1575 SMILES Strings for Mast/stem cell growth factor receptor Kit [D816V]

Compound Name
SMILES String
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccccc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cn[nH]c2)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cnn(C)c2)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccccc2)cc1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)Nc1ccc(cc1)C#N
Cc1ccc(CC(=O)NC2CN(C2)c2ncnn3cc(cc23)-c2cnn(C)c2)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccnn2C)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cn(C)cn2)cc1
C[C@H](NCC1CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)c1ccc(C)cc1 |r|
C[C@@H](NCC1CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)c1ccc(C)cc1 |r|
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)C2=CCOCC2)cc1 |t:25|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(F)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cnn(C)c2)s1
Cc1csc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cnn(C)c2)c1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)Nc1ccc(Cl)cc1
Cc1nn(C)cc1-c1cc2c(ncnn2c1)N1CC(C1)C(=O)Nc1ccc(cc1)C#N
Cc1c(cnn1C)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)Nc1ccc(cc1)C#N
Cc1cc(ccc1NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)C#N
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C)(C1)C(=O)Nc1ccc(cc1)C#N
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(N)nc2)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(F)cc2)cc1
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)c1ccc(C)cc1 |r|
Cc1c(cnn1C)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
Cc1nn(C)cc1-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
Cc1ccc(CNC(=O)C2(C)CN(C2)c2ncnn3cc(cc23)-c2cnn(C)c2)cc1
Cc1n[nH]c(C)c1-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
CCc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cnn(C)c2)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cn(C)nc2N)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cnn(C)c2N)cc1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](CO)c1ccccc1 |r|
COc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cnn(C)c2)cc1
Cc1csc(c1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
Cc1ccc(s1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)c1ccc(F)cc1 |r|
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cnn(C)c2)c(F)c1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cnn(C)c2)cc1F
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(Cl)cc1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)NC(=O)Cc1ccc(Cl)cc1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(F)cc1F
COc1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)Nc1ccc(cc1)C#N
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(\C=C\c4ccccn4)cc23)cc1
CC(C)n1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)Nc1ccc(cc1)C#N
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)NC(=O)Cc1c[nH]c2ccccc12
COc1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
COc1cccc(c1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cnn(c2)C2CC2)cc1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(cc1)C1CC1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cnn3CCCc23)cc1
COc1ccc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
COc1ccc(nc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(=O)n(C)c2)cc1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@H]1[C@@H](O)Cc2ccccc12 |r|
CC(C)n1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
CCC1(CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)C(=O)NCc1ccc(C)cc1
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)c1ccc(C)cc1 |r|
Cc1ccc(CNC(=O)C2(CN)CN(C2)c2ncnn3cc(cc23)-c2cnn(C)c2)cc1
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(N)nc1)c1ccc(F)cc1 |r|
Cc1ccc(CNC(=O)C2(CO)CN(C2)c2ncnn3cc(cc23)-c2cnn(C)c2)cc1
COC1(CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)C(=O)NCc1ccc(C)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(Cl)cc2)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cccc(Cl)c2)cc1
Cc1nc(C)c(s1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
C[C@H](NC(=O)C1(C)CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)c1ccc(F)cc1 |r|
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cn(C)nc1C)c1ccc(F)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)c1ccc(F)cc1 |r|
COC1(CN(C1)c1ncnn2cc(cc12)C1=CCOCC1)C(=O)NCc1ccc(C)cc1 |t:18|
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cn(C)nc1N)c1ccc(F)cc1 |r|
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)c1ccc(Cl)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C)(C1)C(=O)NCc1ccc(Cl)cc1
CC(C(=O)NC1CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)c1ccc(Cl)cc1
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cn[nH]c1)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)c1ccc(Cl)cc1 |r|
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)C2CC2)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc3nonc3c2)cc1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(Cl)cc1F
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)NC(=O)Cc1ccc(Cl)cc1F
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)Nc1ccc(cc1)C(C)(C)C#N
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cnn(c2)C2CCC2)cc1
CN(C)c1ccc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
C[C@H](O)Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)Nc1ccc(cc1)C#N |r|
COc1cc(ccn1)-c1cc2c(ncnn2c1)N1CC(C)(C1)C(=O)NCc1ccc(C)cc1
COc1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NC(CO)c1ccccc1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(cc1)C(C)(C)C
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cnn(c2)C(C)(C)C)cc1
Cc1ccc(CNC(=O)C2(CN(C2)c2ncnn3cc(cc23)-c2cnn(C)c2)C(N)=O)cc1
CC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1 |c:6|
CNCC1(CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)C(=O)NCc1ccc(C)cc1
CC(C)n1cc(c(N)n1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
Cc1ccc(cc1)[C@H](CCN)NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
COc1ccc(-c2cc3c(ncnn3c2)N2CC(C2)C(=O)NCc2ccc(C)cc2)c(F)c1
COc1ccc(cc1F)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
C[C@H](O)Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1 |r|
Cc1ccc(cc1)[C@H](CCO)NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
CC(C)n1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](C)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)NC(=O)C1(CC1)c1ccc(Cl)cc1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NC1CCc2cc(Cl)ccc12
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(CCO)c1)c1ccc(F)cc1 |r|
C[C@H](NC(=O)C1(C)CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)c1ccc(Cl)cc1 |r|
C[C@H](NC(=O)C1(O)CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)c1ccc(Cl)cc1 |r|
COC1(CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)C(=O)N[C@@H](C)c1ccc(Cl)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](CO)c1ccc(Cl)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)Nc1ccc(Br)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc3C(=O)NCc3c2)cc1
CC(C)Oc1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)Nc1ccc(cc1)C#N
CC(C)(O)c1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)Nc1ccc(cc1)C#N
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)C2(N)CC2)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(OC3CC3)cc2)cc1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C)(C1)C(=O)NCc1ccc(Cl)cc1F
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)C(C)(C)N)cc1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(cc1)C(F)(F)F
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc3OCCOc3c2)cc1
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)C1CC1)c1ccc(F)cc1 |r|
CC(C)Oc1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cccc(c2)C(C)(C)O)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)C(C)(C)O)cc1
Cc1ccc(CC(=O)NC2CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)C(C)(C)O)cc1
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)c1ccc(cc1)C1CC1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(Cl)cc1Cl
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)NC(=O)Cc1ccc(Cl)cc1Cl
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cnn(c2)C2CCNC2)cc1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)Nc1ccc(OC(F)(F)F)cc1
COC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C1)C(=O)Nc1ccc(cc1)C#N |c:7|
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)C(O)CO)cc1
CCC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1 |c:7|
CCC(=O)N1CCC=C(C1)c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1 |c:7|
CN(C)CC1(CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)C(=O)NCc1ccc(C)cc1
C[C@H](NC(=O)C1(C)CN(C1)c1ncnn2cc(cc12)-c1cnn2CCCc12)c1ccc(F)cc1 |r|
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cnn(CC(C)(C)O)c2)cc1
Cc1ccc(CC(=O)NC2CN(C2)c2ncnn3cc(cc23)-c2cnn(CC(C)(C)O)c2)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cnn(c2)C(C)(C)CO)cc1
CNCC1(CN(C1)c1ncnn2cc(cc12)-c1cn(C)nc1N)C(=O)NCc1ccc(C)cc1
COC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1 |c:7|
COCCN1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1 |c:7|
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(c1)C1COC1)c1ccc(F)cc1 |r|
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(c1)C(C)(C)C)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](C1CC1)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(N)nc1)c1ccc(Cl)cc1 |r|
CC(C)(O)Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(F)cc1
COCCn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](C)c1ccc(F)cc1 |r|
C[C@H](O)Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](C)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@H]1[C@@H](O)Cc2cc(Cl)ccc12 |r|
CC[C@H](NC(=O)C1(C)CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)c1ccc(Cl)cc1 |r|
CC(C)[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)c1ccc(Cl)cc1 |r|
CC(C)n1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](C)c1ccc(Cl)cc1 |r|
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)C(C)(C)C#N)cc1
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cn(C)nc1N)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1N)c1ccc(Cl)cc1 |r|
COC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)c1ccc(Cl)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](CCO)c1ccc(Cl)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(Br)cc1
Cc1ccc(CNC(=O)C2(C)CN(C2)c2ncnn3cc(cc23)-c2ccc3C(=O)NCc3c2)cc1
Cc1ccc(CNC(=O)C2(C)CN(C2)c2ncnn3cc(cc23)-c2ccc3NC(=O)Cc3c2)cc1
CC(C)(C)Oc1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)Nc1ccc(cc1)C#N
Cc1ccc(CNC(=O)C2CN(C2)c2nccn3nc(cc23)-c2ccc(cc2)C2(CO)CC2)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)C2(O)CCC2)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc3CC(C)(C)Oc3c2)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc3OC(C)(C)Cc3c2)cc1
CC[C@H](NC(=O)N1CC(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)c1ccc(Cl)cc1F |r|
CN(C)C(=O)c1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
Cn1cc(c(N)n1)-c1cc2c(ncnn2c1)N1CC(C)(C1)C(=O)NCc1ccc(Cl)cc1F
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)C2(O)COC2)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(OC(C)(C)C)cc2)cc1
CC(C)Oc1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C)(C1)C(=O)NCc1ccc(C)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cccc(OC(C)(C)C)c2)cc1
Cc1ccc(CNC(=O)C2(C)CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)C(C)(C)O)cc1
CCC(C)(O)c1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)C(C)(C)O)c1ccc(C)cc1 |r|
COC1(CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)C(=O)NCc1ccc(Cl)cc1F
CC(C(=O)NC1CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)c1ccc(Cl)cc1Cl
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)C2=CCN(CC2)C(=O)C2CC2)cc1 |t:25|
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(OC2CC2)cc1)c1ccccc1 |r|
COCCOc1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cnn(CC3(C)COC3)c2)cc1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)NC(=O)C(O)c1ccc(Cl)cc1Cl
CS(=O)(=O)c1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)Nc1ccc(cc1)C#N
CCC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C)(C1)C(=O)NCc1ccc(C)cc1 |c:7|
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc2OCCOc2c1)c1ccc(F)cc1 |r|
CC(C)Oc1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](C)c1ccc(F)cc1 |r|
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)C(C)(C)O)c1ccc(F)cc1 |r|
CC(C)(C)Oc1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(F)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(F)c(c2)C(C)(C)O)cc1
CN(C)C(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1 |c:8|
COC(C)(C)Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(CC(C)(C)O)c1)c1ccc(C)cc1 |r|
CCOC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1 |c:8|
COC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C)(C1)C(=O)NCc1ccc(C)cc1 |c:7|
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)S(C)(=O)=O)cc1
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(=O)n(C)c1)c1ccc(Cl)cc1 |r|
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(CC(C)(C)O)c1)c1ccc(F)cc1 |r|
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cnn(CC(C)(C)O)c2)c(F)c1
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(c1)C(C)(C)CO)c1ccc(F)cc1 |r|
CC[C@H](O)Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](C)c1ccc(F)cc1 |r|
CC(O)C(C)n1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](C)c1ccc(F)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(c1)C(C)C)c1ccc(Cl)cc1 |r|
CC(C)n1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C)(C1)C(=O)N[C@@H](C)c1ccc(Cl)cc1 |r|
COC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](C)c1ccc(F)cc1 |r,c:7|
COC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C)(C1)C(=O)NCc1ccc(F)cc1 |c:7|
Cc1nn(C)cc1-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](CCO)c1ccc(Cl)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C)(C1)C(=O)N[C@@H](CCO)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1(CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)OC)c1ccc(Cl)cc1 |r|
CC(C)(O)Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(Cl)cc1
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(CCO)c1)c1ccc(Cl)cc1 |r|
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)N2CCCC2=O)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)C2=CCN(CC2)S(C)(=O)=O)cc1 |t:25|
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(OC(F)(F)F)cc2)cc1
CC(C)(O)Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(F)cc1F
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)C(C)(O)C2CC2)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)C2(O)CCCC2)cc1
COC1(CN(C1)c1ncnn2cc(cc12)-c1ccc2C(=O)NCc2c1)C(=O)NCc1ccc(C)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)C2(O)CCOC2)cc1
Cc1ccc(CNC(=O)C2(C)CN(C2)c2ncnn3cc(cc23)-c2ccc(OC(C)(C)C)cc2)cc1
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(OC(C)(C)C)cc1)c1ccc(C)cc1 |r|
CCC(C)(C)Oc1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1
CCc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(OC(C)(C)C)cc2)cc1
CN(C)C(=O)c1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](CO)c1ccccc1 |r|
CN(C)C(=O)c1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@H](CO)c1ccccc1 |r|
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)C1(O)CCC1)c1ccc(F)cc1 |r|
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(OCC(C)(C)O)cc2)cc1
COC1(CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)C(C)(C)O)C(=O)NCc1ccc(C)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2cnn(C[C@@H]3CNCCO3)c2)cc1 |r|
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)C2=CCN(CC2)C(=O)C(C)(C)C)cc1 |t:25|
C[C@H](NC(=O)C1(C)CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)C(C)(C)O)c1ccc(F)cc1 |r|
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(OC(C)(C)C)c(F)c2)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(F)c(OC(C)(C)C)c2)cc1
CCC(C)(O)c1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](C)c1ccc(F)cc1 |r|
CC(C)OC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(C)cc1 |c:9|
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(CC2(C)COC2)c1)c1ccc(F)cc1 |r|
COC1(CN(C1)c1ncnn2cc(cc12)-c1cnn(CC(C)(C)O)c1)C(=O)NCc1ccc(C)cc1
Cc1ccc(CNC(=O)C2(C)CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)S(C)(=O)=O)cc1
CC(C)(C)Oc1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(Cl)cc1
CC[C@H](NC(=O)C1(C)CN(C1)c1ncnn2cc(cc12)-c1cnn2CCCc12)c1ccc(Cl)cc1 |r|
COC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C1)(OC)C(=O)NCc1ccc(C)cc1 |c:7|
CCC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C)(C1)C(=O)N[C@@H](C)c1ccc(F)cc1 |r,c:7|
CC(C)(C)Oc1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(F)cc1F
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(c1)[C@@H](C)C(C)(C)O)c1ccc(F)cc1 |r|
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(c1)[C@H](C)C(C)(C)O)c1ccc(F)cc1 |r|
OCC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn2CCCc12)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(c1)C1COC1)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1(C)CN(C1)c1ncnn2cc(cc12)-c1cnn(c1)C(C)C)c1ccc(Cl)cc1 |r|
COC[C@H](O)Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](C)c1ccc(F)cc1 |r|
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)S(C)(=O)=O)c1ccc(F)cc1 |r|
CC(C)(O)c1ccc(cc1)C1=CN2C=CCN(N3CC(C3)C(=O)NCc3ccc(Cl)cc3F)N2C1 |c:14,t:11|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](CC(C)(C)O)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(C[C@H](C)O)c1)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(CCOC)c1)c1ccc(Cl)cc1 |r|
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(CC(C)(C)O)c1)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(C[C@@H](C)O)c1)c1ccc(Cl)cc1 |r|
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)C(=O)N2CCCC2)cc1
Cc1ccc(CNC(=O)C2(C)CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)C(=O)N2CCC2)cc1
Cc1ccc(CNC(=O)C2(C)CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)N2CCCC2=O)cc1
COC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C)(C1)C(=O)NCc1ccc(Cl)cc1 |c:7|
CC(C)(O)Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(cc1)C(F)F
COC1(CN(C1)c1ncnn2cc(cc12)-c1cnn(C)c1)C(=O)NCc1ccc(Br)cc1
COC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C)(C1)C(=O)NCc1ccc(F)cc1F |c:7|
CC(C)(O)Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(Cl)cc1F
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)N1CCCC1=O)c1ccc(F)cc1 |r|
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)C(=O)N1CCC1)c1ccc(F)cc1 |r|
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)C1=CCN(CC1)S(C)(=O)=O)c1ccc(F)cc1 |r,t:21|
COC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(Cl)cc1F |c:7|
COC1(CN(C1)c1ncnn2cc(cc12)-c1ccc(OC(C)(C)C)cc1)C(=O)NCc1ccc(C)cc1
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)C2=CCN(CC2)C(=O)N2CCCC2)cc1 |t:25|
OCC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)C1=CCC(F)(F)CC1)c1ccc(Cl)cc1 |r,t:23|
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)C2=CCN(CC2)C(=O)OC(C)(C)C)cc1 |t:25|
CNCC1(CN(C1)c1ncnn2cc(cc12)-c1cnn(CC(C)(C)O)c1)C(=O)NCc1ccc(C)cc1
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(OC(C)C)cc1)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)C(C)(C)O)c1ccc(Cl)cc1 |r|
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(OC(C)(C)C)cc1)c1ccc(Cl)cc1 |r|
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)C2(CC2)C(F)(F)F)cc1
C[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(OC(C)(C)C)c(F)c1)c1ccc(F)cc1 |r|
COC1(CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)S(C)(=O)=O)C(=O)NCc1ccc(C)cc1
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)[C@@H](O)CO)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)[C@H](O)CO)c1ccc(Cl)cc1 |r|
CC(C)(O)c1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)Nc1ccc(Br)cc1
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(CC(C)(C)N)c1)c1ccc(Cl)cc1 |r|
C[C@H](NC(=O)C1(C)CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)S(C)(=O)=O)c1ccc(F)cc1 |r|
CC(C)(O)c1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C)(C1)C(=O)NCc1ccc(Cl)cc1F
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(CC(C)(C)O)c1)c1ccc(Cl)cc1 |r|
CC[C@H](O)Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](CC)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(c1)C(C)(C)CO)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(c1)[C@H](C)[C@H](C)O)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(c1)[C@@H](C)[C@@H](C)O)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)C1=CCN(CC1)C(=O)OC)c1ccc(Cl)cc1 |r,t:22|
Cc1ccc(CNC(=O)C2CN(C2)c2ncnn3cc(cc23)-c2ccc(cc2)C(C)(O)C(F)(F)F)cc1
CC(C)(O)c1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)NC(=O)Cc1ccc(Cl)cc1Cl
COC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C)(C1)C(=O)NCc1ccc(Cl)cc1F |c:7|
Cc1ccc(cc1)[C@H](CCO)NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(OC(C)(C)C)cc1 |r|
CS(=O)(=O)c1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)NCc1ccc(Cl)cc1F
COC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C1)NC(=O)Cc1ccc(Cl)cc1Cl |c:7|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)C1(O)CCC1)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(OC(C)(C)C)cc1)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1(C)CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)C(C)(C)O)c1ccc(Cl)cc1 |r|
C[C@H](NC(=O)C1(C)CN(C1)c1ncnn2cc(cc12)-c1ccc(OC(C)(C)C)cc1)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)C(C)(O)CC)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(CCC(C)(C)O)c1)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(c1)[C@@H](C)C(C)(C)O)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(c1)[C@H](C)C(C)(C)O)c1ccc(Cl)cc1 |r|
CCC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](CCO)c1ccc(Cl)cc1 |r,c:7|
CCOC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](CC)c1ccc(Cl)cc1 |r,c:8|
CC[C@H](NC(=O)C1(C)CN(C1)c1ncnn2cc(cc12)C1=CCN(CC1)C(=O)OC)c1ccc(Cl)cc1 |r,t:23|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(OC(C)(C)C)cc1)c1ccc(cc1)C1CC1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)S(C)(=O)=O)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(c1)C(C)C(C)O)c1ccc(Cl)cc1 |r|
CC(C)(C)Oc1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)NC(=O)Cc1ccc(Cl)cc1Cl
CC1(CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)S(C)(=O)=O)C(=O)NCc1ccc(Cl)cc1F
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)C1=CCN(CC1)S(C)(=O)=O)c1ccc(Cl)cc1 |r,t:22|
CC(C)(C)Oc1ccc(cc1)-c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](CCO)c1ccc(Cl)cc1 |r|
CCC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C)(C1)C(=O)N[C@@H](CCO)c1ccc(Cl)cc1 |r,c:7|
CC[C@H](NC(=O)C1(CN(C1)c1ncnn2cc(cc12)-c1cnn(CC(C)(C)O)c1)OC)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1(C)CN(C1)c1ncnn2cc(cc12)-c1ccc(cc1)S(C)(=O)=O)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(C[C@@H](O)C(F)(F)F)c1)c1ccc(Cl)cc1 |r|
CC[C@H](NC(=O)C1CN(C1)c1ncnn2cc(cc12)-c1cnn(C[C@H](O)C(F)(F)F)c1)c1ccc(Cl)cc1 |r|
CC(C)(C)OC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C1)C(=O)N[C@@H](CCO)c1ccc(Cl)cc1 |r,c:10|
CC(C)(C)OC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CC(C)(C1)C(=O)N[C@@H](CCO)c1ccc(Cl)cc1 |r,c:10|
Cc1nc([nH]c1-c1ccccc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccccc1
Cc1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccccc1
Cc1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccc(F)cc1
Cc1nc([nH]c1-c1ccc(F)cc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccc(F)cc1
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C2CC2)c([nH]1)-c1ccccc1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C2CC2)c([nH]1)-c1ccccc1
N#Cc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C2CC2)c([nH]1)-c1ccccc1
FC(F)Oc1cccc(c1)-c1nnc([nH]1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Cc1nc([nH]c1-c1cccc(OC(F)(F)F)c1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nnc([nH]1)-c1ccc(F)cc1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nnc([nH]1)-c1ccc(F)cc1
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nnc([nH]1)-c1cccc(OC(F)F)c1
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1cccc(OC(F)(F)F)c1
COc1ccc(cc1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
Cc1nc([nH]c1-c1cccc(F)c1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1ccc(cc1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccnc(OC)c1
COc1ccc(cc1F)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1cccc(F)c1
Cc1nc([nH]c1-c1ccc(F)cc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1cccc(c1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1cccc(c1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccnc(OC)c1
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccc(OC)c(C)c1
CCOc1cccc(c1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
CCOc1cccc(c1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
CCOc1ccc(cc1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
CCOc1ccc(cc1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1ccc(cc1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
COc1ccc(cc1C)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
COc1ccc(cc1C)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
CCOc1ccc(cc1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccnc(OC)c1
Cc1nc([nH]c1-c1ccccc1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1ccccc1
CCOc1cccc(c1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccnc(OC)c1
Cc1nc([nH]c1-c1ccc(Cl)cc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
COc1ccc(cc1OC)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccc(Cl)cc1
Cc1nc([nH]c1-c1ccc(Cl)cc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1ccc(cc1OC)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1ccc(cc1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
COc1ccc(cc1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccnc(OC)c1
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccc(OC)c(OC)c1
COc1ccc(cc1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
Cc1nc([nH]c1-c1ccccc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C(N)=O
COc1ncc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccccc1
Cc1nc([nH]c1-c1ccccc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(C)c1
Cc1nc([nH]c1-c1ccccc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
Cc1nc([nH]c1-c1ccccc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)S(N)(=O)=O
CNC(=O)c1cccc(c1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccccc1
Cc1nc([nH]c1-c1ccccc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
Cc1nc([nH]c1-c1ccccc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cccc(c1)S(N)(=O)=O
COc1ccc(cc1C)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
COc1ccc(cc1C)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1ccc(OC)c(C)c1
CCC1(CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1nc(C)c([nH]1)-c1ccc(OC)cc1
CCC1(CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1nc(C)c([nH]1)-c1ccc(OC)c(C)c1
Cc1nc([nH]c1-c1ccc(F)cc1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Cc1nc([nH]c1-c1ccc(Cl)cc1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
CCc1ccc(cc1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccnc(OC)c1
CCc1ccc(cc1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
CCc1ccc(cc1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
Cc1nc([nH]c1-c1ccc(C)cc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
COc1ccc(cc1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(C)cc12
Cc1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1ccc(F)cc1
CCOc1ccc(cc1C)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
CCOc1ccc(cc1C)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
CCOc1ccc(cc1C)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccnc(OC)c1
Cc1nc([nH]c1-c1ccc2OCOc2c1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Cc1nc([nH]c1-c1ccc2OCOc2c1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccc2OCOc2c1
CC(=O)Nc1cccc(c1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccccc1
COc1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccccc1
Cc1nc([nH]c1-c1ccccc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cn(C)nc1C
Cc1nc([nH]c1-c1ccccc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(C)nc1
CCOc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccccc1
Cc1nc([nH]c1-c1ccccc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccnc(c1)N1CCOCC1
CC1CCN(CC1)c1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccccc1
CC(C)Oc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccccc1
Cc1nc([nH]c1-c1ccccc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccnc(c1)N1CCCC1
Cc1nc([nH]c1-c1ccccc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cccc(OC(F)(F)F)c1
Cc1nc([nH]c1-c1ccccc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cccc(F)c1
Cc1nc([nH]c1-c1ccccc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cccc(Cl)c1
Cc1nc([nH]c1-c1ccccc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cccc(NS(C)(=O)=O)c1
Cc1nc([nH]c1-c1ccc2OCCOc2c1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Cc1nc([nH]c1-c1ccc(OC(F)(F)F)cc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Cc1nc([nH]c1-c1ccc(OC(F)(F)F)cc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccc(OC(F)(F)F)cc1
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccc(C)cc1
Cc1nc([nH]c1-c1ccc(C)cc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
Cc1ccc(s1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccc(OC(C)C)cc1
CC(C)Oc1ccc(cc1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
CC(C)Oc1ccc(cc1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
CCOc1cc(ccc1C)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
CCOc1cc(ccc1C)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
CCOc1cc(ccc1C)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccnc(OC)c1
Cc1nc([nH]c1-c1ccccc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccnc(c1)C(F)(F)F
Cc1nc([nH]c1-c1ccccc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cccc(c1)C(F)(F)F
CCOc1ccc(cc1C)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(C)cc12
COCc1cc(ccc1C)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(C)cc12
CCc1ccc(cc1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(C)cc12
COc1ccc(cc1C)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(C)cc12
COc1cc(ccc1C)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccc(C)c(OC)c1
COc1cc(ccc1C)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(C)cc12
COc1cc(ccc1C)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
Cc1nc([nH]c1-c1ccc(F)cc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
COc1ccc(cc1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
Cc1nc([nH]c1-c1ccc2OC(F)(F)Oc2c1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Cc1nc([nH]c1-c1ccc2OC(F)(F)Oc2c1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccc2OC(F)(F)Oc2c1
COc1ccc(cn1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
Cc1nc([nH]c1-c1ccc(OC(F)F)cc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1cccc(c1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
Cc1nc([nH]c1-c1ccc(OC(F)F)cc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
Cc1nc([nH]c1-c1ccc(OC(F)(F)F)cc1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccc(C)s1
Cc1ccc(s1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Cc1nc([nH]c1-c1ccc(Cl)s1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Cc1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccc2OCOc2c1
Cc1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccc2OCCOc2c1
Cc1nn(C)cc1-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccc(OC(F)(F)F)cc1
COc1cccc(c1)-c1[nH]c(nc1C(F)(F)F)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccnc(OC)c1
COc1cccc(c1)-c1[nH]c(nc1C(F)(F)F)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
CCOc1ccc(cc1C)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(C)cc12
CCOc1cc(ccc1C)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(C)cc12
Cc1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccc2OC(F)(F)Oc2c1
COc1ccc(cc1C)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(C)cc12
COc1cc(ccc1C)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(C)cc12
COc1ccc(cc1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(C)cc12
COc1cccc(c1)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(C)cc12
Cc1nc([nH]c1-c1ccc2OCCOc2c1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
Cc1nc([nH]c1-c1ccc2OCCOc2c1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(c([nH]1)-c1ccc(C)cc1)C(F)(F)F
Cc1ccc(cc1)-c1[nH]c(nc1C(F)(F)F)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Cc1nc([nH]c1-c1ccc(cc1)C(F)(F)F)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Cc1nc([nH]c1-c1ccc(cc1)C(F)(F)F)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
Cc1nc([nH]c1-c1ccc2OCOc2c1)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
CCOc1ccc(cc1C)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
CCC1(CCN(CC1)c1ncnc2[nH]c(C)cc12)c1nc(C)c([nH]1)-c1ccc(OC)cc1
CCC1(CCN(CC1)c1ncnc2[nH]c(C)cc12)c1nc(C)c([nH]1)-c1ccc(OC)c(C)c1
CCOc1ccc(cc1C)-c1[nH]c(nc1C)C1(CC)CCN(CC1)c1ncnc2[nH]c(C)cc12
CCC1(CCN(CC1)c1ncnc2[nH]c(C)cc12)c1nc(C)c([nH]1)-c1ccc2OCOc2c1
CCC1(CCN(CC1)c1ncnc2[nH]c(C)cc12)c1nc(C)c([nH]1)-c1ccc2OCCOc2c1
CCOc1ccc(cc1)-c1[nH]c(nc1C)C1(CC)CCN(CC1)c1ncnc2[nH]c(C)cc12
COc1ccc(cc1)-c1[nH]c(nc1C(F)(F)F)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccnc(OC)c1
COc1ccc(cc1)-c1[nH]c(nc1C(F)(F)F)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
COc1ccc(cc1)-c1[nH]c(nc1C(F)(F)F)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccc(cc1)C(F)(F)F
Cc1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1ccc2OCOc2c1
Cc1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1ccc2OCCOc2c1
Cc1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1ccc2OC(F)(F)Oc2c1
COc1ccc(cc1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
COc1ccc(cc1C)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
Cc1nc([nH]c1-c1ccc2OCOc2c1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
COc1ccc(cc1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(OC)nc1
COc1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1ccc(OC)c(C)c1
COc1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1ccc2OCOc2c1
Cc1nc([nH]c1-c1ccc2OCOc2c1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
CCOc1ccc(cc1C)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
CCOc1ccc(cc1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
Cc1nc([nH]c1-c1ccc(cc1)C(F)F)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1ccc(cc1F)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
Cc1nc([nH]c1-c1ccc(cc1)C(F)F)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
Cc1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nc(C)c([nH]1)-c1ccc(cc1)C(F)(F)F
COc1cccc(c1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(C)cc12
COc1cccc(c1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1cccc(c1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
COc1cccc(c1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(OC)nc1
CCOc1ccc(cc1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
CCOc1ccc(cc1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(OC)nc1
COc1ccc(cn1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1ncc(cc1F)-c1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
Cc1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1ccc(Cl)cc1
Cc1nc([nH]c1-c1ccc(Cl)cc1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
COc1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1ccc(Cl)cc1
Cc1nc([nH]c1-c1ccc(cc1)C(F)(F)F)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1ccc(cc1)C(F)(F)F
Cc1nc([nH]c1-c1ccc(cc1)C(F)(F)F)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
Cc1nc([nH]c1-c1ccc(Cl)cc1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1ncc(cc1F)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
COc1ccc(cn1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
COc1ccc(cc1F)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(C)cc12
Cc1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1ccc(cc1)C(F)F
COc1ncc(cc1F)-c1nc([nH]c1C)C1(C)CCN(CC1)c1ncnc2[nH]c(C)cc12
COc1ccc(cn1)-c1nc([nH]c1C)C1(C)CCN(CC1)c1ncnc2[nH]c(C)cc12
COc1ccc(cc1F)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
COc1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1ccc(OC)c(F)c1
Cc1nc([nH]c1-c1ccc(cc1)C(F)F)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
COc1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1ccc(cc1)C(F)F
Cc1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1cccc(OC(F)F)c1
Cc1nc([nH]c1-c1cccc(OC(F)F)c1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
COc1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1cccc(OC(F)F)c1
Cc1nc([nH]c1-c1cccc(OC(F)F)c1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
Cc1nc([nH]c1-c1ccc(OC(F)F)cc1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
Cc1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1ccc(OC(F)F)cc1
CCc1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
CCc1[nH]c(nc1C)C1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N
Cc1nc([nH]c1-c1ccc(Cl)cc1)C1(C)CCN(CC1)c1ncnc2[nH]nc(C)c12
Cc1nc([nH]c1-c1cccc(OC(F)F)c1)C1(C)CCN(CC1)c1ncnc2[nH]nc(C)c12
COc1ccc(cc1F)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]nc(C)c12
Cc1nc([nH]c1-c1ccc2OC(F)(F)Oc2c1)C1(C)CCN(CC1)c1ncnc2[nH]nc(C)c12
COc1ccc(cc1F)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C(O)=O
CCOc1ccc(cc1F)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(OC)nc1
CCOc1ccc(cc1F)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
COc1ccc(cc1F)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(nc1)C#N
COc1ccc(cc1F)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C(N)=O
COc1ccc(cc1F)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(NS(C)(=O)=O)cc1
COc1ccc(cc1F)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(OCC(O)=O)cc1
COc1ccc(cc1F)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(nc1)N1CCOCC1
COc1ccc(cc1C)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C(N)=O
COc1ccc(cc1C)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(OCC(O)=O)cc1
CNC(=O)c1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1ccc(OC)c(C)c1
COc1ccc(cc1C)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(nc1)N1CCOCC1
CNC(=O)c1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1ccc(OC)c(F)c1
COc1cccc(c1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(OCC(O)=O)cc1
CNC(=O)c1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1cccc(OC)c1
COc1cccc(c1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(nc1)N1CCOCC1
CCOc1ccc(cc1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(OCC(O)=O)cc1
COc1cccc(c1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C(N)=O
CCOc1ccc(cc1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(nc1)C(=O)NC
CCOc1ccc(cc1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(nc1)N1CCOCC1
COc1ccc(cc1C)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(NS(C)(=O)=O)cc1
CCOc1ccc(cc1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C(N)=O
CCOc1ccc(cc1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(NS(C)(=O)=O)cc1
Cc1nc([nH]c1-c1cccc(OC(F)F)c1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C(N)=O
Cc1nc([nH]c1-c1cccc(OC(F)F)c1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(NS(C)(=O)=O)cc1
Cc1nc([nH]c1-c1cccc(OC(F)F)c1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(OCC(O)=O)cc1
COc1cccc(c1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(NS(C)(=O)=O)cc1
CNC(=O)c1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1ccc(cc1)C(F)F
CNC(=O)c1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1cccc(OC(F)F)c1
Cc1nc([nH]c1-c1ccc(cc1)C(F)F)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(nc1)N1CCOCC1
Cc1nc([nH]c1-c1cccc(OC(F)F)c1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(nc1)N1CCOCC1
Cc1nc([nH]c1-c1ccc(cc1)C(F)F)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C(N)=O
Cc1nc([nH]c1-c1ccc(cc1)C(F)F)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(OCC(O)=O)cc1
Cc1nc([nH]c1-c1ccc(OC(F)F)cc1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(OCC(O)=O)cc1
Cc1nc([nH]c1-c1ccc(OC(F)F)cc1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
CCOc1ccc(cc1C)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C(N)=O
CCOc1ccc(cc1C)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(OCC(O)=O)cc1
CCOc1ccc(cc1C)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(c1)C(F)F
CNC(=O)c1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(C)(CC1)c1nc(C)c([nH]1)-c1ccc(OC(F)F)cc1
CCOc1ccc(cc1C)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(nc1)C(=O)NC
Cc1nc([nH]c1-c1ccc(OC(F)F)cc1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(nc1)N1CCOCC1
CCOc1ccc(cc1C)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(nc1)N1CCOCC1
COc1ccc(cc1C)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(nc1)C#N
CCOc1ccc(cc1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(nc1)C#N
Cc1nc([nH]c1-c1ccc(cc1)C(F)F)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(NS(C)(=O)=O)cc1
Cc1nc([nH]c1-c1ccc(OC(F)F)cc1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C(N)=O
Cc1nc([nH]c1-c1ccc(OC(F)F)cc1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(NS(C)(=O)=O)cc1
Cc1nc([nH]c1-c1cccc(OC(F)F)c1)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(nc1)C#N
COc1cccc(c1)-c1[nH]c(nc1C)C1(C)CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(nc1)C#N
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1ccc(C)nc1)c1cccc(Cl)c1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1ccc(C)nc1)c1cccc(OC(F)F)c1 |r|
COc1cccc(c1)[C@H](C)NC(=O)N1CCN(CC1)c1ncnc2[nH]c(C)cc12 |r|
COc1cc(ccc1F)[C@H](C)NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1cccc(F)c1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1cccc(OC(F)F)c1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1ccc(C)nc1)c1cccc(F)c1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1cccc(Cl)c1 |r|
COc1cccc(c1)C(C)NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1ccnc(OC)c1
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)c1nc2ccccc2[nH]1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)c1nc2ccccc2[nH]1
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCN(C(=O)N[C@@H](C)c2cccc(OC(F)F)c2)C(C)(C)C1 |r|
Cc1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)c1nc2ccccc2[nH]1
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1cccc(OC(F)F)c1 |r|
COc1cccc(c1)[C@H](C)NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1cccc(c1)N(C)C |r|
CC(C)(C)Oc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(Cl)cc2)cc1
COc1ccc(cc1)[C@H](C)NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1 |r|
COc1ccc(cc1)[C@@H](C)NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(Cl)cc1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(Cl)cc1)c1ccc(Cl)cc1 |r|
C[C@@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(Cl)cc1)c1ccc(Cl)cc1 |r|
C[C@@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(Cl)cc1)c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(Cl)cc1)c1ccc(F)cc1 |r|
COc1cccc(c1)[C@H](C)NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(Cl)cc1 |r|
COc1cccc(c1)[C@@H](C)NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(Cl)cc1 |r|
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1cccc(Cl)c1 |r|
COc1cccc(c1)[C@H](C)NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1ccc(Cl)cc1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1ccc(F)cc1 |r|
COc1ccc(cc1)[C@@H](C)NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1 |r|
COc1cccc(c1)[C@@H](C)NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1cccc(c1)C(F)(F)F |r|
C[C@@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1ccc(F)cc1 |r|
C[C@@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1ccc(Cl)cc1 |r|
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1cccc(F)c1 |r|
FC(F)Oc1cccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(Cl)cc2)c1
COc1cccc(c1)[C@H](C)NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(Cl)cc1 |r|
C[C@H]1CN(CCN1C(=O)Nc1ccc(C)nc1)c1ncnc2[nH]c(cc12)-c1ccncc1 |r|
C[C@H]1CN(CCN1C(=O)NCc1cccc(Cl)c1)c1ncnc2[nH]c(cc12)-c1ccncc1 |r|
C[C@H]1CN(CCN1C(=O)NCc1ccc(F)cc1)c1ncnc2[nH]c(cc12)-c1ccncc1 |r|
C[C@H]1CN(CCN1C(=O)NCc1ccc(Cl)cc1)c1ncnc2[nH]c(cc12)-c1ccncc1 |r|
C[C@H]1CN(CCN1C(=O)Nc1ccc(Cl)cc1)c1ncnc2[nH]c(cc12)-c1ccncc1 |r|
COc1cccc(c1)[C@H](C)NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)C#CC1CC1 |r|
CCC(NC(=O)N1CCN(C[C@@H]1C)c1ncnc2[nH]c(cc12)-c1ccncc1)c1ccccc1 |r|
CC(NC(=O)N1CCN(C[C@@H]1C)c1ncnc2[nH]c(cc12)-c1ccncc1)c1ccc(F)cc1 |r|
CC(NC(=O)N1CCN(C[C@@H]1C)c1ncnc2[nH]c(cc12)-c1ccncc1)c1ccc(Cl)cc1 |r|
COc1cccc(c1)C(C)NC(=O)N1CCN(C[C@@H]1C)c1ncnc2[nH]c(cc12)-c1ccncc1 |r|
CN(C)c1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)C#CC2CC2)cc1
FC(F)(F)Oc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)C#CC2CC2)cc1
CCC(NC(=O)N1CCN(CC1C)c1ncnc2[nH]c(cc12)-c1ccncc1)c1ccccc1
C[C@@H]1CN(CCN1C(=O)Nc1ccc(C)nc1)c1ncnc2[nH]c(cc12)-c1ccncc1 |r|
C[C@@H]1CN(CCN1C(=O)NCc1cccc(Cl)c1)c1ncnc2[nH]c(cc12)-c1ccncc1 |r|
COc1ccc(NC(=O)N2CCN(C[C@H]2C)c2ncnc3[nH]c(cc23)-c2ccncc2)cn1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccncc1)c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccncc1)c1ccc(Cl)cc1 |r|
COc1cccc(c1)[C@H](C)NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccncc1 |r|
C[C@@H]1CN(CCN1C(=O)NCc1ccc(F)cc1)c1ncnc2[nH]c(cc12)-c1ccncc1 |r|
C[C@@H]1CN(CCN1C(=O)Nc1ccc(F)c(Cl)c1)c1ncnc2[nH]c(cc12)-c1ccncc1 |r|
C[C@@H]1CN(CCN1C(=O)Nc1ccc(OC(F)(F)F)cc1)c1ncnc2[nH]c(cc12)-c1ccncc1 |r|
C[C@@H]1CN(CCN1C(=O)NCc1ccc(Cl)cc1)c1ncnc2[nH]c(cc12)-c1ccncc1 |r|
C[C@@H]1CN(CCN1C(=O)Nc1ccc(Cl)cc1)c1ncnc2[nH]c(cc12)-c1ccncc1 |r|
C[C@@H]1CN(CCN1C(=O)Nc1ccc(cc1)N(C)C)c1ncnc2[nH]c(cc12)-c1ccncc1 |r|
Fc1ccccc1-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)Nc1ccc(OC(F)(F)F)cc1
CC1CN(CCN1C(=O)Nc1ccccc1)c1ncnc2[nH]c(cc12)-c1ccncc1
COc1cccc(c1)[C@H](C)NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N |r|
CN(C)c1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(cc2)C#N)cc1
C[C@H]1CN(CCN1)c1ncnc2[nH]c(cc12)-c1ccncc1 |r|
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1cccc(OC(F)F)c1 |r|
FC(F)Oc1cccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(F)cc2)c1
C[C@@H]1CN(CCN1)c1ncnc2[nH]c(cc12)-c1ccncc1 |r|
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1cccc(OC(F)(F)F)c1 |r|
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NCc1cccc(OC(F)(F)F)c1
CS(=O)(=O)Nc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)Nc1ccc(OC(F)(F)F)cc1
NC(=O)c1cccc(c1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)Nc1ccc(OC(F)(F)F)cc1
Cc1ncc(s1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NCc1ccc(F)cc1
Cc1ncc(s1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)Nc1ccc(OC(F)(F)F)cc1
CNC(=O)c1cccc(c1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NCc1ccc(F)cc1
CC(=O)Nc1cccc(c1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NCc1ccc(F)cc1
NS(=O)(=O)c1cccc(c1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)Nc1ccc(OC(F)(F)F)cc1
CC(=O)Nc1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)Nc1ccc(OC(F)(F)F)cc1
CN(C)C(=O)c1cccc(c1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)Nc1ccc(OC(F)(F)F)cc1
FC(F)(F)Oc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(cc2)C#N)cc1
COc1ncc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(F)cc2)cc1F
CCNC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
CCOc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)C#C)cc1
Fc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(F)cc2)cc1
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)Nc1ccc(OC(F)F)cc1
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)Nc1ccc(OC(F)(F)F)cc1
COc1cccc(c1)[C@H](C)NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(C)c1 |r|
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(C)c1)c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(C)c1)c1ccc(Cl)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)Nc1ccc(F)cc1
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NCc1ccc(Cl)cc1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NS(=O)(=O)c1ccc(Cl)cc1
NS(=O)(=O)c1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NCc1ccc(F)cc1
NS(=O)(=O)c1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)Nc1ccc(OC(F)(F)F)cc1
Fc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccncc2)cc1
FC(F)(F)Oc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccncc2)cc1
Cc1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NCc1ccc(F)cc1
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NCc1ccc(F)cc1
NS(=O)(=O)c1cccc(c1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NCc1ccc(F)cc1
COc1ncc(cn1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NCc1ccc(F)cc1
CS(=O)(=O)Nc1cccc(c1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NCc1ccc(F)cc1
NC(=O)c1cccc(c1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NCc1ccc(F)cc1
Fc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(cc2)C#N)cc1
Fc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2cccc(c2)C#N)cc1
FC(F)(F)Oc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(nc2)C2CC2)cc1
FC(F)(F)Oc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2cnc(nc2)C2CC2)cc1
FC(F)(F)Oc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(cc2)C2(CC2)C#N)cc1
CN(C)c1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)Nc1ccc(OC(F)(F)F)cc1
Cc1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)Nc1ccc(OC(F)(F)F)cc1
CNC(=O)c1cccc(c1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)Nc1ccc(OC(F)(F)F)cc1
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)Nc1ccc(OC(F)(F)F)cc1
COc1ccc(cn1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)Nc1ccc(OC(F)(F)F)cc1
CS(=O)(=O)Nc1cccc(c1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)Nc1ccc(OC(F)(F)F)cc1
CC(=O)Nc1cccc(c1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)Nc1ccc(OC(F)(F)F)cc1
FC(F)(F)Oc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2cccc(c2)C#N)cc1
COc1cccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(F)cc2)n1
Clc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2cccnc2)nc1
Fc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2cccnc2)nc1
FC(F)Oc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(F)cc2)cc1
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1ccc(F)cc1 |r|
COc1cc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2cccnc2)ccn1
COc1cccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2cccnc2)n1
COc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(F)cc2)cn1
NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cccnc1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NCc1cncc(F)c1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)Nc1ccc(OC(F)(F)F)cc1
FC(F)(F)Oc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(Cl)cc2)cc1
Fc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]cc(CC4CC4)c23)cc1
Clc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)C2CC2)cc1
Clc1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NCc1ccc(Cl)cc1
COc1ncc(F)cc1CNC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cccnc1
Cc1ccc(NS(=O)(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(Cl)cc2)cc1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NC(=O)c1ccccc1
COc1ccc(cc1)[C@@H](C)NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1 |r|
C[C@@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1ccc(F)cc1 |r|
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NC(=O)NC1CCCC1
COc1cccc(c1)[C@@H](C)NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1 |r|
Fc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)C#N)cc1
Cc1nc(no1)-c1cccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]ccc23)c1
O=C(Nc1cccnc1)N1CCN(CC1)c1ncnc2[nH]ccc12
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NCc1ccc(Cl)cc1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NCc1ccccc1Cl
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1cccc2ccccc12 |r|
COc1cccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(F)cc2)c1
COc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(F)cc2)cc1
Fc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]cc(C#N)c23)cc1
Cc1ccccc1C(=O)c1c[nH]c2ncnc(N3CCN(CC3)C(=O)NCc3ccc(F)cc3)c12
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NCCc1ccc(Cl)cc1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCN(CC1)C(=O)NCCc1ccccc1
Fc1cccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]ccc23)c1
Fc1ccc(CCNC(=O)N2CCN(CC2)c2ncnc3[nH]ccc23)cc1
Fc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]ccc23)cc1Cl
FC(F)(F)c1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]ccc23)cc1
FC(F)(F)c1cccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]ccc23)c1
Clc1cccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]ccc23)c1
COc1ccc(CCNC(=O)N2CCN(CC2)c2ncnc3[nH]ccc23)cc1
Clc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]ccc23)cc1
Clc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]ccc23)cc1
O=C(Nc1ccc(cc1)C#N)N1CCN(CC1)c1ncnc2[nH]ccc12
Fc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]ccc23)cc1F
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1ccc(Cl)cc1 |r|
FC(F)(F)c1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(Cl)cc2)cn1
Fc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]ccc23)cc1
Fc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]ccc23)cc1
FC(F)(F)Oc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]ccc23)cc1
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(Cl)cc1)c1ccc(Cl)cc1 |r|
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cccnc1)c1ccc(Cl)cc1 |r|
Clc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(Cl)cc2)cc1
Fc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(Cl)cc2)cc1
CCOc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccc(Cl)cc2)cc1
Clc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccccc2)cc1
COc1cc(NC(=O)N2CCN(CC2)c2ncnc3[nH]cc(-c4ccccc4)c23)cc(OC)c1
CCCNS(=O)(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cccnc1
CCCNC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cccnc1
Clc1ccccc1NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cccnc1
CCOc1cccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2cccnc2)c1
Fc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2cccnc2)cc1
FC(F)(F)c1cccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2cccnc2)c1
FC(F)(F)Oc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2cccnc2)cc1
CCOc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2cccnc2)cc1
Fc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]cc(-c4ccccc4)c23)cc1
COc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]cc(-c4ccccc4)c23)cc1
COc1cccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]cc(-c4ccccc4)c23)c1
COc1cc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2cccnc2)cc(OC)c1
COc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2cccnc2)cc1
COc1cccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2cccnc2)c1
CC(C)(C)OC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cccnc1
c1c[nH]c2c1c(ncn2)N3CCNCC3
COc1ccc(cc1)C(=O)N1CCN(CC1)c1ncnc2[nH]ccc12
COc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]ccc23)cc1
CCCNC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccccc1
Clc1ccccc1NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccccc1
COc1cccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccccc2)c1
COc1cc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccccc2)cc(OC)c1
COc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccccc2)cc1
Fc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccccc2)cc1
Fc1ccc(NC(=O)N2CCN(CC2)c2ncnc3[nH]c(cc23)-c2ccccc2)cc1
COc1cc2ncnc(-c3ccc(cc3F)S(=O)(=O)Nc3ccc(Cl)cc3)c2cc1OCCCN1CCOCC1
COc1cc2ncnc(-c3ccc(cc3F)S(=O)(=O)Nc3ccc(F)cc3)c2cc1OCCCN1CCOCC1
COc1ccc(cc1)S(=O)(=O)Nc1ccc(c(F)c1)-c1ncnc2cc(OC)c(OCCCN3CCOCC3)cc12
COc1cc2ncnc(-c3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3F)c2cc1OCCCN1CCOCC1
COc1cc2ncnc(-c3ccc(NS(=O)(=O)C4CC4)cc3F)c2cc1OCCCN1CCOCC1
COc1cc2ncnc(-c3ccc(NS(C)(=O)=O)cc3F)c2cc1OCCCN1CCOCC1
COc1cc2c(ncnc2cc1OCCCN1CCCCC1)-c1ccc(NS(=O)(=O)N2CCCC2)cc1F
COc1cc2c(ncnc2cc1OCCCN1CCCCC1)-c1ccc(NS(C)(=O)=O)cc1F
COc1ccc(cc1)S(=O)(=O)Nc1ccc(c(F)c1)-c1ncnc2cc(OCCCN3CCCCC3)c(OC)cc12
COc1cc2c(ncnc2cc1OCCCN1CCCCC1)-c1ccc(NS(=O)(=O)c2ccc(Cl)cc2)cc1F
COc1cc2c(ncnc2cc1OCCCN1CCCCC1)-c1ccc(NS(=O)(=O)C2CC2)cc1F
COCCOc1cc2ncnc(-c3ccc(NS(=O)(=O)c4ccc(OC(F)F)cc4)cc3F)c2cc1OCCOC
COCCOc1cc2ncnc(-c3ccc(NS(=O)(=O)c4cccc(F)c4)cc3F)c2cc1OCCOC
COCCOc1cc2ncnc(-c3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3F)c2cc1OCCOC
COCCOc1cc2ncnc(-c3ccc(NS(=O)(=O)c4ccc(OC)cc4)cc3F)c2cc1OCCOC
COCCOc1cc2ncnc(-c3ccc(NS(=O)(=O)C4CC4)cc3F)c2cc1OCCOC
COCCOc1cc2ncnc(-c3ccc(NS(C)(=O)=O)cc3F)c2cc1OCCOC
Fc1cc(NS(=O)(=O)C2CC2)ccc1-c1ncnc2cc3OCCOc3cc12
CS(=O)(=O)Nc1ccc(c(F)c1)-c1ncnc2cc3OCCOc3cc12
COc1cc2ncnc(-c3ccc(N)cc3F)c2cc1OC
COc1cc2ncnc(-c3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3F)c2cc1OC
CCCS(=O)(=O)Nc1ccc(c(F)c1)-c1ncnc2cc(OC)c(OC)cc12
COc1cc2ncnc(-c3ccc(NS(=O)(=O)C4CC4)cc3F)c2cc1OC
COc1cc2ncnc(-c3ccc(NS(C)(=O)=O)cc3F)c2cc1OC
COc1cc2ncnc(-c3ccc(NS(C)(=O)=O)c(F)c3)c2cc1OC
COc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1F)-c1ncnc2cc(OC)c(OC)cc12
COc1cc2ncnc(-c3ccc(NS(=O)(=O)N4CCCC4)c(F)c3)c2cc1OC
CCCS(=O)(=O)Nc1ccc(cc1F)-c1ncnc2cc(OC)c(OC)cc12
Cc1ccc(cn1)-c1cc2c(ncnc2[nH]1)C1=CCC(CC1)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1 |t:19|
CCCc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]c(C)cc12
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2cccc(C)c2)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2cccc(OC(F)(F)F)c2)cc1
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)C1=CCC(CC1)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1 |t:18|
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(C)nc2)cc1F
CCCCc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]c(C)cc12
CCCCS(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]c(C)cc12
CCCS(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]c(C)cc12
Fc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]c(cc12)C1CCCC1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(C)s2)cc1F
CCc1ccc(cc1)S(=O)(=O)Nc1ccc(c(F)c1)-c1ncnc2[nH]c(C)cc12
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(C)cc2)cc1F
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc3OCOc3c2)cc1
CC1(C)CC(=CC(C)(C)N1)c1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1 |c:4|
Fc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]c(cc12)C1=CCCC1 |t:30|
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(nc2)C(F)(F)F)cc1
CC1(C)CC(=CC(C)(C)O1)c1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1 |c:4|
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2cc(Cl)c(Cl)s2)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2sc(C)nc2C)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(C)nc2)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc3CCCc3c2)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc3oncc3c2)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2cc(Cl)cs2)cc1
Cc1csc(c1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]c(C)cc12
CC(C)c1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]c(C)cc12
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc3OCCc3c2)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2cc3cc(C)ccc3s2)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2cc3ccccc3s2)cc1
CC(C)Oc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]c(C)cc12
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(cn2)C(F)(F)F)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(C)s2)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(F)c(F)c2)cc1
CCc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]c(C)cc12
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(Cl)c(Cl)c2)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(Br)cc2)cc1
CNS(=O)(=O)c1cccc(c1)-c1ncnc2[nH]c(C)cc12
Cc1cc2c(ncnc2[nH]1)-c1cccc(NS(C)(=O)=O)c1
Fc1ccc(cc1)S(=O)(=O)Nc1ccc(c(F)c1)-c1ncnc2[nH]c(cc12)C1=CCCC1 |t:31|
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2cnn(c2)C(F)F)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(Cl)s2)cc1
COc1ccc(cn1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]c(C)cc12
COc1ccc(cc1F)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]c(C)cc12
COc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]c(C)cc12
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)-c1ccc(cc1F)S(=O)(=O)Nc1ccc(Cl)cc1
Fc1ccc(NS(=O)(=O)c2ccc(c(F)c2)-c2ncnc3[nH]c(cc23)-c2ccc(F)cc2)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(OC(F)F)cc2)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(Cl)cc2)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1
Fc1ccc(cc1)S(=O)(=O)Nc1ccc(c(F)c1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1F
CS(=O)(=O)Nc1ccc(c(F)c1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1F
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2cc(F)ccc2F)cc1F
Cc1cc2c(ncnc2[nH]1)-c1ccc(cc1F)S(=O)(=O)Nc1ccc(F)cc1
Fc1ccc(F)c(c1)-c1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(Cl)cc2)cc1F
Fc1ccc(F)c(c1)-c1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)C2CC2)cc1F
CS(=O)(=O)Nc1ccc(c(F)c1)-c1ncnc2[nH]c(cc12)-c1cc(F)ccc1F
Fc1ccc(-c2cc3c(ncnc3[nH]2)-c2ccc(NS(=O)(=O)C3CC3)cc2F)c(F)c1
Nc1ccc(c(F)c1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1F
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2cc(F)cc(F)c2)cc1F
Cc1cc2c(ncnc2[nH]1)-c1ccc(c(F)c1)S(=O)(=O)Nc1ccc(F)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(Cl)cc2)c(F)c1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2)c(F)c1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(F)cc2)c(F)c1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2cccc(F)c2)c(F)c1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(Cl)cc2)cc1F
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(C)c(F)c2)c(F)c1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2F)c(F)c1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(Cl)cc2F)cc1F
CS(=O)(=O)Nc1ccc(c(F)c1F)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Fc1ccc(CNS(=O)(=O)c2ccc(c(F)c2)-c2ncnc3[nH]c(cc23)-c2ccc(F)cc2)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2)cc1F
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2cccc(F)c2)cc1F
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(OC(F)F)cc2)c(F)c1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(Cl)cc2F)c(F)c1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1F
COc1ccc(cc1)S(=O)(=O)Nc1ccc(c(F)c1)-c1ncnc2[nH]c(C)cc12
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2cccc(Cl)c2F)cc1F
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(C)c(F)c2)cc1F
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(OC(F)F)cc2)cc1F
CS(=O)(=O)Nc1ccc(cc1F)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
CS(=O)(=O)Nc1ccc(c(F)c1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)-c1ccc(cc1F)S(=O)(=O)NCC1CC1
CS(=O)(=O)Nc1ccccc1-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
NS(=O)(=O)c1ccc(c(F)c1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(C)(=O)=O)cc1
Cc1cc2c(ncnc2[nH]1)-c1ccc(cc1)S(=O)(=O)NC1CC1
CCS(=O)(=O)Nc1ccc(c(F)c1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
CS(=O)(=O)Nc1ccc(-c2cc3c(ncnc3[nH]2)-c2ccc(NS(C)(=O)=O)cc2F)c(F)c1
O=S(=O)(Nc1cccc(c1)-c1ncnc2[nH]c(cc12)-c1cnc(nc1)C1CC1)C1CC1
C1CC1c1ncc(cn1)-c1cc2c(ncnc2[nH]1)-c1cnc(nc1)C1CC1
NS(=O)(=O)c1ccc(cc1)-c1ncnc2[nH]c(cc12)-c1cnc(nc1)C1CC1
Fc1cc(NSC2CC2)ccc1-c1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)C2CC2)cc1F
CCCCS(=O)(=O)Nc1ccc(cc1)-c1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)CCCC)cc1
O=S(=O)(Nc1ccc(cc1)-c1ncnc2[nH]c(cc12)-c1ccc(NSC2CC2)cc1)C1CC1
Cc1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(C)cc2)cc1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(Cl)cc2)cc1F
CCCS(=O)(=O)Nc1ccc(c(F)c1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)N2CCCC2)cc1F
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)C2CC2)cc1F
COc1ccc(cc1)S(=O)(=O)Nc1ccc(c(F)c1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
CCCS(=O)(=O)Nc1ccc(cc1F)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)N2CCCC2)c(F)c1
CCS(=O)(=O)Nc1cccc(c1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(F)cc2)c(F)c1
COc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1F)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)C2CC2)c(F)c1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)N2CCCC2)cc1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)-c1cccc(NS(=O)(=O)C2CC2)c1
CS(=O)(=O)Nc1cccc(c1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)-c1ccc(NCc2ccc(nc2)C(F)(F)F)nc1
Nc1ccc(cc1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
CCNc1ccc(cn1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
NS(=O)(=O)c1ccc(cc1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
CCCCS(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)C2CC2)cc1
CCNS(=O)(=O)c1ccc(cc1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
COc1ccc(CNS(=O)(=O)c2ccc(cc2)-c2ncnc3[nH]c(cc23)-c2ccc(F)cc2)cc1
Cc1ccc(NS(=O)(=O)c2ccc(cc2)-c2ncnc3[nH]c(cc23)-c2ccc(F)cc2)cc1
Fc1ccc(NS(=O)(=O)c2ccc(cc2)-c2ncnc3[nH]c(cc23)-c2ccc(F)cc2)cc1
Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)-c1cccc(c1)S(=O)(=O)NC1CC1
CNS(=O)(=O)c1ccc(cc1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
CCS(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
CS(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Cc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
CCCS(=O)(=O)Nc1cccc(c1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Cc1ccc(cc1)S(=O)(=O)Nc1cccc(c1)-c1ncnc2[nH]c(cc12)-c1ccc(F)cc1
Cc1n[nH]c2ncnc(-c3ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)cc3)c12
Cc1n[nH]c2ncnc(-c3ccc(NS(=O)(=O)c4ccc(F)cc4)cc3)c12
Cc1n[nH]c2ncnc(-c3ccc(NS(=O)(=O)c4cccc(F)c4)cc3)c12
Cc1n[nH]c2ncnc(-c3ccc(NS(=O)(=O)c4ccc(nc4)C(F)(F)F)cc3)c12
CCc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]nc(C)c12
Cc1n[nH]c2ncnc(-c3ccc(NS(=O)(=O)c4cccc(Cl)c4)cc3)c12
COc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]nc(C)c12
Cc1n[nH]c2ncnc(-c3ccc(NS(=O)(=O)c4ccc(Cl)cc4)cc3)c12
Cc1n[nH]c2ncnc(-c3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3)c12
Cc1c[nH]c2ncnc(-c3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3)c12
Cc1[nH]c2ncnc(-c3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3)c2c1C
Cc1nc2c(ncnc2[nH]1)-c1ccc(NS(=O)(=O)c2ccc(C)cc2)cc1
Cc1ccc(cc1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(C)c1
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc2CCCc2c1
Cc1csc(c1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(C)c1
Cc1ccc(s1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(C)c1
Cc1ccc2sc(cc2c1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(C)c1
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc2OCOc2c1
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc2OCCc2c1
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(Cl)s1
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1cc(Cl)c(Cl)s1
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1cc(Cl)cs1
Cc1ncc(s1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1
COc1ncc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1
Clc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1cc2ccccc2s1
CC(C)Oc1ccc(cc1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(Cl)cc1
CN(C)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(C)c1
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1cc2ccccc2s1
Clc1ccc(cc1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(cc12)C#CC1CC1
Clc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1cccc(Cl)c1
Fc1ccc(cc1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(Cl)cc1
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(cc1)N1CCCC1=O
CCCn1cc(cn1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(C)c1
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(cc1)C1(CC1)C#N
CC(C)Oc1ccc(cc1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(C)c1
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(F)cc1
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(Cl)cc1
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccccc1OC(F)(F)F
COc1ccc(cc1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(C)c1
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1
FC(F)(F)Oc1cccc(c1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(Cl)cc1
Cn1cc(cn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1cccc(OC(F)(F)F)c1
Cc1nc(no1)-c1cccc(NC(=O)NC2CCN(CC2)c2ncnc3[nH]ccc23)c1
O=C(NC1CCN(CC1)c1ncnc2[nH]ccc12)Nc1cccnc1
Fc1ccc(CNC(=O)NC2CCN(CC2)c2ncnc3[nH]ccc23)cc1
Fc1cccc(CNC(=O)NC2CCN(CC2)c2ncnc3[nH]ccc23)c1
Fc1ccc(CCNC(=O)NC2CCN(CC2)c2ncnc3[nH]ccc23)cc1
Fc1ccc(NC(=O)NC2CCN(CC2)c2ncnc3[nH]ccc23)cc1Cl
FC(F)(F)Oc1ccc(NC(=O)NC2CCN(CC2)c2ncnc3[nH]ccc23)cc1
FC(F)(F)c1ccc(NC(=O)NC2CCN(CC2)c2ncnc3[nH]ccc23)cc1
FC(F)(F)c1cccc(NC(=O)NC2CCN(CC2)c2ncnc3[nH]ccc23)c1
CCc1ccc(cc1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]ccc12
Fc1ccc(F)c(c1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]ccc12
COc1ccc(cc1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]ccc12
NC1CCN(CC1)c1ncnc2[nH]ccc12
COc1ccc(NC(=O)NC2CCN(CC2)c2ncnc3[nH]ccc23)cc1
Fc1ccc(NC(=O)N2CC3CCC2CN3c2ncnc3cc(sc23)-c2ccc(F)cc2)cc1
COc1cccc(CNC(=O)N2CC3CCC2CN3c2ncnc3cc(sc23)-c2ccc(F)cc2)c1
COc1cccc(c1)[C@H](C)NC(=O)N1CC2CCC(C1)N2c1ncnc2cc(sc12)-c1ccc(F)cc1 |r|
COc1cccc(CNC(=O)N2CC3CCC(C2)N3c2ncnc3cc(sc23)-c2ccc(F)cc2)c1
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2cc(sc12)C1=CCN(CC1)C(=O)C1CC1)c1cccc(Cl)c1 |r,t:25|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2cc(sc12)C1=CCN(CC1)S(C)(=O)=O)c1cccc(Cl)c1 |r,t:25|
O=C(N1CCOCC1)N1CCC(=CC1)c1cc2ncnc(-c3ccc(NS(=O)(=O)C4CC4)cc3)c2s1 |c:12|
CS(=O)(=O)Nc1ccc(cc1)-c1ncnc2cc(sc12)C1=CCN(CC1)C(=O)N1CCOCC1 |t:23|
COc1cc(ccn1)-c1cc2ncnc(N3CCN(C(=O)N[C@@H](C)c4cccc(Cl)c4)C(C)(C)C3)c2s1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2cc(sc12)-c1sc(C)nc1C)c1cccc(Cl)c1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2cc(sc12)N1CCOCC1)c1cccc(Cl)c1 |r|
CC(=N)Nc1ccc(cc1)-c1ncnc2cc(sc12)C1=CCN(CC1)C(=O)N1CCOCC1 |t:22|
COc1cccc(c1)[C@H](C)NC(=O)N1CCN(CC1(C)C)c1ncnc2cc(sc12)N1CCOCC1 |r|
Fc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2cc(sc12)C1=CCN(CC1)C(=O)N1CCOCC1 |t:30|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2cc(sc12)-c1cn(C)nc1C)c1cccc(Cl)c1 |r|
COc1cccc(c1)[C@H](C)NC(=O)N1CC2CCC1CN2c1ncnc2cc(sc12)-c1ccc(F)cc1 |r|
COc1cccc(c1)[C@H](C)NC(=O)N1C2CCC1CN(C2)c1ncnc2cc(sc12)-c1ccc(F)cc1 |r|
CS(=O)(=O)N1CCC(=CC1)c1cc2ncnc(N3CCN(CC3)C(=O)NCc3ccc(F)cc3)c2s1 |c:7|
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2cc(sc12)C1=CC(C)(C)NC(C)(C)C1)c1cccc(Cl)c1 |r,t:23|
Fc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2cc(sc12)C1=CCN(CC1)C(=O)C1CC1 |t:30|
O=C(C1CC1)N1CCC(=CC1)c1cc2ncnc(-c3ccc(NS(=O)(=O)C4CC4)cc3)c2s1 |c:9|
CS(=O)(=O)Nc1ccc(cc1)-c1ncnc2cc(sc12)C1=CCN(CC1)C(=O)C1CC1 |t:23|
C[C@H](NC(=O)N1CCC(=CC1)c1ncnc2cc(sc12)-c1ccc(F)cc1)c1cccc(OC(F)F)c1 |r,c:8|
COc1cccc(c1)[C@H](C)NC(=O)N1CCN(CC1)c1ncnc2cc(sc12)C1=CC(C)(C)NC(C)(C)C1 |r,t:32|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2cc(sc12)-c1ccc(F)cc1)c1ccc(Cl)cc1 |r|
COc1ccc(cc1)[C@H](C)NC(=O)N1CCN(CC1(C)C)c1ncnc2cc(sc12)-c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2cc(sc12)-c1ccc(F)cc1)c1cccc(OC(F)F)c1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2cc(sc12)-c1ccc(F)cc1)c1cccc(F)c1 |r|
C[C@H](NC(=O)N1CCC(=CC1)c1ncnc2cc(sc12)-c1ccc(F)cc1)c1cccc(Cl)c1 |r,c:8|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2cc(sc12)-c1ccc(F)cc1)c1cccc(Cl)c1 |r|
COc1cccc(c1)[C@H](C)NC(=O)N1CCC(=CC1)c1ncnc2cc(sc12)-c1ccc(F)cc1 |r,c:17|
COc1cccc(c1)[C@H](C)NC(=O)N1CCC(=CC1)c1ncnc2cc(sc12)-c1cn(C)nc1C |r,c:17|
Cc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2cc(sc12)C1=CCN(CC1)C(=O)C1CC1 |t:30|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2cc(sc12)-c1cn(C)nc1C)c1cccc(F)c1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2cc(sc12)-c1ccc(F)cc1)c1cccc(F)c1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2cc(sc12)-c1ccc(F)cc1)c1cccc(OC(F)F)c1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2cc(sc12)-c1cn(C)nc1C)c1cccc(OC(F)F)c1 |r|
Fc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3cc(sc23)C2CCN(CC2)C(=O)C2CC2)cc1
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2cc(sc12)N1CCOCC1)c1ccc(F)cc1 |r|
Cc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2cc(sc12)C1=CCN(CC1)C(=O)N1CCOCC1 |t:30|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2cc(sc12)-c1cn(C)nc1C)c1cccc(Cl)c1 |r|
Cc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2cc(sc12)C1CCNCC1
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2cc(sc12)-c1ccc(F)cc1)c1ccc(F)cc1 |r|
COc1cccc(c1)[C@H](C)NC(=O)N1CCN(CC1(C)C)c1ncnc2cc(sc12)-c1ccc(F)cc1 |r|
CC1(C)CN(CCN1)c1ncnc2cc(sc12)-c1ccc(F)cc1
Fc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3cc(sc23)C2CCNCC2)cc1
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2cc(Br)sc12)c1ccc(F)cc1 |r|
COc1cccc(c1)[C@H](C)NC(=O)N1CCN(C[C@H]1C)c1ncnc2cc(sc12)-c1cn(C)nc1C |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2cc(sc12)-c1cn(C)nc1C)c1ccc(F)cc1 |r|
COc1cccc(c1)[C@H](C)NC(=O)N1CCN(C[C@H]1C)c1ncnc2cc(sc12)-c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2cc(sc12)-c1ccc(F)cc1)c1ccc(F)cc1 |r|
C[C@@H]1CN(CCN1C(=O)NCc1ccc(F)cc1)c1ncnc2cc(sc12)-c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCC(CC1)c1ncnc2cc(sc12)-c1cn(C)nc1C)c1ccc(F)cc1 |r|
Cc1nn(C)cc1-c1cc2ncnc(C3CCN(CC3)C(=O)NCc3ccc(F)cc3)c2s1
COc1cccc(c1)[C@@H](C)NC(=O)N1CCN(C[C@H]1C)c1ncnc2cc(sc12)-c1ccc(F)cc1 |r|
C[C@@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2cc(sc12)-c1ccc(F)cc1)c1ccc(F)cc1 |r|
Cc1nn(C)cc1-c1cc2ncnc(C3CCNCC3)c2s1
COc1cccc(c1)[C@@H](C)NC(=O)N1CCN(C[C@H]1C)c1ncnc2cc(sc12)-c1cn(C)nc1C |r|
C[C@@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2cc(sc12)-c1cn(C)nc1C)c1ccc(F)cc1 |r|
C[C@@H]1CN(CCN1C(=O)NCc1ccc(F)cc1)c1ncnc2cc(sc12)-c1cn(C)nc1C |r|
Cc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2cc(sc12)C1=CCNCC1 |t:30|
Cc1nn(C)cc1-c1cc2ncnc(C3=CCN(CC3)C(=O)Nc3ccc(Cl)cc3)c2s1 |t:15|
Cc1nn(C)cc1-c1cc2ncnc(C3=CCN(CC3)C(=O)NCc3ccc(F)cc3)c2s1 |t:15|
Cc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2cc(sc12)C1=CCN(CC1)C(=O)OC(C)(C)C |t:30|
Fc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3cc(sc23)C2=CCNCC2)cc1 |t:27|
CC(C)(C)OC(=O)N1CCC(=CC1)c1cc2ncnc(N3CCN(CC3)C(=O)NCc3ccc(F)cc3)c2s1 |c:10|
Cn1cc(cn1)-c1cc2ncnc(N3CC(C)(C)NC(C)(C)C3)c2s1
Cc1nn(C)c(C)c1-c1cc2ncnc(N3CCN(CC3)C(=O)NCc3ccc(F)cc3)c2s1
Cc1nn(C)cc1-c1cc2ncnc(N3CCN(CC3)C(=O)NCc3ccc(F)cc3)c2s1
Cc1c(cnn1C)-c1cc2ncnc(N3CCN(CC3)C(=O)NCc3ccc(F)cc3)c2s1
Cn1cc(cn1)-c1cc2ncnc(-c3ccc(N)nc3)c2s1
Cc1cc2ncnc(-c3ccc(NS(C)(=O)=O)cc3)c2s1
Cc1cc2ncnc(-c3ccc(NS(=O)(=O)c4ccc(C)cc4)cc3)c2s1
Fc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3cc(sc23)-c2cnn(CCN3CCOCC3)c2)cc1
Cn1cc(cn1)-c1cc2ncnc(N3CCN(CC3)C(=O)NCc3ccccc3)c2s1
Brc1cc2ncnc(N3CCN(CC3)C(=O)NCc3ccccc3)c2s1
CCS(=O)Nc1ccc(cc1)-c1ncnc2cc(sc12)-c1ccc(F)cc1
CC(=O)Nc1ccc(cc1)-c1ncnc2cc(sc12)-c1ccc(F)cc1
Nc1ccc(cc1)-c1ncnc2cc(sc12)-c1ccc(F)cc1
Fc1ccc(cc1)-c1cc2ncnc(-c3ccc(cc3)S(=O)(=O)NCc3ccccc3)c2s1
Cc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2cc(sc12)-c1ccc(F)cc1
Fc1ccc(CNC(=O)N2CCN(CC2)c2ncnc3ccsc23)cc1
Fc1ccc(NC(=O)N2CCN(CC2)c2ncnc3ccsc23)cc1
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(C)cc12)c1cccc(Cl)c1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1ccc(F)cc1 |r|
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCN(C(=O)N[C@@H](C)c2ccc(F)cc2)C(C)(C)C1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(C)cc12)c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(C)cc12)c1cccc(OC(F)F)c1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(C)cc12)c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(C)cc12)c1cccc(Cl)c1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(C)cc12)c1cccc(OC(F)F)c1 |r|
COc1cc(ccc1Cl)[C@H](C)NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1 |r|
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCN(C(=O)N[C@@H](C)c2cccc(Cl)c2)C(C)(C)C1 |r|
CCCc1ccc(cc1)S(=O)(=O)NC1CCC(=CC1)c1ncnc2[nH]c(C)cc12 |c:17|
CC(C)Oc1ccc(cc1)S(=O)(=O)NC1CCC(=CC1)c1ncnc2[nH]c(C)cc12 |c:18|
Cc1cc2c(ncnc2[nH]1)C1=CCC(CC1)NS(=O)(=O)c1ccc(OC(F)F)cc1 |t:12|
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)C1=CCC(CC1)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1 |t:20|
FC(F)Oc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1ncnc2[nH]c(Cl)cc12
Cc1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(OC(F)F)cc1
CC(C)c1ccc(cc1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(C)cc12
CCCc1ccc(cc1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(C)cc12
Cc1nn(C)cc1-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(C)cc1
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(C)cc1
Cc1csc(c1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1
CC1(C)CC(=CC(C)(C)N1)c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1 |c:4|
CC1(C)CC(=CC(C)(C)O1)c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1 |c:4|
Cc1nc(C)c(s1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1
CCc1ccc(s1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(C)c1
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(Cl)cc1
Cc1nn(C)cc1-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(Cl)cc1
Cc1nn(C)cc1-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1
FC(F)(F)Oc1ccc(cc1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(cc12)C1=CCCC1 |t:34|
CC1CN(CCC1NS(=O)(=O)c1ccc(C)cc1)c1ncnc2[nH]c(cc12)-c1cnn(C)c1
CN(C)c1ncc(s1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1
CCc1ccc(cc1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(C)cc12
Cc1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(C)cc1
CCc1ccc(cc1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cnn(C)c1
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2ccsc12)c1cccc(Cl)c1 |r|
CC(C)(NC(=O)N1CCN(CC1(C)C)c1ncnc2cc(sc12)-c1ccc(F)cc1)c1ccccc1
CC(C)(NC(=O)N1CCC(=CC1)c1ncnc2cc(sc12)-c1ccc(F)cc1)c1ccccc1 |c:9|
COc1cccc(c1)[C@H](C)NC(=O)N1CCN(CC1(C)C)c1ncnc2cc(sc12)N1CCC(F)(F)CC1 |r|
CCOC(=O)N1CCN(CC1)c1cc2ncnc(N3CCN(C(=O)N[C@@H](C)c4cccc(OC)c4)C(C)(C)C3)c2s1 |r|
COc1cccc(c1)[C@H](C)NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(C)cc12 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(C)cc12)c1cccc(F)c1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N)c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N)c1ccc(Cl)cc1 |r|
COc1cccc(c1)[C@H](C)NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N)c1cccc(F)c1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N)c1cccc(Cl)c1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N)c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N)c1ccc(Cl)cc1 |r|
COc1cccc(c1)[C@H](C)NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N)c1cccc(F)c1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N)c1cccc(Cl)c1 |r|
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCN([C@H](C)C1)C(=O)N[C@@H](C)c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N)c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N)c1cccc(Cl)c1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N)c1cccc(OC(F)F)c1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N)c1cccc(OC(F)F)c1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1ccc(Cl)cc1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1cccc(Cl)c1 |r|
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(cc1)C#N)c1ccc(Cl)cc1 |r|
CC(NC(=O)N1CCN(CC1)c1ncnc2cc(sc12)-c1ccc(F)cc1)c1ccc(C)s1
C[C@@H](NC(=O)N1CC2CCC1CN2c1ncnc2cc(sc12)-c1cn(C)nc1C)c1ccc(F)cc1 |r|
Fc1ccc(cc1)-c1cc2ncnc(N3CCN(CC3)C(=O)NCc3cccs3)c2s1
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCN(C(=O)N[C@@H](C)c2ccc(Cl)cc2)C(C)(C)C1 |r|
COc1cc(ccn1)-c1cc2c(ncnc2[nH]1)N1CCN([C@H](C)C1)C(=O)N[C@@H](C)c1cccc(Cl)c1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1ccc(C)cc1 |r|
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1ccc(C)cc1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1cn(C)nc1C)c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cn(C)nc1C)c1ccc(Cl)cc1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1cnn(C)c1)c1ccc(Cl)cc1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1cn(C)nc1C)c1ccc(Cl)cc1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1ccc(F)cc1)c1ccc(C)cc1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1cnn(C)c1)c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1cn(C)nc1C)c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1cnn(C)c1)c1ccc(Cl)cc1 |r|
C[C@H](NC(=O)N1CCN(CC1(C)C)c1ncnc2[nH]c(cc12)-c1cn(C)nc1C)c1ccc(Cl)cc1 |r|
C[C@H](NC(=O)N1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cn(C)nc1C)c1ccc(F)cc1 |r|
C[C@H](NC(=O)N1CCN(C[C@H]1C)c1ncnc2[nH]c(cc12)-c1cnn(C)c1)c1ccc(F)cc1 |r|
CCc1ccc(cc1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(cc12)-c1cn(C)nc1C
CCc1ccc(cc1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(cc12)-c1ccnc(OC)c1
Cc1cc2c(ncnc2[nH]1)N1CCC(CC1)NS(=O)(=O)c1ccc(Cl)cc1
Cc1cc2c(ncnc2[nH]1)C1=CCC(CC1)NS(=O)(=O)c1ccc(Cl)cc1 |t:12|
CCc1ccc(s1)S(=O)(=O)NC1CCN(CC1)c1ncnc2[nH]c(C)cc12
NC(=O)c1cccc(NC(=O)c2cnc3[nH]c(cc3c2)-c2ccccc2)c1
Brc1cn[nH]c1C(=O)Nc1cnc2[nH]c(cc2c1)-c1ccccc1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccccc2)c1C
O=C(Nc1cnc2[nH]c(cc2c1)-c1ccccc1)c1cc(n[nH]1)C1CC1
Fc1ccc2[nH]nc(C(=O)Nc3cnc4[nH]c(cc4c3)-c3ccccc3)c2c1
O=C(Nc1cnc2[nH]c(cc2c1)-c1ccccc1)c1ccncn1
Fc1cccnc1C(=O)Nc1cnc2[nH]c(cc2c1)-c1ccccc1
Cc1noc(C)c1C(=O)Nc1cnc2[nH]c(cc2c1)-c1ccccc1
O=C(Nc1cnc2[nH]c(cc2c1)-c1ccccc1)c1cn[nH]n1
Cc1cccnc1C(=O)Nc1cnc2[nH]c(cc2c1)-c1ccccc1
Cc1onc(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccccc2)c1C
O=S(=O)(Nc1cnc2[nH]c(cc2c1)-c1ccccc1)c1cn[nH]c1
Cc1cc([nH]n1)C(=O)Nc1cnc2[nH]c(cc2c1)-c1ccc(F)cc1
Fc1ccc(cc1)-c1cc2cc(NC(=O)c3cccc(CC#N)c3)cnc2[nH]1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(F)cc2)c1Cl
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(F)cc2)c1C
Fc1ccc(cc1)-c1cc2cc(NC(=O)c3cccc(c3)C#N)cnc2[nH]1
CC(=O)Nc1cccc(c1)C(=O)Nc1cnc2[nH]c(cc2c1)-c1ccc(F)cc1
Fc1ccc(cc1)-c1cc2cc(NC(=O)c3cccc4n[nH]cc34)cnc2[nH]1
Cc1c[nH]nc1C(=O)Nc1cnc2[nH]c(cc2c1)-c1ccc(F)cc1
CCn1nccc1S(=O)(=O)Nc1cnc2[nH]c(cc2c1)-c1ccc(F)cc1
Cc1cc(n[nH]1)C(=O)Nc1cnc2[nH]c(cc2c1)C1=CCN(CC1)C(=O)N1CCOCC1 |t:21|
Cc1n[nH]c(C(=O)Nc2cnc3[nH]ccc3c2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3n(c(cc3c2)C2=CCN(CC2)C(=O)N2CCOCC2)S(=O)(=O)c2ccccc2)c1C |t:19|
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)C2=CCN(CC2)C(=O)N2CCOCC2)c1C |t:19|
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)C2=CCN(CC2)C(=O)N2CCOCC2)c1Cl |t:19|
Cc1n[nH]cc1C(=O)Nc1cnc2[nH]c(cc2c1)-c1ccc(F)cc1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cn(C)nc2C)c1C
Cc1[nH]nc(C(=O)Nc2cnc3[nH]c(cc3c2)C2=CCN(CC2)C(=O)C2CC2)c1Cl |t:19|
Cc1n[nH]c(C(=O)Nc2cnc3[nH]nc(C)c3c2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]nc(-c4ccc(F)cc4)c3c2)c1C
Cc1cc(n[nH]1)C(=O)Nc1cnc2[nH]c(cc2c1)C1=CCN(CC1)C(=O)C1CC1 |t:21|
Cc1[nH]nc(C(=O)Nc2cnc3[nH]c(cc3c2)C2=CCN(CC2)C(=O)C2CC2)c1C |t:19|
Cc1n[nH]c(C(=O)Nc2cnc(Nc3ccccc3)nc2)c1C
Cc1n[nH]c(C(=O)Nc2ccc(Nc3ccccc3)nc2)c1C
Fc1ccc(cc1)-c1cc2cc(NC(=O)c3n[nH]c4ccccc34)cnc2[nH]1
Fc1ccc(cc1)-c1cc2cc(NC(=O)c3n[nH]c4CCCCc34)cnc2[nH]1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cnn(c2)C2CCNCC2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(Cl)cc3c2)c1C
CCNS(=O)(=O)c1cccc(Nc2ncc(NC(=O)c3[nH]nc(C)c3C)cn2)c1
Cc1n[nH]c(C(=O)Nc2cnc(Nc3cccc(c3)N3CCOCC3)nc2)c1C
CCCS(=O)(=O)Nc1cccc(Nc2ncc(NC(=O)c3[nH]nc(C)c3C)cn2)c1
Cc1n[nH]c(C(=O)Nc2cnc(Nc3cccc(NS(=O)(=O)c4ccccc4)c3)nc2)c1C
CNC(=O)c1cccc(Nc2ncc(NC(=O)c3[nH]nc(C)c3C)cn2)c1
CCOC(=O)Nc1cccc(Nc2ncc(NC(=O)c3[nH]nc(C)c3C)cn2)c1
Fc1ccc(cc1)-c1cc2cc(NC(=O)c3n[nH]c4CCCc34)cnc2[nH]1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)C2=CCN(CC2)S(C)(=O)=O)c1Cl |t:19|
Cc1cc([nH]n1)C(=O)Nc1cnc2[nH]c(cc2c1)N1CCOCC1
Cc1[nH]nc(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(cc2)N2CCOCC2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)C2=CCN(C2)C(=O)C2CC2)c1Cl |t:19|
CC(=O)N1CCC(=CC1)c1cc2cc(NC(=O)c3[nH]nc(C)c3Cl)cnc2[nH]1 |c:6|
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)C2=CCN(C2)C(=O)N2CCOCC2)c1Cl |t:19|
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)C#CCF)c1C
CN(C)c1cccc(c1)-c1cc2cc(NC(=O)c3[nH]nc(C)c3C)cnc2[nH]1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2c(C)noc2C)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cccc(OCCN3CCOCC3)c2)c1C
CNC(=O)c1ccc(cc1)-c1cc2cc(NC(=O)c3[nH]nc(C)c3C)cnc2[nH]1
Cc1cc([nH]n1)C(=O)Nc1cnc2[nH]c(cc2c1)C#CCF
CN1CCN(CC1)c1cc(ccn1)-c1cc2cc(NC(=O)c3n[nH]c(C)c3C)cnc2[nH]1
Cc1[nH]nc(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cccc(c2)N2CCOCC2)c1C
Cc1[nH]nc(NC(=O)c2cnc3[nH]c(cc3c2)-c2ccccc2)c1C
Cc1[nH]nc(C(=O)Nc2cnc3cc(nn3c2)-c2ccc(F)cc2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)C2=CCN(CC2)C(=O)CN2CCOCC2)c1C |t:19|
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)C2=CCN(CC2)C(=O)C(O)CO)c1C |t:19|
COc1ccc(-c2cc3cc(NC(=O)c4[nH]nc(C)c4C)cnc3[nH]2)c(Cl)c1
COc1ccc(-c2cc3cc(NC(=O)c4[nH]nc(C)c4C)cnc3[nH]2)c(F)c1
COc1ccc(Cl)c(c1)-c1cc2cc(NC(=O)c3[nH]nc(C)c3C)cnc2[nH]1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cc(F)cc(c2)N2CCOCC2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cccc(c2)N2CCCC2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)C2=CCC(N)CC2)c1C |t:19|
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(C#N)c(c2)N2CCOCC2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-n2cccn2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cc(OC(F)(F)F)ccc2Cl)c1C
Cc1cc2ncc(NC(=O)c3n[nH]c(C)c3C)cn2n1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)N2CCCC2)c1C
Cc1cc([nH]n1)C(=O)Nc1cnc2[nH]c(cc2c1)-n1cccn1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cccc(c2)N2CCN(CC2)C(=O)C2CC2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(C#N)c(c2)N2CCCC2)c1C
CNS(=O)(=O)c1cccc(c1)-c1cc2cc(NC(=O)c3[nH]nc(C)c3C)cnc2[nH]1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(Cl)cc2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(C)nc2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3sc(nc3c2)-c2ccccc2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2ccccc2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cccc(F)c2C)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(cc2)C(=O)NC2CC2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(OCC3(C)COC3)cc2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2ccccc2)c1Cl
Cc1cc([nH]n1)C(=O)Nc1cnc2[nH]c(nc2c1)-c1ccccc1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2ccccc2F)c1C
CCOc1ncc(cn1)-c1cc2cc(NC(=O)c3[nH]nc(C)c3C)cnc2[nH]1
CC(C)c1ncc(cn1)-c1cc2cc(NC(=O)c3[nH]nc(C)c3C)cnc2[nH]1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cnc(nc2)C2CC2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cnc(NC3CC3)nc2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cnc(nc2)N2CCOCC2)c1C
CCc1cc([nH]n1)C(=O)Nc1cnc2[nH]c(cc2c1)-c1ccc(F)cc1
CN1CCN(CC1)c1ncc(cn1)-c1cc2cc(NC(=O)c3[nH]nc(C)c3C)cnc2[nH]1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(cc2C)C#N)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]nc(-c4cccc(c4)N4CCN(CC4)C(=O)OC(C)(C)C)c3c2)c1C
CC(C)c1cc(ccn1)-c1cc2cc(NC(=O)c3[nH]nc(C)c3C)cnc2[nH]1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2c(C)nn(C)c2C)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]nc(-c4cccc(c4)N4CCNCC4)c3c2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2c(C)n[nH]c2C)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cn(nc2C)C2COC2)c1C
COc1ccc(-c2cc3cc(NC(=O)c4[nH]nc(C)c4C)cnc3[nH]2)c(C)n1
FC(F)c1cc([nH]n1)C(=O)Nc1cnc2[nH]c(cc2c1)-c1ccc(F)cc1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(F)c(c2)-c2nn[nH]n2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccnc(c2)C(=O)NC2CC2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cccnc2C(F)(F)F)c1C
CCc1cc(ccn1)-c1cc2cc(NC(=O)c3[nH]nc(C)c3C)cnc2[nH]1
CCc1ccc(cn1)-c1cc2cc(NC(=O)c3[nH]nc(C)c3C)cnc2[nH]1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccnc3OCCOc23)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccccc2C(F)(F)F)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(C)cc2C)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccccc2OC(F)(F)F)c1C
COc1cncc(c1)-c1cc2cc(NC(=O)c3[nH]nc(C)c3C)cnc2[nH]1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cncc(C)c2)c1C
COc1ccncc1-c1cc2cc(NC(=O)c3[nH]nc(C)c3C)cnc2[nH]1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccnc(c2)N2CCN(CC2)S(C)(=O)=O)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccnc(c2)N2CCN(CC2)C(=O)C2CC2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(I)cc3c2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccnc(c2)N2CCN(CC2)C(=O)CC#N)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(F)cc2OC(F)F)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(F)nc2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cncc(c2)C#N)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)C2=CCOCC2)c1C |t:19|
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cnccc2C(N)=O)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cccc3CCOc23)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cccc(c2)N2CCNCC2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(F)cc2)c1F
CC(C)CNC(=O)c1cccc(c1)-c1cc2cc(NC(=O)c3[nH]nc(C)c3C)cnc2[nH]1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(Cl)cc2C)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccncc2Cl)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(F)nc2F)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cccc3OC(F)(F)Oc23)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cnc(C)c(C)c2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(F)nc2C)c1C
COc1ccc(-c2cc3cc(NC(=O)c4[nH]nc(C)c4C)cnc3[nH]2)c(C)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cn(nc2C)C2CN(C2)C(=O)OC(C)(C)C)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cn(nc2C)C2CNC2)c1C
Cc1c(n[nH]c1C(=O)Nc1cnc2[nH]c(cc2c1)-c1ccc(F)cc1)C(F)F
Ic1cc2cc(NC(=O)c3cccc4n[nH]cc34)cnc2[nH]1
O=C(Nc1cnc2[nH]c(cc2c1)-c1ccccc1)c1cccc2n[nH]cc12
COC(=O)c1cccc(c1)C(=O)Nc1cnc2[nH]c(cc2c1)-c1ccccc1
OC(=O)c1cccc(c1)C(=O)Nc1cnc2[nH]c(cc2c1)-c1ccccc1
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(C(O)=O)c(F)c2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cccc(CC(O)=O)c2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(cc2)C2(CC2)C(O)=O)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(CC(O)=O)cc2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(C(O)=O)c(C)c2)c1C
Cc1n[nH]c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2cccc(C(O)=O)c2C)c1C
C(c1ccccc1)c1cnc(nc1)N1CCN(CC1)c1ncnc2[nH]cnc12
C(c1ccccc1)c1cnc(nc1)N1CCN(CC1)c1ncnc2CNCc12
C(c1ccccc1)c1cnc(nc1)N1CCN(CC1)c1ncnc2ccccc12
COc1ccc2c(ncnc2c1)N1CCN(CC1)c1ncc(Cc2ccccc2)cn1
COc1ccc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2c1
COc1cc2ncnc(N3CCN(CC3)c3ncc(OCC4CC4)cn3)c2cc1OC
COc1ccc2ncnc(N3CCN([C@H](C)C3)c3ncc(Cc4ccccc4)cn3)c2c1 |r|
COc1ccc2c(ncnc2c1)N1CCN(CC1)c1ncc(OCc2ccccc2)cn1
COc1cc2ncnc(N3CCN(CC3)c3ncc(cn3)-c3ccccc3)c2cc1OC
COc1ccc2ncnc(N3CCN(CC3)c3ncc(OCc4ccccc4)cn3)c2c1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3nccc(Cc4ccccc4)n3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Nc4ccccc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Oc4ccccc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Nc4ccccn4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Nc4cccnc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Nc4ccncc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(OCC4CCCC4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(cn3)-c3ccc(cc3)C#N)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1C(N)=O
COc1cc2ncnc(N3CCN(C(=O)C3)c3ncc(Cc4ccccc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(C(=O)C3)c3ncc(Cc4ccc(C)cc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(C(C)C3)c3ncc(Cc4ccccc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(CCc4ccccc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4C)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(C[C@@H]3C)c3ncc(Cc4ccccc4)cn3)c2cc1OC |r|
COc1cc2ncnc(N3CCN(C[C@H]3C)c3ncc(Cc4ccccc4)cn3)c2cc1OC |r|
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)c(N)n3)c2cc1OC
COc1cc2ncnc(N3CCN([C@H](C)C3)c3ncc(Nc4ccccc4)cn3)c2cc1OC |r|
COc1cc2ncnc(N3CCN(CC3)c3ncc(Nc4ccc(C)cc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Nc4ccccc4C)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Nc4cccc(C)c4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(NCc4ccccc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)c(O)n3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(COc4ccccc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(OCc4ccccc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccc(F)cc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4cccc(F)c4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Sc4ccccc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Br)c(OC)n3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Nc4ccc(F)cc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(OCc4cccs4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(OCc4ccsc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccc(cc4)C#N)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4cccc(c4)C#N)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Nc4ccc(cc4)C#N)cn3)c2cc1OC
COc1cc2ncnc(N3CC4CCC(C3)N4c3ncc(Cc4ccccc4)cn3)c2cc1OC |THB:8:9:12.13:16,17:16:10.9.15:12.13|
COc1cc2ncnc(N3CCN(CC3)c3ncc(cn3)N3CCc4ccccc34)c2cc1OC
C(C1CCNCC1)N1Cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2C1
COc1cc2ncnc(N3CCN(CC3)c3ncc(cn3)C(=O)Nc3ccccc3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(cn3)N(C)Cc3ccccc3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(NCc4ccc(C)cc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(NCc4ccccc4C)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(NCc4cccc(C)c4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(NC(C)c4ccccc4)cn3)c2cc1OC
COc1cccc(Cc2cnc(nc2)N2CCN(CC2)c2ncnc3cc(OC)c(OC)cc23)c1
COc1ccc(Cc2cnc(nc2)N2CCN(CC2)c2ncnc3cc(OC)c(OC)cc23)cc1
COc1cc2ncnc(N3CCN(CC3)c3ncc(O[C@H](C)c4ccccc4)cn3)c2cc1OC |r|
COc1cc2ncnc(N3CCN([C@H](C)C3)c3ncc(OCc4ccccc4)cn3)c2cc1OC |r|
COc1cc2ncnc(N3CCN(CC3)c3ncc(OCc4cccc(C)c4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(OCc4ccc(C)cc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(OC(C)c4ccccc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(O[C@@H](C)c4ccccc4)cn3)c2cc1OC |r|
COc1cc2ncnc(N3CCN(CC3)c3ncc(OCc4ccccc4C)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(C(C)C3)c3ncc(OCc4ccccc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(C[C@H]3C)c3ncc(OCc4ccccc4)cn3)c2cc1OC |r|
COc1cc2ncnc(N3CCN(CC3)c3ncc(OCc4ccc(F)cc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Nc4ccc(Cl)cc4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Nc4ccc(F)c(F)c4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(OCc4ccc(cc4)C#N)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(cn3)N3CCCc4ccccc34)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4cccc(c4)C(N)=O)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(NC(=O)Cc4ccccc4)cn3)c2cc1OC
COc1ccc(COc2cnc(nc2)N2CCN(CC2)c2ncnc3cc(OC)c(OC)cc23)cc1
COc1cc2ncnc(N3CCN(CC3)c3ncc(cn3)S(=O)(=O)c3ccccc3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCC1CNC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OC1CCNC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccc(cc4)C(C)(C)C)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Nc4ccc(cc4)C(C)(C)C)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCC(O)CO
COc1cc2c(ncnc2cc1OCC(O)CO)N1CCN(CC1)c1ncc(Cc2ccccc2)cn1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccc(OC(F)F)cc4)cn3)c2cc1OC
CN1CCC(COc2ccc3ncnc(N4CCN(CC4)c4ncc(Cc5ccccc5)cn4)c3c2)CC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccc(cc4)C(F)(F)F)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCC1CCNC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCC1CN(C)C1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OC1CCNCC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OC1CCN(C)C1
COc1cc2c(ncnc2cc1OCC1(C)COC1)N1CCN(CC1)c1ncc(Cc2ccccc2)cn1
COc1cc2ncnc(N3CCN(CC3)c3ncc(OCc4ccc(cc4)C(C)(C)C)cn3)c2cc1OC
CN1CCC(COc2ccc3ncnc(N4CCN(CC4)c4ncc(Cc5ccccc5)c(N)n4)c3c2)CC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCC1CCN(C)C1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCC1CCCNC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCC1CCNCC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OC1CCN(C)CC1
CN1CCC(COc2ccc3ncnc(N4CCN(CC4)c4ncc(Cc5ccccc5)c(=O)[nH]4)c3c2)CC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4cccc(OC(F)(F)F)c4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(OCc4ccc(cc4)C(F)(F)F)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(OCc4cc(Cl)cc(Cl)c4)cn3)c2cc1OC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OC[C@H]1CNCCO1 |r|
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCC1CNCCO1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OC[C@@H]1CNCCO1 |r|
COc1cc2c(ncnc2cc1OCCCN1CCCC1)N1CCN(CC1)c1ncc(Br)cn1
COCCOc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCCOC
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCC1CCNC(=O)C1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCCN1CCCC1=O
COc1cc2c(ncnc2cc1OCCN1CCCC1=O)N1CCN(CC1)c1ncc(Cc2ccccc2)cn1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCC1CCN(C)CC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OC[C@@H]1CCCN(C)C1 |r|
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCC1CCCN(C)C1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OC[C@H]1CCCN(C)C1 |r|
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCCN1CCNCC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCC1CN(C)CCO1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OC1CCN(CCO)C1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)c(=O)[nH]3)c2cc1OCC1CNCCO1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)c(=O)[nH]3)c2cc1OC[C@H]1CNCCO1 |r|
COc1cc2ncnc(N3CC4CCC(C3)N4c3ncc(Cc4ccccc4)cn3)c2cc1OCC1CNCCO1
CCOc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCC1CCN(C)CC1
COc1cc2c(ncnc2cc1OCCCN1CCCCC1)N1CCN(CC1)c1ncc(Cc2ccccc2)cn1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)c(N)n3)c2cc1OC[C@@H]1CCCN(C)C1 |r|
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)c(N)n3)c2cc1OCC1CCN(C)CC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCCN1CCN(C)CC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)c(=O)[nH]3)c2cc1OCC1CCN(C)CC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)c(=O)[nH]3)c2cc1OC[C@@H]1CCCN(C)C1 |r|
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OC1CCN(CCO)CC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)c(=O)[nH]3)c2cc1OCC1CN(C)CCO1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCC1(F)CCN(C)CC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Nc4ccc(F)cc4)cn3)c2cc1OCC1CCN(C)CC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Oc4ccc(F)cc4)cn3)c2cc1OCC1CCN(C)CC1
COc1cc2c(ncnc2cc1OCCCN1CCN(C)CC1)N1CCN(CC1)c1ncc(Cc2ccccc2)cn1
CCOc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)c(N)n3)c2cc1OCC1CCN(C)CC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCCCN1CCN(C)CC1
COc1cc2c(ncnc2cc1OCCCN1CCCCC1)N1CCN(CC1)c1ncc(Nc2ccc(C)cc2)cn1
CCOc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)c(=O)[nH]3)c2cc1OCC1CCN(C)CC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Cc4ccccc4)cn3)c2cc1OCC1CCN(CCO)CC1
COc1cc2ncnc(N3CCN(CC3)c3ncc(Sc4ccc(F)cc4)cn3)c2cc1OCC1CCN(C)CC1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ccccc1
COc1ccc(cc1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ccccc1
COc1cccc(c1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ccccc1
COc1cc(OC)cc(c1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ccccc1
COc1ccc(cc1OC)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ccccc1
CN(C)C(=O)c1ccc(cc1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ccccc1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(Cc2ccccc2)cn1
C[C@@H]1CN(CCN1c1ncc(Cc2ccccc2)cn1)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
C[C@H](c1ccccc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
C[C@@H](c1ccccc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ccc(cn1)C(O)c1ccccc1
C[C@](N)(c1ccccc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cn[nH]c1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@H](N)c1ccccc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(Cc2ccc(F)cc2)cn1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(Oc2ccc(F)cc2)cn1
N#Cc1ccc(cc1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(Cc2ccccc2)cn1
Fc1ccccc1Sc1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cn[nH]c1
COc1ccc(cc1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(Cc2ccccc2)cn1
C[C@@H]1CN(CCN1c1ncc(Cc2ccccc2)cn1)c1ncnn2cc(cc12)-c1cnn(C)c1C |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)C(C)(C)c1ccccc1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](C)(N)c1ccccc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(N)c1ccccc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)C(=C)c1ccc(F)cc1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](C)(O)c1ccccc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(O)c1ccccc1 |r|
C[C@](N)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cn[nH]c1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@H](N)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@H](N)c1ccc(F)cc1 |r|
C[C@@](O)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cn[nH]c1 |r|
C[C@](O)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cn[nH]c1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@H](O)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@H](O)c1ccc(F)cc1 |r|
NC(=O)c1ccc(cc1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(Cc2ccccc2)cn1
C[C@](N)(c1ccccc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1ccc(F)cc1 |r|
CCn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(N)c1ccccc1 |r|
CN(C)[C@@H](c1ccccc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
CN(C)[C@H](c1ccccc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
C[C@](O)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1ccccc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)C(C)(C)c1ccc(F)cc1
CC[C@H](c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
CC[C@@H](c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
Cn1cc(cn1)-c1cc2ncnc(N3CCN(CC3)c3ncc(cn3)C(C)(C)c3ccc(F)cc3)n2n1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](C)(N)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(N)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](C)(O)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(O)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(O)c1ccccc1F |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](C)(O)c1ccccc1F |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@H](CO)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@H](CO)c1ccc(F)cc1 |r|
Cc1cc(no1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](C)(O)c1ccc(F)cc1 |r|
Cc1cc(no1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(O)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](C)(O)c1ccc(F)cn1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(O)c1ccc(F)cn1 |r|
C[C@@H]1CN(CCN1c1ncc(Sc2ccccc2F)cn1)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(Sc2ccccc2F)c(N)n1
C[C@](O)(c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cn[nH]c1)c1ccc(F)cc1F |r|
C[C@@](O)(c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cn[nH]c1)c1ccc(F)cc1F |r|
Cc1ccc(cc1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(O)c1ccc(F)cc1 |r|
Cc1ccc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(O)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)C1(COC1)c1ccc(F)cc1
C[C@](N)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1ccc(F)cc1 |r|
CCn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(N)c1ccc(F)cc1 |r|
C[C@@](O)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1ccc(F)cc1 |r|
C[C@](O)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1ccc(F)cc1 |r|
C[C@](O)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cccc(F)c1 |r|
CO[C@@](C)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
CO[C@](C)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
CC[C@](O)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
CC[C@@](O)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
Cc1nn(C)cc1-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](C)(O)c1ccc(F)cc1 |r|
Cc1nn(C)cc1-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(O)c1ccc(F)cc1 |r|
C[C@@H](c1ccc(F)cc1)c1cnc(nc1)N1CCN(C[C@H]1CO)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
C[C@H](c1ccc(F)cc1)c1cnc(nc1)N1CCN(C[C@H]1CO)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
CCn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(O)c1ccc(F)cc1 |r|
C[C@@H]1CN(CCN1c1ncc(cn1)[C@](C)(O)c1ccc(F)cc1)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
C[C@@H]1CN(CCN1c1ncc(cn1)[C@@](C)(O)c1ccc(F)cc1)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(CO)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](C)(CO)c1ccc(F)cc1 |r|
Cc1cc(F)ccc1[C@](C)(O)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
Cc1ccc(s1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](C)(O)c1ccc(F)cc1 |r|
Cc1ccc(s1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(O)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(O)c1ccc(Cl)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](C)(O)c1ccc(Cl)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(N)c1ccc(F)cc1F |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](C)(N)c1ccc(F)cc1F |r|
Cc1ncc(s1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](C)(O)c1ccc(F)cc1 |r|
Cc1ncc(s1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(O)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cn2ncnc(N3CCN(CC3)c3ncc(cn3)[C@](C)(O)c3ccc(F)cc3)c2c1F |r|
Cn1cc(cn1)-c1cn2ncnc(N3CCN(CC3)c3ncc(cn3)[C@@](C)(O)c3ccc(F)cc3)c2c1F |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](C)(O)c1c(F)cccc1F |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(O)c1c(F)cccc1F |r|
C[C@@H]1CN(CCN1c1ncc(cn1)[C@](C)(O)c1ccc(F)cc1F)c1ncnn2cc(cc12)-c1cnn(C)c1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(O)c1ccc(F)cc1F |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](O)(CF)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](O)(CF)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN([C@H](CO)C1)c1ncc(Sc2ccccc2F)cn1 |r|
CN(C)C(=O)c1ccc(cc1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(Cc2ccccc2)cn1
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)S(=O)(=O)c1ccc(F)cc1
O[C@@](C(F)F)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cn[nH]c1 |r|
COc1cccc(c1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(O)c1ccc(F)cc1 |r|
COc1ccc(cc1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(O)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](O)(C1CC1)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](O)(C1CC1)c1ccc(F)cc1 |r|
C[C@H](O)Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(Sc2ccccc2F)cn1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)C(C)(C)c1c(F)cc(F)cc1F
Cn1cc(cn1)-c1cn2ncnc(N3CCN(CC3)c3ncc(cn3)[C@](C)(O)c3ccc(F)cc3)c2c1Cl |r|
Cn1cc(cn1)-c1cn2ncnc(N3CCN(CC3)c3ncc(cn3)[C@@](C)(O)c3ccc(F)cc3)c2c1Cl |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](C)(O)c1ccc(F)cc1Cl |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(O)c1ccc(F)cc1Cl |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](N)(C(F)F)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](N)(C(F)F)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](C)(N)c1c(F)cc(F)cc1F |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(N)c1c(F)cc(F)cc1F |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](C)(O)c1c(F)cc(F)cc1F |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(O)c1c(F)cc(F)cc1F |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@](O)(C(F)F)c1ccc(F)cc1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](O)(C(F)F)c1ccc(F)cc1 |r|
C[C@](O)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1ccc(cc1)C1CC1 |r|
C([C@@H]1CNCCO1)n1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(Cc2ccccc2)cn1 |r|
C[C@](O)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(c1)C1COC1 |r|
Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](N)(c1ccc(F)cc1)C(F)(F)F |r|
Fc1ccccc1Sc1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(C[C@@H]2CNCCO2)c1 |r|
CC(C)(C)OC(=O)N1CCC(=CC1)c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(O)c1ccc(F)cc1 |r,c:10|
CC(C)(O)Cn1cc(cn1)-c1cc2c(N)ncnn2c1
CC(C)(CO)n1cc(cn1)-c1cc2c(N)ncnn2c1
C[C@@H](O)Cn1cc(cn1)-c1cc2c(N)ncnn2c1 |r|
Nc1ncnn2cc(cc12)-c1cnn(CCO)c1
C[C@H](CO)n1cc(cn1)-c1cc2c(N)ncnn2c1 |r|
C[C@@H](CO)n1cc(cn1)-c1cc2c(N)ncnn2c1 |r|
Nc1ncnn2cc(cc12)-c1cnn(c1)C1COC1
C[C@](N)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(CC2COC2)c1 |r|
C[C@H](O)Cn1cc(cn1)-c1cc2c(ncnn2c1)N1CCN(CC1)c1ncc(cn1)[C@@](C)(N)c1ccc(F)cc1 |r|
C[C@](N)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(c1)C1C[C@H](O)C1 |r,wU:1.0,38.44,wD:1.1,(2.18,-6.48,;3.27,-5.39,;1.78,-4.99,;4.6,-6.16,;4.6,-7.7,;5.93,-8.47,;7.27,-7.7,;8.6,-8.47,;7.27,-6.16,;5.93,-5.39,;3.27,-3.85,;1.93,-3.08,;1.93,-1.54,;3.27,-.77,;4.6,-1.54,;4.6,-3.08,;3.27,.77,;1.93,1.54,;1.93,3.08,;3.27,3.85,;4.6,3.08,;4.6,1.54,;3.27,5.39,;4.6,6.16,;4.6,7.7,;3.27,8.47,;1.93,7.7,;.47,8.18,;-.44,6.93,;.47,5.68,;1.93,6.16,;-1.98,6.93,;-2.88,8.18,;-4.35,7.7,;-4.35,6.16,;-2.88,5.68,;-5.59,5.25,;-7.11,5.5,;-7.36,3.97,;-8.6,3.07,;-5.83,3.73,)|
C[C@](N)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(c1)C1C[C@H](O)C1 |r,wU:1.0,wD:1.1,38.44,(2.18,-6.48,;3.27,-5.39,;1.78,-4.99,;4.6,-6.16,;4.6,-7.7,;5.93,-8.47,;7.27,-7.7,;8.6,-8.47,;7.27,-6.16,;5.93,-5.39,;3.27,-3.85,;1.93,-3.08,;1.93,-1.54,;3.27,-.77,;4.6,-1.54,;4.6,-3.08,;3.27,.77,;1.93,1.54,;1.93,3.08,;3.27,3.85,;4.6,3.08,;4.6,1.54,;3.27,5.39,;4.6,6.16,;4.6,7.7,;3.27,8.47,;1.93,7.7,;.47,8.18,;-.44,6.93,;.47,5.68,;1.93,6.16,;-1.98,6.93,;-2.88,8.18,;-4.35,7.7,;-4.35,6.16,;-2.88,5.68,;-5.59,5.25,;-5.83,3.73,;-7.36,3.97,;-8.6,3.07,;-7.11,5.5,)|
C[C@](N)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(CC2(O)CC2)c1 |r|
C[C@](N)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(c1)C1(CO)CC1 |r|
C[C@](N)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(c1)[C@@H]1CCOC1 |r|
C[C@](N)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(c1)[C@H]1CCOC1 |r|
C[C@](N)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(c1)C1CCOCC1 |r|
C[C@](N)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(c1)[C@@H]1COC[C@@H]1O |r|
C[C@](N)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(c1)[C@H]1COC[C@@H]1O |r|
C[C@](N)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(c1)[C@@H]1COC[C@H]1O |r|
C[C@](N)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(c1)[C@H]1COC[C@H]1O |r|
C[C@](N)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(c1)[C@H]1CC[C@@H]1O |r|
C[C@](N)(c1ccc(F)cc1)c1cnc(nc1)N1CCN(CC1)c1ncnn2cc(cc12)-c1cnn(c1)[C@@H]1CC[C@H]1O |r|