONC(=O)c1ccc(cc1)N(Cc1cccc(c1)C(F)(F)F)C(=O)c1cccc(c1)C(F)(F)F
ONC(=O)c1ccc(cc1)N(Cc1ccccc1)C(=O)c1cccc(c1)C(F)(F)F
ONC(=O)c1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1
CCN(C(=O)c1ccccc1C(F)(F)F)c1ccc(cc1)C(=O)NO
CC(=O)N(Cc1cccc(c1)C(F)(F)F)c1ccc(cc1)C(=O)NO
CC(=O)N(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(cc1)N(CC1CC1)C(=O)c1cccc(c1)C(F)(F)F
CC(C)N(C(=O)c1cccc(c1)C(F)(F)F)c1ccc(cc1)C(=O)NO
CC(C)(C)c1cccc(c1)C(=O)N(CC1CC1)c1ccc(cc1)C(=O)NO
CC(C)(C)c1cc(cc(c1)C(C)(C)C)C(=O)N(CC1CC1)c1ccc(cc1)C(=O)NO
CC(C)(C)c1cc(cc(c1)C(C)(C)C)C(=O)Nc1ccc(cc1)C(=O)NO
CC(C)N(C(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1ccc(cc1)C(=O)NO
CC(C)N(C(=O)c1cccc(OC(F)(F)F)c1)c1ccc(cc1)C(=O)NO
CC(C)N(C(=O)c1cccc(c1F)C(F)(F)F)c1ccc(cc1)C(=O)NO
CC(C)N(C(=O)c1ccc(F)c(c1)C(F)(F)F)c1ccc(cc1)C(=O)NO
CC(C)N(C(=O)c1cc(cc(c1)C(C)(C)C)C(C)(C)C)c1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(NC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)cc1
CC(C)(C)c1cccc(NC(=O)c2ccc(cc2)C(=O)NO)c1
CCN(C(=O)c1ccc(cc1)C(=O)NO)c1cccc(c1)C(C)(C)C
NCCCNCCCCCC(=O)C(F)(F)F
CN(C)S(=O)(=O)c1ccc(NCCCCCC(=O)NO)c2nonc12
CN(C)S(=O)(=O)c1ccc(NCCCCCCC(=O)NO)c2nonc12
CCC(=O)CCCCC[C@H](NC(=O)[C@@H]1CC11CN(C)C1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CN(C)C1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)C1CC2(C1)CN(C)C2)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)CC1CC2(C1)CN(C)C2)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)C1CCC2(CN(C)C2)CC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1C[C@]11CCN(C)C1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1C[C@@]11CCN(C)C1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@@H]1C[C@]11CCN(C)C1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@@H]1C[C@@]11CCN(C)C1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@@H]1CC11CCCN(C)C1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCCN(C)C1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCN1CCC2(CC[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2cc3ccccc3nc2OC)CC1 |r|
CCN1CCC2(CC[C@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2cc3ccccc3nc2OC)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)C1=NOC2(C1)CCN(C)CC2)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r,t:13|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCC(CC1)N(C)C)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r,wD:9.9,13.12,(21.19,-2.07,;19.64,-2.07,;18.88,-3.41,;19.65,-4.74,;17.34,-3.41,;16.57,-4.75,;15.03,-4.75,;14.26,-6.09,;12.72,-6.09,;11.95,-7.43,;12.72,-8.76,;14.27,-8.76,;15.03,-7.42,;15.03,-10.08,;15.04,-11.61,;16.36,-10.84,;17.12,-12.17,;18.64,-12.17,;19.41,-10.85,;18.65,-9.53,;17.12,-9.52,;20.94,-10.86,;21.7,-12.19,;21.72,-9.54,;10.41,-7.43,;9.64,-6.1,;8.13,-6.43,;7.98,-7.96,;9.39,-8.57,;6.66,-8.74,;5.32,-7.97,;3.99,-8.75,;2.65,-7.98,;1.32,-8.76,;1.32,-10.3,;2.66,-11.07,;3.99,-10.3,;5.33,-11.06,;6.66,-10.29,;8,-11.05,;8.01,-12.59,)|
CCC(=O)CCCCC[C@H](NC(=O)[C@@H]1CC11CCC(CC1)N(C)C)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r,wU:13.12,wD:9.9,(49.9,-2.06,;48.36,-2.06,;47.6,-3.4,;48.37,-4.74,;46.06,-3.4,;45.28,-4.74,;43.74,-4.74,;42.98,-6.08,;41.44,-6.08,;40.66,-7.42,;41.44,-8.75,;42.98,-8.75,;43.75,-7.41,;43.75,-10.08,;43.76,-11.61,;45.08,-10.83,;45.84,-12.16,;47.35,-12.16,;48.13,-10.85,;47.37,-9.52,;45.84,-9.51,;49.66,-10.85,;50.42,-12.19,;50.43,-9.53,;39.13,-7.42,;38.35,-6.09,;36.85,-6.42,;36.7,-7.95,;38.1,-8.57,;35.37,-8.73,;34.03,-7.97,;32.7,-8.74,;31.37,-7.98,;30.04,-8.75,;30.03,-10.3,;31.37,-11.06,;32.71,-10.29,;34.04,-11.05,;35.38,-10.28,;36.72,-11.04,;36.72,-12.58,)|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCOCC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@@H]1CC11CCOCC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2cc3ccccc3nc2OC)CC1 |r|
CCCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2cc3ccccc3nc2OC)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC1)C(C)C)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC2CC2)CC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC1)C(C)=O)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC(F)(F)F)CC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CCC(F)(F)F)CC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(Cc2ccccc2)CC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(Cc2ccc(OC)cc2)CC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(Cc2cccnc2)CC1)c1ncc([nH]1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc(o1)-c1cc2ccccc2nc1OC |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc(o2)-c2cc3ccccc3nc2OC)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC1)C(C)C)c1ncc(o1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1nnc(o1)-c1cc2ccccc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1nnc([nH]1)-c1cc2ccccc2nc1OC |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2nnc([nH]2)-c2cc3ccccc3nc2OC)CC1 |r|
CN1CCN(CC1)c1ccc(c(N)c1)[N+]([O-])=O
CN1CC(C1)C(=O)N[C@@H](CCCCCC(=O)c1ncco1)c1ncc([nH]1)-c1ccc(F)cc1 |r|
CN1CCC(CC1)C(=O)N[C@@H](CCCCCC(=O)c1nccs1)c1ncc([nH]1)-c1ccc(F)cc1 |r|
CN1CCC(CC1)C(=O)N[C@@H](CCCCCC(=O)c1nc(C)co1)c1ncc([nH]1)-c1ccc(F)cc1 |r|
CN1CC(C1)C(=O)N[C@@H](CCCCCC(=O)c1cc(C)on1)c1ncc([nH]1)-c1ccccc1F |r|
CN1CCC(CC1)C(=O)N[C@@H](CCCCCC(=O)c1ccccn1)c1ncc([nH]1)-c1ccccc1 |r|
N[C@@H](CCCCCC(=O)c1ccon1)c1ncc([nH]1)-c1ccccc1F |r|
N[C@@H](CCCCCC(=O)c1cocn1)c1ncc([nH]1)-c1ccccc1F |r|
COc1nc2ccccc2cc1-c1cnc([nH]1)[C@@H](N)CCCCCC(=O)c1cnoc1C |r|
N[C@@H](CCCCCC(=O)c1ccon1)c1cnn(n1)-c1ccc(F)cc1 |r|
N[C@@H](CCCCCC(=O)c1ccon1)c1cnn(c1)-c1ccc(F)cc1 |r|
CN1CC(C1)C(=O)N[C@@H](CCCCCC(=O)c1ccon1)c1ncc(o1)-c1ccccc1F |r|
O=C(NC(c1ccccc1)c1ccccc1)c1cc(nc2ccccc12)-c1cc2ccccc2o1
CCc1nc(N)nc(N)c1-c1ccc(cc1)-c1cn(CCCCCC(=O)NO)nn1
CCc1nc(N)nc(N)c1-c1ccc(cc1)-c1cn(CCCCCCC(=O)NO)nn1
CCc1nc(N)nc(N)c1-c1ccc(cc1)-c1cn(CCCCCCCC(=O)NO)nn1
CCc1nc(N)nc(N)c1-c1ccc(\C=C\C(=O)NO)cc1
CCc1nc(N)nc(N)c1-c1ccc(cc1)-c1ccc(\C=C\C(=O)NO)cc1
COc1cc(ccc1O)C(=O)OCCCCCCCOC(=O)c1ccc(O)c(OC)c1
[H][C@@]12CCCC[C@]1([H])N(Cc1ccc(cc1)C(=O)NO)c1ccccc1S(=O)(=O)C2 |r|
ONC(=O)c1ccc(Cn2c(=O)c(F)cn(C3CCCO3)c2=O)cc1
CN(C)c1ccc(cc1)C(=O)N(CC(=O)NC1CCCCC1)Cc1ccc(cc1)C(=O)NO
C\C(\C=C\C(=O)NO)=C/c1ccc(NS(=O)(=O)c2ccc(cc2)N(CCCl)CCCl)cc1
CN(C)c1cccc2c(cccc12)S(=O)(=O)NCCCCCC(=O)NO
COC(=O)[C@@H](Cc1ccccn1)NC(=O)CCCCCCC(=O)NO |r|
COC(=O)[C@H](Cc1ccccn1)NC(=O)CCCCCCC(=O)NO |r|
O=C(NC1=CC(=O)c2ccccc2C1=O)c1ccccc1 |t:3|
Nc1cc(F)ccc1NC(=O)\C=C\c1cnn(C\C=C\c2ccccc2)c1
Nc1ccccc1NC(=O)CCCCCCCNC(=O)C(\Cc1ccc(O)c(Br)c1)=N\O
Nc1ccccc1NC(=O)CCCCCCNC(=O)C(\Cc1ccc(O)c(Br)c1)=N\O
Nc1ccccc1NC(=O)CCCCCNC(=O)C(\Cc1ccc(O)c(Br)c1)=N\O
Nc1ccccc1NC(=O)CCCCNC(=O)C(\Cc1ccc(O)c(Br)c1)=N\O
Nc1ccccc1NC(=O)CCCNC(=O)C(\Cc1ccc(O)c(Br)c1)=N\O
Nc1ccccc1NC(=O)CCNC(=O)C(\Cc1ccc(O)c(Br)c1)=N\O
Nc1ccccc1NC(=O)CNC(=O)C(\Cc1ccc(O)c(Br)c1)=N\O
ONC(=O)CCCCNC(=O)C(\Cc1ccc(O)c(Br)c1)=N\O
ONC(=O)CNC(=O)C(\Cc1ccc(O)c(Br)c1)=N\O
O\N=C(/Cc1ccc(O)c(Br)c1)C(=O)NCCC(O)=O
OCCNC(=O)C(\Cc1ccc(O)c(Br)c1)=N\O
CCCCNC(=O)C(\Cc1ccc(O)c(Br)c1)=N\O
CCCNC(=O)C(\Cc1ccc(O)c(Br)c1)=N\O
CCCCCCCC(=O)SCC\C=C\[C@@H]1CC(=O)NCc2cccc(n2)-c2cccc(n2)C(=O)N[C@@H](C(C)C)C(=O)O1 |r|
[H][C@@]12C[C@](C)(CC[C@]1(C)CC[C@]1(C)C2=CC(=O)[C@@]2([H])[C@@]1(C)CC[C@@]1([H])C(C)(C)C(=O)C(=C[C@]21C)C#N)C(=O)N1CCN(CC1)c1ccc(NC(=O)CCCCCCC(=O)NO)cc1 |r,c:33,t:15|
COc1ccc(\C=C\C(=O)c2nnn(c2C)-c2ccc(Cl)cc2)cc1OC
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1cnccn1)B(O)O |r|
Nc1ccccc1NC(=O)c1ccc(CNC(=O)c2n[nH]cc2NC(=O)c2c(Cl)cccc2Cl)cc1
Nc1ccccc1NC(=O)Cc1ccc(NC(=O)c2n[nH]cc2NC(=O)c2c(Cl)cccc2Cl)cc1
CC(C)c1cc(C(=O)N2Cc3ccc(NCc4ccc(cc4)C(=O)NO)cc3C2)c(O)cc1O
CC(C)c1cc(C(=O)N2Cc3ccc(NC(=O)CCC(=O)NO)cc3C2)c(O)cc1O
CC(C)c1cc(C(=O)N2Cc3ccc(NC(=O)CCCC(=O)NO)cc3C2)c(O)cc1O
CC(C)c1cc(C(=O)N2Cc3ccc(NC(=O)CCCCC(=O)NO)cc3C2)c(O)cc1O
CC(C)c1cc(C(=O)N2Cc3ccc(NC(=O)CCCCCC(=O)NO)cc3C2)c(O)cc1O
CC(C)c1cc(C(=O)N2Cc3ccc(NC(=O)CCCCCCC(=O)NO)cc3C2)c(O)cc1O
CC(C)c1cc(C(=O)N2Cc3ccc(NC(=O)CCCCCCCC(=O)NO)cc3C2)c(O)cc1O
CC(C)c1cc(C(=O)N2Cc3ccc(NC(=O)CCCCCCCCC(=O)NO)cc3C2)c(O)cc1O
CC(C)c1cc(C(=O)N2Cc3ccc(\C=C\C(=O)NO)cc3C2)c(O)cc1O
ONC(=O)c1ccc(Nc2c3ccccc3nc3ccccc23)cc1
ONC(=O)Cc1ccc(Nc2c3ccccc3nc3ccccc23)cc1
ONC(=O)c1cccc(Nc2c3ccccc3nc3ccccc23)c1
ONC(=O)c1ccc(Nc2c3ccccc3nc3ccc(F)cc23)cc1
ONC(=O)c1ccc(Nc2c3ccccc3nc3ccc(Br)cc23)cc1
ONC(=O)c1ccc(Nc2c3ccccc3nc3ccc(OC(F)(F)F)cc23)cc1
ONC(=O)c1ccc(Nc2c3ccccc3nc3ccc(OCc4ccccc4)cc23)cc1
COc1cc2nc3ccccc3c(Nc3ccc(cc3)C(=O)NO)c2c(OC)c1OC
COc1ccc2nc3cc(Cl)ccc3c(Nc3ccc(cc3)C(=O)NO)c2n1
ONC(=O)c1ccc(Nc2c3CCCCc3nc3ccccc23)cc1
ONC(=O)c1ccc(Nc2ccnc3ccccc23)cc1
FC(F)(F)c1nc(no1)-c1ccc(cc1)C(=O)NCCN1CCCC1
C[C@H](CN1CCC[C@@H]1C)NC(=O)c1ccc(cc1)-c1noc(n1)C(F)(F)F |r|
ONC(=O)c1ccc(CN2C(=O)\C(=C3/Nc4ccccc4/C/3=N\O)c3ccccc23)cc1
ONC(=O)c1ccc(CN2C(=O)\C(=C3/Nc4ccccc4/C/3=N\O)c3cc(F)ccc23)cc1
ONC(=O)c1ccc(CN2C(=O)\C(=C3/Nc4ccccc4/C/3=N\O)c3cc(Cl)ccc23)cc1
ONC(=O)c1ccc(CN2C(=O)\C(=C3/Nc4ccccc4/C/3=N\O)c3cccc(Cl)c23)cc1
ONC(=O)c1ccc(CN2C(=O)\C(=C3/Nc4ccccc4/C/3=N\O)c3cc(Br)ccc23)cc1
Cc1ccc2N(Cc3ccc(cc3)C(=O)NO)C(=O)\C(=C3/Nc4ccccc4/C/3=N\O)c2c1
COc1ccc2N(Cc3ccc(cc3)C(=O)NO)C(=O)\C(=C3/Nc4ccccc4/C/3=N\O)c2c1
C\C(=N/NC(=S)NCCCCCC(=O)NO)c1ccc(Br)cc1
C\C(=N/NC(=S)NCCCCCC(=O)NO)c1ccc(F)cc1
C\C(=N/NC(=S)NCCCCCC(=O)NO)c1cccc(Br)c1
ONC(=O)CCCCCNC(=S)N\N=C(/c1ccccc1)c1cccc(c1)[N+]([O-])=O
[#6]-[#7](-[#6])-[#6](=S)-[#7]\[#7]=[#6](\c1ccccn1)-c1ccccn1
Nc1ccc(cn1)-c1nc(N2CCOCC2)c2ncn(CCCCCCC(=O)NO)c2n1
OCc1cccc(c1)-c1nc(N2CCOCC2)c2ncn(CCCCCCC(=O)NO)c2n1
Nc1ncc(cn1)-c1nc(N2CCOCC2)c2ccn(CCCCCCC(=O)NO)c2n1
CS(=O)(=O)N1CCN(Cc2cc3nc(nc(N4CCOCC4)c3s2)-c2cccc3[nH]ncc23)CC1
Cc1ccc(cc1)C(=O)Nc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(NC(=O)c2ccc(cc2)C2CC2)cc1
ONC(=O)c1ccc(NC(=O)c2ccc(cc2)C2CCCCC2)cc1
ONC(=O)c1ccc(NC(=O)c2ccc(cc2)N2CCOCC2)cc1
ONC(=O)c1ccc(NC(=O)c2ccc(cc2)C(F)(F)F)cc1
ONC(=O)c1ccc(NC(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(NC(=O)c2ccc(F)cc2)cc1
CC(C)(C)c1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)C(=O)NO
CC(C)(C)c1ccc(CC(=O)Nc2ccc(cc2)C(=O)NO)cc1
ONC(=O)c1ccc(CNC(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
CC(C)(C)c1ccc(cc1)C(=O)NCc1ccc(cc1)C(=O)NO
CC(C)(C)c1ccc(cc1)S(=O)(=O)NCc1ccc(cc1)C(=O)NO
CC(C)N(Cc1ccc(cc1)C(=O)NO)C(=O)c1c(F)c(F)c(F)c(F)c1F
CC(C)(C)c1ccc(cc1)C(=O)N(Cc1ccc(cc1)C(=O)NO)C1CC1
ONC(=O)c1ccc(CN(C2CC2)C(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
ONC(=O)\C=C\c1ccc(CNC(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
ONC(=O)\C=C\c1ccc(CN(C2CC2)C(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
CC(C)(C)c1ccc(NC(=O)c2ccc(cc2)C(=O)NO)cc1
CC(C)(C)c1ccc(NS(=O)(=O)c2ccc(cc2)C(=O)NO)cc1
CCN(C(=O)c1ccc(cc1)C(C)(C)C)c1ccc(cc1)C(=O)NO
CN(Cc1ccc(cc1)C(=O)NO)C(=O)c1c(F)c(F)c(F)c(F)c1F
ONC(=O)Cc1ccc(OCCCn2c3CNCCc3c3cccc(Cl)c23)cc1
ONC(=O)c1cnc(nc1)N1CCC2(CCN(Cc3c[nH]c4ccccc34)C2)CC1
ONC(=O)c1ccc(NC(=O)Nc2ccc(Cl)cc2)cc1
ONC(=O)\C=C\c1ccc(NC(=O)Nc2ccc(Cl)cc2)cc1
ONC(=O)CCc1ccc(NC(=O)Nc2ccc(Cl)cc2)cc1
CC(C)(Nc1ncc(cc1F)C(=O)NO)c1ccccc1
[H][C@]12CC(=O)N[C@H](C(C)C)C(=O)N[C@]([H])(CSSCC\C=C\1)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)O2 |r,t:20|
[H][C@]12CC(=O)N[C@H](C(C)C)C(=O)N[C@]([H])(CSSCC\C=C\1)C(=O)N[C@H](CC(C)C)C(=O)NCC(=O)O2 |r,t:20|
[H][C@]12CC(=O)N[C@H](C(C)C)C(=O)N[C@]([H])(CSSCC\C=C\1)C(=O)N[C@@H](Cc1ccccc1)C(=O)NCC(=O)O2 |r,t:20|
[H][C@]12CC(=O)N[C@H](C(C)C)C(=O)N[C@]([H])(CSSCC\C=C\1)C(=O)N[C@H](Cc1ccccc1)C(=O)NCC(=O)O2 |r,t:20|
[H][C@]12CC(=O)N[C@H](C(C)C)C(=O)N[C@]([H])(CSSCC\C=C\1)C(=O)N[C@@H](C)C(=O)NCC(=O)O2 |r,t:20|
[H][C@]12CC(=O)N[C@H](C(C)C)C(=O)N[C@]([H])(CSSCC\C=C\1)C(=O)N[C@H](C)C(=O)NCC(=O)O2 |r,t:20|
[H][C@]12CC(=O)N[C@H](C(C)C)C(=O)N[C@]([H])(CSSCC\C=C\1)C(=O)NCC(=O)NCC(=O)O2 |r,t:20|
[H][C@]12CC(=O)N[C@H](C(C)C)C(=O)N[C@]([H])(CSSCC\C=C\1)C(=O)N\C(=C/C)C(=O)NCC(=O)O2 |r,t:20|
OC(=O)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 |r|
ONC(=O)c1cnc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)s1 |r|
ONC(=O)c1coc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)n1 |r|
ONC(=O)c1csc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)n1 |r|
ONC(=O)c1ccc(CCCN2CCc3cc(CN[C@H]4C[C@@H]4c4ccc(F)cc4)ccc3C2)cc1 |r|
COc1ccc(cc1)[C@H]1C[C@@H]1NCc1cn2CCN(CCCc3ccc(cc3)C(=O)NO)Cc2n1 |r|
ONC(=O)c1ccc(CCCN2CC(CN[C@H]3C[C@@H]3c3ccccc3)C2)cc1 |r|
ONC(=O)c1ccc(CCN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 |r|
CN(C)CCNC(=O)c1ccc(cc1)[C@H]1C[C@@H]1NCC1CCN(CCCc2ccc(cc2)C(=O)NO)CC1 |r|
ONC(=O)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccc(cc3)C(=O)N3CCCCC3)CC2)cc1 |r|
ONC(=O)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccc(cc3)C(=O)N3CCOCC3)CC2)cc1 |r|
Cc1noc(C)c1-c1ccc(cc1)[C@H]1C[C@@H]1NCC1CCN(CCCc2ccc(cc2)C(=O)NO)CC1 |r|
Cn1cc(cn1)-c1ccc(cc1)[C@H]1C[C@@H]1NCC1CCN(CCCc2ccc(cc2)C(=O)NO)CC1 |r|
ONC(=O)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccc(cc3)-c3ccc(nc3)C(F)(F)F)CC2)cc1 |r|
Cn1ccc(cc1=O)-c1ccc(cc1)[C@H]1C[C@@H]1NCC1CCN(CCCc2ccc(cc2)C(=O)NO)CC1 |r|
ONC(=O)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccc(cc3)-c3ccc(cc3)C#N)CC2)cc1 |r|
ONC(=O)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccc(cc3)-c3ccc(F)cc3)CC2)cc1 |r|
ONC(=O)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccc(cc3)-c3ccc(Cl)cc3)CC2)cc1 |r|
ONC(=O)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccc(OCc4ccc(F)cc4)cc3)CC2)cc1 |r|
COc1ccc(cc1)[C@H]1C[C@@H]1NCC1CCN(CCCc2ccc(cc2)C(=O)NO)CC1 |r|
ONC(=O)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccc(F)cc3)CC2)cc1 |r|
COCCOc1cc2ncnc(Nc3ccc(\C=C\C(=O)NO)cc3)c2cc1OCCOC
CC[N+]1=C(C=CC2=C3Oc4cc(O)cc(OCCCCCCCC(O)=O)c4C=C3CCC2)C(C)(C)c2ccccc12
CC[N+]1=C(C=CC2=C3Oc4cc(O)cc(OCCCCCCCC(=O)NO)c4C=C3CCC2)C(C)(C)c2ccccc12
CC(C)(C)n1nnnc1CNCc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(CNCc2nnnn2Cc2ccccc2)cc1
ONC(=O)c1ccc(CNCc2nnnn2C2CCCCC2)cc1
ONC(=O)c1ccc(CNC(c2nnnn2C2CCCCC2)c2ccccc2)cc1
ONC(=O)c1ccc(CNC(c2nnnn2Cc2ccccc2)c2ccccc2)cc1
CCCCC(NCc1ccc(cc1)C(=O)NO)c1nnnn1Cc1ccccc1
ONC(=O)c1ccc(CN(Cc2nnnn2C2CCCCC2)C(=O)c2ccccc2)cc1
Cc1ccccc1C(=O)N(Cc1nnnn1C1CCCCC1)Cc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(CN(Cc2nnnn2Cc2ccccc2)C(=O)c2ccccc2)cc1
Cc1cc(C)cc(c1)C(=O)N(Cc1nnnn1Cc1ccccc1)Cc1ccc(cc1)C(=O)NO
CC(C)c1ccc(cc1)C(=O)N(Cc1nnnn1Cc1ccccc1)Cc1ccc(cc1)C(=O)NO
c1ccc(cc1)Cn2c(nnn2)CN(Cc3ccc(cc3)C(=O)NO)C(=O)c4ccccc4C(F)(F)F
C[C@H](NC(=O)[C@H](CC(=O)NC(C)(C)C)NC(=O)c1ccc(cc1)C(=O)NO)C(=O)NCc1ccccc1 |r|
OCCCN(Cc1ccc(cc1)C(=O)NO)C(=O)Cc1ccccc1
c1cc(ccc1CN)NC(=O)N(CCCCO)Cc2ccc(cc2)C(=O)NO
CCCCN(Cc1ccc(cc1)C(=O)NO)C(=O)Nc1ccc(CN)cc1
CN1CC2(CCN(CC2)Cc3ccc(cc3)C(=O)NO)c4c1cccc4
ONC(=O)c1ccc(CN2CCC3(CN(Cc4ccccc4)c4ccccc34)CC2)cc1
ONC(=O)c1ccc(CN2CCC3(CN(C(=O)c4ccccc4)c4ccccc34)CC2)cc1
ONC(=O)c1ccc(CN2CCC3(CN(C(=O)c4ccccc4)c4c3cccc4-c3ccccc3)CC2)cc1
ONC(=O)c1ccc(CC(=O)N2CCC3(CN(Cc4ccccc4)c4ccccc34)CC2)cc1
ONC(=O)c1ccc(CNC(=O)N2CCC3(CN(Cc4ccccc4)c4ccccc34)CC2)cc1
ONC(=O)c1ccc(COC(=O)N2CCC3(CN(Cc4ccccc4)c4ccccc34)CC2)cc1
CNc1ccccc1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
Nc1cccc(F)c1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
Nc1cccnc1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
CSc1ccccc1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
COc1ccccc1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
Oc1ccccc1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
Oc1cccc(F)c1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
COc1cccc(F)c1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
COc1cccc(O)c1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
COc1ccc(O)c(c1)C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
Oc1cccnc1C(=O)NCCCC[C@H](NC(=O)c1cncs1)c1ncc([nH]1)-c1ccc2ccccc2c1 |r|
Cn1cc(-c2ccccc2Oc2ccccc2)c2cc([nH]c2c1=O)C(=O)NCCCC(=O)NO
Cn1cc(-c2ccccc2Oc2ccccc2)c2cc([nH]c2c1=O)C(=O)NCCCCC(=O)NO
Cn1cc(-c2ccccc2Oc2ccccc2)c2cc([nH]c2c1=O)C(=O)NCCCCCC(=O)NO
Cn1cc(-c2ccccc2Oc2ccccc2)c2cc([nH]c2c1=O)C(=O)NCCCCCCC(=O)NO
Cn1cc(-c2ccccc2Oc2ccccc2)c2cc([nH]c2c1=O)C(=O)NCc1ccc(cc1)C(=O)NO
Cn1cc(-c2ccccc2Oc2ccccc2)c2cc([nH]c2c1=O)C(=O)NCCCCC(=O)Nc1ccccc1N
Cn1cc(-c2ccccc2Oc2ccccc2)c2cc([nH]c2c1=O)C(=O)NCCCCCC(=O)Nc1ccccc1N
Cn1cc(-c2ccccc2Oc2ccccc2)c2cc([nH]c2c1=O)C(=O)NCCCCCCC(=O)Nc1ccccc1N
Cn1cc(-c2ccccc2Oc2ccccc2)c2cc([nH]c2c1=O)C(=O)NCc1ccc(cc1)C(=O)Nc1ccccc1N
CC(C)Oc1ccc(cc1-c1cn(C)c(=O)c2[nH]c(cc12)C(=O)NCc1ccc(cc1)C(=O)NO)C(C)(C)O
Cn1cc(-c2cc(ccc2OC2CC2)C(C)(C)O)c2cc([nH]c2c1=O)C(=O)NCc1ccc(cc1)C(=O)NO
Cn1cc(-c2cc(ccc2Oc2ccc(F)cc2F)C(C)(C)O)c2cc([nH]c2c1=O)C(=O)NCc1ccc(cc1)C(=O)NO
Cc1cc(F)cc(C)c1Oc1ccc(cc1-c1cn(C)c(=O)c2[nH]c(cc12)C(=O)NCc1ccc(cc1)C(=O)NO)C(C)(C)O
CC(C)Oc1ccc(cc1-c1cn(C)c(=O)c2[nH]c(cc12)C(=O)NCCCCCCC(=O)NO)C(C)(C)O
Cn1cc(-c2cc(ccc2OC2CC2)C(C)(C)O)c2cc([nH]c2c1=O)C(=O)NCCCCCCC(=O)NO
Cn1cc(-c2cc(ccc2Oc2ccc(F)cc2F)C(C)(C)O)c2cc([nH]c2c1=O)C(=O)NCCCCCCC(=O)NO
Cc1cc(F)cc(C)c1Oc1ccc(cc1-c1cn(C)c(=O)c2[nH]c(cc12)C(=O)NCCCCCCC(=O)NO)C(C)(C)O
ONC(=O)CCCCCCC(=O)Nc1cnc(nc1)N(c1ccccc1)c1ccccc1
[H][C@@]1(CC(=O)Nc2ccc(O)cc2)N=C(c2c(C)c(C)sc2-n2c(C)nnc12)c1ccc(Cl)cc1 |r,c:14|
CCNC(=O)c1cc2c([nH]1)C(=O)N(C=C2c3cc(ccc3Oc4c(cc(cc4C)F)C)C(C)(C)O)C
ONC(=O)c1ccc(Cn2c3ccccc3c(-c3ccccc3)c(O)c2=O)cc1
COc1c(-c2ccccc2)c2ccccc2n(Cc2ccc(cc2)C(=O)NO)c1=O
ONC(=O)c1ccc(Cn2c3ccccc3c(-c3ccccc3)c(OCc3ccccc3)c2=O)cc1
ONC(=O)c1ccc(Cn2c3ccccc3c(-c3cccnc3)c(O)c2=O)cc1
ONC(=O)c1ccc(COc2c(-c3ccccc3)c3ccccc3[nH]c2=O)cc1
Cn1c2ccccc2c(-c2ccccc2)c(OCc2ccc(cc2)C(=O)NO)c1=O
ONC(=O)c1ccc(COc2c(-c3ccccc3)c3ccccc3n(CC#C)c2=O)cc1
ONC(=O)c1ccc(COc2c(-c3ccccc3)c3ccccc3n(Cc3ccccc3)c2=O)cc1
ONC(=O)c1ccc(COc2c(-c3ccccc3)c3ccccc3n(Cc3ccncc3)c2=O)cc1
ONC(=O)c1ccc(COc2c(-c3ccccc3)c3ccccc3n(C3CCN(Cc4ccccc4)CC3)c2=O)cc1
CCN(CC)Cc1ccc(Cn2c3ccccc3c(-c3ccccc3)c(OCc3ccc(cc3)C(=O)NO)c2=O)cc1
Cn1c2ccccc2c(-c2cccnc2)c(OCc2ccc(cc2)C(=O)NO)c1=O
ONC(=O)c1ccc(COc2c(-c3cccnc3)c3ccccc3n(Cc3ccccc3)c2=O)cc1
ONC(=O)c1ccc(COc2c(-c3cccnc3)c3ccccc3n(Cc3ccncc3)c2=O)cc1
CCN(CC)Cc1ccc(Cn2c3ccccc3c(-c3cccnc3)c(OCc3ccc(cc3)C(=O)NO)c2=O)cc1
Cn1c2ccccc2c(C2CCCCC2)c(OCc2ccc(cc2)C(=O)NO)c1=O
ONC(=O)c1ccc(CN2C(=O)c3ccccc3C2=O)cc1-c1ccccc1
ONC(=O)c1ccc(CN2C(=O)c3cccc(F)c3C2=O)cc1-c1ccccc1
ONC(=O)c1ccc(CN2C(=O)c3ccccc3S2(=O)=O)cc1-c1ccccc1
CC(C)[C@@H](c1ccccc1)C(=O)Nc2ccc(cc2)C(=O)NO
Nc1ccccc1NC(=O)c1ccc(Cn2cnc3c(Nc4ccc(F)c(Cl)c4)nc(Cl)nc23)cc1
Nc1ccccc1NC(=O)c1ccc(Cn2cnc3c(Nc4ccc(cc4)C(=O)NO)nc(Cl)nc23)cc1
Cc1c[nH]nc1Nc1nc(Cl)nc2n(Cc3ccc(cc3)C(=O)Nc3ccccc3N)cnc12
Nc1ccccc1NC(=O)c1ccc(Cn2ccc3c(Cl)nc(Cl)nc23)cc1
Nc1nc(Cl)c2ncn(Cc3ccc(cc3)C(=O)Nc3ccccc3N)c2n1
Nc1ccccc1NC(=O)c1ccc(Cn2cnc3c(Nc4ccc(F)c(Cl)c4)nc(N)nc23)cc1
COc1cc(Nc2nc(N)nc3n(Cc4ccc(cc4)C(=O)Nc4ccccc4N)cnc23)cc(OC)c1
Nc1nc(Nc2ccc(F)c(Cl)c2)c2ccn(Cc3ccc(cc3)C(=O)Nc3ccccc3N)c2n1
Nc1nc(Cl)c2ccn(Cc3ccc(cc3)C(=O)Nc3cc(F)ccc3N)c2n1
COc1ccc(cc1C(=O)Nc1ccc2n(C)c(=O)c(C)cc2c1)C(=O)NO
Cc1cc2cc(NS(=O)(=O)c3ccc(cc3)C(=O)NO)ccc2n(C)c1=O
Cc1cc2cc(NS(=O)(=O)Cc3ccc(cc3)C(=O)NO)ccc2n(C)c1=O
CC(C)OC(=O)N[C@@H]1C[C@H](C)N(C(C)=O)c2ccc(cc12)-c1ccc(NC(=O)CCCCCCC(=O)NO)cc1 |r|
Cn1cc(cn1)-c1ccc(cc1)S(=O)(=O)n1ccc(\C=C\C(=O)Nc2ccccc2N)c1
N=C1Sc2ccccc2C2=NCCCN12 |t:10|
Nc1ccc(cc1NC(=O)c1ccc2nc(ccc2c1)N1CCNCC1)-c1cccs1
ONC(=O)c1cnc(nc1)C1(CCC(F)(F)CC1)c1ccccc1
CCCCCCCCCCCCCCCCNNC(=O)c1cccs1
Nc1cc(F)ccc1NC(=O)c1ccc(CNC(=O)\C=C\c2cccnc2)cc1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCC(=O)NO)c(C)c1)N1CCCC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCC(=O)NO)c(C)c1)N1CCCCC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCC(=O)NO)c(C)c1)N1CCSCC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCC(=O)NO)c(C)c1)N1CCOCC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCC(=O)NO)c(C)c1)N1CCOC[C@@H]1C |r|
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCC(=O)NO)c(C)c1)N1CCOC[C@H]1C |r|
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCC(=O)NO)c(C)c1)N1CCN(C)CC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCC(=O)NO)c(C)c1)N1CCS(=O)(=O)CC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCC(=O)NO)c(C)c1)N1CCC(F)(F)CC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCC(=O)NO)c(C)c1)N1CCCC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCC(=O)NO)c(C)c1)N1CCCCC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCC(=O)NO)c(C)c1)N1CCSCC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCC(=O)NO)c(C)c1)N1CCOCC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCC(=O)NO)c(C)c1)N1CCOC[C@@H]1C |r|
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCC(=O)NO)c(C)c1)N1CCOC[C@H]1C |r|
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCC(=O)NO)c(C)c1)N1CCN(C)CC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCC(=O)NO)c(C)c1)N1CCS(=O)(=O)CC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCC(=O)NO)c(C)c1)N1CCC(F)(F)CC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCC(=O)NO)c(C)c1)N1CCCC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCC(=O)NO)c(C)c1)N1CCCCC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCC(=O)NO)c(C)c1)N1CCSCC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCC(=O)NO)c(C)c1)N1CCOCC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCC(=O)NO)c(C)c1)N1CCOC[C@@H]1C |r|
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCC(=O)NO)c(C)c1)N1CCOC[C@H]1C |r|
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCC(=O)NO)c(C)c1)N1CCN(C)CC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCC(=O)NO)c(C)c1)N1CCS(=O)(=O)CC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCC(=O)NO)c(C)c1)N1CCC(F)(F)CC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCCC(=O)NO)c(C)c1)N1CCCC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCCC(=O)NO)c(C)c1)N1CCCCC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCCC(=O)NO)c(C)c1)N1CCSCC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCCC(=O)NO)c(C)c1)N1CCOCC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCCC(=O)NO)c(C)c1)N1CCOC[C@@H]1C |r|
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCCC(=O)NO)c(C)c1)N1CCOC[C@H]1C |r|
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCCC(=O)NO)c(C)c1)N1CCN(C)CC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCCC(=O)NO)c(C)c1)N1CCS(=O)(=O)CC1
COc1cc(OC)c2c(nc(nc2c1)-c1cc(C)c(OCCCCCC(=O)NO)c(C)c1)N1CCC(F)(F)CC1
CN(C)CCOc1ccc(cc1)-c1cc(=O)c2c(O)cc(OCCCCCC(=O)NO)cc2o1
Nc1nc2cc(ccc2o1)-c1nn(CCCCCCC(=O)NO)c2ncnc(N)c12
Nc1nc2cc(ccc2o1)-c1nn(CC2CCN(CC2)c2ncc(cn2)C(=O)NO)c2ncnc(N)c12
ONC(=O)c1cccc(c1)C(=O)NOCc1ccc(Cl)cc1Cl
CN1CCN(CC1)NC(=O)c1cccc(c1)C(=O)NO
CCCCCCC(=O)N(O)C1CC(=O)C(C1=O)c1ccc(Cl)cc1
ONC(=O)\C=C\c1ccccc1Oc1c(Cl)cccc1Cl
c1ccc(c(c1)/C=C/C(=O)NO)Sc2ccc(cc2)Cl
ONC(=O)c1ccc(CN(CC(=O)NCc2ccccc2)C(=O)c2cccc3ccccc23)cc1
Cc1ccccc1C(=O)N(CC(=O)NCc1ccccc1)Cc1ccc(cc1)C(=O)NO
Cc1ccc(C(=O)N(CC(=O)NCc2ccccc2)Cc2ccc(cc2)C(=O)NO)c(C)c1
ONC(=O)c1ccc(CN(CC(=O)NCc2ccccc2)C(=O)Cc2ccccc2)cc1
CC(C)c1ccc(CC(=O)N(CC(=O)NCc2ccccc2)Cc2ccc(cc2)C(=O)NO)cc1
Cc1ccc(C(=O)N(CC(=O)NC2CCCCC2)Cc2ccc(cc2)C(=O)NO)c(C)c1
ONC(=O)c1ccc(CN(CC(=O)NC2CCCCC2)C(=O)Cc2ccccc2)cc1
CC(C)c1ccc(CC(=O)N(CC(=O)NC2CCCCC2)Cc2ccc(cc2)C(=O)NO)cc1
CC(C)c1ccc(cc1)C(=O)N(CC(=O)NC12CC3CC(CC(C3)C1)C2)Cc1ccc(cc1)C(=O)NO |TLB:15:16:19:23.22.21,THB:17:18:21:25.16.24,17:16:19.18.23:21,24:16:19:23.22.21,24:22:19:25.17.16|
Cc1ccccc1C(=O)N(CC(=O)NC12CC3CC(CC(C3)C1)C2)Cc1ccc(cc1)C(=O)NO |TLB:13:14:17:21.20.19,THB:15:16:19:23.14.22,15:14:17.16.21:19,22:14:17:21.20.19,22:20:17:23.15.14|
CC(C)c1ccc(cc1)C(=O)N(Cc1ccc(cc1)C(=O)NO)C(C)(C)C(=O)NCc1ccccc1
CN(C)c1ccc(cc1)C(=O)N(Cc1ccc(cc1)C(=O)NO)C(C)(C)C(=O)NCc1ccccc1
CC(C)c1ccc(cc1)C(=O)N(Cc1ccc(cc1)C(=O)NO)C(C)(C)C(=O)NC1CCCCC1
CNC(=O)CN(Cc1ccc(cc1)C(=O)NO)C(=O)c1ccc(cc1)C(C)C
Cc1cc(C)cc(c1)C(=O)N(CC(=O)N1CCCCC1)Cc1ccc(cc1)C(=O)NO
CN(C)C(=O)CN(Cc1ccc(cc1)C(=O)NO)C(=O)c1cc(C)cc(C)c1
ONC(=O)c1ccc(CN2CCc3ccccc3CC2)cc1
ONC(=O)c1ccc(CN2CCCc3ccccc3C2)cc1
ONC(=O)c1ccc(CN2CCCCc3ccccc23)cc1
ONC(=O)c1ccc(CN2CCCOc3ccccc23)cc1
ONC(=O)c1ccc(CN2CCCSc3ccccc23)cc1
ONC(=O)c1ccc(CN2CCC[S+]([O-])c3ccccc23)cc1
COc1ccc2CCN(Cc3ccc(cc3)C(=O)NO)CCc2c1
COc1cccc2CCN(Cc3ccc(cc3)C(=O)NO)CCc12
COc1ccc(Br)c2CCN(Cc3ccc(cc3)C(=O)NO)CCc12
COc1ccc(C2CC2)c2CCN(Cc3ccc(cc3)C(=O)NO)CCc12
COc1ccc(-c2ccccc2)c2CCN(Cc3ccc(cc3)C(=O)NO)CCc12
ONC(=O)c1ccc(CN2CCCCc3cc(Cl)ccc23)cc1
ONC(=O)c1ccc(CN2CCCCc3ccc(Cl)cc23)cc1
ONC(=O)c1ccc(CN2CCCCc3ccc(F)cc23)cc1
ONC(=O)c1ccc(CN2CCCCc3ccc(Br)cc23)cc1
COc1cccc2N(Cc3ccc(cc3)C(=O)NO)CCCCc12
COc1ccc2N(Cc3ccc(cc3)C(=O)NO)CCCCc2c1
COc1ccc2CCCCN(Cc3ccc(cc3)C(=O)NO)c2c1
COc1cc2CCCCN(Cc3ccc(cc3)C(=O)NO)c2cc1OC
Cc1ccc2CCCCN(Cc3ccc(cc3)C(=O)NO)c2c1
ONC(=O)c1ccc(CN2CCCCc3ccc(cc23)C2CC2)cc1
ONC(=O)c1ccc(CN2CCCCc3ccc(cc23)-c2ccccc2)cc1
ONC(=O)c1ccc(NCc2nc(nn2-c2ccccc2)-c2ccccc2)cc1
Cc1cccc(c1)-c1nc(CNc2ccc(cc2)C(=O)NO)n(n1)-c1ccccc1
Cc1ccc(cc1)-c1nc(CNc2ccc(cc2)C(=O)NO)n(n1)-c1ccccc1
COc1ccc(cc1)-c1nc(CNc2ccc(cc2)C(=O)NO)n(n1)-c1ccccc1
ONC(=O)c1ccc(NCc2nc(nn2-c2ccccc2)-c2ccc(F)cc2)cc1
ONC(=O)c1ccc(NCc2nc(nn2-c2ccccc2)-c2ccccc2Cl)cc1
ONC(=O)c1ccc(NCc2nc(nn2-c2ccccc2)-c2cccc(Cl)c2)cc1
ONC(=O)c1ccc(NCc2nc(nn2-c2ccccc2)-c2ccc(Cl)cc2)cc1
ONC(=O)c1ccc(NCc2nc(nn2-c2ccccc2)-c2cc3ccccc3s2)cc1
Cc1ccsc1-c1nc(CNc2ccc(cc2)C(=O)NO)n(n1)-c1ccccc1
ONC(=O)c1ccc(NCc2nc(nn2-c2ccccc2)-c2sccc2Br)cc1
Cc1ccc(s1)-c1nc(CNc2ccc(cc2)C(=O)NO)n(n1)-c1ccccc1
ONC(=O)c1ccc(NCc2nc(nn2-c2ccc(O)cc2)-c2cccs2)cc1
ONC(=O)c1ccc(NCc2nc(nn2-c2ccc(F)cc2)-c2ccccc2)cc1
ONC(=O)c1ccc(NCc2nc(nn2-c2ccccc2Cl)-c2ccccc2)cc1
ONC(=O)c1ccc(NCc2nc(nn2-c2cccc(Cl)c2)-c2ccccc2)cc1
ONC(=O)c1ccc(NCc2nc(nn2-c2ccc(Br)cc2)-c2ccccc2)cc1
Cc1ccc(cc1)-n1nc(nc1CNc1ccc(cc1)C(=O)NO)-c1ccccc1
Cc1cccc(c1)-n1nc(nc1CNc1ccc(cc1)C(=O)NO)-c1ccccc1
COc1ccc(cc1)-n1nc(nc1CNc1ccc(cc1)C(=O)NO)-c1ccccc1
COc1ccc(cc1)-n1nc(nc1CNc1ccc(cc1)C(=O)NO)-c1ccc(O)cc1
CC[C@@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)CC)NC(=O)[C@H]2CCCCN2C1=O |r|
CCC(=O)CCCCC[C@H](NC(=O)C1CN(C)C1)c1ncc([nH]1)-c1ccccc1 |r|
CCC(=O)CCCCC[C@@H]1NC(=O)C2CCN2CCCCCOc2ccccc2-c2cnc1[nH]2 |r|
CCC(=O)CCCCC[C@@H]1NC(=O)C2CCN2CCCCCCOc2ccccc2-c2cnc1[nH]2 |r|
CCC(=O)CCCCC[C@@H]1NC(=O)C2CCN2CCCCCCc2ccccc2-c2cnc1[nH]2 |r|
CCC(=O)CCCCC[C@H](NC(=O)C1CN(C)C1)c1[nH]c(nc1C(N)=O)-c1ccccc1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2[nH]c(nc2C(N)=O)-c2ccc(F)cc2)CC1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2[nH]c-3nc2C(=O)NCCC\C=C/c2cccc-3c2)CC1 |r,c:34|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2[nH]c-3nc2C(=O)NCCC\C=C\c2cccc-3c2)CC1 |r,t:34|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2[nH]c-3nc2C(=O)NCCCCCc2cccc-3c2)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2C3CCC(C3)c2c1 |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)C\C=C\CN2C3CCC2c2cc(ccc32)-c2cnc1[nH]2 |r,wU:13.12,wD:9.8,t:24,TLB:24:25:30.35:27.28,(23.45,-24.5,;22.06,-23.86,;20.81,-24.75,;20.95,-26.28,;19.42,-24.11,;18.17,-25,;16.77,-24.37,;15.52,-25.25,;14.13,-24.61,;12.87,-25.5,;13.01,-27.03,;14.4,-27.67,;15.66,-26.78,;14.57,-29.2,;15.45,-30.45,;13.92,-30.58,;12.54,-29.79,;11.18,-30.58,;11.18,-32.16,;12.55,-32.95,;13.93,-32.17,;4.16,-31.99,;3.9,-30.43,;2.43,-29.87,;2.17,-28.31,;3.4,-27.31,;2.98,-25.79,;2.48,-27.25,;3.5,-28.41,;5.02,-28.11,;5.51,-26.65,;7.02,-26.34,;7.51,-24.88,;6.49,-23.73,;5,-24.02,;4.5,-25.49,;9.01,-24.58,;9.64,-23.19,;11.17,-23.36,;11.48,-24.86,;10.14,-25.62,)|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)CCCCN2C3CCC2c2cc(ccc32)-c2cnc1[nH]2 |r,wU:13.12,wD:9.8,TLB:24:25:30.35:27.28,(51.92,-23.44,;50.53,-22.8,;49.28,-23.69,;49.42,-25.23,;47.89,-23.06,;46.63,-23.95,;45.24,-23.31,;43.98,-24.2,;42.6,-23.56,;41.34,-24.45,;41.48,-25.97,;42.87,-26.62,;44.13,-25.73,;43.03,-28.14,;43.92,-29.39,;42.39,-29.53,;41.01,-28.74,;39.65,-29.52,;39.64,-31.11,;41.02,-31.9,;42.4,-31.11,;33.18,-31.04,;32.37,-29.37,;30.9,-28.81,;30.64,-27.26,;31.86,-26.25,;31.45,-24.73,;30.95,-26.19,;31.97,-27.36,;33.49,-27.06,;33.97,-25.6,;35.49,-25.29,;35.98,-23.83,;34.96,-22.68,;33.47,-22.96,;32.96,-24.43,;37.48,-23.53,;38.11,-22.13,;39.64,-22.3,;39.95,-23.81,;38.61,-24.56,)|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)CCCCN2C3CCC2c2c3cccc2-c2cnc1[nH]2 |r,wU:13.12,wD:9.8,TLB:24:25:30.31:27.28,(78.21,-22.01,;76.81,-21.36,;75.57,-22.25,;75.7,-23.79,;74.16,-21.62,;72.91,-22.51,;71.51,-21.87,;70.25,-22.75,;68.86,-22.12,;67.6,-23.01,;67.75,-24.54,;69.14,-25.19,;70.4,-24.29,;69.3,-26.71,;70.19,-27.96,;68.66,-28.1,;67.28,-27.31,;65.91,-28.1,;65.91,-29.68,;67.28,-30.48,;68.67,-29.69,;61.98,-30.85,;60.45,-30.26,;60.19,-28.64,;61.47,-27.61,;61.21,-26,;59.75,-25.61,;60.77,-26.76,;62.28,-26.46,;62.77,-25,;61.74,-23.85,;60.24,-24.16,;59.22,-22.99,;59.72,-21.52,;61.21,-21.24,;62.24,-22.39,;63.74,-22.09,;64.38,-20.69,;65.91,-20.86,;66.21,-22.37,;64.87,-23.12,)|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2c(ccn(C)c2=O)c1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2ccc3c(ccn(CC)c3=O)c2)CC1 |r|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)CCOCCn2ccc3cc(ccc3c2=O)-c2cnc1[nH]2 |r,wU:13.12,wD:9.8,(78.93,-40.88,;77.54,-40.24,;76.29,-41.13,;76.43,-42.66,;74.89,-40.49,;73.64,-41.38,;72.24,-40.74,;70.98,-41.63,;69.6,-40.99,;68.34,-41.88,;68.48,-43.41,;69.88,-44.06,;71.14,-43.16,;70.04,-45.57,;70.92,-46.83,;69.39,-46.96,;68.01,-46.18,;66.65,-46.96,;66.65,-48.55,;68.02,-49.34,;69.41,-48.55,;65.26,-49.35,;61.83,-47.66,;57.1,-47.99,;54.94,-45.64,;55.51,-42.82,;57.41,-41.01,;57.91,-39.53,;59.43,-39.23,;60.46,-40.39,;61.95,-40.11,;62.97,-41.26,;62.48,-42.72,;60.98,-43.03,;59.96,-41.87,;58.44,-42.17,;57.93,-43.7,;64.48,-40.96,;65.11,-39.56,;66.64,-39.74,;66.94,-41.24,;65.61,-41.99,)|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)CCCCCn2c3ccc(cc3ccc2=O)-c2cnc1o2 |r,wU:13.12,wD:9.8,(24.65,-55.17,;23.25,-54.53,;22.01,-55.41,;22.14,-56.95,;20.6,-54.78,;19.35,-55.67,;17.96,-55.03,;16.7,-55.92,;15.31,-55.28,;14.05,-56.17,;14.2,-57.69,;15.59,-58.35,;16.85,-57.45,;15.75,-59.86,;16.63,-61.12,;15.1,-61.25,;13.72,-60.47,;12.36,-61.25,;12.36,-62.84,;13.73,-63.63,;15.12,-62.84,;6.84,-61.59,;5.26,-61.91,;4.2,-60.71,;4.71,-59.19,;3.65,-57.99,;4.16,-56.46,;5.67,-56.16,;6.69,-57.32,;8.2,-57.01,;8.69,-55.55,;7.67,-54.4,;6.17,-54.68,;5.15,-53.52,;3.62,-53.82,;3.13,-55.3,;1.55,-55.62,;10.19,-55.25,;10.83,-53.85,;12.36,-54.03,;12.66,-55.53,;11.32,-56.28,)|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)CCCOCCn2ccc3cc(ccc3c2=O)-c2cnc1[nH]2 |r,wU:13.12,wD:9.8,(53.94,-55.95,;52.55,-55.3,;51.3,-56.19,;51.44,-57.72,;49.9,-55.56,;48.65,-56.45,;47.25,-55.81,;45.99,-56.69,;44.61,-56.06,;43.35,-56.95,;43.49,-58.47,;44.88,-59.12,;46.14,-58.23,;45.04,-60.64,;45.93,-61.89,;44.4,-62.03,;43.02,-61.24,;41.66,-62.03,;41.66,-63.61,;43.03,-64.41,;44.41,-63.62,;40.26,-64.41,;38.55,-63.17,;36.55,-63.64,;33.33,-59.89,;30.34,-58.69,;30.85,-56.4,;32.42,-56.08,;32.92,-54.6,;34.44,-54.29,;35.47,-55.46,;36.96,-55.18,;37.98,-56.33,;37.49,-57.79,;35.99,-58.09,;34.97,-56.93,;33.45,-57.24,;32.94,-58.76,;39.48,-56.03,;40.12,-54.63,;41.65,-54.8,;41.95,-56.31,;40.62,-57.06,)|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)CCCCCOc2ccc3cc(ccc3n2)-c2cnc1o2 |r,wU:13.12,wD:9.8,(79.6,-58.13,;78.2,-57.48,;76.96,-58.37,;77.1,-59.91,;75.56,-57.74,;74.31,-58.63,;72.91,-57.99,;71.65,-58.87,;70.27,-58.24,;69.01,-59.13,;69.15,-60.65,;70.55,-61.31,;71.8,-60.41,;70.7,-62.82,;71.59,-64.07,;70.06,-64.21,;68.68,-63.43,;67.32,-64.21,;67.32,-65.79,;68.69,-66.59,;70.07,-65.8,;65.92,-66.59,;64.48,-65.02,;62.43,-65.43,;59.65,-62.19,;56.5,-60.66,;56.51,-58.58,;58.08,-58.26,;58.58,-56.78,;60.1,-56.48,;61.13,-57.64,;62.62,-57.36,;63.64,-58.51,;63.15,-59.97,;61.65,-60.28,;60.63,-59.12,;59.11,-59.42,;65.15,-58.21,;65.78,-56.81,;67.31,-56.98,;67.61,-58.49,;66.28,-59.24,)|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)CCCOCCCn2ccc3cc(ccc3c2=O)-c2cnc1[nH]2 |r,wU:13.12,wD:9.8,(27.19,-4.47,;25.79,-3.82,;24.56,-4.71,;24.69,-6.24,;23.15,-4.08,;21.91,-4.96,;20.51,-4.33,;19.26,-5.21,;17.87,-4.58,;16.62,-5.46,;16.76,-6.99,;18.16,-7.64,;19.41,-6.74,;18.31,-9.15,;19.19,-10.4,;17.67,-10.54,;16.29,-9.76,;14.94,-10.54,;14.93,-12.12,;16.3,-12.91,;17.68,-12.12,;13.54,-12.91,;12.05,-11.67,;10.16,-12.03,;8.16,-8.93,;4.6,-8.03,;3.64,-6.43,;4.15,-4.92,;5.72,-4.6,;6.21,-3.12,;7.73,-2.82,;8.75,-3.98,;10.24,-3.69,;11.27,-4.85,;10.77,-6.31,;9.28,-6.61,;8.26,-5.45,;6.74,-5.75,;6.23,-7.27,;12.76,-4.55,;13.4,-3.15,;14.93,-3.33,;15.22,-4.83,;13.9,-5.58,)|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)CCCCCCCCn2ccc3cc(ccc3c2=O)-c2cnc1[nH]2 |r,wU:13.12,wD:9.8,(54.03,-3.3,;52.63,-2.65,;51.39,-3.55,;51.52,-5.08,;49.99,-2.91,;48.73,-3.8,;47.34,-3.16,;46.08,-4.04,;44.69,-3.4,;43.44,-4.3,;43.59,-5.82,;44.98,-6.47,;46.23,-5.57,;45.14,-7.99,;46.02,-9.24,;44.49,-9.38,;43.11,-8.59,;41.76,-9.38,;41.75,-10.96,;43.12,-11.75,;44.51,-10.96,;40.36,-11.76,;38.97,-10.95,;37.58,-11.75,;36.09,-10.67,;34.26,-10.81,;32.5,-6.91,;30.88,-5.99,;31.12,-4.14,;32.53,-3.43,;33.01,-1.95,;34.54,-1.65,;35.57,-2.81,;37.06,-2.53,;38.07,-3.68,;37.59,-5.14,;36.08,-5.44,;35.07,-4.29,;33.55,-4.59,;33.04,-6.11,;39.58,-3.38,;40.22,-1.98,;41.75,-2.16,;42.05,-3.66,;40.71,-4.41,)|
CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC22CCN(CC2)CCCCCCCCn2ccc3cc(-c4cnc1[nH]4)c(OC)cc3c2=O |r,wU:13.12,wD:9.8,(81.04,-4.01,;79.64,-3.37,;78.4,-4.27,;78.53,-5.8,;77,-3.63,;75.75,-4.52,;74.35,-3.88,;73.09,-4.76,;71.71,-4.12,;70.45,-5.02,;70.6,-6.54,;71.99,-7.19,;73.24,-6.29,;72.15,-8.71,;73.03,-9.95,;71.5,-10.1,;70.13,-9.31,;68.77,-10.1,;68.77,-11.67,;70.13,-12.47,;71.52,-11.68,;67.37,-12.47,;65.99,-11.67,;64.6,-12.47,;63.21,-11.22,;61.32,-11.48,;59.29,-7.36,;57.73,-6.26,;58.02,-4.74,;59.54,-4.15,;60.03,-2.67,;61.55,-2.37,;62.58,-3.53,;64.07,-3.25,;65.09,-4.4,;66.6,-4.1,;67.23,-2.7,;68.76,-2.88,;69.06,-4.38,;67.72,-5.13,;64.6,-5.85,;65.62,-7,;65.13,-8.45,;63.1,-6.16,;62.08,-5.01,;60.56,-5.31,;60.05,-6.83,)|
CCC(=O)CCCCC[C@@H]1NC(=O)CN(C)CCCCOCCCCn2ccc3cc(ccc3c2=O)-c2cnc1[nH]2 |r|
CN1CCN(CC1)c1nc(nc2cc(Cl)ccc12)-c1ccc(cc1)C(=O)NO
Cn1c2cnc3ccc(cc3c2n(-c2ccc(cc2)C(C)(C)C#N)c1=O)-c1cnc2ccccc2c1
CCc1c(C)c2cc3[nH]c(cc4nc([C@@H](CCC(=O)Nc5ccc(cc5)C(=O)Nc5ccccc5N)[C@@H]4C)c(C(=O)OC)c4[nH]c(cc1n2)c(C)c4C(=O)OC)c(C)c3C=C |r|
CC12CC3CC(C)(C1)CC(C3)(C2)NCc1ccc(cc1)C(=O)NO |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NCc1ccc(\C=C\C(=O)NO)cc1 |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NS(=O)(=O)c1ccc(\C=C\C(=O)NO)cc1 |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NS(=O)(=O)c1cccc(\C=C\C(=O)NO)c1 |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NC(=O)CCCCCC(=O)NO |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NC(=O)CCCCCCC(=O)NO |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NC(=O)CCCCCCCC(=O)NO |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NC(=O)CCCCCCCCC(=O)NO |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NCc1cccc(NC(=O)CCCCCCC(=O)NO)c1 |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NCc1ccc(NC(=O)CCCCCCC(=O)NO)cc1 |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
CC12CC3CC(C)(C1)CC(C3)(C2)NCc1ccc(NCc2ccc(cc2)C(=O)NO)cc1 |TLB:12:9:4:7.2.1,0:1:4:10.9.8,THB:2:3:8:7.1.11,2:1:4.3.10:8,11:1:4:10.9.8,11:9:4:7.2.1|
ONC(=O)CCCCCCn1cc(nn1)-c1ccc2ncnc(Nc3ccc(Br)cc3F)c2c1
CSc1ccc2Sc3ccccc3N(Cc3ccc(cc3)C(=O)NO)c2c1
NC(=O)c1ccc2Sc3ccccc3N(Cc3ccc(cc3)C(=O)NO)c2c1
C\C(=N/O)c1ccc2Sc3ccccc3N(Cc3ccc(cc3)C(=O)NO)c2c1
ONC(=O)c1ccc(CN2c3ccccc3[S+]([O-])c3ccc(Cl)cc23)cc1
ONC(=O)c1ccc(CN2c3ccccc3[S+]([O-])c3ccc(cc23)C(F)(F)F)cc1
COc1ccc2[S+]([O-])c3ccccc3N(Cc3ccc(cc3)C(=O)NO)c2c1
CSc1ccc2[S+]([O-])c3ccccc3N(Cc3ccc(cc3)C(=O)NO)c2c1
NC(=O)c1ccc2[S+]([O-])c3ccccc3N(Cc3ccc(cc3)C(=O)NO)c2c1
C\C(=N/O)c1ccc2[S+]([O-])c3ccccc3N(Cc3ccc(cc3)C(=O)NO)c2c1
NC(=O)c1ccc2Sc3ccccc3N(Cc3ccc(\C=C\C(=O)NO)cc3)c2c1
ONC(=O)c1ccc(CN2c3ccccc3Sc3ccc(cc23)C(=O)Nc2ccccn2)cc1
Cc1ccc(NC(=O)c2ccc3Sc4ccccc4N(Cc4ccc(cc4)C(=O)NO)c3c2)nc1
ONC(=O)c1ccc(CN2c3ccccc3Sc3ccc(cc23)C(=O)Nc2ccc(Br)cn2)cc1
CN(c1ccccc1Cl)S(=O)(=O)C1CC2OC1C(=C2c1ccc(O)cc1)c1ccc(NC(=O)CCCCCCC(O)=O)cc1 |c:19|
CN(c1cccc2ccccc12)S(=O)(=O)C1CC2OC1C(=C2c1ccc(O)cc1)c1ccc(NC(=O)CCCCCCC(O)=O)cc1 |c:23|
ONC(=O)CCCCCONC(=O)c1cc2ccccc2[nH]1
ONC(=O)CCCCCONC(=O)c1ccc2ccccc2n1
ONC(=O)CCCCCONC(=O)c1nccc2ccccc12
ONC(=O)CCCCCONC(=O)c1cnc2ccccc2n1
ONC(=O)CCCCCONC(=O)c1ccc2ccccc2c1
CC(N1CCCc2cc(Cl)ccc12)c1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(cc1)C(=O)N1CCCc2cc(Cl)ccc12
ONC(=O)c1ccc(cc1)C(=O)N1CCCc2cc(F)ccc12
ONC(=O)c1ccc(CN2c3ccc(Cl)cc3CCCC2=O)cc1
ONC(=O)c1ccc(CN2CCCCc3cc(Br)ccc23)cc1
ONC(=O)c1ccc(CN2CCCCc3cc(ccc23)-c2cc[nH]n2)cc1
ONC(=O)c1ccc(CN2CCCCc3cc(ccc23)C#N)cc1
NC(=O)c1ccc2N(Cc3ccc(cc3)C(=O)NO)CCCCc2c1
ONC(=O)c1ccc(CN2C(=O)CCc3cc(Cl)ccc23)cc1
ONC(=O)c1ccc(CN2C(=O)CCc3cc(Br)ccc23)cc1
ONC(=O)c1ccc(CN2C(=O)CCc3cc(ccc23)C2CC2)cc1
CCCc1ccc2N(Cc3ccc(cc3)C(=O)NO)C(=O)CCc2c1
ONC(=O)c1ccc(CN2CCCc3cc(ccc23)-c2cc[nH]n2)cc1
ONC(=O)c1ccc(CN2CCCc3cc(ccc23)C#N)cc1
c1cc(ccc1CN2CCCc3c2ccc(c3)C(=O)N)C(=O)NO
Cn1c(SCCCCCC(O)=O)nnc1-c1ccncc1
CCn1c(SCCCCCC(O)=O)nnc1-c1ccncc1
OC(=O)CCCCCSc1nnc(-c2ccncc2)n1CC=C
OC(=O)CCCCCSc1nnc(-c2ccncc2)n1-c1ccccc1
Cn1c(SCCCCCC(=O)NO)nnc1-c1ccncc1
CCn1c(SCCCCCC(=O)NO)nnc1-c1ccncc1
ONC(=O)CCCCCSc1nnc(-c2ccncc2)n1CC=C
ONC(=O)CCCCCSc1nnc(-c2ccncc2)n1-c1ccccc1
Cn1c(SCCCCCC(=O)Nc2ccccc2N)nnc1-c1ccncc1
CCn1c(SCCCCCC(=O)Nc2ccccc2N)nnc1-c1ccncc1
Nc1ccccc1NC(=O)CCCCCSc1nnc(-c2ccncc2)n1CC=C
Nc1ccccc1NC(=O)CCCCCSc1nnc(-c2ccncc2)n1-c1ccccc1
Cn1c(SCc2ccc(cc2)C(=O)NO)nnc1-c1ccncc1
CCn1c(SCc2ccc(cc2)C(=O)NO)nnc1-c1ccncc1
ONC(=O)c1ccc(CSc2nnc(-c3ccncc3)n2CC=C)cc1
ONC(=O)c1ccc(CSc2nnc(-c3ccncc3)n2-c2ccccc2)cc1
Cn1c(SCc2ccc(cc2)C(=O)Nc2ccccc2N)nnc1-c1ccncc1
CCn1c(SCc2ccc(cc2)C(=O)Nc2ccccc2N)nnc1-c1ccncc1
Nc1ccccc1NC(=O)c1ccc(CSc2nnc(-c3ccncc3)n2CC=C)cc1
Nc1ccccc1NC(=O)c1ccc(CSc2nnc(-c3ccncc3)n2-c2ccccc2)cc1
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc(o1)-c1cc2cccnc2cc1OC |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc(o2)-c2cc3cccnc3cc2OC)CC1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2cc3cccnc3cc2OC)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccc(nc2cc1OC)N1CCCC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC2CC2)CC1)c1ncc([nH]1)-c1cc2cccnc2cc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC2CC2)CC1)c1ncc(o1)-c1cc2ccc(C)nc2cc1OC |r|
ONC(=O)c1cc(F)c2CN(CCc2c1)C1CCC1
Cn1c2CN(Cc3ccc(cc3F)C(=O)NO)CCc2c2ccccc12
ONC(=O)c1ccc(CN2CC3(C2)CCOC3)c(F)c1
CN1Cc2cc(ccc2CN1Cc1ccccc1)C(=O)NO
ONC(=O)c1cc(F)c2-c3cccn3CCc2c1
CN1CC2(CCCCC2)CC[C@H]1Cc1cc(F)cc(c1)C(=O)NO |r|
ONC(=O)c1cc(F)c(Cn2nnnc2-c2cccs2)c(F)c1
ONC(=O)c1cccnc1
ONC(=O)c1cccc(F)c1
Cc1ccc(cc1)C(=O)NO
Cc1ccc(cn1)C(=O)NO
Cc1ccc(cc1F)C(=O)NO
Cc1c(F)cc(cc1F)C(=O)NO
Nc1ccc(cn1)C(=O)NO
Nc1ncc(cn1)C(=O)NO
Nc1ccc(cc1F)C(=O)NO
Nc1c(F)cc(cc1F)C(=O)NO
CC(=O)Nc1ccc(cc1F)C(=O)NO
CCN(CC)Cc1ccc2cc(COC(=O)Nc3c(F)cc(cc3F)C(=O)NO)ccc2c1
CC(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)C(=O)NCCCCCCC(=O)NO)ncc1Cl
CC(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(NC(=O)CCCCCCC(=O)NO)cc2)ncc1Cl
COc1cc2c(NC3CCN(C)CC3)cc(nc2cc1OCCCN1CCCC1)-c1ccc(C)o1
COc1cc2c(NCC3CCN(C)CC3)cc(nc2cc1OCCCN1CCCC1)-c1ccc(C)o1
COc1cc2c(NCC3CCN(CC3)c3ncc(cn3)C(=O)NO)cc(nc2cc1OCCCN1CCCC1)-c1ccc(C)o1
COc1cc2c(NCc3ccc(cc3)C(=O)NO)cc(nc2cc1OCCCN1CCCC1)-c1ccc(C)o1
COc1cc2c(NCC3CCC(CC3)C(=O)NO)cc(nc2cc1OCCCN1CCCC1)-c1ccc(C)o1 |(23,-19.22,;24.34,-18.45,;25.68,-19.22,;27.01,-18.45,;28.34,-19.21,;29.67,-18.44,;29.66,-16.9,;30.99,-16.12,;32.33,-16.89,;32.32,-18.44,;33.65,-19.21,;34.99,-18.44,;34.99,-16.89,;33.65,-16.12,;36.33,-19.21,;36.33,-20.75,;37.66,-18.44,;38.99,-19.21,;31.01,-19.2,;31.01,-20.75,;29.68,-21.52,;28.34,-20.76,;27.01,-21.53,;25.68,-20.76,;24.34,-21.53,;24.34,-23.07,;23.01,-23.84,;23.01,-25.38,;21.67,-26.15,;20.26,-25.52,;19.23,-26.67,;20,-28,;21.5,-27.68,;32.35,-21.51,;33.76,-20.88,;34.79,-22.02,;34.03,-23.35,;34.66,-24.76,;32.52,-23.04,)|
COc1cc2c(NCC3CCN(Cc4ccc(cc4)C(=O)NO)CC3)cc(nc2cc1OCCCN1CCCC1)-c1ccc(C)o1
COc1cc2c(NC3CCN(Cc4ccc(cc4)C(=O)NO)CC3)cc(nc2cc1OCCCN1CCCC1)-c1ccc(C)o1
COc1cc2c(NCC3CCN(CC3)c3ccc(cc3)C(=O)NO)cc(nc2cc1OCCCN1CCCC1)-c1ccc(C)o1
COc1cc2c(NCC3CCN(CC3)C3CCC(CC3)C(=O)NO)cc(nc2cc1OCCCN1CCCC1)-c1ccc(C)o1 |(44.4,-30.77,;45.73,-30,;47.08,-30.78,;48.4,-30.01,;49.74,-30.77,;51.07,-30,;51.06,-28.46,;52.39,-27.68,;53.72,-28.45,;53.72,-30,;55.04,-30.78,;56.39,-30.01,;56.39,-28.47,;55.05,-27.69,;57.72,-30.79,;57.71,-32.33,;59.03,-33.1,;60.37,-32.34,;60.37,-30.79,;59.04,-30.02,;61.7,-33.11,;61.7,-34.65,;63.04,-32.34,;64.37,-33.12,;52.4,-30.76,;52.41,-32.31,;51.08,-33.08,;49.74,-32.31,;48.41,-33.09,;47.07,-32.32,;45.74,-33.09,;45.74,-34.63,;44.4,-35.4,;44.4,-36.94,;43.07,-37.71,;41.66,-37.08,;40.62,-38.22,;41.39,-39.56,;42.9,-39.24,;53.75,-33.07,;55.15,-32.43,;56.19,-33.57,;55.42,-34.91,;56.05,-36.32,;53.91,-34.6,)|
COc1cc2c(NCC3CCC(CC3)c3ccc(cc3)C(=O)NO)cc(nc2cc1OCCCN1CCCC1)-c1ccc(C)o1 |(5.35,-49.68,;6.68,-48.91,;8.02,-49.68,;9.35,-48.91,;10.69,-49.68,;12.01,-48.9,;12.01,-47.36,;13.34,-46.59,;14.67,-47.36,;14.66,-48.91,;15.99,-49.68,;17.33,-48.92,;17.34,-47.37,;16,-46.59,;18.66,-49.69,;18.65,-51.23,;19.98,-52.01,;21.32,-51.24,;21.32,-49.69,;19.99,-48.93,;22.65,-52.02,;22.65,-53.56,;23.99,-51.25,;25.32,-52.02,;13.35,-49.66,;13.36,-51.21,;12.02,-51.99,;10.69,-51.22,;9.36,-52,;8.02,-51.23,;6.69,-52,;6.69,-53.54,;5.35,-54.3,;5.35,-55.84,;4.02,-56.61,;2.61,-55.98,;1.57,-57.13,;2.34,-58.46,;3.85,-58.14,;14.69,-51.97,;16.1,-51.34,;17.13,-52.48,;16.37,-53.82,;17,-55.22,;14.86,-53.5,)|
COc1cc2c(NCc3ccc(cc3)-c3ccc(cc3)C(=O)NO)cc(nc2cc1OCCCN1CCCC1)-c1ccc(C)o1
COc1cc2c(NCc3ccc(cc3)[C@H]3CC[C@@H](CC3)C(=O)NO)cc(nc2cc1OCCCN1CCCC1)-c1ccc(C)o1 |r,wU:14.14,wD:17.21,(52.14,-46.19,;53.47,-45.42,;54.82,-46.19,;56.15,-45.42,;57.48,-46.19,;58.81,-45.41,;58.8,-43.87,;60.13,-43.1,;61.47,-43.87,;61.46,-45.42,;62.79,-46.19,;64.13,-45.43,;64.13,-43.88,;62.79,-43.1,;65.46,-46.2,;66.79,-45.44,;68.12,-46.21,;68.12,-47.75,;66.78,-48.52,;65.45,-47.74,;69.45,-48.53,;69.44,-50.07,;70.78,-47.76,;72.12,-48.54,;60.14,-46.17,;60.15,-47.72,;58.82,-48.5,;57.48,-47.73,;56.15,-48.51,;54.81,-47.74,;53.48,-48.51,;53.48,-50.05,;52.14,-50.82,;52.14,-52.36,;50.81,-53.13,;49.4,-52.5,;48.37,-53.64,;49.14,-54.97,;50.64,-54.66,;61.49,-48.48,;62.89,-47.85,;63.93,-48.99,;63.16,-50.33,;63.8,-51.73,;61.66,-50.01,)|
COc1cc2c(NCc3ccc(cc3)[C@@H]3CC[C@@H](CC3)C(=O)NO)cc(nc2cc1OCCCN1CCCC1)-c1ccc(C)o1 |r,wU:14.14,17.21,(5.03,-4.91,;6.36,-4.14,;7.71,-4.92,;9.03,-4.14,;10.37,-4.91,;11.7,-4.14,;11.69,-2.6,;13.02,-1.82,;14.35,-2.59,;14.35,-4.14,;15.67,-4.92,;17.02,-4.15,;17.02,-2.61,;15.68,-1.83,;18.35,-4.93,;18.34,-6.47,;19.66,-7.24,;21,-6.48,;21.01,-4.93,;19.68,-4.16,;22.34,-7.25,;22.33,-8.79,;23.67,-6.48,;25,-7.26,;13.03,-4.9,;13.04,-6.44,;11.71,-7.22,;10.37,-6.45,;9.04,-7.23,;7.7,-6.46,;6.37,-7.23,;6.37,-8.77,;5.03,-9.54,;5.03,-11.08,;3.7,-11.85,;2.29,-11.22,;1.25,-12.36,;2.02,-13.7,;3.53,-13.38,;14.38,-7.21,;15.78,-6.57,;16.82,-7.71,;16.05,-9.05,;16.68,-10.45,;14.54,-8.74,)|
COc1cc2c(NC3CCN(CC3)c3ccc(cc3)C(=O)NO)cc(nc2cc1OCCCN1CCCC1)-c1ccc(C)o1
COc1cc2c(NCC3CCN(CC3)c3ncc(cn3)C(=O)NO)cc(C)nc2cc1OCCCN1CCCC1
COc1cc2c(NC3CCN(CC3)c3ncc(cn3)C(=O)NO)cc(C)nc2cc1OCCCN1CCCC1
COc1cc2c(NCC3CCN(CC3)c3ncc(cn3)C(=O)NO)cc(nc2cc1OCC1CCNCC1)-c1ccc(C)o1
COc1cc2nc(cc(NCC3CCN(CC3)c3ncc(cn3)C(=O)NO)c2cc1OC)-c1ccc(C)o1
COc1cc2nc(cc(NC3CCN(CC3)c3ncc(cn3)C(=O)NO)c2cc1OC)-c1ccc(C)o1
COc1cc2nc(cc(NCC3C4CCC3CN(C4)c3ncc(cn3)C(=O)NO)c2cc1OC)-c1ccc(C)o1
COc1cc2nc(cc(NCc3ccc(cc3)C(=O)NO)c2cc1OC)-c1ccc(C)o1
COc1cc2nc(cc(NCC3CCC(CC3)C(=O)NO)c2cc1OC)-c1ccc(C)o1 |(18.22,-51.09,;18.22,-49.55,;19.56,-48.78,;20.89,-49.55,;22.22,-48.77,;23.56,-49.54,;24.89,-48.76,;24.88,-47.21,;23.55,-46.45,;23.54,-44.91,;24.87,-44.14,;26.21,-44.91,;26.2,-46.46,;27.53,-47.23,;28.87,-46.47,;28.87,-44.92,;27.54,-44.14,;30.2,-47.24,;30.19,-48.78,;31.53,-46.48,;32.87,-47.25,;22.22,-47.23,;20.89,-46.46,;19.56,-47.23,;18.21,-46.46,;16.88,-47.23,;26.23,-49.52,;27.63,-48.88,;28.67,-50.02,;27.91,-51.36,;28.54,-52.76,;26.4,-51.05,)|
COc1cc2nc(cc(NCc3ccc(cn3)C(=O)NO)c2cc1OC)-c1ccc(C)o1
COc1cc2nc(cc(NCC3CCN(Cc4ccc(cc4)C(=O)NO)CC3)c2cc1OC)-c1ccc(C)o1
COc1cc2nc(cc(NCC3CCN(Cc4ccc(s4)C(=O)NO)CC3)c2cc1OC)-c1ccc(C)o1
COc1cc2nc(cc(NCC3CCN(CC3)C3CC(C3)C(=O)NO)c2cc1OC)-c1ccc(C)o1 |(23.21,-8.51,;23.21,-6.97,;24.55,-6.2,;25.88,-6.97,;27.22,-6.2,;28.55,-6.96,;29.89,-6.19,;29.88,-4.64,;28.54,-3.88,;28.53,-2.34,;29.86,-1.56,;31.2,-2.33,;31.19,-3.89,;32.52,-4.66,;33.86,-3.89,;33.87,-2.35,;32.53,-1.57,;35.19,-4.67,;35.58,-6.17,;37.07,-5.77,;36.68,-4.28,;38.4,-6.55,;38.39,-8.09,;39.74,-5.78,;41.07,-6.56,;27.22,-4.65,;25.88,-3.89,;24.55,-4.66,;23.21,-3.89,;21.87,-4.66,;31.22,-6.95,;32.63,-6.31,;33.66,-7.45,;32.9,-8.78,;33.54,-10.19,;31.4,-8.47,)|
COc1cc2nc(cc(N[C@H]3CC[C@H](CC3)C(=O)NO)c2cc1OC)-c1ccc(C)o1 |r,wU:10.9,13.16,(4.91,-22.33,;4.91,-20.79,;6.24,-20.02,;7.57,-20.79,;8.91,-20.02,;10.24,-20.78,;11.58,-20.01,;11.57,-18.46,;10.23,-17.7,;10.22,-16.16,;11.55,-15.38,;11.54,-13.84,;12.88,-13.07,;14.21,-13.83,;14.21,-15.37,;12.89,-16.14,;15.55,-13.06,;16.88,-13.83,;15.54,-11.52,;16.88,-10.75,;8.91,-18.47,;7.57,-17.71,;6.24,-18.48,;4.9,-17.71,;3.56,-18.48,;12.91,-20.77,;14.32,-20.13,;15.35,-21.27,;14.59,-22.6,;15.23,-24.01,;13.09,-22.29,)|
COc1cc2nc(cc(N[C@H]3CC[C@@H](CC3)C(=O)NO)c2cc1OC)-c1ccc(C)o1 |r,wU:10.9,wD:13.16,(17.68,-22.69,;17.68,-21.15,;19.01,-20.38,;20.35,-21.15,;21.68,-20.37,;23.01,-21.14,;24.35,-20.37,;24.34,-18.82,;23,-18.06,;23,-16.52,;24.33,-15.74,;24.31,-14.2,;25.65,-13.42,;26.98,-14.19,;26.98,-15.73,;25.66,-16.5,;28.32,-13.42,;29.65,-14.19,;28.31,-11.88,;29.65,-11.11,;21.68,-18.83,;20.34,-18.07,;19.01,-18.84,;17.67,-18.06,;16.34,-18.83,;25.69,-21.13,;27.09,-20.49,;28.12,-21.63,;27.36,-22.96,;28,-24.36,;25.86,-22.65,)|
COc1cc2nc(cc(NCC3CCN(CC3)c3ccc(cn3)C(=O)NO)c2cc1OC)-c1ccc(C)o1
COc1cc2nc(C)cc(NCC3CCN(CC3)c3ncc(cn3)C(=O)NO)c2cc1OC
COc1cc2nc(cc(NCC3CCN(CC3)c3ncc(cn3)C(=O)NO)c2cc1OC)C1CCCCC1
COc1cc2nc(cc(NCC3CCN(CC3)c3ncc(cn3)C(=O)NO)c2cc1OC)-c1ccccc1
COc1cc2nc(cc(NCC3CCN(CC3)c3ncc(cn3)C(=O)NO)c2cc1OC)N1CCCCC1
COc1cc2nc(cc(NCC3CCN(CC3)c3ncc(cn3)C(=O)NO)c2cc1OC)-c1cc(C)oc1C
COc1cc2nc(cc(NCC3CCN(CC3)c3ncc(cn3)C(=O)NO)c2cc1OC)-c1ccc(C)s1
COc1cc2nc(nc(NCC3CCN(CC3)c3ncc(cn3)C(=O)NO)c2cc1OC)-c1ccc(C)o1
CCCNc1ccc2C(=O)N(CCCC(=O)NO)C(=O)c3cccc1c23
ONC(=O)CCCCCN1C(=O)c2cccc3c(OCc4ccc(cc4)C(F)(F)F)ccc(C1=O)c23
CN1CC(=O)N(Cc2ccc(cc2)C(=O)NO)C1=O
CCCN1CC(=O)N(Cc2ccc(cc2)C(=O)NO)C1=O
ONC(=O)c1ccc(CN2C(=O)CN(Cc3ccccc3)C2=O)cc1
ONC(=O)c1ccc(CN2C(=O)CN(Cc3ccc(Cl)cc3)C2=O)cc1
Cc1ccc(CN2CC(=O)N(Cc3ccc(cc3)C(=O)NO)C2=O)cc1
COc1ccc(CN2CC(=O)N(Cc3ccc(cc3)C(=O)NO)C2=O)cc1
CC(C)(C)c1ccc(CN2CC(=O)N(Cc3ccc(cc3)C(=O)NO)C2=O)cc1
ONC(=O)c1ccc(CN2C(=O)CN(CCc3ccccc3)C2=O)cc1
Cc1ccc2ccccc2c1N1CC(=O)N(Cc2ccc(cc2)C(=O)NO)C1=O
CC1(NC(=O)N(Cc2ccc(cc2)C(=O)NO)C1=O)c1ccccc1
CCCC1(NC(=O)N(Cc2ccc(cc2)C(=O)NO)C1=O)c1ccccc1
ONC(=O)c1ccc(CN2C(=O)NC(Cc3ccccc3)(C2=O)c2ccccc2)cc1
ONC(=O)c1ccc(CN2C(=O)NC(Cc3ccc(Cl)cc3)(C2=O)c2ccccc2)cc1
Cc1ccc(CC2(NC(=O)N(Cc3ccc(cc3)C(=O)NO)C2=O)c2ccccc2)cc1
COc1ccc(CC2(NC(=O)N(Cc3ccc(cc3)C(=O)NO)C2=O)c2ccccc2)cc1
CC(C)(C)c1ccc(CC2(NC(=O)N(Cc3ccc(cc3)C(=O)NO)C2=O)c2ccccc2)cc1
ONC(=O)c1ccc(CN2C(=O)NC(CCc3ccccc3)(C2=O)c2ccccc2)cc1
ONC(=O)c1ccc(CN2C(=O)NC(Cc3cccc4ccccc34)(C2=O)c2ccccc2)cc1
ONC(=O)c1ccc(CN2C(=O)NC(Cc3ccc4ccccc4c3)(C2=O)c2ccccc2)cc1
CN1C(Cc2ccccc2)C(=O)N(Cc2ccc(cc2)C(=O)NO)C1=O
CCCN1C(Cc2ccccc2)C(=O)N(Cc2ccc(cc2)C(=O)NO)C1=O
ONC(=O)c1ccc(CN2C(=O)C(Cc3ccccc3)N(Cc3ccccc3)C2=O)cc1
ONC(=O)c1ccc(CN2C(=O)C(Cc3ccccc3)N(Cc3ccc(Cl)cc3)C2=O)cc1
Cc1ccc(CN2C(Cc3ccccc3)C(=O)N(Cc3ccc(cc3)C(=O)NO)C2=O)cc1
COc1ccc(CN2C(Cc3ccccc3)C(=O)N(Cc3ccc(cc3)C(=O)NO)C2=O)cc1
CC(C)(C)c1ccc(CN2C(Cc3ccccc3)C(=O)N(Cc3ccc(cc3)C(=O)NO)C2=O)cc1
ONC(=O)c1ccc(CN2C(=O)C(Cc3ccccc3)N(CCc3ccccc3)C2=O)cc1
ONC(=O)c1ccc(CN2C(=O)C(Cc3ccccc3)N(Cc3cccc4ccccc34)C2=O)cc1
ONC(=O)c1ccc(CN2C(=O)C(Cc3ccccc3)N(Cc3ccc4ccccc4c3)C2=O)cc1
ONC(=O)c1ccc(CN2C(=O)C(Cc3ccccc3)N(Cc3ccccn3)C2=O)cc1
ONC(=O)c1ccc(CN2C(=O)C(Cc3ccccc3)N(Cc3cccnc3)C2=O)cc1
ONC(=O)c1ccc(CN2C(=O)C(Cc3ccccc3)N(Cc3ccncc3)C2=O)cc1
CC(C)CC1N(C)C(=O)N(Cc2ccc(cc2)C(=O)NO)C1=O
CCCN1C(CC(C)C)C(=O)N(Cc2ccc(cc2)C(=O)NO)C1=O
CC(C)CC1N(Cc2ccccc2)C(=O)N(Cc2ccc(cc2)C(=O)NO)C1=O
CC(C)(C)OC(=O)Nc1ccc(cc1)-c1cc(NC(=O)CCCCCCC(=O)NO)no1
ONC(=O)c1ccc(Cl)c(NC(=O)c2ccc(cc2)-c2ccccc2)c1
CSc1ccc(cc1NC(=O)c1ccc(cc1)-c1ccccc1)C(=O)NO
ONC(=O)c1ccc(Cl)c(NC(=O)c2ccc(cc2Cl)-c2ccccc2)c1
CCOc1ccc(cc1NC(=O)c1ccc(Cl)cc1Cl)C(=O)NO
CCCOc1ccc(cc1C(=O)Nc1cc(ccc1C)C(=O)NO)C(C)=O
COc1ccc(cc1NC(=O)c2cccc3c2oc4c3cccc4)C(=O)NO
Cc1ccc(cc1C(=O)Nc1ccc(Cl)cc1)C(=O)NO
CCOc1ccc(cc1NC(=O)c1cccc(c1)C(=O)NO)C(C)=O
COc1ccc(cc1NC(=O)c1cc(ccc1OC)C(=O)NO)C(C)=O
CCOc1ccc(cc1NC(=O)c1cc(ccc1Cl)C(=O)NO)C(C)=O
CNC(=O)CCCCCCCn1nc(-c2ccc3oc(N)nc3c2)c2c(N)ncnc12
Nc1ncnc2n(CCCCCCCCC(=O)NO)nc(-c3cnc4[nH]ccc4c3)c12
ONC(=O)\C=C\c1ccc(CN2c3ccccc3Sc3ccccc23)cc1
ONC(=O)CCc1ccc(CN2c3ccccc3Sc3ccccc23)cc1
ONC(=O)c1coc(CN2c3ccccc3Sc3ccccc23)n1
ONC(=O)c1ccc(CN2c3ccccc3Sc3ccccc23)nc1
CNC(=O)c1ccc(CN2c3ccccc3Sc3ccccc23)nc1
CCNC(=O)c1ccc(CN2c3ccccc3Sc3ccccc23)nc1
ONC(=O)Cn1cc(CN2c3ccccc3Sc3ccccc23)cn1
CNC(=O)Cn1cc(CN2c3ccccc3Sc3ccccc23)cn1
CCNC(=O)Cn1cc(CN2c3ccccc3Sc3ccccc23)cn1
C[C@@]12CC3C[C@@](C)(C1)CC(C3)(C2)NCc1ccc(cn1)C(=O)NO |r,TLB:4:3:11:7.5.8,4:5:2.3.10:11,6:5:2:10.9.11,12:9:2:7.4.5,THB:8:5:2:10.9.11,8:9:2:7.4.5|
CN(Cc1ccc(cn1)C(=O)NO)C12CC3C[C@](C)(C[C@](C)(C3)C1)C2 |r,TLB:22:15:24:19.20.23,22:20:16.15.14:24,21:20:16:14.13.24,1:13:16:19.22.20,THB:23:20:16:14.13.24,23:13:16:19.22.20|
CCCN(Cc1ccc(cn1)C(=O)NO)C12CC3C[C@](C)(C[C@](C)(C3)C1)C2 |r,TLB:24:17:26:21.22.25,24:22:18.17.16:26,23:22:18:16.15.26,3:15:18:21.24.22,THB:25:22:18:16.15.26,25:15:18:21.24.22|
CNC(=O)c1ccc(CN(C)C23CC4C[C@](C)(C[C@](C)(C4)C2)C3)nc1 |r,TLB:20:13:22:17.18.21,20:18:14.13.12:22,19:18:14:12.11.22,9:11:14:17.20.18,THB:21:18:14:12.11.22,21:11:14:17.20.18|
CCCN(Cc1ccc(cn1)C(=O)NC)C12CC3C[C@](C)(C[C@](C)(C3)C1)C2 |r,TLB:24:17:26:21.22.25,24:22:18.17.16:26,23:22:18:16.15.26,3:15:18:21.24.22,THB:25:22:18:16.15.26,25:15:18:21.24.22|
CN1CCc2c(C1)c1cc(C)ccc1n2Cc1ccc(cn1)C(=O)NO
COc1ccc2n(Cc3ccc(cn3)C(=O)NO)c3CCN(C)Cc3c2c1
ONC(=O)CCCO\N=C1\C(\Nc2ccccc\12)=C1\C(=O)Nc2ccccc12
OC(=O)CCCO\N=C1\C(\Nc2ccccc\12)=C1\C(=O)Nc2ccccc12
ONC(=O)CCCO\N=C1\C(\Nc2ccccc\12)=C1\C(=O)N(CC#C)c2ccccc12
COc1ccc(cc1OC(C)C(=O)NO)N(C)c1nc(C)nc2ccccc12
CCCC(Oc1cc(ccc1OC)N(C)c1nc(C)nc2ccccc12)C(=O)NO
CCCCC(Oc1cc(ccc1OC)N(C)c1nc(C)nc2ccccc12)C(=O)NO
COc1ccc(cc1OC(C)(C)C(=O)NO)N(C)c1nc(C)nc2ccccc12
COc1ccc(cc1OC(C(C)C)C(=O)NO)N(C)c1nc(C)nc2ccccc12
COc1ccc(cc1OC(C(=O)NO)c1ccccc1)N(C)c1nc(C)nc2ccccc12
COc1ccc(cc1OC1(CCC1)C(=O)NO)N(C)c1nc(C)nc2ccccc12
CCCCCCCSSCC\C=C\[C@@H]1CC(=O)NCc2nc(cs2)C(=O)N\C(=C/C)C(=O)N[C@@H](CCCCN)C(=O)O1 |r|
CCCCCCCSSCC\C=C\[C@@H]1CC(=O)NCc2nc(cs2)C(=O)N\C(=C/C)C(=O)N[C@@H](CCCCNC(=O)CCCCC[N+]2=C(\C=C\C=C\C=C3\N(CC)c4ccc5c(cc(cc5c4C3(C)C)S(O)(=O)=O)S(O)(=O)=O)C(C)(C)c3c2ccc2c(cc(cc32)S(O)(=O)=O)S([O-])(=O)=O)C(=O)O1 |r,c:47|
Nc1nc(NCCc2ccc(cc2)C(=O)NO)nc2nc(nn12)-c1ccco1
Nc1nc(NCCc2ccc(\C=C\C(=O)NO)cc2)nc2nc(nn12)-c1ccco1
Nc1nc(NCCc2ccc(OCCCC(=O)NO)cc2)nc2nc(nn12)-c1ccco1
Nc1nc(NCCc2ccc(OCCCCC(=O)NO)cc2)nc2nc(nn12)-c1ccco1
Nc1nc(NCCc2ccc(OCCCCCC(=O)NO)cc2)nc2nc(nn12)-c1ccco1
Nc1nc(NCCc2ccc(NC(=O)CCCCCCC(=O)NO)cc2)nc2nc(nn12)-c1ccco1
CN(CCc1ccc(cc1)C(=O)NO)c1nc(N)n2nc(nc2n1)-c1ccco1
CCN(CCc1ccc(cc1)C(=O)NO)c1nc(N)n2nc(nc2n1)-c1ccco1
Nc1nc(NCc2ccc(cc2)C(=O)NO)nc2nc(nn12)-c1ccco1
Nc1nc(NCc2ccc(\C=C\C(=O)NO)cc2)nc2nc(nn12)-c1ccco1
Nc1nc(NCc2ccc(OCCCCC(=O)NO)cc2)nc2nc(nn12)-c1ccco1
Nc1nc(NCCCc2ccc(cc2)C(=O)NO)nc2nc(nn12)-c1ccco1
Nc1nc(NCCOc2ccc(cc2)C(=O)NO)nc2nc(nn12)-c1ccco1
CN(CCOc1ccc(cc1)C(=O)NO)c1nc(N)n2nc(nc2n1)-c1ccco1
Nc1nc(NCCCCCCC(=O)NO)nc2nc(nn12)-c1ccco1
Nc1nc(nc2nc(nn12)-c1ccco1)N1CCN(CCc2ccc(cc2)C(=O)NO)CC1
Nc1nc2n(CCc3ccc(cc3)C(=O)NO)ncc2c2nc(nn12)-c1ccco1
Nc1nc2n(CCc3ccc(OCCCCCC(=O)NO)cc3)ncc2c2nc(nn12)-c1ccco1
Nc1nc2n(CCc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)ncc2c2nc(nn12)-c1ccco1
Nc1nc2n(CCCCC(=O)NO)ncc2c2nc(nn12)-c1ccco1
Nc1nc2n(CCCCCC(=O)NO)ncc2c2nc(nn12)-c1ccco1
Nc1nc2n(CCCCCCC(=O)NO)ncc2c2nc(nn12)-c1ccco1
Nc1nc2n(CCN3CCC(CC3)c3ccc(cc3)C(=O)NO)ncc2c2nc(nn12)-c1ccco1
Nc1nc2n(CCN3CCc4ccc(cc4C3)C(=O)NO)ncc2c2nc(nn12)-c1ccco1
Nc1ccccc1NC(=O)c1ccc(CCNc2nc(N)n3nc(nc3n2)-c2ccco2)cc1
Nc1ccccc1NC(=O)c1ccc(CNc2nc(N)n3nc(nc3n2)-c2ccco2)cc1
Nc1ccccc1NC(=O)c1ccc(CCCNc2nc(N)n3nc(nc3n2)-c2ccco2)cc1
Nc1ccccc1NC(=O)c1ccc(OCCNc2nc(N)n3nc(nc3n2)-c2ccco2)cc1
Nc1ccccc1NC(=O)c1ccc(CCn2ncc3c2nc(N)n2nc(nc32)-c2ccco2)cc1
Nc1ccccc1NC(=O)c1ccc(Cn2ncc3c2nc(N)n2nc(nc32)-c2ccco2)cc1
Nc1cc(F)ccc1NC(=O)c1ccc(CCNc2nc(N)n3nc(nc3n2)-c2ccco2)cc1
Nc1nc(NCCc2ccc(O)cc2)nc2nc(nn12)-c1ccco1
CC(C)(F)CN1CCc2cc(O)ccc2C1c1ccc(OCCCCCC(=O)NO)cc1
CC(C)(F)CN1CCc2cc(O)ccc2C1c1ccc(OCCCCCCC(=O)NO)cc1
CC(C)(F)CN1CCc2cc(O)ccc2C1c1ccc(OC2CN(CC(=O)NO)C2)cc1
CCN(CC)CCNC(=O)c1ccc(NC(=O)CCCCCCC(=O)NO)cc1
ONC(=O)CCCCCCC(=O)Nc1ccc(cc1)C(=O)NC1CCNCC1
COc1ccc2[nH]cc(CCNCc3ccc(\C=C\C(=O)NO)cc3)c2c1
COc1ccc2[nH]cc(CCNC(=O)c3ccc(\C=C\C(=O)NO)cc3)c2c1
COc1ccc2[nH]cc(CCNC(=O)\C=C\c3ccc(cc3)C(=O)NO)c2c1
COc1ccc2n(Cc3ccc(\C=C\C(=O)NO)cc3)cc(CCNC(C)=O)c2c1
COc1ccc2n(Cc3ccc(cc3)C(=O)NO)cc(CCNC(C)=O)c2c1
COc1ccc2n(CCCCCC(=O)NO)cc(CCNC(C)=O)c2c1
COc1ccc2[nH]cc(CCN(Cc3ccc(\C=C\C(=O)NO)cc3)C(=O)\C=C\c3ccc(O)c(OC)c3)c2c1
COc1ccc2[nH]cc(CCN(Cc3ccc(cc3)C(=O)NO)C(=O)\C=C\c3ccc(O)c(OC)c3)c2c1
COc1ccc2[nH]cc(CCN(CCCCCC(=O)NO)C(=O)\C=C\c3ccc(O)c(OC)c3)c2c1
COc1ccc2[nH]cc(CCNC(=O)CN(Cc3ccc(\C=C\C(=O)NO)cc3)C(=O)\C=C\c3ccc(O)c(OC)c3)c2c1
COc1ccc2[nH]cc(CCNC(=O)CN(CCCCCC(=O)NO)C(=O)\C=C\c3ccc(O)c(OC)c3)c2c1
CS(=O)(=O)c1ccc(cc1)-n1ccc2cnc(Nc3cnn(CCCCCCC(=O)NO)c3)nc12
ONC(=O)CCCCCCn1cc(Nc2ncc3ccn(Cc4ccccc4F)c3n2)cn1
CS(=O)(=O)c1ccc(cc1)-n1ccc2cnc(Nc3cnn(CCCCCC(=O)NO)c3)nc12
ONC(=O)CCCCCn1cc(Nc2ncc3ccn(-c4ccc(Br)cc4)c3n2)cn1
ONC(=O)CCCCCCn1cc(Nc2ncc3ccn(Cc4ccccc4)c3n2)cn1
ONC(=O)CCCCCCn1cc(Nc2ncc3ccn(-c4ccccc4)c3n2)cn1
ONC(=O)CCCCCn1cc(Nc2ncc3ccn(Cc4cccc(F)c4)c3n2)cn1
ONC(=O)CCCCCn1cc(Nc2ncc3ccn(Cc4ccccc4)c3n2)cn1
ONC(=O)CCCCCCn1cc(Nc2ncc3ccn(Cc4cccc(F)c4)c3n2)cn1
ONC(=O)CCCCCn1cc(Nc2ncc3ccn(Cc4ccccc4F)c3n2)cn1
ONC(=O)CCCCCCn1cc(Nc2ncc3ccn(-c4ccc(Br)cc4)c3n2)cn1
ONC(=O)CCCCCCn1cc(Nc2ncc3ccn(-c4ccc(F)cc4)c3n2)cn1
COc1cccc(Cn2ccc3cnc(Nc4cnn(CCCCCCC(=O)NO)c4)nc23)c1
ONC(=O)CCCCCCn1cc(Nc2ncc3ccn(-c4ccc(Cl)cc4)c3n2)cn1
ONC(=O)CCCCCn1cc(Nc2ncc3ccn(Cc4cccc(Cl)c4)c3n2)cn1
ONC(=O)CCCCCCn1cc(Nc2ncc3ccn(Cc4cccc(Cl)c4)c3n2)cn1
COc1cccc(Cn2ccc3cnc(Nc4cnn(CCCCCC(=O)NO)c4)nc23)c1
ONC(=O)CCCCCCn1cc(Nc2ncc3ccn(Cc4ccccc4Cl)c3n2)cn1
ONC(=O)CCCCCn1cc(Nc2ncc3ccn(Cc4ccccc4Cl)c3n2)cn1
ONC(=O)CCCCCCn1cc(Nc2ncc3ccn(C4CCCC4)c3n2)cn1
ONC(=O)CCCCCCn1cc(Nc2ncc3ccn(CC4CC4)c3n2)cn1
ONC(=O)CCCCCCn1cc(Nc2ncc3ccn(CC4CCCCC4)c3n2)cn1
ONC(=O)c1cccc(\C=C\c2ccnc(c2)-c2ccccc2O)c1
ONC(=O)c1ccc(\C=C\c2ccnc(c2)-c2cc(F)ccc2O)cc1
COc1ccccc1-c1cc(\C=C\c2ccc(cc2)C(=O)NO)ccn1
ONC(=O)c1ccc(\C=C\c2ccnc(c2)-c2cccc(O)c2)cc1
OCc1cccc(c1)-c1cc(\C=C\c2ccc(cc2)C(=O)NO)ccn1
ONC(=O)c1ccc(\C=C\c2ccnc(c2)-c2cccnc2)cc1
Cc1ccc(cc1)-c1cc(\C=C\c2ccc(cc2)C(=O)NO)ccn1
COc1ccc(cc1)-c1cc(\C=C\c2ccc(cc2)C(=O)NO)ccn1
ONC(=O)c1ccc(\C=C\c2cccc(c2)-c2ccccc2O)cc1
ONC(=O)c1ccc(\C=C\c2cccc(c2)-c2cccc(O)c2)cc1
ONC(=O)c1ccc(\C=C\c2cccc(c2)-c2cc(F)ccc2O)cc1
ONC(=O)c1ccc(\C=C\c2ccnc(Br)c2)cc1
ONC(=O)c1ccc(\C=C\c2ccncc2)cc1
ONC(=O)c1ccc(\C=C\c2ccnc(c2)-c2ccsc2)cc1
Cc1ccc(c(F)c1)-c1cncc(\C=C\c2ccc(cc2)C(=O)NO)c1
ONC(=O)c1ccc(\C=C\c2cncc(c2)-c2ccccc2O)cc1
COc1ccc(F)cc1-c1cncc(\C=C\c2ccc(cc2)C(=O)NO)c1
ONC(=O)CCCCCCOc1ccc(cc1)-c1nc2ccc(cc2[nH]1)-c1nc2ccccc2[nH]1
ONC(=O)CCCCCCCOc1cccc(c1)-c1nc2ccc(cc2[nH]1)-c1nc2ccccc2[nH]1
ONC(=O)CCCCCCOc1cccc(c1)-c1nc2ccccc2[nH]1
ONC(=O)CCCCCCCOc1cccc(c1)-c1nc2ccccc2[nH]1
ONC(=O)c1ccc(CNS(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2ccccc2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2ccc(F)cc2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2ccc(cc2)C(F)(F)F)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
CN(C)c1ccc(CN(Cc2ccc(cc2)C(=O)NO)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
Cc1ccc(CN(Cc2ccc(cc2)C(=O)NO)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
CC(C)(C)c1ccc(CN(Cc2ccc(cc2)C(=O)NO)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2ccncc2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2ccncc2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2ccccc2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2ccc(F)cc2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2cccc(F)c2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2ccccc2F)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(Cc2ccccn2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
c1cc(cnc1)CN(Cc2ccc(cc2)C(=O)NO)S(=O)(=O)c3cc(c(c(c3F)F)F)F
ONC(=O)CCCCCCC(=O)N\N=C\c1ccc(cc1)N(c1ccccc1)c1ccccc1
CCCNNC(=O)c1ccc(CNC(=O)c2cc3cc(OCC=C)ccc3o2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2cc3cc(O)ccc3o2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2cc3cc(OC)ccc3o2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2cc3cc(Br)ccc3o2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2cc3cc(Cl)ccc3o2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2cc3cc(F)ccc3o2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2cc3cc(OC)ccc3[nH]2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2cc3cc(Br)ccc3[nH]2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2nc3ccccc3s2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2cc3cc(Cl)ccc3[nH]2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2nc3ccccc3[nH]2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2cc3cc(F)ccc3[nH]2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2cc3ccccc3s2)cc1
CCCNNC(=O)\C=C\c1ccc(CNCCc2c(C)[nH]c3ccccc23)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2cc3ccccc3o2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2cc3ccccc3[nH]2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2ccc3cnccc3n2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2ccc3ccncc3c2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2ccc3cnccc3c2)cc1
CCCNNC(=O)c1ccc(CNC(=O)\C=C\c2ccccc2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2ccc3ccccc3n2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2cc3ccccc3cn2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2cnc3ccccc3c2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2ccc3ccccc3c2)cc1
ONC(=O)CCCCCCNc1nn2c(nc3ccc(Br)cc3c2=O)c2ccccc12
ONC(=O)CCCCCCCNc1nn2c(nc3ccc(Br)cc3c2=O)c2ccccc12
ONC(=O)CCCCCCNc1nn2c(nc3ccc(Cl)cc3c2=O)c2ccccc12
ONC(=O)CCCCCCNc1nn2c(nc3ccc(F)cc3c2=O)c2ccccc12
Cc1ccc2nc3c4ccccc4c(NCCCCCCC(=O)NO)nn3c(=O)c2c1
ONC(=O)CCCCCCNc1nn2c(nc3ccccc3c2=O)c2ccccc12
ONC(=O)CCCCCCCNc1nn2c(nc3ccc(Cl)cc3c2=O)c2ccccc12
ONC(=O)CCCCCCCNc1nn2c(nc3ccc(F)cc3c2=O)c2ccccc12
Cc1ccc2nc3c4ccccc4c(NCCCCCCCC(=O)NO)nn3c(=O)c2c1
ONC(=O)CCCCCCCNc1nn2c(nc3ccccc3c2=O)c2ccccc12
COc1ccccc1-c1ncc(s1)C(=O)NCCCCCCC(=O)NO
COc1ccc(cc1)-c1ncc(s1)C(=O)NCCCCCCC(=O)NO
COc1cccc(c1)-c1ncc(s1)C(=O)NCCCCCCC(=O)NO
COc1cc(OC)cc(c1)-c1ncc(s1)C(=O)NCCCCCCC(=O)NO
COc1ccc(-c2ncc(s2)C(=O)NCCCCCCC(=O)NO)c(OC)c1
COc1cc(cc(OC)c1OC)-c1ncc(s1)C(=O)NCCCCCCC(=O)NO
ONC(=O)CCCCCCNC(=O)c1cnc(s1)-c1ccc(OC(F)(F)F)cc1
COc1ccc(-c2ncc([nH]2)C(=O)NCCCCCCC(=O)NO)c(OC)c1
CC(C)(C)OC(=O)Nc1ccc(cc1)-c1ncc(s1)C(=O)NCCCCCCC(=O)NO
COc1ccc(-c2ncc(s2)C(=O)NCCCCCC(=O)NO)c(OC)c1
COc1ccc(-c2ncc(s2)C(=O)NCCCCC(=O)NO)c(OC)c1
Cc1ccc(cc1)-c1ncc(\C=C\C(=O)Nc2ccccc2N)s1
COc1cccc(c1)-c1ncc(\C=C\C(=O)Nc2ccccc2N)s1
COc1ccc(cc1)-c1ncc(\C=C\C(=O)Nc2ccccc2N)s1
COc1ccc(cc1OC)-c1ncc(\C=C\C(=O)Nc2ccccc2N)s1
COc1ccc(-c2ncc(\C=C\C(=O)Nc3ccccc3N)s2)c(OC)c1OC
COc1cc(cc(OC)c1OC)-c1ncc(\C=C\C(=O)Nc2ccccc2N)s1
Nc1ccccc1NC(=O)\C=C\c1cnc(s1)-c1ccc2cc[nH]c2c1
COc1ccc(cc1)-c1ncc(\C=C\C(=O)NO)s1
ONC(=O)\C=C\c1cnc(s1)-c1ccc2OCCOc2c1
COc1cc(OC)cc(c1)-c1ncc(\C=C\C(=O)NO)s1
COc1ccc(-c2ncc(\C=C\C(=O)NO)s2)c(OC)c1OC
COc1cc(cc(OC)c1OC)-c1ncc(\C=C\C(=O)NO)s1
ONC(=O)\C=C\c1cnc(s1)-c1ccc(cc1)N1CCOCC1
CC(C)(C)OC(=O)CC(O)\C=C\CCSSCC\C=C\C(O)CC(=O)OC(C)(C)C
Cn1cc(CN2CC3(C2)CCN(C3)c2ncc(cn2)C(=O)NO)c2ccc(cc12)C#N
CN1C2N(CCc3c2[nH]c2ccc(OCc4ccc(\C=C\C(=O)NO)cc4)cc32)C(=O)c2cc(F)ccc12
CN1C2N(CCc3c2[nH]c2ccc(OCc4ccc(\C=C\C(=O)Nc5ccccc5N)cc4)cc32)C(=O)c2cc(F)ccc12
ONC(=O)CCCSC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1cccc2ccccc12 |r|
ONC(=O)CCCSC[C@H](NC(=O)c1ccccc1)C(=O)Nc1ccccc1 |r|
ONC(=O)CCCSC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1ccccc1 |r|
CCc1c(c([nH]c1C(=O)Nc2cccc(c2)CCC(=O)NO)C)C(=O)C
CCc1c([nH]c(C)c1C(C)=O)C(=O)Nc1cccc(\C=C\C(=O)NO)c1
CCc1c([nH]c(C)c1C(C)=O)C(=O)Nc1cccc(CCC(=O)Nc2ccccc2N)c1
CCc1c([nH]c(C)c1C(C)=O)C(=O)Nc1cccc(CCC(=O)OC)c1
Cn1cccc1C(=O)Nc1cccc(CCC(=O)NO)c1
CCc1c([nH]c(C)c1C(C)=O)C(=O)Nc1cc(\C=C\C(=O)NO)ccc1OC
CCc1c([nH]c(C)c1C(C)=O)C(=O)Nc1cc(\C=C\C(=O)NO)ccc1O
CCc1c([nH]c(C)c1C(C)=O)C(=O)Nc1cc(ccc1OC)S(=O)(=O)Nc1cccc(\C=C\C(=O)NO)c1
COc1ccc(cc1NC(=O)c1[nH]c(C)c2c1CCCCC2=O)S(=O)(=O)n1ccc(\C=C\C(=O)NO)c1
Cc1[nH]c(C(=O)Nc2cc(ccc2OCCCCCCCC(=O)NO)S(=O)(=O)N2CCOCC2)c2CCCCC(=O)c12
Cc1c2c(CCCCC2=O)c(C(=O)Nc2cc(ccc2OCCCCCCCC(=O)NO)S(=O)(=O)N2CCOCC2)n1C
COC(=O)CCCCCCCOc1ccc(cc1NC(=O)c1c2CCCCC(=O)c2c(C)n1C)S(=O)(=O)N1CCOCC1
ONC(=O)\C=C\c1ccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)cc1
ONC(=O)c1ccc(cc1)N1CCc2cc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)ccc12
ONC(=O)c1ccc(cc1)N1CCCc2cc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)ccc12
ONC(=O)c1ccc(CN2CCc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)cc23)cc1
ONC(=O)\C=C\c1ccc(CN2CCc3cc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)ccc23)cc1
ONC(=O)CCCCCCC(=O)N\N=C\c1cnc(nc1)N(c1ccccc1)c1ccccc1
OCCN(C(=O)Cc1ccccc1)C(=O)Cc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(Cn2sc3ccccc3c2=O)cc1
ONC(=O)c1ccc(CN2C(=O)CSC2=O)cc1
COc1ccc2C(=O)N(Cc3ccc(cc3)C(=O)NO)C(=O)c3cccc1c23
CCCC1=C(Nc2ccc(cc2)C(=O)NO)C2N=CC=CC2=N1 |c:3,18,20,23|
CC(C)(C)OC(=O)Nc1cccc(c1)-c1cc(no1)C(=O)NCCc1cc(no1)C(=O)NO
Fc1ccc(cc1Cl)N(Cc1ccc(cn1)-c1nnc(o1)C(F)(F)F)S(=O)(=O)N1CCN(CC1)C1COC1
Fc1cc(ccc1CN(c1cccnc1)S(=O)(=O)N1CCNCC1)-c1nnc(o1)C(F)(F)F
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(OCCCCCCC(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(OCCCC(=O)NO)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(OCc2ccc(cc2)C(=O)NO)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(O\C=C\c2ccc(CC(=O)NO)cc2)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)CC(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)CCCC(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)CCCCC(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)CCCCCC(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)CCCCCCC(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)c2ccc(cc2)C(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)\C=C\C(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)CCC(=O)NO)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)CCCC(=O)NO)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)CCCCC(=O)NO)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)CCCCCC(=O)NO)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NC(=O)\C=C\C(=O)NO)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NCC(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(NCCC(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(cc1)C#CCCC(=O)Nc1ccccc1N
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(\C=C\C(=O)Nc2ccccc2N)cc1
COc1cc(cc(OC)c1OC)C(=O)c1csc(n1)-c1ccc(\C=C\C(=O)NO)cc1
CC(C)(C)OC(=O)Nc1cccc(c1)C(=O)\C=C\c1ccc(\C=C\C(=O)NO)cc1
CN(CC#C)Cc1cccc(NC(=O)CCCCCCC(=O)NO)c1
Nc1ncc(cn1)-c1cc(N2CCOCC2)c(=O)n(Cc2ccc(cc2)C(=O)NO)n1
Nc1ncc(cn1)-c1cc(N2CCOCC2)c(=O)n(Cc2ccc(cc2)C(=O)NO)c1
Nc1ncc(cn1)-c1cn(Cc2ccc(cc2)C(=O)NO)c(=O)c(n1)N1CCOCC1
Nc1ncc(cn1)-c1cn(Cc2cccc(c2)C(=O)NO)c(=O)c(n1)N1CCOCC1
Nc1ncc(cn1)-c1cn(CCCCCC(=O)NO)c(=O)c(n1)N1CCOCC1
Nc1ncc(cn1)-c1cn(CCCCCCC(=O)NO)c(=O)c(n1)N1CCOCC1
Nc1ncc(cn1)-c1cn(CCCCCCCC(=O)NO)c(=O)c(n1)N1CCOCC1
Nc1ccc(cn1)-c1cn(Cc2ccc(cc2)C(=O)NO)c(=O)c(n1)N1CCOCC1
Nc1ccc(cc1)-c1cn(Cc2ccc(cc2)C(=O)NO)c(=O)c(n1)N1CCOCC1
CNc1ncc(cn1)-c1cn(Cc2ccc(cc2)C(=O)NO)c(=O)c(n1)N1CCOCC1
ONC(=O)c1ccc(Cn2cc(nc(N3CCOCC3)c2=O)-c2cccnc2)cc1
ONC(=O)c1ccc(Cn2cc(nc(N3CCOCC3)c2=O)-c2cncnc2)cc1
ONC(=O)c1ccc(Cn2cc(nc(N3CCOCC3)c2=O)-c2ccc(O)cc2)cc1
ONC(=O)c1ccc(Cn2cc(nc(N3CCOCC3)c2=O)-c2cccc(O)c2)cc1
OCc1ccc(cc1)-c1cn(Cc2ccc(cc2)C(=O)NO)c(=O)c(n1)N1CCOCC1
OCc1cccc(c1)-c1cn(Cc2ccc(cc2)C(=O)NO)c(=O)c(n1)N1CCOCC1
Cn1cc(cn1)-c1cn(Cc2ccc(cc2)C(=O)NO)c(=O)c(n1)N1CCOCC1
ONC(=O)c1ccc(Cn2cc(nc(N3CCOCC3)c2=O)-c2cn[nH]c2)cc1
ONC(=O)c1ccc(Cn2cc(nc(N3CCOCC3)c2=O)-c2ccoc2)cc1
Cc1noc(C)c1-c1cn(Cc2ccc(cc2)C(=O)NO)c(=O)c(n1)N1CCOCC1
ONC(=O)c1ccc(Cn2cc(nc(N3CCOCC3)c2=O)-c2cccc3[nH]ncc23)cc1
Nc1ncc(cn1)-c1cn(Cc2ccc(cc2)C(=O)NO)c(=O)c(n1)N1CCCCC1
CN1CCN(CC1)c1nc(cn(Cc2ccc(cc2)C(=O)NO)c1=O)-c1cnc(N)nc1
COC1CCN(CC1)c1nc(cn(Cc2ccc(cc2)C(=O)NO)c1=O)-c1cnc(N)nc1
Nc1ncc(cn1)-c1cn(Cc2ccc(cc2)C(=O)NO)c(=O)c(Nc2ccccc2)n1
ONC(=O)CCCCCCNC(=O)c1csc(n1)C#C
ONC(=O)CCCCC\C=C/c1csc(n1)C#C
ONC(=O)CCCCC\C=C\c1csc(n1)C#C
ONC(=O)\C=C\C=C\c1csc(n1)C#C
ONC(=O)\C=C\c1csc(n1)C#C
ONC(=O)CCCCCCNC(=O)c1csc(Br)n1
ONC(=O)CCCCC\C=C/c1csc(Br)n1
ONC(=O)CCCCC\C=C\c1csc(Br)n1
ONC(=O)\C=C\C=C\c1csc(Br)n1
ONC(=O)\C=C\c1csc(Br)n1
Cc1cc(C)cc(c1)C(=O)N(CC(=O)NC1CCCCC1)Cc1ccc(cc1F)C(=O)NO
CN(C)c1ccc(cc1)C(=O)N(CC(=O)NC1CCCCC1)Cc1ccc(cc1F)C(=O)NO
ONC(=O)c1ccc(CN(CC(=O)NC2CCCCC2)C(=O)c2ccccc2F)c(F)c1
Cc1ccccc1C(=O)N(CC(=O)NC1CCCCC1)Cc1ccc(cc1F)C(=O)NO
COc1ccccc1C(=O)N(CC(=O)NC1CCCCC1)Cc1ccc(cc1F)C(=O)NO
ONC(=O)c1ccc(CN(CC(=O)NC2CCCCC2)C(=O)c2ccccc2C(F)(F)F)c(F)c1
Cc1cc(C)cc(c1)C(=O)N(CC(=O)NCc1ccccc1)Cc1ccc(cc1F)C(=O)NO
CN(C)c1ccc(cc1)C(=O)N(Cc2ccc(cc2F)C(=O)NO)CC(=O)NCc3ccccc3
Cc1cc(C)cc(c1)C(=O)N(CC(=O)NC(C)(C)C)Cc1ccc(cc1F)C(=O)NO
CN(C)c1ccc(cc1)C(=O)N(CC(=O)NC(C)(C)C)Cc1ccc(cc1F)C(=O)NO
CC(C)(C)NC(=O)CN(Cc1ccc(cc1F)C(=O)NO)C(=O)c1ccccc1F
Cc1ccccc1C(=O)N(CC(=O)NC(C)(C)C)Cc1ccc(cc1F)C(=O)NO
COc1ccccc1C(=O)N(CC(=O)NC(C)(C)C)Cc1ccc(cc1F)C(=O)NO
CC(C)(C)NC(=O)CN(Cc1ccc(cc1F)C(=O)NO)C(=O)c1ccccc1C(F)(F)F
CC(C)(C)NC(=O)CN(Cc1ccc(cc1F)C(=O)NO)C(=O)c1ccccc1Cl
CC(C)c1ccccc1C(=O)N(CC(=O)NC(C)(C)C)Cc1ccc(cc1F)C(=O)NO
Cc1ccccc1C(=O)N(CC(=O)NC(C)(C)C)Cc1ccc(cc1)C(=O)NO
COc1ccccc1C(=O)N(CC(=O)NC(C)(C)C)Cc1ccc(cc1)C(=O)NO
ONC(=O)\C=C\c1ccc(CCCCCCc2n[nH]c(=O)c3cc(F)ccc23)cc1
ONC(=O)CCCCCCOc1ccc(cc1)-c1nnc(s1)-c1ccccc1
ONC(=O)CCCCOc1cccc(c1)-c1nnc(s1)-c1ccccc1
ONC(=O)CCCCCOc1cccc(c1)-c1nnc(s1)-c1ccccc1
ONC(=O)CCCCCCOc1cccc(c1)-c1nnc(s1)-c1ccccc1
ONC(=O)CCCCCCOc1cccc(c1)-c1nnc(s1)-c1ccccc1Cl
CCCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](CCCCCS)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CO)NC(=O)[C@H](C)NC(=O)[C@H](CCCCN)NC1=O |r|
CC(C)n1ncc2c(cc(cc12)-c1ccc(nc1)N1CCN(CCCC(=O)NO)CC1)C(=O)NCc1c(C)cc(C)[nH]c1=O
CC(C)n1ncc2c(cc(cc12)-c1ccc(nc1)N1CCN(CCCCC(=O)NO)CC1)C(=O)NCc1c(C)cc(C)[nH]c1=O
CC(C)n1ncc2c(cc(cc12)-c1ccc(nc1)N1CCN(CCCCCC(=O)NO)CC1)C(=O)NCc1c(C)cc(C)[nH]c1=O
CC(C)n1ncc2c(cc(cc12)-c1ccc(nc1)N1CCN(CCCCCCC(=O)NO)CC1)C(=O)NCc1c(C)cc(C)[nH]c1=O
CC(C)n1ncc2c(cc(cc12)-c1ccc(nc1)N1CCN(CCCCCCCC(=O)NO)CC1)C(=O)NCc1c(C)cc(C)[nH]c1=O
CC(C)n1ncc2c(cc(cc12)-c1ccc(nc1)N1CCN(CCCCCCCCC(=O)NO)CC1)C(=O)NCc1c(C)cc(C)[nH]c1=O
CC(C)n1ncc2c(cc(cc12)-c1ccc(nc1)N1CCN(CCCCCCCCCC(=O)NO)CC1)C(=O)NCc1c(C)cc(C)[nH]c1=O
CC(C)n1ncc2c(cc(cc12)-c1ccc(nc1)N1CCN(Cc2ccc(cc2)C(=O)NO)CC1)C(=O)NCc1c(C)cc(C)[nH]c1=O
CC(C)n1ncc2c(cc(cc12)-c1ccc(nc1)N1CCN(Cc2ccc(o2)C(=O)NO)CC1)C(=O)NCc1c(C)cc(C)[nH]c1=O
CC(C)n1ncc2c(cc(cc12)-c1ccc(nc1)N1CCN(Cc2ccc(NC(=O)CCCCCCC(=O)NO)cc2)CC1)C(=O)NCc1c(C)cc(C)[nH]c1=O
CC(C)n1ncc2c(cc(cc12)-c1ccc(nc1)N1CCN(CC1)c1ncc(cn1)C(=O)NO)C(=O)NCc1c(C)cc(C)[nH]c1=O
CC(C)n1ncc2c(cc(cc12)-c1ccc(nc1)N1CCN(CC1)C(=O)CCCC(=O)NO)C(=O)NCc1c(C)cc(C)[nH]c1=O
CC(C)n1ncc2c(cc(cc12)-c1ccc(nc1)N1CCN(CC1)C(=O)CCCCC(=O)NO)C(=O)NCc1c(C)cc(C)[nH]c1=O
CC(C)n1ncc2c(cc(cc12)-c1ccc(nc1)N1CCN(CC1)C(=O)CCCCCC(=O)NO)C(=O)NCc1c(C)cc(C)[nH]c1=O
CC(C)n1ncc2c(cc(cc12)-c1ccc(nc1)N1CCN(CC1)C(=O)CCCCCCC(=O)NO)C(=O)NCc1c(C)cc(C)[nH]c1=O
CC(C)n1ncc2c(cc(cc12)-c1ccc(NC(=O)CCCCCCC(=O)NO)cc1)C(=O)NCc1c(C)cc(C)[nH]c1=O
CC(C)n1ncc2c(cc(cc12)-c1ccc(NC(=O)CCCCCC(=O)NO)cc1)C(=O)NCc1c(C)cc(C)[nH]c1=O
Cc1cc(C)c(CNC(=O)c2cc(cc(NCCCCC(=O)NO)c2C)-c2ccc(nc2)N2CCN(CC2)C(=O)OC(C)(C)C)c(=O)[nH]1
Cc1cc(C)c(CNC(=O)c2cc(cc(NCCCCCC(=C)NO)c2C)-c2ccc(nc2)N2CCN(CC2)C(=O)OC(C)(C)C)c(=O)[nH]1
Cc1cc(C)c(CNC(=O)c2cc(cc(NCCCCCCC(=O)NO)c2C)-c2ccc(nc2)N2CCN(CC2)C(=O)OC(C)(C)C)c(=O)[nH]1
Cc1cc(C)c(CNC(=O)c2cc(cc(NCCCCCCCC(=O)NO)c2C)-c2ccc(nc2)N2CCN(CC2)C(=O)OC(C)(C)C)c(=O)[nH]1
Cc1cc(C)c(CNC(=O)c2cc(cc(NC(=O)CCCC(=O)NO)c2C)-c2ccc(nc2)N2CCN(CC2)C(=O)OC(C)(C)C)c(=O)[nH]1
Cc1cc(C)c(CNC(=O)c2cc(cc(NC(=O)CCCCC(=O)NO)c2C)-c2ccc(nc2)N2CCN(CC2)C(=O)OC(C)(C)C)c(=O)[nH]1
CC[C@@H](C)n1cc(C)c2c(cc(cc12)-c1ccc(nc1)N1CCN(CCCCCCCCC(=O)NO)CC1)C(=O)NCc1c(C)cc(C)[nH]c1=O |r|
CC[C@@H](C)n1cc(C)c2c(cc(cc12)-c1ccc(nc1)N1CCN(CC1)c1ncc(cn1)C(=O)NO)C(=O)NCc1c(C)cc(C)[nH]c1=O |r|
CCN(C1CCOCC1)c1cc(cc(C(=O)NCc2c(C)cc(C)[nH]c2=O)c1C)-c1ccc(nc1)N1CCN(CCCCCCCCC(=O)NO)CC1
CCN(C1CCOCC1)c1cc(cc(C(=O)NCc2c(C)cc(C)[nH]c2=O)c1C)-c1ccc(nc1)N1CCN(CC1)c1ncc(cn1)C(=O)NO
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(CC2CC(C2)C(=O)NO)ccc1OCC |(22.02,-12.67,;21.55,-11.21,;20.04,-10.88,;19.56,-9.42,;20.47,-8.18,;19.56,-6.94,;20.04,-5.47,;18.11,-7.41,;18.11,-8.95,;16.78,-9.72,;15.45,-8.95,;15.45,-7.41,;16.78,-6.63,;16.78,-5.09,;14.12,-9.72,;14.12,-11.26,;12.8,-12.03,;12.8,-13.57,;14.14,-14.34,;14.54,-15.82,;16.02,-15.42,;15.62,-13.93,;17.36,-16.18,;18.69,-15.4,;17.37,-17.72,;16.04,-18.5,;11.45,-11.27,;11.45,-9.72,;12.78,-8.95,;12.78,-7.41,;11.45,-6.64,;11.45,-5.1,)|
CCCc1nn(C)c2c1nc([nH]c2=O)-c1cc(Cc2ccc(cc2)C(=O)Nc2ccccc2N)ccc1OCC
C[C@H]1CN(Cc2ccc(cc2)C(=O)NO)C[C@@H]1c1nc2n(ncc2c(=O)[nH]1)C1CCCC1 |r|
C[C@H]1CN(Cc2ccc(\C=C\C(=O)NO)cc2)C[C@@H]1c1nc2n(ncc2c(=O)[nH]1)C1CCOCC1 |r|
C[C@H](N1CC(Cc2ccc(cc2)C(=O)Nc2ccccc2N)C1)c1nc2n(ncc2c(=O)[nH]1)C1CCCC1 |r|
ONC(=O)CCCCNC(=S)Nc1ccc(\C=C\C(=O)c2cccnc2)cc1
COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](O[C@H]5C[C@H](N)[C@H](O)[C@H](C)O5)c4c(O)c3C(=O)c12)C(C)=O |r|
ONC(=O)CCCCc1cn(nn1)-c1ccc(cc1)C(=O)c1c(sc2cc(O)ccc12)-c1ccc(O)cc1
ONC(=O)CCCCCCN1CC(N=N1)c1ccc2ncnc(Nc3ccc(Br)cc3F)c2c1 |c:13|
ONC(=O)c1ccc(\C=N\NC(=O)c2cc(nc(n2)-c2cccc(O)c2)N2CCOCC2)cc1
ONC(=O)c1ccc(\C=N\NC(=O)c2cc(nc(n2)-c2cccc3[nH]ncc23)N2CCOCC2)cc1
CC(C)n1c(C)nc2c(F)cc(cc12)-c1nc(Nc2ccc(CNC(=O)CCCCCCC(=O)NO)cc2)ncc1F
ONC(=O)CCCCCNC(=O)c1cccc2cc3ccccc3nc12
C[C@H]1COc2c(N3CCN(C)CC3)c(F)cc3c2n1cc(C(=O)NCC1CN(CC(=O)NO)N=N1)c3=O |r,c:36|
CCC(CC)(c1ccc(OCC(O)C(C)(C)C)c(C)c1)c1ccc(OCC(=O)NO)c(C)c1
ONC(=O)c1ccc(NC(=O)N2CCC(CC2)N2[C@@H]([C@H](C2=O)c2ccccc2)c2ccccc2)cc1 |r|
ONC(=O)c1ccc(CC(=O)N2CCC(CC2)N2[C@@H]([C@H](C2=O)c2ccccc2)c2ccccc2)cc1 |r|
ONC(=O)c1ccc(CNC(=O)N2CCC(CC2)N2[C@@H]([C@H](C2=O)c2ccccc2)c2ccccc2)cc1 |r|
ONC(=O)c1ccc(\C=C\C(=O)N2CCC(CC2)N2[C@@H]([C@H](C2=O)c2ccccc2)c2ccccc2)cc1 |r|
ONC(=O)\C=C\c1ccc(cc1)C(=O)N1CCC(CC1)N1[C@@H]([C@H](C1=O)c1ccccc1)c1ccccc1 |r|
ONC(=O)c1ccc(CC(=O)N2CCC(CC2)N2CC(C2=O)(c2ccccc2)c2ccccc2)cc1
ONC(=O)c1ccc(CNC(=O)N2CCC(CC2)N2CC(C2=O)(c2ccccc2)c2ccccc2)cc1
ONC(=O)c1ccc(COC(=O)N2CCC(CC2)N2CC(C2=O)(c2ccccc2)c2ccccc2)cc1
Cc1cccc(c1)C1CC(=O)N1C1CCN(CC1)C(=O)NCc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(CNC(=O)N2CCC(CC2)N2C(CC2=O)c2cccc(Cl)c2)cc1
CCCNNC(=O)c1ccc(NC(=O)Cc2ccccc2)cc1
CCCNNC(=O)c1ccc(Nc2ccccc2)cc1
Nc1ccccc1NC(=O)c1cnc(NCc2ccccc2)cn1
NC(=O)c1ccc(COc2ccc(cc2)-n2cc3cccc(C(N)=O)c3n2)cc1
NC(=O)\C=C\c1ccc(COc2ccc(cc2)-n2cc3cccc(C(N)=O)c3n2)cc1
ONC(=O)COc1ccc(CNCCc2c[nH]c3ccccc23)c(F)c1
Cc1[nH]c2ccccc2c1C1=CCC(CC1)NCc1ccc(OCC(=O)NO)cc1F |t:12|
COc1ccc(cc1\C=C\C(=O)NO)N(C)c1cc(nc2ccccc12)C#N
COc1ccc(cc1\C=C\C(=O)NO)N(C)c1nc(C)nc2ccccc12
CC(C)c1cc(C(=O)N(C)Cc2ccc(cc2)C(=O)NO)c(O)cc1O
CN(Cc1ccc(cc1)C(=O)NO)C(=O)c1ccccc1
ONC(=O)\C=C\c1ccc(CNc2ccc3nc4CCCCCn4c(=O)c3c2)cc1
CN(C)CCCNC(=O)c1ccc(C=C2/CCn3c2nc2cc(N4CCN(CCCCCCCC(=O)NO)CC4)c(F)cc2c3=O)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2ccccc2)cc1
CCNNC(=O)c1ccc(CNC(=O)c2ccccc2)cc1
CNNC(=O)c1ccc(CNC(=O)c2ccccc2)cc1
CCCCN(Cc1ccc(cc1)C(=O)NNCC)C(=O)c1ccccc1
CCCCN(Cc1ccc(cc1)C(=O)NNCC)C(=O)Nc1ccccc1
CCNNC(=O)c1ccc(CNc2cccc3cccnc23)cc1
CCNNC(=O)c1ccc(CNC(=O)Nc2cccc3cccnc23)cc1
CCNNC(=O)c1ccc(NC(=O)Nc2cccc3cccnc23)cc1
CCNNC(=O)c1ccc(Cn2ccc3cc(ccc23)C(=O)c2ccc(OC)cc2)cc1
CCNNC(=O)c1csc(n1)-c1cccnc1
CCNNC(=O)c1coc(c1)-c1ccc(Br)cc1
CCNNC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3ccccc3)c2=O)cc1
CCNNC(=O)c1ccc(Cn2nnnc2-c2cccs2)cc1
CCNNC(=O)c1ccc(CN2c3ccccc3Sc3ccccc23)cc1
CCNNC(=O)c1ccc(CN2c3ccccc3Sc3cccnc23)cc1
CCNNC(=O)c1ccc(Cn2c3ccccc3c3ccccc23)cc1
CCNNC(=O)c1ccc(Cn2c3CCCCc3c3ccccc23)cc1
CCNNC(=O)c1ccc(Cn2c3ccccc3c3cccnc23)cc1
CCNNC(=O)c1ccc(Cn2c3ccccc3c3ccncc23)cc1
CCNNC(=O)c1ccc(Cn2c3ccccc3c3cnccc23)cc1
CCNNC(=O)c1ccc(CN2c3ccccc3Oc3ccccc23)cc1
CCNNC(=O)c1ccc(CN2c3ccccc3Cc3ccccc23)cc1
CCNNC(=O)c1ccc(CN2c3ccccc3C=Cc3ccccc23)cc1 |c:19|
CCNNC(=O)c1ccc(CN2c3ccccc3C=Cc3ccncc23)cc1 |c:19|
CCNNC(=O)c1ccc(CN2c3ccccc3C=Cc3nc(C)nc(C)c23)cc1 |c:19|
CCNNC(=O)c1ccc(CN2c3ccccc3C=Cc3ccc(C)cc23)cc1 |c:19|
CCNNC(=O)c1ccc(CN2c3ccccc3C=Cc3ccc(F)cc23)cc1 |c:19|
CCNNC(=O)c1ccc(CN2c3ccccc3C=Cc3ccc(cc23)C(F)(F)F)cc1 |c:19|
CCNNC(=O)c1ccc(CN2c3ccccc3CCc3ccccc23)cc1
CCNNC(=O)c1ccc(CN2c3ccccc3CC(=O)c3ccccc23)cc1
CC1(CCN(CC1)c1cnc(c(N)n1)-c1cccc(Cl)c1Cl)NCC(=O)NCc1ccc(\C=C\C(=O)NO)cc1
CC1(CCN(CC1)c1cnc(c(N)n1)-c1cccc(Cl)c1Cl)NCc1ccc(cc1)C(=O)NCc1ccc(\C=C\C(=O)NO)cc1
Clc1ccc(cc1Cl)C1CC(=NN1C(=O)COc1ccc(\C=C2\SC(=O)NC2=O)cc1)c1ccccc1 |c:11|
Fc1ccc(cc1)C1=NN(C(C1)c1ccco1)C(=O)COc1ccc(\C=C2\SC(=O)NC2=O)cc1 |t:8|
Fc1ccc(cc1)C1=NN(C(C1)c1ccc(Cl)c(Cl)c1)C(=O)COc1ccc(\C=C2\SC(=O)NC2=O)cc1 |t:8|
CC(N1CCN(Cc2ccc(cc2)C(=O)NO)CC1)c1ccccc1
ONC(=O)c1ccc(CN2CCN(CC2)C(c2ccccc2)c2ccccc2)cc1
ONC(=O)c1ccc(CCN2CCN(CC2)C(c2ccccc2)c2ccccc2)cc1
ONC(=O)c1ccc(CCCN2CCN(CC2)C(c2ccccc2)c2ccccc2)cc1
ONC(=O)c1ccc(CCCCN2CCN(CC2)C(c2ccccc2)c2ccccc2)cc1
ONC(=O)c1ccccc1CN1CCN(CC1)C(c1ccccc1)c1ccccc1
ONC(=O)c1cccc(CN2CCN(CC2)C(c2ccccc2)c2ccccc2)c1
ONC(=O)c1ccc(CN2CCN(Cc3ccccc3)CC2)cc1
ONC(=O)c1ccc(\C=N\NC(=O)c2ccnc(n2)-c2ccccc2)cc1
Nc1ccccc1NC(=O)CCCCCCC(=O)Nc1ccccc1
CCCNNC(=O)CCCCCCC(=O)Nc1ccccc1
COc1ccc(Cn2ccc3ccc(cc23)C(=O)NO)cc1C(=O)NCCNc1ccc(c2nonc12)S(=O)(=O)N(C)C
COc1ccc(Cn2ccc3ccc(cc23)C(=O)NO)cc1C(=O)NCCCNc1ccc(c2nonc12)S(=O)(=O)N(C)C
COc1ccc(Cn2ccc3ccc(cc23)C(=O)NO)cc1C(=O)NCCCCNc1ccc(c2nonc12)S(=O)(=O)N(C)C
CN(Cc1ccc(cc1)C(=O)NO)S(=O)(=O)c1c(F)c(F)c(F)c(F)c1F
CC(C)N(Cc1ccc(cc1)C(=O)NO)S(=O)(=O)c1c(F)c(F)c(F)c(F)c1F
ONC(=O)c1ccc(CN(C2CC2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc(CN(C2CC2)S(=O)(=O)c2c(F)c(F)cc(F)c2F)cc1
ONC(=O)c1ccc(CN(C2CC2)S(=O)(=O)c2ccc(F)cc2)cc1
ONC(=O)c1ccc(CN(C2CC2)S(=O)(=O)c2cc(F)c(F)c(F)c2)cc1
ONC(=O)c1ccc(CN(C2CC2)S(=O)(=O)c2c(F)cc(F)cc2F)cc1
ONC(=O)c1cccc(CN(C2CC2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)c1
ONC(=O)c1ccc(CN(C2CC2)S(=O)(=O)c2c(F)c(Cl)c(F)c(Cl)c2F)cc1
ONC(=O)c1ccc(CN(C2CC2)S(=O)(=O)c2c(F)cc(F)c(Cl)c2F)cc1
ONC(=O)c1ccc(CN(C2CC2)S(=O)(=O)c2c(F)c(F)c(Cl)c(F)c2F)cc1
ONC(=O)c1ccc(CN(C2CC2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
ONC(=O)CCCCCCn1cc(C(=O)NC23CC4CC(CC(C4)C2)C3)c2ccccc12 |TLB:19:20:17.18.23:24,THB:19:18:24:25.20.21,21:20:17:23.22.24,21:22:17:25.19.20|
ONC(=O)CCCCCCn1cc(C(=O)NC2C3CC4CC(C3)CC2C4)c2ccccc12 |TLB:15:16:18:22.20.21,THB:20:19:16:22.21.23,20:21:18.19.25:16,23:21:18:25.24.16,23:24:18:22.20.21,(6.06,-7.06,;5.65,-5.57,;4.16,-5.17,;3.06,-6.27,;3.76,-3.68,;2.27,-3.28,;1.87,-1.79,;.37,-1.38,;-.02,.11,;-1.52,.51,;-1.92,2,;-1,3.25,;-1.88,4.48,;-1.48,5.97,;-2.57,7.06,;.01,6.37,;1.11,5.27,;1.12,4.23,;.28,3.34,;1.32,3.63,;2.31,3.24,;3.02,4.14,;2.04,3.89,;3.03,5.2,;2.05,5.61,;1.31,4.75,;-3.38,4.01,;-4.72,4.78,;-6.06,4.01,;-6.06,2.45,;-4.72,1.69,;-3.38,2.46,)|
ONC(=O)CCCCCCn1cc(C(=O)NCc2ccc(Cl)cc2)c2ccccc12
ONC(=O)CCCCCCn1cc(C(=O)Nc2ccc(Cl)cc2Cl)c2ccccc12
ONC(=O)CCCCCCn1cc(C(=O)N2CCOCC2)c2ccccc12
ONC(=O)CCCCCCn1cc(C(=O)NC2CCCCC2)c2ccccc12
ONC(=O)CCCCCCn1cc(C(=O)NC2CCCCCC2)c2ccccc12
ONC(=O)CCCCCCn1cc(C(=O)NC2CCCCCCC2)c2ccccc12
ONC(=O)CCCCn1cc(C(=O)NC2C3CC4CC(C3)CC2C4)c2ccccc12 |TLB:13:14:16.23.17:21.19.20,23:22:20:16.17.18,THB:13:14:20:16.17.18,23:17:14.22.21:20,18:17:14:21.19.20,18:19:14:16.23.17,(5.03,-6.59,;4.55,-5.13,;3.05,-4.81,;2.02,-5.96,;2.57,-3.34,;1.06,-3.03,;.58,-1.56,;-.93,-1.25,;-1.4,.22,;-.5,1.47,;-1.4,2.71,;-.93,4.17,;-1.96,5.32,;.58,4.49,;1.61,3.35,;2.8,4.63,;4.13,4.14,;5.53,4.48,;5.54,6.01,;4.14,6.59,;2.8,6.11,;3.1,5.35,;3.11,3.77,;4.51,3.2,;-2.87,2.24,;-4.21,3,;-5.54,2.23,;-5.54,.68,;-4.21,-.09,;-2.87,.69,)|
ONC(=O)CCCCCn1cc(C(=O)NC2C3CC4CC(C3)CC2C4)c2ccccc12 |TLB:14:15:17.24.18:22.20.21,24:23:21:17.18.19,THB:14:15:21:17.18.19,24:18:15.23.22:21,19:18:15:22.20.21,19:20:15:17.24.18,(6.04,-6.75,;4.53,-6.43,;4.05,-4.97,;5.08,-3.82,;2.55,-4.65,;2.07,-3.19,;.56,-2.87,;.08,-1.41,;-1.43,-1.09,;-1.9,.37,;-1,1.63,;-1.9,2.87,;-1.43,4.33,;-2.46,5.48,;.08,4.65,;1.11,3.51,;2.3,4.78,;3.62,4.29,;5.03,4.64,;5.04,6.17,;3.64,6.75,;2.3,6.27,;2.6,5.51,;2.61,3.93,;4.01,3.36,;-3.37,2.39,;-4.71,3.16,;-6.04,2.39,;-6.04,.84,;-4.71,.07,;-3.37,.85,)|
ONC(=O)c1ccc(Cn2cc(C(=O)NC3C4CC5CC(C4)CC3C5)c3ccccc23)cc1 |TLB:14:15:17.24.18:22.20.21,24:23:21:17.18.19,THB:14:15:21:17.18.19,24:18:15.23.22:21,19:18:15:22.20.21,19:20:15:17.24.18,(6.31,-5.44,;4.8,-5.13,;4.32,-3.66,;5.35,-2.51,;2.82,-3.35,;1.78,-4.5,;.28,-4.18,;-.19,-2.72,;-1.7,-2.4,;-2.18,-.93,;-1.27,.31,;-2.18,1.56,;-1.7,3.02,;-2.73,4.17,;-.19,3.34,;.83,2.2,;2.03,3.48,;3.35,2.98,;4.76,3.33,;4.77,4.86,;3.37,5.44,;2.02,4.96,;2.32,4.2,;2.33,2.62,;3.74,2.06,;-3.65,1.08,;-4.98,1.84,;-6.31,1.08,;-6.31,-.47,;-4.98,-1.24,;-3.65,-.46,;.82,-1.57,;2.33,-1.88,)|
ONC(=O)\C=C\c1ccc(Cn2cc(C(=O)NC3C4CC5CC(C4)CC3C5)c3ccccc23)cc1 |TLB:16:17:19.26.20:24.22.23,26:25:23:19.20.21,THB:16:17:23:19.20.21,26:20:17.25.24:23,21:20:17:24.22.23,21:22:17:19.26.20,(7.57,-3.88,;6.07,-3.56,;5.05,-4.71,;5.53,-6.16,;3.55,-4.4,;3.07,-2.94,;1.56,-2.63,;.53,-3.78,;-.98,-3.45,;-1.45,-2,;-2.95,-1.67,;-3.44,-.21,;-2.53,1.04,;-3.44,2.28,;-2.96,3.74,;-3.99,4.89,;-1.45,4.06,;-.42,2.92,;.77,4.2,;2.1,3.71,;3.5,4.05,;3.51,5.58,;2.11,6.16,;.77,5.68,;1.06,4.93,;1.08,3.34,;2.48,2.78,;-4.91,1.81,;-6.24,2.57,;-7.57,1.8,;-7.57,.26,;-6.23,-.52,;-4.91,.26,;-.44,-.85,;1.07,-1.16,)|
ONC(=O)CCCCCCn1c(cc2ccccc12)C(=O)NC1C2CC3CC(C2)CC1C3 |TLB:31:30:28:24.25.26,21:22:24.31.25:29.27.28,THB:31:25:22.30.29:28,26:25:22:29.27.28,26:27:22:24.31.25,21:22:28:24.25.26,(5.94,-5.95,;5.54,-4.46,;4.04,-4.06,;2.94,-5.16,;3.64,-2.57,;2.15,-2.17,;1.75,-.67,;.25,-.27,;-.15,1.22,;-1.64,1.62,;-2.05,3.12,;-1.12,4.38,;-2,5.6,;-3.51,5.13,;-4.84,5.91,;-6.19,5.13,;-6.19,3.57,;-4.85,2.81,;-3.51,3.58,;.39,4.36,;1.16,5.66,;1.13,3.04,;2.65,3.03,;3.73,4.18,;4.93,3.74,;6.18,4.06,;6.19,5.43,;4.94,5.95,;3.72,5.52,;3.99,4.84,;4,3.41,;5.26,2.9,)|
ONC(=O)CCCCCCn1c(cc2cc(Cl)ccc12)C(=O)NC1C2CC3CC(C2)CC1C3 |TLB:32:31:29:25.26.27,22:23:25.32.26:30.28.29,THB:32:26:23.31.30:29,27:26:23:30.28.29,27:28:23:25.32.26,22:23:29:25.26.27,(6.58,-5.95,;6.18,-4.46,;4.68,-4.06,;3.58,-5.16,;4.28,-2.57,;2.79,-2.17,;2.39,-.67,;.89,-.27,;.49,1.22,;-1,1.62,;-1.41,3.12,;-.48,4.37,;-1.36,5.6,;-2.87,5.13,;-4.2,5.91,;-5.55,5.13,;-6.83,5.87,;-5.55,3.57,;-4.2,2.81,;-2.87,3.58,;1.03,4.36,;1.8,5.66,;1.78,3.04,;3.29,3.03,;4.37,4.18,;5.57,3.74,;6.82,4.05,;6.83,5.43,;5.58,5.95,;4.36,5.52,;4.63,4.83,;4.64,3.41,;5.9,2.9,)|
COc1ccc2n(CCCCCCC(=O)NO)c(cc2c1)C(=O)NC1C2CC3CC(C2)CC1C3 |TLB:33:32:30:26.27.28,23:24:26.33.27:31.29.30,THB:33:27:24.32.31:30,28:27:24:31.29.30,28:29:24:26.33.27,23:24:30:26.27.28,(-6.83,6.65,;-6.83,5.17,;-5.55,4.43,;-5.55,2.87,;-4.2,2.11,;-2.87,2.88,;-1.41,2.42,;-1,.92,;.49,.52,;.89,-.97,;2.39,-1.37,;2.79,-2.87,;4.28,-3.27,;4.68,-4.76,;3.58,-5.86,;6.18,-5.16,;6.58,-6.65,;-.48,3.67,;-1.36,4.9,;-2.87,4.43,;-4.2,5.2,;1.03,3.66,;1.8,4.96,;1.78,2.34,;3.29,2.33,;4.37,3.48,;5.57,3.04,;6.82,3.35,;6.83,4.73,;5.58,5.25,;4.36,4.82,;4.64,4.13,;4.64,2.71,;5.91,2.2,)|
ONC(=O)CCCCCCn1c(cc2ccc(Br)cc12)C(=O)NC1C2CC3CC(C2)CC1C3 |TLB:32:31:29:25.26.27,22:23:25.32.26:30.28.29,THB:32:26:23.31.30:29,27:26:23:30.28.29,27:28:23:25.32.26,22:23:29:25.26.27,(6.58,-5.95,;6.18,-4.46,;4.68,-4.06,;3.58,-5.16,;4.28,-2.57,;2.79,-2.17,;2.39,-.67,;.89,-.27,;.49,1.22,;-1,1.62,;-1.41,3.12,;-.48,4.38,;-1.36,5.6,;-2.87,5.13,;-4.2,5.91,;-5.55,5.13,;-5.55,3.57,;-6.83,2.82,;-4.21,2.81,;-2.87,3.58,;1.03,4.36,;1.8,5.66,;1.77,3.04,;3.29,3.03,;4.37,4.18,;5.56,3.74,;6.82,4.05,;6.83,5.43,;5.58,5.95,;4.36,5.52,;4.63,4.83,;4.64,3.41,;5.9,2.9,)|
ONC(=O)CCCCCCn1c(nc2ccccc12)C(=O)NC1C2CC3CC(C2)CC1C3 |TLB:31:30:28:24.25.26,21:22:24.31.25:29.27.28,THB:31:25:22.30.29:28,26:25:22:29.27.28,26:27:22:24.31.25,21:22:28:24.25.26,(5.94,-5.95,;5.54,-4.46,;4.04,-4.06,;2.94,-5.16,;3.64,-2.57,;2.15,-2.17,;1.75,-.67,;.25,-.27,;-.15,1.22,;-1.64,1.62,;-2.05,3.12,;-1.12,4.38,;-2,5.6,;-3.51,5.13,;-4.84,5.91,;-6.19,5.13,;-6.19,3.57,;-4.85,2.81,;-3.51,3.58,;.39,4.36,;1.16,5.66,;1.13,3.04,;2.65,3.03,;3.73,4.18,;4.92,3.74,;6.18,4.05,;6.19,5.43,;4.93,5.95,;3.72,5.52,;3.99,4.84,;4,3.41,;5.26,2.9,)|
ONC(=O)CCCCCCn1nc(C(=O)NC2C3CC4CC(C3)CC2C4)c2ccccc12 |TLB:25:24:22:18.19.20,15:16:22:18.19.20,THB:25:19:16.24.23:22,20:19:16:23.21.22,20:21:16:18.25.19,15:16:18.25.19:23.21.22,(6.06,-8.79,;5.66,-7.3,;4.16,-6.9,;3.07,-8,;3.76,-5.41,;2.27,-5.01,;1.87,-3.51,;.37,-3.11,;-.03,-1.62,;-1.52,-1.22,;-1.92,.28,;-.99,1.53,;-1.88,2.76,;-1.41,4.17,;-2.39,5.28,;.05,4.46,;.52,5.87,;1.59,7.02,;2.79,6.58,;4.05,6.89,;4.06,8.27,;2.8,8.79,;1.59,8.36,;1.86,7.67,;1.87,6.25,;3.13,5.74,;-3.38,2.29,;-4.72,3.06,;-6.06,2.29,;-6.06,.73,;-4.72,-.03,;-3.38,.74,)|
CC(=O)SCCCCCCn1cc(C(=O)NC2C3CC4CC(C3)CC2C4)c2ccccc12 |TLB:25:24:22:18.19.20,15:16:22:18.19.20,THB:25:19:16.24.23:22,20:19:16:23.21.22,20:21:16:18.25.19,15:16:18.25.19:23.21.22,(5.74,-8.79,;5.34,-7.3,;6.39,-6.25,;3.84,-6.9,;3.44,-5.41,;1.95,-5.01,;1.55,-3.51,;.05,-3.11,;-.35,-1.62,;-1.84,-1.22,;-2.25,.28,;-1.32,1.53,;-2.2,2.76,;-1.73,4.17,;-2.72,5.28,;-.28,4.46,;.19,5.87,;1.27,7.02,;2.47,6.59,;3.72,6.9,;3.73,8.27,;2.48,8.79,;1.26,8.36,;1.54,7.68,;1.54,6.26,;2.81,5.74,;-3.71,2.29,;-5.04,3.06,;-6.39,2.29,;-6.39,.73,;-5.05,-.03,;-3.71,.74,)|
CC(=O)SCCCCCCCn1cc(C(=O)NC2C3CC4CC(C3)CC2C4)c2ccccc12 |TLB:26:25:23:19.20.21,16:17:23:19.20.21,THB:26:20:17.25.24:23,21:20:17:24.22.23,21:22:17:19.26.20,16:17:19.26.20:24.22.23,(6.81,-8.69,;5.37,-8.31,;4.32,-9.36,;4.97,-6.81,;3.46,-6.41,;3.06,-4.91,;1.56,-4.51,;1.16,-3,;-.34,-2.6,;-.75,-1.1,;-2.24,-.7,;-2.65,.81,;-1.72,2.07,;-2.61,3.3,;-2.13,4.71,;-3.12,5.83,;-.67,5.01,;-.2,6.43,;.88,7.58,;2.09,7.14,;3.35,7.46,;3.36,8.84,;2.1,9.36,;.87,8.93,;1.15,8.24,;1.15,6.81,;2.43,6.29,;-4.12,2.83,;-5.46,3.61,;-6.81,2.82,;-6.81,1.26,;-5.46,.5,;-4.12,1.27,)|
SCCCCCCn1cc(C(=O)NC2C3CC4CC(C3)CC2C4)c2ccccc12 |TLB:22:21:19:15.16.17,12:13:19:15.16.17,THB:22:16:13.21.20:19,17:16:13:20.18.19,17:18:13:15.16.22,12:13:15.16.22:20.18.19,(5.2,-7.97,;4.81,-6.51,;3.29,-6.1,;2.88,-4.57,;1.36,-4.16,;.95,-2.64,;-.57,-2.24,;-.98,-.71,;-.04,.57,;-.94,1.82,;-.46,3.25,;-1.46,4.39,;1.02,3.56,;1.5,4.99,;2.6,6.16,;3.82,5.72,;5.1,6.03,;5.11,7.44,;3.83,7.97,;2.59,7.53,;2.87,6.83,;2.88,5.38,;4.17,4.86,;-2.47,1.34,;-3.83,2.13,;-5.2,1.34,;-5.2,-.25,;-3.83,-1.02,;-2.47,-.24,)|
SCCCCCCCn1cc(C(=O)NC2C3CC4CC(C3)CC2C4)c2ccccc12 |TLB:23:22:20:16.17.18,13:14:20:16.17.18,THB:23:17:14.22.21:20,18:17:14:21.19.20,18:19:14:16.17.23,13:14:16.17.23:21.19.20,(5.93,-8.16,;4.47,-7.77,;4.08,-6.31,;2.56,-5.9,;2.15,-4.38,;.63,-3.97,;.22,-2.45,;-1.3,-2.04,;-1.71,-.51,;-.77,.77,;-1.67,2.02,;-1.19,3.45,;-2.19,4.58,;.29,3.75,;.77,5.19,;1.87,6.36,;3.09,5.91,;4.37,6.23,;4.38,7.63,;3.1,8.16,;1.86,7.72,;2.14,7.03,;2.15,5.58,;3.44,5.05,;-3.2,1.53,;-4.56,2.32,;-5.93,1.53,;-5.93,-.05,;-4.56,-.83,;-3.2,-.04,)|
ONC(=O)c1ccc(CNCc2ccccc2)cc1
ONC(=O)c1ccc(CNCc2cccs2)cc1
c1cc(ccc1CNCc2ccsc2)C(=O)NO
CN1CCN(CC1)Cc2ccc(cc2)C(=O)NO
c1ccc(cc1)CCN2CCC(CC2)/C=C/C(=O)NO
c1ccc2c(c1)c(c[nH]2)CCN3CCC(CC3)/C=C/C(=O)NO
ONC(=O)\C=C\C1CCN(Cc2cccc3ccccc23)CC1
ONC(=O)\C=C\C1CCN(Cc2csc3ccccc23)CC1
Cn1cc(CN2CCC(CC2)\C=C\C(=O)NO)c2ccccc12
ONC(=O)\C=C\C1CCN(Cc2ccc(Cl)cc2)CC1
CC(C)n1cnc2c(nc(nc12)N1CCOCC1)-c1cccc(OCCCC(=O)NO)c1
ONC(=O)CCCCCCC(=O)Nc1nc2CC[C@@H](Cc2s1)NC(=O)c1cccc2ccccc12 |r|
C[C@@H]1CN(Cc2ccc(cc2)C(=O)NO)C[C@H]1c1nc2n(ncc2c(=O)[nH]1)C1CCCC1 |r|
C[C@H]1CN(Cc2ccc(cc2)C(=O)NO)C[C@@H](C)N1Cc1cccc(Cl)c1 |r|
COc1ccc(CNC(=O)c2cc(F)ccc2N2CCOCC2)cc1OCC(=O)NO
COc1ccc(CNC(=O)c2cc(F)ccc2N2CCOCC2)cc1\C=C\C(=O)NO
COc1ccc(CNC(=O)c2cc(ccc2N2CCOCC2)C(=O)Nc2ccccc2N)cc1O
COc1cc2nc(NCCCCCC(=O)NO)nc(NC3CCN(C)CC3)c2cc1OC
COc1cc2nc(NCCCCCCC(=O)NO)nc(NC3CCN(C)CC3)c2cc1OC
COc1cc2nc(NCCCCCC(=O)NO)nc(NC3CCN(CC3)C(C)C)c2cc1OC
COc1cc2nc(NCCCCCCC(=O)NO)nc(NC3CCN(CC3)C(C)C)c2cc1OC
COc1cc2nc(nc(NC3CCN(CC3)C(C)C)c2cc1OC)N1CCN(CCCCCC(=O)NO)CC1
COc1cc2nc(NCCCCCC(=O)NO)nc(NC3CCN(Cc4ccccc4)CC3)c2cc1OC
COc1cc2nc(nc(NC3CCN(Cc4ccccc4)CC3)c2cc1OC)N1CCN(CCCCCC(=O)NO)CC1
COc1cc2nc(nc(NC3CCN(Cc4ccccc4)CC3)c2cc1OC)N1CCN(Cc2ccc(\C=C\C(=O)NO)cc2)CC1
Cc1c(COc2ccc(CNCCC(=O)NO)c(F)c2)cccc1-c1ccccc1
CN(CCCC(=O)NO)Cc1ccc(OCc2cccc(c2C)-c2ccccc2)cc1F
CN(CCCCC(=O)NO)Cc1ccc(OCc2cccc(c2C)-c2ccccc2)cc1F
Cc1c(COc2ccc(CNCCCCCC(=O)NO)c(F)c2)cccc1-c1ccccc1
Cc1c(COc2ccc(CNCCCCCCC(=O)NO)c(F)c2)cccc1-c1ccccc1
COc1cc(OCc2cccc(c2C)-c2ccccc2)cc(OC)c1CNCCC(=O)NO
COc1cc(OCc2cccc(c2C)-c2ccccc2)cc(OC)c1CN(C)CCCC(=O)NO
COc1cc(OCc2cccc(c2C)-c2ccccc2)cc(OC)c1CN(C)CCCCC(=O)NO
COc1cc(OCc2cccc(c2C)-c2ccccc2)cc(OC)c1CNCCCCCC(=O)NO
COc1cc(OCc2cccc(c2C)-c2ccccc2)cc(OC)c1CNCCCCCCC(=O)NO
Cc1c(COc2ccc(CNCCC(=O)NO)c(OCc3cccc(c3)C#N)c2)cccc1-c1ccccc1
CN(CCCC(=O)NO)Cc1ccc(OCc2cccc(c2C)-c2ccccc2)cc1OCc1cccc(c1)C#N
CN(CCCCC(=O)NO)Cc1ccc(OCc2cccc(c2C)-c2ccccc2)cc1OCc1cccc(c1)C#N
Cc1c(COc2ccc(CNCCCCCC(=O)NO)c(OCc3cccc(c3)C#N)c2)cccc1-c1ccccc1
Cc1c(COc2ccc(CNCCCCCCC(=O)NO)c(OCc3cccc(c3)C#N)c2)cccc1-c1ccccc1
Cc1c(COc2ccc(CNCCCCCC(=O)NO)c(F)c2)cccc1-c1ccc2OCCOc2c1
Cc1c(COc2ccc(CNCCCCCCC(=O)NO)c(F)c2)cccc1-c1ccc2OCCOc2c1
COc1cc(OCc2cccc(c2C)-c2ccc3OCCOc3c2)cc(OC)c1CNCCCCCC(=O)NO
COC1C=C(OCc2cccc(c2C)-c2ccc3OCCOc3c2)C=C(OC)C1CNCCCCCCC(=O)NO |t:3,27|
ONC(=O)CCCCc1nnc(o1)-c1cc2c3ccccc3[nH]c2c(n1)-c1ccc(cc1)C(F)(F)F
COc1cc(cc(OC)c1OC)-c1nc(cc2c3ccccc3[nH]c12)-c1nnc(CCCCC(=O)NO)o1
CCN(CC)c1ccc(cc1)C(=O)NCCCCCCC(=O)NO
CC12CC3CC(C)(C1)CC(C3)(C2)NC(=O)\C=C\c1ccc(cc1)C(=O)NO |TLB:4:5:11:2.3.10,4:3:11:8.5.7,0:1:8:3.10.4,THB:2:1:8:3.10.4,2:3:8:11.7.1,6:5:11:2.3.10|
COc1ccc(Cn2ccc3cc(ccc23)C(=O)NO)cc1
CCCNNC(=O)c1ccc(cc1)-c1ccc(CNC(C)=O)cc1
CCCCCCNNC(=O)c1ccc(cc1)-c1ccc(CNC(C)=O)cc1
CCCCCCNNC(=O)c1cccc(NCc2ccccc2)c1
CCCNNC(=O)c1cnc(NCc2ccccc2)nc1
CCCNNC(=O)c1cnc(nc1)N1CCN(Cc2c[nH]c3ccccc23)CC1
CCCCCCNNC(=O)c1cnc(nc1)N1CCN(Cc2c[nH]c3ccccc23)CC1
COc1cc(OC)cc(c1)N(CCCCC(=O)NO)c1ccc2ncc(nc2c1)-c1cnn(C)c1
COc1cc(OC)cc(c1)N(CCCCCC(=O)NO)c1ccc2ncc(nc2c1)-c1cnn(C)c1
COc1cc(OC)cc(c1)N(CCCCCCC(=O)NO)c1ccc2ncc(nc2c1)-c1cnn(C)c1
COc1cc(OC)cc(c1)N(CCNC(C)C)c1ccc2ncc(nc2c1)-c1cnn(CCCCCCC(=O)NO)c1
COc1cc(OC)cc(c1)N(CCNC(C)C)c1ccc2ncc(nc2c1)-c1cnn(CCOc2ccc(cc2)C(=O)NO)c1
ONC(=O)CCCCCCNC(=O)c1ccc(NC(=O)COCCNC(=O)COc2cccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c23)cc1
ONC(=O)CCCCCCNC(=O)c1ccc(NC(=O)COCCOCCNC(=O)COc2cccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c23)cc1
ONC(=O)CCCCCCNC(=O)c1ccc(NC(=O)CCOCCOCCOCCNC(=O)COc2cccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c23)cc1
ONC(=O)CCCCCCNC(=O)c1ccc(NC(=O)CCOCCOCCOCCOCCNC(=O)COc2cccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c23)cc1
ONC(=O)CCCCCCNC(=O)c1ccc(NC(=O)CCOCCOCCOCCOCCNC(=O)CNc2cccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c23)cc1
ONC(=O)CCCCCCNC(=O)c1ccc(NC(=O)CCCCCCCNC(=O)COc2cccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c23)cc1
Cc1nc2cc(NC(=O)CCOCCOCCOCCNC(=O)COc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)ccc2n1Cc1ccc(cc1F)C(=O)NO
Cc1nc2cc(NC(=O)CCOCCOCCOCCOCCNC(=O)COc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)ccc2n1Cc1ccc(cc1F)C(=O)NO
Cc1nc2cc(NC(=O)CCOCCOCCOCCOCCNC(=O)CNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)ccc2n1Cc1ccc(cc1F)C(=O)NO
Cc1nc2cc(NC(=O)CCCCCCCNC(=O)COc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)ccc2n1Cc1ccc(cc1F)C(=O)NO
COc1cc(OC)cc(\C=C\c2ccc(OCCCCCCC(=O)NO)cc2)c1
CC(C)(CNC(=O)c1cccc(c1)-c1noc(n1)C(F)(F)F)c1coc(n1)-c1ccccc1
CN(CCCOc1ccc(NC(=O)CCCCCCC(=O)NO)cc1Cl)CC#C
CN(CCCOc1cccc(NC(=O)CCCCCCC(=O)NO)c1Cl)CC#C
CN(CCCOc1cc(NC(=O)CCCCCCC(=O)NO)ccc1Cl)CC#C
CN(CCCOc1cc(NC(=O)CCCCCCC(=O)NO)c(Cl)cc1Cl)CC#C
CN(CCCOc1cc(NC(=O)CCCCCCCCC(=O)NO)ccc1Cl)CC#C
CN(CCCOc1cc(NC(=O)CCCCCCCC(=O)NO)ccc1Cl)CC#C
CN(CCCOc1cc(NCc2ccc(\C=C\C(=O)NO)cc2)ccc1Cl)CC#C
CN(CCCOc1cc(NCc2ccc(cc2)C(=O)NO)ccc1Cl)CC#C
ONC(=O)c1cnc(nc1)N1CCC(CC1)NC(=O)c1cnc(nc1O)-n1cccn1
CNc1nc(Cl)nc2n(Cc3ccc(cc3)C(=O)Nc3ccccc3N)cnc12
CCNc1nc(Cl)nc2n(Cc3ccc(cc3)C(=O)Nc3ccccc3N)cnc12
CCCNc1nc(Cl)nc2n(Cc3ccc(cc3)C(=O)Nc3ccccc3N)cnc12
CCCCNc1nc(Cl)nc2n(Cc3ccc(cc3)C(=O)Nc3ccccc3N)cnc12
CC(C)N(Cc1ccc(cc1)C(=O)NO)S(=O)(=O)c2cc(c(c(c2F)F)F)F
CC(C)N(Cc1ccc(cc1)C(=O)NO)Cc1cc(F)c(F)c(F)c1F
CC(C)CN(Cc1ccc(cc1)C(=O)NO)S(=O)(=O)c1cc(F)c(F)c(F)c1F
COCCN(Cc1ccc(cc1)C(=O)NO)S(=O)(=O)c1cc(F)c(F)c(F)c1F
ONC(=O)c1ccc(CN(C2CCCC2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
ONC(=O)c1ccc2CN(CCc2c1)S(=O)(=O)c1cc(F)c(F)c(F)c1F
CC(C)N(Cc1ccc(cn1)C(=O)NO)S(=O)(=O)c1cc(F)c(F)c(F)c1F
CC(C)N(Cc1ccc(CC(=O)NO)cc1)S(=O)(=O)c1cc(F)c(F)c(F)c1F
COc1cc(ccc1CN(C(C)C)S(=O)(=O)c1cc(F)c(F)c(F)c1F)C(=O)NO
Nc1nc(-c2ccco2)c2cnn(CCc3ccc(cc3)C(=O)Nc3ccccc3N)c2n1
Nc1nc(-c2ccco2)c2cnn(Cc3cccc(OCCCCCCC(=O)NO)c3)c2n1
CN(C)c1nc2c(Br)c(Br)c(Br)c(Br)c2n1CCCCCC(=O)NO
CN(C)c1nc2c(Br)c(Br)c(Br)c(Br)c2n1CCCCCCCC(=O)NO
CC(C)n1c(C)nc2c(F)cc(cc12)-c1nc(Nc2ccc(CNC(=O)CC(=O)NO)cc2)ncc1F
CN(CCOc1no[n+]([O-])c1S(=O)(=O)c1ccccc1)C(=O)c1ccc(\C=C\C(=O)NO)cc1
C[C@H]1COc2c(N3CCN(C)CC3)c(F)cc3c2n1cc(C(=O)OCc1cn(CCCCCC(=O)NO)nn1)c3=O |r|
C[C@H]1COc2c(N3CCN(C)CC3)c(F)cc3c2n1cc(C(=O)OCc1cn(CCCCCCC(=O)NO)nn1)c3=O |r|
C[C@H]1COc2c(N3CCN(C)CC3)c(F)cc3c2n1cc(C(=O)OCc1cn(CCCCCCCC(=O)NO)nn1)c3=O |r|
C[C@H]1COc2c(N3CCN(C)CC3)c(F)cc3c2n1cc(C(=O)NCc1cn(CCCCCC(=O)NO)nn1)c3=O |r|
C[C@H]1COc2c(N3CCN(C)CC3)c(F)cc3c2n1cc(C(=O)NCc1cn(CCCCCCC(=O)NO)nn1)c3=O |r|
C[C@H]1COc2c(N3CCN(C)CC3)c(F)cc3c2n1cc(C(=O)NCc1cn(CCCCCCCC(=O)NO)nn1)c3=O |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccccc2[nH]c1=O |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccccc2n(C)c1=O |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cn(C)c2ccccc2c1=O |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cnc2ccccc2c1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2ncccc2c1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2ccc3cnccc3c2)CC1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2ccc3ccncc3c2)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nccnc2c1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nnccc2c1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cnc2ncccc2c1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)C1=CC2SC=NC2C=C1 |r,c:34,38,t:30|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)C1=CC2OC=NC2C=C1 |r,c:34,38,t:30|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nn(C)cc2c1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2n(C)c(=O)ccc2c1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2ccc([nH]c2=O)-c2ccccc2)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc(cc1)-c1ccncc1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc(cc1)-c1cccnc1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc(cc1)-c1cnccn1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nc(C)ccc2c1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nc(CC)ccc2c1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nc(ccc2c1)C1CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nc(OC)ccc2c1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nc(ccc2c1)N1CCCC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nc(ccc2c1)-c1ncco1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1ccc2nc(ccc2c1)-n1cccn1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2cccnc2cc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccc(C)nc2cc1OC |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2cc3ccc(C)nc3cc2OC)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC1)C(C)C)c1ncc([nH]1)-c1cc2ccc(C)nc2cc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC2CC2)CC1)c1ncc([nH]1)-c1cc2ccc(C)nc2cc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC1)C1CCC1)c1ncc([nH]1)-c1cc2ccc(C)nc2cc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC2CC2)CC1)c1ncc([nH]1)-c1cc2ccc(CC)nc2cc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(CC2CC2)CC1)c1ncc([nH]1)-c1cc2ccc(nc2cc1OC)C1CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccc(nc2cc1OC)C1CC1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2cc3ccc(=O)n(C)c3cc2OC)CC1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2cc3cn(C)nc3cc2OC)CC1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc([nH]2)-c2cc3nccnc3cc2OC)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccncc2nc1OC |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccc(C)nc2cc1F |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccc(C)nc2cc1Cl |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccc(C)nc2cc1C |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc([nH]1)-c1cc2ccc(C)nc2cc1CC |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc(o2)-c2cc3ccncc3nc2OC)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc(o1)-c1cc2ccc(C)nc2cc1OC |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc(o2)-c2cc3ccc(C)nc3cc2OC)CC1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc(o2)-c2cc3ccc(=O)n(C)c3cc2OC)CC1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc(o2)-c2cc3cccnc3nc2OC)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc(o1)-c1cc2ccc(C)nc2cc1F |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc(o1)-c1cc2ccc(nc2cc1F)C1CC1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc(o2)-c2cc3cn(C)nc3cc2OC)CC1 |r|
CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC11CCN(C)CC1)c1ncc(o1)-c1ccc(cc1)-c1cccnc1 |r|
CCN1CCC2(C[C@@H]2C(=O)N[C@@H](CCCCCC(=O)CC)c2ncc(o2)-c2cc3ccn(CC)c(=O)c3cc2OC)CC1 |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(F)c2c(=O)n1CCCCCC(=O)NO |r|
CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(F)c2c(=O)n1Cc1ccc(cc1)C(=O)NO |r|
ONC(=O)c1ccc(Cn2c(nc3cccc(F)c3c2=O)[C@@H]2CC3(CC3)CN2c2ncnc3[nH]cnc23)cc1 |r|
Nc1nc(N)c(C#N)c(n1)N1CC2(CC2)C[C@H]1c1nc2cccc(F)c2c(=O)n1Cc1ccc(cc1)C(=O)NO |r|
Nc1nc(N)c(C#N)c(n1)N1CC2(CC2)C[C@H]1c1nc2cccc(F)c2c(=O)n1Cc1ccc(s1)C(=O)NO |r|
Nc1nc(N)c(C#N)c(n1)N1CCC[C@H]1c1nc2cccc(Cl)c2c(=O)n1Cc1ccc(cc1)C(=O)NO |r|
Nc1nc(N)c(C#N)c(n1)N1CC2(CC2)C[C@H]1c1nc2cccc(Cl)c2c(=O)n1Cc1ccc(cc1)C(=O)NO |r|
C[C@H](Nc1nc(N)nc(N)c1C#N)c1nc2cccc(Cl)c2c(=O)n1Cc1ccc(s1)C(=O)NO |r|
CC[C@H](Nc1nc(N)nc(N)c1C#N)c1nc2cccc(Cl)c2c(=O)n1Cc1ccc(s1)C(=O)NO |r|
Nc1nc(N)c(C#N)c(n1)N1CCC[C@H]1c1nc2cccc(Cl)c2c(=O)n1Cc1ccc(s1)C(=O)NO |r|
Nc1nc(N)c(C#N)c(n1)N1CC2(CC2)C[C@H]1c1nc2cccc(Cl)c2c(=O)n1Cc1ccc(s1)C(=O)NO |r|
Nc1nc(N)c(C#N)c(n1)N1CC2(CC2)C[C@H]1c1nc2cccc(Cl)c2c(=O)n1Cc1cc(no1)C(=O)NO |r|
Nc1nc(N)c(C#N)c(n1)N1CCC[C@H]1c1nc(NCc2ccc(cc2)C(=O)NO)c2c(Cl)cccc2n1 |r|
Nc1nc(N)c(C#N)c(n1)N1CC2(CC2)C[C@H]1c1nc(NCc2ccc(cc2)C(=O)NO)c2c(Cl)cccc2n1 |r|
Nc1nc(N)c(C#N)c(n1)N1CC2(CC2)C[C@H]1c1nc(NCCc2ccc(cc2)C(=O)NO)c2c(Cl)cccc2n1 |r|
Nc1nc(N)c(C#N)c(n1)N1C[C@@H](C[C@H]1c1nc2cccc(Cl)c2c(=O)n1-c1ccccc1)OC(=O)NCc1ccc(cc1)C(=O)NO |r|
Nc1nc(N)c(C#N)c(n1)N1C[C@H](C[C@H]1c1nc2cccc(Cl)c2c(=O)n1-c1ccccc1)OC(=O)NCc1ccc(cc1)C(=O)NO |r|
Cn1c(nc2cccc(Cl)c2c1=O)[C@@H]1C[C@H](CN1c1nc(N)nc(N)c1C#N)OCc1ccc(cc1)C(=O)NO |r|
Cn1c(nc2cccc(Cl)c2c1=O)[C@@H]1C[C@H](CN1c1nc(N)nc(N)c1C#N)OCc1ccc(s1)C(=O)NO |r|
Cn1c(nc2cccc(Cl)c2c1=O)[C@@H]1C[C@H](CN1c1nc(N)nc(N)c1C#N)OC(=O)NCc1ccc(cc1)C(=O)NO |r|
CN(Cc1ccc(cc1)C(=O)NO)C(=O)O[C@@H]1C[C@H](N(C1)c1nc(N)nc(N)c1C#N)c1nc2cccc(Cl)c2c(=O)n1C |r|
Cn1c(nc2cccc(Cl)c2c1=O)[C@@H]1C[C@H](CN1c1nc(N)nc(N)c1C#N)OC(=O)NCCc1ccc(cc1)C(=O)NO |r|
Cn1c(nc2cccc(Cl)c2c1=O)[C@@H]1C[C@H](CN1c1nc(N)nc(N)c1C#N)OC(=O)NCc1ccc(s1)C(=O)NO |r|
ONC(=O)c1ccc(CN2CC(=O)N[C@@H](Cc3ccccc3)C2=O)cc1 |r|
ONC(=O)c1ccc(CN2CC(=O)N[C@H](Cc3ccccc3)C2=O)cc1 |r|
ONC(=O)c1cccc(CN2CC(=O)N[C@@H](Cc3ccccc3)C2=O)c1 |r|
CN1C(Cc2ccccc2)C(=O)N(Cc2ccc(cc2)C(=O)NO)CC1=O
ONC(=O)c1ccc(CN2CC(=O)N(C=C)C(Cc3ccccc3)C2=O)cc1
ONC(=O)c1ccc(CN2CC(=O)N(C(CCc3ccccc3)C2=O)c2ccccc2)cc1
ONC(=O)c1ccc(CN2CC(=O)N(Cc3ccccc3)[C@H](Cc3ccccc3)C2=O)cc1 |r|
ONC(=O)c1ccc(CN2CC(=O)N(Cc3ccccc3Cl)[C@H](Cc3ccccc3)C2=O)cc1 |r|
ONC(=O)c1ccc(CN2CC(=O)N(Cc3ccc(Cl)cc3)[C@H](Cc3ccccc3)C2=O)cc1 |r|
ONC(=O)c1ccc(CN2CC(=O)N(Cc3cccc(Cl)c3)[C@H](Cc3ccccc3)C2=O)cc1 |r|
COc1cccc(CN2[C@H](Cc3ccccc3)C(=O)N(Cc3ccc(cc3)C(=O)NO)CC2=O)c1 |r|
ONC(=O)c1ccc(CN2CC(=O)N[C@@H](Cc3c[nH]c4ccccc34)C2=O)cc1 |r|
ONC(=O)c1ccc(CN2CC(=O)N[C@H](Cc3c[nH]c4ccccc34)C2=O)cc1 |r|
ONC(=O)c1cn(nn1)C1CCN(CC1)C(=O)Cc1ccc2ccccc2c1
ONC(=O)\C=C\c1cccn(CCCCCCn2cc(nn2)-c2cccc(c2)C#N)c1=O
Cc1[nH]c2ccccc2c1CCNS(=O)(=O)c1ccc(\C=C\C(=O)NO)cc1
ONC(=O)CCCCCC(=O)N(Cc1ccc(Br)s1)c1ccc(OCCN2CCOCC2)cc1
ONC(=O)\C=C\c1ccc(cc1)S(=O)(=O)Nc1cc(F)cc(F)c1
COc1ccc(\C=N\NC(=O)CCCCCCCC(=O)NO)cc1
[H][C@]12Cc3c([nH]c4ccccc34)[C@H](N1C(=O)CN(CC1CCN(CC1)c1ncc(CC(=O)NO)cn1)C2=O)c1ccc2OCOc2c1 |r|
COc1ccccc1NC(=O)N[C@H](C(=O)Nc1ccc(cc1)C(=O)NO)c1ccccc1 |r|
Nc1ccccc1NC(=O)CCCCCCC(=O)NO
ONC(=O)c1ccc(NC(=O)[C@@H](NC(=O)c2ccc3ccccc3c2)c2ccccc2)cc1 |r|
ONC(=O)c1ccc(NC(=O)[C@@H](NS(=O)(=O)c2cccc3ccccc23)c2ccccc2)cc1 |r|
ONC(=O)c1ccc(NC(=O)[C@@H](NC(=O)c2cccc(Br)c2)c2ccccc2)cc1 |r|
CN(C)c1cccc2c(cccc12)S(=O)(=O)N[C@H](C(=O)Nc1ccc(cc1)C(=O)NO)c1ccccc1 |r|
COC(=O)\C=C\c1ccc(OCCNc2cc3c4ccccc4[nH]c3c(n2)-c2ccc(OC)cc2)c(OC)c1
COC(=O)\C=C\c1ccc(OCCCNc2cc3c4ccccc4[nH]c3c(n2)-c2ccc(OC)cc2)c(OC)c1
ONC(=O)\C=C\c1ccc(cc1)N1CC(=O)N2C(Cc3c([nH]c4ccccc34)C2c2ccc3OCOc3c2)C1=O
ONC(=O)CCCN1CCC(CC1)N1CC(=O)N2C(Cc3c([nH]c4ccccc34)C2c2ccc3OCOc3c2)C1=O
ONC(=O)c1cnc(nc1)N1CCC(CN2CC(=O)N3C(Cc4c([nH]c5ccccc45)C3c3ccc4OCOc4c3)C2=O)CC1
ONC(=O)c1ccc(CN2CCN(CC2)C(=O)c2c[nH]c3ccccc23)cc1
ONC(=O)c1ccc(CN2CCN(CC2)C(=O)c2c[nH]c3ccc(Cl)cc23)cc1
Cc1cccc2c(c[nH]c12)C(=O)N1CCN(Cc2ccc(cc2)C(=O)NO)CC1
ONC(=O)c1ccc(CN2CCN(CC2)C(=O)c2c[nH]c3cc(OCc4ccccc4)ccc23)cc1
Cn1cc(C(=O)N2CCN(Cc3ccc(cc3)C(=O)NO)CC2)c2ccccc12
ONC(=O)c1ccc(CN2CCN(CC2)C(=O)c2c[nH]c3cccc(Cc4ccccc4)c23)cc1
ONC(=O)c1ccc(CN2CCN(CC2)C(=O)c2c[nH]c3cc(F)ccc23)cc1
ONC(=O)c1ccc(CN2CCN(CC2)C(=O)c2cc3ccccc3[nH]2)cc1
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)Nc1ccc(cc1)C(=O)NO)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
CN(C)c1ccc(cc1)-c1nc(cc2c3ccccc3[nH]c12)C(=O)NCc1ccc(\C=C\C(=O)NO)cc1
CCC(=O)CCCCC[C@H](NC(=O)C1CN(C)C1)c1ncc(o1)-c1cc2ccccc2nc1OC |r|
CNC(=O)CCCCC[C@H](NC(=O)Cn1ccc2cc(ccc12)C#N)c1ncc([nH]1)-c1ccc(CN(C)C)cc1 |r|
COc1ccc(\C=C2/SC(=O)N(CCNC(=O)Nc3c(C)n(C)n(-c4ccccc4)c3=O)C2=O)cc1
Cc1c(NC(=O)NCCN2C(=O)S\C(=C/c3ccc(cc3)[N+]([O-])=O)C2=O)c(=O)n(-c2ccccc2)n1C
COc1cc(\C=C2/SC(=O)N(CCNC(=O)Nc3c(C)n(C)n(-c4ccccc4)c3=O)C2=O)cc(OC)c1OC
Cc1c(NC(=O)CN2C(=O)S\C(=C/c3ccc(Br)cc3)C2=O)c(=O)n(-c2ccccc2)n1C
COc1ccc(NC(=O)CCCCCCNC(=O)C(O)(O)C(F)(F)F)cc1
OC(O)(C(=O)NCCCCCCC(=O)Nc1ncc(s1)-c1ccccc1)C(F)(F)F
OC(O)(C(=O)NCCCCCCC(=O)Nc1nc2ccccc2s1)C(F)(F)F
COc1ccc2sc(NC(=O)CCCCCCNC(=O)C(O)(O)C(F)(F)F)nc2c1
Oc1ccc(cc1)-c1cnc(NC(=O)CCCCCCNC(=O)C(O)(O)C(F)(F)F)s1
OC(O)(C(=O)NCCCCCCC(=O)Nc1ccc(Cl)cc1)C(F)(F)F
OC(O)(C(=O)NCCCCCCC(=O)Nc1ccc(Br)cc1)C(F)(F)F
OC(O)(C(=O)NCCCCCCC(=O)Nc1ccc(cc1)-c1ccccc1)C(F)(F)F
COc1ccc(cc1)-c1cnc(NC(=O)CCCCCCNC(=O)C(O)(O)C(F)(F)F)s1
OC(O)(C(=O)NCCCCCCC(=O)Nc1ncc(s1)-c1ccc(Br)cc1)C(F)(F)F
COc1ccc(CC2C=Cc3cc(ccc23)C(=O)NO)cc1 |c:8|
CN(C)c1cccc2c(SNCCCCCC(=O)NO)cccc12
CC(C)Cc1c(OCCOc2cccc(\C=C\C(=O)NO)c2)ccc2CCC(=O)Oc12
COc1cc2c(Nc3cccc(\C=C\C(=O)NO)c3)ncnc2cc1OCCCN1CCOCC1
ONC(=O)\C=C\c1cccc(Nc2ncnc3cc4OCCOc4cc23)c1
Cc1ccc(COc2cccc3ccc(nc23)C(=O)NCc2ccc(cc2)C(=O)NO)cc1
COc1ccc(COc2cccc3ccc(nc23)C(=O)NCc2ccc(cc2)C(=O)NO)cc1
ONC(=O)c1ccc(CNC(=O)c2ccc3cccc(OCc4ccc(F)cc4)c3n2)cc1
COc1cccc2ccc(nc12)C(=O)NCc1ccc(cc1)C(=O)NO
ONC(=O)CCCCCCNc1nc2ccccc2nc1-c1nc2ccccc2o1
COc1cc2c(cc1-c1c(C)noc1C)[nH]c1ncnc(NCCCCCCC(=O)NO)c21 |(3.05,-2.83,;3.05,-4.37,;1.72,-5.15,;.38,-4.38,;-.95,-5.15,;-.95,-6.69,;.38,-7.46,;1.72,-6.69,;3.05,-7.46,;3.19,-8.98,;2.04,-10,;4.7,-9.31,;5.48,-7.97,;4.44,-6.82,;4.76,-5.31,;-2.41,-7.16,;-3.32,-5.92,;-4.85,-5.76,;-5.48,-4.35,;-4.57,-3.1,;-3.04,-3.26,;-2.14,-2.02,;-2.76,-.61,;-1.86,.64,;-2.49,2.04,;-1.59,3.29,;-2.21,4.7,;-1.31,5.94,;-1.94,7.35,;-3.47,7.51,;-1.03,8.6,;-1.66,10,;-2.41,-4.67,)|
COc1cc2c(cc1-c1c(C)noc1C)[nH]c1nc(C)nc(NCCCCCCC(=O)NO)c21 |(3.82,-2.83,;3.82,-4.37,;2.48,-5.15,;1.15,-4.38,;-.18,-5.15,;-.18,-6.69,;1.15,-7.46,;2.48,-6.69,;3.82,-7.46,;3.96,-8.98,;2.8,-10,;5.47,-9.31,;6.24,-7.97,;5.21,-6.82,;5.52,-5.31,;-1.65,-7.16,;-2.55,-5.92,;-4.08,-5.76,;-4.71,-4.35,;-6.24,-4.19,;-3.81,-3.1,;-2.27,-3.26,;-1.37,-2.02,;-2,-.61,;-1.1,.64,;-1.72,2.04,;-.82,3.29,;-1.45,4.7,;-.54,5.94,;-1.17,7.35,;-2.7,7.51,;-.27,8.6,;-.9,10,;-1.65,-4.67,)|
[H][C@]12CCCN1C(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCCCC(=O)NO)NC2=O
[H][C@]12CCCCN1C(=O)[C@@]([H])(NC(=O)[C@H](Cc1c[nH]c3ccccc13)NC(=O)[C@H](CCCCCC(=O)NO)NC2=O)[C@@H](C)CC |r|
FC(F)c1nnc(o1)-c1ccc(Cn2cc(nn2)-c2ccc(NC3NCC=N3)cc2)cc1 |c:28|
COc1cc2CC(CC3CCN(Cc4ccc(\C=C\C(=O)NO)cc4)CC3)C(=O)c2cc1OC
COc1cc2CC(CC3CCN(CC3)S(=O)(=O)c3cccc(\C=C\C(=O)NO)c3)C(=O)c2cc1OC
COc1cc2CC(CC3CCN(Cc4cccc(NC(=O)CCCCCCC(=O)NO)c4)CC3)C(=O)c2cc1OC
COc1cc2CC(CC3CCN(Cc4ccc(NC(=O)CCCCCCC(=O)NO)cc4)CC3)C(=O)c2cc1OC
COc1cc2CC(CC3CCN(Cc4ccc(NCc5ccc(cc5)C(=O)NO)cc4)CC3)C(=O)c2cc1OC
COc1ccc(cc1)-c1cc(ccn1)C(=O)NCc1ccc(cc1)C(=O)NO
COc1ccc(cc1)-c1cc(ccn1)-c1ccn(Cc2ccc(cc2)C(=O)NO)n1
COc1cc(NCc2ccc(cc2)C(=O)NO)c2ncccc2c1
ONC(=O)c1ccc(CNc2cccc3ccc(F)nc23)cc1
ONC(=O)c1ccc(CNC2CCCc3cccnc23)cc1
ONC(=O)c1ccc(CN2CCc3cccnc23)cc1
ONC(=O)c1ccc(CN2CCCc3cccnc23)cc1
COc1cc(ccc1CN1CCCc2cccnc12)C(=O)NO
COc1cc(CN2CCCc3cccnc23)ccc1C(=O)NO
ONC(=O)c1ccc(CN2CCCc3cccnc23)c(F)c1
ONC(=O)c1ccc(CNC2CCCc3cccnc23)c(F)c1
ONC(=O)c1ccc(CN2CCc3cccnc23)c(F)c1
COc1ccc(cc1O)[C@H]1[C@H](COC(=O)CCC(=O)NO)C(=O)N1c1cc(OC)c(OC)c(OC)c1 |r|
COc1ccc(cc1O)[C@H]1[C@H](COC(=O)c2ccc(cc2)C(=O)NO)C(=O)N1c1cc(OC)c(OC)c(OC)c1 |r|
ONC(=O)CNC(=O)c1ncc(o1)-c1ccccc1
ONC(=O)CCCCNC(=O)c1ncc(o1)-c1ccccc1
ONC(=O)CCCCCNC(=O)c1ncc(o1)-c1ccccc1
ONC(=O)CCCCCCNC(=O)c1ncc(o1)-c1ccccc1
ONC(=O)CCCCCCCNC(=O)c1ncc(o1)-c1ccccc1
COc1ccc(cc1)-c1cnc(o1)C(=O)NCCCCCCC(=O)NO
COc1ccc(cc1)-c1cnc(o1)C(=O)NCC(=O)NO
COc1ccc(cc1)-c1cnc(o1)C(=O)NCCCC(=O)NO
COc1ccc(cc1)-c1cnc(o1)C(=O)NCCCCC(=O)NO
COc1ccc(cc1)-c1cnc(o1)C(=O)NCCCCCC(=O)NO
COc1ccc(cc1)-c1cnc(o1)C(=O)NCCCCCCCC(=O)NO
COc1cccc(c1)-c1cnc(o1)C(=O)NCCCCCCC(=O)NO
COc1cccc(c1)-c1cnc(o1)C(=O)NCCCCCCCC(=O)NO
COc1ccccc1-c1cnc(o1)C(=O)NCCCCCCC(=O)NO
ONC(=O)CCCCCCNC(=O)c1ncc(o1)-c1ccc(F)cc1
ONC(=O)CCCCCCNC(=O)c1ncc(o1)-c1ccc(Br)cc1
ONC(=O)CCCCCCCNC(=O)c1ncc(o1)-c1ccc(Br)cc1
ONC(=O)CCCCCCNC(=O)c1ncc(o1)-c1cccc(Br)c1
ONC(=O)CCCCCCNC(=O)c1ncc(o1)-c1ccc(Cl)cc1
ONC(=O)CCCCCCNC(=O)c1ncc(o1)-c1cccc(Cl)c1
ONC(=O)CCCCCCNC(=O)c1ncc(o1)-c1ccccc1Cl
Cc1ccc(cc1)-c1cnc(o1)C(=O)NCCCCCC(=O)NO
Cc1ccc(cc1)-c1cnc(o1)C(=O)NCCCCCCC(=O)NO
Cc1cccc(c1)-c1cnc(o1)C(=O)NCCCCCCC(=O)NO
Cc1ccccc1-c1cnc(o1)C(=O)NCCCCCCC(=O)NO
ONC(=O)CCCCCCNC(=O)c1ncc(o1)-c1ccc(cc1)C(F)(F)F
ONC(=O)CCCCCCCNC(=O)c1ncc(o1)-c1ccc(cc1)C(F)(F)F
ONC(=O)CCCCCCNC(=O)c1ncc(o1)-c1cccc(c1)C(F)(F)F
ONC(=O)CCCCCNC(=O)c1ncc(s1)-c1ccccc1
ONC(=O)CCCCCCNC(=O)c1ncc(s1)-c1ccccc1
ONC(=O)CCCCCCNC(=O)c1ncc(s1)-c1ccc(F)cc1
ONC(=O)CCCCCCNC(=O)c1ncc(s1)-c1ccc(Cl)cc1
ONC(=O)CCCCCCNC(=O)c1ncc(s1)-c1cccc(Cl)c1
ONC(=O)CCCCCCNC(=O)c1ncc(s1)-c1ccccc1Cl
COc1ccc(cc1)-c1cnc(s1)C(=O)NCCCCCC(=O)NO
COc1ccc(cc1)-c1cnc(s1)C(=O)NCCCCCCC(=O)NO
COc1ccc(cc1)-c1cnc(s1)C(=O)NCCCCCCCC(=O)NO
COc1cccc(c1)-c1cnc(s1)C(=O)NCCCCCCC(=O)NO
COc1cccc(c1)-c1cnc(s1)C(=O)NCCCCCCCC(=O)NO
COc1ccccc1-c1cnc(s1)C(=O)NCCCCCCC(=O)NO
Cc1ccc(cc1)-c1cnc(s1)C(=O)NCCCCCCC(=O)NO
Cc1cccc(c1)-c1cnc(s1)C(=O)NCCCCCCC(=O)NO
Cc1ccccc1-c1cnc(s1)C(=O)NCCCCCCC(=O)NO
ONC(=O)CCCCCCNC(=O)c1ncc(s1)-c1ccc(cc1)C(F)(F)F
ONC(=O)CCCCCCNC(=O)c1ncc(s1)-c1cccc(c1)C(F)(F)F
Cc1cc(-c2ccc(C=c3c(=C)[nH]n(-c4ccc(cc4)C(O)=O)c3=O)o2)c(cc1C)[N+]([O-])=O |w:8.7|
Nc1ccccc1NC(=O)c1ccc(NC(=O)c2n[nH]cc2NC(=O)c2c(Cl)cccc2Cl)cc1
ONC(=O)c1ccc(COc2no[n+]([O-])c2S(=O)(=O)c2ccccc2)cc1
ONC(=O)\C=C\COc1no[n+]([O-])c1S(=O)(=O)c1ccccc1
ONC(=O)c1ccc(Oc2no[n+]([O-])c2S(=O)(=O)c2ccccc2)cc1
ONC(=O)c1cccc(Oc2no[n+]([O-])c2S(=O)(=O)c2ccccc2)c1
COc1cc(ccc1Oc1no[n+]([O-])c1S(=O)(=O)c1ccccc1)C(=O)NO
ONC(=O)\C=C\c1ccc(Oc2no[n+]([O-])c2S(=O)(=O)c2ccccc2)cc1
ONC(=O)CCn1c2cc(Cl)ccc2c(=O)n(Cc2ccccc2)c1=O
ONC(=O)CCn1c2ccccc2c(=O)n(CCc2ccccc2)c1=O
ONC(=O)c1ccc(Cn2c3ccccc3c(=O)n(CCc3ccccc3)c2=O)c(F)c1
CCc1nc2c(Cc3ccc(cc3)C(=O)NO)cccc2c(=O)n1CCc1ccccc1
ONC(=O)c1ccc(Cn2c3cc(ccc3c(=O)[nH]c2=O)C(F)(F)F)cc1
ONC(=O)c1ccc(Cn2c3ccc(Br)cc3c(=O)[nH]c2=O)cc1
ONC(=O)c1ccc(Cn2c3cccc(Cl)c3c(=O)[nH]c2=O)cc1
ONC(=O)c1cccc(Cn2c3c(Cl)cccc3c(=O)[nH]c2=O)c1
ONC(=O)c1ccc(Cn2c3c(Cl)cccc3c(=O)[nH]c2=O)cc1
ONC(=O)c1ccc(\C=C\c2nc3ccccc3c(=O)[nH]2)cc1
ONC(=O)c1ccc(cc1)-c1nc2ccccc2c(=O)[nH]1
ONC(=O)c1ccc(Cn2c3cc(F)ccc3c(=O)[nH]c2=O)cc1
ONC(=O)c1ccc(Cn2c3ccc(F)cc3c(=O)[nH]c2=O)cc1
Cc1nc2cc(\C=C\C(=O)NO)ccc2c(=O)n1-c1ccccc1
Cc1nc2ccc(\C=C\CC(=O)NO)cc2c(=O)n1-c1ccccc1
CCc1nc2ccc(\C=C\CC(=O)NO)cc2c(=O)n1-c1ccccc1
Cn1c(CCC(=O)NO)nc2ccccc2c1=O
SCC(=O)Nc1ccc(Cn2c3c(Cl)cccc3c(=O)[nH]c2=O)cc1
COc1ccc2c3CCN(Cc3oc2c1)[C@@H](Cc1ccccc1)C(=O)Nc1ccc(cc1)C(=O)NO |r|
ONC(=O)\C=C\c1ccc(NC(=O)Cc2ccccc2)cn1
CCC(C(=O)Nc1ccc(\C=C\C(=O)NO)nc1)c1ccccc1
CC(C)C(C(=O)Nc1ccc(\C=C\C(=O)NO)nc1)c1ccccc1
ONC(=O)\C=C\c1ccc(NC(=O)Cc2ccc3ccccc3c2)cn1
CCC(C(=O)Nc1ccc(nc1)C(=O)NO)c1ccccc1
CC(C)C(C(=O)Nc1ccc(nc1)C(=O)NO)c1ccccc1
ONC(=O)c1ccc(NC(=O)C(Cc2ccccc2)c2ccccc2)cn1
ONC(=O)c1ccc(NC(=O)Cc2ccc3ccccc3c2)cn1
C[C@@H](O)C(=O)CCCCCCC(=O)Nc1ccccc1 |r|
C[C@H](O)C(=O)CCCCCCC(=O)Nc1ccccc1 |r|
C[C@@H](OC(C)=O)C(=O)CCCCCCC(=O)Nc1ccccc1 |r|
c1ccc(cc1)NC(=O)CCCCCCC(=O)C(F)(F)F
C[Si](O)(O)CCCCCCC(=O)Nc1ccccc1
CCC(=O)CCCCCCC(=O)Nc1ccccc1
OCC(=O)CCCCCCC(=O)Nc1ccccc1
CCN(CC)C(=S)SSCCCCCC(=O)Nc1ccccc1
ON1C[C@@H](CCCCCC(=O)Nc2ccccc2)C1=O |r|
ON1C[C@H](CCCCCC(=O)Nc2ccccc2)C1=O |r|
O=C(CCCCCC1CNC1=O)Nc1ccccc1
Nc1ccccc1N1CC(CCCCCC(=O)Nc2ccccc2)C1=O
Cc1onc(c1C(=O)NCCCCCCC(=O)NO)-c1ccccc1
CNC(=O)CN1C(=Nc2ccccc2C1=O)CCC(=O)O
CCNC(=O)Cn1c(CCC(O)=O)nc2ccccc2c1=O
OC(=O)CCc1nc2ccccc2c(=O)n1CC(=O)NC1CC1
CC(C)(C)NC(=O)Cn1c(CCC(O)=O)nc2ccccc2c1=O
OC(=O)CCc1nc2ccccc2c(=O)n1CC(=O)NC12CC3CC(CC(C3)C1)C2 |TLB:27:22:29:26.28.25,27:26:29:23.22.21,THB:28:20:23:27.26.25,28:26:23:20.29.21|
OC(=O)CCc1nc2ccccc2c(=O)n1CC(=O)NCC1CCCCC1
c1ccc(cc1)CNC(=O)CN2C(=Nc3ccccc3C2=O)CCC(=O)O
COc1ccccc1CNC(=O)Cn1c(CCC(O)=O)nc2ccccc2c1=O
OC(=O)CCc1nc2ccccc2c(=O)n1CC(=O)NCc1ccccc1Cl
OC(=O)CCc1nc2ccccc2c(=O)n1CC(=O)NCc1ccc(cc1)C(F)(F)F
OC(=O)CCc1nc2ccccc2c(=O)n1CC(=O)NCc1cccnc1
COc1ccc(CNC(=O)Cn2c(CCC(O)=O)nc3ccccc3c2=O)cc1
OC(=O)CCc1nc2ccccc2c(=O)n1CC(=O)NCCc1ccccc1
COc1ccccc1CCNC(=O)Cn1c(CCC(O)=O)nc2ccccc2c1=O
COc1ccccc1CNC(=O)Cn1c(CCC(O)=O)nc2c(F)cccc2c1=O
COc1ccccc1CNC(=O)Cn1c(CCC(O)=O)nc2c(C)cccc2c1=O
COc1ccccc1CNC(=O)CN2C(=Nc3c(cccc3Cl)C2=O)CCC(=O)O
COc1ccccc1CNC(=O)Cn1c(CCC(O)=O)nc2c(Cl)cc(I)cc2c1=O
Cc1ccccc1CNC(=O)Cn1c(CCC(O)=O)nc2c(Cl)cccc2c1=O
OC(=O)CCc1nc2c(Cl)cccc2c(=O)n1CC(=O)NCc1ccccc1F
OC(=O)CCc1nc2c(Cl)cccc2c(=O)n1CC(=O)NCc1ccccc1Cl
OC(=O)CCc1nc2c(Cl)cccc2c(=O)n1CC(=O)NCC1CCCCO1
OC(=O)CCc1nc2c(Cl)cccc2c(=O)n1CC(=O)NCC1CCCO1
COc1ccccc1CN(C)C(=O)Cn1c(CCC(O)=O)nc2c(Cl)cccc2c1=O
ONC(=O)CCCCCN1c2ccccc2S(=O)(=O)C(CC1=O)c1ccccc1
ONC(=O)CCCCCN1c2ccccc2S(=O)(=O)C(CC1=O)c1ccc(Cl)c(Cl)c1
Cc1nc(NC(=O)N2C[C@@H](C[C@H]2C(N)=O)NC(=O)CCCC(=O)NO)sc1-c1ccnc(c1)C(C)(C)C(F)(F)F |r|
Cc1nc(NC(=O)N2C[C@@H](C[C@H]2C(N)=O)NC(=O)CCCCC(=O)NO)sc1-c1ccnc(c1)C(C)(C)C(F)(F)F |r|
Cc1nc(NC(=O)N2C[C@@H](C[C@H]2C(N)=O)NC(=O)CCCCCCC(=O)NO)sc1-c1ccnc(c1)C(C)(C)C(F)(F)F |r|
Cc1nc(NC(=O)N2C[C@@H](C[C@H]2C(N)=O)NC(=O)c2ccc(cc2)C(=O)NO)sc1-c1ccnc(c1)C(C)(C)C(F)(F)F |r|
Cc1nc(NC(=O)N2C[C@@H](C[C@H]2C(N)=O)NC(=O)Cc2ccc(cc2)C(=O)NO)sc1-c1ccnc(c1)C(C)(C)C(F)(F)F |r|
Cc1nc(NC(=O)N2C[C@@H](C[C@H]2C(N)=O)NC(=O)c2ccc(cn2)C(=O)NO)sc1-c1ccnc(c1)C(C)(C)C(F)(F)F |r|
Cc1nc(NC(=O)N2C[C@@H](C[C@H]2C(N)=O)Nc2ccc(cn2)C(=O)NO)sc1-c1ccnc(c1)C(C)(C)C(F)(F)F |r|
Cc1nc(NC(=O)N2C[C@@H](C[C@H]2C(N)=O)Nc2ncc(cn2)C(=O)NO)sc1-c1ccnc(c1)C(C)(C)C(F)(F)F |r|
Cc1nc(NC(=O)N2C[C@@H](C[C@H]2C(N)=O)NS(=O)(=O)c2ccc(cc2)C(=O)NO)sc1-c1ccnc(c1)C(C)(C)C(F)(F)F |r|
Cc1nc(NC(=O)N2C[C@@H](C[C@H]2C(N)=O)NS(=O)(=O)Cc2ccc(cc2)C(=O)NO)sc1-c1ccnc(c1)C(C)(C)C(F)(F)F |r|
CCCNNC(=O)c1cnc(NCc2ccc(OC)cc2)cn1
ONC(=O)CCCCCNc1cc(nc(n1)-c1ccccn1)N1CCc2ccccc2CC1
ONC(=O)CCCCNc1cc(nc(n1)-c1ccccn1)N1CCc2ccccc2CC1
ONC(=O)CNc1cc(nc(n1)-c1ccccn1)N1CCc2ccccc2CC1
ONC(=O)CCNc1cc(nc(n1)-c1ccccn1)N1CCc2ccccc2CC1
ONC(=O)CCCNc1cc(nc(n1)-c1ccccn1)N1CCc2ccccc2CC1
ONC(=O)CNc1cc(nc(n1)-c1ccccn1)N1CCCCCC1
ONC(=O)CCNc1cc(nc(n1)-c1ccccn1)N1CCCCCC1
ONC(=O)CCCNc1cc(nc(n1)-c1ccccn1)N1CCCCCC1
CN(Cc1ccccc1)c1cc(NCC(=O)NO)nc(n1)-c1ccccn1
CN(Cc1ccccc1)c1cc(NCCC(=O)NO)nc(n1)-c1ccccn1
CN(Cc1ccccc1)c1cc(NCCCC(=O)NO)nc(n1)-c1ccccn1
ONC(=O)CNc1cc(nc(n1)-c1ccccn1)N1CCN(CC1)c1ccc(F)cc1
ONC(=O)CCNc1cc(nc(n1)-c1ccccn1)N1CCN(CC1)c1ccc(F)cc1
ONC(=O)CCCNc1cc(nc(n1)-c1ccccn1)N1CCN(CC1)c1ccc(F)cc1
ONC(=O)CNc1cc(nc(n1)-c1cccnc1)N1CCCCCC1
ONC(=O)CCNc1cc(nc(n1)-c1cccnc1)N1CCCCCC1
ONC(=O)CCCNc1cc(nc(n1)-c1cccnc1)N1CCCCCC1
CN(Cc1ccccc1)c1cc(NCC(=O)NO)nc(n1)-c1cccnc1
CN(Cc1ccccc1)c1cc(NCCC(=O)NO)nc(n1)-c1cccnc1
CN(Cc1ccccc1)c1cc(NCCCC(=O)NO)nc(n1)-c1cccnc1
ONC(=O)CNc1cc(cc(c1)-c1cccnc1)N1CCN(CC1)c1ccc(F)cc1
ONC(=O)CCNc1cc(cc(c1)-c1cccnc1)N1CCN(CC1)c1ccc(F)cc1
ONC(=O)CCCNc1cc(cc(c1)-c1cccnc1)N1CCN(CC1)c1ccc(F)cc1
ONC(=O)CCCCCCNc1cc(nc(n1)-c1ccccn1)N1CCc2ccccc2CC1
ONC(=O)CCCCNc1cc(nc(n1)-c1ccccn1)N1CCCCCC1
ONC(=O)CCCCCNc1cc(nc(n1)-c1ccccn1)N1CCCCCC1
ONC(=O)CCCCCCNc1cc(nc(n1)-c1ccccn1)N1CCCCCC1
CN(Cc1ccccc1)c1cc(NCCCCC(=O)NO)nc(n1)-c1ccccn1
CN(Cc1ccccc1)c1cc(NCCCCCC(=O)NO)nc(n1)-c1ccccn1
CN(Cc1ccccc1)c1cc(NCCCCCCC(=O)NO)nc(n1)-c1ccccn1
ONC(=O)CCCCCCNc1cc(nc(n1)-c1cccnc1)N1CCCCCC1
CN(Cc1ccccc1)c1cc(NCCCCCCC(=O)NO)nc(n1)-c1cccnc1
OC(=O)CCNc1cc(nc(n1)-c1ccccn1)N1CCc2ccccc2CC1
FC(F)c1nnc(o1)-c1cnc(NCc2ccccc2)nc1
COc1ccc(CNc2ncc(cn2)-c2nnc(o2)C(F)F)cc1
FC(F)(F)c1nnc(o1)-c1cnc(NCc2ccccc2)nc1
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CNC(=O)[C@@H]3CCC(=O)N3Cc3ccccc3)cc2)cc1 |r|
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CNC(=O)[C@H]3CCC(=O)N3Cc3ccccc3)cc2)cc1 |r|
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CNC(=O)[C@@H]3CCC(=O)N3Cc3ccc(F)cc3)cc2)cc1 |r|
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CNC(=O)[C@@H]3CCC(=O)N3Cc3ccc(Br)cc3)cc2)cc1 |r|
Nc1ccccc1NC(=O)c1ccc(COc2ccc(NC(=O)[C@@H]3CCC(=O)N3Cc3ccccc3)cc2)cc1 |r|
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CN3[C@H](CC(=O)NCc4ccccc4)CCC3=O)cc2)cc1 |r|
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CNC(=O)[C@@H]3CCCN3Cc3ccccc3)cc2)cc1 |r|
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CNC(=O)[C@H]3CCCN3Cc3ccccc3)cc2)cc1 |r|
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CNC(=O)[C@@H]3CCCN3)cc2)cc1
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CNC(=O)[C@H]3CCCN3)cc2)cc1
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CNC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)cc1 |r|
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CNC(=O)[C@@H]3CCCN3C(=O)c3ccccc3)cc2)cc1 |r|
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CNC(=O)[C@@H]3CCCN3Cc3ccc(F)cc3)cc2)cc1 |r|
OC(=O)c1ccc(COc2ccc(CNC(=O)[C@@H]3CCCN3Cc3ccccc3)cc2)cc1 |r|
O=C(NCc1ccc(OCc2ccc(cc2)C(=O)NCc2ccccc2)cc1)[C@@H]1CCC(=O)N1Cc1ccccc1 |r|
O=C(NCc1ccc(OCc2ccc(cc2)C(=O)Nc2ccccc2)cc1)[C@@H]1CCC(=O)N1Cc1ccccc1 |r|
ONC(=O)c1ccc(COc2ccc(CNC(=O)[C@@H]3CCC(=O)N3Cc3ccccc3)cc2)cc1 |r|
OB(O)c1ccc(COc2ccc(CNC(=O)[C@@H]3CCC(=O)N3Cc3ccccc3)cc2)cc1 |r|
OC(=O)c1ccc(COc2ccc(CNC(=O)[C@@H]3CCC(=O)N3Cc3ccccc3)cc2)cc1 |r|
OC(=O)c1ccc(COc2ccc(CNC(=O)[C@@H]3CCC(=O)N3Cc3ccc(Br)cc3)cc2)cc1 |r|
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CNC(=O)C3CCCO3)cc2)cc1
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CNC(=O)c3ccccn3)cc2)cc1
Nc1ccccc1NC(=O)c1ccc(COc2ccc(CNC(=O)c3cc4ccccc4[nH]3)cc2)cc1
CC(C)(C)OC(=O)NCc1ccc(OCc2ccc(cc2)C(=O)Nc2ccccc2N)cc1
NCc1ccc(OCc2ccc(cc2)C(=O)Nc2ccccc2N)cc1
Cc1cnc(Nc2ccc(OCCN3CCCC3)cc2)nc1Nc1ccc(cc1)C(=O)NO
FC(F)c1nnc(o1)-c1ccc(Cn2nnc(n2)-c2ccccn2)nc1
COc1ccccc1-c1nnn(Cc2ccc(cn2)-c2nnc(o2)C(F)F)n1
CS(=O)(=O)NCC(Nc1ncc(cn1)-c1nnc(o1)C(F)F)c1ccc(OC(F)(F)F)cc1
COc1cc(NCC(=O)NCCCCCCCC(=O)Nc2ccc(cc2)C(=O)NCCCCCCC(=O)NO)ccc1C(=O)NC1CCC(=O)NC1=O
Cc1cc(nc(n1)SCC(=O)Nc2ncc(s2)Cc3cccc(c3)OCc4cn(nn4)CCOC)C
Cc1cc(C)nc(SCC(=O)Nc2ncc(Cc3cccc(c3)C(=O)NO)s2)n1
Cc1cc(C)nc(SCC(=O)Nc2ncc(Cc3ccc(cc3)C(=O)NO)s2)n1
Cc1cc(C)nc(SCC(=O)Nc2ncc(Cc3cccc(OCc4cn(Cc5ccc(cc5)C(=O)NO)nn4)c3)s2)n1
Cc1cc(C)nc(SCC(=O)Nc2ncc(Cc3cccc(OCc4cn(CCCCC(=O)NCc5ccc(cc5)C(=O)NO)nn4)c3)s2)n1
CCCCN(Cc1ccc(cc1)C(=O)NO)C(=O)CCCCn1cc(COc2cccc(Cc3cnc(NC(=O)CSc4nc(C)cc(C)n4)s3)c2)nn1
Cc1cc(C)nc(SCC(=O)Nc2ncc(Cc3cccc(OCc4cn(CCOCCOCCOCCOCCC(=O)Nc5ccc(cc5)C(=O)NCc5ccc(cc5)C(=O)NO)nn4)c3)s2)n1
Cc1cc(C)nc(SCC(=O)Nc2ncc(Cc3cccc(OCc4cn(CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCC(=O)Nc5ccc(cc5)C(=O)NCc5ccc(cc5)C(=O)NO)nn4)c3)s2)n1
Cc1cc(C)nc(SCC(=O)Nc2ncc(Cc3cccc(OCc4cn(CCOCCOCCOCCOCCC(=O)Nc5ccc(cc5)C(=O)NCCCCCCC(=O)NO)nn4)c3)s2)n1
CC(=O)NCc1ccc(cc1)C(=O)NO
ONC(=O)c1ccc(CNC(=O)c2ccccc2)cc1
CCCCC(=O)N(CCCC)Cc1ccc(cc1)C(=O)NO
CN1CCC2C(C1)c1ccccc1N2Cc1ccc(cc1)C(=O)NO
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(cc5)C(=O)NO)ccc4c1)(C2)C3 |r,TLB:8:6:36:2.1.35,8:1:36:6.9.5,5:3:6.9.8:35,THB:5:6:36.3.2:35|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(cc5F)C(=O)NO)ccc4c1)(C2)C3 |r,TLB:8:6:37:2.1.36,8:1:37:6.9.5,5:3:6.9.8:36,THB:5:6:37.3.2:36|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(C(=O)NO)c(F)c5)ccc4c1)(C2)C3 |r,TLB:8:6:37:2.1.36,8:1:37:6.9.5,5:3:6.9.8:36,THB:5:6:37.3.2:36|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(cc5OC)C(=O)NO)ccc4c1)(C2)C3 |r,TLB:8:6:38:2.1.37,8:1:38:6.9.5,5:3:6.9.8:37,THB:5:6:38.3.2:37|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(C(=O)NO)c(OC)c5)ccc4c1)(C2)C3 |r,TLB:8:6:38:2.1.37,8:1:38:6.9.5,5:3:6.9.8:37,THB:5:6:38.3.2:37|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(C(=O)NO)c(C)c5)ccc4c1)(C2)C3 |r,TLB:8:6:37:2.1.36,8:1:37:6.9.5,5:3:6.9.8:36,THB:5:6:37.3.2:36|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(C(=O)NO)c(O)c5)ccc4c1)(C2)C3 |r,TLB:8:6:37:2.1.36,8:1:37:6.9.5,5:3:6.9.8:36,THB:5:6:37.3.2:36|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(C(=O)NO)c(OCC)c5)ccc4c1)(C2)C3 |r,TLB:8:6:39:2.1.38,8:1:39:6.9.5,5:3:6.9.8:38,THB:5:6:39.3.2:38|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(C(=O)NO)c(Cl)c5)ccc4c1)(C2)C3 |r,TLB:8:6:37:2.1.36,8:1:37:6.9.5,5:3:6.9.8:36,THB:5:6:37.3.2:36|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(C(=O)NO)c(Br)c5)ccc4c1)(C2)C3 |r,TLB:8:6:37:2.1.36,8:1:37:6.9.5,5:3:6.9.8:36,THB:5:6:37.3.2:36|
COc1cc(ccc1C(=O)NO)C(=O)NCC12CC3CC(CC(C3)C1)C2 |TLB:23:22:25:19.18.17,23:18:25:22.24.21,THB:21:22:25.20.19:17,21:20:22.24.23:17|
COc1cc(ccc1C(=O)NO)C(=O)NCCC12CC3CC(CC(C3)C1)C2 |TLB:24:23:26:20.19.18,24:19:26:23.25.22,THB:22:23:26.21.20:18,22:21:23.25.24:18|
COc1cc(CN(C)CC23CC4CC(CC(C4)C2)C3)ccc1C(=O)NO |TLB:16:15:18:12.11.10,16:11:18:15.17.14,THB:14:15:18.13.12:10,14:13:15.17.16:10|
COc1cc(CN(C)CCC23CC4CC(CC(C4)C2)C3)ccc1C(=O)NO |TLB:17:16:19:13.12.11,17:12:19:16.18.15,THB:15:16:19.14.13:11,15:14:16.18.17:11|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CNC(=O)c1ccc4n(Cc5ccc(cc5)C(=O)NNCCC)ccc4c1)(C2)C3 |r,TLB:8:6:39:2.1.38,8:1:39:6.9.5,5:3:6.9.8:38,THB:5:6:39.3.2:38|
Nc1ccccc1NC(=O)c1ccc(CNC(=O)OC2CCN(CC2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
Nc1nn(nc1C(=O)NCc1ccc(cc1)C(=O)NO)-c1ccccc1
Nc1nn(nc1C(=O)NCc1ccc(cc1)C(=O)Nc1ccccc1N)-c1ccccc1Cl
Cc1cnc(Nc2ccc(OCCCCCCC(=O)NO)cc2)nc1Nc1cccc(c1)S(=O)(=O)NC(C)(C)C
Cc1cnc(Nc2ccc(OCCCCCCC(=O)NO)c(F)c2)nc1Nc1cccc(c1)S(=O)(=O)NC(C)(C)C
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CC(=O)Nc1ccc(cc1)C(=O)NCCCCCCC(=O)NO)(C2)C3 |r,TLB:5:3:9.6.8:34,THB:2:1:9:3.5.35,2:3:9:8.1.34,5:6:2.3.35:34|
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CC(=O)NCC(=O)Nc1ccc(cc1)C(=O)NCCCCCCC(=O)NO)(C2)C3 |r,TLB:5:3:9.6.8:38,THB:2:1:9:3.5.39,2:3:9:8.1.38,5:6:2.3.39:38|
ONC(=O)CCCCCCNC(=O)c1ccc(NC(=O)CNC(=O)CC2c3ccccc3-c3ccccc23)cc1
[H][C@]12C[C@]3([H])C[C@]([H])(C1)CC(CC(=O)NCCOCCOCCCCCCn1cc(nn1)-c1ccc(cc1)C(=O)NCCCCCCC(=O)NO)(C2)C3 |r,TLB:11:10:8.1.2:5,THB:51:10:8.1.2:5,51:1:5:10.9.52,2:1:9:3.5.52,2:3:9:8.1.51|
COc1ccc(-c2nc3ccccc3s2)cc1OCCCCCCC(=O)NO
Cc1c2ccc(Nc3ccnc(Nc4ccc(NC(=O)CCCCCCC(=O)NO)cc4)n3)cc2nn1C
Cc1c2ccc(Nc3ccnc(Nc4ccc(OCCCCCCC(=O)NO)cc4)n3)cc2nn1C
CCCNNC(=O)c1ccc(Nc2nccc(N(C)c3ccc4c(C)n(C)nc4c3)n2)cc1
CCCNNC(=O)c1ccc(CNC(=O)\C=C\c2cccnc2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2cc3cnccc3[nH]2)cc1
N#CC(C#N)=C1C=C(/C=C/c2ccc(O)c(NC(=O)CCCCCCC(=O)NO)c2)Oc2ccccc21
N#CC(C#N)=C1C=C(/C=C/c2ccc(O)c(NC(=O)CCCCCCC(=O)NO)c2)Oc2ccc(O)cc21
COc1ccc(/C=C/C(=O)c2ccc(OC)c3c2OC(C)(C)C=C3)cc1NCC(=O)NO
COc1ccc(/C=C/C(=O)c2ccc(Br)c3c2OC(C)(C)C=C3)cc1OCC(=O)NO
COc1ccc(/C=C/C(=O)c2ccc(Br)c3c2OC(C)(C)C=C3)cc1NCC(=O)NO
COc1ccc(C(=O)NO)cc1NCc1ccc(OCc2cn(CCCCCC(=O)Nc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)nn2)cc1
COc1ccccc1/C=C1CC(=O)N(CCCCCCC(=O)NO)C1=O
CCOc1ccc(-c2nc(C(=O)NCc3ccc(C(=O)NO)cc3)c3[nH]c(=O)n(-c4cccnc4OC)c3n2)cn1
CCN(Cc1ccc(C(=O)NO)cc1)C(=O)c1ccccc1
CCCN(Cc1ccc(C(=O)NO)cc1)C(=O)c1ccccc1
CCCCN(Cc1ccc(C(=O)NO)cc1)C(=O)c1ccccc1
O=C(NO)c1ccc(CN(CC2CC2)C(=O)c2ccccc2)cc1
O=C(NO)c1ccc(CN(CC2CCCCC2)C(=O)c2ccccc2)cc1
O=C(NO)c1ccc(CN(Cc2ccccc2)C(=O)c2ccccc2)cc1
O=C(NO)c1ccc(CN(Cc2ccco2)C(=O)c2ccccc2)cc1
O=C(NO)c1ccc(CN(Cc2cccs2)C(=O)c2ccccc2)cc1
O=C(NO)c1ccc(CN(CC23CC4CC(CC(C4)C2)C3)C(=O)c2ccccc2)cc1
O=C(NO)c1ccc(CN(Cc2cccc3ccccc23)C(=O)c2ccccc2)cc1
C[C@@H](COCCC(=O)N1CCN(c2ncc(C(=O)NO)cn2)CC1)Nc1cn[nH]c(=O)c1C(F)(F)F
C[C@@H](COCCC(=O)N1CCN(c2ccc(C(=O)NO)cn2)CC1)Nc1cn[nH]c(=O)c1C(F)(F)F
C[C@@H](COCCC(=O)N1CCN(c2cnc(C(=O)NO)cn2)CC1)Nc1cn[nH]c(=O)c1C(F)(F)F
C[C@@H](COCCC(=O)N1CC2CN(c3ncc(C(=O)NO)cn3)CC2C1)Nc1cn[nH]c(=O)c1C(F)(F)F
C[C@@H](COCCC(=O)NC1CCN(c2ncc(C(=O)NO)cn2)CC1)Nc1cn[nH]c(=O)c1C(F)(F)F
C[C@@H](COCCC(=O)N1CCC(Nc2ncc(C(=O)NO)cn2)CC1)Nc1cn[nH]c(=O)c1C(F)(F)F
C[C@@H](COCCC(=O)N1CCC2(CCN(c3ncc(C(=O)NO)cn3)C2)C1)Nc1cn[nH]c(=O)c1C(F)(F)F
C[C@@H](COCCC(=O)NCCN(C)c1ncc(C(=O)NO)cn1)Nc1cn[nH]c(=O)c1C(F)(F)F
C[C@@H](COCCC(=O)N1CCN(c2ncc(C(=O)NCCCC(=O)NO)cn2)CC1)Nc1cn[nH]c(=O)c1C(F)(F)F
C[C@@H](COCCC(=O)N1CCN(c2ncc(C(=O)NCCCCC(=O)NO)cn2)CC1)Nc1cn[nH]c(=O)c1C(F)(F)F
C[C@@H](COCCC(=O)N1CCN(c2ncc(C(=O)NCCCCCC(=O)NO)cn2)CC1)Nc1cn[nH]c(=O)c1C(F)(F)F
C[C@@H](COCCC(=O)N1CCN(c2ncc(C(=O)NCCCCCCC(=O)NO)cn2)CC1)Nc1cn[nH]c(=O)c1C(F)(F)F
C[C@@H](COCCC(=O)N1CCN(c2ncc(NC(=O)CCCCCC(=O)NO)cn2)CC1)Nc1cn[nH]c(=O)c1C(F)(F)F
C[C@@H](COCCC(=O)N1CCN(c2ncc(NC(=O)CCCCCCC(=O)NO)cn2)CC1)Nc1cn[nH]c(=O)c1C(F)(F)F
C[C@@H](COCCC(=O)N1CCN(c2ncc(-c3cnn(CCCCCC(=O)NO)c3)cn2)CC1)Nc1cn[nH]c(=O)c1C(F)(F)F
C[C@@H](COCCC(=O)N1CCN(c2ncc(-c3cnn(CCCCCCC(=O)NO)c3)cn2)CC1)Nc1cn[nH]c(=O)c1C(F)(F)F
C[C@@H](COCCC(=O)N1CCN(c2ncc(OCCCCCC(=O)NO)cn2)CC1)Nc1cn[nH]c(=O)c1C(F)(F)F
C[C@@H](COCCC(=O)N1CCN(c2ncc(OCCCCCCC(=O)NO)cn2)CC1)Nc1cn[nH]c(=O)c1C(F)(F)F
C[C@@H](COCCC(=O)N1CCN(c2ncc(OCc3ccc(C(=O)NO)cc3)cn2)CC1)Nc1cn[nH]c(=O)c1C(F)(F)F
C[C@@H](COCCC(=O)N1CCN(c2ncc(OCc3ccc(/C=C/C(=O)NO)cc3)cn2)CC1)Nc1cn[nH]c(=O)c1C(F)(F)F
O=C(NO)c1ccc(Cn2c3c(c4ccccc42)C(=O)CCC3)cc1
CC1(C)CC(=O)c2c(n(Cc3ccc(C(=O)NO)cc3)c3ccc(Br)cc23)C1
CC1(C)CC(=O)c2c(n(Cc3ccc(C(=O)NO)cc3)c3ccccc23)C1
O=C(NO)c1ccc(Cn2c3c(c4cc(F)ccc42)C(=O)CCC3)cc1
O=C(NO)c1ccc(Cn2c3c(c4ccccc42)C(=O)C(CN2CCCCC2)CC3)cc1
CC1CN(CC2CCc3c(c4ccccc4n3Cc3ccc(C(=O)NO)cc3)C2=O)CC(C)O1
CN1CCN(CC2CCc3c(c4ccccc4n3Cc3ccc(C(=O)NO)cc3)C2=O)CC1
CCN1CCN(CC2CCc3c(c4ccccc4n3Cc3ccc(C(=O)NO)cc3)C2=O)CC1
CC1(C)Cc2c(c3ccccc3n2Cc2ccc(C(=O)NO)cc2)C(=O)C1CN1CCOCC1
Cc1nccn1CC1C(=O)c2c(n(Cc3ccc(C(=O)NO)cc3)c3ccccc23)CC1(C)C
O=C(NO)c1ccc(Cn2c3c(c4ccccc42)C(=O)C(CN2CCN(c4ccc(F)cc4)CC2)CC3)cc1
Cc1ccc(N2CCN(CC3CCc4c(c5ccccc5n4Cc4ccc(C(=O)NO)cc4)C3=O)CC2)cc1C
CC(C)(C)OC(=O)N1CCN(CC2CCc3c(c4ccccc4n3Cc3ccc(C(=O)NO)cc3)C2=O)CC1
O=C(NO)c1ccc(Cn2c3c(c4cc(F)ccc42)C(=O)C(CN2CCOCC2)CC3)cc1
CN1CCN(CC2CCc3c(c4cc(F)ccc4n3Cc3ccc(C(=O)NO)cc3)C2=O)CC1
CC(C)(C)OC(=O)N1CCN(CC2CCc3c(c4cc(F)ccc4n3Cc3ccc(C(=O)NO)cc3)C2=O)CC1
Cc1nccn1CC1CCc2c(c3cc(F)ccc3n2Cc2ccc(C(=O)NO)cc2)C1=O
CC(C)N1CCN(CC2CCc3c(c4cc(F)ccc4n3Cc3ccc(C(=O)NO)cc3)C2=O)CC1
CCN1CCN(CC2CCc3c(c4cc(F)ccc4n3Cc3ccc(C(=O)NO)cc3)C2=O)CC1
CCCCN1CCN(CC2CCc3c(c4cc(F)ccc4n3Cc3ccc(C(=O)NO)cc3)C2=O)CC1
CC1(C)Cc2c(c3cc(F)ccc3n2Cc2ccc(C(=O)NO)cc2)C(=O)C1CN1CCOCC1
CN1CCN(CC2C(=O)c3c(n(Cc4ccc(C(=O)NO)cc4)c4ccc(F)cc34)CC2(C)C)CC1
CC1(C)CC(=O)c2c(C(F)(F)F)nn(Cc3ccc(C(=O)NO)cc3)c2C1
Cc1c2c(n(Cc3ccc(C(=O)NO)cc3)c1C)CCCC2=O
Cc1c2c(n(Cc3ccc(C(=O)NO)cc3)c1C)CC(C)(C)CC2=O
Cc1nn(Cc2ccc(C(=O)NO)cc2)c2c1C(=O)CC(C)(C)C2
Cc1cn(Cc2ccc(C(=O)NO)cc2)c2c1C(=O)CC(C)(C)C2
Cc1cn(Cc2ccc(C(=O)NO)cc2)c2c1C(=O)CCC2
O=C(CN(C(=O)Cc1ccc(C(=O)NO)cc1)c1ccccc1)NC1CCCCC1
O=C(CN(C(=O)Cc1ccc(C(=O)NO)cc1)c1ccccc1)NCc1ccccc1
CCCCNC(=O)CN(C(=O)Cc1ccc(C(=O)NO)cc1)c1ccccc1
CC(C)(C)NC(=O)CN(C(=O)Cc1ccc(C(=O)NO)cc1)c1ccccc1
Cc1ccccc1N(CC(=O)NC1CCCCC1)C(=O)Cc1ccc(C(=O)NO)cc1
Cc1cccc(N(CC(=O)NC2CCCCC2)C(=O)Cc2ccc(C(=O)NO)cc2)c1
Cc1ccc(N(CC(=O)NC2CCCCC2)C(=O)Cc2ccc(C(=O)NO)cc2)cc1
CCc1ccccc1N(CC(=O)NC1CCCCC1)C(=O)Cc1ccc(C(=O)NO)cc1
O=C(CN(C(=O)Cc1ccc(C(=O)NO)cc1)c1ccccc1C(F)(F)F)NC1CCCCC1
O=C(CN(C(=O)Cc1ccc(C(=O)NO)cc1F)c1ccccc1)NC1CCCCC1
Cc1ccccc1N(CC(=O)NC1CCCCC1)C(=O)Cc1ccc(C(=O)NO)cc1F
CCc1ccccc1N(CC(=O)NC1CCCCC1)C(=O)Cc1ccc(C(=O)NO)cc1F
O=C(CN(C(=O)Cc1ccc(C(=O)NO)cc1F)c1ccccc1C(F)(F)F)NC1CCCCC1
Nc1ccccc1NC(=O)/C=C/c1ccc(-c2ncc(CNc3ccccc3)s2)cc1
Nc1ccccc1NC(=O)c1ccc(-c2ncc(CNc3ccccc3)s2)cc1
Nc1ccccc1NC(=O)c1ccc(CNC(=O)c2ccc(-c3ncc(CNc4ccccc4)s3)cc2)cc1
Nc1ccccc1NC(=O)c1ccc(NC(=O)c2ccc(-c3ncc(CNc4ccccc4)s3)cc2)cc1
Nc1ccccc1NC(=O)/C=C/c1ccc(CNC(=O)c2ccc(-c3ncc(CNc4ccccc4)s3)cc2)cc1
Nc1ccccc1NC(=O)CCCCCC(=O)Nc1ccc(-c2ncc(CNc3ccccc3)s2)cc1
Nc1ccccc1NC(=O)c1ccc(CNC(=O)c2ncc(CNc3ccccc3)s2)cc1
CCCNNC(=O)c1ccc(CNC(=O)c2ncc(CNc3ccccc3)s2)cc1
CCCNNC(=O)c1ccc(Nc2nccc(N(C)c3ccc4c(C)n(C)cc4c3)n2)cc1
NNC(=O)c1ccc(COc2ccccc2Cl)cc1
O=C(NO)c1ccc(Cn2cnc3c(Nc4ccc(F)c(Cl)c4)ncnc32)cc1
O=C(NO)c1ccc(Cn2cnc3c(Nc4ccc(Br)cc4F)ncnc32)cc1
COc1ccc(Nc2ncnc3c2ncn3Cc2ccc(C(=O)NO)cc2)cc1
Cc1noc(C)c1-c1ccc2n(CCCCCCC(=O)NO)cc(Cc3ccc(F)cc3)c2c1
Cn1c(CCCCCCC(=O)NO)nc2cc(ccc12)N(CCCl)CCCl
Nc1ncnc2c1ncn2Cc1ccc(-c2cn(CCCCCCC(=O)NO)nn2)cc1
O=C(NO)C1CCN(C[C@@H](O)COC(Cn2c3ccccc3c3ccccc32)Cn2c3ccccc3c3ccccc32)CC1
Nc1ccccc1NC(=O)c1ccc(CNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1
Nc1cc(F)ccc1NC(=O)c1ccc(CNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1
CC1=C(NCc2ccc(C(=O)Nc3ccccc3N)cc2)C(=O)c2ccccc2C1=O
CC1=C(NCCCCNC(=O)CS)C(=O)c2ccccc2C1=O
CN(Cc1ccccc1)C(=O)c1ccc(-c2noc(C(F)(F)F)n2)cc1
CCN(CC)CCCCNC(=O)c1ccc(-c2noc(C(F)(F)F)n2)cc1
CCN(CC)CCN(C)C(=O)c1ccc(-c2noc(C(F)(F)F)n2)cc1
O=C(NCCc1c[nH]c2ccccc12)c1ccc(-c2noc(C(F)(F)F)n2)cc1
CN(C(=O)c1ccc(-c2noc(C(F)(F)F)n2)cc1)c1ccccc1
CN(C)c1ccc(CNC(=O)c2ccc(-c3noc(C(F)(F)F)n3)cc2)cc1
O=C(Nc1cnc2ccccc2c1)c1ccc(-c2noc(C(F)(F)F)n2)cc1
O=C(NOCc1coc(-c2ccccc2)n1)c1ccc(-c2noc(C(F)(F)F)n2)cc1
O=C(NOCCN1CCCCC1)c1ccc(-c2noc(C(F)(F)F)n2)cc1
O=C(NOCCN1CCOCC1)c1ccc(-c2noc(C(F)(F)F)n2)cc1
COc1ncc(-c2cc(OCCCCCCC(=O)Nc3ccccc3N)c3ncnc(C)c3c2)cc1NS(=O)(=O)c1ccc(F)cc1F
COc1ncc(-c2cc(OCCCc3ccc(C(=O)Nc4ccccc4N)cc3)c3ncnc(C)c3c2)cc1NS(=O)(=O)c1ccc(F)cc1F
COC(=O)/C=C/c1ccc(CN(C(=O)OC(C)(C)C)C2CC2c2ccc(F)cc2)cc1
CC12CC3CC(C)(C1)CC(NC(=O)Nc1ccc(C(=O)NCCCCCC(=O)NO)cc1F)(C3)C2
CC12CC3CC(C)(C1)CC(NC(=O)Nc1ccc(C(=O)NCCCCCCC(=O)NO)cc1F)(C3)C2
CC12CC3CC(C)(C1)CC(NC(=O)Nc1ccc(C(=O)NCCCCC(=O)NO)cc1F)(C3)C2
CC12CC3CC(C)(C1)CC(NC(=O)Nc1ccc(C(=O)NCCCCC(=O)NO)cc1)(C3)C2
CC12CC3CC(C)(C1)CC(NC(=O)Nc1ccc(C(=O)NCCCCCC(=O)NO)cc1)(C3)C2
CC12CC3CC(C)(C1)CC(NC(=O)Nc1ccc(C(=O)NCCCCCCC(=O)NO)cc1)(C3)C2
O=C(CCNC(=O)[C@H]1CCCN(S(=O)(=O)c2ccc(NC(=O)Nc3ccc(OC(F)(F)F)cc3)c(F)c2)C1)NO
COc1cc(OC)c(/C=C/S(=O)(=O)Cc2ccc(OC)c(NC(=O)CCC(=O)NO)c2)c(OC)c1
COc1cc(OC)c(/C=C/S(=O)(=O)Cc2ccc(OC)c(NCC(=O)NO)c2)c(OC)c1
COc1ccc(cc1NCC(=O)O)CS(=O)(=O)/C=C/c2c(cc(cc2OC)OC)OC
O=C(Cc1ccc(C(=O)NO)cc1)Nc1ccc2ncnc(Nc3ccc(Br)c(F)c3)c2c1
O=C(COc1ccc2c(c1)OC1(CCN(Cc3cc(F)cc(F)c3)CC1)CC2=O)NO
O=C(COc1ccc2c(c1)OC1(CCN(Cc3cc(Cl)cc(Cl)c3)CC1)CC2=O)NO
Cc1ccccc1/C=C/C(=O)Nc1ccc(C(=O)NS(=O)(=O)c2ccc(NCCCCCCC(=O)NO)c([N+](=O)[O-])c2)c(Oc2ccccc2)c1
CN(c1ccccc1)c1ncc(NC(=O)CS)cn1
Cc1c2ccc(N(C)c3ccnc(Nc4ccc(NC(=O)CCCCCCC(=O)NO)cc4)n3)cc2nn1C
O=C(CCCCCCN1CCN(c2ccc(Nc3ncc(F)c(-c4cn(C5CCCC5)nn4)n3)cc2)CC1)NO
O=C(CS)Nc1ccc(Cn2c3c(c4ccccc42)CS(=O)(=O)CC3)cc1
C[C@H](NC(=O)[C@H](CC(=O)NCC(C)(C)C)NC(=O)CCC(=O)Nc1ccc(C(=O)NO)cc1)C(=O)NCc1ccc(F)cc1F
C[C@H](NC(=O)[C@H](CC(=O)NCC(C)(C)C)NC(=O)CCCCCCC(=O)NO)C(=O)NCc1ccc(F)cc1F
C[C@H](NC(=O)[C@H](CC(=O)NCC(C)(C)C)NC(=O)c1ccc(C(=O)NO)cc1)C(=O)NCc1ccc(F)cc1F
C[C@H](NC(=O)[C@H](CC(=O)NCC(C)(C)C)NC(=O)c1ccc(/C=C/C(=O)NO)cc1)C(=O)NCc1ccc(F)cc1F
C[C@H](NC(=O)[C@H](CC(=O)NCC(C)(C)C)NC(=O)c1c[nH]c2ccccc12)C(=O)NCc1ccc(F)cc1F
O=C(CCc1ccc(-c2sc3cc(O)ccc3c2C(=O)c2ccc(OCCN3CCCCC3)cc2)cc1)NO
O=C(CCCCc1ccc(-c2sc3cc(O)ccc3c2C(=O)c2ccc(OCCN3CCCCC3)cc2)cc1)NO
O=C(CCCCCc1ccc(-c2sc3cc(O)ccc3c2C(=O)c2ccc(OCCN3CCCCC3)cc2)cc1)NO
O=C(CCCCCCc1ccc(-c2sc3cc(O)ccc3c2C(=O)c2ccc(OCCN3CCCCC3)cc2)cc1)NO
O=C(CCCOc1ccc(-c2sc3cc(O)ccc3c2C(=O)c2ccc(OCCN3CCCCC3)cc2)cc1)NO
O=C(CCCCOc1ccc(-c2sc3cc(O)ccc3c2C(=O)c2ccc(OCCN3CCCCC3)cc2)cc1)NO
O=C(CCCCCOc1ccc(-c2sc3cc(O)ccc3c2C(=O)c2ccc(OCCN3CCCCC3)cc2)cc1)NO
O=C(NO)c1ccc(NCc2cc(-c3cccc(Cl)c3)cn3ccnc23)cc1
O=C(NO)c1ccc(NCc2cc(-c3cccc(Br)c3)cn3ccnc23)cc1
Cc1ccc(-c2cc(C(=O)NCc3ccc(C(=O)NO)cc3)c3nccn3c2)cc1
O=C(NO)c1ccc(CNC(=O)c2cc(-c3ccc(F)cc3)cn3ccnc23)cc1
Cc1cccc(-c2cc(C(=O)NCc3ccc(C(=O)NO)cc3)c3nccn3c2)c1
Cc1ccccc1-c1cc(C(=O)NCc2ccc(C(=O)NO)cc2)c2nccn2c1
C=C1C(=O)N(C)[C@H](C)[C@H](O)N1C(=O)/C=C/C=C[C@@H](CO)[C@H](O)[C@H](C)CCC
C#CCN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NO)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NO)cc1
O=C1CNC(=O)/C(=C/c2ccc(C(=O)NO)cc2)N1
C#CCN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCCCCCCCC(=O)NO)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCCCCCCC(=O)NO)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCCC(=O)NO)cc1
C#CCN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)Nc2ccc(C(=O)NO)cc2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)Nc2ccc(C(=O)NO)cc2)cc1
C#CCN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCc2ccc(C(=O)NO)cc2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCc2ccc(C(=O)NO)cc2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(NCc2ccc(C(=O)NO)cc2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(OCc2ccc(C(=O)NO)cc2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(OCC(=O)NO)cc1
C#CCN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)Nc2cccc(C(=O)NO)c2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)Nc2cccc(C(=O)NO)c2)cc1
C#CCN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCc2cccc(C(=O)NO)c2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCc2cccc(C(=O)NO)c2)cc1
C#CCN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCCNC(=O)c2ccc(C(=O)NO)cc2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCCNC(=O)c2ccc(C(=O)NO)cc2)cc1
C#CCN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCCCNC(=O)c2ccc(C(=O)NO)cc2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(C(=O)NCCCNC(=O)c2ccc(C(=O)NO)cc2)cc1
CN1C(=O)CNC(=O)/C1=C/c1ccc(/C=C/C(=O)NO)cc1
Cc1cc(/C=C/C(=O)NO)ccc1/C=C1/C(=O)NCC(=O)N1C
Cc1cc(/C=C2/C(=O)NCC(=O)N2C)ccc1/C=C/C(=O)NO
CCOc1cc(/C=C2/C(=O)NCC(=O)N2C)ccc1/C=C/C(=O)NO
COc1cc(/C=C2/C(=O)NCC(=O)N2C)ccc1/C=C/C(=O)NO
CN1C(=O)CNC(=O)/C1=C/c1ccc(/C=C/C(=O)NO)cc1F
CN1C(=O)CNC(=O)/C1=C/c1ccc(/C=C/C(=O)NO)cc1C(F)(F)F
CN1C(=O)CNC(=O)/C1=C/c1ccc(N(C)C)c(/C=C/C(=O)NO)c1
CN1C(=O)CNC(=O)/C1=C/c1ccc(-c2ccc(/C=C/C(=O)NO)cc2)cc1
COc1ccc(CN2[C@H](C(=O)NCc3ccc(C(=O)NO)cc3)Cc3c([nH]c4ccccc34)[C@H]2C2CC2)cc1
O=C(NO)c1ccc(CNC(=O)[C@@H]2Cc3c([nH]c4ccccc34)[C@@H](C3CC3)N2Cc2ccccc2)cc1
COc1ccc(CN2[C@H](C)c3[nH]c4ccccc4c3C[C@H]2C(=O)NCc2ccc(C(=O)NO)cc2)cc1
O=C(NO)c1ccc(CNC(=O)[C@@H]2Cc3c([nH]c4ccccc34)[C@@H](C3CC3)N2Cc2ccc(Cl)cc2)cc1
O=C(NO)c1ccc(CNC(=O)[C@@H]2Cc3c([nH]c4ccccc34)[C@@H](c3ccc(Cl)cc3)N2CC2CC2)cc1
O=C(NO)c1ccc(CNC(=O)[C@@H]2Cc3c([nH]c4ccccc34)[C@@H](c3ccc(Cl)cc3)N2)cc1
COc1ccc([C@H]2N[C@H](C(=O)NCc3ccc(C(=O)NO)cc3)Cc3c2[nH]c2ccccc32)cc1OC
O=C(NO)c1ccc(CNC(=O)[C@@H]2Cc3c([nH]c4ccccc34)[C@@H](c3ccccc3)N2)cc1
O=C(NO)c1ccc(CNC(=O)[C@@H]2Cc3c([nH]c4ccccc34)[C@@H](C3CC3)N2)cc1
O=C(NO)c1ccc(CNC(=O)[C@@H]2Cc3c([nH]c4ccccc34)[C@@H](C3CCCC3)N2)cc1
O=C(NO)c1ccc(CNC(=O)[C@@H]2Cc3c([nH]c4ccccc34)[C@@H](c3ccc4c(c3)OCO4)N2)cc1
CCN(CC)Cc1ccccc1CNC(=O)c1cccc(NC(=O)c2cccc(NC(=O)CCCCCCC(=O)NO)c2)c1
CCN(CC)Cc1ccccc1CNC(=O)c1cccc(NC(=O)c2cccc(C(=O)NO)c2)c1
O=C(NO)c1ccc(CC(=O)N2CCc3c([nH]c4ccccc34)C2)cc1
O=C(CCCCCC(=O)N1CCc2c([nH]c3ccccc23)C1)NO
O=C(CCCCCCC(=O)N1CCc2c([nH]c3ccccc23)C1)NO
O=C(NO)c1ccc(CN2CCc3c([nH]c4ccccc34)C2)cc1
COc1ccc2[nH]c3c(c2c1)CCN(Cc1ccc(C(=O)NO)cc1)C3
COc1ccc2[nH]c3c(c2c1)CCN(Cc1ccc(/C=C/C(=O)NO)cc1)C3
O=C(NO)c1ccc(CN2CCc3c(n(CC4CC4)c4ccc(F)cc34)C2)cc1
O=C(NO)c1ccc(C2NCCc3c2[nH]c2ccccc32)cc1
O=C(NO)c1ccc(C2c3[nH]c4ccccc4c3CCN2Cc2ccccc2)cc1
O=C(NO)c1ccc(CN2CCc3[nH]c4ccccc4c3C2)cc1
O=C(NO)c1cccc(CN2CCc3[nH]c4ccccc4c3C2)c1
O=C(/C=C/c1ccc(CN2CCc3[nH]c4ccccc4c3C2)cc1)NO
O=C(NO)c1ccc(CN2CCc3[nH]c4ccc(F)cc4c3C2)cc1
Cc1ccc2[nH]c3c(c2c1)CN(Cc1ccc(C(=O)NO)cc1)CC3
COc1ccc(CN2[C@@H](C(=O)NCc3ccc(C(=O)NO)cc3)Cc3c([nH]c4ccccc34)[C@@H]2C2CC2)cc1
Cn1c2c(c3ccccc31)CN(Cc1ccc(C(=O)NO)cc1)CC2
Cn1c2c(c3ccccc31)CN(C(=O)NCc1ccc(C(=O)NO)cc1)CC2
O=C(NO)c1ccc(CN2CCc3c(c4ccccc4n3Cc3ccccc3)C2)cc1
O=C(NO)c1ccc(CNC(=O)N2CCc3c(c4ccccc4n3Cc3ccccc3)C2)cc1
O=C(NO)c1ccc(CNC(=S)N2CCc3c(c4ccccc4n3Cc3ccccc3)C2)cc1
O=C(NO)c1ccc(COC(=O)N2CCc3c(c4ccccc4n3Cc3ccccc3)C2)cc1
CCN(CC)Cc1ccc(Cn2c3c(c4ccccc42)CN(C(=O)NCc2ccc(C(=O)NO)cc2)CC3)cc1
Cn1c2c(c3ccccc31)CN(C(=O)OCc1ccc(C(=O)NO)cc1)CC2
O=C(NO)c1ccc(CC(=O)N2CCc3c(c4ccccc4n3Cc3ccccc3)C2)cc1
O=C(NO)c1ccc(C(=O)N2CCc3c(c4ccccc4n3Cc3ccccc3)C2)cc1
O=C(NO)c1ccc(NC(=O)N2CCc3c(c4ccccc4n3Cc3ccccc3)C2)cc1
O=C(CS)Nc1ccc(CN2CCc3c(c4ccccc4n3Cc3ccccc3)C2)cc1
O=C(CS)Nc1ccc(CNC(=O)N2CCc3c(c4ccccc4n3Cc3ccccc3)C2)cc1
O=C(CS)NCCCCCNC(=O)N1CCc2c(c3ccccc3n2Cc2ccccc2)C1
O=C(NO)c1cccc(CN2CCc3c(c4ccccc4n3Cc3ccccc3)C2)c1
O=C(NO)c1cccc(CNC(=O)N2CCc3c(c4ccccc4n3Cc3ccccc3)C2)c1
O=C(NCC[Se][Se]CCNC(=O)/C(Cc1ccc(Br)s1)=N/O)/C(Cc1ccc(Br)s1)=N/O
O=C(NCC[Se][Se]CCNC(=O)/C(Cc1ccsc1)=N/O)/C(Cc1ccsc1)=N/O
O=C(NCC[Se][Se]CCNC(=O)/C(Cc1ccc(O)c(Br)c1)=N/O)/C(Cc1ccc(O)c(Br)c1)=N/O
O=C(CCCCCCCN1C(=O)[C@@H]2CCC(=O)N2Cc2ccccc21)NO
O=C(CCCCCCCN1C(=O)[C@@H]2CCCN2Cc2ccccc21)NO
COc1cc2c(cc1OCc1ccccc1)CN1C(=O)CC[C@H]1C(=O)N2CCCCCCCC(=O)NO
COc1cc2c(cc1O)CN1C(=O)CC[C@H]1C(=O)N2CCCCCCCC(=O)NO
O=C(CCCCCN1C(=O)[C@@H]2CCCN2Cc2ccccc21)NO
COc1cc2c(cc1OCc1ccccc1)CN1C(=O)CC[C@H]1C(=O)N2CCCCCC(=O)NO
COc1cc2c(cc1O)CN1C(=O)CC[C@H]1C(=O)N2CCCCCC(=O)NO
O=C(CCCCCCN1C(=O)[C@@H]2CCCN2Cc2ccccc21)NO
COc1cc2c(cc1OCc1ccccc1)CN1C(=O)CC[C@H]1C(=O)N2CCCCCCC(=O)NO
COc1cc2c(cc1O)CN1C(=O)CC[C@H]1C(=O)N2CCCCCCC(=O)NO
O=C(NO)c1ccc(CN2C(=O)[C@@H]3CCCN3Cc3ccccc32)cc1
COc1cc2c(cc1OCc1ccccc1)CN1C(=O)CC[C@H]1C(=O)N2Cc1ccc(C(=O)NO)cc1
COc1cc2c(cc1O)CN1C(=O)CC[C@H]1C(=O)N2Cc1ccc(C(=O)NO)cc1
O=C(Cc1ccc(CN2C(=O)[C@@H]3CCCN3Cc3ccccc32)cc1)NO
COc1cc2c(cc1OCc1ccccc1)CN1C(=O)CC[C@H]1C(=O)N2Cc1ccc(CC(=O)NO)cc1
COc1cc2c(cc1O)CN1C(=O)CC[C@H]1C(=O)N2Cc1ccc(CC(=O)NO)cc1
O=C(NO)c1ccccc1CN1C(=O)[C@@H]2CCCN2Cc2ccccc21
COc1cc2c(cc1OCc1ccccc1)CN1C(=O)CC[C@H]1C(=O)N2Cc1ccccc1C(=O)NO
COc1cc2c(cc1O)CN1C(=O)CC[C@H]1C(=O)N2Cc1ccccc1C(=O)NO
O=C(NO)c1cccc(CN2C(=O)[C@@H]3CCCN3Cc3ccccc32)c1
COc1cc2c(cc1OCc1ccccc1)CN1C(=O)CC[C@H]1C(=O)N2Cc1cccc(C(=O)NO)c1
COc1cc2c(cc1O)CN1C(=O)CC[C@H]1C(=O)N2Cc1cccc(C(=O)NO)c1
CN(C)CCCn1c(SCc2ccc(/C=C/C(=O)NO)cc2)nc2ccccc21
N#CC1(CNc2cccc(-c3cc(Nc4cnn(CCCCCCC(=O)NO)c4)ncc3Cl)n2)CCOCC1
N#CC1(CNc2cccc(-c3cc(Nc4cnn(CCCCCC(=O)NO)c4)ncc3Cl)n2)CCOCC1
N#CC1(CNc2cccc(-c3cc(Nc4cnn(Cc5ccc(C(=O)NO)cc5)c4)ncc3Cl)n2)CCOCC1
N#CC1(CNc2cccc(-c3cc(Nc4cnn(CCCCCCC(=O)Nc5ccccc5N)c4)ncc3Cl)n2)CCOCC1
N#CC1(CNc2cccc(-c3cc(Nc4cnn(CCCCCC(=O)Nc5ccccc5N)c4)ncc3Cl)n2)CCOCC1
N#CC1(CNc2cccc(-c3cc(Nc4cnn(Cc5ccc(C(=O)Nc6ccccc6N)cc5)c4)ncc3Cl)n2)CCOCC1
CCCCNNC(=O)c1ccc(Cn2cc(Nc3cc(-c4cccc(NCC5(C#N)CCOCC5)n4)c(Cl)cn3)cn2)cc1
O=C(CCCCCCn1cc(Nc2cc(-c3cccc(NCC4CCOCC4)n3)c(Cl)cn2)cn1)NO
O=C(CCCCCn1cc(Nc2cc(-c3cccc(NCC4CCOCC4)n3)c(Cl)cn2)cn1)NO
O=C(NO)c1ccc(Cn2cc(Nc3cc(-c4cccc(NCC5CCOCC5)n4)c(Cl)cn3)cn2)cc1
O=C(CCCCCCn1cc(Nc2cc(-c3cccc(NCc4cccc(F)c4)n3)c(Cl)cn2)cn1)NO
O=C(CCCCCn1cc(Nc2cc(-c3cccc(NCc4cccc(F)c4)n3)c(Cl)cn2)cn1)NO
O=C(NO)c1ccc(Cn2cc(Nc3cc(-c4cccc(NCc5cccc(F)c5)n4)c(Cl)cn3)cn2)cc1
COc1cc(F)ccc1-c1cc(Nc2cnn(CCCCCCC(=O)NO)c2)ncc1F
COc1cc(F)ccc1-c1cc(Nc2cnn(CCCCCC(=O)NO)c2)ncc1F
COc1cc(F)ccc1-c1cc(Nc2ccc(NC(=O)CCCCCCC(=O)NO)cc2)ncc1F
COc1cc(F)ccc1-c1cc(Nc2ccc(/C=C/C(=O)Nc3ccccc3N)cc2)ncc1F
COc1cc(F)ccc1-c1cc(Nc2cnn(CCCCCC(=O)Nc3ccccc3N)c2)ncc1F
COc1cc(F)ccc1-c1cc(Nc2ccc(NC(=O)CCCCCCC(=O)Nc3ccccc3N)cc2)ncc1F
O=C(CCCCCCn1cc(Nc2ncc(Cl)c(-c3cnc4ccccn34)n2)cn1)NO
O=C(CCCCCn1cc(Nc2ncc(Cl)c(-c3cnc4ccccn34)n2)cn1)NO
CCCNNC(=O)CCCCCCn1cc(Nc2ncc(Cl)c(-c3cnc4ccccn34)n2)cn1
CCCNNC(=O)CCCCCn1cc(Nc2ncc(Cl)c(-c3cnc4ccccn34)n2)cn1
CCCNNC(=O)c1ccc(Cn2cc(Nc3ncc(Cl)c(-c4cnc5ccccn45)n3)cn2)cc1
CCCNNC(=O)c1ccc(Cn2cc(Nc3ncc(Cl)c(-c4cnc5ccc(-c6ccccc6)cn45)n3)cn2)cc1
CCCNNC(=O)CCCCCn1cc(Nc2ncc(Cl)c(-c3cnc4ccc(-c5ccccc5)cn34)n2)cn1
O=C(CCCCCCn1cc(Nc2ncc(Cl)c(OC3CCCCC3)n2)cn1)NO
O=C(CCCCCn1cc(Nc2ncc(Cl)c(OC3CCCCC3)n2)cn1)NO
O=C(/C=C/c1ccc(Nc2ncc(Cl)c(OC3CCCCC3)n2)cc1)NO
O=C(NO)c1ccc(Cn2cc(Nc3ncc(Cl)c(OC4CCCCC4)n3)cn2)cc1
O=C(CCCCCCC(=O)Nc1ccc(Nc2ncc(Cl)c(OC3CCCCC3)n2)cc1)NO
O=C(CCCC(=O)Nc1ccc(Nc2ncc(Cl)c(OC3CCCCC3)n2)cc1)NO
CCCCNNC(=O)CCCCCCC(=O)Nc1ccc(Nc2ncc(Cl)c(OC3CCCCC3)n2)cc1
CCCCN(CCc1c(C)[nH]c2ccccc12)Cc1ccc(/C=C/C(=O)NNCCC)cc1
CN1C(=O)N2Cc3c(c4cc(OCCN5CCOCC5)ccc4n3Cc3ccc(C(=O)NO)cc3)C(c3ccccc3)(C2)C1=O
CN1C(=O)N2Cc3c(c4cc(OCCN5CCOCC5)ccc4n3Cc3ccc(C(=O)NO)cc3)[C@@](c3ccccc3)(C2)C1=O
CN1C(=O)N2Cc3c(c4ccccc4n3Cc3ccc(C(=O)NO)cc3)C(c3ccccc3)(C2)C1=O
CN1C(=O)N2Cc3c(c4ccccc4n3Cc3ccc(C(=O)NO)cc3)[C@@](c3ccccc3)(C2)C1=O
CN1C(=O)N2Cc3c(c4cc(OCCN5CCOCC5)ccc4n3Cc3ccc(C(=O)NO)cc3)C(C)(C2)C1=O
C[C@@]12CN(Cc3c1c4cc(ccc4n3Cc5ccc(cc5)C(=O)NO)OCCN6CCOCC6)C(=O)N(C2=O)C
CN1C(=O)N2Cc3c(c4cc(OCCN5CCOCC5)ccc4n3Cc3ccc(C(=O)NO)cc3)[C@](C)(C2)C1=O
CN1C(=O)N2Cc3c(c4cc(OCCN5CCOCC5)ccc4n3Cc3ccc(C(=O)NO)cc3)C(C3CCCCC3)(C2)C1=O
CN1C(=O)N2Cc3c(c4cc(OCCN5CCOCC5)ccc4n3Cc3ccc(C(=O)NO)cc3)C(c3ccco3)(C2)C1=O
CN1C(=O)N2Cc3c(c4cc(O)ccc4n3Cc3ccc(C(=O)NO)cc3)C(c3cccs3)(C2)C1=O
COc1ccc2c(ccn2S(=O)(=O)c2ccc(C(=O)NO)cc2)c1
O=C(NO)c1ccc(S(=O)(=O)n2ccc3cc(OCc4ccccc4)ccc32)cc1
O=C(NO)c1ccc(S(=O)(=O)n2ccc3cc(OCCCN4CCCCC4)ccc32)cc1
C#CCN1CCN(CCCOc2ccc3c(ccn3S(=O)(=O)c3ccc(C(=O)NO)cc3)c2)CC1
COc1ccc2c(ccn2S(=O)(=O)c2ccc(C(=O)NN)cc2)c1
NNC(=O)c1ccc(S(=O)(=O)n2ccc3cc(OCc4ccccc4)ccc32)cc1
NNC(=O)c1ccc(S(=O)(=O)n2ccc3cc(OCCCN4CCCCC4)ccc32)cc1
C#CCN1CCN(CCCOc2ccc3c(ccn3S(=O)(=O)c3ccc(C(=O)NN)cc3)c2)CC1
CCCNNC(=O)c1ccc(S(=O)(=O)n2ccc3cc(OC)ccc32)cc1
CCCN(CCC)NC(=O)c1ccc(S(=O)(=O)n2ccc3cc(OC)ccc32)cc1
CCCNNC(=O)c1ccc(S(=O)(=O)n2ccc3cc(OCCCN4CCCCC4)ccc32)cc1
C#CCN1CCN(CCCOc2ccc3c(ccn3S(=O)(=O)c3ccc(C(=O)NNCCC)cc3)c2)CC1
Nc1ccccc1NC(=O)c1ccc(S(=O)(=O)n2ccc3cc(OCc4ccccc4)ccc32)cc1
Nc1ccccc1NC(=O)c1ccc(S(=O)(=O)n2ccc3cc(OCCCN4CCCCC4)ccc32)cc1
C#CCN1CCN(CCCOc2ccc3c(ccn3S(=O)(=O)c3ccc(C(=O)Nc4ccccc4N)cc3)c2)CC1
CN(CC#C)Cc1cc2cc(OCCCN3CCCCC3)ccc2n1C
CCc1c(C#N)c(SC(C(N)=O)c2ccccc2)nc(N(C)C2CCN(c3ncc(C(=O)NO)cn3)CC2)c1C#N
CCc1c(C#N)c(S[C@@H](C(N)=O)c2ccccc2)nc(N2CCC(CNCc3ccc(/C=C/C(=O)NO)cc3)CC2)c1C#N
CNC(=O)c1ccccc1Nc1nc(Nc2ccc(NC(=O)CCCCCCC(=O)NO)cc2)ncc1Cl
Nc1ccn(Cc2ccc(-c3cn(CCCCCCC(=O)NO)nn3)cc2)c(=O)n1
COc1ccc2c3ccnc(C)c3n(CC3CCN(c4ncc(C(=O)NO)cn4)CC3)c2c1
COc1ccc(-c2cc(-c3ccc(C(C)C)cc3)cnc2NCc2ccc(C(=O)NO)cc2)cc1
O=C(Cc1ccc(C(=O)NO)cc1)Nc1ccc2ncnc(Nc3ccc(Cl)c(F)c3)c2c1
O=C(Cc1ccc(C(=O)NO)cc1)Nc1ccc2ncnc(Nc3ccc(I)cc3)c2c1
COc1cc(OCCCCCCC(=O)NO)ccc1C1c2ccc(O)cc2CCN1CC(C)(C)F
COc1ccc(-c2ccc(C(=O)N3CCc4c(cc(Cl)c(C(=O)NO)c4Cl)C3)cc2)cc1
O=C(NO)c1c(Cl)cc2c(c1Cl)CCN(C(=O)c1cc3ccccc3[nH]1)C2
CC(C)(C)c1nc(-c2cccc(NS(=O)(=O)c3c(F)cccc3F)c2F)c(-c2ccnc(NCCCCCCC(=O)NO)n2)s1
O=C(CCCCCCNc1nccc(-c2sc(-c3ccccc3)nc2-c2cccc(NS(=O)(=O)c3c(F)cccc3F)c2F)n1)NO
CC(C)(C)OC(=O)Nc1cccc(c1)-c1cc(no1)C(=O)NCCCCCCC(=O)NO
O=C(/C=C/c1ccc2nn(Cc3ccc(Cl)cc3)cc2c1)NO
CNCCOc1ccc(-c2cc(=O)c3cc(OCCCCCC(=O)NO)cc(O)c3o2)cc1
O=C(NO)c1ccc(CNc2ncnc3[nH]ccc23)cc1
Cn1cc(CCCC(=O)Nc2ccc(C(=O)NO)cc2)c2ccccc21
Cc1ccc(Cn2cnc3cc(/C=C/C(=O)NO)ccc3c2=O)cc1
O=C(/C=C/c1ccc2c(=O)n(Cc3ccc(Cl)cc3)cnc2c1)NO
O=C(NO)c1ccc(CNc2cccc3cc(-c4cccnc4)cnc23)cc1
O=C(NO)c1ccc(CNc2cccc3cc(-c4ccncc4)cnc23)cc1
ONC(=O)CCCCCCC(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1
C=C[C@@]1(C)CC[C@H](C(=C)CN2CCN(C(=O)CCCCCCC(=O)NO)CC2)C[C@@H]1C(=C)Cn1cccn1
C=C[C@]1(C)CC[C@@H](C(=C)Cn2cccn2)C[C@H]1C(=C)CN1CCN(C(=O)CCCCCCC(=O)NO)CC1
COc1ccc(-c2cn(CCCCCC(=O)NO)c(C)c2C(C)=O)cc1
CC(=O)c1c(-c2ccc([N+](=O)[O-])cc2)cn(CCCCCC(=O)NO)c1C
COc1cc(/C=C/C(=O)CC(=O)/C=C/c2ccc(/C=C/C(=O)NO)cc2)ccc1O
COc1cc(/C=C/C(=O)c2ccc(OCCCCCC(=O)NO)cc2)cc(OC)c1OC
C[C@@H]1CC[C@H]2[C@@H](C)C(OCC(=O)NO)C[C@@H]3O[C@]4(C)CC[C@@H]1[C@]32OO4
C[C@@H]1CC[C@H]2[C@@H](C)C(SCCC(=O)NO)C[C@@H]3O[C@]4(C)CC[C@@H]1[C@]32OO4
O=C(CCCc1ccc(N(CCCl)CCCl)cc1)NO
Cc1nc(C)c(C(=O)Nc2cccc(C(=O)NO)c2)nc1C
C[C@]12CC[C@H](OC(=O)CCCCCC(=O)NO)CC1=CCC1C2CC[C@]2(C)C(c3cccnc3)=CCC12
O=C(CCCCCn1c(=O)c(-c2ccc(Cl)cc2Cl)cc2cnc(NC3CC3)nc21)NO
C[C@@H]1CN(Cc2ccc(C(=O)NO)cc2)C[C@H]1c1nc2c(cnn2C2CCOCC2)c(=O)[nH]1
CC(C)NC(=O)[C@H]1CC[C@@H](n2/c(=N/C(=O)c3ccccc3)[nH]c3cc(/C=C/C(=O)NO)ccc32)CC1
CC(C)(C)NC(=O)CN(Cc1ccc(C(=O)NO)cc1)C(=O)c1cc2ccccc2[nH]1
CC(C)(C)NC(=O)CN(Cc1ccc(C(=O)NO)cc1)C(=O)c1ccc2ccccc2n1
CC(C)(C)NC(=O)CN(Cc1ccc(C(=O)NO)cc1)C(=O)c1nccc2ccccc12
CC(C)(C)NC(=O)CN(Cc1ccc(C(=O)NO)cc1)C(=O)c1c[nH]c2ccccc12
Cn1c(C(=O)N(CC(=O)NC(C)(C)C)Cc2ccc(C(=O)NO)cc2)cc2ccccc21
Cn1cc(C(=O)N(CC(=O)NC(C)(C)C)Cc2ccc(C(=O)NO)cc2)c2ccccc21
Cn1cc(C(=O)N(CC(=O)NC(C)(C)C)Cc2ccc(C(=O)NO)cc2)c2ncccc21
O=C(CN(Cc1ccc(C(=O)NO)cc1)C(=O)c1c[nH]c2ccccc12)NCc1ccccc1
Cn1cc(C(=O)N(CC(=O)NCc2ccccc2)Cc2ccc(C(=O)NO)cc2)c2ccccc21
O=C(CN(Cc1ccc(C(=O)NO)cc1)C(=O)c1cc2ccccc2[nH]1)NCc1ccccc1
O=C(CN(Cc1ccc(C(=O)NO)cc1)C(=O)c1c[nH]c2ccccc12)NC1CCCCC1
Cn1cc(C(=O)N(CC(=O)NC2CCCCC2)Cc2ccc(C(=O)NO)cc2)c2ccccc21
O=C(CN(Cc1ccc(C(=O)NO)cc1)C(=O)c1cc2ccccc2[nH]1)NC1CCCCC1
O=C(CN(Cc1ccc(C(=O)NO)cc1)C(=O)c1c[nH]c2ccccc12)NC1CCCC1
CC(C)(C)CC(C)(C)NC(=O)CN(Cc1ccc(C(=O)NO)cc1)C(=O)c1c[nH]c2ccccc12
COC(=O)CNC(=O)CN(Cc1ccc(C(=O)NO)cc1)C(=O)c1cc2ccccc2[nH]1
O=C(CCCCCCCCCCCc1cccc(O)c1)NO
C=C(c1ccc(OC)c(OC(C)C(=O)NO)c1)c1cc(C)nc2ccccc12
C=C(c1ccc(OC)c(OC(F)C(=O)NO)c1)c1cc(C)nc2ccccc12
COc1cc(-c2nc(C(=O)NCc3ccc(C(=O)NO)cc3)cc3c2[nH]c2ccccc23)cc(OC)c1OC
CN1CCC2c3ccccc3N(Cc3ccc(C(=O)NO)cc3)C2C1
COc1cc2c(cc1OCc1ccc(C(=O)Nc3ccccc3N)cc1)CC[C@@H]1[C@H]3CC[C@@H](O)[C@]3(C)CC[C@@H]21
Nc1nc(Cl)c2ccn(Cc3ccc(-c4noc(C(F)(F)F)n4)cc3)c2n1
Nc1nc(Cl)c2ncn(Cc3ccc(-c4noc(C(F)(F)F)n4)cc3)c2n1
Nc1nc(Cl)c2ccn(Cc3ccc(-c4noc(C(F)(F)F)n4)cc3F)c2n1
Nc1nc(Cl)c2ncn(Cc3ccc(-c4noc(C(F)(F)F)n4)cc3F)c2n1
Nc1nc(Cl)c2ccn(Cc3ccc(-c4noc(C(F)(F)F)n4)c(F)c3)c2n1
Nc1nc(Cl)c2ncn(Cc3ccc(-c4noc(C(F)(F)F)n4)c(F)c3)c2n1
FC(F)(F)c1nc(-c2ccc(Cn3cnc4c(Cl)ncnc43)cc2)no1
Fc1cc(-c2noc(C(F)(F)F)n2)ccc1Cn1cnc2c(Cl)ncnc21
Fc1cc(Cn2cnc3c(Cl)ncnc32)ccc1-c1noc(C(F)(F)F)n1
Nc1nc(Cl)c2ncn(Cc3ccc(-c4noc(C(F)(F)F)n4)c(Cl)c3)c2n1
Nc1nc(Cl)c2ccn(Cc3ccc(C(=O)NO)cc3)c2n1
Nc1nc(Cl)c2ncn(Cc3ccc(C(=O)NO)cc3)c2n1
Nc1ncc2ncn(Cc3ccc(C(=O)NO)cc3)c2n1
Nc1nc(Cl)c2ccn(Cc3ccc(C(=O)NO)cc3F)c2n1
Nc1nc(Cl)c2ncn(Cc3ccc(C(=O)NO)cc3F)c2n1
Nc1ncc2ncn(Cc3ccc(C(=O)NO)cc3F)c2n1
O=C(NO)c1ccc(Cn2cnc3c(Cl)ncnc32)c(F)c1
O=C(NO)c1ccc(Cn2cnc3c(Cl)ncnc32)cc1
Nc1nc(Cl)c2ccn(Cc3ccc(C(=O)NO)cn3)c2n1
Nc1nc(Cl)c2ncn(Cc3ccc(C(=O)NO)cn3)c2n1
Nc1nc(Cl)c2ccn(Cc3ccc(CC(=O)NO)cc3)c2n1
Nc1nc(Cl)c2ncn(Cc3ccc(CC(=O)NO)cc3)c2n1
Nc1nc(Cl)c2ccn(Cc3nc(C(=O)NO)co3)c2n1
Nc1nc(Cl)c2ccn(Cc3ccc(NC(=O)CS)cc3)c2n1
Nc1nc(Cl)c2ncn(Cc3ccc(NC(=O)CS)cc3)c2n1
Nc1nc(Cl)c2ncn(Cc3ccc(CNC(=O)CS)cc3)c2n1
Nc1nc(Cl)c2ccn(Cc3cccc(-c4noc(C(F)(F)F)n4)c3)c2n1
Nc1nc(Cl)c2ncn(Cc3cccc(-c4noc(C(F)(F)F)n4)c3)c2n1
COc1ccc([C@@H]2N[C@@H](C(=O)NCc3ccc(C(=O)NO)cc3)Cc3c2[nH]c2ccccc32)cc1
COc1ccc([C@H]2N[C@H](C(=O)NCc3ccc(C(=O)NO)cc3)Cc3c2[nH]c2ccccc32)cc1
COc1ccc(CN2[C@@H](C(=O)NCc3ccc(C(=O)NO)cc3)Cc3c([nH]c4ccccc34)[C@@H]2C)cc1
O=C(NO)c1ccc(CNC(=O)[C@H]2Cc3c([nH]c4ccccc34)[C@H](C3CC3)N2Cc2ccc(Cl)cc2)cc1
O=C(NO)c1ccc(CNC(=O)[C@H]2Cc3c([nH]c4ccccc34)[C@H](c3ccc(Cl)cc3)N2CC2CC2)cc1
O=C(NO)c1ccc(CNC(=O)[C@H]2Cc3c([nH]c4ccccc34)[C@H](c3ccc(Cl)cc3)N2)cc1
COc1ccc([C@@H]2N[C@@H](C(=O)NCc3ccc(C(=O)NO)cc3)Cc3c2[nH]c2ccccc32)cc1OC
O=C(NO)c1ccc(CNC(=O)[C@H]2Cc3c([nH]c4ccccc34)[C@H](c3ccccc3)N2)cc1
O=C(NO)c1ccc(CNC(=O)[C@H]2Cc3c([nH]c4ccccc34)[C@H](C3CC3)N2)cc1
O=C(NO)c1ccc(CNC(=O)[C@H]2Cc3c([nH]c4ccccc34)[C@H](C3CCCC3)N2)cc1
CCCNNC(=O)c1ccc(CNC(=O)[C@H](CC(C)C)NC(=O)[C@@H](O)[C@H](N)Cc2ccccc2)cc1
CC(C)C[C@H](NC(=O)[C@@H](O)[C@H](N)Cc1ccccc1)C(=O)NCc1ccc(C(=O)NO)cc1
O=C(NO)c1ccc2nc[nH]c2c1
O=C(NO)c1ccc2nc(CCc3ccccc3)[nH]c2c1
O=C(NO)c1ccc2[nH]c(CNc3ccccc3)nc2c1
Cn1c(CNc2ccccc2)nc2cc(C(=O)NO)ccc21
CCn1c(CNc2ccccc2)nc2cc(C(=O)NO)ccc21
CC(C)n1c(CNc2ccccc2)nc2cc(C(=O)NO)ccc21
O=C(NO)c1ccc2c(c1)nc(CNc1ccccc1)n2C1CC1
Cn1c(CSc2ccccc2)nc2cc(C(=O)NO)ccc21
Cn1c(COc2ccccc2)nc2cc(C(=O)NO)ccc21
Cn1c(CN2CCC3(CC2)OCCO3)nc2cc(C(=O)NO)ccc21
Cn1c(CN2CCCCC2)nc2cc(C(=O)NO)ccc21
Cn1c(CNc2cccc3ccccc23)nc2cc(C(=O)NO)ccc21
Cc1ccccc1NCc1nc2cc(C(=O)NO)ccc2n1C
Cc1cccc(NCc2nc3cc(C(=O)NO)ccc3n2C)c1
Cc1ccc(NCc2nc3cc(C(=O)NO)ccc3n2C)cc1
Cn1c(CNc2ccccc2F)nc2cc(C(=O)NO)ccc21
Cn1c(CNc2cccc(F)c2)nc2cc(C(=O)NO)ccc21
Cn1c(CNc2ccc(F)cc2)nc2cc(C(=O)NO)ccc21
CN(Cc1nc2cc(C(=O)NO)ccc2n1C)c1ccccc1
CCN(Cc1nc2cc(C(=O)NO)ccc2n1C)c1ccccc1
CCCN(Cc1nc2cc(C(=O)NO)ccc2n1C)c1ccccc1
CCCCN(Cc1nc2cc(C(=O)NO)ccc2n1C)c1ccccc1
CCCCN(Cc1nc2cc(C(=O)NO)ccc2n1C)c1cccc(F)c1
Cn1c(CNCc2ccccc2)nc2cc(C(=O)NO)ccc21
C[C@H](NCc1ccccc1)c1nc2cc(C(=O)NO)ccc2n1C
C[C@@H](NCc1ccccc1)c1nc2cc(C(=O)NO)ccc2n1C
Cn1c([C@H](Cc2ccccc2)NCc2ccccc2)nc2cc(C(=O)NO)ccc21
Cn1c([C@@H](Cc2ccccc2)NCc2ccccc2)nc2cc(C(=O)NO)ccc21
COc1nc(-c2ccc(NC(=O)Nc3ccc(C(=O)NCCCCCC(=O)Nc4ccccc4N)cc3)cc2)nc(N2CCOCC2)n1
Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1Nc1nc(-c2cccnc2)nc2nn(C)cc12
CCNC(=O)C[C@@H]1N=C(c2ccc(Cl)cc2)c2cc(OC)ccc2-n2c(C)nnc12 |r,t:7|