10751 SMILES Strings for Nuclear receptor ROR-gamma

Compound Name
SMILES String
CC(=O)N1CCN(CC1)c1ccc(CN2CCCN(c3ccccc3)S2(=O)=O)c(F)c1
CN(c1ccccc1)S(=O)(=O)N(Cc1ccc(cc1F)N1CCN(CC1)C(C)=O)C1CCC1
CS(=O)(=O)N1CCC(CC1)Oc1ccc(cc1)N1CCN(Cc2ccc(F)cc2)S1(=O)=O
CC(C)CN(Cc1ccc(F)cc1)S(=O)(=O)Nc1ccc(OC2CCN(CC2)S(C)(=O)=O)cc1
CC(C)CN(Cc1ccc(F)cc1)S(=O)(=O)N(C)c1ccc(OC2CCN(CC2)S(C)(=O)=O)cc1
CC(C)CN(c1ccc(OC2CCN(CC2)S(C)(=O)=O)cc1)S(=O)(=O)N(C)Cc1ccc(F)cc1
CC1CCN(c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)C(C)=O
CC(=O)N1CCN(CC1)c1ccc(CN2CCCCN(c3ccccc3)S2(=O)=O)c(F)c1
CC1CCN(Cc2ccc(cc2F)N2CCN(CC2)C(C)=O)S(=O)(=O)N1c1ccccc1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)Oc2ccccc2)c(F)c1
CC(C)CN(Cc1ccc(cc1)N1CCCC1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCC(O)CC1)S(=O)(=O)Cc1ccccc1
COCCNc1ccc(CN(CC(C)C)S(=O)(=O)Cc2ccccc2)cc1
CC(C)CN(Cc1ccc(cc1)N1CCOCC1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCN(C)CC1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(NCCO)cc1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCNC(=O)C1)S(=O)(=O)Cc1ccccc1
CC(C)CN([C@@H](C)c1ccc(cc1)N1CCOCC1)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN([C@H](C)c1ccc(cc1)N1CCOCC1)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN([C@@H](C)c1ccc(cc1)N1CCC(O)CC1)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN([C@@H](C)c1ccc(cc1)N1CCN(C)CC1)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN([C@H](C)c1ccc(cc1)N1CCC(O)CC1)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN([C@H](C)c1ccc(cc1)N1CCN(C)CC1)S(=O)(=O)Cc1ccccc1 |r|
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2cc(Cl)ccc2Cl)c(F)c1
CC(c1ccccc1)S(=O)(=O)N(Cc1ccc(cc1F)N1CCN(CC1)C(C)=O)CC(F)(F)F
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2cccc(OC(F)(F)F)c2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2ccc(cc2)C(C)(C)C)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2cccc(Cl)c2)c(F)c1
CC(C)CN(Cc1ccc(cc1)N1CCC(CC1)C(=O)N(C)C)S(=O)(=O)Cc1ccccc1
COCC1CCN(CC1)c1ccc(CN(CC(C)C)S(=O)(=O)Cc2ccccc2)cc1
CC(C)CN(Cc1ccc(cc1)N1CCC(CO)CC1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCC(CC1)C(N)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCC(CC1)N(C)C)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCC(CC1)C#N)S(=O)(=O)Cc1ccccc1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2ccc(OC(F)(F)F)cc2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2cccc(c2)C(C)(C)C)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2cccc(Cl)c2Cl)c(F)c1
CC(C)c1ccc(cc1)S(=O)(=O)N(Cc1ccc(cc1F)N1CCN(CC1)C(C)=O)C1CCC1
COc1cccc(c1)S(=O)(=O)N(Cc1ccc(cc1F)N1CCN(CC1)C(C)=O)C1CCC1
CC(C)CN(Cc1ccc(cc1)N1CC[C@@H](C1)C(N)=O)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN(Cc1ccc(cc1)N1CCS(=O)(=O)CC1)S(=O)(=O)Cc1ccccc1
COC(=O)N1CCN(CC1)c1ccc(CN(CC(C)C)S(=O)(=O)Cc2ccccc2)cc1
CC(C)CN(Cc1ccc(cc1)N1CCC(CC1)NC(C)=O)S(=O)(=O)Cc1ccccc1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2ccccc2Cl)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2cccc(F)c2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2ccccc2C)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2ccccc2F)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2ccc(Cl)cc2Cl)c(F)c1
CC(C)CN(Cc1ccc(cc1)N1CC[C@@H](C1)N(C)C)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN(Cc1ccc(cc1)N1CCN(CC1)S(=O)(=O)N(C)C)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCN(CC1)C(=O)C1CC1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCN(CCO)CC1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCC(C1)N(C)C)S(=O)(=O)Cc1ccccc1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)CCc2ccccc2)c(F)c1
COc1ccc(cc1)S(=O)(=O)N(Cc1ccc(cc1F)N1CCN(CC1)C(C)=O)C1CCC1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2ccc(C)cc2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2ccccc2C(F)(F)F)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2c(F)cccc2F)c(F)c1
COCCN(Cc1ccc(cc1)N1CCN(CC1)C(C)=O)S(=O)(=O)Cc1ccccc1
CC(C)N(Cc1ccc(cc1)N1CCN(CC1)C(C)=O)S(=O)(=O)Cc1ccccc1
CCCN(Cc1ccc(cc1)N1CCN(CC1)C(C)=O)S(=O)(=O)Cc1ccccc1
CCN(Cc1ccc(cc1)N1CCN(CC1)C(C)=O)S(=O)(=O)Cc1ccccc1
CN(Cc1ccc(cc1)N1CCN(CC1)C(C)=O)S(=O)(=O)Cc1ccccc1
CC(=O)N1CCN(CC1)c1ccc(CN(CC(F)(F)F)S(=O)(=O)Cc2ccccc2)cc1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)Cc2ccccc2)cc1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CC2)S(=O)(=O)Cc2ccccc2)cc1
CC(=O)N1CCN(CC1)c1ccc(CN(C2COC2)S(=O)(=O)Cc2ccccc2)cc1
CC(=O)N1CCN(CC1)c1ccc2CN(CCOc2c1)S(=O)(=O)Cc1ccccc1
NC(=O)N1CCC(CC1)c1ccc(CN(CC(F)(F)F)S(=O)(=O)Cc2ccccc2)c(F)c1
CN(C)S(=O)(=O)N1CCC(CC1)c1ccc(CN(CC(F)(F)F)S(=O)(=O)Cc2ccccc2)c(F)c1
CS(=O)(=O)N1CCC(CC1)c1ccc(CN(CC(F)(F)F)S(=O)(=O)Cc2ccccc2)c(F)c1
CC(=O)N1CCC(CC1)c1ccc(CN(CC(F)(F)F)S(=O)(=O)Cc2ccccc2)c(F)c1
CS(=O)(=O)NC1CCN(CC1)c1ccc(CN(CC(F)(F)F)S(=O)(=O)Cc2ccccc2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2ccc(F)c(F)c2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2ccc(cc2)C#N)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2cccc(c2)C#N)c(F)c1
COc1ccc(c(OC)c1)S(=O)(=O)N(Cc1ccc(cc1F)N1CCN(CC1)C(C)=O)C1CCC1
NC(=O)C1CCN(CC1)c1ccc(CN(CC(F)(F)F)S(=O)(=O)Cc2ccccc2)c(F)c1
CC(C)CN(Cc1ccc(cc1C)N1CCN(CC1)C(C)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(N2CCN(CC2)C(C)=O)c(C)c1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1F)N1CCN(CC1)C(C)=O)S(=O)(=O)Cc1ccccc1
CC(=O)N1CCN(CC1)c1ccc(CN(CC(F)(F)F)S(=O)(=O)Cc2ccccc2)c(F)c1
CS(=O)(=O)N1CCN(CC1)c1ccc(CN(CC(F)(F)F)S(=O)(=O)Cc2ccccc2)c(F)c1
CN(C)S(=O)(=O)N1CCN(CC1)c1ccc(CN(CC(F)(F)F)S(=O)(=O)Cc2ccccc2)c(F)c1
CC(=O)N1C[C@@H]2C[C@H](C1)N2c1ccc(CN(CC(F)(F)F)S(=O)(=O)Cc2ccccc2)c(F)c1 |r,THB:10:9:3.4.8:6|
CC(=O)N1[C@H]2C[C@@H]1CN(C2)c1ccc(CN(CC(F)(F)F)S(=O)(=O)Cc2ccccc2)c(F)c1 |r,THB:1:3:8.9.7:5|
CC(=O)N1CCN(CC1)c1ccc(CN(C(C)(C)C)S(=O)(=O)Cc2ccccc2)cc1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)Cc2cc(Cl)cc(Cl)c2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)Cc2ccc(Cl)c(Cl)c2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)Cc2ccc(cc2)C(F)(F)F)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)Cc2ccc(Cl)cc2Cl)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)Cc2ccccc2C(F)(F)F)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)Cc2ccccc2Cl)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)Cc2ccc(Cl)cc2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)Cc2cc(F)ccc2F)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)Cc2ccc(F)cc2F)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)Cc2cccc(Cl)c2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)Cc2cccc(F)c2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)Cc2ccc(F)cc2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)Cc2ccccc2F)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2(C)COC2)S(=O)(=O)Cc2ccccc2)cc1
Fc1cc(ccc1CN(CC(F)(F)F)S(=O)(=O)Cc1ccccc1)N1CCS(=O)(=O)CC1
CC(=O)N1C[C@@H]2C[C@H]1CN2c1ccc(CN(CC(F)(F)F)S(=O)(=O)Cc2ccccc2)c(F)c1 |r|
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)Cc2ccccc2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2cc(Cl)cc(Cl)c2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2ccc(Cl)c(Cl)c2)c(F)c1
CC(C)CN(Cc1ccc(cc1)N1CCC(O)C1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCN(CC1)S(C)(=O)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N2CCN(CC2)C(=O)C)S(=O)(=O)Cc3ccccc3
COC1CCN(CC1)c1ccc(CN(CC(C)C)S(=O)(=O)Cc2ccccc2)cc1
CC(C)CN(Cc1ccc(cc1)N1CCCC(O)C1)S(=O)(=O)Cc1ccccc1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2cc(C)cc(C)c2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2cccc(C)c2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(CC(F)(F)F)S(=O)(=O)C(C)(C)c2ccccc2)c(F)c1
CC(C)CN(Cc1ccc(cc1)N1CCC(C1)S(C)(=O)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CC(O)C1)S(=O)(=O)Cc1ccccc1
CCOC(=O)N1CCN(CC1)c1ccc(CN(CC(C)C)S(=O)(=O)Cc2ccccc2)cc1
CC(C)CN(Cc1ccc(cc1)N1CC(C1)C(N)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CC(C1)C(=O)N(C)C)S(=O)(=O)Cc1ccccc1
CC(=O)N1C[C@H]2C[C@@H]1CN2c1ccc(CN(CC(F)(F)F)S(=O)(=O)Cc2ccccc2)c(F)c1 |r|
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2ccc(F)cc2F)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2c(Cl)cccc2Cl)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2cc(F)ccc2F)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2cc(F)cc(F)c2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1
CC(C)CN(Cc1ccc(cc1)N1CCCOCC1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCC(CC1)NS(C)(=O)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCC(CS(C)(=O)=O)CC1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCC(CC1)S(=O)(=O)N(C)C)S(=O)(=O)Cc1ccccc1
CC(=O)N1CCN(CC1)c1ccc(CN(CC#N)S(=O)(=O)Cc2ccccc2)cc1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2cccc(OC(F)F)c2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2ccc(Cl)cc2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2cccc(c2)C(F)(F)F)c(F)c1
CC(C)CN([C@@H](C)c1ccc(cc1)N1CCN(CC1)S(=O)(=O)N(C)C)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN([C@@H](C)c1ccc(cc1)N1CCC(CC1)C(N)=O)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN([C@H](C)c1ccc(cc1)N1CCN(CC1)C(C)=O)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN([C@H](C)c1ccc(cc1)N1CCN(CC1)S(=O)(=O)N(C)C)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN([C@H](C)c1ccc(cc1)N1CCC(CC1)C(N)=O)S(=O)(=O)Cc1ccccc1 |r|
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)CCc2ccc(F)cc2)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)CCc2cccc(F)c2)c(F)c1
COc1ccccc1S(=O)(=O)N(Cc1ccc(cc1F)N1CCN(CC1)C(C)=O)C1CCC1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2ccc(F)cc2)c(F)c1
CC(=O)N1CCN(CC1)c2ccc(c(c2)F)CN(C3CCC3)S(=O)(=O)c4ccccc4
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2ccccc2C#N)c(F)c1
CS(=O)(=O)N(Cc1ccc(cc1F)N1CCN(CC1)C(=O)C1CC1)S(=O)(=O)CCc1ccccc1
CC(C)CN(Cc1ccc(cn1)N1CCN(CC1)C(C)=O)S(=O)(=O)Cc1ccccc1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)Cc2ccccc2)cc1F
CC(C)CN(Cc1ccc(nc1)N1CCN(CC1)C(C)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1cnc(cn1)N1CCN(CC1)C(C)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1C#N)N1CCN(CC1)C(C)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(N2CCN(CC2)C(C)=O)c(c1)C#N)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ncc(cn1)N1CCN(CC1)C(C)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1cnc(nc1)N1CCN(CC1)C(C)=O)S(=O)(=O)Cc1ccccc1
CC(=O)N1CCN(CC1)c1ccc(CN(C2(C)CC2)S(=O)(=O)Cc2ccccc2)cc1
CC(=O)N1CCN(CC1)c1ccc(CN(C2(C)CCC2)S(=O)(=O)Cc2ccccc2)cc1
CC(C)CN(Cc1ccc(cc1)N1CCN(CC1=O)C(C)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(OC2CCN(CC2)C(C)=O)cc1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(NC2CCN(CC2)C(C)=O)cc1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCCS(=O)(=O)CC1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCCN(CC1)C(C)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CC2(C1)CCN(C2)C(C)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(NC2CCN(CC2)S(C)(=O)=O)cc1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCC2(CN(C2)C(C)=O)CC1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N(C)C1CCN(CC1)S(C)(=O)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(OC2CCN(CC2)S(C)(=O)=O)cc1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CC2(C1)CCN(CC2)C(C)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCC2(CCN(C2)C(C)=O)C1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCC2(CN(C2)C(C)=O)C1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CC2(CN(C2)C(C)=O)C1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCN(CC1)C(=O)CO)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCN(CC1)C(=O)CC#N)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCN(CC1)C(=O)[C@H](C)O)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN(Cc1ccc(cc1)N1CCN(CC1)C(=O)[C@@H](C)O)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN(Cc1ccc(cc1)N1CCN(CC1)C(=O)C1(O)CC1)S(=O)(=O)Cc1ccccc1
COCC(=O)N1CCN(CC1)c1ccc(CN(CC(C)C)S(=O)(=O)Cc2ccccc2)cc1
CO[C@@H](C)C(=O)N1CCN(CC1)c1ccc(CN(CC(C)C)S(=O)(=O)Cc2ccccc2)cc1 |r|
CO[C@H](C)C(=O)N1CCN(CC1)c1ccc(CN(CC(C)C)S(=O)(=O)Cc2ccccc2)cc1 |r|
CC(C)CN(Cc1ccc(cc1)N1CCN(CC1)C(=O)C1COC1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCN(CC1)C(=O)C1(C)COC1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(O[C@@H]2C[C@@H]3CC[C@H](C2)N3S(C)(=O)=O)cc1)S(=O)(=O)Cc1ccccc1 |r,TLB:19:18:11.12.17:15.14|
CC(C)CN(Cc1ccc(O[C@@H]2CCN(C2)S(C)(=O)=O)cc1)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN(Cc1ccc(O[C@H]2CCN(C2)S(C)(=O)=O)cc1)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN(Cc1ccc(NC2CCN(CC2)C(=O)N(C)C)cc1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCC(C1)C#N)S(=O)(=O)Cc1ccccc1
CNC(=O)C1CCN(CC1)c1ccc(CN(CC(C)C)S(=O)(=O)Cc2ccccc2)cc1
CC(C)CN(Cc1ccc(cc1)N1CC[C@@H](O)C1)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN(Cc1ccc(cc1)N1CC[C@H](O)C1)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN(Cc1ccc(cc1)N1CCC2(COC2)C1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCC2(COC2)CC1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCC2(CCOC2)C1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCC2(CCCO2)C1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CC2(C1)CCOC2)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CC2COC[C@@H]2C1)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN(Cc1ccc(cc1)N1CC2(C1)CCOCC2)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCC2(CCNC2=O)C1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCC2(CCNC2)C1=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCC(CC1)N1CCS(=O)(=O)CC1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCC(CC1)C(C)(C)O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCN(CC1)C1COC1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(N[C@H]2CC[C@H](CC2)C#N)cc1)S(=O)(=O)Cc1ccccc1 |r,wU:11.10,14.17,(4.67,-3.47,;4.67,-1.93,;6,-1.16,;3.33,-1.16,;3.33,.38,;2,1.15,;.67,.38,;-.67,1.15,;-2,.38,;-2,-1.16,;-3.33,-1.93,;-4.67,-1.16,;-6,-1.93,;-7.34,-1.16,;-7.34,.38,;-6,1.15,;-4.67,.38,;-8.67,1.15,;-10,1.92,;-.67,-1.93,;.67,-1.16,;4.67,1.15,;3.9,2.49,;5.44,2.49,;6,.38,;7.34,1.15,;8.67,.38,;10,1.15,;10,2.7,;8.67,3.47,;7.34,2.7,)|
CC(C)CN(Cc1ccc(NC2(C)CCN(CC2)S(C)(=O)=O)cc1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CC(C1)C1CCOCC1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(N[C@H]2CCC[C@H](O)C2)cc1)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN(Cc1ccc(N[C@@H]2CCN(C[C@@H]2F)S(C)(=O)=O)cc1)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN(Cc1ccc(N[C@@H]2CCN(C[C@H]2F)S(C)(=O)=O)cc1)S(=O)(=O)Cc1ccccc1 |r|
CC(C)CN(Cc1ccc(NC2CCCOC2)cc1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(NC2CCOCC2)cc1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(N[C@@H]2CC[C@H](O)CC2)cc1)S(=O)(=O)Cc1ccccc1 |r,wD:11.10,14.14,(4,-3.47,;4,-1.93,;5.33,-1.16,;2.67,-1.16,;2.67,.38,;1.33,1.15,;,.38,;-1.33,1.15,;-2.67,.38,;-2.67,-1.16,;-4,-1.93,;-5.33,-1.16,;-6.67,-1.93,;-8,-1.16,;-8,.38,;-9.34,1.15,;-6.67,1.16,;-5.33,.38,;-1.33,-1.93,;,-1.16,;4,1.15,;3.23,2.49,;4.77,2.49,;5.33,.38,;6.67,1.15,;8,.38,;9.34,1.15,;9.34,2.7,;8,3.47,;6.67,2.7,)|
CC(C)CN(Cc1ccc(N[C@H]2CC[C@H](O)CC2)cc1)S(=O)(=O)Cc1ccccc1 |r,wU:11.10,wD:14.14,(4,-3.47,;4,-1.93,;5.33,-1.16,;2.67,-1.16,;2.67,.38,;1.33,1.15,;,.38,;-1.33,1.15,;-2.67,.38,;-2.67,-1.16,;-4,-1.93,;-5.33,-1.16,;-6.67,-1.93,;-8,-1.16,;-8,.38,;-9.34,1.15,;-6.67,1.16,;-5.33,.38,;-1.33,-1.93,;,-1.16,;4,1.15,;3.23,2.49,;4.77,2.49,;5.33,.38,;6.67,1.15,;8,.38,;9.34,1.15,;9.34,2.7,;8,3.47,;6.67,2.7,)|
CC(C)CN(Cc1ccc(N[C@@H]2CC[C@H](CC#N)C2)cc1)S(=O)(=O)Cc1ccccc1 |r|
CCN1CC[C@H](Nc2ccc(CN(CC(C)C)S(=O)(=O)Cc3ccccc3)cc2)C(F)(F)C1 |r|
CCN1CC[C@@H](Nc2ccc(CN(CC(C)C)S(=O)(=O)Cc3ccccc3)cc2)[C@@H](F)C1 |r|
CCN1CC[C@H](Nc2ccc(CN(CC(C)C)S(=O)(=O)Cc3ccccc3)cc2)[C@H](F)C1 |r|
CC(C)CN(c1ccccc1C(F)(F)F)S(=O)(=O)c1ccc(cc1)-c1ccc(cc1)S(C)(=O)=O
CC(C)CN(c1ccccc1Cl)S(=O)(=O)c1ccc(cc1)-c1ccc(NS(C)(=O)=O)cc1
CC(C)CN(Cc1ccccc1Cl)S(=O)(=O)c1ccc(cc1)-c1ccc(cc1)S(C)(=O)=O
CC(C)CN(Cc1cccc(Cl)c1)S(=O)(=O)c1ccc(cc1)-c1ccc(cc1)S(C)(=O)=O
CC(C)CN(c1cccc(Cl)c1)S(=O)(=O)c1ccc(Oc2ccc(cc2)S(C)(=O)=O)cc1
CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(cc1)-c1ccc(NS(C)(=O)=O)cc1
CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(cc1)-c1ccc(cc1)C(N)=O
CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(cc1)-c1ccc(cc1)S(C)(=O)=O
CC(C)CN(c1ccccc1Cl)S(=O)(=O)c1cccc(c1)-c1ccc(cc1)S(C)(=O)=O
CC(C)CN(c1cccc(Cl)c1)S(=O)(=O)c1cccc(c1)-c1ccc(cc1)S(C)(=O)=O
CC(C)CN(c1ccc(Cl)cc1)S(=O)(=O)c1ccc(cc1)-c1ccc(cc1)S(C)(=O)=O
CC(C)CN(c1cccc(c1)C(F)(F)F)S(=O)(=O)c1ccc(cc1)-c1ccc(cc1)S(C)(=O)=O
CC(C)CN(c1ccccc1Cl)S(=O)(=O)c1ccc(cc1)-c1ccc(cc1)S(N)(=O)=O
CC(C)CN(c1cccc(Cl)c1)S(=O)(=O)c1ccc(cc1)-c1ccc(cc1)S(N)(=O)=O
CC(C)CN(c1cccc(Cl)c1)S(=O)(=O)c1ccc(cc1)-c1ccc(cc1)C(N)=O
CC(C)CN(c1ccccc1Cl)S(=O)(=O)c1ccc(cc1)-c1ccc(cc1)C(N)=O
CC(C)CN(c1cccc(Cl)c1)S(=O)(=O)c1ccc(cc1)-c1ccc(NS(C)(=O)=O)cc1
CC(=O)Nc1ccc2N(Cc3ccc(cc3)C(O)(C(F)(F)F)C(F)(F)F)CCCc2c1
CC(=O)Nc1ccc2N(Cc3ccc(cc3)C(O)(C(F)(F)F)C(F)(F)F)C(=O)CCc2c1
CC(=O)Nc1ccc2N(Cc3ccc(cc3)C(O)(C(F)(F)F)C(F)(F)F)CCc2c1
CS(=O)(=O)Nc1ccc2N(Cc3ccc(cc3)C(O)(C(F)(F)F)C(F)(F)F)CCCc2c1
CS(=O)(=O)Nc1ccc2N(Cc3ccc(cc3)C(O)(C(F)(F)F)C(F)(F)F)C(=O)CCc2c1
COc1cc(cc(c1)C(=O)Nc1cnc2n(C)cc(C3CCN(CC3)C(=O)C3CCCC3)c2c1C(F)(F)F)C#N
Cc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc(C3CCN(CC3)C(=O)C3CCCC3)c2c1C(F)(F)F
Cn1cc(C2CCN(CC2)C(=O)C2CCCC2)c2c(c(NC(=O)c3ccc(F)c(c3)C#N)cnc12)C(F)(F)F
COc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc(C3CCN(CC3)C(=O)C3CCCC3)c2c1C(F)(F)F
CC(C)C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(c12)C(F)(F)F
COc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc(C3CCN(CC3)C(=O)C(C)C)c2c1C(F)(F)F
CC(C)C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3ccc(C)c(c3)C#N)c(c12)C(F)(F)F
COc1cc(cc(c1)C(=O)Nc1cnc2n(C)cc(C3CCN(CC3)C(=O)C(C)C)c2c1C(F)(F)F)C#N
CC(C)C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3ccc(F)c(c3)C#N)c(c12)C(F)(F)F
COc1ccc(cc1Cl)C(=O)Nc1cnc2n(C)cc(C3CCN(CC3)C(=O)C(C)C)c2c1C(F)(F)F
CC(C)C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3ccc(Cl)c(c3)C#N)c(c12)C(F)(F)F
CC(C)C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3ccc(F)c(Cl)c3)c(c12)C(F)(F)F
COc1cc(Cl)cc(c1)C(=O)Nc1cnc2n(C)cc(C3CCN(CC3)C(=O)C(C)C)c2c1C(F)(F)F
Cn1cc(C2CCN(CC2)C(=O)CC2CCCC2)c2c(c(NC(=O)c3cccc(c3)C#N)cnc12)C(F)(F)F
CC(C)CC(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(c12)C(F)(F)F
Cn1cc(C2CCN(CC2)C(=O)[C@H]2C[C@H]3CCCC[C@H]3C2)c2c(c(NC(=O)c3cccc(c3)C#N)cnc12)C(F)(F)F |r|
CC(C)C(C)(C)CC(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(c12)C(F)(F)F
Cn1cc(C2CCN(CC2)C(=O)CC2CCC2)c2c(c(NC(=O)c3cccc(c3)C#N)cnc12)C(F)(F)F
Cn1cc(C2CCN(CC2)C(=O)C2CCCCC2)c2c(c(NC(=O)c3cccc(c3)C#N)cnc12)C(F)(F)F
Cn1cc(C2CCN(CC2)C(=O)CC2CCCCC2)c2c(c(NC(=O)c3cccc(c3)C#N)cnc12)C(F)(F)F
C[C@@H](C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(c12)C(F)(F)F)C(C)(C)C |r|
C[C@H](C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(c12)C(F)(F)F)C(C)(C)C |r|
Cn1cc(C2CCN(CC2)C(=O)C2CCCC2)c2c(c(NC(=O)c3cccc(c3)C#N)cnc12)C(F)(F)F
Cn1cc(C2CCN(CC2)C(=O)CC2CC2)c2c(c(NC(=O)c3cccc(c3)C#N)cnc12)C(F)(F)F
CC(C1CC1)C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(c12)C(F)(F)F |w:1.0|
C[C@@H]1CCC[C@H]1C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(c12)C(F)(F)F |r|
C[C@@H]1CCC[C@@H]1C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(c12)C(F)(F)F |r|
Cn1cc(C2CCN(CC2)C(=O)[C@H]2CCCS2)c2c(c(NC(=O)c3cccc(c3)C#N)cnc12)C(F)(F)F |r|
Cn1cc(C2CCN(CC2)C(=O)[C@@H]2CCCS2)c2c(c(NC(=O)c3cccc(c3)C#N)cnc12)C(F)(F)F |r|
COc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc(C3CCN(CC3)C(=O)[C@H](C)C(C)(C)C)c2c1C(F)(F)F |r|
COc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc(C3CCN(CC3)C(=O)[C@@H](C)C(C)(C)C)c2c1C(F)(F)F |r|
C[C@@H](C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12)C(C)(C)C |r|
Cc1cccc(F)c1C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12
Cc1c(NC(=O)c2cccc(c2)C#N)cnc2n(C)cc(C3CCN(CC3)C(=O)c3cccc4CCCc34)c12
Cc1c(NC(=O)c2cccc(c2)C#N)cnc2n(C)cc(C3CCN(CC3)C(=O)C3C[C@H]4CCC3C4)c12 |r|
Cc1c(NC(=O)c2cccc(c2)C#N)cnc2n(C)cc(C3CCN(CC3)C(=O)C3C[C@@H]4CCC3C4)c12 |r|
CC(C)[C@@H](C)C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12 |r|
COc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc(C3CCN(CC3)C(=O)[C@H](C)C(C)(C)C)c2c1C |r|
COc1cc(cc(c1)C(=O)Nc1cnc2n(C)cc(C3CCN(CC3)C(=O)[C@H](C)C(C)(C)C)c2c1C)C#N |r|
COc1ccc(cc1C(=O)Nc1cnc2n(C)cc(C3CCN(CC3)C(=O)[C@H](C)C(C)(C)C)c2c1C)C#N |r|
C[C@@H](C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cc(Cl)ccc3F)c(C)c12)C(C)(C)C |r|
COc1cc(Cl)cc(c1)C(=O)Nc1cnc2n(C)cc(C3CCN(CC3)C(=O)[C@H](C)C(C)(C)C)c2c1C |r|
COCCOc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc(C3CCN(CC3)C(=O)[C@H](C)C(C)(C)C)c2c1C |r|
COc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc(C3CCN(CC3)C(=O)[C@@H](C)C(F)(F)F)c2c1C |r|
COc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc(C3CCN(CC3)C(=O)[C@H](C)C(F)(F)F)c2c1C |r|
C[C@H]1CCC[C@@H]1C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12 |r|
C[C@@H]1CCC[C@H]1C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12 |r|
CC(C)[C@@H]1CCC[C@H]1C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12 |r|
C[C@@H](C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12)C12CC(C1)C2 |r|
C[C@H](C1CCCC1)C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12 |r|
COc1cc(cc(c1)C(=O)Nc1cnc2n(C)cc(C3CCN(CC3)C(=O)C3CCCC3)c2c1C)C#N
Cc1c(NC(=O)c2cc(O)cc(c2)C#N)cnc2n(C)cc(C3CCN(CC3)C(=O)C3CCCC3)c12
C[C@@H](C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cc(O)cc(c3)C#N)c(c12)C(F)(F)F)C(C)(C)C |r|
Cn1cc(C2CCN(CC2)C(=O)C2CCCC2)c2c(c(NC(=O)c3cc(O)cc(c3)C#N)cnc12)C(F)(F)F
C[C@@H](C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cc(O)cc(c3)C#N)c(C)c12)C(C)(C)C |r|
COCCOc1cc(cc(c1)C(=O)Nc1cnc2n(C)cc(C3CCN(CC3)C(=O)C3CCCC3)c2c1C)C#N
COc1cc(cc(c1)C(=O)Nc1cnc2n(C)cc([C@@H]3CCN(C(=O)C4CCCC4)C(C)(C)C3)c2c1C)C#N |r|
Cc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc([C@@H]3CCN(C(=O)C4CCCC4)C(C)(C)C3)c2c1C |r|
COc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc([C@@H]3CCN(C(=O)C4CCCC4)C(C)(C)C3)c2c1C |r|
Cc1c(NC(=O)c2ccc(F)c(c2)C#N)cnc2n(C)cc([C@@H]3CCN(C(=O)C4CCCC4)C(C)(C)C3)c12 |r|
COc1cc(Cl)cc(c1)C(=O)Nc1cnc2n(C)cc([C@@H]3CCN(C(=O)C(C)C)C(C)(C)C3)c2c1C |r|
COc1cc(Cl)cc(c1)C(=O)Nc1cnc2n(C)cc([C@@H]3CCN(C(=O)C4CCCC4)C(C)(C)C3)c2c1C |r|
Cc1c(NC(=O)c2cc(O)cc(c2)C#N)cnc2n(C)cc([C@@H]3CCN(C(=O)C4CCCC4)C(C)(C)C3)c12 |r|
Cn1cc([C@@H]2CCN(C(=O)C3CCCC3)C(C)(C)C2)c2c(c(NC(=O)c3cccc(c3)C#N)cnc12)C(F)(F)F |r|
CC(C)C(=O)N1CC[C@H](CC1(C)C)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(c12)C(F)(F)F |r|
COc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc([C@@H]3CCN(C(=O)C(C)C)C(C)(C)C3)c2c1C(F)(F)F |r|
C[C@@H](C(=O)N1CC[C@H](CC1(C)C)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12)C(C)(C)C |r|
COc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc([C@@H]3CCN(C(=O)[C@H](C)C(C)(C)C)C(C)(C)C3)c2c1C |r|
COc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc([C@@H]3CCN(C(=O)C(C)C)C(C)(C)C3)c2c1C |r|
Cc1c(NC(=O)c2cccc(c2)C#N)cnc2n(C)cc([C@@H]3CCN(C(=O)C4CCCC4)C(C)(C)C3)c12 |r|
CC(C)C(=O)N1CC[C@H](CC1(C)C)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12 |r|
Cc1c(NC(=O)c2cccc(c2)C#N)cnc2n(C)cc([C@@H]3CCN(C(=O)C[C@@H](O)C(F)(F)F)C(C)(C)C3)c12 |r|
Cc1c(NC(=O)c2cccc(c2)C#N)cnc2n(C)cc([C@@H]3CCN(C(=O)CC4CCCC4)C(C)(C)C3)c12 |r|
Cc1c(NC(=O)c2cccc(c2)C#N)cnc2n(C)cc([C@@H]3CCN(C(=O)CC4CCCCC4)C(C)(C)C3)c12 |r|
Cc1c(NC(=O)c2cccc(c2)C#N)cnc2n(C)cc([C@@H]3CCN(C(=O)CC4CCC4)C(C)(C)C3)c12 |r|
CC(C)C(=O)N1C[C@@H]2CC[C@H](C1)[C@H]2c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(c12)C(F)(F)F |r|
COc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc(C3C4CC[C@H]3CN(C4)C(=O)C(C)C)c2c1C(F)(F)F |r|
Cn1cc(C2[C@H]3CC[C@@H]2CN(C3)C(=O)C2CCCC2)c2c(c(NC(=O)c3cccc(c3)C#N)cnc12)C(F)(F)F |r|
CC(C)C(=O)N1CC[C@H]([C@@H](C)C1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(c12)C(F)(F)F |r|
C[C@H]1CN(CC[C@H]1c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(c12)C(F)(F)F)C(=O)C1CCCC1 |r|
CC(C)C(=O)N1CC[C@H]([C@@H](C)C1)c1cn(C)c2ncc(NC(=O)c3cccc(C#N)c3F)c(c12)C(F)(F)F |r|
C[C@H]1CN(CC[C@H]1c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12)C(=O)CC1CC1 |r|
C[C@H]1CN(CC[C@H]1c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12)C(=O)C1CCCC1 |r|
CC(C)C(=O)N1CC[C@H]([C@@H](C)C1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12 |r|
CC(C1CC1)C(=O)N1CC[C@H]([C@@H](C)C1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12 |r,w:1.0|
COCCOc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc([C@@H]3CCN(C[C@@H]3C)C(=O)C3CCCC3)c2c1C |r|
C[C@H](C(=O)N1CC[C@H]([C@@H](C)C1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12)C(F)(F)F |r|
C[C@@H](C(=O)N1CCC([C@@H](C)C1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12)C(F)(F)F |r|
COc1cc(cc(c1)C(=O)Nc1cnc2n(C)cc([C@@H]3CCN([C@@H](C)C3)C(=O)C3CCCC3)c2c1C)C#N |r|
C[C@@H](C(=O)N1CC[C@H](C[C@@H]1C)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12)C(F)(F)F |r|
C[C@H](C(=O)N1CC[C@H](C[C@@H]1C)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12)C(F)(F)F |r|
COc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc([C@@H]3CCN([C@@H](C)C3)C(=O)[C@H](C)C(F)(F)F)c2c1C |r|
COc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc([C@@H]3CCN([C@@H](C)C3)C(=O)[C@@H](C)C(F)(F)F)c2c1C |r|
CC(C)C(=O)N1CC[C@H](C[C@@H]1C)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(c12)C(F)(F)F |r|
CC(C)C(=O)N1CCC(CC11CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12
C[C@@H]1CN([C@@H](C)CC1c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12)C(=O)C1CCCC1 |r|
CC(C)C(=O)N1CC2CC[C@@H](C1)C2c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12 |r|
COc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc(C3C4CC[C@H]3CN(C4)C(=O)C3CCCC3)c2c1C |r|
Cc1c(NC(=O)c2cccc(c2)C#N)cnc2n(C)cc([C@@H]3C[C@H]4CC[C@@H]3CN4C(=O)C3CCCC3)c12 |r,THB:29:28:21.22:25.24|
CC(C)CC(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12
COc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc(C3CCN(CC3)C(=O)C(C)C)c2c1C
C[C@H](C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12)C(F)(F)F |r|
COc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc([C@@H]3CCN(C[C@@H]3C)C(=O)C(C)C)c2c1C |r|
CC(C)C(=O)N1CC[C@H](C[C@@H]1C)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12 |r|
COC(=O)c1ccc(-c2nn(Cc3c(Cl)cccc3C(F)(F)F)c3cnccc23)c(F)c1
OC(=O)c1ccc(-c2nn(Cc3c(F)cccc3Br)c3cccnc23)c(F)c1
OC(=O)c1ccc(-c2nn(Cc3c(Cl)cccc3C(F)(F)F)c3cccc(F)c23)c(F)c1
OC(=O)c1ccc(cc1)-c1nn(Cc2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
OC(=O)c1c(F)cc(cc1F)-c1nn(Cc2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
CC(c1c(Cl)cccc1C(F)(F)F)n1nc(-c2ccc(cc2F)C(O)=O)c2c(F)cccc12
C[C@H](c1c(Cl)cccc1C(F)(F)F)n1nc(-c2ccc(cc2F)C(O)=O)c2c(F)cccc12 |r|
C[C@@H](c1c(Cl)cccc1C(F)(F)F)n1nc(-c2ccc(cc2F)C(O)=O)c2c(F)cccc12 |r|
OC(=O)c1ccc(-c2nn(Cc3cccc(F)c3Br)c3cccnc23)c(F)c1
OC(=O)c1ccc(-c2nn(Cc3cc(Cl)ccc3C#N)c3cccnc23)c(F)c1
CC(c1ccccc1C(F)(F)F)n1nc(-c2ccc(cc2F)C(O)=O)c2ncccc12
Cc1ccc(Cl)c(Cn2nc(-c3ccc(cc3F)C(O)=O)c3ncccc23)c1F
OC(=O)c1ccc(-c2nn(Cc3c(Cl)ccc(F)c3F)c3cccnc23)c(F)c1
OC(=O)c1ccc(-c2nn(Cc3c(F)ccc(F)c3F)c3cccnc23)c(F)c1
OC(=O)c1ccc(-c2nn(Cc3c(F)cccc3C(F)(F)F)c3cccnc23)c(F)c1
OC(=O)c1ccc(-c2nn(Cc3c(F)cccc3F)c3cccnc23)c(F)c1
OC(=O)c1ccc(-c2nn(Cc3c(F)cccc3Cl)c3cccnc23)c(F)c1
COc1ccc(Cl)c(Cn2nc(-c3ccc(cc3F)C(O)=O)c3ncccc23)c1F
COc1ccc(F)c(Cn2nc(-c3ccc(cc3F)C(O)=O)c3ncccc23)c1Cl
OC(=O)c1ccc(-c2nn(Cc3c(F)ccc(Cl)c3Cl)c3cccnc23)c(F)c1
OC(=O)c1ccc(-c2nn(Cc3cccc4ccsc34)c3cccnc23)c(F)c1
OC(=O)c1ccc(-c2nn(Cc3c(Cl)ccc(c3Cl)C(F)(F)F)c3cccnc23)c(F)c1
OC(=O)c1ccc(-c2nn(Cc3c(Cl)ccc(Cl)c3F)c3cccnc23)c(F)c1
COC(=O)c1cccc(Cl)c1Cn1nc(-c2ccc(cc2F)C(O)=O)c2ncccc12
OC(=O)c1ccc(-c2nn(Cc3c(Cl)cccc3Br)c3cccnc23)c(F)c1
OC(=O)c1ccc(-c2nn(Cc3c(Cl)cccc3C(F)(F)F)c3cccnc23)c(F)c1
OC(=O)c1ccc(cc1O)-c1nn(Cc2c(Cl)cccc2C(F)(F)F)c2ccccc12
OC(=O)c1ccc(-c2cn(Cc3c(Cl)cccc3C(F)(F)F)c3cccnc23)c(F)c1
OC(=O)c1ccc(-c2cn(Cc3c(Cl)cccc3C(F)(F)F)c3cnccc23)c(F)c1
OC(=O)c1ccc(-c2nn(Cc3cc(F)ccc3F)c3cccc(F)c23)c(F)c1
OC(=O)c1ccc(-c2nn(Cc3cccc(OC(F)(F)F)c3)c3cccc(F)c23)c(F)c1
COc1ccccc1Cn1nc(-c2ccc(cc2F)C(O)=O)c2c(F)cccc12
OC(=O)c1ccc(-c2nn(Cc3ccccc3-n3cccn3)c3cccc(F)c23)c(F)c1
OC(=O)c1ccc(-c2nn(Cc3ccccc3C#N)c3cccc(F)c23)c(F)c1
OC(=O)c1ccc(-c2nn(Cc3cc(OC(F)(F)F)ccc3F)c3cccc(F)c23)c(F)c1
OC(=O)c1ccc(cc1)-c1nn(Cc2c(Cl)cccc2Cl)c2cccc(F)c12
OC(=O)c1ccc(-c2nn(Cc3c(Cl)cccc3Cl)c3cccnc23)c(F)c1
OC(=O)c1cc(F)c(cc1O)-c1nn(Cc2c(Br)cccc2C(F)(F)F)c2cccc(F)c12
OC(=O)c1cc(F)c(cc1O)-c1nn(Cc2c(F)cccc2Cl)c2cccc(F)c12
OC(=O)c1cc(F)c(cc1O)-c1nn(Cc2ccccc2)c2cccc(F)c12
OC(=O)c1cc(F)c(cc1O)-c1nn(Cc2cc(F)ccc2Cl)c2cccc(F)c12
OC(=O)c1cc(F)c(cc1O)-c1nn(Cc2ccc(F)cc2Cl)c2cccc(F)c12
OC(=O)c1cc(F)c(cc1O)-c1nn(Cc2cc(F)ccc2Br)c2cccc(F)c12
OC(=O)c1cc(F)c(cc1O)-c1nn(Cc2cc(F)cc(Cl)c2)c2cccc(F)c12
OC(=O)c1cc(F)c(cc1O)-c1nn(Cc2cc(Cl)cc(Cl)c2)c2cccc(F)c12
OC(=O)c1cc(F)c(cc1O)-c1nn(Cc2ccc(Br)cc2F)c2cccc(F)c12
OC(=O)c1cc(F)c(cc1O)-c1nn(Cc2cc(Cl)ccc2Cl)c2cccc(F)c12
OC(=O)c1cc(F)c(cc1O)-c1nn(Cc2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
OC(=O)c1cc(F)c(cc1O)-c1nn(Cc2cc(F)cc(c2)C(F)(F)F)c2cccc(F)c12
OC(=O)c1cc(F)c(cc1O)-c1nn(Cc2c(F)cccc2C(F)(F)F)c2cccc(F)c12
OC(=O)c1cc(F)c(cc1O)-c1nn(Cc2c(Cl)cccc2C2CC2)c2cccc(F)c12
Cc1cccc(Cl)c1Cn1nc(-c2cc(O)c(cc2F)C(O)=O)c2c(F)cccc12
OC(=O)c1ccc(-c2nn(Cc3c(Cl)cccc3C3(O)CCC3)c3cccc(F)c23)c(F)c1
COC(=O)c1cc(F)c(cc1O)-c1nn(Cc2c(C)cccc2C(F)(F)F)c2cccc(F)c12
OC(=O)c1cc(F)c(cc1O)-c1nn(Cc2ccccc2C(F)(F)F)c2cccc(F)c12
CCc1cccc(c1Cn1nc(-c2cc(O)c(cc2F)C(O)=O)c2c(F)cccc12)C(F)(F)F
CC(C)c1cccc(c1Cn1nc(-c2cc(O)c(cc2F)C(O)=O)c2c(F)cccc12)C(F)(F)F
COC1CN(C1)C(=O)c1cc(F)c2c(nn(Cc3c(Cl)cccc3C(F)(F)F)c2c1)-c1cc(O)c(cc1F)C([O-])=O
OC(=O)c1cc(F)c(cc1O)-c1nn(Cc2c(Cl)cccc2C(F)(F)F)c2cc(cc(F)c12)C(=O)N1CCC1
OC(=O)c1ccc(-c2nn(Cc3c(Cl)cccc3C(F)(F)F)c3cc(cc(F)c23)C(=O)N2CCC2)c(F)c1
[#8]\[#7]=[#6]-1/[#6]-[#6]C([#6]-[#6]-1)(c1ccc(cc1)C([#8]-[#6]-c1ccccc1)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
COC(=O)C1CC(CCC1=O)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CC(C)(C)OC(=O)C1CC(CCC1=O)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
O[C@H]1CC[C@@](CC1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:4.7,wD:1.0,(-1.52,12.33,;-2.38,11.05,;-3.92,11.16,;-4.78,9.88,;-4.1,8.5,;-2.57,8.39,;-1.71,9.67,;-2.77,7.73,;-2.77,6.19,;-1.44,5.42,;-.1,6.19,;-.1,7.73,;-1.44,8.5,;1.23,5.42,;2.56,4.65,;3.9,5.42,;5.23,4.65,;6.57,5.42,;6.57,6.96,;7.9,4.65,;7.9,3.11,;6.57,2.34,;5.23,3.11,;3.9,2.34,;2,6.75,;2.77,8.08,;.67,7.52,;3.33,5.98,;.46,4.08,;-.31,2.75,;-.87,4.85,;1.79,3.31,;-5.58,8.07,;-7.06,7.65,;-6.01,9.55,;-5.16,6.59,;-3.67,6.22,;-3.24,4.74,;-4.31,3.63,;-3.89,2.15,;-5.81,4,;-6.23,5.48,)|
O[C@H]1CC[C@](CC1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:4.7,1.0,(-1.52,12.33,;-2.38,11.05,;-1.71,9.67,;-2.57,8.39,;-4.1,8.5,;-4.78,9.88,;-3.92,11.16,;-2.77,7.73,;-2.77,6.19,;-1.44,5.42,;-.1,6.19,;-.1,7.73,;-1.44,8.5,;1.23,5.42,;2.56,4.65,;3.9,5.42,;5.23,4.65,;6.57,5.42,;6.57,6.96,;7.9,4.65,;7.9,3.11,;6.57,2.34,;5.23,3.11,;3.9,2.34,;2,6.75,;2.77,8.08,;.67,7.52,;3.33,5.98,;.46,4.08,;-.31,2.75,;-.87,4.85,;1.79,3.31,;-5.58,8.07,;-7.06,7.65,;-6.01,9.55,;-5.16,6.59,;-3.67,6.22,;-3.24,4.74,;-4.31,3.63,;-3.89,2.15,;-5.81,4,;-6.23,5.48,)|
OC1CCC(CC1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |(-1.52,5.82,;-2.38,4.55,;-1.71,3.16,;-2.57,1.89,;-4.1,1.99,;-4.78,3.38,;-3.92,4.65,;-2.77,1.22,;-2.77,-.32,;-1.44,-1.09,;-.1,-.32,;-.1,1.22,;-1.44,1.99,;1.23,-1.09,;2.56,-1.86,;3.9,-1.09,;5.23,-1.86,;6.57,-1.09,;6.57,.45,;7.9,-1.86,;7.9,-3.4,;6.57,-4.17,;5.23,-3.4,;3.9,-4.17,;2,.25,;2.77,1.58,;.67,1.02,;3.33,-.52,;.46,-2.42,;-.31,-3.75,;-.87,-1.65,;1.79,-3.19,;-5.58,1.57,;-7.06,1.14,;-6.01,3.05,;-5.16,.09,;-3.67,-.28,;-3.24,-1.76,;-4.31,-2.87,;-3.89,-4.35,;-5.81,-2.5,;-6.23,-1.02,)|
[#8]\[#7]=[#6]-1\[#6]-[#6]C([#6]-[#6]-1)(c1ccc(cc1)C([#8]-[#6]-c1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
Fc1ccc(cc1)S(=O)(=O)[C@@]1(CC[C@@H](CC1)N1CCOCC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r,wU:10.24,wD:10.10,13.17,(-1.35,-8.2,;-.83,-6.75,;.69,-6.48,;1.22,-5.03,;.23,-3.85,;-1.29,-4.12,;-1.82,-5.57,;.75,-2.41,;1.28,-.96,;2.2,-2.93,;-.69,-1.88,;-.96,-3.4,;-2.41,-3.92,;-3.59,-2.93,;-3.32,-1.42,;-1.87,-.89,;-5.04,-3.46,;-5.3,-4.98,;-6.75,-5.5,;-7.93,-4.51,;-7.66,-3,;-6.22,-2.47,;.08,-.55,;1.62,-.55,;2.39,.79,;1.62,2.12,;.08,2.12,;-.69,.79,;2.39,3.45,;3.72,2.68,;3.72,1.14,;5.05,.37,;6.39,1.14,;6.39,2.68,;7.72,.37,;7.72,-1.17,;6.39,-1.94,;5.05,-1.17,;3.72,-1.94,;3.16,4.79,;3.93,6.12,;1.82,5.56,;4.49,4.02,;1.05,4.22,;-.28,4.99,;.89,5.76,;.28,2.89,)|
NC1CCC(CC1)(c1ccc(cc1)C(OCc1ccccc1)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |(4.85,3.7,;3.31,3.81,;2.45,2.53,;.92,2.64,;.24,4.02,;1.1,5.3,;2.64,5.19,;.24,2.48,;-1.09,1.71,;-1.09,.17,;.24,-.6,;1.58,.17,;1.58,1.71,;.24,-2.14,;.24,-3.68,;1.58,-4.45,;1.58,-5.99,;.24,-6.76,;.24,-8.3,;1.58,-9.07,;2.91,-8.3,;2.91,-6.76,;1.78,-2.14,;3.32,-2.14,;1.78,-.6,;1.78,-3.68,;-1.3,-2.14,;-2.84,-2.14,;-1.3,-.6,;-1.3,-3.68,;-.87,5.09,;-1.97,6.16,;.2,6.2,;-1.94,3.98,;-1.51,2.5,;-2.58,1.39,;-4.07,1.77,;-5.14,.66,;-4.5,3.25,;-3.43,4.36,)|
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CC(=O)N1CCC(CC1)C(=O)N[C@H]1CC[C@@](CC1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:15.19,wD:12.12,(-11.14,-2.7,;-10.46,-4.08,;-11.32,-5.36,;-8.93,-4.19,;-8.25,-5.57,;-6.71,-5.68,;-5.85,-4.41,;-6.53,-3.02,;-8.06,-2.91,;-4.32,-4.51,;-3.64,-5.9,;-3.46,-3.24,;-1.92,-3.34,;-1.24,-4.73,;.29,-4.83,;1.15,-3.56,;.48,-2.17,;-1.06,-2.07,;1.15,-2.02,;2.49,-1.25,;2.49,.29,;1.15,1.06,;-.18,.29,;-.18,-1.25,;1.15,2.6,;-.39,2.6,;1.15,4.14,;1.15,5.68,;2.69,4.14,;-.39,4.14,;2.69,2.6,;4.23,2.6,;2.69,1.06,;3.6,3.85,;2.26,-4.63,;1.19,-5.74,;3.37,-5.7,;3.33,-3.52,;2.91,-2.04,;3.98,-.93,;5.47,-1.3,;6.54,-.2,;5.89,-2.78,;4.82,-3.89,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(CC[C@@H](CC1)NC(=O)C1CCN(CC1)C(=O)CC#N)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:10.32,wD:13.17,(6.8,.07,;5.73,-1.04,;4.24,-.66,;3.17,-1.77,;3.59,-3.25,;5.09,-3.63,;6.16,-2.52,;2.52,-4.36,;1.45,-5.47,;3.63,-5.43,;1.42,-3.29,;.55,-4.57,;-.98,-4.46,;-1.66,-3.08,;-.8,-1.8,;.74,-1.91,;-3.19,-2.97,;-4.05,-4.25,;-3.38,-5.63,;-5.59,-4.14,;-6.45,-5.41,;-7.99,-5.31,;-8.66,-3.92,;-7.8,-2.65,;-6.27,-2.75,;-10.2,-3.82,;-10.87,-2.43,;-11.06,-5.09,;-12.6,-4.99,;-14.13,-4.88,;1.42,-1.75,;2.75,-.98,;2.75,.56,;1.42,1.33,;.08,.56,;.08,-.98,;1.42,2.87,;2.96,2.87,;-.12,2.87,;-1.66,2.87,;-.12,4.41,;-.12,1.33,;1.42,4.41,;1.42,5.95,;2.96,4.41,;.17,5.31,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(CC[C@@H](CC1)NC(=O)c1ccncc1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:10.27,wD:13.17,(6.55,.22,;5.48,-.89,;3.99,-.52,;2.92,-1.63,;3.34,-3.11,;4.84,-3.48,;5.91,-2.37,;2.28,-4.21,;1.21,-5.32,;3.38,-5.28,;1.17,-3.14,;.31,-4.42,;-1.23,-4.31,;-1.91,-2.93,;-1.04,-1.65,;.49,-1.76,;-3.44,-2.82,;-4.3,-4.1,;-3.63,-5.48,;-5.84,-3.99,;-6.7,-5.27,;-8.24,-5.16,;-8.91,-3.78,;-8.05,-2.5,;-6.51,-2.61,;1.17,-1.6,;2.5,-.83,;2.5,.71,;1.17,1.48,;-.17,.71,;-.17,-.83,;1.17,3.02,;2.71,3.02,;-.37,3.02,;-1.91,3.02,;-.37,4.56,;-.37,1.48,;1.17,4.56,;1.17,6.1,;2.71,4.56,;-.08,5.46,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(CC[C@@H](CC1)NC(=O)c1cccnc1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:10.27,wD:13.17,(6.55,.22,;5.48,-.89,;3.99,-.52,;2.92,-1.63,;3.34,-3.11,;4.84,-3.48,;5.91,-2.37,;2.28,-4.21,;1.21,-5.32,;3.38,-5.28,;1.17,-3.14,;.31,-4.42,;-1.23,-4.31,;-1.91,-2.93,;-1.04,-1.65,;.49,-1.76,;-3.44,-2.82,;-4.3,-4.1,;-3.63,-5.48,;-5.84,-3.99,;-6.51,-2.61,;-8.05,-2.5,;-8.91,-3.78,;-8.24,-5.16,;-6.7,-5.27,;1.17,-1.6,;2.5,-.83,;2.5,.71,;1.17,1.48,;-.17,.71,;-.17,-.83,;1.17,3.02,;2.71,3.02,;-.37,3.02,;-1.91,3.02,;-.37,4.56,;-.37,1.48,;1.17,4.56,;1.17,6.1,;2.71,4.56,;-.08,5.46,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(CC[C@@H](CC1)NC(=O)c1cccnn1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:10.27,wD:13.17,(6.55,.22,;5.48,-.89,;3.99,-.52,;2.92,-1.63,;3.34,-3.11,;4.84,-3.48,;5.91,-2.37,;2.28,-4.21,;1.21,-5.32,;3.38,-5.28,;1.17,-3.14,;.31,-4.42,;-1.23,-4.31,;-1.91,-2.93,;-1.04,-1.65,;.49,-1.76,;-3.44,-2.82,;-4.3,-4.1,;-3.63,-5.48,;-5.84,-3.99,;-6.51,-2.61,;-8.05,-2.5,;-8.91,-3.78,;-8.24,-5.16,;-6.7,-5.27,;1.17,-1.6,;2.5,-.83,;2.5,.71,;1.17,1.48,;-.17,.71,;-.17,-.83,;1.17,3.02,;2.71,3.02,;-.37,3.02,;-1.91,3.02,;-.37,4.56,;-.37,1.48,;1.17,4.56,;1.17,6.1,;2.71,4.56,;-.08,5.46,)|
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Fc1ccc(cc1)S(=O)(=O)[C@@]1(CC[C@@H](CC1)NC(=O)Cc1ccncc1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:10.28,wD:13.17,(-8.02,.89,;-6.51,.62,;-5.98,-.82,;-4.46,-1.09,;-3.47,.09,;-4,1.53,;-5.52,1.8,;-1.96,-.18,;-2.22,-1.7,;-1.69,1.34,;-.44,-.45,;1.08,-.18,;2.07,-1.36,;1.54,-2.81,;.02,-3.07,;-.97,-1.89,;2.53,-3.99,;2,-5.43,;.49,-5.7,;2.99,-6.61,;2.47,-8.06,;3.46,-9.24,;2.93,-10.69,;1.41,-10.95,;.42,-9.77,;.95,-8.33,;-.44,1.09,;.89,1.86,;.89,3.4,;-.44,4.17,;-1.77,3.4,;-1.77,1.86,;-.44,5.71,;-.44,7.25,;1.1,5.71,;2.64,5.71,;1.1,4.17,;1.1,7.25,;-1.98,5.71,;-3.52,5.71,;-1.98,7.25,;-1.98,4.17,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(CC[C@@H](CC1)NC(=O)N1CCOCC1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:10.27,wD:13.17,(6.55,.22,;5.48,-.89,;3.99,-.52,;2.92,-1.63,;3.34,-3.11,;4.84,-3.48,;5.91,-2.37,;2.28,-4.21,;1.21,-5.32,;3.38,-5.28,;1.17,-3.14,;.31,-4.42,;-1.23,-4.31,;-1.91,-2.93,;-1.04,-1.65,;.49,-1.76,;-3.44,-2.82,;-4.3,-4.1,;-3.63,-5.48,;-5.84,-3.99,;-6.7,-5.27,;-8.24,-5.16,;-8.91,-3.78,;-8.05,-2.5,;-6.51,-2.61,;1.17,-1.6,;2.5,-.83,;2.5,.71,;1.17,1.48,;-.17,.71,;-.17,-.83,;1.17,3.02,;2.71,3.02,;-.37,3.02,;-1.91,3.02,;-.37,4.56,;-.37,1.48,;1.17,4.56,;1.17,6.1,;2.71,4.56,;-.08,5.46,)|
Cn1cc2CC(CCc2n1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
Cn1ncc2CC(CCc12)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CCn1ncc2CC(CCc12)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CCn1cc2CC(CCc2n1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CC(C)n1cc2CC(CCc2n1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CC(C)n1ncc2CC(CCc12)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
Fc1ccc(cc1)S(=O)(=O)C1(CCc2nn(Cc3ccncc3)cc2C1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCc2c(C1)cnn2Cc1ccncc1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCc2c(C1)cnn2C1CCOCC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
CC(=O)Nc1nc2CCC(Cc2s1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
Fc1ccc(cc1)S(=O)(=O)C1(CCc2nn(cc2C1)-c1ccncc1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)[C@@]1(CCc2nn(cc2C1)-c1ccncc1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r|
CC(=O)N1CCC(CC1)n1cc2C[C@](CCc2n1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCC(CC1)n1cc2C[C@@](CCc2n1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)c1ccc(cc1)-n1cc2CC(CCc2n1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CCOC(=O)Cn1cc2CC(CCc2n1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(=O)Cn1ncc2CC(CCc12)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CCOC(=O)CCn1ncc2CC(CCc12)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(=O)CCn1ncc2CC(CCc12)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
Fc1ccc(cc1)S(=O)(=O)C1(CCC(CC1)N1CCN(Cc2ccccc2)CC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |(8.35,-1.38,;6.83,-1.64,;5.84,-.46,;4.33,-.73,;3.8,-2.18,;4.79,-3.36,;6.31,-3.09,;2.28,-2.45,;2.55,-3.96,;2.02,-.93,;.77,-2.71,;1.29,-4.16,;.3,-5.34,;-1.21,-5.07,;-1.74,-3.63,;-.75,-2.45,;-2.2,-6.25,;-1.68,-7.7,;-2.67,-8.88,;-4.18,-8.61,;-5.17,-9.79,;-6.69,-9.52,;-7.68,-10.7,;-9.2,-10.44,;-9.72,-8.99,;-8.73,-7.81,;-7.22,-8.08,;-4.71,-7.17,;-3.72,-5.99,;.77,-1.17,;2.1,-.4,;2.1,1.14,;.77,1.91,;-.57,1.14,;-.57,-.4,;.77,3.45,;.77,4.99,;2.1,5.76,;2.1,7.3,;.77,8.07,;-.57,7.3,;.77,9.61,;2.1,10.38,;3.43,9.61,;3.43,8.07,;4.77,7.3,;2.31,3.45,;3.85,3.45,;2.31,1.91,;2.31,4.99,;-.77,3.45,;-2.31,3.45,;-.77,1.91,;-.77,4.99,)|
CC(=O)N1CCN(CC1)C1CCC(CC1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |(-4.86,-12.57,;-5.39,-11.13,;-6.9,-10.86,;-4.4,-9.95,;-2.88,-10.21,;-1.89,-9.03,;-2.42,-7.59,;-3.93,-7.32,;-4.92,-8.5,;-1.43,-6.41,;.09,-6.67,;1.08,-5.49,;.55,-4.05,;-.96,-3.78,;-1.95,-4.96,;.55,-2.51,;1.89,-1.74,;1.89,-.2,;.55,.57,;-.78,-.2,;-.78,-1.74,;.55,2.11,;.55,3.65,;1.89,4.42,;1.89,5.96,;.55,6.73,;-.78,5.96,;.55,8.27,;1.89,9.04,;3.22,8.27,;3.22,6.73,;4.55,5.96,;-.99,2.11,;-2.53,2.11,;-.99,.57,;-.99,3.65,;2.09,2.11,;3.63,2.11,;2.09,.57,;2.09,3.65,;2.07,-3.78,;2.34,-5.3,;1.8,-2.26,;3.59,-3.51,;4.11,-2.07,;5.63,-1.8,;6.62,-2.98,;8.14,-2.71,;6.09,-4.42,;4.58,-4.69,)|
CN1CCN(CC1)C1CCC(CC1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(=O)c1ccc(cc1)-n1ncc2CC(CCc12)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(=O)C1CCC(CC1)n1cc2CC(CCc2n1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |(-13.67,.38,;-12.9,-.95,;-13.67,-2.29,;-11.36,-.95,;-10.59,-2.29,;-9.05,-2.29,;-8.28,-.95,;-9.05,.38,;-10.59,.38,;-6.74,-.95,;-5.84,-2.2,;-4.37,-1.72,;-3.04,-2.49,;-1.7,-1.72,;-1.7,-.18,;-3.04,.59,;-4.37,-.18,;-5.84,.29,;-.19,-1.46,;.8,-2.63,;2.32,-2.37,;2.85,-.92,;1.86,.26,;.34,-.01,;4.36,-.65,;5.88,-.39,;6.41,1.06,;7.92,1.33,;8.45,2.78,;7.46,3.96,;9.97,3.04,;10.95,1.86,;10.43,.42,;8.91,.15,;8.38,-1.3,;4.09,.86,;3.83,2.38,;2.58,.6,;5.61,1.13,;4.63,-2.17,;4.9,-3.69,;3.11,-2.44,;6.15,-1.9,;-1.18,-3.17,;.27,-2.64,;-2.62,-3.7,;-.65,-4.62,;.87,-4.88,;1.39,-6.33,;.4,-7.51,;.93,-8.96,;-1.11,-7.24,;-1.64,-5.8,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(CCC(CC1)C#N)c1ccc(cc1)C(OCc1ccccc1)(C(F)(F)F)C(F)(F)F |r,wU:10.19,(-6.98,-4.21,;-5.46,-3.94,;-4.47,-5.12,;-2.95,-4.86,;-2.43,-3.41,;-3.42,-2.23,;-4.93,-2.5,;-.91,-3.14,;-1.18,-1.63,;-.64,-4.66,;.61,-2.87,;.08,-1.43,;1.07,-.25,;2.59,-.52,;3.11,-1.96,;2.12,-3.14,;3.58,.66,;4.57,1.84,;.61,-4.41,;-.73,-5.18,;-.73,-6.72,;.61,-7.49,;1.94,-6.72,;1.94,-5.18,;.61,-9.03,;.61,-10.57,;1.94,-11.34,;1.94,-12.88,;.61,-13.65,;.61,-15.19,;1.94,-15.96,;3.27,-15.19,;3.27,-13.65,;2.15,-9.03,;3.69,-9.03,;2.15,-7.49,;2.15,-10.57,;-.93,-9.03,;-2.47,-9.03,;-.93,-7.49,;-.93,-10.57,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(CCC(CC1)C#N)c1ccc(cc1)C(OCc1ccccc1)(C(F)(F)F)C(F)(F)F |r,wD:10.19,(-6.98,-4.21,;-5.46,-3.94,;-4.47,-5.12,;-2.95,-4.86,;-2.43,-3.41,;-3.42,-2.23,;-4.93,-2.5,;-.91,-3.14,;-1.18,-1.63,;-.64,-4.66,;.61,-2.87,;2.12,-3.14,;3.11,-1.96,;2.59,-.52,;1.07,-.25,;.08,-1.43,;3.58,.66,;4.57,1.84,;.61,-4.41,;-.73,-5.18,;-.73,-6.72,;.61,-7.49,;1.94,-6.72,;1.94,-5.18,;.61,-9.03,;.61,-10.57,;1.94,-11.34,;1.94,-12.88,;.61,-13.65,;.61,-15.19,;1.94,-15.96,;3.27,-15.19,;3.27,-13.65,;2.15,-9.03,;3.69,-9.03,;2.15,-7.49,;2.15,-10.57,;-.93,-9.03,;-2.47,-9.03,;-.93,-7.49,;-.93,-10.57,)|
Fc1ccc(cc1)S(=O)(=O)C1(CCC(CC1)N1CCN(Cc2ccccc2)CC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |(-4.27,-7.84,;-3.74,-6.39,;-2.22,-6.12,;-1.7,-4.67,;-2.69,-3.49,;-4.2,-3.76,;-4.73,-5.21,;-2.16,-2.05,;-.71,-2.57,;-3.61,-1.52,;-1.63,-.6,;-3.15,-.33,;-3.68,1.11,;-2.69,2.29,;-1.17,2.03,;-.64,.58,;-3.21,3.74,;-4.73,4.01,;-5.26,5.46,;-4.27,6.64,;-4.79,8.08,;-6.31,8.35,;-7.3,7.17,;-8.82,7.44,;-9.34,8.89,;-8.35,10.07,;-6.84,9.8,;-2.75,6.37,;-2.22,4.92,;-.3,-1.37,;-.3,-2.91,;1.03,-3.68,;2.37,-2.91,;2.37,-1.37,;1.03,-.6,;3.7,-3.68,;5.03,-4.45,;6.37,-3.68,;7.7,-4.45,;9.04,-3.68,;9.04,-2.14,;10.37,-4.45,;10.37,-5.99,;9.04,-6.76,;7.7,-5.99,;6.37,-6.76,;4.47,-2.35,;5.24,-1.01,;3.14,-1.58,;5.8,-3.12,;2.93,-5.01,;2.16,-6.35,;1.6,-4.24,;4.26,-5.78,)|
Fc1ccc(cc1)S(=O)(=O)C1(CCC(CC1)C#N)c1ccc(cc1)C(OCc1ccccc1)(C(F)(F)F)C(F)(F)F |w:13.17,(-6.98,1.46,;-5.46,1.72,;-4.47,.54,;-2.95,.81,;-2.43,2.26,;-3.42,3.44,;-4.93,3.17,;-.91,2.52,;-1.18,4.04,;-.64,1.01,;.61,2.79,;.08,4.24,;1.07,5.42,;2.59,5.15,;3.11,3.7,;2.12,2.52,;3.58,6.33,;4.57,7.51,;.61,1.25,;-.73,.48,;-.73,-1.06,;.61,-1.83,;1.94,-1.06,;1.94,.48,;.61,-3.37,;.61,-4.91,;1.94,-5.68,;1.94,-7.22,;.61,-7.99,;.61,-9.53,;1.94,-10.3,;3.27,-9.53,;3.27,-7.99,;2.15,-3.37,;3.69,-3.37,;2.15,-1.83,;2.15,-4.91,;-.93,-3.37,;-2.47,-3.37,;-.93,-1.83,;-.93,-4.91,)|
C[C@@H]1C[C@](CCC1NC(=O)OC(C)(C)C)(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
[#6]C([#6])([#6])[S@](=O)\[#7]=[#6]-1/[#6]-[#6]C([#6]-[#6]-1)(c1ccc(cc1)C([#8]-[#6]-c1ccccc1)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(C)OC(=O)NC1(C)CCC(CC1)(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |(-8.34,-2.39,;-7.13,-3.34,;-6.18,-2.12,;-8.07,-4.55,;-5.91,-4.29,;-4.48,-3.71,;-4.27,-2.18,;-3.27,-4.66,;-1.84,-4.08,;-2.16,-5.59,;-2.37,-2.63,;-1.38,-1.45,;.14,-1.72,;.66,-3.17,;-.33,-4.35,;.14,-.18,;1.47,.59,;1.47,2.13,;.14,2.9,;-1.2,2.13,;-1.2,.59,;.14,4.44,;.14,5.98,;1.68,4.44,;3.22,4.44,;1.68,2.9,;1.68,5.98,;-1.4,4.44,;-2.94,4.44,;-1.4,5.98,;-1.4,2.9,;1.65,-1.45,;1.39,.06,;1.92,-2.97,;3.17,-1.19,;3.7,.26,;5.21,.53,;6.2,-.65,;7.72,-.38,;5.68,-2.1,;4.16,-2.37,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(CC[C@@H](CC1)N1C(=O)c2ccncc2C1=O)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:13.17,wD:10.30,(-5.57,-6.34,;-4.39,-5.35,;-2.95,-5.88,;-1.77,-4.89,;-2.04,-3.37,;-3.48,-2.85,;-4.66,-3.84,;-.86,-2.38,;.13,-3.56,;-1.85,-1.2,;.32,-1.39,;1.09,-2.73,;2.63,-2.73,;3.4,-1.39,;2.63,-.06,;1.09,-.06,;4.94,-1.39,;5.85,-2.64,;5.37,-4.1,;7.31,-2.16,;8.65,-2.93,;9.98,-2.16,;9.98,-.62,;8.65,.15,;7.31,-.62,;5.85,-.15,;5.37,1.32,;-.86,-.4,;-.59,1.11,;-1.77,2.1,;-3.22,1.58,;-3.48,.06,;-2.3,-.93,;-4.39,2.57,;-5.57,3.56,;-3.4,3.75,;-2.42,4.92,;-2.23,2.76,;-4.58,4.74,;-5.38,1.39,;-6.37,.21,;-6.56,2.38,;-4.21,.4,)|
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CCOC(=O)c1cn(nn1)[C@H]1CC[C@@](CC1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:10.10,wD:13.17,(1.48,-14.22,;2.1,-12.81,;1.2,-11.57,;1.83,-10.16,;3.36,-10,;.92,-8.92,;1.4,-7.45,;.15,-6.55,;-1.1,-7.45,;-.62,-8.92,;.15,-5.01,;-1.18,-4.24,;-1.18,-2.7,;.15,-1.93,;1.48,-2.7,;1.48,-4.24,;-.84,-.75,;-.31,.7,;-1.3,1.88,;-2.82,1.61,;-3.35,.17,;-2.36,-1.01,;-3.81,2.79,;-4.8,3.97,;-2.63,3.78,;-1.45,4.77,;-1.64,2.6,;-3.62,4.96,;-4.99,1.8,;-6.17,.81,;-5.98,2.98,;-4,.62,;1.14,-.75,;-.04,.24,;2.32,-1.74,;2.13,.43,;1.6,1.88,;2.59,3.06,;4.11,2.79,;5.1,3.97,;4.64,1.35,;3.65,.17,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(CC[C@@H](CC1)n1cc(nn1)-c1cccnc1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:10.30,wD:13.17,(1.64,5.81,;.46,4.82,;-.98,5.35,;-2.16,4.36,;-1.9,2.84,;-.45,2.32,;.73,3.31,;-3.08,1.85,;-4.07,3.03,;-4.26,.86,;-2.09,.67,;-.75,-.1,;-.75,-1.64,;-2.09,-2.41,;-3.42,-1.64,;-3.42,-.1,;-2.09,-3.95,;-3.33,-4.85,;-2.86,-6.32,;-1.32,-6.32,;-.84,-4.85,;-3.76,-7.56,;-5.29,-7.4,;-6.2,-8.65,;-5.57,-10.05,;-4.04,-10.22,;-3.14,-8.97,;-.55,.57,;.12,-.82,;1.66,-.93,;2.52,.35,;1.85,1.74,;.31,1.84,;4.06,.24,;5.59,.14,;3.95,-1.29,;3.84,-2.83,;2.41,-1.19,;5.49,-1.4,;4.17,1.78,;4.27,3.32,;5.7,1.67,;2.63,1.89,)|
CC(C)(C)OC(=O)N1CC(C1)c1cn(nn1)[C@H]1CC[C@@](CC1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:16.17,wD:19.24,(-5.21,-15.33,;-5.21,-13.79,;-3.67,-13.79,;-6.75,-13.79,;-5.21,-12.25,;-3.87,-11.48,;-2.54,-12.25,;-3.87,-9.94,;-2.78,-8.85,;-3.87,-7.76,;-4.96,-8.85,;-3.87,-6.22,;-2.63,-5.31,;-3.1,-3.85,;-4.64,-3.85,;-5.12,-5.31,;-2.2,-2.6,;-2.82,-1.2,;-1.92,.05,;-.39,-.11,;.24,-1.52,;-.67,-2.76,;-.49,1.42,;.78,2.29,;.67,3.82,;-.71,4.5,;-1.99,3.64,;-1.88,2.1,;-.82,6.03,;-.92,7.57,;.72,6.14,;2.26,6.25,;.83,4.6,;.61,7.68,;-2.35,5.93,;-3.89,5.82,;-2.46,7.46,;-2.25,4.39,;1.11,.26,;.73,1.76,;1.48,-1.23,;2.6,.63,;3.03,2.11,;4.52,2.49,;5.59,1.38,;7.08,1.75,;5.17,-.1,;3.67,-.47,)|
OC(=O)c1cn(nn1)[C@H]1CC[C@@](CC1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:8.8,wD:11.15,(-.64,7.93,;.69,7.16,;2.03,7.93,;.69,5.62,;-.55,4.71,;-.08,3.25,;1.46,3.25,;1.94,4.71,;-.98,2,;-.36,.6,;-1.26,-.65,;-2.79,-.49,;-3.42,.92,;-2.51,2.17,;-1.49,-1.3,;-1.54,-2.84,;-.23,-3.66,;1.13,-2.94,;1.18,-1.4,;-.13,-.58,;2.43,-3.75,;1.62,-5.06,;3.25,-2.45,;4.06,-1.14,;4.55,-3.26,;1.94,-1.63,;3.74,-4.57,;5.04,-5.38,;2.92,-5.87,;5.17,-3.99,;-4.29,-.86,;-4.66,.63,;-5.78,-1.23,;-3.91,-2.35,;-2.43,-2.78,;-2.06,-4.27,;-3.17,-5.34,;-2.8,-6.84,;-4.65,-4.92,;-5.02,-3.42,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(CC[C@@H](CC1)n1cc(nn1)C(=O)N1CCOCC1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:13.17,wD:10.32,(-2.94,-8.61,;-3.31,-7.12,;-2.2,-6.05,;-2.57,-4.55,;-4.05,-4.13,;-5.16,-5.2,;-4.79,-6.69,;-4.43,-2.63,;-4.8,-1.14,;-5.92,-3.01,;-2.93,-2.26,;-1.4,-2.42,;-.5,-1.18,;-1.12,.23,;-2.65,.39,;-3.56,-.85,;-.22,1.48,;-.69,2.94,;.55,3.85,;1.8,2.94,;1.32,1.48,;.55,5.39,;-.78,6.16,;1.89,6.16,;1.89,7.7,;3.22,8.47,;4.55,7.7,;4.55,6.16,;3.22,5.39,;-1.63,-3.08,;-1.68,-4.62,;-.37,-5.43,;.99,-4.71,;1.04,-3.17,;-.27,-2.35,;2.29,-5.52,;1.48,-6.83,;3.11,-4.22,;3.92,-2.91,;4.41,-5.03,;1.8,-3.4,;3.6,-6.34,;4.9,-7.16,;2.78,-7.65,;5.03,-5.76,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(CC[C@@H](CC1)n1cc(nn1)C(=O)Nc1cccnc1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:10.33,wD:13.17,(-8.89,-3.75,;-7.4,-3.37,;-6.33,-4.48,;-4.83,-4.11,;-4.41,-2.63,;-5.48,-1.52,;-6.97,-1.89,;-2.91,-2.26,;-3.29,-.76,;-2.54,-3.75,;-1.42,-1.88,;-2.05,-.48,;-1.14,.77,;.39,.61,;1.02,-.8,;.11,-2.04,;1.3,1.85,;.82,3.32,;2.07,4.22,;3.31,3.32,;2.84,1.85,;2.07,5.76,;.73,6.53,;3.4,6.53,;3.4,8.07,;4.73,8.84,;4.73,10.38,;3.4,11.15,;2.07,10.38,;2.07,8.84,;-1.31,-3.42,;-2.59,-4.28,;-2.48,-5.82,;-1.1,-6.49,;.18,-5.63,;.07,-4.1,;-.99,-8.03,;-.88,-9.57,;.55,-7.92,;2.08,-7.81,;.65,-9.46,;.44,-6.39,;-2.53,-8.14,;-4.06,-8.24,;-2.63,-6.6,;-2.42,-9.67,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(CC[C@@H](CC1)n1cc(nn1)C1CNC1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:10.28,wD:13.17,(2.94,-6.14,;2.57,-4.64,;3.68,-3.57,;3.31,-2.08,;1.83,-1.66,;.72,-2.73,;1.09,-4.22,;1.45,-.16,;1.08,1.33,;2.95,.21,;-.04,-.53,;.59,-1.94,;-.32,-3.19,;-1.85,-3.03,;-2.48,-1.62,;-1.57,-.37,;-2.76,-4.27,;-2.28,-5.74,;-3.53,-6.64,;-4.77,-5.74,;-4.3,-4.27,;-3.53,-8.18,;-2.44,-9.27,;-3.53,-10.36,;-4.61,-9.27,;-.15,1,;1.13,1.86,;1.02,3.4,;-.36,4.07,;-1.64,3.21,;-1.53,1.68,;-.47,5.61,;-.58,7.15,;-2.01,5.5,;-3.54,5.4,;-2.11,7.04,;-1.9,3.97,;1.07,5.72,;2.6,5.83,;1.17,4.18,;.96,7.25,)|
C[C@@H]1C[C@](CCC1NC(=O)OC(C)(C)C)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@@H]1C[C@](CCC1NC(=O)Cc1ccncc1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
COC(=O)C1CCC(CC1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |(-3.73,-8.52,;-2.74,-7.34,;-3.27,-5.89,;-4.79,-5.63,;-2.28,-4.71,;-2.81,-3.27,;-1.82,-2.09,;-.3,-2.35,;.23,-3.8,;-.76,-4.98,;-.3,-.81,;1.03,-.04,;1.03,1.5,;-.3,2.27,;-1.63,1.5,;-1.63,-.04,;-.3,3.81,;1.24,3.81,;-.3,5.35,;-.3,6.89,;1.24,5.35,;-1.84,5.35,;-1.84,3.81,;-3.38,3.81,;-2.74,5.05,;-1.84,2.27,;1.22,-2.09,;2.73,-1.82,;.95,-.57,;1.48,-3.6,;2.93,-4.13,;3.2,-5.65,;2.02,-6.64,;2.29,-8.15,;.57,-6.11,;.3,-4.59,)|
Fc1ccc(cc1)S(=O)(=O)C1(CCC(CC1)C(=O)Nc1ccnnc1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |(-6.43,-.44,;-5.36,-1.54,;-5.79,-3.02,;-4.72,-4.13,;-3.22,-3.76,;-2.8,-2.28,;-3.87,-1.17,;-2.15,-4.87,;-3.26,-5.94,;-1.08,-5.98,;-1.05,-3.8,;-.37,-2.41,;1.17,-2.31,;2.03,-3.58,;1.35,-4.97,;-.18,-5.07,;3.56,-3.48,;4.24,-2.09,;4.42,-4.75,;5.96,-4.64,;6.64,-3.26,;8.17,-3.15,;9.03,-4.43,;8.36,-5.81,;6.82,-5.92,;-1.05,-2.26,;.29,-1.49,;.29,.05,;-1.05,.82,;-2.38,.05,;-2.38,-1.49,;-1.05,2.36,;-2.59,2.36,;-1.05,3.9,;-1.05,5.44,;.49,3.9,;-2.59,3.9,;.49,2.36,;2.03,2.36,;.49,.82,;1.4,3.61,)|
CC1(O)CCN(CC1)C(=O)C1CCC(CC1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |(7.25,-7.77,;5.89,-7.05,;6.06,-8.58,;6.57,-5.66,;5.71,-4.39,;4.17,-4.5,;3.5,-5.88,;4.36,-7.16,;3.31,-3.22,;3.99,-1.83,;1.77,-3.33,;.91,-2.05,;-.62,-2.16,;-1.3,-3.54,;-.44,-4.82,;1.1,-4.71,;-1.3,-2,;.04,-1.23,;.04,.31,;-1.3,1.08,;-2.63,.31,;-2.63,-1.23,;-1.3,2.62,;-2.84,2.62,;-1.3,4.16,;-1.3,5.7,;.24,4.16,;-2.84,4.16,;.24,2.62,;1.78,2.62,;.24,1.08,;1.15,3.86,;-2.41,-4.61,;-3.51,-5.68,;-1.34,-5.72,;-3.48,-3.5,;-4.97,-3.88,;-6.04,-2.77,;-5.61,-1.29,;-6.68,-.18,;-4.12,-.91,;-3.05,-2.02,)|
Fc1ccc(cc1)S(=O)(=O)C1(CCC(CC1)C(=O)NCc1ccnnc1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |(7.56,-1.05,;6.04,-1.32,;5.05,-.14,;3.54,-.41,;3.01,-1.86,;4,-3.04,;5.51,-2.77,;1.49,-2.12,;1.22,-.61,;1.76,-3.64,;-.02,-2.39,;.5,-3.84,;-.49,-5.02,;-2,-4.75,;-2.53,-3.3,;-1.54,-2.12,;-2.99,-5.93,;-4.51,-5.66,;-2.47,-7.38,;-3.46,-8.56,;-2.93,-10,;-3.92,-11.18,;-3.39,-12.63,;-1.88,-12.9,;-.89,-11.72,;-1.41,-10.27,;-.02,-.85,;1.31,-.08,;1.31,1.46,;-.02,2.23,;-1.36,1.46,;-1.36,-.08,;-.02,3.77,;-.02,5.31,;1.52,3.77,;3.06,3.77,;1.52,2.23,;1.52,5.31,;-1.56,3.77,;-3.1,3.77,;-1.56,5.31,;-1.56,2.23,)|
Fc1ccc(cc1)S(=O)(=O)C1(CCC(CC1)C(=O)N1CCS(=O)(=O)CC1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |(-7.34,-.9,;-5.83,-1.17,;-5.3,-2.62,;-3.78,-2.89,;-2.79,-1.71,;-3.32,-.26,;-4.84,.01,;-1.28,-1.97,;-1.55,-3.49,;-1.01,-.46,;.24,-2.24,;1.76,-1.97,;2.74,-3.15,;2.22,-4.6,;.7,-4.87,;-.29,-3.69,;3.21,-5.78,;4.72,-5.51,;2.68,-7.23,;3.67,-8.41,;3.14,-9.85,;1.63,-10.12,;1.84,-11.65,;.48,-11.15,;.64,-8.94,;1.16,-7.5,;.24,-.7,;1.57,.07,;1.57,1.61,;.24,2.38,;-1.1,1.61,;-1.1,.07,;.24,3.92,;.24,5.46,;1.78,3.92,;3.32,3.92,;1.78,2.38,;1.78,5.46,;-1.3,3.92,;-2.84,3.92,;-1.3,5.46,;-1.3,2.38,)|
Fc1ccc(cc1)S(=O)(=O)C1(CCC(CC1)C(=O)N1CCC(C1)c1ccncc1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |(-.35,-9.89,;-1.02,-8.5,;-.16,-7.23,;-.83,-5.84,;-2.37,-5.74,;-3.23,-7.01,;-2.56,-8.4,;-3.05,-4.35,;-3.72,-2.97,;-4.43,-5.03,;-1.66,-3.68,;-2.57,-2.43,;-1.94,-1.02,;-.41,-.86,;.5,-2.11,;-.13,-3.52,;.22,.54,;1.75,.71,;-.69,1.79,;-2.23,1.79,;-2.7,3.26,;-1.46,4.16,;-.21,3.26,;-1.46,5.7,;-2.79,6.47,;-2.79,8.01,;-1.46,8.78,;-.12,8.01,;-.12,6.47,;-.21,-4.2,;.05,-5.72,;1.5,-6.25,;2.68,-5.26,;2.41,-3.74,;.96,-3.21,;4.13,-5.78,;3.6,-7.23,;4.65,-4.34,;5.18,-2.89,;6.1,-4.86,;3.21,-3.81,;5.57,-6.31,;7.02,-6.84,;5.05,-7.76,;6.85,-5.45,)|
Fc1ccc(cc1)S(=O)(=O)C1(CCC(CC1)C(=O)NCC1CCOCC1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |(7.56,-1.05,;6.04,-1.32,;5.05,-.14,;3.54,-.41,;3.01,-1.86,;4,-3.04,;5.51,-2.77,;1.49,-2.12,;1.22,-.61,;1.76,-3.64,;-.02,-2.39,;.5,-3.84,;-.49,-5.02,;-2,-4.75,;-2.53,-3.3,;-1.54,-2.12,;-2.99,-5.93,;-4.51,-5.66,;-2.47,-7.38,;-3.46,-8.56,;-2.93,-10,;-1.41,-10.27,;-.89,-11.72,;-1.88,-12.9,;-3.39,-12.63,;-3.92,-11.18,;-.02,-.85,;1.31,-.08,;1.31,1.46,;-.02,2.23,;-1.36,1.46,;-1.36,-.08,;-.02,3.77,;-.02,5.31,;1.52,3.77,;3.06,3.77,;1.52,2.23,;1.52,5.31,;-1.56,3.77,;-3.1,3.77,;-1.56,5.31,;-1.56,2.23,)|
CC(=O)N1CCN(CC1)C(=O)C1CCC(CC1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |(8.15,-8.35,;6.61,-8.45,;5.93,-9.84,;5.75,-7.18,;6.42,-5.79,;5.56,-4.52,;4.03,-4.62,;3.35,-6.01,;4.21,-7.28,;3.17,-3.35,;3.84,-1.96,;1.63,-3.45,;.77,-2.18,;-.77,-2.28,;-1.44,-3.67,;-.58,-4.94,;.95,-4.84,;-1.44,-2.13,;-.11,-1.36,;-.11,.18,;-1.44,.95,;-2.78,.18,;-2.78,-1.36,;-1.44,2.49,;-2.98,2.49,;-1.44,4.03,;-1.44,5.57,;.1,4.03,;-2.98,4.03,;.1,2.49,;1.64,2.49,;.1,.95,;1,3.74,;-2.55,-4.74,;-3.66,-5.81,;-1.48,-5.85,;-3.62,-3.63,;-5.12,-4,;-6.19,-2.9,;-5.76,-1.41,;-6.83,-.31,;-4.27,-1.04,;-3.2,-2.15,)|
Cc1n[nH]c(C)c1CNC(=O)C1CCC(CC1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
Fc1ccc(cc1)S(=O)(=O)C1(CCC(CC1)C(=O)NCC1CCS(=O)(=O)CC1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |(7.49,-.51,;6.42,-1.62,;4.93,-1.25,;3.86,-2.35,;4.29,-3.83,;5.78,-4.21,;6.85,-3.1,;3.22,-4.94,;2.15,-6.05,;4.32,-6.01,;2.11,-3.87,;1.25,-5.15,;-.29,-5.04,;-.96,-3.66,;-.1,-2.38,;1.43,-2.49,;-2.5,-3.55,;-3.18,-2.17,;-3.36,-4.83,;-4.9,-4.72,;-5.76,-6,;-5.08,-7.38,;-5.95,-8.66,;-7.48,-8.55,;-7.64,-10.08,;-8.84,-9.27,;-8.16,-7.17,;-7.3,-5.89,;2.11,-2.33,;3.44,-1.56,;3.44,-.02,;2.11,.75,;.77,-.02,;.77,-1.56,;2.11,2.29,;3.65,2.29,;.57,2.29,;-.97,2.29,;.57,3.83,;.57,.75,;2.11,3.83,;2.11,5.37,;3.65,3.83,;.86,4.73,)|
Fc1ccc(cc1)S(=O)(=O)C1(CCC(CC1)C(=O)NC1(CC1)c1ccncc1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |(1.7,5.55,;1.43,4.04,;-.01,3.51,;-.28,1.99,;.9,1,;2.35,1.53,;2.61,3.05,;.63,-.51,;-.88,-.25,;2.15,-.78,;.36,-2.03,;.63,-3.55,;-.55,-4.54,;-1.99,-4.01,;-2.26,-2.49,;-1.08,-1.5,;-3.17,-5,;-2.91,-6.52,;-4.62,-4.47,;-5.8,-5.46,;-5.03,-6.8,;-6.57,-6.8,;-6.98,-4.47,;-8.43,-5,;-9.61,-4.01,;-9.34,-2.49,;-7.89,-1.97,;-6.71,-2.96,;1.9,-2.03,;2.67,-3.36,;4.21,-3.36,;4.98,-2.03,;4.21,-.7,;2.67,-.7,;6.52,-2.03,;8.06,-2.03,;6.52,-3.57,;6.52,-5.11,;4.98,-3.57,;8.06,-3.57,;6.52,-.49,;6.52,1.05,;8.06,-.49,;4.98,-.49,)|
Fc1ccc(cc1)S(=O)(=O)C1(CCC(CC1)C(=O)NCc1cn[nH]c1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |(7.32,-3.78,;5.81,-3.52,;5.28,-2.07,;3.76,-1.8,;2.77,-2.98,;3.3,-4.43,;4.82,-4.7,;1.26,-2.72,;1.52,-1.2,;.99,-4.23,;-.26,-2.45,;-1.59,-1.68,;-2.93,-2.45,;-2.93,-3.99,;-1.59,-4.76,;-.26,-3.99,;-4.26,-4.76,;-5.6,-3.99,;-4.26,-6.3,;-5.6,-7.07,;-5.6,-8.61,;-4.35,-9.51,;-4.83,-10.98,;-6.37,-10.98,;-6.84,-9.51,;.27,-1,;1.78,-.73,;2.31,.71,;1.32,1.89,;-.2,1.63,;-.72,.18,;1.85,3.34,;2.37,4.79,;3.29,2.81,;4.74,2.29,;2.77,1.37,;3.82,4.26,;.4,3.87,;-1.05,4.39,;.93,5.31,;-.13,2.42,)|
Fc1ccc(cc1)S(=O)(=O)C1(CCC(CC1)C(=O)NCCc1ccncc1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F
OC(c1ccc(CBr)cc1)(C(F)(F)F)C(F)(F)F
O=COCc1ccc2NCCCc2c1
OC(c1ccc(CN2CCCc3cc(COC=O)ccc23)cc1)(C(F)(F)F)C(F)(F)F
CN(C)C(=O)c1ccc2N(Cc3ccc(cc3)C(O)(C(F)(F)F)C(F)(F)F)CCCc2c1
Brc1ccc2NC(=O)CCc2c1
OC(c1ccc(CN2C(=O)CCc3cc(COC=O)ccc23)cc1)(C(F)(F)F)C(F)(F)F
CN(C)C(=O)c1ccc2N(Cc3ccc(cc3)C(O)(C(F)(F)F)C(F)(F)F)C(=O)CCc2c1
Brc1ccc(NC(=O)\C=C\c2ccccc2)cc1
OC(c1ccc(Cn2c3ccc(COC=O)cc3ccc2=O)cc1)(C(F)(F)F)C(F)(F)F
CC(C)(C)NS(=O)(=O)c1ccc(cc1C(F)(F)F)-c1sc(nc1CC1CCCCC1)-c1nnc(o1)C(C)(C)O
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)-c2nnc(o2)C(C)(C)O)c2ccccc12
Cc1nnc(o1)-c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2nnc(CC(C)(C)C(O)=O)o2)c(Cl)c1Cl
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)-c2nnc(CC(C)(C)C(O)=O)o2)c2ccccc12
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)-c2nnc(CC(C)(C)C(O)=O)o2)c(Cl)c1Cl
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2nnc(CC(C)(C)C(O)=O)o2)c2ccccc12)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2nnc(CC(C)(C)C(O)=O)o2)c(Cl)c1Cl)C(F)(F)F |r|
CC(C)(Cc1nnc(o1)-c1nc(CC2CCC2)c(s1)-c1ccc(c(Cl)c1Cl)S(=O)(=O)NCC(F)(F)F)C(O)=O
CC(C)(Cc1nnc(o1)-c1nc(CC2CCC2)c(s1)-c1ccc(CN2CCOCC2(C)C)c(Cl)c1Cl)C(O)=O
CC(C)(Cc1nnc(o1)-c1nc(CC2CCC2)c(s1)-c1ccc(CN2CCOCC2(C)C)c2ccccc12)C(O)=O
CC(N1CCOCC1(C)C)c1ccc(-c2sc(nc2CC2CCC2)-c2nnc(CC(C)(C)C(O)=O)o2)c2ccccc12
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2nnc(CC(C)(C)OC=O)o2)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2nnc(CC(C)(C)OC=O)o2)c(Cl)c1)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2nnc(CC(C)(C)OC=O)o2)c(OC(F)(F)F)c1)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2nnc(CC(C)(C)OC=O)o2)c(c1)C(F)(F)F)C(F)(F)F |r|
CC(C)Cc1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)N[C@@H](C)C(F)(F)F)-c1nnc(CC(C)(C)OC=O)o1 |r|
CC(C)Cc1nc(sc1-c1ccc(cc1OC(F)(F)F)S(=O)(=O)N[C@@H](C)C(F)(F)F)-c1nnc(CC(C)(C)OC=O)o1 |r|
C[C@H](NS(=O)(=O)c1ncc(-c2sc(nc2CC2CCCCC2)-c2nnc(CC(C)(C)OC=O)o2)c2ccccc12)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2nnc(CC(C)(C)OC=O)o2)c2ccncc12)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2nnc(CC(C)(C)OC=O)o2)c2cnccc12)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2nnc(CC(C)(C)OC=O)o2)c(OC(F)(F)F)c1)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2nnc(CC(C)(C)OC=O)o2)c(Cl)c1)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)-c2nnc(CC(C)(C)OC=O)o2)c2ccccc12)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)-c2nnc(CC(C)(C)OC=O)o2)c(OC(F)(F)F)c1)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)-c2nnc(CC(C)(C)C(O)=O)o2)c2ccncc12)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)-c2nnc(CC(C)(C)C(O)=O)o2)c2ccncc12)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)-c2nnc(CC(C)(C)C(O)=O)o2)c(C(F)F)c1F)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2nnc(CC(C)(C)C(O)=O)o2)c(C(F)F)c1F)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)-c2nnc(CC(C)(C)C(O)=O)o2)c(C(F)F)c1F)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC(C)(C)OC)-c2nnc(CC(C)(C)OC=O)o2)c2ccccc12)C(F)(F)F |r|
COC(C)(C)Cc1nc(sc1-c1ccc(c2ccccc12)S(=O)(=O)N[C@@H](C)C(F)(F)F)-c1nnc(CC(C)(C)OC=O)o1 |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CC(C)(C)C2)-c2nnc(CC(C)(C)C(O)=O)o2)c(Cl)c1Cl)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CC(F)(F)C2)-c2nnc(CC(C)(C)C(O)=O)o2)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CC(F)(F)C2)-c2nnc(CC(C)(C)C(O)=O)o2)c2ccccc12)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2Cc2ccc(F)cc2)-c2nnc(CC(C)(C)C(O)=O)o2)c(C(F)F)c1F)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2Cc2ccc(F)cc2)-c2nnc(CC(C)(C)C(O)=O)o2)c(Cl)c1Cl)C(F)(F)F |r|
CC(C)(Cc1nnc(o1)-c1nc(CC2CCC2)c(s1)-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(O)=O
C[C@H](NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCC1)-c1nnc(CC(C)(C)OC=O)o1)C(F)(F)F |r|
CC(C)(C)c1cc(cc(c1)C(O)(C(F)(F)F)C(F)(F)F)-c1sc(nc1CC1CCC1)-c1nnc(CC(C)(C)C(O)=O)o1
C[C@H](NC(=O)c1cc(cc(c1)C1(CC1)C(F)(F)F)-c1sc(nc1CC1CCC1)-c1nnc(CC(C)(C)C(O)=O)o1)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCC2)-c2nnc(CC(C)(C)C(O)=O)o2)c(C(F)F)c1F)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2COC(C)C)-c2nnc(CC(C)(C)C(O)=O)o2)c2ccccc12)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCC2)-c2nnc(CC(C)(C)C(O)=O)o2)c(C(F)F)c1Cl)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCC2)-c2nnc(CC(C)(C)C(O)=O)o2)c(F)c1C(F)F)C(F)(F)F |r|
CC(C)(Cc1nnc(o1)-c1nc(Cc2ccc(F)cc2)c(s1)-c1ccc(cc1C(F)F)C(O)(C(F)(F)F)C(F)(F)F)C(O)=O
CC[C@@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2nnc(CC(C)(C)C(O)=O)o2)c(C(F)F)c1F)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC(C)(C)OC)-c2nnc(CC(C)(C)OC=O)o2)c(Cl)c1Cl)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CC(F)(F)C2)-c2nnc(CC(C)(C)C(O)=O)o2)c2ccccc12)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2nnc(o2)[C@H]2C[C@@H](C2)OC=O)c(Cl)c1Cl)C(F)(F)F |r,wU:1.0,27.32,wD:25.27,(2.83,-6.51,;1.36,-6.99,;.22,-5.96,;.54,-4.45,;-.97,-4.13,;2.05,-4.77,;.86,-2.94,;2.32,-2.47,;2.64,-.96,;1.5,.07,;1.82,1.57,;.79,2.72,;1.56,4.05,;3.07,3.73,;3.23,2.2,;4.56,1.43,;4.56,-.11,;5.65,-1.2,;4.56,-2.29,;3.47,-1.2,;.93,5.46,;-.57,5.78,;-.73,7.31,;.67,7.94,;1.7,6.79,;.99,9.44,;2.28,10.28,;1.45,11.57,;.15,10.74,;1.77,13.08,;3.23,13.56,;3.55,15.06,;.04,-.41,;-1.11,.62,;-.28,-1.91,;-1.75,-2.39,;1.04,-8.49,;.72,-10,;2.55,-8.81,;-.46,-8.17,)|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CN2CCCC(F)(F)C2)-c2nnc(o2)C(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CN2CCCC(F)(F)C2)-c2nnc(CC(C)(C)C(O)=O)o2)c(Cl)c1Cl)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CN2CCC[C@@H](F)C2)-c2nnc(CC(C)(C)C(O)=O)o2)c2ccccc12)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CN2CCCC(F)(F)C2)-c2nnc(CC(C)(C)C(O)=O)o2)c2ccccc12)C(F)(F)F |r|
CC(C)(Cc1nnc(o1)-c1nc(CN2CCCC(F)(F)C2)c(s1)-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(O)=O
CC(C)(Cc1nnc(o1)-c1nc(CN2CCC[C@@H](F)C2)c(s1)-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(O)=O |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2nnc(CC(C)(C)OC=O)s2)c(Cl)c1Cl)C(F)(F)F |r|
Cc1nc(no1)-c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2noc(CC(C)(C)OC=O)n2)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2noc(CC(C)(C)OC=O)n2)c(OC(F)(F)F)c1)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)-c2noc(CC(C)(C)OC=O)n2)c2ccncc12)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)-c2noc(CC(C)(C)OC=O)n2)c2cnccc12)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)-c2noc(CC(C)(C)OC=O)n2)c(OC(F)(F)F)c1)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ncc(-c2sc(nc2CC2CCC2)-c2noc(CC(C)(C)OC=O)n2)c2ccccc12)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2noc(CC(C)(C)OC=O)n2)c(C(F)F)c1F)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2noc(CC(C)(C)OC=O)n2)c(c1F)C(F)(F)F)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC(C)(C)OC)-c2noc(CC(C)(C)OC=O)n2)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)-c1noc(CC(C)(C)OC=O)n1)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2(CCC2)OC)-c2noc(CC(C)(C)OC=O)n2)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2noc(CC(C)(C)C(O)=O)n2)c(C(F)F)c1Cl)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CN2CCCC(F)(F)C2)-c2noc(CC(C)(C)C(O)=O)n2)c(C(F)F)c1F)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CN2CCCC(F)(F)C2)-c2noc(CC(C)(C)OC=O)n2)c(Cl)c1Cl)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CN2CC(F)(F)C[C@@H]2C)-c2noc(CC(C)(C)OC=O)n2)c(Cl)c1Cl)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CN2CC(F)(F)C[C@@H]2C)-c2noc(CC(C)(C)C(O)=O)n2)c(C(F)F)c1F)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CN2CCC[C@@H]2C)-c2noc(CC(C)(C)C(O)=O)n2)c(C(F)F)c1F)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CN2CCC(F)(F)[C@@H]2C)-c2noc(CC(C)(C)C(O)=O)n2)c(C(F)F)c1F)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CN2CC(F)(F)CC2(C)C)-c2noc(CC(C)(C)C(O)=O)n2)c(C(F)F)c1F)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CN2CCC[C@@H]2CF)-c2noc(CC(C)(C)C(O)=O)n2)c(C(F)F)c1F)C(F)(F)F |r|
Cc1noc(n1)-c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC(C)(C)C
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2cc(CC(C)(C)C)on2)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2cccc(CC(C)(C)OC=O)c2)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2cccc(CC(C)(C)OC=O)n2)c2ccncc12)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2cc(CC(C)(C)OC=O)ncn2)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2cc(CC(C)(C)OC=O)ncn2)c2ccncc12)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2cnc(CC(C)(C)C(O)=O)s2)c(Cl)c1Cl)C(F)(F)F |r|
COCCN1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2cc3c(C)cc(cc3n2C)C(F)(F)F)c1Cl
Cc1cc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCN(CC4)C4COC4)c3Cl)cc12)C(F)(F)F
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CC(C)n1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2c(C)cc(cc12)C#N
Cc1cc(nc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)nc12)C#N
Cn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)cc2c(Cl)cc(cc12)C#N
Cn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)cc2cccnc12
Cc1cc(nc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)cc12)C#N
Cc1cc(nc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(O)CC4)c3Cl)cc12)C#N
Cc1cc(nc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC4)C4COC4)c3Cl)cc12)C#N
Cc1cc(nc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)cc12)C(F)(F)F
Cc1cc(Cl)nc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)cc12
Cn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)cc2ncc(cc12)C(F)(F)F
Cn1c(cc2ncc(cc12)C(F)(F)F)C(=O)c1c(Cl)ccc(C(=O)N2CCOCC2)c1Cl
Cn1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)cc2cnc(cc12)C(F)(F)F
Cc1nc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)cc12)C(F)(F)F
Cc1nc(cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)cc12)C#N
Cc1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2c(C)cc(cn12)C(F)(F)F
Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(O)CC3)c2Cl)nc2c(C)cc(cn12)C(F)(F)F
Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(CCO)CC3)c2Cl)nc2c(C)cc(cn12)C(F)(F)F
Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC3)C(C)(C)O)c2Cl)nc2c(C)cc(cn12)C(F)(F)F
Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(O)C3)c2Cl)nc2c(C)cc(cn12)C(F)(F)F
CN(C)C1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cn3c2C)C(F)(F)F)c1Cl
COC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cn3c2C)C(F)(F)F)c1Cl
COCCC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cn3c2C)C(F)(F)F)c1Cl
Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC3)C3COC3)c2Cl)nc2c(C)cc(cn12)C(F)(F)F
Cc1c(Cc2c(Cl)ccc(C(=O)N3CCN(CC3)C3COC3)c2Cl)nc2c(C)cc(cn12)C(F)(F)F
Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(CO)CC3)c2Cl)nc2c(C)cc(cn12)C(F)(F)F
CC(O)C1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cn3c2C)C(F)(F)F)c1Cl
Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)nc2c(C)cc(cn12)C(F)(F)F
Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(CCO)CC3)c2Cl)nc2c(C)cc(cn12)C#N
Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(CO)CC3)c2Cl)nc2c(C)cc(cn12)C#N
COC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cn3c2C)C#N)c1Cl
Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC3)C(C)(C)O)c2Cl)nc2c(C)cc(cn12)C#N
CC(O)C1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cn3c2C)C#N)c1Cl
Cc1c(Cc2c(Cl)ccc(C(=O)N3CCC(CC3)C3COC3)c2Cl)nc2c(C)cc(cn12)C#N
COCCC1CCN(CC1)C(=O)c1ccc(Cl)c(Cc2nc3c(C)cc(cn3c2C)C#N)c1Cl
Cc1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2c(C)cc(Cl)nn12
Cc1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2cc(C)c(Cl)nn12
Cc1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2c(C)cc(nn12)C(F)(F)F
Cc1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2c(C)cc(nn12)C#N
Cc1c(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2cc(C)c(nn12)C#N
Cc1cc(nc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCOCC4)c3Cl)nc12)C(F)(F)F
Cc1nn(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)c2c(C)cc(cc12)C(F)(F)F
Cc1nn(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2c(C)cc(cc12)C(F)(F)F
Cc1n(Cc2c(Cl)ccc(C(=O)N3CCOCC3)c2Cl)nc2c(C)cc(cc12)C(F)(F)F
Cc1n(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)nc2c(C)cc(cc12)C(F)(F)F
Cc1cn(Cc2c(Cl)ccc(C(=O)N3CCC(CC3)C(O)=O)c2Cl)c2c(C)cc(cc12)C(F)(F)F
Cc1cn(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2c(C)cc(cc12)C(F)(F)F
Cc1cn(C(=O)c2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2c(C)cc(cc12)C(F)(F)F
Cc1cn(Cc2c(Cl)ccc(C(=O)N3CCC(O)CC3)c2Cl)c2c(C)cc(cc12)C#N
Cc1cn(Cc2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2c(C)cc(cc12)C#N
Cc1cn(C(=O)c2c(Cl)ccc(C(=O)N3CCC(O)CC3)c2Cl)c2c(C)cc(cc12)C#N
Cc1cn(C(=O)c2c(Cl)ccc(C(=O)N3CCC(CC(O)=O)CC3)c2Cl)c2c(C)cc(cc12)C#N
Cc1cc(nc2n(C)c(Cc3c(Cl)ncc(C(=O)N4CCC(O)CC4)c3Cl)cc12)C(F)(F)F
Cc1cc(OC(F)(F)F)cc2n(C)c(Cc3c(Cl)ccc(C(=O)N4CCC(CC(O)=O)CC4)c3Cl)cc12
CCC(CC)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(CC)ncnc1C1CC1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C3CCCC3)c2=O)-c2c(C)ncnc2C2CC2)nc1
CCc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(=O)(=O)CC)c(=O)n(C3CCCC3)c2n1
CCC(CC)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(OC)ncnc1C1CC1
CCc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(=O)(=O)CC)c(=O)n([C@@H](C)C(C)C)c2n1 |r|
CC[C@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(CC)ncnc1C1CC1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)C(C)C)c2=O)-c2c(ncnc2C2CC2)C2CC2)nc1 |r|
CC[C@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(OC)ncnc1C1CC1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C(C)C)c2=O)-c2c(OC)ncnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C3CCCC3)c2=O)-c2c(OC)ncnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C(C)C)c2=O)-c2c(C)ncnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)C(C)C)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C3CCCC3)c2=O)-c2c(ncnc2C2CC2)C2CC2)nc1
CCC(C)n1c2nc(ncc2nc(NCc2ccc(cc2)S(C)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C(C)C)c2=O)-c2c(ncnc2C2CC2)C2CC2)nc1
CCC(CC)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(ncnc1C1CC1)C1CC1
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(OC)ncnc1C1CC1 |r|
CCc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(=O)(=O)CC)c(=O)n([C@H](C)C(C)C)c2n1 |r|
CC[C@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(ncnc1C1CC1)C1CC1 |r|
CC[C@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(C)ncnc1C1CC1 |r|
CCc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(=O)(=O)CC)c(=O)n(C(C)C)c2n1
CCC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(OC)ncnc1C1CC1 |r|
CCC(C)n1c2nc(ncc2nc(NCc2ccc(cc2)S(C)(=O)=O)c1=O)-c1c(ncnc1C1CC1)C1CC1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H](C)C(C)C)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H](C)C(C)C)c2=O)-c2c(ncnc2C2CC2)C2CC2)nc1 |r|
CCC(C)n1c2nc(ncc2nc(NCc2ccc(cc2)S(C)(=O)=O)c1=O)-c1c(OC)ncnc1C1CC1
CCC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(C)ncnc1C1CC1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(c2=O)C2(C)CC2)-c2c(ncnc2C2CC2)C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)COC)c2=O)-c2c(ncnc2C2CC2)C2CC2)nc1 |r|
CCc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(=O)(=O)CC)c(=O)n([C@@H](C)COC)c2n1 |r|
CCC[C@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(C)ncnc1C1CC1 |r|
CCc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(=O)(=O)CC)c(=O)n(c2n1)C1(C)CC1
CCC[C@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(OC)ncnc1C1CC1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)COC)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C(C)C)c2=O)-c2c(OC)ncnc2C2CC2)cn1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(c2=O)C2(C)CC2(F)F)-c2c(OC)ncnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(c2=O)C2(C)CC2)-c2c(OC)ncnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(c2=O)C2(C)CC2)-c2c(ncnc2C2CC2)C2CC2)cc1
CCc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(=O)(=O)CC)c(=O)n([C@H](C)COC)c2n1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(CC3CCCO3)c2=O)-c2c(ncnc2C2CC2)C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H](C)COC)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(c2=O)C2(C)CC2)-c2c(C)ncnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C3CC3)c2=O)-c2c(OC)ncnc2C2CC2)cc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(CC3CCCO3)c2=O)-c2c(OC)ncnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C3CC3)c2=O)-c2c(C)ncnc2C2CC2)cc1
CS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C3CC3)c2=O)-c2c(ncnc2C2CC2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C3CC3)c2=O)-c2c(ncnc2C2CC2)C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(-c3ccccc3)c2=O)-c2c(C)ncnc2C2CC2)nc1
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cc3)S(C)(=N)=O)c(=O)n(C(C)C)c2n1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(c2=O)C2(CC2)C#N)-c2c(OC)ncnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C3CC3)c2=O)-c2c(ncnc2C2CC2)C2CC2)cn1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C3CCC3)c2=O)-c2c(OC)ncnc2C2CC2)nc1
CCS(=O)(=O)c1cnc(CNc2nc3cnc(nc3n([C@H](C)C(C)C)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C3CCC3)c2=O)-c2c(C)ncnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H](C)COC)c2=O)-c2c(ncnc2C2CC2)C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(c2=O)C2(C)CC2)-c2c(C)ncnc2C2CC2)cc1
CCc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cc3)S(=O)(=O)CC)c(=O)n(c2n1)C1(C)CC1
CC[C@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(C)ncnc1C(F)(F)F |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H](C)C(F)(F)F)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H](C)C(F)(F)F)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)C(F)(F)F)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)C(F)(F)F)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(c2=O)C2(C)CC2)-c2c(OC)ncnc2C2CC2)cc1
CCC1(CC1)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(C)ncnc1C1CC1
CCS(=O)(=O)c1cnc(CNc2nc3cnc(nc3n([C@@H](C)C(C)C)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)C(C)C)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H](C)C(C)C)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1cnc(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1cnc(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r|
CCc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(=O)(=O)CC)c(=O)n([C@@H](C)C3CC3)c2n1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(ncnc2C2CC2)C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H](C)C3CC3)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)N1CCC(CNc2nc3cnc(nc3n([C@H](C)C3CC3)c2=O)-c2c(OC)ncnc2C2CC2)CC1 |r|
CCS(=O)(=O)c1cnc(CNc2nc3cnc(nc3n([C@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1cnc(CNc2nc3cnc(nc3n([C@H](C)C3CC3)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1cnc(CNc2nc3cnc(nc3n(C3CCCC3)c2=O)-c2c(C)ncnc2C2CC2)nc1
CCS(=O)(=O)c1cnc(CNc2nc3cnc(nc3n(C3CCCC3)c2=O)-c2c(OC)ncnc2C2CC2)nc1
CCS(=O)(=O)c1cnc(CNc2nc3cnc(nc3n(C3CCC3)c2=O)-c2c(C)ncnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(cc1)[C@@H](C)Nc1nc2cnc(nc2n(C2CCC2)c1=O)-c1c(C)ncnc1C1CC1 |r|
CCS(=O)(=O)c1ccc(cc1)[C@H](C)Nc1nc2cnc(nc2n(C2CCC2)c1=O)-c1c(C)ncnc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(C)ncnc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(CC)ncnc1C1CC1 |r|
CC[C@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(ncnc1C1CC1)C(C)C |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(ncnc1C1CC1)C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1cncnc1C(C)C |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H]3CCOC3)c2=O)-c2c(ncnc2C2CC2)C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H]3CCOC3)c2=O)-c2c(ncnc2C2CC2)C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(CC3CC3)c2=O)-c2c(OC)ncnc2C2CC2)nc1
COCCS(=O)(=O)N1CCC(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)CC1 |r|
CC[C@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(C)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(nc2)S(C)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
CC[C@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(C)(=O)=O)c1=O)-c1c(OC)ncnc1C1CC1 |r|
CC[C@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(N)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
CC[C@H](C)n1c2nc(ncc2nc(NCc2ccc(nc2)S(C)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
CC[C@H](C)n1c2nc(ncc2nc(NCc2ccc(nc2)S(=O)(=O)CC)c1=O)-c1c(C)ncnc1C1CC1 |r|
CC[C@@H](n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(C)ncnc1C1CC1)C(F)(F)F |r|
CCS(=O)(=O)c1cnc(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)s1 |r|
CCn1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(C)ncnc1C1CC1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(CC(C)(C)F)c2=O)-c2c(C)ncnc2C2CC2)nc1
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(C)(=O)=O)c(=O)n(CC(C)(C)F)c2n1
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(nc3)S(C)(=O)=O)c(=O)n(CC(C)C)c2n1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H]3CCC[C@H]3C#N)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H]3CCC[C@@H]3C#N)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H]3CC3C(F)(F)F)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r,@@:23|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H]3CCC[C@H]3C#N)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H]3CCC[C@@H]3C#N)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H](C3CC3)C(F)(F)F)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1sc(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)nc1C |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(CC3CCC3)c2=O)-c2c(C)ncnc2C2CC2)cc1
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(N)(=O)=O)c(=O)n(CC3CCC3)c2n1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(CC3CCC3)c2=O)-c2c(OC)ncnc2C2CC2)nc1
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(C)(=O)=O)c(=O)n(CC3CCC3)c2n1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C3CCCC3=O)c2=O)-c2c(C)ncnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C3CCCC3=O)c2=O)-c2c(OC)ncnc2C2CC2)nc1
CC[C@H](C)n1c2nc(ncc2nc(NCc2ccc(nc2)S(=O)(=O)CC)c1=O)-c1c(OC)ncnc1C1CC1 |r|
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(N)(=O)=O)c(=O)n(C(C)C)c2n1 |@:32|
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(nc3)S(C)(=O)=O)c(=O)n([C@@H](C)C3CC3)c2n1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(OC)ncnc2C2CC2)cn1 |r|
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(C)(=O)=O)c(=O)n([C@@H](C)C3CC3)c2n1 |r|
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(N)(=O)=O)c(=O)n([C@@H](C)C3CC3)c2n1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(CC3(C)CC3)c2=O)-c2c(C)ncnc2C2CC2)nc1
C[C@@H](C1CC1)n1c2nc(ncc2nc(NCc2ccc(nc2)S(C)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(N)(=O)=O)c1=O)-c1c(C)nc(N)nc1C1CC1 |r|
CCS(=O)(=O)N5CCC(CNc4nc3cnc(c1c(C)ncnc1C2CC2)nc3n(C(C)C)c4=O)CC5
CCS(=O)(=O)N5CCC(CNc4nc3cnc(c1c(OC)ncnc1C2CC2)nc3n(C(C)C)c4=O)CC5
CC[C@H](C)n1c2nc(ncc2nc(NCc2ccc(cc2)S(N)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
COc1cc(ccc1CNc1nc2cnc(nc2n([C@@H](C)C2CC2)c1=O)-c1c(C)ncnc1C1CC1)C#N |r|
CNS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)cc1 |r|
C[C@@H](C1CC1)n1c2nc(ncc2nc(NCc2ccc(cn2)S(C)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
C[C@@H](C1CC1)n1c2nc(ncc2nc(NCc2ccc(cc2)S(C)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
CCS(=O)(=O)N1CCC(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)CC1 |r|
CCS(=O)(=O)c5ccc(CNc4nc3cnc(c1c(C)ncnc1C2CC2)nc3n(C(C)(C)C)c4=O)nc5
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C(C)C)c2=O)-c2cnc(N)nc2C(C)C)nc1
CCS(=O)(=O)c4ccc(CNc3nc2cnc(c1c(OC)ncnc1OC)nc2n(C(C)C)c3=O)nc4
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C(C)C)c2=O)-c2c(C)nc(N)nc2C2CC2)nc1
CCS(=O)(=O)c5ccc(CNc4nc3cnc(c1c(OC)ncnc1C2CC2)nc3n(C(C)C)c4=O)cc5
C[C@@H](C1CC1)n1c2nc(ncc2nc(NCc2ccc(cc2)S(=O)(=O)CC#N)c1=O)-c1c(C)ncnc1C1CC1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C(C)C)c2=O)-c2cncnc2C(C)C)nc1
COc2ncnc(C1CC1)c2c5ncc4nc(NCc3ccc(S(=O)(=O)CC#N)cc3)c(=O)n(C(C)C)c4n5
CCS(=O)(=O)N1CC[C@H](CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)C1 |r|
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(C)(=O)=O)c(=O)n(C(C)C)c2n1
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cc3)S(C)(=O)=O)c(=O)n(C(C)C)c2n1
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cc3)S(N)(=O)=O)c(=O)n(C(C)C)c2n1
CCS(=O)(=O)N1CC2(CC(CNc3nc4cnc(nc4n([C@@H](C)C4CC4)c3=O)-c3c(OC)ncnc3C3CC3)C2)C1 |r|
CCS(=O)(=O)N1CC2(CC(CNc3nc4cnc(nc4n([C@@H](C)C4CC4)c3=O)-c3c(C)ncnc3C3CC3)C2)C1 |r|
CCS(=O)(=O)c5ccc(CNc4nc3cnc(c1c(OC)ncnc1C2CC2)nc3n(CC(C)C)c4=O)cn5
CNS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C(C)C)c2=O)-c2c(OC)ncnc2C2CC2)nc1
CCS(=O)(=O)c5ccc(CNc4nc3cnc(c1c(C)ncnc1C2CC2)nc3n(CC(C)C)c4=O)cn5
CCS(=O)(=O)c6ccc(CNc5nc3cnc(c1c(OC)ncnc1C2CC2)nc3n([C@@H](C)C4CC4)c5=O)cn6
CCS(=O)(=O)c6ccc(CNc5nc3cnc(c1c(C)ncnc1C2CC2)nc3n([C@@H](C)C4CC4)c5=O)cn6
Cc2ncnc(C1CC1)c2c7ncc6nc(NCC4CCN(S(=O)(=O)C3CC3)CC4)c(=O)n([C@@H](C)C5CC5)c6n7
Cc2ncnc(C1CC1)c2c6ncc5nc(NCc3ccc(S(C)(=N)=O)cc3)c(=O)n([C@@H](C)C4CC4)c5n6
CCc2ncnc(C1CC1)c2c5ncc4nc(NCc3ccc(S(=O)(=O)CC)cn3)c(=O)n([C@@H](C#N)C(C)C)c4n5
CCS(=O)(=O)c5ccc(CNc4nc3cnc(c1c(C)ncnc1C2CC2)nc3n([C@@H](C#N)C(C)C)c4=O)nc5
CCS(=O)(=O)N7C[C@@H]6C(CNc5nc3cnc(c1c(C)ncnc1C2CC2)nc3n([C@@H](C)C4CC4)c5=O)[C@@H]6C7
Cc2ncnc(C1CC1)c2c6ncc5nc(NCc3ccc(NS(C)(=O)=O)cc3)c(=O)n([C@@H](C)C4CC4)c5n6
C[C@@H](C1CC1)n1c2nc(ncc2nc(NCC2CCN(CC2)S(=O)(=O)CC#N)c1=O)-c1c(C)ncnc1C1CC1 |r|
C[C@@H](C1CC1)n1c2nc(ncc2nc(NCC2CCN(CC2)C(C)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
CCc2ncnc(C1CC1)c2c5ncc4nc(NCc3ccc(S(=O)(=O)CC)cn3)c(=O)n([C@H](C#N)C(C)C)c4n5
CCS(=O)(=O)c5ccc(CNc4nc3cnc(c1c(C)ncnc1C2CC2)nc3n([C@H](C#N)C(C)C)c4=O)nc5
COCCS(=O)(=O)N1CCC(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(OC)ncnc2C2CC2)CC1 |r|
CCS(=O)(=O)c5ccc(CNc4nc3cnc(c1c(OC(C)C)ncnc1C2CC2)nc3n(C(C)C)c4=O)nc5
Cc2ncnc(C1CC1)c2c5ncc4nc(NCc3ccc(S(=O)(=O)CC#N)cc3)c(=O)n(C(C)C)c4n5
CCCc1ncnc(C)c1c4ncc3nc(NCc2ccc(S(=O)(=O)CC)cn2)c(=O)n(C(C)C)c3n4
CCc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(=O)(=O)CC)c(=O)n(CC)c2n1
CCS(=O)(=O)c7ccc(CNc6nc4cnc(c2c(C1CC1)ncnc2C3CC3)nc4n([C@H]5CCOC5)c6=O)cc7
CCc2ncnc(C1CC1)c2c6ncc5nc(NCc3ccc(S(=O)(=O)CC)cc3)c(=O)n([C@H]4CCOC4)c5n6
CCS(=O)(=O)c6ccc(CNc5nc3cnc(c1c(OC)ncnc1C2CC2)nc3n([C@H]4CCOC4)c5=O)cc6
CCS(=O)(=O)c5ccc(CNc4nc3cnc(c1c(C)ncnc1C2CC2)nc3n([C@@H](C)C(F)(F)F)c4=O)cc5
CCS(=O)(=O)c4ccc(CNc3nc2cnc(c1c(C)ncnc1C(C)C)nc2n(C(C)C)c3=O)nc4
CCS(=O)(=O)c5ccc(CNc4nc3cnc(c1c(C)ncnc1C2CCC2)nc3n(C(C)C)c4=O)nc5
C[C@H](n1c2nc(ncc2nc(NCc2ccc(cn2)S(C)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1)C(F)(F)F |r|
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(C)(=O)=O)c(=O)n([C@@H](C)C(F)(F)F)c2n1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H](C)C3CCC3)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ncc(cn2)S(=O)(=O)CC)c1=O)-c1c(C)ncnc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ncc(cn2)S(=O)(=O)CC)c1=O)-c1c(OC)ncnc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ncc(cn2)S(=O)(=O)CC)c1=O)-c1c(CC)ncnc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ncc(cn2)S(=O)(=O)CC)c1=O)-c1c(ncnc1C1CC1)C1CC1 |r|
CCS(=O)(=O)c1cnc(CNc2nc3cnc(nc3n([C@@H](C)C(F)(F)F)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1cnc(CNc2nc3cnc(nc3n([C@@H](C)C(F)(F)F)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cc2)S(C)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cc2)S(C)(=O)=O)c1=O)-c1c(OC)ncnc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cc2)S(C)(=O)=O)c1=O)-c1c(CC)ncnc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cc2)S(C)(=O)=O)c1=O)-c1c(ncnc1C1CC1)C1CC1 |r|
C[C@H](C1CCC1)n1c2nc(ncc2nc(NCc2ccc(cc2)S(C)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
C[C@H](C1CCC1)n1c2nc(ncc2nc(NCc2ccc(cc2)S(N)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cc2)S(N)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cc2)S(N)(=O)=O)c1=O)-c1c(OC)ncnc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(nc2)S(=O)(=O)CC)c1=O)-c1c(C)ncnc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(nc2)S(=O)(=O)CC)c1=O)-c1c(OC)ncnc1C1CC1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)C3CCC3)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
C[C@@H](C1CC1)n1c2nc(ncc2nc(NCc2ccc(cc2)C(O)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
CCCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)N[C@H]1C[C@H](CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)C1 |r,wU:20.21,8.8,wD:6.5,(5.61,-7.37,;6.94,-6.6,;6.94,-5.06,;8.28,-5.83,;5.61,-5.83,;6.94,-3.52,;5.61,-2.75,;5.21,-1.26,;3.72,-1.66,;2.39,-.89,;2.39,.65,;1.06,1.42,;-.28,.65,;-1.61,1.42,;-2.94,.65,;-4.28,1.42,;-4.28,2.96,;-2.94,3.73,;-1.61,2.96,;-.28,3.73,;-.28,5.27,;-1.61,6.04,;1.06,6.04,;2.6,6.04,;1.83,7.37,;1.06,2.96,;2.39,3.73,;-5.61,3.73,;-5.61,5.27,;-4.28,6.04,;-6.94,6.04,;-8.28,5.27,;-8.28,3.73,;-6.94,2.96,;-6.94,1.42,;-7.71,.08,;-6.17,.08,;4.12,-3.15,)|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc3c(CCS3(=O)=O)c2)c1=O)-c1c(C)ncnc1C1CC1 |r|
C[C@@H](C1CC1)n1c2nc(ncc2nc(NCc2ccc(cc2)C(N)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cc3)S(N)(=O)=O)c(=O)n([C@@H](C)C3CC3)c2n1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(N[C@@H](C)c2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(OC)ncnc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(N[C@H](C)c2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(OC)ncnc1C1CC1 |r|
CNS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r|
COCCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)cc1 |r|
CCc2ncnc(C1CC1)c2c6ncc5nc(NCc3ccc(S(C)(=N)=O)cc3)c(=O)n([C@@H](C)C4CC4)c5n6
CCS(=O)(=O)N1CC[C@@H](CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)C1 |r|
C[C@@H](C1CC1)n1c2nc(ncc2nc(NCc2ccc3c(CCS3(=O)=O)c2)c1=O)-c1c(C)ncnc1C1CC1 |r|
CCS(=O)(=O)c1cnc(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)cn1 |r|
C[C@@H](C1CC1)n1c2nc(ncc2nc(NCc2ccc(cn2)S(N)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
COCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)cc1 |r|
COC(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)cc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(C)nc(N)nc2C2CC2)nc1 |r|
CCS(=O)(=O)c1cnc(CNc2nc3cnc(nc3n([C@@H](C)C3CCC3)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1cnc(CNc2nc3cnc(nc3n([C@H](C)C3CCC3)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
[H][C@]12CC[C@]([H])(C1)[C@@H](C2)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(C)ncnc1C1CC1 |r,TLB:9:7:3.2:6|
[H][C@]12CC[C@]([H])(C1)[C@@H](C2)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(OC)ncnc1C1CC1 |r,TLB:9:7:3.2:6|
[H][C@@]12CC[C@@]([H])(O1)[C@@H](C2)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(OC)ncnc1C1CC1 |r,THB:9:7:2.3:6|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(nc2)S(=O)(=O)CC)c1=O)-c1c(CC)ncnc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(nc2)S(=O)(=O)CC)c1=O)-c1c(ncnc1C1CC1)C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(C)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(C)(=O)=O)c1=O)-c1c(OC)ncnc1C1CC1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H]3CCC[C@@H]3OC)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H]3CCC[C@@H]3OC)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r|
CO[C@H]1CCC[C@@H]1n1c2nc(ncc2nc(NCc2ccc(cc2)S(C)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
CO[C@H]1CCC[C@@H]1n1c2nc(ncc2nc(NCc2ccc(cc2)S(C)(=O)=O)c1=O)-c1c(OC)ncnc1C1CC1 |r|
CCc1nc(N)nc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(=O)(=O)CC)c(=O)n(C(C)C)c2n1
C[C@@H](C1CCC1)n1c2nc(ncc2nc(NCc2ccc(cc2)S(C)(=N)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
CCS(=O)(=O)c6ccc(CNc5nc3cnc(c1c(C)nc(N)nc1C2CC2)nc3n([C@H](C)C4CCC4)c5=O)nc6
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(N)(=O)=O)c(=O)n(CC3CC3)c2n1
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(N)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(N)(=O)=O)c1=O)-c1c(OC)ncnc1C1CC1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(CC3CC3)c2=O)-c2c(C)ncnc2C2CC2)nc1
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(N)(=O)=O)c(=O)n(C3CCC3)c2n1
CNS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C3CCC3)c2=O)-c2c(OC)ncnc2C2CC2)nc1
CCS(=O)(=O)c1cnc(CNc2nc3cnc(nc3n(C3CCC3)c2=O)-c2c(OC)ncnc2C2CC2)nc1
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(C)(=O)=O)c(=O)n(C3CCC3)c2n1
Cc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(C)(=O)=O)c(=O)n(C3CCC3)c2n1
CNS(=O)(=O)c6ccc(CNc5nc3cnc(c1c(C)ncnc1C2CC2)nc3n(C4CCC4)c5=O)nc6
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cc2)S(C)(=O)=O)c1=O)-c1c(C)nc(N)nc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cc2)S(N)(=O)=O)c1=O)-c1c(C)nc(N)nc1C1CC1 |r|
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(C)(=O)=O)c(=O)n(CC3CC3)c2n1
Cc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(C)(=O)=O)c(=O)n(CC3CC3)c2n1
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(=O)(=O)C3CC3)c(=O)n([C@@H](C)C3CC3)c2n1 |r|
C[C@@H](C1CC1)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)C2CC2)c1=O)-c1c(C)ncnc1C1CC1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C3CCC3)c2=O)-c2c(C)ncnc2C2CC2)cc1
CCc1nc(N)nc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(=O)(=O)C3CC3)c(=O)n([C@@H](C)C3CC3)c2n1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(CC(C)C)c2=O)-c2c(C)ncnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(CC(C)C)c2=O)-c2c(OC)ncnc2C2CC2)nc1
CC(C)Cn1c2nc(ncc2nc(NCc2ccc(cn2)S(N)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(N)(=O)=O)c(=O)n(CC(C)C)c2n1
CCS(=O)(=O)c1csc(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)n1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(C)nc(N)nc1C1CC1 |r|
CC(C)Cn1c2nc(ncc2nc(NCc2ccc(cn2)S(C)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1
COc1ncnc(C2CC2)c1-c1ncc2nc(NCc3ccc(cn3)S(C)(=O)=O)c(=O)n(CC(C)C)c2n1
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(nc2)S(=O)(=O)CC)c1=O)-c1c(C)nc(N)nc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cn2)S(C)(=O)=O)c1=O)-c1c(C)nc(N)nc1C1CC1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H]3C[C@@H](C3)OC)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r,wU:20.20,22.25,(10,-5.04,;8.67,-4.27,;7.34,-5.04,;6.57,-6.38,;8.11,-6.38,;6,-4.27,;4.67,-5.04,;3.33,-4.27,;3.33,-2.73,;2,-1.96,;.67,-2.73,;-.67,-1.96,;-2,-2.73,;-3.33,-1.96,;-4.67,-2.73,;-6,-1.96,;-6,-.42,;-4.67,.35,;-3.33,-.42,;-2,.35,;-2,1.89,;-.91,2.98,;-2,4.07,;-3.09,2.98,;-2,5.61,;-.67,6.38,;-.67,-.42,;.67,.35,;-7.34,.35,;-7.34,1.89,;-6,2.66,;-6,4.2,;-8.67,2.66,;-10,1.89,;-10,.35,;-8.67,-.42,;-8.67,-1.96,;-9.44,-3.3,;-7.9,-3.3,;4.67,-1.96,;6,-2.73,)|
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@H]3C[C@@H](C3)OC)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r,wU:20.20,wD:22.25,(10,-5.04,;8.67,-4.27,;7.34,-5.04,;6.57,-6.38,;8.11,-6.38,;6,-4.27,;4.67,-5.04,;3.33,-4.27,;3.33,-2.73,;2,-1.96,;.67,-2.73,;-.67,-1.96,;-2,-2.73,;-3.33,-1.96,;-4.67,-2.73,;-6,-1.96,;-6,-.42,;-4.67,.35,;-3.33,-.42,;-2,.35,;-2,1.89,;-3.09,2.98,;-2,4.07,;-.91,2.98,;-2,5.61,;-.67,6.38,;-.67,-.42,;.67,.35,;-7.34,.35,;-7.34,1.89,;-6,2.66,;-6,4.2,;-8.67,2.66,;-10,1.89,;-10,.35,;-8.67,-.42,;-8.67,-1.96,;-9.44,-3.3,;-7.9,-3.3,;4.67,-1.96,;6,-2.73,)|
C[C@@H](C1CC1)n1c2nc(ncc2nc(NCC2CC3(C2)CN(C3)C(=O)OC(C)(C)C)c1=O)-c1c(C)ncnc1C1CC1 |r|
CC[C@@H](C)n1c2nc(ncc2nc(NCc2ccc(cc2)S(=O)(=O)N2CCOCC2)c1=O)-c1c(OC)ncnc1C1CC1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cc3CC(C)OC4(CCN(CC4)C(C)c4cnc(nc4)C(F)(F)F)c3s2)nc1 |$;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;$|
CCS(=O)(=O)c1ccc(CNC(=O)c2cc3C[C@H](C)OC4(CCN(CC4)[C@@H](C)c4cnc(nc4)C(F)(F)F)c3s2)nc1 |r,$;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;$|
CCS(=O)(=O)c1ccc(CNC(=O)c2cc3C[C@H](C)OC4(CCN(CC4)[C@H](C)c4cnc(nc4)C(F)(F)F)c3s2)nc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cc3C[C@@H](C)OC4(CCN(CC4)C(C)c4cnc(nc4)C(F)(F)F)c3s2)nc1 |r|
Fc1cccc(Cl)c1C(=O)Nc1cnc2cnn(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)n1ncc2cnc(NC(=O)c3c(F)cccc3Cl)cc12
Fc1cccc(Cl)c1C(=O)Nc1cnc2cnn(c2c1)S(=O)(=O)c1cccc(c1)C#N
Fc1ccc(cc1)S(=O)(=O)n1ncc2cnc(NC(=O)c3c(F)cccc3F)cc12
Fc1ccc(cc1)S(=O)(=O)n1ncc2cnc(NC(=O)c3c(Cl)cccc3Cl)cc12
Fc1ccc(cc1)S(=O)(=O)n1ncc2cnc(NC(=O)c3c(Cl)cccc3C(F)(F)F)cc12
Fc1cccc(Cl)c1C(=O)Nc1cc2n(ncc2cn1)S(=O)(=O)c1cccc(Cl)c1
FC(F)Oc1cccc(c1)S(=O)(=O)n1ncc2cnc(NC(=O)c3c(F)cccc3Cl)cc12
CC(C)(C)c1cccc(c1)S(=O)(=O)n1ncc2cnc(NC(=O)c3c(F)cccc3Cl)cc12
Fc1cccc(Cl)c1C(=O)Nc1cc2n(ncc2cn1)S(=O)(=O)c1cccc(c1)C(F)(F)F
Cc1nn(cc1S(=O)(=O)n1ncc2cnc(NC(=O)c3c(F)cccc3Cl)cc12)C(F)F
CC1COc2ncc(NC(=O)c3c(F)cccc3Cl)cc2N1S(=O)(=O)c1ccc(F)cc1
Fc1ccc(cc1)S(=O)(=O)N1CCOc2ncc(NC(=O)c3c(F)cccc3Cl)cc12
C[C@H]1CN(c2cc(NC(=O)c3c(F)cccc3Cl)cnc2O1)S(=O)(=O)c1cccc(C)c1 |r|
CCc1cccc(c1)S(=O)(=O)N1C[C@H](C)Oc2ncc(NC(=O)c3c(F)cccc3Cl)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)c3c(F)cccc3Cl)cnc2O1)S(=O)(=O)c1cccc(C)c1 |r|
C[C@H](C(=O)Nc1cnc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1cccc(C)c1)c1ccccc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2O1)S(=O)(=O)c1cccc(c1)C1CC1
CC1COc2ncc(NC(=O)c3c(Cl)cccc3C(F)(F)F)cc2N1S(=O)(=O)c1ccc(F)cc1
CC1COc2ncc(NC(=O)c3c(F)cccc3Cl)cc2N1S(=O)(=O)c1cccc(c1)C#N
Fc1cccc(Cl)c1C(=O)Nc1cnc2OCCN(c2c1)S(=O)(=O)c1cccc(c1)C#N
Fc1cccc(Cl)c1C(=O)Nc1cnc2OCCN(c2c1)S(=O)(=O)c1ccc(Cl)cc1
Fc1ccc(cc1F)S(=O)(=O)N1CCOc2ncc(NC(=O)c3c(F)cccc3Cl)cc12
C[C@H]1CN(c2cc(NC(=O)c3c(F)cccc3C(F)(F)F)cnc2O1)S(=O)(=O)c1cccc(C)c1 |r|
C[C@H]1CN(c2cc(NC(=O)c3c(F)cccc3Cl)cnc2O1)S(=O)(=O)c1cccc(c1)C#N |r|
C[C@H]1CN(c2cc(NC(=O)c3c(F)cccc3Cl)cnc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@H]1CN(c2cc(NC(=O)c3c(F)cccc3Cl)cnc2O1)S(=O)(=O)c1cccc(c1)C1CC1 |r|
C[C@H](C(=O)Nc1cnc2O[C@@H](C)CN(c2c1)S(=O)(=O)c1cccc(C)c1)c1ccccc1 |r|
C[C@H](C(=O)Nc1cnc2O[C@@H](C)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)c1ccccc1 |r|
CC(C(=O)Nc1cnc2O[C@@H](C)CN(c2c1)S(=O)(=O)c1cccc(C)c1)C(F)(F)F |r|
CC(C(=O)Nc1cnc2O[C@@H](C)CN(c2c1)S(=O)(=O)c1cccc(C)c1)c1ccccc1C |r|
CC(C(=O)Nc1cnc2O[C@@H](C)CN(c2c1)S(=O)(=O)c1cccc(C)c1)c1ccc(F)cc1 |r|
CCC(C)C(=O)Nc1cnc2O[C@@H](C)CN(c2c1)S(=O)(=O)c1cccc(C)c1 |r|
CC(C(=O)Nc1cnc2O[C@@H](C)CN(c2c1)S(=O)(=O)c1cccc(C)c1)c1ccc(Cl)cc1 |r|
C[C@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2O1)S(=O)(=O)c1cccc(c1)C1CC1 |r|
Fc1ccc(cc1)S(=O)(=O)N1CCCc2ncc(NC(=O)c3c(F)cccc3F)cc12
Cc1cccc(c1)S(=O)(=O)N1CCCc2ncc(NC(=O)c3c(F)cccc3Cl)cc12
C[C@H](C(=O)Nc1cnc2CCCN(c2c1)S(=O)(=O)c1cccc(C)c1)c1ccccc1 |r|
Cc1cccc(c1)S(=O)(=O)N1C[C@@H](Cc2ncc(NC(=O)c3c(Cl)cccc3Cl)cc12)NC(=O)OC(C)(C)C |r|
Cc1cccc(c1)S(=O)(=O)N1C[C@H](N)Cc2ncc(NC(=O)c3c(Cl)cccc3Cl)cc12 |r|
CC(=O)N[C@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(C)c1 |r|
COC(=O)N[C@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(C)c1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2O1)S(=O)(=O)c1cccc(c1)C1CC1 |r|
CC(C)(C)OC(=O)N[C@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(Cl)c1 |r|
CC(=O)NC1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(Cl)c1
CC(C)OC(=O)N[C@@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CN(C)C(=O)NC1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(c1)C(F)(F)F
Cc1nn(cc1S(=O)(=O)N1C[C@H](Cc2ncc(NC(=O)c3c(F)cccc3Cl)cc12)NC(=O)C(F)(F)F)C(F)F |r|
Cc1nn(cc1S(=O)(=O)N1C[C@@H](Cc2ncc(NC(=O)c3c(F)cccc3Cl)cc12)NC(=O)C(F)(F)F)C(F)F |r|
C[C@H](N)C(=O)N[C@@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
C[C@H](O)C(=O)N[C@@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
N[C@@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)N[C@@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
C[C@H](N)C(=O)N[C@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
C[C@H](O)C(=O)N[C@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)OC(=O)N[C@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)N[C@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
N[C@H](CO)C(=O)NC1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)OC(=O)N[C@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)OC(=O)N[C@@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1ccc(F)cc1 |r|
CCOC(=O)N[C@@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CCOC(=O)N[C@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)OC(=O)N[C@@H]1CN(c2cc(NC(=O)c3c(F)cccc3Cl)cnc2C1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(C)OC(=O)N[C@H]1CN(c2cc(NC(=O)c3c(F)cccc3Cl)cnc2C1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
C[C@H](O)C(=O)N[C@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(C)c1 |r|
CC(=O)NC1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(c1)C1CC1
CC(C)(C)OC(=O)NC1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(c1)C1CC1
NC1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(c1)C1CC1
Cc1cccc(c1)S(=O)(=O)N1CC(N)COc2ncc(NC(=O)C(F)(F)F)cc12
Cc1cccc(c1)S(=O)(=O)N1CC(N)COc2ncc(NC(=O)c3c(Cl)cccc3Cl)cc12
CC(=O)NC1COc2ncc(NC(=O)c3c(Cl)cccc3Cl)cc2N(C1)S(=O)(=O)c1cccc(C)c1
CN(C)C1COc2ncc(NC(=O)c3c(Cl)cccc3Cl)cc2N(C1)S(=O)(=O)c1cccc(C)c1
CCNC1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(C)c1
CCN(CC)[C@@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(C)c1 |r|
CCN(CC)[C@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2C1)S(=O)(=O)c1cccc(C)c1 |r|
Clc1cccc(c1)S(=O)(=O)N1C[C@H](CN2CCCC2=O)Oc2ccc(NC(=O)c3c(Cl)cccc3Cl)cc12 |r|
FC(F)(F)c1cccc(c1)S(=O)(=O)N1C[C@H](Cc2ncc(NC(=O)c3c(Cl)cccc3Cl)cc12)N1CCCC1=O |r|
FC(F)(F)c1cccc(c1)S(=O)(=O)N1C[C@@H](Cc2ncc(NC(=O)c3c(Cl)cccc3Cl)cc12)N1CCCC1=O |r|
Fc1cccc(Cl)c1C(=O)Nc1cnc2C[C@@H](CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)N1CCCC1=O |r|
Fc1cccc(Cl)c1C(=O)Nc1cnc2C[C@H](CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)N1CCCC1=O |r|
Clc1cccc(c1)S(=O)(=O)N1C[C@H](CN2C(=O)COC2=O)Oc2ncc(NC(=O)c3c(Cl)cccc3Cl)cc12 |r|
CN1CC(=O)N(C[C@H]2CN(c3cc(NC(=O)c4c(Cl)cccc4Cl)cnc3O2)S(=O)(=O)c2cccc(Cl)c2)C1=O |r|
CN1CCN(C[C@H]2CN(c3cc(NC(=O)c4c(Cl)cccc4Cl)cnc3O2)S(=O)(=O)c2cccc(Cl)c2)CC1=O |r|
CN(C)C[C@H]1CN(c2cc(NC(=O)c3c(Cl)cccc3Cl)cnc2O1)S(=O)(=O)c1cccc(Cl)c1 |r|
O[C@@H]1CCN(C[C@H]2CN(c3cc(NC(=O)c4c(Cl)cccc4Cl)cnc3O2)S(=O)(=O)c2cccc(Cl)c2)C1 |r|
Clc1cccc(c1)S(=O)(=O)N1C[C@H](CN2CCOCC2)Oc2ncc(NC(=O)c3c(Cl)cccc3Cl)cc12 |r|
CN1CCN(C[C@H]2CN(c3cc(NC(=O)c4c(Cl)cccc4Cl)cnc3O2)S(=O)(=O)c2cccc(Cl)c2)CC1 |r|
C[C@H](C(=O)Nc1cnc2C[C@@H](CO)CN(c2c1)S(=O)(=O)c1cn(nc1C)C(F)F)C(C)(C)C |r|
Cc1cccc(c1)S(=O)(=O)N1CC(CO)Cc2ncc(NC(=O)c3c(Cl)cccc3Cl)cc12
C[C@H](C(=O)Nc1cnc2C[C@@H](CN3CC[C@@H](O)C3)CN(c2c1)S(=O)(=O)c1cn(nc1C)C(F)F)C(C)(C)C |r|
C[C@H](C(=O)Nc1cnc2C[C@H](CN3CC[C@@H](O)C3)CN(c2c1)S(=O)(=O)c1cn(nc1C)C(F)F)C(C)(C)C |r|
FC(F)(F)c1cccc(c1)S(=O)(=O)N1C[C@H](Cc2ncc(NC(=O)c3c(Cl)cccc3Cl)cc12)N1CCOC1=O |r|
CC1CCN(CC1)C(=O)c1nc(sc1-c1ccc(c2ccccc12)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O
CC(C)(O)CNC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F
C[C@H]1C[C@@H](F)CCN1C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(C)(F)C2)c(s1)-c1ccc(c(Cl)c1Cl)C(N)(C(F)(F)F)C(F)(F)F
CC(C)(O)CNC(=O)c1nc(C(=O)N2CC3CC2C3)c(s1)-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F |THB:11:13:16:18,(4.03,-8.43,;2.62,-7.8,;1.21,-7.18,;2,-9.21,;3.25,-6.4,;2.34,-5.15,;2.97,-3.74,;4.5,-3.58,;2.06,-2.5,;.52,-2.5,;.05,-1.03,;-1.42,-.56,;-2.56,-1.59,;-1.74,.95,;-.61,2,;-2.05,2.53,;-3.32,3.48,;-3.07,1.47,;-4.57,1.09,;1.29,-.13,;2.54,-1.03,;1.29,1.41,;-.04,2.18,;-.04,3.72,;1.29,4.49,;2.63,3.72,;3.96,4.49,;2.63,2.18,;3.96,1.41,;1.29,6.03,;2.83,6.03,;1.29,7.57,;1.29,9.11,;2.83,7.57,;-.25,7.57,;-.25,6.03,;-1.79,6.03,;-1.15,7.28,;-.25,4.49,)|
CCN(CC(F)(F)F)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O
CCCN(C)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O
CC(C)CN(C)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O
C[C@H]1CCCN1C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
CC(C)(O)CNC(=O)c1nc(C(=O)N2CC(C2)C(F)(F)F)c(s1)-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)CC2)c(s1)-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F
CC(C)N(C)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)(F)C2)c(s1)-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F
CN(C1CCC1)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O
CCN(CCOC)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O
CCN(C1CCC1)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O
C[C@@H]1CCCN1C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
CCN(CC)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O
CCN(CC)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)[N+]#[C-]
CCN(CC)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)C(N)=O
CCN(CC)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)N[C@H]1CC11CCOCC1 |r|
CCN(CC)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)N1C[C@@H](O)C[C@@H](O)C1 |r|
CCN(CC)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC1(O)COC1
CCN(CC)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NC[C@H](C)O |r|
CCN(CC)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NC[C@@H](C)O |r|
CCN(CC)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NC1COC1
CCN(CC)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC1(O)CC1
OC(c1ccc(-c2sc(nc2C(=O)N2C3CCC2CC3)C(=O)N2CCNC(=O)C2)c(Cl)c1Cl)(C(F)(F)F)C(F)(F)F
OC(c1ccc(-c2sc(nc2C(=O)N2C3CCC2CC3)C(=O)N2CC(=O)NC(=O)C2)c(Cl)c1Cl)(C(F)(F)F)C(F)(F)F
CCN(CC)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(N)=O
CCN(CC)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)N1CC(O)(C1)C(C)(C)O
OC(c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(=O)N2CC3(C2)CS(=O)(=O)C3)c(Cl)c1Cl)(C(F)(F)F)C(F)(F)F
OC(c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(=O)NC2CS(=O)(=O)C2)c(Cl)c1Cl)(C(F)(F)F)C(F)(F)F
CC(C)(O)CCNC(=O)c1nc(C(=O)N2CCC(F)CC2)c(s1)-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)CC2)c(s1)-c1cc(cc(c1)C(O)(C(F)(F)F)C(F)(F)F)C(C)(C)C
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)N1C[C@@H](O)C[C@@H](O)C1 |r|
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1ccc(cc1OC(F)(F)F)C(O)(C(F)(F)F)C(F)(F)F)C(=O)N1C[C@@H](O)C[C@@H](O)C1 |r|
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1ccc(cc1C(F)(F)F)C(O)(C(F)(F)F)C(F)(F)F)C(=O)N1C[C@@H](O)C[C@@H](O)C1 |r|
CC(C)Oc1cc(ccc1-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)N1C[C@@H](O)C[C@@H](O)C1)C(O)(C(F)(F)F)C(F)(F)F |r|
CCN(CC)C(=O)c1nc(sc1-c1ccc(cc1CC)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O
CCN(CC)C(=O)c1nc(sc1-c1ccc(cc1OC(F)(F)F)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O
CCN(CC)C(=O)c1nc(sc1-c1ccc(c(F)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O
O[C@H]1C[C@@H](O)CN(C1)C(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F |r|
O[C@H]1CN(C[C@H]1O)C(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F |r|
CC(C)(O)C(O)CNC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F
C[C@H]1CCCN1C(=O)c1nc(sc1-c1ccc(cc1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)N1CC(O)(C1)C(C)(C)O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1ccc(cc1C(F)(F)F)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1ccc(cc1C(F)(F)F)C(O)(C(F)(F)F)C(F)(F)F)C(=O)N1C[C@@H](O)C[C@@H](O)C1 |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1ccc(cc1C(F)(F)F)C(O)(C(F)(F)F)C(F)(F)F)C(=O)N1CC(O)(C1)C(C)(C)O |r|
CCN(CC)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(CC)C(F)(F)F)C(=O)NCC(C)(C)O
CCN(CC)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)[C@](O)(CC)C(F)(F)F)C(=O)NCC(C)(C)O |r|
CCN(CC(F)(F)F)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)N[C@H]1C[C@@H](C1)C(O)=O |r,wU:36.37,wD:38.42,(-.81,7.98,;-.18,6.58,;-1.09,5.33,;-2.62,5.49,;-3.53,4.25,;-5.06,4.41,;-2.9,2.84,;-1.99,4.09,;-.46,3.92,;-1.37,2.68,;1.07,3.76,;2.1,4.91,;3.51,4.28,;3.35,2.75,;1.84,2.43,;1.21,1.02,;2.12,-.22,;1.49,-1.63,;-.04,-1.79,;-.95,-.55,;-2.48,-.71,;-.32,.86,;-1.22,2.11,;-.67,-3.2,;-2.07,-2.57,;-1.29,-4.61,;-1.92,-6.01,;-2.7,-3.98,;.11,-5.23,;.74,-3.82,;2.15,-4.45,;1.06,-5.33,;1.37,-2.42,;4.84,5.05,;4.84,6.59,;6.17,4.28,;6.17,2.74,;7.26,1.65,;6.17,.56,;5.08,1.65,;6.17,-.98,;7.51,-1.75,;4.84,-1.75,)|
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)CC2)c(s1)-c1ccc(c2ncccc12)C(O)(C(F)(F)F)C(F)(F)F
CCN(CC)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)N1CCS(=N)(=O)CC1
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)N1CC2(C1)CS(=N)(=O)C2 |r|
CN=S1(=O)CC2(CN(C2)C(=O)c2nc(C(=O)N3CC(F)(F)C[C@@H]3C)c(s2)-c2ccc(c(Cl)c2Cl)C(O)(C(F)(F)F)C(F)(F)F)C1 |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1ccc(cc1C(F)F)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@@H]1CCCN1C(=O)c1nc(sc1-c1ccc(cc1C(F)F)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCCN1C(=O)c1nc(sc1-c1ccc(cc1C(F)F)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
CC(C)(O)CNC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1ccc(cc1C(F)F)C(O)(C(F)(F)F)C(F)(F)F
C[C@H]1CCCN1C(=O)c1nc(sc1-c1ccc(c(F)c1C(F)F)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1ccc(c(Cl)c1F)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1ccc(cc1OC(F)F)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
COc1cc(ccc1-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NCC(C)(C)O)C(O)(C(F)(F)F)C(F)(F)F |r|
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1ccc(cc1C(F)F)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
CCc1cc(ccc1-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NCC(C)(C)O)C(O)(C(F)(F)F)C(F)(F)F |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1ccc(cc1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCCN1C(=O)c1nc(sc1-c1cnc(cc1C)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1ccc(cc1F)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCCN1C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)c1noc(=O)[nH]1 |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(cc1C(F)(F)F)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCCN1C(=O)c1nc(sc1-c1cnc(cc1C(F)(F)F)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)CC2)c(s1)-c1cnc(cc1C(F)(F)F)C(O)(C(F)(F)F)C(F)(F)F
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(cc1C)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1ccc(cc1C)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@@H]1CCCN1C(=O)c1nc(sc1-c1ccc(cc1C)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1ccc(cc1OC(F)(F)F)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1ccc(cc1C)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1ccc(c(F)c1F)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCCN1C(=O)c1nc(sc1-c1ccc(cc1C)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCC(C)(C)O |r|
Cc1cc(ccc1-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)NCC(C)(C)O)C(O)(C(F)(F)F)C(F)(F)F
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(CC2)[N+]#[C-])c(s1)-c1ccc(cc1C(F)F)C(O)(C(F)(F)F)C(F)(F)F
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC[C@@H]2CO)c(s1)-c1ccc(cc1C(F)F)C(O)(C(F)(F)F)C(F)(F)F |r|
COc1cc(ccc1-c1sc(nc1C(=O)N1CCCC[C@@H]1C)C(=O)NCC(C)(C)O)C(O)(C(F)(F)F)C(F)(F)F |r|
COc1cc(ccc1-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)NCC(C)(C)O)C(O)(C(F)(F)F)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(C[C@H]4CC[C@@H](CC4)C(F)(F)F)Cc3c2)cc1 |r,wU:26.29,wD:23.22,17.17,(10.83,-2.3,;9.5,-3.07,;8.16,-2.3,;8.93,-.96,;7.39,-3.63,;6.83,-1.53,;5.5,-2.3,;4.16,-1.53,;4.16,.01,;2.83,.78,;1.49,.01,;.16,.78,;.16,2.32,;-1.17,.01,;-1.17,-1.53,;-2.51,-2.3,;-3.84,-1.53,;-5.3,-2,;-5.7,-3.49,;-7.19,-3.89,;-4.61,-4.58,;-6.21,-.76,;-7.75,-.76,;-8.52,.58,;-7.75,1.91,;-8.52,3.24,;-10.06,3.24,;-10.83,1.91,;-10.06,.58,;-10.83,4.58,;-12.37,4.58,;-10.06,5.91,;-9.29,4.58,;-5.3,.49,;-3.84,.01,;-2.51,.78,;5.5,.78,;6.83,.01,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(Cl)cc4)Cc3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C#N)Cc3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(OC(F)F)cc4)Cc3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc3c2)c2nccc(n2)C(F)(F)F)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(F)cc4)Cc3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc3c2)c2ncc(cn2)C(F)(F)F)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(Cl)cc4)C(=O)c3c2)cc1 |r|
CCOC(=O)c1cnc(nc1C(F)(F)F)N1Cc2cc(cnc2[C@@H]1C(C)C)C(=O)NCc1ccc(cc1)S(=O)(=O)CC |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3c(c2)C(=O)N(Cc2ccc(Cl)cc2)C3(O)C(C)C)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc3c2)c2ncc(CO)c(n2)C(F)(F)F)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(C(=O)c3c2)S(=O)(=O)c2ccc(cc2)C#N)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc3c2)c2ncc([C@@H](C)O)c(n2)C(F)(F)F)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc3c2)C(=O)OC(C)(C)C)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc3c2)C(=O)OCc2ccccc2)cc1 |r|
CC(C)[C@@H]1N(Cc2ccc(Cl)cc2)Cc2cc(cnc12)C(=O)NCc1ccc(cc1)S(C)(=O)=O |r|
CC(C)[C@H]1N(Cc2ccc(Cl)cc2)Cc2cc(cnc12)C(=O)NCc1ccc(cc1)S(C)(=O)=O |r|
CC(C)[C@H]1N(Cc2ccc(cc2)C#N)Cc2cc(cnc12)C(=O)NCc1ccc(cc1)S(C)(=O)=O |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(C[C@H]4CC[C@@H](CC4)C(F)(F)F)Cc3c2)cc1 |r,wU:26.29,wD:23.22,17.17,(11.6,-2.96,;10.27,-3.73,;8.93,-2.96,;9.7,-1.63,;8.16,-4.3,;7.6,-2.19,;6.27,-2.96,;4.93,-2.19,;4.93,-.65,;3.6,.12,;2.26,-.65,;.93,.12,;.93,1.66,;-.4,-.65,;-.4,-2.19,;-1.74,-2.96,;-3.07,-2.19,;-4.54,-2.67,;-4.93,-4.16,;-6.42,-4.56,;-3.84,-5.25,;-5.44,-1.42,;-6.98,-1.42,;-7.75,-.09,;-6.98,1.24,;-7.75,2.58,;-9.29,2.58,;-10.06,1.24,;-9.29,-.09,;-10.06,3.91,;-9.29,5.25,;-11.6,3.91,;-10.83,5.25,;-4.54,-.18,;-3.07,-.65,;-1.74,.12,;6.27,.12,;7.6,-.65,)|
CC(C)[C@@H]1N(Cc2ccc(cc2)C#N)Cc2cc(cnc12)C(=O)NCc1ccc(cc1)S(C)(=O)=O |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCc1ccc(cc1)S(C)(=O)=O |r|
CC(C)[C@@H]1N(Cc2ccc(Cl)cn2)Cc2cc(cnc12)C(=O)NCc1ccc(cc1)S(C)(=O)=O |r|
CC(C)[C@@H]1N(Cc2ccc(F)cc2)Cc2cc(cnc12)C(=O)NCc1ccc(cc1)S(C)(=O)=O |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc3c2)C(=O)OCc2ccc(Cl)cc2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4cnc(nc4)C(F)(F)F)Cc3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cn4)C(F)(F)F)Cc3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(Cl)cc4)[C@H](C)c3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(Cl)cc4)[C@@H](C)c3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)[C@H](C)c3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)[C@@H](C)c3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)C(=O)c3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)nc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(Cl)cc4)Cc3c2)nc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C#N)Cc3c2)nc1 |r|
CC(C)[C@@H]1N(Cc2ccc(cn2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCc1ccc(cc1)S(C)(=O)=O |r|
CC(C)[C@H]1N(Cc2ccc(cn2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCc1ccc(cc1)S(C)(=O)=O |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)-c4nnn(C)n4)Cc3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(nc4)C(F)(F)F)Cc3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@@H](C(C)C)N(Cc4ccc(nc4)C(F)(F)F)Cc3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(C[C@H]4CC[C@H](CC4)C(F)(F)F)Cc3c2)cc1 |r,wU:23.22,26.29,wD:17.17,(11.6,-2.96,;10.27,-3.73,;8.93,-2.96,;9.7,-1.63,;8.16,-4.3,;7.6,-2.19,;6.27,-2.96,;4.93,-2.19,;4.93,-.65,;3.6,.12,;2.26,-.65,;.93,.12,;.93,1.66,;-.4,-.65,;-.4,-2.19,;-1.74,-2.96,;-3.07,-2.19,;-4.54,-2.67,;-4.93,-4.16,;-6.42,-4.56,;-3.84,-5.25,;-5.44,-1.42,;-6.98,-1.42,;-7.75,-.09,;-9.29,-.09,;-10.06,1.24,;-9.29,2.58,;-7.75,2.58,;-6.98,1.24,;-10.06,3.91,;-9.29,5.25,;-11.6,3.91,;-10.83,5.25,;-4.54,-.18,;-3.07,-.65,;-1.74,.12,;6.27,.12,;7.6,-.65,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(CC4CCC(F)(F)CC4)Cc3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(CC4CCC(F)(F)CC4)Cc3c2)nc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(C[C@H]4CC[C@@H](CC4)C(=O)OC)Cc3c2)cc1 |r,wU:26.29,wD:23.22,17.17,(11.42,-1.63,;9.88,-1.63,;9.11,-2.96,;10.45,-3.73,;8.34,-4.3,;7.78,-2.19,;6.44,-2.96,;5.11,-2.19,;5.11,-.65,;3.78,.12,;2.44,-.65,;1.11,.12,;1.11,1.66,;-.22,-.65,;-.22,-2.19,;-1.56,-2.96,;-2.89,-2.19,;-4.36,-2.67,;-4.75,-4.16,;-6.24,-4.56,;-3.67,-5.25,;-5.26,-1.42,;-6.8,-1.42,;-7.57,-.09,;-6.8,1.24,;-7.57,2.58,;-9.11,2.58,;-9.88,1.24,;-9.11,-.09,;-9.88,3.91,;-11.42,3.91,;-9.11,5.25,;-7.57,5.25,;-4.36,-.18,;-2.89,-.65,;-1.56,.12,;6.44,.12,;7.78,-.65,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(C[C@H]4CC[C@@H](CC4)OC)Cc3c2)cc1 |r,wU:26.29,wD:23.22,17.17,(11.42,-.96,;9.88,-.96,;9.11,-2.3,;10.44,-3.07,;8.34,-3.63,;7.78,-1.53,;6.44,-2.3,;5.11,-1.53,;5.11,.01,;3.78,.78,;2.44,.01,;1.11,.78,;1.11,2.32,;-.22,.01,;-.22,-1.53,;-1.56,-2.3,;-2.89,-1.53,;-4.36,-2,;-4.75,-3.49,;-6.24,-3.89,;-3.67,-4.58,;-5.26,-.76,;-6.8,-.76,;-7.57,.58,;-6.8,1.91,;-7.57,3.24,;-9.11,3.24,;-9.88,1.91,;-9.11,.58,;-9.88,4.58,;-11.42,4.58,;-4.36,.49,;-2.89,.01,;-1.56,.78,;6.44,.78,;7.78,.01,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc3c2)C(=O)OC(C)(C)C)nc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(C[C@H]4CC[C@@H](CC4)C(F)(F)F)C(=O)c3c2)nc1 |r,wU:26.29,wD:23.22,17.17,(11.6,-2.96,;10.27,-2.19,;8.93,-2.96,;9.7,-4.3,;8.16,-4.3,;7.6,-2.19,;7.6,-.65,;6.27,.12,;4.93,-.65,;3.6,.12,;2.26,-.65,;.93,.12,;.93,1.66,;-.4,-.65,;-.4,-2.19,;-1.74,-2.96,;-3.07,-2.19,;-4.54,-2.67,;-4.93,-4.16,;-6.42,-4.56,;-3.84,-5.25,;-5.44,-1.42,;-6.98,-1.42,;-7.75,-.09,;-6.98,1.24,;-7.75,2.58,;-9.29,2.58,;-10.06,1.24,;-9.29,-.09,;-10.06,3.91,;-9.29,5.25,;-11.6,3.91,;-10.83,5.25,;-4.54,-.18,;-4.93,1.31,;-3.07,-.65,;-1.74,.12,;4.93,-2.19,;6.27,-2.96,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H]([C@@H]4CCOC4)N(Cc4ccc(cc4)C#N)Cc3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(CC4CCN(CC(F)(F)F)CC4)Cc3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H]([C@H]4CCOC4)N(Cc4ccc(cc4)C#N)Cc3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@@H]([C@@H]4CCOC4)N(Cc4ccc(cc4)C#N)Cc3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@@H]([C@H]4CCOC4)N(Cc4ccc(cc4)C#N)Cc3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@@H](C(C)C)N(C[C@H]4CC[C@@H](CC4)C(F)(F)F)Cc3c2)nc1 |r,wU:26.29,17.17,wD:23.22,(11.42,-1.63,;9.88,-1.63,;9.11,-2.96,;10.45,-3.73,;8.34,-4.3,;7.78,-2.19,;7.78,-.65,;6.44,.12,;5.11,-.65,;3.78,.12,;2.44,-.65,;1.11,.12,;1.11,1.66,;-.22,-.65,;-.22,-2.19,;-1.56,-2.96,;-2.89,-2.19,;-4.36,-2.67,;-4.75,-4.16,;-6.24,-4.56,;-3.67,-5.25,;-5.26,-1.42,;-6.8,-1.42,;-7.57,-.09,;-6.8,1.24,;-7.57,2.58,;-9.11,2.58,;-9.88,1.24,;-9.11,-.09,;-9.88,3.91,;-9.11,5.25,;-11.42,3.91,;-10.65,5.25,;-4.36,-.18,;-2.89,-.65,;-1.56,.12,;5.11,-2.19,;6.44,-2.96,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc5OC(F)(F)Oc5c4)Cc3c2)nc1 |r|
CCS(=O)(=O)c1ccc(CC(=O)Nc2cnc3[C@H](C(C)C)N(C[C@H]4CC[C@@H](CC4)C(F)(F)F)Cc3c2)cc1 |r,wU:26.29,wD:23.22,17.17,(11.6,-2.96,;10.27,-3.73,;8.93,-2.96,;9.7,-1.63,;8.16,-4.3,;7.6,-2.19,;6.27,-2.96,;4.93,-2.19,;4.93,-.65,;3.6,.12,;2.26,-.65,;2.26,-2.19,;.93,.12,;-.4,-.65,;-.4,-2.19,;-1.74,-2.96,;-3.07,-2.19,;-4.54,-2.67,;-4.93,-4.16,;-6.42,-4.56,;-3.84,-5.25,;-5.44,-1.42,;-6.98,-1.42,;-7.75,-.09,;-6.98,1.24,;-7.75,2.58,;-9.29,2.58,;-10.06,1.24,;-9.29,-.09,;-10.06,3.91,;-9.29,5.25,;-11.6,3.91,;-10.83,5.25,;-4.54,-.18,;-3.07,-.65,;-1.74,.12,;6.27,.12,;7.6,-.65,)|
CCS(=O)(=O)c1ccc(CC(=O)Nc2cnc3[C@H](C(C)C)N(Cc4ccc(Cl)cc4)Cc3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CC(=O)Nc2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C#N)Cc3c2)cc1 |r|
CCS(=O)(=O)c1ccc(CC(=O)Nc2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)cc1 |r|
CCS(=O)(=O)c1ccc(nc1)[C@@H](C)NC(=O)c1cnc2[C@H](C(C)C)N(Cc3ccc(cc3)C(F)(F)F)Cc2c1 |r|
CCS(=O)(=O)c1ccc(nc1)[C@H](C)NC(=O)c1cnc2[C@H](C(C)C)N(Cc3ccc(cc3)C(F)(F)F)Cc2c1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC1CCS(=O)(=O)CC1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCCC1CCS(=O)(=O)CC1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC1CCN(CC1)S(C)(=O)=O |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCc1ccc(cc1)C#N |r|
COC(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)cc1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCCC1CN(C1)C(=O)OC(C)(C)C |r|
CNS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)cc1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC1CN(C1)C(=O)OC(C)(C)C |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCc1cn2cccnc2n1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC(O)c1ccc(cc1)C(F)(F)F |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)N[C@@H](CCO)c1ccc(Cl)cc1 |r|
COc1cccc(c1)C(C)(C)CNC(=O)c1cnc2[C@H](C(C)C)N(Cc3ccc(cc3)C(F)(F)F)Cc2c1 |r|
CN\C(CNC(=O)c1cnc2[C@H](C(C)C)N(Cc3ccc(cc3)C(F)(F)F)Cc2c1)=C/C=N |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC1CCN(C1)C(=O)OC(C)(C)C |r|
COC(=O)[C@H]1CC[C@H](CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)CC1 |r,wU:7.7,wD:16.16,4.3,(10.93,-.65,;10.93,-2.19,;9.6,-2.96,;9.6,-4.5,;8.27,-2.19,;8.27,-.65,;6.93,.12,;5.6,-.65,;4.26,.12,;2.93,-.65,;1.6,.12,;1.6,1.66,;.26,-.65,;.26,-2.19,;-1.07,-2.96,;-2.4,-2.19,;-3.87,-2.67,;-4.27,-4.16,;-5.75,-4.56,;-3.18,-5.25,;-4.77,-1.42,;-6.31,-1.42,;-7.08,-.09,;-6.31,1.24,;-7.08,2.58,;-8.62,2.58,;-9.39,1.24,;-8.62,-.09,;-9.39,3.91,;-8.62,5.25,;-10.93,3.91,;-10.16,5.25,;-3.87,-.18,;-2.4,-.65,;-1.07,.12,;5.6,-2.19,;6.93,-2.96,)|
CN\C=C(\CNC(=O)c1cnc2[C@H](C(C)C)N(Cc3ccc(cc3)C(F)(F)F)Cc2c1)C=N |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCCN1CCOCC1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCc1ccccn1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCCCN1CCCC1=O |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC1(CC1)c1ccc(Cl)cc1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCc1ccccc1CN1CCN(C)CC1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCc1ccn(C)n1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCc1ccnnc1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCc1cccnn1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC1COCCO1 |r|
CCS(=O)(=O)CCNC(=O)c1cnc2[C@H](C(C)C)N(Cc3ccc(cc3)C(F)(F)F)Cc2c1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NC1(CO)Cc2ccccc2C1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC(N1CCOCC1)c1cccnc1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCCc1ccc2CCCNc2n1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCCC1CCOCC1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCCCS(=O)(=O)c1ccccc1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC(N(C)C)c1ccncc1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC(N1CCOCC1)c1ccc(cc1)C(F)(F)F |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCc1nnc2CCCn12 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC1CCN(CC1)C(=O)OC(C)(C)C |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCCCn1ccnc1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCCc1ccccn1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCc1ccccc1OCCN(C)C |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCCN1CCN(C)CC1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC1CCN(C)CC1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCCc1ccnc(O)c1 |r|
CCS(=O)(=O)N1CC(CCNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)C1 |r|
COC(=O)N1CC(CCNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)C1 |r|
CCS(=O)(=O)N1CC(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)C1 |r|
COC(=O)N1CC(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)C1 |r|
CCS(=O)(=O)N1CCC(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)C1 |r|
COC(=O)N1CCC(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)C1 |r|
CNC(=O)[C@H]1CC[C@H](CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)CC1 |r,wU:4.3,wD:16.16,7.7,(11.6,-2.96,;10.27,-2.19,;8.93,-2.96,;8.93,-4.5,;7.6,-2.19,;6.27,-2.96,;4.93,-2.19,;4.93,-.65,;3.6,.12,;2.26,-.65,;.93,.12,;.93,1.66,;-.4,-.65,;-.4,-2.19,;-1.74,-2.96,;-3.07,-2.19,;-4.54,-2.67,;-4.93,-4.16,;-6.42,-4.56,;-3.84,-5.25,;-5.44,-1.42,;-6.98,-1.42,;-7.75,-.09,;-6.98,1.24,;-7.75,2.58,;-9.29,2.58,;-10.06,1.24,;-9.29,-.09,;-10.06,3.91,;-9.29,5.25,;-11.6,3.91,;-10.83,5.25,;-4.54,-.18,;-3.07,-.65,;-1.74,.12,;6.27,.12,;7.6,-.65,)|
CCS(=O)(=O)N1CCC(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)CC1 |r|
COC(=O)N1CCC(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)CC1 |r|
CNS(=O)(=O)N1CCC(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)CC1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC1CCN(CC1)C(=O)C(C)O |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC1CCN(CC1)C(=O)CO |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC1CCN(CC1)C(C)=O |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCc1ccncc1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCc1cccc(c1)S(C)(=O)=O |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC(F)(F)F |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC1(O)CCC2(CC1)OCCO2 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)N[C@H](C)c1ccc(Br)cc1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NC1(CC1)c1cnccn1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCCC1C(=O)Nc2ccc(Cl)cc12 |r|
CC(C)NC(=O)c1cnc2[C@H](C(C)C)N(Cc3ccc(cc3)C(F)(F)F)Cc2c1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NC(CO)c1ccc(Br)cc1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC(F)F |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)N[C@@H]1[C@H](O)Cc2ccccc12 |r|
COC(=O)C(Cc1ccc(F)cc1)NC(=O)c1cnc2[C@H](C(C)C)N(Cc3ccc(cc3)C(F)(F)F)Cc2c1 |r|
COC(=O)C[C@H]1CC[C@H](CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)CC1 |r,wU:8.8,wD:17.17,5.4,(12.27,-2.19,;10.93,-2.96,;9.6,-2.19,;9.6,-.65,;8.27,-2.96,;6.93,-2.19,;6.93,-.65,;5.6,.12,;4.26,-.65,;2.93,.12,;1.6,-.65,;.26,.12,;.26,1.66,;-1.07,-.65,;-1.07,-2.19,;-2.4,-2.96,;-3.74,-2.19,;-5.2,-2.67,;-5.6,-4.16,;-7.09,-4.55,;-4.51,-5.25,;-6.11,-1.42,;-7.65,-1.42,;-8.42,-.09,;-7.65,1.24,;-8.42,2.58,;-9.96,2.58,;-10.73,1.24,;-9.96,-.09,;-10.73,3.91,;-9.96,5.25,;-12.27,3.91,;-11.5,5.25,;-5.2,-.18,;-3.74,-.65,;-2.4,.12,;4.26,-2.19,;5.6,-2.96,)|
COC(=O)CC(NC(=O)c1cnc2[C@H](C(C)C)N(Cc3ccc(cc3)C(F)(F)F)Cc2c1)c1ccc(Br)cc1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NC[C@H]1CC[C@@H](CC1)C#N |r,wU:27.29,wD:3.2,30.36,(-5.75,-4.56,;-4.27,-4.16,;-3.18,-5.25,;-3.87,-2.67,;-4.77,-1.42,;-6.31,-1.42,;-7.08,-.09,;-6.31,1.24,;-7.08,2.58,;-8.62,2.58,;-9.39,1.24,;-8.62,-.09,;-9.39,3.91,;-8.62,5.25,;-10.93,3.91,;-10.16,5.25,;-3.87,-.18,;-2.4,-.65,;-1.07,.12,;.26,-.65,;.26,-2.19,;-1.07,-2.96,;-2.4,-2.19,;1.6,.12,;1.6,1.66,;2.93,-.65,;4.26,.12,;5.6,-.65,;6.93,.12,;8.27,-.65,;8.27,-2.19,;6.93,-2.96,;5.6,-2.19,;9.6,-2.96,;10.93,-3.73,)|
CCS(=O)(=O)N\C=C(\CNC(=O)c1cnc2[C@H](C(C)C)N(Cc3ccc(cc3)C(F)(F)F)Cc2c1)C=N |r|
COC(=O)C1(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)CCOCC1 |r|
COC(=O)C(Cc1cc(=O)[nH]c2ccccc12)NC(=O)c1cnc2[C@H](C(C)C)N(Cc3ccc(cc3)C(F)(F)F)Cc2c1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NC(Cc1cc(=O)[nH]c2ccccc12)C(O)=O |r|
COC(=O)CC1(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)CCCCC1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NC(Cc1ccc(F)cc1)C(O)=O |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NC[C@H]1CC[C@H](CC(O)=O)CC1 |r,wU:27.29,wD:3.2,30.33,(-6.42,-4.56,;-4.93,-4.16,;-3.84,-5.25,;-4.54,-2.67,;-5.44,-1.42,;-6.98,-1.42,;-7.75,-.09,;-6.98,1.24,;-7.75,2.58,;-9.29,2.58,;-10.06,1.24,;-9.29,-.09,;-10.06,3.91,;-9.29,5.25,;-11.6,3.91,;-10.83,5.25,;-4.54,-.18,;-3.07,-.65,;-1.74,.12,;-.4,-.65,;-.4,-2.19,;-1.74,-2.96,;-3.07,-2.19,;.93,.12,;.93,1.66,;2.26,-.65,;3.6,.12,;4.93,-.65,;6.27,.12,;7.6,-.65,;7.6,-2.19,;8.93,-2.96,;10.27,-2.19,;11.6,-2.96,;10.27,-.65,;6.27,-2.96,;4.93,-2.19,)|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NC(CC(O)=O)c1ccc(Br)cc1 |r|
CCS(=O)(=O)c1ccc(nc1)C1(CC1)NC(=O)c1cnc2[C@H](C(C)C)N(Cc3ccc(cc3)C(F)(F)F)Cc2c1 |r|
CCS(=O)(=O)c1cnc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)c(C)c1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)nc1C |r|
CCS(=O)(=O)c1cnc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)c(F)c1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC1(CC(O)=O)CCCCC1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC1(CCOCC1)C(O)=O |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCc1ccc(cc1)C(O)=O |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NC[C@H]1CC[C@@H](CC1)C(O)=O |r,wU:27.29,wD:3.2,30.36,(-5.75,-4.56,;-4.27,-4.16,;-3.18,-5.25,;-3.87,-2.67,;-4.77,-1.42,;-6.31,-1.42,;-7.08,-.09,;-6.31,1.24,;-7.08,2.58,;-8.62,2.58,;-9.39,1.24,;-8.62,-.09,;-9.39,3.91,;-8.62,5.25,;-10.93,3.91,;-10.16,5.25,;-3.87,-.18,;-2.4,-.65,;-1.07,.12,;.26,-.65,;.26,-2.19,;-1.07,-2.96,;-2.4,-2.19,;1.6,.12,;1.6,1.66,;2.93,-.65,;4.26,.12,;5.6,-.65,;6.93,.12,;8.27,-.65,;8.27,-2.19,;6.93,-2.96,;5.6,-2.19,;9.6,-2.96,;10.93,-2.19,;9.6,-4.5,)|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)N[C@@H](CO)c1ccc(cc1)C#N |r|
COC(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)nc1 |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCc1ccc(cn1)C(O)=O |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCCC1CN(C1)S(C)(=O)=O |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC1CN(C1)S(C)(=O)=O |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCC1CCN(C1)S(C)(=O)=O |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCc1ccc(cn1)C#N |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NC[C@@H]1CCN(C[C@H]1O)C(=O)OC(C)(C)C |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NC[C@@H]1CCN(C[C@H]1OC(C)=O)C(C)=O |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)N[C@H](CO)c1ccc(cc1)C#N |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)nn1 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CN)CN(c2c1)S(=O)(=O)c1ccc(F)cc1
CCn1cc(c(C)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cnn(C)c1C
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc2nccn2c1
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc2nccn12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(C)c(c1)C#N |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cc(Br)ccc1Cl |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cnn(C(F)F)c1C |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1c(C)nn2CCCOc12 |r|
COc1c(c(C)nn1C)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1c(C)nn2CCCCc12 |r|
COc1nn(C)c(C)c1S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cnc2sccn12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(Cl)c1Cl |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1c(C)nc2ncccn12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cnn2CCCOc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1c(C)nn2cccnc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(Cl)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1Cl |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(Cl)c1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C#N |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)S(C)(=O)=O |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C#N |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)c(C)c1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cc(cnc1Cl)C(F)(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cc(C)cnc1Cl |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cc(C)c[nH]c1=O |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cncc(C)c1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)c(F)c1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cncc(c1)C(F)(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(Cl)c(c1)C#N |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cc(ccc1C)C#N |r|
CC(C)n1nc(C)c(c1C)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cnc2ccccn12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1c(C)nc2ccccn12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1c(C)nc2sccn12 |r|
COc1nn2CCCCc2c1S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
COc1nn2CCCc2c1S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1c(Cl)nn2CCCCc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(n1)C(F)(F)F |r|
CCn1cc(c(OC)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CCn1cc(c(OCC(=O)OC)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CCn1cc(c(OCC(F)F)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CCn1cc(c(OCC(O)=O)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CCn1cc(c(OCC(=O)NC)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CCn1cc(c(OCC(F)(F)F)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1c(Cl)nn2CCCc12 |r|
CCNc1nn(CC)cc1S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CCn1cc(c(n1)C1CC1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CCn1cc(c(OC(F)F)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CCn1cc(c(n1)N(C)C)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1
CCn1cc(c(O)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(OC(C)C)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(F)c1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(C)c1 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(Cl)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C#N |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(Cl)c(c1)C#N |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cc(ccc1C)C#N |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(C)c1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cc(ccc1Cl)C#N |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cc(Cl)cc(c1)C#N |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cnn(C(F)F)c1C |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(C)nc1C(F)(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1sc(C)nc1C |r|
CCOc1cc(ccc1F)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(OC(F)F)c1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(OC(F)(F)F)c1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cnc(C)s1 |r|
CCn1ncc(c1C)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1nc(C)c(c1C)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCCn1cc(c(C)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1sc(C)nc1C(F)(F)F |r|
CCCn1nc(C)c(c1C)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1c(C)nn(CC(F)(F)F)c1C |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1c(C)nn(CC(F)F)c1C |r|
CCn1cc(c(n1)C(F)(F)F)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(C)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cnn(C)c1C |r|
Cc1c(cnn1C)S(=O)(=O)N1C[C@H](CNS(C)(=O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1nn2CCCc2c1S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1nn2CCCCc2c1S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1c(C)nn(C(F)F)c1C |r|
CCn1cc(c(OC)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cncc(c1)C1CC1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1c(Cl)nn2CCCCc12 |r|
COc1nn(C)c(C)c1S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1c(Cl)nn2CCCc12 |r|
CCn1cc(c(OCC(F)F)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC(F)F)cc1S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(n1)C1CC1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OC(F)F)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(NC)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCNc1nn(CC)cc1S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1C)C1CC1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cnn(C2CC2)c1C |r|
CCOc1nn(cc1S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cnc2ccccn12 |r|
CCn1cc(c(OCc2ccccc2)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCCCOCc2ccccc2)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCCCO)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCCn1nc(C)cc1S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COCCn1cc(c(C)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COCCn1ncc(c1C)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)n1cc(c(C)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)n1ncc(c1C)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1c(OCCO)nn2CCCCc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1Cl)C(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1C)C1CCC1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cnn(C2COC2)c1C |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(CCO)nc1Cl |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cnn(CCO)c1C |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(CC(C)(C)O)nc1C |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cnn(CC(C)(C)O)c1C |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@H](CNC(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@H](CNC(=O)[C@@H]2C[C@@H]2F)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@H](CNC(=O)C(C)(C)O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@H](CNC(=O)C(C)(O)C(F)(F)F)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@H](CNC(=O)C(C)(N)C(F)(F)F)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@H](CNS(=O)(=O)CC(F)(F)F)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@H](CNS(C)(=O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C1CC1
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C1CC1
C[C@@H](NC(C)=O)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1
C[C@H](NC(C)=O)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1
C[C@@H](NC(C)=O)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
C[C@H](NC(C)=O)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
C[C@@H](NC(C)=O)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(F)c1 |r|
C[C@H](NC(C)=O)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(F)c1 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@@H](C)NC(C)=O |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@H](C)NC(C)=O |r|
COc1nn(C)c(C)c1S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@@H](C)NC(C)=O |r|
COc1nn(C)c(C)c1S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@H](C)NC(C)=O |r|
C[C@H](NC(C)=O)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@H](NC(C)=O)[C@@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@@H](NC(C)=O)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N[C@H](C1CC1)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N[C@@H](C1CC1)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC(C)(C)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1
CC(=O)NC(C)(C)[C@@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1
CC(=O)NC(C)(C)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC(=O)NC(C)(C)[C@@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC(=O)NC(C)(C)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(NS(C)(=O)=O)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC(C)(NS(=O)(=O)C1CC1)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC(C)(NS(C)(=O)=O)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(F)c1 |r|
CC(C)(NS(C)(=O)=O)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CN(C)C(=O)C(=O)NC(C)(C)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(NS(=O)(=O)C1CC1)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(C)(C)NC(C)=O |r|
CC(=O)NC(C)(C)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(=O)NC(C)(C)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F |r|
COc1nn(C)c(C)c1S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(C)(C)NC(C)=O |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(C)(C)NC(C)=O |r|
CC(=O)NC(C)(C)[C@@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(=O)NC(C)(C)[C@@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F |r|
CCC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
CCC(C)(C)OC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)C(C)(C)OC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C#N)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC3(C)CCC3)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC3(C)CC3)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC(F)(F)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C3CC3)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C(F)(F)F)C(C)(C)c3ccccc3)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C(F)(F)F)C3(C)CCCCC3)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C3CCCCC3)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C3CCCCC3)C(F)(F)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@@H](OC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)C(F)(F)F |r|
C[C@H](OC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)C(F)(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C(F)(F)F)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC3(CCCCC3)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC3(CCC(C)(C)CC3)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(c3ccccc3)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(c3ccc(Cl)cc3)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(c3ccccc3)C(F)(F)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(c3ccccc3)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CCC(OC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)C(F)(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(Cc3ccccc3)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC3(CC3)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC3(CC3)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
Fc1ccc(cc1)S(=O)(=O)N1C[C@H](CNC(=O)C2CC2)Oc2ccc(NC(=O)OCC3(CC3)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC3(CC3)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(F)c1 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OCC3(CC3)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC3(CC3)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(C)c1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC3(CC3)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC3CCC(F)(F)CC3)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC3CC3(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC3CCCC3)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC3CCCC3)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC3CCCCC3)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC3CCCCC3C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC3CC4CCC3C4)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC3(CC(F)(F)F)C4CCCC34)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)O[C@@H]3CCCC[C@@H]3C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)O[C@H]3CCCC[C@H]3C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(OC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(C)(C)C |r|
CC(OC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
C[C@@H](OC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(C)(C)C |r|
C[C@H](OC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(C)(C)C |r|
C[C@H](OC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1cn(nc1C)C(F)F)C(C)(C)C |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)O[C@H](C(C)(C)C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)O[C@@H](C(C)(C)C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@@H](OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3CC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(C)(C)C |r|
C[C@H](OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3CC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(C)(C)C |r|
C[C@@H](OC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1cn(nc1C)C(F)F)C(C)(C)C |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC(F)(F)c3ccccc3)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC3CC(F)(F)C3(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC(C)(C)C#N)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC(C)(C)C)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(C)COC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(C)COC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC3(C)CC3)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CCC(C)OC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC3(C)CCCC3)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC3(C)CN(C3)C(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCc3ccccc3)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCc3ccccc3Cl)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CCC(C)(C)C(F)(F)COC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC(F)(F)C(C)(C)C=C)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC3(CC3(F)F)c3ccccc3)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCCC(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC[Si](C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC(Cl)(Cl)Cl)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC(Cl)(Cl)Cl)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
Fc1ccc(cc1)S(=O)(=O)N1C[C@H](CNC(=O)C2CC2)Oc2ccc(NC(=O)OCC(Cl)(Cl)Cl)cc12 |r|
COC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(C)OC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)Oc3ccccc3)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)Oc3ccc(Cl)cc3)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)Oc3ccccc3Cl)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC3CC3)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCC3CC3)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OCCS(C)(=O)=O)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(OC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C1CC1 |r|
CC(OC(=O)Nc1ccc2O[C@@H](CNC(C)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(F)CC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CNC(=O)C(C)(C)C)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(C)CC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
CCC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CCCC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3CC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3CC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
Cc1nn(cc1S(=O)(=O)N1C[C@H](CNC(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C)cc12)C(F)F |r|
CC(C)(C)COC(=O)Nc1ccc2O[C@@H](CNC(=O)C3CC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
Cc1nn(cc1S(=O)(=O)N1C[C@H](CNC(=O)C2CC2)Oc2ccc(NC(=O)OCC(C)(C)C)cc12)C(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3C[C@@H]3F)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3CC(F)C3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r,wD:12.12,(-7.51,-3.64,;-8.28,-2.31,;-9.05,-3.64,;-6.94,-1.54,;-5.61,-2.31,;-5.61,-3.85,;-4.28,-1.54,;-2.94,-2.31,;-2.94,-3.85,;-1.61,-4.62,;-.28,-3.85,;1.06,-4.62,;2.39,-3.85,;3.72,-4.62,;5.06,-3.85,;6.39,-4.62,;6.39,-6.16,;7.73,-3.85,;9.21,-4.25,;9.61,-2.76,;10.95,-1.99,;8.12,-2.36,;2.39,-2.31,;1.06,-1.54,;-.28,-2.31,;-1.61,-1.54,;1.06,,;2.6,,;-.48,,;1.06,1.54,;2.39,2.31,;2.39,3.85,;1.06,4.62,;1.06,6.16,;-.28,3.85,;-.28,2.31,;-9.61,-1.54,;-9.61,,;-10.95,-2.31,;-10.95,-.77,)|
CC(C)(OC(=O)Nc1ccc2O[C@H](CNC(=O)C3CC(F)(F)C3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC1CC1C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3CC3(F)F)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C34CC(C3)C4)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(C)CC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC1CC(C1)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r,wD:9.9,(10.95,-1.99,;9.61,-2.76,;9.21,-4.25,;7.73,-3.85,;8.12,-2.36,;6.39,-4.62,;6.39,-6.16,;5.06,-3.85,;3.72,-4.62,;2.39,-3.85,;2.39,-2.31,;1.06,-1.54,;-.28,-2.31,;-1.61,-1.54,;-2.94,-2.31,;-4.28,-1.54,;-5.61,-2.31,;-5.61,-3.85,;-6.94,-1.54,;-8.28,-2.31,;-7.51,-3.64,;-9.05,-3.64,;-9.61,-1.54,;-9.61,,;-10.95,-2.31,;-10.95,-.77,;-2.94,-3.85,;-1.61,-4.62,;-.28,-3.85,;1.06,-4.62,;1.06,,;2.6,,;-.48,,;1.06,1.54,;2.39,2.31,;2.39,3.85,;1.06,4.62,;1.06,6.16,;-.28,3.85,;-.28,2.31,)|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3CC3(C)C)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)[C@H]3C[C@@H]3F)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CN(C)C1(CC1)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(C)CCC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(N)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C(O)C(F)(F)F)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C(C)(N)C(F)(F)F)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(N)CCCC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(F)C(N)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C(N)C(F)(F)F)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(N)CC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C(C)(O)C(F)(F)F)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(O)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(N(C)C)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CN(C)C(=O)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CN(C)C(C)(C)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CNC(C)(C)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(C)N1CCC1C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3CC33CCC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(C)CC3(F)F)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3COC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(C)COC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CN1CC(C1)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(N)COC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3CCCOC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@H](CNC(=O)CC3CCOCC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@H](CNC(=O)C3CCOCC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
Cn1cc(cn1)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)c3cn[nH]c3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(CC3)C(F)(F)F)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
Cn1cccc1C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(CC3)C#N)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)c3ccno3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)c3c[nH]cn3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(O)CC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)c3ncc[nH]3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)c3nc[nH]n3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)c3cnn[nH]3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)c3ccco3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3CCN3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3CNC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3CCCO3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(C)CCC(=O)N3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(O)CCC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
COC1CC(C1)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r,wD:10.10,(11.61,-2.76,;10.28,-1.99,;8.95,-2.76,;8.55,-4.25,;7.06,-3.85,;7.46,-2.36,;5.73,-4.62,;5.73,-6.16,;4.39,-3.85,;3.06,-4.62,;1.72,-3.85,;1.72,-2.31,;.39,-1.54,;-.94,-2.31,;-2.28,-1.54,;-3.61,-2.31,;-4.94,-1.54,;-6.28,-2.31,;-6.28,-3.85,;-7.61,-1.54,;-8.95,-2.31,;-8.18,-3.64,;-9.72,-3.64,;-10.28,-1.54,;-10.28,,;-11.61,-2.31,;-11.61,-.77,;-3.61,-3.85,;-2.28,-4.62,;-.94,-3.85,;.39,-4.62,;.39,,;1.93,,;-1.15,,;.39,1.54,;1.72,2.31,;1.72,3.85,;.39,4.62,;.39,6.16,;-.94,3.85,;-.94,2.31,)|
CC(C)N1CC(C1)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@H](CNC(=O)C3(C)CCCC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3CCO3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)c3nnc[nH]3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(O)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
Cc1noc(C)c1CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)[C@@H]3C[C@@H]3C#N)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)c3ccc[nH]3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
Cc1noc(C)c1C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
Cc1nc[nH]c1C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
Cc1nc(c[nH]1)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CCS(=O)(=O)c1cccc(c1)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CCS(=O)(=O)c1ccc(cc1)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CCS(=O)(=O)c1ccc(CC(=O)NC[C@H]2CN(c3cc(NC(=O)OC(C)(C)C(F)(F)F)ccc3O2)S(=O)(=O)c2ccc(F)cc2)cc1 |r|
COC(C)(C)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3CCOCC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3COC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CCn1cc(c(OC)n1)S(=O)(=O)N1C[C@H](CNC(=O)C2COC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1nn2CCCc2c1S(=O)(=O)N1C[C@H](CNC(=O)C2COC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)[C@@H]3C[C@@H]3F)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(C)COC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(N)COC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(C)CCCO3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)C1CC(CCO1)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(CCOCC3)C#N)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(C)CCCCO3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
Cn1cc(cn1)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)c3cn[nH]c3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(CC3)C(F)(F)F)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(C)CC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(CC3)C#N)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(O)CC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)c3ncc[nH]3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC1CC1C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)[C@@H]3CCCO3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3CCCO3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)[C@@H]3C[C@@H]3C#N)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(C)CCC(=O)N3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(O)CCC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
COC1CC(C1)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r,wD:10.10,(10.95,-.45,;10.95,-1.99,;9.61,-2.76,;9.21,-4.25,;7.73,-3.85,;8.12,-2.36,;6.39,-4.62,;6.39,-6.16,;5.06,-3.85,;3.72,-4.62,;2.39,-3.85,;2.39,-2.31,;1.06,-1.54,;-.28,-2.31,;-1.61,-1.54,;-2.94,-2.31,;-4.28,-1.54,;-5.61,-2.31,;-5.61,-3.85,;-6.94,-1.54,;-8.28,-2.31,;-7.51,-3.64,;-9.05,-3.64,;-9.61,-1.54,;-9.61,,;-10.95,-2.31,;-10.95,-.77,;-2.94,-3.85,;-1.61,-4.62,;-.28,-3.85,;1.06,-4.62,;1.06,,;2.6,,;-.48,,;1.06,1.54,;-.28,2.31,;-.28,3.85,;1.06,4.62,;1.06,6.16,;2.39,3.85,;3.72,4.62,;2.39,2.31,)|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3CC(F)(F)C3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C34CC(C3)C4)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3CCCOC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(C)CCCC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)[C@H]3C[C@@H]3F)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3CCOC(C)(C)C3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(C)CCOCC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CCC1(COC1)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(F)CCOCC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3(C)CCC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CCn1cc(c(C)n1)S(=O)(=O)N1C[C@H](CNC(=O)C2COC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3COC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(F)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)[C@@H]3C[C@@H]3C#N)CN(c2c1)S(=O)(=O)c1ccc(F)c(F)c1)C(F)(F)F |r|
CCn1cc(c(C)n1)S(=O)(=O)N1C[C@H](CNC(=O)[C@@H]2C[C@@H]2C#N)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)[C@H]3C[C@@H]3F)CN(c2c1)S(=O)(=O)c1ccc(F)c(F)c1)C(F)(F)F |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CNC(=O)C2COC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)CC3CCCOC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC1OCCC1C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CCn1cc(c(OC(F)F)n1)S(=O)(=O)N1C[C@H](CNC(=O)[C@@H]2C[C@@H]2F)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OC(F)F)n1)S(=O)(=O)N1C[C@H](CNC(=O)C(C)(C)O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OC(F)F)n1)S(=O)(=O)N1C[C@H](CNC(=O)C(C)(N)C(F)(F)F)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(cc1S(=O)(=O)N1C[C@H](CNC(=O)[C@@H]2C[C@@H]2F)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(F)F |r|
CCOc1nn(cc1S(=O)(=O)N1C[C@H](CNC(=O)C(C)(C)O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(F)F |r|
CCOc1nn(cc1S(=O)(=O)N1C[C@H](CNC(=O)C(C)(N)C(F)(F)F)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(F)F |r|
CCn1cc(c(OCC(F)F)n1)S(=O)(=O)N1C[C@H](CNC(=O)C(C)(C)O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC(F)F)cc1S(=O)(=O)N1C[C@H](CNC(=O)C(C)(C)O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(C)n1)S(=O)(=O)N1C[C@H](CNC(=O)C(C)(C)O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1nn2CCCc2c1S(=O)(=O)N1C[C@H](CNC(=O)C(C)(C)O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)C3CC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
Cc1nn(cc1S(=O)(=O)N1C[C@H](CNS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)C3CC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(F)c1)C(F)(F)F |r|
CCOc1cc(ccc1F)S(=O)(=O)N1C[C@H](CNS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
Cc1c(cnn1C(F)F)S(=O)(=O)N1C[C@H](CNS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CNS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)C3CC3)CN(c2c1)S(=O)(=O)c1cccc(c1)S(C)(=O)=O)C(F)(F)F |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CNS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)C3CC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(F)c1 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CNS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)C3CC3)CN(c2c1)S(=O)(=O)c1cccc(c1)C#N)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)C3CC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)C3CC3)CN(c2c1)S(=O)(=O)c1cccc(c1)C#N |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)C3CC3)CN(c2c1)S(=O)(=O)c1cccc(c1)S(C)(=O)=O |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)C3CC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)C3CC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
Fc1ccc(cc1)S(=O)(=O)N1C[C@H](CNS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OCC3(CC3)C(F)(F)F)cc12 |r|
Cc1nn(cc1S(=O)(=O)N1C[C@H](CNS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C)cc12)C(F)F |r|
COc1nn2CCCCc2c1S(=O)(=O)N1C[C@H](CNS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OC)n1)S(=O)(=O)N1C[C@H](CNS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1nn2CCCc2c1S(=O)(=O)N1C[C@H](CNS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(C)n1)S(=O)(=O)N1C[C@H](CNS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@H](CNS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CNS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(cc1S(=O)(=O)N1C[C@H](CNS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(F)F |r|
CCn1cc(c(OC(F)F)n1)S(=O)(=O)N1C[C@H](CNS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCC(=O)OC)n1)S(=O)(=O)N1C[C@H](CNS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CNS(C)(=O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)c(F)c1 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CNS(C)(=O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)S(C)(=O)=O |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CNS(C)(=O)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
Cc1nn(cc1S(=O)(=O)N1C[C@H](CNS(C)(=O)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12)C(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CNS(C)(=O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C#N |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CNS(C)(=O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(C)(=O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CNS(C)(=O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CCn1cc(c(C)n1)S(=O)(=O)N1C[C@H](CNS(C)(=O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(C)(=O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)c3cccnc3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
Cc1ncc(s1)S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
Cn1cnc(c1)S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)c3cccs3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)C3(C)CC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CCS(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)CC(F)(F)F)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)C(F)(F)F)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
Cc1nc(C)c(s1)S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)CC3CCCCC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
Cc1noc(C)c1S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CCCS(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)c3ccccc3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)CCl)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)c3ccc(Cl)s3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)Cc3ccccn3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)Cc3cccnc3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)CS(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
Cn1cc(c(n1)C(F)(F)F)S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)Cc3ccccc3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)c3ccccc3C#N)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
Cc1c(cnn1C(F)F)S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)CC(F)(F)F)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CCC1CC1S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CCOCCS(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)CC3CCCCO3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)CC3CC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CCC1CC1S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
Cc1noc(C)c1S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CCCS(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)c3ccccc3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)CS(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@H](CNS(=O)(=O)CC(F)(F)F)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CN(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1)S(C)(=O)=O
CC(C)(OC(=O)Nc1ccc2O[C@@H](CN3CCCS3(=O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
CN(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1)S(C)(=O)=O |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)N1CCC(CC1)C(F)(F)F
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)N1CCC(C1)C(F)(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)N1CCCC(C1)C(F)(F)F |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)N1CCC(F)CC1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)cc(F)c2O1)S(=O)(=O)c1ccc(F)cc1
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)cc(F)c2O1)S(=O)(=O)c1ccc(F)cc1
Cc1nn(cc1S(=O)(=O)N1C[C@H](CNS(C)(=O)=O)Oc2c(F)cc(NC(=O)OC(C)(C)C)cc12)C(F)F |r|
CC(C)(C)OC(=O)Nc1cc(F)c2O[C@@H](CNS(=O)(=O)C3CC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
Cc1nn(cc1S(=O)(=O)N1C[C@H](CNS(=O)(=O)C2CC2)Oc2c(F)cc(NC(=O)OC(C)(C)C)cc12)C(F)F |r|
CC(C)(C)OC(=O)Nc1cc(F)c2O[C@@H](CNS(C)(=O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)cc(F)c2O1)S(=O)(=O)c1ccc(F)c(F)c1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)cc(F)c2O1)S(=O)(=O)c1ccc(F)c(F)c1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)cc(Cl)c2O1)S(=O)(=O)c1ccc(F)cc1
CC(C)(OC(=O)Nc1cc(Cl)c2O[C@@H](CNS(C)(=O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
C[C@@H]1[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc2N1S(=O)(=O)c1ccc(F)cc1
C[C@@H]1[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1ccc(F)cc1
C[C@@H]1[C@@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc2N1S(=O)(=O)c1ccc(F)cc1
C[C@H]1[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc2N1S(=O)(=O)c1ccc(F)cc1
C[C@@H]1[C@@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1ccc(F)cc1 |r|
C[C@H]1[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1ccc(F)cc1 |r|
CC[C@H]1[C@@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1ccc(F)cc1 |r|
CCOc1nn(CC)cc1S(=O)(=O)N1[C@H](C)[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
C[C@H]1[C@@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1cn(nc1C)C(F)F |r|
C[C@@H]1[C@H](CNC(=O)C(C)(C)O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1ccc(F)cc1 |r|
C[C@@H]1[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1cn(nc1C)C(F)F |r|
CCc1nc(c(OCC(F)(F)F)s1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1ccc(cn1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1scnc1C |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cncc(F)c1 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1nccn1C |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1nc(C)sc1C |r|
CCc1ncc(s1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1c(C)nn(CCC(F)(F)F)c1C |r|
CCOc1sc(CC)nc1S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1sc(nc1S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C1CC1 |r|
CCOc1sc(nc1S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(F)(F)F |r|
CCc1nc(c(OC(C)C)s1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OC[C@@H](O)CO)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OC[C@H](C)O)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCCOC)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCC(C)(C)CO)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1c(OCc2ccccc2)nn2CCCCc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(CCNC(=O)OC(C)(C)C)nc1C |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cnn(CCNC(=O)OC(C)(C)C)c1C |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1c(Cl)nc2ccccn12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccnn1C |r|
C[C@@H](O)COc1nn2CCCCc2c1S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
C[C@H](O)COc1nn2CCCCc2c1S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)[C@@H]3C[C@@H]3C#N)CN(c2c1)S(=O)(=O)c1cn(nc1OCCO)C(F)F)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)CC(F)(F)F)CN(c2c1)S(=O)(=O)c1cn(nc1OCCO)C(F)F)C(F)(F)F |r|
CC(C)(O)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1OCCO)C(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C(C)(N)C(F)(F)F)CN(c2c1)S(=O)(=O)c1cn(nc1OCCO)C(F)F)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)[C@H]3C[C@H]3F)CN(c2c1)S(=O)(=O)c1cn(nc1OCCO)C(F)F)C(F)(F)F |r|
CC(C)n1cc(c(OCCO)n1)S(=O)(=O)N1C[C@H](CNC(=O)C(C)(C)O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1OCCO)C1CC1 |r|
CC(C)(O)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1OCCO)C1CC1 |r|
CC(C)(O)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1c(OCCO)nn2ccccc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)C3COC3)CN(c2c1)S(=O)(=O)c1cn(nc1OCCO)C(F)F)C(F)(F)F |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@H](CNS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1OCCO)C(F)F |r|
CC(C)n1cc(c(OCCO)n1)S(=O)(=O)N1C[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1c(OCCO)nn2ccccc12 |r|
CCn1cc(c(OCC(=O)OC)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@H](NC(C)=O)C1CC1 |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@H](NC(C)=O)C1CC1 |r|
CCn1cc(c(OCC(=O)OC)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@@H](NC(C)=O)C1CC1 |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(NC(C)=O)C1CC1 |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@H](NC(=O)C(C)(C)O)C1CC1 |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@@H](NC(=O)C(C)(C)O)C1CC1 |r|
CCn1cc(c(OCC(=O)OC)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@H](NC(=O)C(C)(C)O)C1CC1 |r|
CCn1cc(c(OCC(=O)OC)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@@H](NC(=O)C(C)(C)O)C1CC1 |r|
C[C@H](NC(C)=O)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1OCCO)C(F)F |r|
CC[C@@H](NC(C)=O)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC[C@H](NC(C)=O)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CCOc1nn(cc1S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@@H](C)NC(C)=O)C(F)F |r|
CCOc1nn(cc1S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@H](C)NC(C)=O)C(F)F |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@@H](C)NC(C)=O |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@H](C)NC(C)=O |r|
CC(C)n1cc(c(C)n1)S(=O)(=O)N1C[C@H](CNC(=O)C(C)(C)O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)n1ncc(c1C)S(=O)(=O)N1C[C@H](CNC(=O)C(C)(C)O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
Cc1nn(cc1S(=O)(=O)N1C[C@H](CNC(=O)C(C)(C)O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C1CC1 |r|
Cc1c(cnn1C1CC1)S(=O)(=O)N1C[C@H](CNC(=O)C(C)(C)O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(O)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1c(Cl)nc2sccn12 |r|
CC(C)(O)C(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)S(F)(F)(F)(F)F |r|
Cn1nccc1S(=O)(=O)N1C[C@H](CNC(=O)C(C)(C)O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCNc1nn(CC)cc1S(=O)(=O)N1C[C@H](CNC(=O)C(C)(C)O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
Cc1nn(cc1S(=O)(=O)N1C[C@H](CNC(=O)C(C)(C)O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)C3CC3)CN(c2c1)S(=O)(=O)c1cccc(c1)S(F)(F)(F)(F)F)C(F)(F)F |r|
C[C@@H]1[C@H](CNS(C)(=O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1cn(nc1C)C(F)F |r|
CCS(=O)(=O)NC[C@@H]1Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N([C@@H]1C)S(=O)(=O)c1cn(nc1C)C(F)F |r|
C[C@@H]1[C@H](CNS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1cn(nc1C)C(F)F |r|
C[C@@H]1[C@H](CNS(=O)(=O)CC(F)(F)F)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1cn(nc1C)C(F)F |r|
C[C@@H]1[C@H](CNC(=O)C(C)(C)O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1cn(nc1C)C(F)F |r|
C[C@@H]1[C@H](CNC(=O)[C@H]2C[C@H]2F)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1cn(nc1C)C(F)F |r|
C[C@@H]1[C@H](CNC(=O)C(C)(N)C(F)(F)F)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1cn(nc1C)C(F)F |r|
C[C@@H]1[C@H](CNC(=O)C(C)(O)C(F)(F)F)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1cn(nc1C)C(F)F |r|
C[C@@H]1[C@H](CNC(=O)[C@H]2C[C@@H]2C#N)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1cn(nc1C)C(F)F |r|
C[C@@H]1[C@H](CNC(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1cn(nc1C)C(F)F |r|
C[C@@H]1[C@H](CNC(=O)[C@H]2C[C@H]2F)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1cn(nc1OCCO)C(F)F |r|
C[C@@H]1[C@H](CNS(C)(=O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1cn(nc1OCCO)C(F)F |r|
CCOc1nn(CC)cc1S(=O)(=O)N1[C@H](C)[C@H](CNS(C)(=O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC)cc1S(=O)(=O)N1[C@H](C)[C@H](CNC(=O)[C@H]2C[C@H]2F)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC)cc1S(=O)(=O)N1[C@H](C)[C@H](CNC(=O)[C@@H]2C[C@@H]2C#N)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC)cc1S(=O)(=O)N1[C@H](C)[C@H](CNC(=O)C(C)(C)O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1[C@H](C)[C@H](CNS(C)(=O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1[C@H](C)[C@H](CNC(=O)[C@H]2C[C@H]2F)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1[C@H](C)[C@H](CNC(=O)[C@@H]2C[C@@H]2C#N)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1[C@H](C)[C@H](CNC(=O)C(C)(C)O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1[C@H](C)[C@H](CNC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
C[C@H](NC(C)=O)[C@@H]1Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N([C@@H]1C)S(=O)(=O)c1ccc(F)c(F)c1
CC(=O)N[C@@H]([C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
CC(=O)N[C@H]([C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
CC(=O)N[C@@H]([C@@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
CC(=O)N[C@H]([C@@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
CC[C@@H]1N(C[C@H]2CC[C@@H](CC2)C(F)(F)F)Cc2cc(cnc12)C(=O)N[C@@H](COC)c1ccc(cc1)S(=O)(=O)CC |r,wU:25.27,8.11,wD:2.1,5.4,(-5.94,-18.02,;-4.43,-17.7,;-3.95,-16.24,;-4.86,-14.99,;-6.4,-14.99,;-7.17,-13.66,;-6.4,-12.33,;-7.17,-10.99,;-8.71,-10.99,;-9.48,-12.33,;-8.71,-13.66,;-9.48,-9.66,;-8.71,-8.32,;-11.02,-9.66,;-10.25,-8.32,;-3.95,-13.75,;-2.49,-14.22,;-1.16,-13.45,;.18,-14.22,;.18,-15.76,;-1.16,-16.53,;-2.49,-15.76,;1.51,-13.45,;1.51,-11.91,;2.85,-14.22,;4.18,-13.45,;4.18,-11.91,;5.51,-11.14,;5.51,-9.6,;5.51,-14.22,;5.51,-15.76,;6.85,-16.53,;7.91,-15.61,;8.18,-14.22,;6.85,-13.45,;9.11,-16.3,;8.42,-17.5,;9.8,-15.1,;10.3,-16.99,;11.5,-16.3,)|
CC[C@@H]1N(C[C@H]2CC[C@@H](CC2)C(F)(F)F)Cc2cc(cnc12)C(=O)N[C@@H](COC(N)=O)c1ccc(cc1)S(=O)(=O)CC |r,wU:25.27,8.11,wD:2.1,5.4,(-1.61,-24.6,;-.1,-24.28,;.38,-22.82,;-.53,-21.57,;-2.07,-21.57,;-2.84,-20.24,;-2.07,-18.91,;-2.84,-17.57,;-4.38,-17.57,;-5.15,-18.91,;-4.38,-20.24,;-5.15,-16.24,;-4.38,-14.9,;-6.69,-16.24,;-5.92,-14.9,;.38,-20.33,;1.84,-20.8,;3.17,-20.03,;4.51,-20.8,;4.51,-22.34,;3.17,-23.11,;1.84,-22.34,;5.84,-20.03,;5.84,-18.49,;7.18,-20.8,;8.51,-20.03,;8.51,-18.49,;9.84,-17.72,;9.84,-16.07,;11.27,-15.25,;8.41,-15.25,;9.84,-20.8,;9.84,-22.34,;11.18,-23.11,;12.51,-22.34,;12.51,-20.8,;11.18,-20.03,;13.84,-23.11,;13.02,-24.54,;14.67,-24.54,;15.27,-22.29,;16.7,-23.11,)|
CC[C@@H]1N(C[C@H]2CC[C@@H](OC2)C(F)(F)F)Cc2cc(cnc12)C(=O)N[C@@H](COC)c1ccc(cc1)S(=O)(=O)CC |r|
CC[C@@H]1N(C[C@@H]2CC[C@H](OC2)C(F)(F)F)Cc2cc(cnc12)C(=O)N[C@@H](COC)c1ccc(cc1)S(=O)(=O)CC |r|
CC[C@@H]1N(C[C@@H]2CC[C@@H](OC2)C(F)(F)F)Cc2cc(cnc12)C(=O)N[C@@H](COC)c1ccc(cc1)S(=O)(=O)CC |r|
CC[C@@H]1N(C[C@H]2CC[C@H](OC2)C(F)(F)F)Cc2cc(cnc12)C(=O)N[C@@H](COC)c1ccc(cc1)S(=O)(=O)CC |r|
CCOC[C@H](NC(=O)c1cnc2[C@H](CC)N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)Cc2c1)c1ccc(cc1)S(=O)(=O)CC |r,wU:20.23,4.4,wD:17.16,12.12,(6.93,4.75,;5.6,3.98,;5.6,2.44,;4.26,1.67,;4.26,.13,;2.93,-.64,;1.6,.13,;1.6,1.67,;.26,-.64,;.26,-2.18,;-1.07,-2.95,;-2.4,-2.18,;-3.87,-2.66,;-4.64,-3.99,;-5.97,-4.76,;-4.77,-1.41,;-6.31,-1.41,;-7.08,-.08,;-6.31,1.26,;-7.08,2.59,;-8.62,2.59,;-9.39,1.26,;-8.62,-.08,;-9.39,3.93,;-8.62,5.26,;-10.93,3.93,;-10.16,5.26,;-3.87,-.16,;-2.4,-.64,;-1.07,.13,;5.6,-.64,;5.6,-2.18,;6.93,-2.95,;8.31,-2.21,;8.27,-.64,;6.93,.13,;9.65,-2.98,;8.88,-4.31,;10.42,-1.64,;10.98,-3.75,;12.31,-2.98,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](COC)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@H]3CC[C@H](CC3)C(F)(F)F)Cc2c1 |r,wU:31.35,28.28,11.15,wD:22.23,(12.31,-2.95,;10.98,-3.72,;9.65,-2.95,;8.88,-4.28,;10.42,-1.61,;8.31,-2.18,;6.93,-2.92,;5.6,-2.15,;5.6,-.61,;6.93,.16,;8.27,-.61,;4.26,.16,;4.26,1.7,;2.93,2.47,;2.93,4.01,;2.93,-.61,;1.6,.16,;1.6,1.7,;.26,-.61,;.26,-2.15,;-1.07,-2.92,;-2.4,-2.15,;-3.87,-2.62,;-4.64,-3.96,;-5.97,-4.73,;-3.87,-5.29,;-4.77,-1.38,;-6.31,-1.38,;-7.08,-.04,;-8.62,-.04,;-9.39,1.29,;-8.62,2.62,;-7.08,2.62,;-6.31,1.29,;-9.39,3.96,;-8.62,5.29,;-10.93,3.96,;-10.16,5.29,;-3.87,-.13,;-2.4,-.61,;-1.07,.16,)|
CCS(=O)(=O)c1ccc(nc1)[C@@H](COC(N)=O)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@H]3CC[C@H](CC3)C(F)(F)F)Cc2c1 |r,wU:33.37,30.30,wD:11.17,24.25,(12.31,-2.95,;10.98,-3.72,;9.65,-2.95,;8.88,-4.28,;10.42,-1.61,;8.31,-2.18,;8.27,-.61,;6.93,.16,;5.6,-.61,;5.6,-2.15,;6.93,-2.92,;4.26,.16,;4.26,1.7,;5.6,2.47,;5.6,4.01,;6.93,4.78,;4.27,4.78,;2.93,-.61,;1.6,.16,;1.6,1.7,;.26,-.61,;.26,-2.15,;-1.07,-2.92,;-2.4,-2.15,;-3.87,-2.62,;-4.64,-3.96,;-5.97,-4.73,;-3.87,-5.29,;-4.77,-1.38,;-6.31,-1.38,;-7.08,-.04,;-8.62,-.04,;-9.39,1.29,;-8.62,2.62,;-7.08,2.62,;-6.31,1.29,;-9.39,3.96,;-8.62,5.29,;-10.93,3.96,;-10.16,5.29,;-3.87,-.13,;-2.4,-.61,;-1.07,.16,)|
CCS(=O)(=O)c1ccc(nc1)[C@H](COC(N)=O)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)Cc2c1 |r,wU:33.37,11.17,wD:30.30,24.25,(12.31,-2.95,;10.98,-3.72,;9.65,-2.95,;8.88,-4.28,;10.42,-1.61,;8.31,-2.18,;8.27,-.61,;6.93,.16,;5.6,-.61,;5.6,-2.15,;6.93,-2.92,;4.26,.16,;4.26,1.7,;5.6,2.47,;5.6,4.01,;6.93,4.78,;4.27,4.78,;2.93,-.61,;1.6,.16,;1.6,1.7,;.26,-.61,;.26,-2.15,;-1.07,-2.92,;-2.4,-2.15,;-3.87,-2.62,;-4.64,-3.96,;-5.97,-4.73,;-3.87,-5.29,;-4.77,-1.38,;-6.31,-1.38,;-7.08,-.04,;-6.31,1.29,;-7.08,2.62,;-8.62,2.62,;-9.39,1.29,;-8.62,-.04,;-9.39,3.96,;-8.62,5.29,;-10.93,3.96,;-10.16,5.29,;-3.87,-.13,;-2.4,-.61,;-1.07,.16,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](COC(N)=O)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@H]3CC[C@H](CC3)C(F)(F)F)Cc2c1 |r,wU:33.37,30.30,11.17,wD:24.25,(12.31,-2.95,;10.98,-3.72,;9.65,-2.95,;8.88,-4.28,;10.42,-1.61,;8.31,-2.18,;6.93,-2.92,;5.6,-2.15,;5.6,-.61,;6.93,.16,;8.27,-.61,;4.26,.16,;4.26,1.7,;5.6,2.47,;5.6,4.01,;6.93,4.78,;4.27,4.78,;2.93,-.61,;1.6,.16,;1.6,1.7,;.26,-.61,;.26,-2.15,;-1.07,-2.92,;-2.4,-2.15,;-3.87,-2.62,;-4.64,-3.96,;-5.97,-4.73,;-3.87,-5.29,;-4.77,-1.38,;-6.31,-1.38,;-7.08,-.04,;-8.62,-.04,;-9.39,1.29,;-8.62,2.62,;-7.08,2.62,;-6.31,1.29,;-9.39,3.96,;-8.62,5.29,;-10.93,3.96,;-10.16,5.29,;-3.87,-.13,;-2.4,-.61,;-1.07,.16,)|
CCS(=O)(=O)c1ccc(cc1)[C@@H](COC(N)=O)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)Cc2c1 |r,wU:33.37,wD:30.30,11.17,24.25,(12.31,-2.95,;10.98,-3.72,;9.65,-2.95,;8.88,-4.28,;10.42,-1.61,;8.31,-2.18,;6.93,-2.92,;5.6,-2.15,;5.6,-.61,;6.93,.16,;8.27,-.61,;4.26,.16,;4.26,1.7,;5.6,2.47,;5.6,4.01,;6.93,4.78,;4.27,4.78,;2.93,-.61,;1.6,.16,;1.6,1.7,;.26,-.61,;.26,-2.15,;-1.07,-2.92,;-2.4,-2.15,;-3.87,-2.62,;-4.64,-3.96,;-5.97,-4.73,;-3.87,-5.29,;-4.77,-1.38,;-6.31,-1.38,;-7.08,-.04,;-6.31,1.29,;-7.08,2.62,;-8.62,2.62,;-9.39,1.29,;-8.62,-.04,;-9.39,3.96,;-8.62,5.29,;-10.93,3.96,;-10.16,5.29,;-3.87,-.13,;-2.4,-.61,;-1.07,.16,)|
CC[C@H]1N(C[C@H]2CC[C@@H](CC2)C(F)(F)F)Cc2cc(cnc12)C(=O)N[C@@H](COC(N)=O)c1ccc(cc1)S(=O)(=O)CC |r,wU:8.11,25.27,2.1,wD:5.4,(-5.97,-4.76,;-4.64,-3.99,;-3.87,-2.66,;-4.77,-1.41,;-6.31,-1.41,;-7.08,-.08,;-6.31,1.26,;-7.08,2.59,;-8.62,2.59,;-9.39,1.26,;-8.62,-.08,;-9.39,3.93,;-8.62,5.26,;-10.93,3.93,;-10.16,5.26,;-3.87,-.16,;-2.4,-.64,;-1.07,.13,;.26,-.64,;.26,-2.18,;-1.07,-2.95,;-2.4,-2.18,;1.6,.13,;1.6,1.67,;2.93,-.64,;4.26,.13,;4.26,1.67,;5.6,2.44,;5.6,3.98,;6.93,4.75,;4.27,4.75,;5.6,-.64,;5.6,-2.18,;6.93,-2.95,;8.31,-2.21,;8.27,-.64,;6.93,.13,;9.65,-2.98,;8.88,-4.31,;10.42,-1.64,;10.98,-3.75,;12.31,-2.98,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](COCC(O)=O)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)Cc2c1 |r,wU:31.31,11.18,wD:34.38,25.26,(12.31,-2.95,;10.98,-3.72,;9.65,-2.95,;8.88,-4.28,;10.42,-1.61,;8.31,-2.18,;6.93,-2.92,;5.6,-2.15,;5.6,-.61,;6.93,.16,;8.27,-.61,;4.26,.16,;4.26,1.7,;2.93,2.47,;2.93,4.01,;1.6,4.78,;1.6,6.32,;.26,4.01,;2.93,-.61,;1.6,.16,;1.6,1.7,;.26,-.61,;.26,-2.15,;-1.07,-2.92,;-2.4,-2.15,;-3.87,-2.62,;-4.64,-3.96,;-5.97,-4.73,;-3.87,-5.29,;-4.77,-1.38,;-6.31,-1.38,;-7.08,-.04,;-8.62,-.04,;-9.39,1.29,;-8.62,2.62,;-7.08,2.62,;-6.31,1.29,;-9.39,3.96,;-8.62,5.29,;-10.93,3.96,;-10.16,5.29,;-3.87,-.13,;-2.4,-.61,;-1.07,.16,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](COC)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)Cc2c1 |r,wU:31.35,11.15,wD:28.28,22.23,(12.31,-2.95,;10.98,-3.72,;9.65,-2.95,;8.88,-4.28,;10.42,-1.61,;8.31,-2.18,;6.93,-2.92,;5.6,-2.15,;5.6,-.61,;6.93,.16,;8.27,-.61,;4.26,.16,;4.26,1.7,;2.93,2.47,;2.93,4.01,;2.93,-.61,;1.6,.16,;1.6,1.7,;.26,-.61,;.26,-2.15,;-1.07,-2.92,;-2.4,-2.15,;-3.87,-2.62,;-4.64,-3.96,;-5.97,-4.73,;-3.87,-5.29,;-4.77,-1.38,;-6.31,-1.38,;-7.08,-.04,;-6.31,1.29,;-7.08,2.62,;-8.62,2.62,;-9.39,1.29,;-8.62,-.04,;-9.39,3.96,;-8.62,5.29,;-10.93,3.96,;-10.16,5.29,;-3.87,-.13,;-2.4,-.61,;-1.07,.16,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](COC(N)=O)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)Cc2c1 |r,wU:33.37,11.17,wD:30.30,24.25,(12.31,-2.95,;10.98,-3.72,;9.65,-2.95,;8.88,-4.28,;10.42,-1.61,;8.31,-2.18,;6.93,-2.92,;5.6,-2.15,;5.6,-.61,;6.93,.16,;8.27,-.61,;4.26,.16,;4.26,1.7,;5.6,2.47,;5.6,4.01,;6.93,4.78,;4.27,4.78,;2.93,-.61,;1.6,.16,;1.6,1.7,;.26,-.61,;.26,-2.15,;-1.07,-2.92,;-2.4,-2.15,;-3.87,-2.62,;-4.64,-3.96,;-5.97,-4.73,;-3.87,-5.29,;-4.77,-1.38,;-6.31,-1.38,;-7.08,-.04,;-6.31,1.29,;-7.08,2.62,;-8.62,2.62,;-9.39,1.29,;-8.62,-.04,;-9.39,3.96,;-8.62,5.29,;-10.93,3.96,;-10.16,5.29,;-3.87,-.13,;-2.4,-.61,;-1.07,.16,)|
C[C@@H]1CN(CC[C@@H]1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccnc12
C[C@H]1CN(CC[C@@H]1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccnc12
OC(=O)C1CCN(C1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
C[C@@H]1CN(CC[C@@H]1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
CC1(CCN(CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12)C(O)=O
OC1(CCN(CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12)C(F)(F)F
OC(=O)C1(CCN(CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12)c1ccccc1
OC(=O)[C@@H]1CC[C@@H](CC1)Nc1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12 |r,wU:6.9,3.2,(5.3,7.45,;5.77,5.99,;7.28,5.67,;4.74,4.84,;3.23,5.16,;2.2,4.02,;2.68,2.55,;4.19,2.23,;5.22,3.38,;1.65,1.41,;2.13,-.06,;1.22,-1.3,;2.13,-2.55,;1.65,-4.01,;2.68,-5.16,;.14,-4.33,;-.89,-3.19,;-.41,-1.72,;-2.39,-3.51,;-2.87,-4.97,;-1.84,-6.12,;-.33,-5.8,;.7,-6.94,;1.73,-8.09,;-.45,-7.97,;1.84,-5.91,;3.59,-2.07,;4.92,-2.84,;6.26,-2.07,;6.26,-.53,;4.92,.24,;4.92,1.78,;3.59,-.53,)|
OC(=O)C1CCN(CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
OC(=O)CC1CCN(CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
OC(=O)C1=CCN(CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccnc12 |t:3|
OC(=O)C1CCN(CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccnc12
OC(=O)C1(F)CCN(CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccnc12
OC(=O)C1CCN(CC1F)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccnc12
OC1(CCN(CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccnc12)C(F)(F)F
OC(=O)CC1CN(C1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccnc12
CN(C)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)N1CCC(CC1)C(O)=O
OCc1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)N1CCC(CC1)C(O)=O
Cc1cccc2n(nc(N3CCC(CC3)C(O)=O)c12)C(=O)c1c(Cl)cccc1C(F)(F)F
OC(=O)C1CCN(CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2cccc(F)c12
OC(=O)C1CCN(CC1)c1nn(C(=O)c2c(Cl)cccc2C2CCC2)c2cccc(F)c12
C[C@@H]1CN(CC[C@H]1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
OC(=O)C1CC2CCC(C1)N2c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12 |TLB:1:3:10:6.7|
OC(=O)C1C[C@@H]2CCC[C@H](C1)N2c1nn(Cc2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
CCC1CC(CCN1c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12)C(O)=O
OC(=O)C1(O)CCN(CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
O[C@H]1CN(CC[C@@H]1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2cccc(F)c12
c1cc(c(c(c1)Cl)C(=O)n2c3cccc(c3c(n2)N4CC[C@H]([C@@H](C4)O)C(=O)O)F)C5CC5
O[C@H]1CN(CC[C@@H]1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
O[C@@H]1CN(CC[C@H]1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
O[C@@H]1CN(CC[C@@H]1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
C[C@]1(CCN(C[C@@H]1O)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2cccc(F)c12)C(O)=O
C[C@@]1(CCN(C[C@@H]1O)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2cccc(F)c12)C(O)=O
C[C@]1(CCN(C[C@H]1O)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2cccc(F)c12)C(O)=O
OC(=O)C1CCN(c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cccc(F)c23)C(=O)C1
CC1CC(CCN1c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12)C(O)=O
COC1CN(C1)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)N1CCC(CC1)C(O)=O
C[C@H]1CCCN1C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)N1CCC(CC1)C(O)=O |r|
CO[C@H]1CCN(C1)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)N1CCC(CC1)C(O)=O |r|
CO[C@@H]1CCN(C1)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)N1CCC(CC1)C(O)=O |r|
CC(C)(O)C(=O)NNC(=O)C[C@@H]1CCc2cc(ccc2N1S(=O)(=O)c1ccc(F)cc1)C(O)(C(F)(F)F)C(F)(F)F |r|
OC(c1ccc2N([C@H](Cc3nnc(CC#N)o3)CCc2c1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F |r|
C\C(C[C@@H]1CCc2cc(ccc2N1S(=O)(=O)c1ccc(F)cc1)C(O)(C(F)(F)F)C(F)(F)F)=N/Oc1ccccc1 |r|
CCO\N=C(\C)C[C@@H]1CCc2cc(ccc2N1S(=O)(=O)c1ccc(F)cc1)C(O)(C(F)(F)F)C(F)(F)F |r|
CCON=C(C)CC1CCc2cc(ccc2N1S(=O)(=O)c1ccc(F)cc1)C(O)(C(F)(F)F)C(F)(F)F |w:3.2|
CSc1nnc(C[C@@H]2CCc3cc(ccc3N2S(=O)(=O)c2ccc(F)cc2)C(O)(C(F)(F)F)C(F)(F)F)s1 |r|
CS(=O)(=O)c1nnc(C[C@@H]2CCc3cc(ccc3N2S(=O)(=O)c2ccc(F)cc2)C(O)(C(F)(F)F)C(F)(F)F)s1 |r|
CC(C)(O)c1nnc(C[C@@H]2CCc3cc(ccc3N2S(=O)(=O)c2ccc(F)cc2)C(O)(C(F)(F)F)C(F)(F)F)o1 |r|
CC(C)(N)CC(=O)NNC(=O)C[C@@H]1CCc2cc(ccc2N1S(=O)(=O)c1ccc(F)cc1)C(O)(C(F)(F)F)C(F)(F)F |r|
CC(C)(N)CC(=O)NNC(=O)C[C@@H]1CCc2cc(ccc2N1S(=O)(=O)c1ccc(F)cc1)C(O)(C(F)(F)F)C(F)(F)F
OC(c1ccc2N([C@H](CC(=O)NNC(=O)c3ccncc3)CCc2c1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F |r|
NC1(CC1)c1nnc(C[C@@H]2CCc3cc(ccc3N2S(=O)(=O)c2ccc(F)cc2)C(O)(C(F)(F)F)C(F)(F)F)o1 |r|
OC(c1ccc2N([C@H](Cc3nnc(o3)-c3ccncc3)CCc2c1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F |r|
CC(=C)c1nnc(C[C@@H]2CCc3cc(ccc3N2S(=O)(=O)c2ccc(F)cc2)C(O)(C(F)(F)F)C(F)(F)F)o1
CC(O)(CO)c1nnc(C[C@@H]2CCc3cc(ccc3N2S(=O)(=O)c2ccc(F)cc2)C(O)(C(F)(F)F)C(F)(F)F)o1
CCC(O)Cn1ccc(C[C@@H]2CCc3cc(ccc3N2S(=O)(=O)c2ccc(F)cc2)C(O)(C(F)(F)F)C(F)(F)F)n1 |r|
OC(c1ccc2N([C@H](Cc3ccnn3Cc3ccc(F)cc3)CCc2c1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F |r|
OCC(O)Cc1nnc(C[C@@H]2CCc3cc(ccc3N2S(=O)(=O)c2ccc(F)cc2)C(O)(C(F)(F)F)C(F)(F)F)o1 |r|
OCC(O)Cn1nccc1C[C@@H]1CCc2cc(ccc2N1S(=O)(=O)c1ccc(F)cc1)C(O)(C(F)(F)F)C(F)(F)F |r|
OCC(O)Cn1ccc(C[C@@H]2CCc3cc(ccc3N2S(=O)(=O)c2ccc(F)cc2)C(O)(C(F)(F)F)C(F)(F)F)n1 |r|
OC(c1ccc2N([C@H](Cc3nnc(CC(=O)OCc4ccccc4)o3)CCc2c1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F |r|
CN(C)C(=O)Cc1nnc(C[C@@H]2CCc3cc(ccc3N2S(=O)(=O)c2ccc(F)cc2)C(O)(C(F)(F)F)C(F)(F)F)o1 |r|
NC(=O)Cc1nnc(C[C@@H]2CCc3cc(ccc3N2S(=O)(=O)c2ccc(F)cc2)C(O)(C(F)(F)F)C(F)(F)F)o1 |r|
OC(c1ccc2N([C@H](CNS(=O)(=O)c3ccc(F)cc3)CCc2c1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F |r|
OC(c1ccc2N([C@H](CNS(=O)(=O)c3ccc(Cl)nc3)CCc2c1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F |r|
OC(c1ccc2N([C@H](CNS(=O)(=O)C3CC3)CCc2c1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F |r|
CCOC(=O)CNC[C@@H]1CCc2cc(ccc2N1S(=O)(=O)c1ccc(F)cc1)C(O)(C(F)(F)F)C(F)(F)F |r|
OC(c1ccc2N([C@H](CNCc3ccccc3)CCc2c1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F |r|
OC(c1ccc2N(C(CNC(=O)NC3CC3)CCc2c1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
OC(c1ccc2N(C(CNC(=O)Nc3ccccc3)CCc2c1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
OC(c1ccc2N(C(CNC(=O)NCc3ccccc3)CCc2c1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
C\C=C\c1cccc(Cl)c1C(=O)n1nc(-c2ccc(cc2F)C(O)=O)c2ncccc12
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(C=O)c12
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3CC3)c3cccnc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3ccccn3)c3ccccc23)c(F)c1
CC(C(=O)n1nc(-c2ccc(cc2F)C(O)=O)c2ccccc12)c1ccccc1
COCC(=O)n1nc(-c2ccc(cc2F)C(O)=O)c2ccccc12
OC(=O)c1ccc(-c2nn(C(=O)c3cccnc3)c3ccccc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)CN3CCCC3=O)c3ccccc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3cccc4ccccc34)c3ccccc23)c(F)c1
Cn1c(cc2ccccc12)C(=O)n1nc(-c2ccc(cc2F)C(O)=O)c2ccccc12
Cc1cccc(C(=O)n2nc(-c3ccc(cc3F)C(O)=O)c3ccccc23)c1Br
OC(=O)c1ccc(-c2nn(C(=O)c3cccc4CCCc34)c3ccccc23)c(F)c1
CC(C)(C)OC(=O)N1CC2C(C1)C2C(=O)n1nc(-c2ccc(cc2F)C(O)=O)c2ccccc12
OC(=O)c1ccc(-c2nn(C(=O)c3cccc4CCOc34)c3ccccc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3cccc4ccoc34)c3ccccc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3cccc(Cl)c3Br)c3ccccc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)C3CCCO3)c3ccccc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C=C)c3cccnc23)c(F)c1
CC(=C)c1cccc(Cl)c1C(=O)n1nc(-c2ccc(cc2F)C(O)=O)c2ncccc12
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)ccc4OCCOc34)c3cccnc23)c(F)c1
CN(C)c1cccc(C)c1C(=O)n1nc(-c2ccc(cc2F)C(O)=O)c2ncccc12
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3CC3)c3cccc(Cl)c23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3CC3)c3cccc(F)c23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3CCC3)c3cccnc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3CC3)c3ccccc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3N3CCOCC3)c3cccnc23)c(F)c1
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)C(=O)N1CCOCC1
C[C@H]1CN(C[C@@H](C)O1)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(ccc23)C(=O)N2CCC(=O)CC2)c(F)c1
CC(=O)Nc1cc(ccc1C(O)=O)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2ccccc12
CS(=O)(=O)Nc1cc(ccc1C(O)=O)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccnc12
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(Br)ccc12
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(ccc23)N2CCC2)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(NC4CC4)ccc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(NC4COC4)ccc23)c(F)c1
OC1CCN(C1)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)N1CCOCC1
Nc1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
CN(C(C)=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(NC(=O)C4CC4)ccc23)c(F)c1
CS(=O)(=O)Nc1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
CNC(=O)Nc1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
CC(=O)Nc1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
CN(c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O)S(C)(=O)=O
CNC(=O)N(C)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(ccc23)N2CCNC2=O)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(Br)ccc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(ccc23)N2CCC2=O)c(F)c1
CN1CCN(C1=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(ccc23)N2CCCC2=O)c(F)c1
OC(=O)c1cnc2c(I)nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1
CON(C)C(=O)c1cnc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(cnc23)C(=O)NC2CC2)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(cnc23)C(=O)NCC2CC2)c(F)c1
CC1COCCN1C(=O)c1cnc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
CC1COCC(C)N1C(=O)c1cnc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OCc1cnc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OC(C1CC1)c1cnc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OC(c1ncco1)c1cnc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(cnc23)C(=O)c2ncco2)c(F)c1
OC(=O)c1ccc2c(I)nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1
Cc1cnc(o1)-c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)C#CCOC1CCCCO1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(ccc23)C#CCOC2CCCCO2)c(F)c1
NCC#Cc1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)C#C
Cc1noc(n1)-c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OCc1cnc(o1)-c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
Cn1cnc(c1)-c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(ccc23)-c2ncco2)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(ccc23)-c2ncc(Br)o2)c(F)c1
CN(C)C(=N/C#N)\c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(ccc23)-c2n[nH]c(=O)o2)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(ccc23)-c2nnc[nH]2)c(F)c1
Cc1nnc(o1)-c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
Cn1ccnc1-c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)-c1nccs1
Cn1cncc1-c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1)C(O)=O
Cc1cc(cs1)-c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1)C(O)=O
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)-c1ncccn1
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)-c1ccncn1
Cn1cnc(c1)-c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1)C(O)=O
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)-c1cscn1
NCc1ccnc(c1)-c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1)C(O)=O
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)-c1ccccn1
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)-c1cncs1
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)-c1cccnc1
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)-c1ccncc1
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)-c1ccc(cc1)C#N
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)-c1cccc(c1)C#N
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)-c1ccccc1C#N
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)-c1cccs1
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)-c1ccccc1F
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)-c1cccc(F)c1
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)-c1ccc(F)cc1
Cn1nccc1-c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1)C(O)=O
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)-c1ccc(O)cc1
CS(=O)(=O)NCc1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1)C(O)=O
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(ccc23)C2NC(=O)NC2=O)c(F)c1
CC(C)(C)OC(=O)Nc1cc2c(cn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2cn1)-c1ccc(cc1F)C(O)=O
CC(C)(C)OC(=O)Nc1cnc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
CNc1cnc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
CC(=O)Nc1cc2c(cn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2cn1)-c1ccc(cc1F)C(O)=O
CNc1cc2c(cn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2cn1)-c1ccc(cc1F)C(O)=O
COCCNc1cc2c(cn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2cn1)-c1ccc(cc1F)C(O)=O
Cc1c(-c2ccc(cc2F)C(O)=O)c2ccccc2n1C(=O)c1c(Cl)cccc1C(F)(F)F |(.45,-6.63,;-.89,-7.4,;-1.79,-6.15,;-1.39,-4.67,;-2.48,-3.58,;-2.08,-2.09,;-.6,-1.69,;.49,-2.78,;.09,-4.27,;1.18,-5.36,;-.2,-.2,;1.29,.2,;-1.29,.89,;-3.26,-6.63,;-4.59,-5.86,;-5.92,-6.63,;-5.92,-8.17,;-4.59,-8.94,;-3.26,-8.17,;-1.79,-8.65,;-1.39,-10.13,;-2.48,-11.22,;.09,-10.53,;1.18,-9.44,;.78,-7.95,;2.67,-9.84,;3.07,-11.33,;1.98,-12.42,;.49,-12.02,;-.6,-13.11,;-2.08,-12.71,;-.2,-14.6,;-1.69,-14.2,)|
Cc1c(-c2ccc(cc2)C(O)=O)c2ccccc2n1C(=O)c1ccccc1C(F)(F)F
OC(=O)c1cc(F)c(-c2nn(C(=O)c3c(Cl)cccc3C3CC3)c3cccnc23)c(F)c1 |(8.53,-.51,;7.04,-.91,;5.95,.18,;6.64,-2.4,;7.73,-3.49,;7.33,-4.98,;8.42,-6.07,;5.84,-5.38,;5.45,-6.86,;6.35,-8.11,;5.45,-9.35,;5.84,-10.84,;4.76,-11.93,;7.33,-11.24,;8.42,-10.15,;8.02,-8.66,;9.91,-10.55,;10.31,-12.04,;9.22,-13.13,;7.73,-12.73,;6.64,-13.82,;5.15,-14.22,;6.24,-15.3,;3.98,-8.88,;2.65,-9.65,;1.31,-8.88,;1.31,-7.34,;2.65,-6.57,;3.98,-7.34,;4.76,-4.29,;3.27,-4.68,;5.15,-2.8,)|
OC(=O)c1cc(F)c(-c2nn(C(=O)c3c(Cl)cccc3C3CC3)c3ccccc23)c(F)c1 |(2.72,7.05,;1.23,6.65,;.14,7.74,;.83,5.16,;-.66,4.77,;-1.06,3.28,;-2.54,2.88,;.03,2.19,;-.36,.7,;.54,-.54,;-.36,-1.79,;.03,-3.28,;-1.06,-4.37,;1.52,-3.68,;2.61,-2.59,;2.21,-1.1,;4.1,-2.99,;4.5,-4.47,;3.41,-5.56,;1.92,-5.16,;.83,-6.25,;-.66,-6.65,;.43,-7.74,;-1.83,-1.31,;-3.16,-2.08,;-4.5,-1.31,;-4.5,.23,;-3.16,1,;-1.83,.23,;1.52,2.59,;2.61,1.5,;1.92,4.08,)|
OC(=O)c1cc(F)c(-c2nn(C(=O)c3c(Cl)cccc3C3CC3)c3cccc(F)c23)c(F)c1 |(2.72,7.05,;1.23,6.65,;.14,7.74,;.83,5.16,;-.66,4.77,;-1.06,3.28,;-2.54,2.88,;.03,2.19,;-.36,.7,;.54,-.54,;-.36,-1.79,;.03,-3.28,;-1.06,-4.37,;1.52,-3.68,;2.61,-2.59,;2.21,-1.1,;4.1,-2.99,;4.5,-4.47,;3.41,-5.56,;1.92,-5.16,;.83,-6.25,;-.66,-6.65,;.43,-7.74,;-1.83,-1.31,;-3.16,-2.08,;-4.5,-1.31,;-4.5,.23,;-3.16,1,;-3.93,2.33,;-1.83,.23,;1.52,2.59,;2.61,1.5,;1.92,4.08,)|
OC(=O)c1cc(F)c(-c2cn(C(=O)c3c(Cl)cccc3C3CC3)c3cccnc23)c(F)c1 |(2.72,7.05,;1.23,6.65,;.14,7.74,;.83,5.16,;-.66,4.77,;-1.06,3.28,;-2.54,2.88,;.03,2.19,;-.36,.7,;.54,-.54,;-.36,-1.79,;.03,-3.28,;-1.06,-4.37,;1.52,-3.68,;2.61,-2.59,;2.21,-1.1,;4.1,-2.99,;4.5,-4.47,;3.41,-5.56,;1.92,-5.16,;.83,-6.25,;-.66,-6.65,;.43,-7.74,;-1.83,-1.31,;-3.16,-2.08,;-4.5,-1.31,;-4.5,.23,;-3.16,1,;-1.83,.23,;1.52,2.59,;2.61,1.5,;1.92,4.08,)|
OC(=O)c1cc(F)c(-c2nn(C(=O)c3c(Cl)cccc3C3CCC3)c3cccnc23)c(F)c1 |(-3.13,8,;-2.04,6.91,;-.56,7.31,;-2.44,5.42,;-1.37,4.28,;-1.77,2.79,;-.68,1.7,;-3.25,2.39,;-3.65,.91,;-2.75,-.34,;-3.65,-1.59,;-3.25,-3.07,;-4.34,-4.16,;-1.77,-3.47,;-.68,-2.38,;-1.08,-.9,;.81,-2.78,;1.21,-4.27,;.12,-5.36,;-1.37,-4.96,;-2.46,-6.05,;-4,-6.05,;-4,-7.59,;-2.46,-7.59,;-5.12,-1.11,;-6.45,-1.88,;-7.78,-1.11,;-7.78,.43,;-6.45,1.2,;-5.12,.43,;-4.34,3.48,;-5.83,3.08,;-3.94,4.97,)|
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(cnc23)C(=O)N2CCCOC2)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(cnc23)C(=O)N2CCOC2)c(F)c1
OC(=O)c1ccc(-c2cn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(ccc23)C(=O)N2CCC2)c(F)c1
COC1CN(C1)C(=O)c1ccc2c(cn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
NC(=O)Cc1cnc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(CC(=O)N4CCC4)cnc23)c(F)c1
CNC(=O)Cc1cnc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
CN(C)C(=O)Cc1cnc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(ccc23)C2COC2)c(F)c1
COCCOc1cc(C)c(C(=O)n2nc(-c3ccc(cc3F)C(O)=O)c3ncccc23)c(Cl)c1
Cc1cc(cc(Cl)c1C(=O)n1nc(-c2ccc(cc2F)C(O)=O)c2ncccc12)N1CCOCC1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(cnc23)C(=O)N(C2CC2)C2CC2)c(F)c1
CN(C)c1cc(C)c(C(=O)n2nc(-c3ccc(cc3F)C(O)=O)c3ncccc23)c(Cl)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3CCCC3)c3cccnc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3CCCCC3)c3cccnc23)c(F)c1
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2OC2CC2)c2ccccc12
OC1CN(C1)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1)C(O)=O
COC(=O)Nc1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OC(=O)CCNc1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cc(ccc12)C(O)=O
CN(C1CC1)C(=O)c1cnc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(cnc23)C(=O)C2CC2)c(F)c1
Cc1cnc(o1)-c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1)C([O-])=O
OCC#Cc1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1)C(O)=O
CC(O)C#Cc1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
CN(C)C(=N\C#N)\c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
COCCNc1cnc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1F)C(O)=O
Cc1cc(N)cc(Cl)c1C(=O)n1nc(-c2ccc(cc2F)C(O)=O)c2ncccc12
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCC(CO)(CC1)n1cnnc1 |r|
C[C@H]1CC[C@@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCC(CO)(CC1)n1cnnc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(OCC2CCOCC2)cc1F |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(OCC2CCS(=O)(=O)CC2)cc1 |r|
C[C@H]1CC[C@@](C)(c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCC(CC1)n1cnnc1 |r|
C[C@H]1CC[C@@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCC(CC1)n1cnnc1C |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CC[C@H](C[C@@H]1C)n1cnnc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(C[C@@H]1CO)C(C)=O |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCC(CC1)n1cnnc1C |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CC[C@@H](C[C@@H]1C)n1cnnc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCC(CC1)n1cnnc1CC#N |r|
COC(=O)[C@@H]1CN(CC[C@H]1n1cnnc1)c1ccc(CN2[C@@H](C)CC[C@H](c3ccccc3)S2(=O)=O)c(F)c1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)N1CCC(CC1)n1cnnc1 |r|
COCc1nncn1C1CCN(CC1)c1ccc(CN2[C@@H](C)CC[C@H](c3ccccc3)S2(=O)=O)c(F)c1 |r|
COC(=O)[C@H]1CN(CC[C@H]1n1cnnc1)c1ccc(CN2[C@@H](C)CC[C@H](c3ccccc3)S2(=O)=O)c(F)c1 |r|
C[C@H]1CN(CC[C@H]1n1cnnc1)c1ccc(CN2[C@@H](C)CC[C@H](c3ccccc3)S2(=O)=O)c(F)c1 |r|
C[C@@H]1CN(CC[C@@H]1n1cnnc1)c1ccc(CN2[C@@H](C)CC[C@H](c3ccccc3)S2(=O)=O)c(F)c1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(N2C[C@H]3[C@@H](C2)[C@@H]3n2cnnc2)c(F)c1F |r|
C[C@H]1CC[C@@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(N2C[C@H]3[C@@H](C2)[C@@H]3n2cnnc2)c(F)c1F |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(N2CCC(CC2)n2cnnc2)c(F)c1F |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)N1C[C@H]2[C@@H](C1)C2n1cnnc1 |r|
C[C@H]1CC[C@@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)N1C[C@H]2[C@@H](C1)C2n1cnnc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(N2C[C@H]3[C@@H](C2)[C@@H]3n2cnnc2)c(F)c1 |r|
C[C@@H]1CN(CC[C@H]1n1cnnc1)c1ccc(CN2[C@@H](C)CC[C@H](c3ccccc3)S2(=O)=O)c(F)c1 |r|
C[C@H]1CN(CC[C@@H]1n1cnnc1)c1ccc(CN2[C@@H](C)CC[C@H](c3ccccc3)S2(=O)=O)c(F)c1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CC2CC2C(C1)n1cnnc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(N2CCC(CC2)n2cnnc2)c(F)c1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)C1(CCN(CC1)C(C)=O)OC(N)=O |r|
C[C@H]1CC[C@@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(N2CCC(CC2)n2cnnc2)c(F)c1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1[C@H]2CC[C@@H]1C[C@H](C2)n1cnnc1 |r,THB:19:23:30.29.28:25.26|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1C[C@@H]2CC[C@H](C1)[C@@H]2n1cnnc1 |r|
C[C@H]1CC[C@@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1C[C@@H]2CC[C@H](C1)[C@@H]2n1cnnc1 |r|
COC(=O)[C@@H]1C[C@@H](CCN1c1ccc(CN2[C@@H](C)CC[C@H](c3ccccc3)S2(=O)=O)c(F)c1)n1cnnc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(OC2CCN(CC2)S(C)(=N)=O)cc1F |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(N2CC3[C@H](C2)[C@H]3n2cnnc2)c(F)c1 |r|
C[C@H]1CC[C@@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(N2CC3[C@H](C2)[C@H]3n2cnnc2)c(F)c1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CC[C@H]([C@H](CO)C1)n1cnnc1 |r|
C[C@H]1CCC(c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1)C12CCC(CC1)NC2=O |r,wD:1.0,(,-1.54,;1.33,-.77,;2.67,-1.54,;4,-.77,;4,.77,;5.33,1.54,;6.67,.77,;8,1.54,;8,3.08,;6.67,3.85,;5.33,3.08,;2.67,1.54,;1.9,2.87,;3.44,2.87,;1.33,.77,;,1.54,;-1.33,.77,;-2.67,1.54,;-4,.77,;-4,-.77,;-2.67,-1.54,;-1.33,-.77,;-5.33,-1.54,;-5.33,-3.08,;-6.67,-3.85,;-8,-3.08,;-6.9,-3.08,;-5.89,-2.5,;-8,-1.54,;-6.67,-.77,;-6.67,.77,)|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1C[C@@H]2C[C@H](C1)[C@H]2n1cnnc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CC[C@H]([C@@H](CO)C1)n1cnnc1 |r|
COC(=O)[C@H]1C[C@@H](CCN1c1ccc(CN2[C@@H](C)CC[C@H](c3ccccc3)S2(=O)=O)c(F)c1)n1cnnc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCC(CC1)n1cnnc1CO |r|
C[C@H]1CC[C@@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCC(CC1)n1cnnc1CO |r|
COC(=O)[C@@H]1C[C@H](CCN1c1ccc(CN2[C@@H](C)CC[C@H](c3ccccc3)S2(=O)=O)c(F)c1)n1cnnc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)c1ccc(cc1)C(O)=O |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)[N+]1([O-])CCC(CC1)n1cnnc1 |r,wU:4.4,wD:1.0,(1.85,-.53,;3.19,.24,;4.52,-.53,;5.85,.24,;5.85,1.78,;7.19,2.55,;8.52,1.78,;9.85,2.55,;9.85,4.09,;8.52,4.86,;7.19,4.09,;4.52,2.55,;3.75,3.88,;5.29,3.88,;3.19,1.78,;1.85,2.55,;.52,1.78,;.52,.24,;-.82,-.53,;-2.15,.24,;-2.15,1.78,;-.82,2.55,;-.82,4.09,;-3.48,-.53,;-3.48,1.01,;-4.82,.24,;-6.15,-.53,;-6.15,-2.07,;-4.82,-2.84,;-3.48,-2.07,;-7.48,-2.84,;-7.48,-4.38,;-8.95,-4.86,;-9.85,-3.61,;-8.95,-2.37,)|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCC2(CC1)OCCO2 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(N2CCN(CC2)C(C)=O)c(CO)c1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CC[C@@H]([C@H](CO)C1)n1cnnc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CC[C@@H]([C@@H](CO)C1)n1cnnc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)C1CCOCC1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCC2(CCCO2)CC1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCC2(CC1)OCCCO2 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCC2(CCO2)CC1 |r|
COC(=O)[C@@H]1CC2(CCN1c1ccc(CN3[C@@H](C)CC[C@H](c4ccccc4)S3(=O)=O)c(F)c1)OCCO2 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCOCC1 |r|
COC(=O)[C@H]1CC2(CCN1c1ccc(CN3[C@@H](C)CC[C@H](c4ccccc4)S3(=O)=O)c(F)c1)OCCO2 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCC[C@@H](C1)n1cnnc1 |r|
FC(F)[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCC(CC1)n1cnnc1 |r|
FC(F)[C@H]1CC[C@@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCC(CC1)n1cnnc1 |r|
FC(F)[C@H]1CC[C@@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)N1CCC(CC1)n1cnnc1 |r|
FC(F)[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)N1CCC(CC1)n1cnnc1 |r|
Fc1cc(N2CCC(CC2)n2cnnc2)c(F)cc1CN1[C@H](CC[C@@H](c2ccccc2)S1(=O)=O)C(F)(F)F |r|
Fc1cc(N2CCC(CC2)n2cnnc2)c(F)cc1CN1[C@H](CC[C@H](c2ccccc2)S1(=O)=O)C(F)(F)F |r|
Fc1cc(N2CC3[C@H](C2)[C@H]3n2cnnc2)c(F)cc1CN1[C@H](CC[C@H](c2ccccc2)S1(=O)=O)C(F)(F)F |r|
Fc1cc(N2CC3[C@H](C2)[C@H]3n2cnnc2)c(F)cc1CN1[C@H](CC[C@@H](c2ccccc2)S1(=O)=O)C(F)(F)F |r|
Fc1cc(ccc1CN1[C@H](CC[C@H](c2ccccc2)S1(=O)=O)C(F)(F)F)N1CCC(CC1)n1cnnc1 |r|
Fc1cc(ccc1CN1[C@H](CC[C@@H](c2ccccc2)S1(=O)=O)C(F)(F)F)N1CCC(CC1)n1cnnc1 |r|
Fc1cc(ccc1CN1[C@H](CC[C@H](c2ccccc2)S1(=O)=O)C(F)(F)F)N1CC2[C@H](C1)[C@H]2n1cnnc1 |r|
Fc1cc(ccc1CN1[C@H](CC[C@@H](c2ccccc2)S1(=O)=O)C(F)(F)F)N1C[C@H]2[C@@H](C1)[C@@H]2n1cnnc1 |r|
COC(=O)C1CN(CCC1n1cnnc1)c1cc(F)c(CN2C(C)CCC(c3ccccc3)S2(=O)=O)cc1F
COC1CN(CCC1n1cnnc1)c1ccc(CN2C(C)CCC(c3ccccc3)S2(=O)=O)c(F)c1
CC1CCC(c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)N1CC2CC1CC2n1cnnc1
CC1CCC(c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCC(C(F)C1)n1cnnc1
CC1CC2(CCN(CC2)c2ccc(CN3[C@@H](C)CC[C@H](c4ccccc4)S3(=O)=O)c(F)c2)OC1=O |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CC[C@H]([C@H](F)C1)n1cnnc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CC2(CCO2)C1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)C1Cc1ccc(cc1F)N1CCC2(CC1)N(C)C(=O)N(C)C2=O |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)C(O)C1CCN(CC1)C(C)=O |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CC[C@H]([C@@H](F)C1)n1cnnc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CC[C@@H]([C@H](F)C1)n1cnnc1 |r|
CO[C@H]1CN(CC[C@H]1n1cnnc1)c1ccc(CN2[C@@H](C)CC[C@H](c3ccccc3)S2(=O)=O)c(F)c1 |r|
CO[C@@H]1CN(CC[C@@H]1n1cnnc1)c1ccc(CN2[C@@H](C)CC[C@H](c3ccccc3)S2(=O)=O)c(F)c1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CC[C@@H]([C@@H](F)C1)n1cnnc1 |r|
C[C@H]1CCC(c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)c1ccc(C(O)=O)c(O)c1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)c1ccc(C(O)=O)c(O)c1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)N1C[C@@H]2C[C@H]1C[C@@H]2n1cnnc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)N1C[C@H]2C[C@@H]1C[C@H]2n1cnnc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(CC2=CCOCC2)cc1F |r,t:23|
[#6]-[#6@H]-1-[#6]-[#6]-[#6@H](-c2ccccc2)S(=O)(=O)[#7]-1-[#6]-c1ccc(\[#6]=[#6]-2/[#6]-[#6]-[#8]-[#6]-[#6]-2)cc1F |r|
COC(=O)C1CCOCC1c1cc(F)c(CN2[C@@H](C)CC[C@H](c3ccccc3)S2(=O)=O)cc1F |r|
COC(=O)[C@H]1CCOC[C@@H]1c1cc(F)c(CN2[C@@H](C)CC[C@H](c3ccccc3)S2(=O)=O)cc1F |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)N1CC[C@H]([C@H](O)C1)n1cnnc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)N1CC[C@H]([C@@H](O)C1)n1cnnc1 |r|
COC(=O)Cc1cc(F)c(CN2[C@@H](C)CC[C@H](c3ccccc3)S2(=O)=O)cc1F |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)C1COCCC1C(O)=O |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)[C@@H]1COCC[C@H]1C(O)=O |r|
COC(=O)[C@@H]1CCOC[C@H]1c1cc(F)c(CN2[C@@H](C)CC[C@H](c3ccccc3)S2(=O)=O)cc1F |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)N1CC[C@H]([C@@H](F)C1)n1cnnc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)N1CC[C@@H]([C@H](F)C1)n1cnnc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(CCO)cc1F |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(CC(=O)N[C@H]2C[C@H](O)C2)cc1F |r,wU:4.4,25.26,wD:1.0,27.29,(2.28,-1.93,;3.61,-1.15,;4.94,-1.92,;6.28,-1.15,;6.28,.38,;7.61,1.15,;8.95,.38,;10.28,1.15,;10.28,2.69,;8.95,3.46,;7.61,2.69,;4.94,1.15,;4.17,2.49,;5.71,2.49,;3.61,.38,;2.28,1.15,;.94,.38,;.94,-1.16,;-.39,-1.92,;-.39,-3.46,;-1.72,-1.16,;-3.06,-1.93,;-4.39,-1.16,;-4.39,.38,;-5.73,-1.93,;-7.06,-1.16,;-8.55,-1.55,;-8.95,-.07,;-10.28,.7,;-7.46,.33,;-1.72,.38,;-.39,1.15,;-.39,2.69,)|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(CC(N)=O)cc1F |r|
CC(CO)c1cc(F)c(CN2[C@@H](C)CC[C@H](c3ccccc3)S2(=O)=O)cc1F |r|
CCOC(=O)C(C(=O)OCC)c1cc(F)c(CN2[C@@H](C)CC[C@H](c3ccccc3)S2(=O)=O)cc1F |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)C(CO)CO |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(CC(=O)OC(C)(C)C)cc1F |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)C(CO)CCC#N |r|
CC(=O)N1CCN(CC1)c1ccc(CN2C3(CC3)CC[C@@H](c3ccccc3)S2(=O)=O)c(F)c1 |r|
CC(=O)N1CCN(CC1)c1ccc(CN2C3(CC3)CC[C@H](c3ccccc3)S2(=O)=O)c(F)c1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)C(C)(C)OCC(O)=O |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)C(C)(C)OCC(N)=O |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)C(CO)CC1COC1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)C(CO)CC#N |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)C(CO)CC(N)=O |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)C(CO)C1COC1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)C(C)(C)OCC(O)CO |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)C(CO)c1ccccc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)C(C)(C)OC[C@H](O)CO |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)C(C)(C)OC[C@@H](O)CO |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)C(CO)C1CCN(C)C1=O |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)C(CO)CCC(N)=O |r|
CC[C@@H](CC[C@H](c1ccccc1)S(=O)=O)NCc1cc(F)c(cc1F)N1CCC(CC1)N(C=N)C=N |r|
CC[C@H]1CC[C@@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)N1C[C@H]2[C@@H](C1)[C@@H]2n1cnnc1 |r|
CC[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)N1C[C@H]2[C@@H](C1)[C@@H]2n1cnnc1 |r|
CC1[C@H]2CC[C@@H](c3ccccc3)S(=O)(=O)N2Cc2c(F)cc(N3CCC(CC3)n3cnnc3)c(F)c12 |r|
CC[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1C[C@H]2[C@@H](C1)[C@@H]2n1cnnc1 |r|
CC[C@H]1CC[C@@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1C[C@H]2[C@@H](C1)[C@@H]2n1cnnc1 |r|
[H][C@@]12CN(C[C@]1([H])[C@H]2n1cnnc1)c1cc(F)c(CN2CCCC[C@@H](c3ccccc3)S2(=O)=O)cc1F |r|
Fc1cc(N2CCC(CC2)n2cnnc2)c(F)cc1CN1CCCC[C@@H](c2ccccc2)S1(=O)=O |r|
Fc1cc(N2CCC(CC2)n2cnnc2)c(F)cc1CN1CCCC[C@H](c2ccccc2)S1(=O)=O |r|
Fc1cc(N2C[C@H]3[C@@H](C2)[C@@H]3n2cnnc2)c(F)cc1CN1CCCC[C@H](c2ccccc2)S1(=O)=O |r|
Fc1cc(ccc1CN1CCCC[C@@H](c2ccccc2)S1(=O)=O)N1C[C@H]2[C@@H](C1)[C@@H]2n1cnnc1 |r|
Fc1cc(ccc1CN1CCCC[C@H](c2ccccc2)S1(=O)=O)N1C[C@H]2[C@@H](C1)[C@@H]2n1cnnc1 |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(cc1F)[C@H]1COCC[C@@H]1C(O)=O |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1cc(F)c(CC(=O)N[C@@H]2C[C@H](O)C2)cc1F |r,wU:4.4,25.26,27.29,wD:1.0,(2.28,-1.93,;3.61,-1.15,;4.94,-1.92,;6.28,-1.15,;6.28,.38,;7.61,1.15,;8.95,.38,;10.28,1.15,;10.28,2.69,;8.95,3.46,;7.61,2.69,;4.94,1.15,;4.17,2.49,;5.71,2.49,;3.61,.38,;2.28,1.15,;.94,.38,;.94,-1.16,;-.39,-1.92,;-.39,-3.46,;-1.72,-1.16,;-3.06,-1.93,;-4.39,-1.16,;-4.39,.38,;-5.73,-1.92,;-7.06,-1.15,;-7.46,.33,;-8.95,-.07,;-10.28,.7,;-8.55,-1.55,;-1.72,.38,;-.39,1.15,;-.39,2.69,)|
C[C@H]1CC[C@@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)c1ccc(cc1)C(O)=O |r|
C[C@H]1CC[C@@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)c1ccc(C(O)=O)c(O)c1 |r|
COc1nc2ccc(cc2c(Cl)c1CC1CCC(F)(F)CC1)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CC1CCC(F)(F)CC1)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CC1CCS(=O)(=O)CC1)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2nc(Cl)c(CN3CCOCC3)c(Cl)c2c1
COc1nc2ccc(cc2c(Cl)c1CC1CCOCC1)C(O)(C1CCN(CC1)C(C)=O)c1ccccc1
COc1nc2ccc(cc2c(Cl)c1CC1CCOCC1)[C@](O)(C1CCN(CC1)C(C)=O)c1ccccc1 |r|
COc1nc2ccc(cc2c(Cl)c1CC1CCOCC1)[C@@](O)(C1CCN(CC1)C(C)=O)c1ccccc1 |r|
COc1nc2ccc(cc2c(Cl)c1CC1CCOCC1)C(O)(C1CCN(CC1)C(C)=O)c1cncn1C
COc1nc2ccc(cc2c(Cl)c1CC1CCOCC1)[C@@](O)(C1CCN(CC1)C(C)=O)c1cncn1C |r|
COc1nc2ccc(cc2c(Cl)c1CC1CCOCC1)[C@](O)(C1CCN(CC1)C(C)=O)c1cncn1C |r|
COc1nc2ccc(cc2c(Cl)c1CC1CCOCC1)C(O)(C1CCN(CC1)S(C)(=O)=O)c1cncn1C
COc1nc2ccc(cc2c(Cl)c1CC1CCOCC1)[C@@](O)(C1CCN(CC1)S(C)(=O)=O)c1cncn1C |r|
COc1nc2ccc(cc2c(Cl)c1CC1CCOCC1)[C@](O)(C1CCN(CC1)S(C)(=O)=O)c1cncn1C |r|
COc1nc2ccc(cc2c(Cl)c1C1CCOCC1)C(O)(C1CCN(CC1)C(C)=O)c1ccccc1
COc1nc2ccc(cc2c(Cl)c1C1CCOCC1)[C@](O)(C1CCN(CC1)C(C)=O)c1ccccc1 |r|
COc1nc2ccc(cc2c(Cl)c1C1CCOCC1)[C@@](O)(C1CCN(CC1)C(C)=O)c1ccccc1 |r|
CCOC(=O)c1c(nc2ccc(cc2c1C(F)(F)F)C(O)(c1cccnc1)c1cccnc1)C(F)(F)F
CC(=O)N1CCC(CC1)C(O)(c1cncn1C)c1ccc2nc(c(C(=O)N3CCCCC3)c(c2c1)C(F)(F)F)C(F)(F)F
COc1cc2cc(ccc2nc1-c1ccccc1)C(O)(c1cnnn1C)c1sc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1C)C(O)(C1CCN(CC1)C(C)=O)c1ccccc1
COc1nc2ccc(cc2c(Cl)c1C)[C@@](O)(C1CCN(CC1)C(C)=O)c1ccccc1 |r|
COc1nc2ccc(cc2c(Cl)c1C)[C@](O)(C1CCN(CC1)C(C)=O)c1ccccc1 |r|
COc1nc2ccc(cc2c(Cl)c1C)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1C)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1C)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1C)C(O)(c1cnnn1C)c1sc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1C)[C@@](O)(c1cnnn1C)c1sc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1C)[C@](O)(c1cnnn1C)c1sc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CC1CC1)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1CC1CC1)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CC1CC1)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CC1CC1)C(O)(C1CCN(CC1)C(C)=O)c1ccccc1
COc1nc2ccc(cc2c(Cl)c1CC1CC1)[C@@](O)(C1CCN(CC1)C(C)=O)c1ccccc1 |r|
COc1nc2ccc(cc2c(Cl)c1CC1CC1)[C@](O)(C1CCN(CC1)C(C)=O)c1ccccc1 |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(O)(CC1)C(F)(F)F)C(O)(c1cncn1C)c1ccnc(c1)C(F)(F)F
COc1nc2ccc(cc2c(Cl)c1CN1CCN(CC(F)(F)F)CC1)[C@@](O)(c1cnnn1C)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCN(CC(F)(F)F)CC1)[C@](O)(c1cnnn1C)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1C)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F
CC(C)c1c(Cl)nc2ccc(cc2c1Cl)C(O)(c1cccnc1)c1cccc(Cl)c1
CC(C)c1c(Cl)c2cc(ccc2nc1-c1cncnc1)C(O)(c1cccnc1)c1cccc(Cl)c1
Cc1c(Cl)nc2ccc(cc2c1Cl)C(O)(c1cccnc1)c1cccc(Cl)c1
Cc1c(Cl)c2cc(ccc2nc1-c1cncnc1)C(O)(c1cccnc1)c1cccc(Cl)c1
CC(C)c1c(Cl)c2cc(ccc2nc1-c1ccsc1)C(O)(c1cccnc1)c1cccc(Cl)c1
Cc1c(Cl)c2cc(ccc2nc1-c1ccc2n(C)ncc2c1)C(O)(c1cccnc1)c1cccc(Cl)c1
Cc1c(Cl)c2cc(ccc2nc1-c1ccc2cnn(C)c2c1)C(O)(c1cccnc1)c1cccc(Cl)c1
CC(C)(C)c1c(Cl)nc2ccc(cc2c1Cl)C(O)(c1cccnc1)c1cccc(Cl)c1
CC(C)(C)c1c(\C=C\c2ccccc2)nc2ccc(cc2c1Cl)C(O)(c1cccnc1)c1cccc(Cl)c1
CC(C)(C)c1c(nc2ccc(cc2c1-c1ccco1)C(O)(c1cccnc1)c1cccc(Cl)c1)-c1ccco1
OC(c1cccnc1)(c1cccc(Cl)c1)c1ccc2nc(Cl)c(C3CCCCC3)c(Cl)c2c1
OC(c1cccnc1)(c1cccc(Cl)c1)c1ccc2nc(-c3cncnc3)c(C3CCCCC3)c(Cl)c2c1
Cn1cncc1C(O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(N3CCC3)c(OCc3ccccc3)c(Cl)c2c1
COc1nc2ccc(cc2c(Cl)c1CCC1CCN(CC1)C(C)=O)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F
COc1nc2ccc(cc2c(Cl)c1C1=CCN(C)CC1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |t:15|
COc1nc2ccc(cc2c(Cl)c1OCC1CCCO1)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1OC)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1OCC1(C)COC1)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1OCC1(C)COC1)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OCC1(C)COC1)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OCCN1CCOCC1)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1OCCN1CCOCC1)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
CC(C)Oc1c(Cl)c2cc(ccc2nc1N1CCC1)C(O)(c1cnnn1C)c1ccc(C)nc1C
CC(C)Oc1c(Cl)c2cc(ccc2nc1N1CCC1)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
CC(C)Oc1c(Cl)c2cc(ccc2nc1N1CCC1)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
Cn1cncc1C(O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(Cl)c(OCC(F)(F)F)c(Cl)c2c1
Cn1cncc1C(O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(Cl)c(OCC3CC3)c(Cl)c2c1
CC(C)Oc1c(Cl)nc2ccc(cc2c1Cl)C(O)(c1cnnn1C)c1cnc(C)n1C
CC(C)Oc1c(Cl)nc2ccc(cc2c1Cl)C(O)(c1cnnn1C)c1ccc(C)nc1C
CC(C)Oc1c(Cl)nc2ccc(cc2c1Cl)C(O)(c1cnnn1C)c1sc(C)nc1C
CC(C)Oc1c(Cl)nc2ccc(cc2c1Cl)C(O)(C1CCN(CC1)C(C)=O)c1ccccc1
Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2nc(Cl)c(OCC(F)(F)F)c(Cl)c2c1
CCOc1c(Cl)nc2ccc(cc2c1Cl)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F
CCOc1c(Cl)nc2ccc(cc2c1Cl)C(O)(c1cncn1C)c1ccc(Cl)nc1
CC(C)Oc1c(Cl)nc2ccc(cc2c1Cl)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F
CC(C)Oc1c(Cl)nc2ccc(cc2c1Cl)C(O)(c1cncn1C)c1ccc(Cl)nc1
CC(C)Oc1c(Cl)nc2ccc(cc2c1Cl)[C@](O)(c1cncn1C)c1ccc(Cl)nc1 |r|
CC(C)Oc1c(Cl)nc2ccc(cc2c1Cl)[C@@](O)(c1cncn1C)c1ccc(Cl)nc1 |r|
COc1nc2ccc(cc2c(Cl)c1OCC(C)(C)O)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1OCC(C)(C)O)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OCC(C)(C)O)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OC1CCCN(C)C1)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1OCC1CCCN1C)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1OCC1CCOC1)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1OCC(C)(C)O)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1OCC1CCO1)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1OCC1CC1(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1OC(C)C1CC1)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1OCc1cc(C)nn1C)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1OC1CCOCC1)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1OCC1COC1)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1OCC1(C)CC1)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1OCc1c(C)noc1C)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1OCC1(C)COC1)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1OCC1CC1)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1OC1CCN(C)CC1)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OCc1ncccn1)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1OCc1ncccn1)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OCc1ncccn1)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OCC1CC1)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1OCC1CC1)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OCC1CC1)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OC1CCOCC1)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1OC1CCOCC1)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OC1CCOCC1)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OCCS(C)(=O)=O)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1OCCS(C)(=O)=O)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OCc1c(C)noc1C)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1OCc1c(C)noc1C)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OCC1CC1(F)F)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1OCC1CC1(F)F)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OCC1CC1(F)F)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OCc1nccs1)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OCc1nccs1)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OCCN(C)C)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OCc1ccccc1)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
CC(C)Oc1c(Cl)c2cc(ccc2nc1N1CCC1)[C@](O)(c1cnnn1C)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1OCC1(C)COC1)[C@@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1OCC1(C)COC1)[C@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
COCCOc1c(OC)nc2ccc(cc2c1Cl)[C@@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
COCCOc1c(OC)nc2ccc(cc2c1Cl)[C@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1OC(C)C)C(O)(c1cnnn1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1OC(C)C)[C@](O)(c1cnnn1C)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1OC(C)C)[C@@](O)(c1cnnn1C)c1cnc(C)n1C |r|
CC(C)Oc1c(Cl)c2cc(ccc2nc1N1CCC1)C(O)(c1cnnn1C)c1sc(C)nc1C
CC(C)Oc1c(Cl)c2cc(ccc2nc1N1CCC1)[C@](O)(c1cnnn1C)c1sc(C)nc1C |r|
CC(C)Oc1c(Cl)c2cc(ccc2nc1N1CCC1)[C@@](O)(c1cnnn1C)c1sc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1C(=O)N1CCC(CC1)C(F)(F)F)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1OC(C)C)C(O)(C1CCN(CC1)C(C)=O)c1ccccc1
COc1nc2ccc(cc2c(Cl)c1OC(C)C)[C@@](O)(C1CCN(CC1)C(C)=O)c1ccccc1 |r|
COc1nc2ccc(cc2c(Cl)c1OC(C)C)[C@](O)(C1CCN(CC1)C(C)=O)c1ccccc1 |r|
COc1nc2ccc(cc2c(Cl)c1OC(C)C)[C@](O)(c1cnnn1C)c1sc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OC(C)C)[C@@](O)(c1cnnn1C)c1sc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OCC(F)(F)F)[C@](O)(c1cncn1C)c1ccc(Cl)cc1 |r|
COc1nc2ccc(cc2c(Cl)c1OCC(F)(F)F)[C@@](O)(c1cncn1C)c1ccc(Cl)cc1 |r|
Cn1cncc1[C@@](O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(N3CCC3)c(OCC3CC3)c(Cl)c2c1 |r|
Cn1cncc1[C@](O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(N3CCC3)c(OCC3CC3)c(Cl)c2c1 |r|
COc1nc2ccc(cc2c(Cl)c1OCC1CC1)[C@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1OCC1CC1)[C@@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
Cn1cncc1[C@@](O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(N3CCC3)c(OCC(F)(F)F)c(Cl)c2c1 |r|
Cn1cncc1[C@](O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(N3CCC3)c(OCC(F)(F)F)c(Cl)c2c1 |r|
Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2nc(N3CCC3)c(OCC(F)(F)F)c(Cl)c2c1
Cn1cncc1[C@@](O)(c1ccc(Cl)cc1)c1ccc2nc(N3CCC3)c(OCC(F)(F)F)c(Cl)c2c1 |r|
Cn1cncc1[C@](O)(c1ccc(Cl)cc1)c1ccc2nc(N3CCC3)c(OCC(F)(F)F)c(Cl)c2c1 |r|
CCOc1c(OC)nc2ccc(cc2c1Cl)[C@@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
CCOc1c(OC)nc2ccc(cc2c1Cl)[C@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
CCOc1c(OC)nc2ccc(cc2c1Cl)C(O)(c1cncn1C)c1ccc(Cl)cc1
CCOc1c(OC)nc2ccc(cc2c1Cl)[C@@](O)(c1cncn1C)c1ccc(Cl)cc1 |r|
CCOc1c(OC)nc2ccc(cc2c1Cl)[C@](O)(c1cncn1C)c1ccc(Cl)cc1 |r|
CC(C)Oc1c(Cl)c2cc(ccc2nc1N1CCC1)[C@@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
CC(C)Oc1c(Cl)c2cc(ccc2nc1N1CCC1)[C@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
CC(C)Oc1c(Cl)c2cc(ccc2nc1N1CCC1)[C@](O)(c1cncn1C)c1ccc(Cl)cc1 |r|
CC(C)Oc1c(Cl)c2cc(ccc2nc1N1CCC1)[C@@](O)(c1cncn1C)c1ccc(Cl)cc1 |r|
COc1nc2ccc(cc2c(Cl)c1OC(C)C)[C@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1OC(C)C)[C@@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
COc1nc2ccc(cc2c(OC)c1OCC(F)(F)F)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F
COc1nc2ccc(cc2c(Cl)c1OC)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F
COc1nc2ccc(cc2c(Cl)c1OCC(F)(F)F)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F
COc1nc2ccc(cc2c(Cl)c1OC(C)C)[C@](O)(c1cncn1C)c1ccc(Cl)cc1 |r|
COc1nc2ccc(cc2c(Cl)c1OC(C)C)[C@@](O)(c1cncn1C)c1ccc(Cl)cc1 |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)n1cccn1)C(O)(c1cncn1C)c1ccc(Cl)cc1
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)n1cccn1)[C@](O)(c1cncn1C)c1ccc(Cl)cc1 |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)n1cccn1)[C@@](O)(c1cncn1C)c1ccc(Cl)cc1 |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)n1cccn1)C(O)(C1CCN(CC1)C(C)=O)c1ccccc1
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)n1cccn1)[C@@](O)(C1CCN(CC1)C(C)=O)c1ccccc1 |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)n1cccn1)[C@](O)(C1CCN(CC1)C(C)=O)c1ccccc1 |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)n1cccn1)[C@@](O)(c1cnnn1C)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)n1cccn1)[C@](O)(c1cnnn1C)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)n1cccn1)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)n1cccn1)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@@](O)(c1cnnn1C)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@](O)(c1cnnn1C)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(F)(F)CC1)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1CN1CCC(F)(F)CC1)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(F)(F)CC1)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(F)CC1)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(F)CC1)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CC(F)(F)C1)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CC(F)(F)C1)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CC(F)C1)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CC(F)C1)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)C(O)(c1cnc(C)n1C)c1ncc(C)n1C
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1C(C)(C)CCCC1(C)C)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CC(C1)C(F)(F)F)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CC(C1)C(F)(F)F)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)S(C)(=O)=O)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)C(O)(C1CCN(CC1)C(C)=O)c1ccccc1
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@@](O)(C1CCN(CC1)C(C)=O)c1ccccc1 |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@](O)(C1CCN(CC1)C(C)=O)c1ccccc1 |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@@](O)(c1cnnn1C)c1cc(C)nc(C)c1 |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@](O)(c1cnnn1C)c1cc(C)nc(C)c1 |r|
COc1nc2ccc(cc2c(Cl)c1CN1CC(C1)C(F)(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1CN1CC(C1)C(F)(F)F)[C@](O)(c1cnnn1C)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CC(C1)C(F)(F)F)[C@@](O)(c1cnnn1C)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CC(C1)C(F)(F)F)[C@@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1CC(C1)C(F)(F)F)[C@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1CC(C1)C(F)(F)F)[C@@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1CC(C1)C(F)(F)F)[C@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@@](O)(C1CCOCC1)c1cnnn1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@](O)(C1CCOCC1)c1cnnn1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@@](O)(C1CN(C1)C(C)=O)c1cnnn1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@](O)(C1CN(C1)C(C)=O)c1cnnn1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@@](O)(C1CN(C1)C(C)=O)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@](O)(C1CN(C1)C(C)=O)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@@](O)(C1CN(C1)C(C)=O)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@](O)(C1CN(C1)C(C)=O)c1ccnc(c1)C(F)(F)F |r|
Cc1ncc(n1C)[C@](c2ccc3c(c2)c(c(c(n3)OC)CN4CCC(CC4)C(F)(F)F)Cl)(c5ccnc(c5)C(F)(F)F)O
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@](O)(c1cnc(C)n1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@@](O)(C1CN(C1)S(C)(=O)=O)c1cnnn1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@](O)(C1CN(C1)S(C)(=O)=O)c1cnnn1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@@](O)(C1CCOCC1)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@](O)(C1CCOCC1)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@@](O)(c1cnnn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@](O)(c1cnnn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@@](O)(C1CCOCC1)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@](O)(C1CCOCC1)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@@](O)(C1CN(C1)C(C)=O)c1ccc(nc1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@](O)(C1CN(C1)C(C)=O)c1ccc(nc1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1C(C)C)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1C(C)C)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1C(C)C)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CC(C)C)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1CC(C)C)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CC(C)C)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CC(C)C)C(O)(c1cnnn1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1CC(C)C)[C@@](O)(c1cnnn1C)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1CC(C)C)[C@](O)(c1cnnn1C)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1C1CCCC1)C(O)(c1cnnn1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1C1CCCC1)[C@@](O)(c1cnnn1C)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1C1CCCC1)[C@](O)(c1cnnn1C)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1C1CCCC1)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1C1CCCC1)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1C1CCCC1)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CC(F)(F)F)C(O)(c1cnnn1C)c1cnc(C)n1C
COc1c(CC(F)(F)F)c(Cl)nc2ccc(cc12)C(O)(c1cnnn1C)c1cnc(C)n1C
Cn1cncc1C(O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(N3CCC3)c(CC(F)(F)F)c(Cl)c2c1
Cn1cncc1[C@@](O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(N3CCC3)c(CC(F)(F)F)c(Cl)c2c1 |r|
Cn1cncc1[C@](O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(N3CCC3)c(CC(F)(F)F)c(Cl)c2c1 |r|
Cn1cncc1C(O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(Cl)c(CC(F)(F)F)c(N3CCC3)c2c1
Cn1cncc1[C@@](O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(Cl)c(CC(F)(F)F)c(N3CCC3)c2c1 |r|
Cn1cncc1[C@](O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(Cl)c(CC(F)(F)F)c(N3CCC3)c2c1 |r|
Cc1ccc(c(C)n1)C(O)(c1cnnn1C)c1ccc2nc(Cl)c(CC(F)(F)F)c(Cl)c2c1
Cc1ccc(c(C)n1)C(O)(c1cnnn1C)c1ccc2nc(N3CCC3)c(CC(F)(F)F)c(Cl)c2c1
Cc1ccc(c(C)n1)[C@@](O)(c1cnnn1C)c1ccc2nc(N3CCC3)c(CC(F)(F)F)c(Cl)c2c1 |r|
Cc1ccc(c(C)n1)[C@](O)(c1cnnn1C)c1ccc2nc(N3CCC3)c(CC(F)(F)F)c(Cl)c2c1 |r|
COc1nc2ccc(cc2c(Cl)c1CC(F)(F)F)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1CC(F)(F)F)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
Cc1ncc(n1C)C(O)(c1cnc(C)n1C)c1ccc2nc(Cl)c(CC(F)(F)F)c(Cl)c2c1
COc1nc2ccc(cc2c(Cl)c1CC(F)(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1C(=O)N1CCC(CC1)C(F)(F)F)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F
COc1nc2ccc(cc2c(Cl)c1C(=O)NCC1CC1)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1C(=O)N(C)C)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1C(=O)NC1CC1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F
COc1nc2ccc(cc2c(Cl)c1C(=O)NC1CC1)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1C(=O)N1CCCC1)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1C(=O)NCC(F)(F)F)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1C(=O)N1CC(F)(F)C1)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1OCC1CCOCC1)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1OCC1CCOCC1)[C@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OCC1CCOCC1)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OC(C)C)C(O)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1OC(C)C)C(O)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1CC(C)C)C(O)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1CC(C)C)C(O)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1C1CCCC1)C(O)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1OC(C)C)[C@@](C)(O)c1ccc(C)nc1C |r|
COc1nc2ccc(cc2c(Cl)c1OC(C)C)[C@](C)(O)c1ccc(C)nc1C |r|
CC(C)Oc1c(Cl)nc2ccc(cc2c1Cl)C(O)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1CN1CCC(O)(CC1)C(F)(F)F)[C@@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(O)(CC1)C(F)(F)F)[C@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CNC(=O)C1(CCC1)C(F)(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1CNC(=O)C1(CC1)C(F)(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1CNC(=O)CC(F)(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1CNC(=O)CCC(F)(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)C(O)c1ccc(cc1)C#N
COc1nc2ccc(cc2c(Cl)c1CN1CCn2nc(nc2C1)C(F)(F)F)[C@@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCn2nc(nc2C1)C(F)(F)F)[C@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCn2c(C1)nnc2C(F)(F)F)[C@@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCn2c(C1)nnc2C(F)(F)F)[C@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN(C)CC(F)(F)F)[C@@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN(C)CC(F)(F)F)[C@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@@](O)(c1cncn1C)c1ccc(cc1)C#N |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)[C@](O)(c1cncn1C)c1ccc(cc1)C#N |r|
COc1nc2ccc(cc2c(Cl)c1CNCCC(F)(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1CNCCOCC(F)(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1CNCCCC(F)(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)n1ccc(n1)C(F)(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
CCC(NCc1c(OC)nc2ccc(cc2c1Cl)C(O)(c1cnc(C)n1C)c1cnc(C)n1C)C(F)(F)F
COc1nc2ccc(cc2c(Cl)c1CN(C)CC(F)(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1CN[C@H](C)C(F)(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1CN[C@@H](C)C(F)(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C |r|
COc1nc2ccc(cc2c(Cl)c1CNC1CCCC(C1)C(F)(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
CC[C@@H](NCc1c(OC)nc2ccc(cc2c1Cl)C(O)(c1cnc(C)n1C)c1cnc(C)n1C)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CNCC1CCC(CC1)C(F)(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C |(4.42,-7.31,;4.42,-5.78,;3.08,-5,;1.75,-5.78,;.41,-5,;-.92,-5.78,;-2.25,-5,;-2.25,-3.47,;-1.07,-2.54,;.41,-3.47,;1.75,-2.69,;1.75,-1.15,;3.08,-3.47,;4.42,-2.69,;4.42,-1.15,;5.75,-.38,;5.75,1.15,;7.08,1.93,;7.08,3.47,;5.75,4.29,;4.42,3.47,;4.42,1.93,;5.75,5.83,;5.75,7.37,;7.29,5.83,;4.21,5.83,;-3.59,-2.69,;-4.36,-4.03,;-4.92,-1.93,;-6.38,-2.4,;-7.29,-1.15,;-6.38,.09,;-7.15,1.42,;-4.92,-.38,;-3.59,.38,;-2.82,-1.36,;-3.14,-.05,;-2.05,1.01,;-.8,.1,;.53,.87,;-1.28,-1.36,;-.51,-2.69,)|
COc1nc2ccc(cc2c(Cl)c1CNC(C)(C)C(F)(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
Cn1cncc1[C@@](O)(c1ccnc(c1)C(F)(F)F)c1ccc2nc(C3CC3)c(CN3CCC(CC3)C(F)(F)F)c(Cl)c2c1 |r|
Cn1cncc1[C@](O)(c1ccnc(c1)C(F)(F)F)c1ccc2nc(C3CC3)c(CN3CCC(CC3)C(F)(F)F)c(Cl)c2c1 |r|
COc1nc2ccc(cc2c(C#N)c1CC(F)(F)F)C(O)(c1cnnn1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1CC(F)(F)F)C(O)(c1cncn1C)c1ccc(cc1)C#N
COc1nc2ccc(cc2c(Cl)c1CC(F)(F)F)[C@](O)(c1cncn1C)c1ccc(cc1)C#N |r|
COc1nc2ccc(cc2c(Cl)c1CC(F)(F)F)[C@@](O)(c1cncn1C)c1ccc(cc1)C#N |r|
COc1nc2ccc(cc2c(C#N)c1OCC(F)(F)F)[C@@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
COc1nc2ccc(cc2c(C#N)c1OCC(F)(F)F)[C@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
COc1nc2ccc(cc2c(C#N)c1OCC1CC1)[C@@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(C#N)c1OCC1CC1)[C@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(C#N)c1OCC(F)(F)F)[C@@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(C#N)c1OCC(F)(F)F)[C@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(C#N)c1OCC(F)(F)F)C(O)(c1cncn1C)c1ccc(cc1)C#N
COc1nc2ccc(cc2c(C#N)c1OCC(F)(F)F)[C@](O)(c1cncn1C)c1ccc(cc1)C#N |r|
COc1nc2ccc(cc2c(C#N)c1OCC1CC1)[C@@](O)(c1cncn1C)c1ccc(cc1)C#N |r|
COc1nc2ccc(cc2c(C#N)c1OCC1CC1)[C@](O)(c1cncn1C)c1ccc(cc1)C#N |r|
COc1nc2ccc(cc2c(Cl)c1OCC(F)(F)F)[C@@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1OCC(F)(F)F)[C@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1OCC1CC1)[C@@](O)(c1cncn1C)c1ccc(cc1)C#N |r|
COc1nc2ccc(cc2c(Cl)c1OCC1CC1)[C@](O)(c1cncn1C)c1ccc(cc1)C#N |r|
COc1nc2ccc(cc2c(Cl)c1OCC1CC1)C(O)(c1cncn1C)c1ccc(Cl)cc1
COc1nc2ccc(cc2c(Cl)c1OCC1CC1)[C@@](O)(c1cncn1C)c1ccc(Cl)cc1 |r|
COc1nc2ccc(cc2c(Cl)c1OCC1CC1)[C@](O)(c1cncn1C)c1ccc(Cl)cc1 |r|
COc1nc2ccc(cc2c(Cl)c1OCC1CC1)[C@@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1OCC1CC1)[C@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(C#N)c1CC(F)(F)F)[C@@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(C#N)c1CC(F)(F)F)[C@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
CCc1nc2ccc(cc2c(C#N)c1OCC1CC1)[C@](O)(C1CN(C1)C(C)=O)c1cnnn1C |r|
CCc1nc2ccc(cc2c(C#N)c1OCC1CC1)[C@@](O)(C1CN(C1)C(C)=O)c1cnnn1C |r|
COc1nc2c(C)cc(cc2c(Cl)c1OCC(F)(F)F)C(O)(c1cnc(C)n1C)c1c(C)nn(C)c1C
COc1nc2ccc(cc2c(Cl)c1OCC(F)(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
CCc1nc2ccc(cc2c(Cl)c1OCC1CC1)C(O)(C1CN(C1)C(C)=O)c1cnnn1C
COc1nc2ccc(cc2c(Cl)c1CC(F)(F)F)[C@](O)(C1CN(C1)C(C)=O)c1cnnn1C |r|
COc1nc2ccc(cc2c(Cl)c1CC(F)(F)F)[C@@](O)(C1CN(C1)C(C)=O)c1cnnn1C |r|
CCc1nc2ccc(cc2c(CC)c1CC(F)(F)F)[C@@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
CCc1nc2ccc(cc2c(CC)c1CC(F)(F)F)[C@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CC(F)(F)F)[C@@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CC(F)(F)F)[C@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
CCc1nc2ccc(cc2c(C#N)c1CC(F)(F)F)[C@@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
CCc1nc2ccc(cc2c(C#N)c1CC(F)(F)F)[C@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
CCc1nc2ccc(cc2c(Cl)c1CC(F)(F)F)[C@@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
CCc1nc2ccc(cc2c(Cl)c1CC(F)(F)F)[C@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
Cc1ccc(c(C)n1)C(O)(c1cnnn1C)c1ccc2nc(Cl)c(CC(F)(F)F)c(N3CCC3)c2c1
Cc1ccc(c(C)n1)[C@](O)(c1cnnn1C)c1ccc2nc(Cl)c(CC(F)(F)F)c(N3CCC3)c2c1 |r|
Cc1ncc(n1C)C(O)(c1cnc(C)n1C)c1ccc2nc(Cl)c(CC(F)(F)F)c(N3CCC3)c2c1
COc1nc2ccc(cc2c(Cl)c1CC(F)(F)F)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F
COc1nc2ccc(cc2c(Cl)c1CC(F)(F)F)[C@@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CC(F)(F)F)[C@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
COc1nc2ccc(cc2c(C#N)c1CC(F)(F)F)[C@@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
COc1nc2ccc(cc2c(C#N)c1CC(F)(F)F)[C@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CC(F)(F)F)[C@@](O)(c1cncn1C)c1ccc(Cl)cc1 |r|
COc1nc2ccc(cc2c(Cl)c1CC(F)(F)F)[C@](O)(c1cncn1C)c1ccc(Cl)cc1 |r|
COc1nc2ccc(cc2c(Cl)c1CCC(F)(F)F)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F
COc1nc2ccc(cc2c(Cl)c1CCC(F)(F)F)[C@@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CCC(F)(F)F)[C@](O)(c1cncn1C)c1ccc(nc1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CCC(F)(F)F)C(O)(c1cncn1C)c1ccnc(c1)C(F)(F)F
COc1nc2ccc(cc2c(Cl)c1CCC(F)(F)F)[C@@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CCC(F)(F)F)[C@](O)(c1cncn1C)c1ccnc(c1)C(F)(F)F |r|
COc1nc2ccc(cc2c(Cl)c1CCC(F)(F)F)C(O)(c1cncn1C)c1ccc(Cl)cc1
COc1nc2ccc(cc2c(Cl)c1CCC(F)(F)F)[C@@](O)(c1cncn1C)c1ccc(Cl)cc1 |r|
COc1nc2ccc(cc2c(Cl)c1CCC(F)(F)F)[C@](O)(c1cncn1C)c1ccc(Cl)cc1 |r|
COc1nc2ccc(cc2c(Cl)c1OCC(F)(F)F)C(O)(c1cnc(C)n1C)c1c(C)nn(C)c1C
FC(F)(F)C(OCc1ccccc1)(c1ccc(cc1)C1(CC=CC1)S(=O)(=O)c1ccccc1)C(F)(F)F |c:23|
OC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccccc1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CC=CC1)c1ccc(cc1)C(OCc1ccccc1)(C(F)(F)F)C(F)(F)F |c:13|
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccccc1)(C(F)(F)F)C(F)(F)F
c1cc(ccc1C2(CCCC2)S(=O)(=O)c3ccc(cc3)F)C(C(F)(F)F)(C(F)(F)F)O
COC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(Cl)(C(F)(F)F)C(F)(F)F
NC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
CC(O)(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
CC(OCc1c(F)cccc1F)(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(F)(F)c1ccccc1
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(Oc1ccccc1)(C(F)(F)F)C(F)(F)F
O[C@H]1CC[C@](C1)(c1ccc(cc1)C(OCc1ccccc1)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
O[C@H]1CC[C@](C1)(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
O[C@@H]1CC[C@](C1)(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
O[C@H]1CC[C@@](C1)(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)C1(CC=CC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |c:13|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(C[C@H]2O[C@H]2C1)c1ccc(cc1)C(OCc1ccccc1)(C(F)(F)F)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(C[C@H]2O[C@H]2C1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r|
O[C@H]1C[C@](C[C@H]1O)(c1ccc(cc1)C(OCc1ccccc1)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
O[C@H]1C[C@](C[C@H]1O)(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(c1ccc(cc1)[C@]1(C[C@H]2OC(=O)O[C@H]2C1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)C1(CCC(=C)C1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
OCC1CCC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(=O)C1CCC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CC(=O)N1CCN(CC1)C(=O)[C@@H]1CC[C@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCN(CC1)C(=O)[C@H]1CC[C@@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCN(CC1)C(=O)[C@@H]1CC[C@@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCN(CC1)C(=O)[C@H]1CC[C@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(C)OC(=O)NC1CCC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
Fc1ccc(cc1)S(=O)(=O)C1(CCC(C1)NCc1ccccc1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
Fc1cccc(F)c1COC(c1ccc(cc1)C1(CC1)S(=O)(=O)c1ccccc1)(C(F)(F)F)C(F)(F)F
OC[C@H]1C[C@]1(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(C)OC(=O)[C@H]1C[C@]1(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN(C)C(=O)[C@H]1C[C@]1(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)C1(CCC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CC(=C)C1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
OCC1CC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |(-3.89,-8.36,;-2.55,-7.59,;-2.55,-6.05,;-1.46,-4.96,;-2.55,-3.87,;-3.64,-4.96,;-1.46,-2.78,;.02,-3.18,;1.11,-2.09,;.71,-.6,;-.77,-.21,;-1.86,-1.3,;1.8,.48,;2.89,1.57,;2.49,3.06,;3.58,4.15,;3.18,5.64,;1.7,6.04,;4.27,6.73,;5.76,6.33,;6.16,4.84,;5.07,3.75,;5.47,2.26,;.71,1.57,;-.37,2.66,;-.37,.48,;1.8,2.66,;2.89,-.6,;3.98,-1.69,;1.8,-1.69,;3.98,.48,;-3.64,-2.78,;-2.55,-1.69,;-4.73,-3.87,;-4.73,-1.69,;-6.22,-2.09,;-7.31,-1,;-6.91,.48,;-8,1.57,;-5.42,.88,;-4.33,-.21,)|
OC(=O)[C@H]1C[C@@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:5.7,wD:3.2,(-3.76,-13.91,;-2.42,-13.14,;-1.09,-13.91,;-2.42,-11.6,;-1.33,-10.51,;-2.42,-9.42,;-3.51,-10.51,;-1.33,-8.33,;.15,-8.73,;1.24,-7.64,;.84,-6.15,;-.64,-5.75,;-1.73,-6.84,;1.93,-5.06,;3.02,-3.97,;2.62,-2.49,;3.71,-1.4,;3.31,.09,;1.83,.49,;4.4,1.18,;5.89,.78,;6.29,-.71,;5.2,-1.8,;5.6,-3.28,;.84,-3.97,;-.25,-2.89,;-.25,-5.06,;1.93,-2.89,;3.02,-6.15,;4.11,-7.24,;1.93,-7.24,;4.11,-5.06,;-3.51,-8.33,;-2.42,-7.24,;-4.6,-9.42,;-4.6,-7.24,;-6.09,-7.64,;-7.18,-6.55,;-6.78,-5.06,;-7.87,-3.97,;-5.29,-4.66,;-4.2,-5.75,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(C[C@@H](C1)C(=O)NC1CCOCC1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:10.25,wD:12.15,(-6.08,4.02,;-4.99,2.93,;-5.39,1.44,;-4.3,.35,;-2.81,.75,;-2.42,2.24,;-3.51,3.33,;-1.73,-.34,;-2.81,-1.43,;-.64,.75,;-.64,-1.43,;.45,-2.52,;-.64,-3.6,;-1.73,-2.52,;-.64,-5.14,;.7,-5.91,;-1.97,-5.91,;-1.97,-7.45,;-.64,-8.22,;-.64,-9.76,;-1.97,-10.53,;-3.3,-9.76,;-3.3,-8.22,;.45,-.34,;1.94,-.74,;3.03,.35,;2.63,1.84,;1.14,2.24,;.05,1.15,;3.72,2.93,;4.81,4.02,;4.81,1.84,;5.9,.75,;3.72,.75,;5.9,2.93,;2.63,4.02,;1.54,5.11,;3.72,5.11,;1.54,2.93,)|
NC1CC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |(-2.81,-13.01,;-2.81,-11.47,;-1.72,-10.38,;-2.81,-9.29,;-3.9,-10.38,;-1.72,-8.21,;-.23,-8.6,;.86,-7.52,;.46,-6.03,;-1.03,-5.63,;-2.12,-6.72,;1.55,-4.94,;2.64,-3.85,;2.24,-2.36,;3.33,-1.27,;2.93,.21,;1.44,.61,;4.02,1.3,;5.51,.9,;5.9,-.58,;4.82,-1.67,;5.21,-3.16,;.46,-3.85,;-.63,-2.76,;-.63,-4.94,;1.55,-2.76,;2.64,-6.03,;3.73,-7.12,;1.55,-7.12,;3.73,-4.94,;-3.9,-8.21,;-2.81,-7.12,;-4.98,-9.29,;-4.98,-7.12,;-6.47,-7.52,;-7.56,-6.43,;-7.16,-4.94,;-8.25,-3.85,;-5.67,-4.54,;-4.59,-5.63,)|
Cn1cc(cn1)-c1ccc2CC(Cc2c1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCC=C)(C(F)(F)F)C(F)(F)F
COCCOC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
COCCOCCOC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
OCCCOC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
CN(C)CCOC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
NC(=O)COC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
CNC(=O)COC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCC(=O)Nc1ccccc1Cl)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCC1CCOCC1)(C(F)(F)F)C(F)(F)F
Cc1ccccc1COC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccccc1F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccccc1Cl)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccccc1C#N)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccccc1C(F)(F)F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccccc1OC(F)(F)F)(C(F)(F)F)C(F)(F)F
FC(F)Oc1ccccc1COC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccccc1-c1ccccc1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccccc1CS(=O)(=O)c1ccccc1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1cccc(c1)C#N)(C(F)(F)F)C(F)(F)F
CC(C)(C)OC(=O)Nc1cccc(COC(c2ccc(cc2)C2(CCCC2)S(=O)(=O)c2ccc(F)cc2)(C(F)(F)F)C(F)(F)F)c1
Nc1cccc(COC(c2ccc(cc2)C2(CCCC2)S(=O)(=O)c2ccc(F)cc2)(C(F)(F)F)C(F)(F)F)c1
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccc(cc1)C(F)(F)F)(C(F)(F)F)C(F)(F)F
COC(=O)c1ccc(COC(c2ccc(cc2)C2(CCCC2)S(=O)(=O)c2ccc(F)cc2)(C(F)(F)F)C(F)(F)F)cc1
NC(=O)c1ccc(COC(c2ccc(cc2)C2(CCCC2)S(=O)(=O)c2ccc(F)cc2)(C(F)(F)F)C(F)(F)F)cc1
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccc(cc1)C(=O)c1ccccc1)(C(F)(F)F)C(F)(F)F
CS(=O)(=O)c1ccc(COC(c2ccc(cc2)C2(CCCC2)S(=O)(=O)c2ccc(F)cc2)(C(F)(F)F)C(F)(F)F)cc1
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccc(cc1)-c1ccccc1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccc(cc1)-c1csnn1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1cccc(Cl)c1Cl)(C(F)(F)F)C(F)(F)F
Cc1ccc(COC(c2ccc(cc2)C2(CCCC2)S(=O)(=O)c2ccc(F)cc2)(C(F)(F)F)C(F)(F)F)c(F)c1
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccc(F)cc1F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccc(cc1F)C#N)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccc(cc1F)-c1ncon1)(C(F)(F)F)C(F)(F)F
CS(=O)(=O)c1ccc(COC(c2ccc(cc2)C2(CCCC2)S(=O)(=O)c2ccc(F)cc2)(C(F)(F)F)C(F)(F)F)c(Cl)c1
COc1cc(ccc1COC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F)C#N
COc1cc(ccc1COC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F)C(F)(F)F
COc1cc(OC(F)(F)F)ccc1COC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccc(F)cc1C#N)(C(F)(F)F)C(F)(F)F
CS(=O)(=O)c1cc(Cl)ccc1COC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1cc(F)ccc1F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1cc(Cl)ccc1F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1cc(ccc1F)C#N)(C(F)(F)F)C(F)(F)F
COC(=O)c1ccc(F)c(COC(c2ccc(cc2)C2(CCCC2)S(=O)(=O)c2ccc(F)cc2)(C(F)(F)F)C(F)(F)F)c1
FC(F)Oc1ccc(F)c(COC(c2ccc(cc2)C2(CCCC2)S(=O)(=O)c2ccc(F)cc2)(C(F)(F)F)C(F)(F)F)c1
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1cc(F)ccc1C#N)(C(F)(F)F)C(F)(F)F
COC(=O)c1ccc(C#N)c(COC(c2ccc(cc2)C2(CCCC2)S(=O)(=O)c2ccc(F)cc2)(C(F)(F)F)C(F)(F)F)c1
COc1ccc(F)cc1COC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
COc1ccc(OC(F)(F)F)cc1COC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
COc1ccc(cc1COC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F)[N+]([O-])=O
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1c(Cl)cccc1Cl)(C(F)(F)F)C(F)(F)F
COC(=O)c1cccc(F)c1COC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccc(Cl)c(Cl)c1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccc(C#N)c(F)c1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccc(F)c(c1)C#N)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccc(-c2ncco2)c(F)c1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccc(-c2ncon2)c(F)c1)(C(F)(F)F)C(F)(F)F
COc1cc(F)cc(COC(c2ccc(cc2)C2(CCCC2)S(=O)(=O)c2ccc(F)cc2)(C(F)(F)F)C(F)(F)F)c1
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1c(F)cc(F)cc1F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1c(F)ccc(F)c1F)(C(F)(F)F)C(F)(F)F
Cc1ccc(F)c(COC(c2ccc(cc2)C2(CCCC2)S(=O)(=O)c2ccc(F)cc2)(C(F)(F)F)C(F)(F)F)c1F
COc1ccc(F)c(COC(c2ccc(cc2)C2(CCCC2)S(=O)(=O)c2ccc(F)cc2)(C(F)(F)F)C(F)(F)F)c1F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1cccc2ccccc12)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccc2ccccc2c1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1cc(Cl)nc(Cl)c1)(C(F)(F)F)C(F)(F)F
Cc1ccc(COC(c2ccc(cc2)C2(CCCC2)S(=O)(=O)c2ccc(F)cc2)(C(F)(F)F)C(F)(F)F)c(C)n1
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1cccnc1Br)(C(F)(F)F)C(F)(F)F
COC(=O)c1ncccc1COC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccccn1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccc(cn1)C#N)(C(F)(F)F)C(F)(F)F
CSc1nccc(COC(c2ccc(cc2)C2(CCCC2)S(=O)(=O)c2ccc(F)cc2)(C(F)(F)F)C(F)(F)F)n1
Cc1noc(C)c1COC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1ccno1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1cc(no1)-c1ccccc1C#N)(C(F)(F)F)C(F)(F)F
Cc1cc(COC(c2ccc(cc2)C2(CCCC2)S(=O)(=O)c2ccc(F)cc2)(C(F)(F)F)C(F)(F)F)n(n1)-c1ccc(Cl)cc1
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCC1COc2ccccc2O1)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCCn1cccn1)(C(F)(F)F)C(F)(F)F
CCC(O)(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
CCC(OCc1c(F)cccc1F)(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
CCC(OCc1c(F)cccc1F)(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(OC)cc1)C(F)(F)F
OC(c1ccccc1)(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
COC(c1ccccc1)(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
OC(Cc1ccccc1)(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
OC(CCc1ccccc1)(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(Oc1ccccc1F)(C(F)(F)F)C(F)(F)F
Cc1ccc(OC(c2ccc(cc2)C2(CCCC2)S(=O)(=O)c2ccc(F)cc2)(C(F)(F)F)C(F)(F)F)cc1
Fc1ccc(OC(c2ccc(cc2)C2(CCCC2)S(=O)(=O)c2ccc(F)cc2)(C(F)(F)F)C(F)(F)F)cc1
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(Oc1ccc(cc1)C#N)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(Oc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
CC(Oc1ccccc1)(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
COc1ccc(OC(C)(c2ccc(cc2)C2(CCCC2)S(=O)(=O)c2ccc(F)cc2)C(F)(F)F)cc1
O[C@H]1CC[C@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
O[C@@H]1CC[C@@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
O[C@H]1CC[C@](C1)(c1ccc(cc1)C(OCc1cccc(c1)C#N)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
O[C@H]1CC[C@](C1)(c1ccc(cc1)C(OCc1cc(F)ccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
O[C@H]1CC[C@](C1)(c1ccc(cc1)C(OCc1c(Cl)cccc1Cl)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Cc1noc(C)c1COC(c1ccc(cc1)[C@@]1(CC[C@H](O)C1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F |r|
O[C@H]1C[C@](C[C@H]1O)(c1ccc(cc1)C(OCc1cc(F)ccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
O[C@H]1C[C@](C[C@H]1O)(c1ccc(cc1)C(OCc1cccc(c1)C#N)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
O[C@H]1C[C@](C[C@H]1O)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(C[C@H]2OC(=O)O[C@H]2C1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@]1(CC[C@@H](C1)C(=O)Nc1ccncc1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@]1(CC[C@H](C1)C(=O)Nc1ccncc1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@]1(CC[C@@H](C1)C(=O)NCc1ccncc1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@]1(CC[C@H](C1)C(=O)NCc1ccncc1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@]1(CC[C@@H](C1)C(=O)NC1CCOCC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@]1(CC[C@H](C1)C(=O)NC1CCOCC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r|
OC(=O)C1CCN(CC1)C(=O)C1CCC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(=O)C1CCN(CC1)C(=O)[C@H]1CC[C@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C1CCN(CC1)C(=O)[C@@H]1CC[C@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC1(O)CCN(CC1)C(=O)C1CCC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CC1(O)CCN(CC1)C(=O)[C@H]1CC[C@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC1(O)CCN(CC1)C(=O)[C@@H]1CC[C@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OCC1(O)CCN(CC1)C(=O)C1CCC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
Fc1ccc(cc1)S(=O)(=O)[C@]1(CC[C@@H](C1)C(=O)N1CCOCC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@]1(CC[C@H](C1)C(=O)N1CCOCC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r|
CC1(O)CCN(CC1)C(=O)[C@@H]1CC[C@](C1)(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC1(O)CCN(CC1)C(=O)[C@H]1CC[C@](C1)(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCN(CC1)C(=O)[C@@H]1CC[C@](C1)(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCN(CC1)C(=O)[C@H]1CC[C@](C1)(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCN(CC1)C(=O)[C@@H]1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCN(CC1)C(=O)[C@H]1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC1(O)CCN(CC1)C(=O)[C@@H]1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@]1(CC[C@H](C1)C(=O)NC1CCOCC1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@]1(CC[C@@H](C1)C(=O)NC1CCOCC1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
CCN(CC)C(=O)[C@H]1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)NC1CCC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CC(C)CNC1CCC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
COc1ccc(NC2CCC(C2)(c2ccc(cc2)C(OCc2c(F)cccc2F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)cc1
Fc1ccc(cc1)S(=O)(=O)C1(CCC(C1)NCc1ccc(Cl)cc1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCC(C1)N1CCOCC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
CC(=O)NC1CCC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)NC1CCC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:3.2,wD:6.9,(6.89,-12.02,;7.52,-10.61,;9.05,-10.45,;6.61,-9.36,;5.08,-9.53,;4.18,-8.28,;4.8,-6.87,;6.34,-6.71,;7.24,-7.96,;3.9,-5.63,;4.53,-4.22,;2.37,-5.79,;1.46,-4.54,;-.08,-4.54,;-.55,-3.08,;.69,-2.17,;1.94,-3.08,;-.34,-1.03,;.14,.44,;-.89,1.58,;-2.4,1.26,;-2.88,-.2,;-1.84,-1.35,;-3.43,2.41,;-4.46,3.55,;-5.97,3.23,;-7,4.37,;-8.5,4.05,;-8.98,2.59,;-9.53,5.2,;-9.06,6.66,;-7.55,6.98,;-6.52,5.84,;-5.01,6.16,;-4.57,1.37,;-5.72,.34,;-3.54,.23,;-5.6,2.52,;-2.29,3.44,;-1.14,4.47,;-1.25,2.29,;-3.32,4.58,;1.72,-1.03,;.58,0,;2.87,-2.06,;2.75,.12,;2.28,1.58,;3.31,2.73,;4.81,2.41,;5.84,3.55,;5.29,.94,;4.26,-.2,)|
Fc1ccc(cc1)S(=O)(=O)C1(CCC(C1)NC(=O)C1CCOCC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
CC(=O)N1CCC(CC1)C(=O)NC1CCC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
Fc1ccc(cc1)S(=O)(=O)C1(CCC(C1)NC(=O)c1ccncc1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(CCC(C1)N1CCCC1=O)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
NC(=O)[C@H]1C[C@]1(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CNC(=O)[C@H]1C[C@]1(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC1(O)CCN(CC1)C(=O)[C@H]1C[C@]1(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CNC(=O)[C@H]1C[C@@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:6.8,wD:4.3,(-.83,-9.54,;-.83,-8,;-2.16,-7.23,;-3.5,-8,;-2.16,-5.69,;-1.07,-4.61,;-2.16,-3.52,;-3.25,-4.61,;-1.07,-2.43,;.41,-2.83,;1.5,-1.74,;1.1,-.25,;-.38,.15,;-1.47,-.94,;2.19,.84,;3.28,1.93,;2.88,3.42,;3.97,4.5,;3.57,5.99,;2.09,6.39,;4.66,7.08,;6.15,6.68,;6.55,5.19,;5.46,4.11,;5.86,2.62,;3.28,-.25,;4.37,-1.34,;2.19,-1.34,;4.37,.84,;1.1,1.93,;.01,3.02,;.01,.84,;2.19,3.02,;-3.25,-2.43,;-4.34,-3.52,;-2.16,-1.34,;-4.34,-1.34,;-5.83,-1.74,;-6.92,-.65,;-6.52,.84,;-7.61,1.93,;-5.03,1.24,;-3.94,.15,)|
CC(C)(O)CNC(=O)[C@H]1C[C@@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:10.12,wD:8.7,(-2.82,-10.55,;-1.48,-9.78,;-2.25,-8.44,;-.71,-11.11,;-.15,-9.01,;-.15,-7.47,;-1.48,-6.7,;-2.82,-7.47,;-1.48,-5.16,;-.39,-4.07,;-1.48,-2.98,;-2.57,-4.07,;-.39,-1.89,;1.09,-2.29,;2.18,-1.2,;1.78,.29,;.3,.69,;-.79,-.4,;2.87,1.38,;3.96,2.47,;3.56,3.95,;4.65,5.04,;4.25,6.53,;2.77,6.93,;5.34,7.62,;6.83,7.22,;7.23,5.73,;6.14,4.64,;6.54,3.16,;1.78,2.47,;.69,3.55,;.69,1.38,;2.87,3.55,;3.96,.29,;5.05,-.8,;2.87,-.8,;5.05,1.38,;-2.57,-1.89,;-3.66,-2.98,;-1.48,-.8,;-3.66,-.8,;-5.15,-1.2,;-6.24,-.11,;-5.84,1.38,;-6.93,2.47,;-4.35,1.78,;-3.26,.69,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(C[C@@H](C1)C(=O)NCc1ccncc1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r,wU:10.26,wD:12.15,(-6.63,3.06,;-5.54,1.98,;-5.94,.49,;-4.85,-.6,;-3.37,-.2,;-2.97,1.29,;-4.06,2.37,;-2.28,-1.29,;-3.37,-2.38,;-1.19,-.2,;-1.19,-2.38,;-.1,-3.47,;-1.19,-4.56,;-2.28,-3.47,;-1.19,-6.1,;.14,-6.87,;-2.52,-6.87,;-2.52,-8.41,;-3.86,-9.18,;-3.86,-10.72,;-5.19,-11.49,;-6.52,-10.72,;-6.52,-9.18,;-5.19,-8.41,;-.1,-1.29,;1.39,-1.69,;2.48,-.6,;2.08,.89,;.59,1.29,;-.5,.2,;3.17,1.98,;4.26,3.06,;3.86,4.55,;4.95,5.64,;4.55,7.13,;3.06,7.53,;5.64,8.22,;7.12,7.82,;7.52,6.33,;6.43,5.24,;6.83,3.75,;2.08,3.06,;.99,4.15,;.99,1.98,;3.17,4.15,;4.26,.89,;5.34,-.2,;3.17,-.2,;5.34,1.98,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(C[C@@H](C1)C(=O)Nc1ccncc1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r,wU:10.25,wD:12.15,(-6.62,2.33,;-5.53,1.24,;-5.93,-.25,;-4.84,-1.34,;-3.36,-.94,;-2.96,.55,;-4.05,1.64,;-2.27,-2.03,;-3.36,-3.12,;-1.18,-.94,;-1.18,-3.12,;-.09,-4.21,;-1.18,-5.3,;-2.27,-4.21,;-1.18,-6.84,;-2.51,-7.61,;.16,-7.61,;.16,-9.15,;1.49,-9.92,;1.49,-11.46,;.16,-12.23,;-1.18,-11.46,;-1.18,-9.92,;-.09,-2.03,;1.4,-2.43,;2.49,-1.34,;2.09,.15,;.6,.55,;-.49,-.54,;3.18,1.24,;4.27,2.33,;3.87,3.81,;4.96,4.9,;4.56,6.39,;3.07,6.79,;5.65,7.48,;7.13,7.08,;7.53,5.59,;6.44,4.51,;6.84,3.02,;2.09,2.33,;1,3.42,;1,1.24,;3.18,3.42,;4.27,.15,;5.36,-.94,;3.18,-.94,;5.36,1.24,)|
Cc1nnc(NC(=O)[C@H]2C[C@@](C2)(c2ccc(cc2)C(OCc2c(F)cccc2F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)s1 |r,wU:10.12,wD:8.7,(1.33,-12.6,;.42,-11.36,;-1.12,-11.36,;-1.59,-9.89,;-.35,-8.99,;-.35,-7.45,;-1.68,-6.68,;-3.01,-7.45,;-1.68,-5.14,;-.59,-4.05,;-1.68,-2.96,;-2.77,-4.05,;-.59,-1.87,;.9,-2.27,;1.99,-1.18,;1.59,.31,;.1,.71,;-.99,-.38,;2.68,1.4,;3.77,2.49,;3.37,3.97,;4.46,5.06,;4.06,6.55,;2.57,6.95,;5.15,7.64,;6.63,7.24,;7.03,5.75,;5.94,4.66,;6.34,3.18,;1.59,2.49,;.5,3.57,;.5,1.4,;2.68,3.57,;3.77,.31,;4.85,-.78,;2.68,-.78,;4.85,1.4,;-2.77,-1.87,;-3.86,-2.96,;-1.68,-.78,;-3.86,-.78,;-5.34,-1.18,;-6.43,-.09,;-6.04,1.4,;-7.12,2.49,;-4.55,1.8,;-3.46,.71,;.9,-9.89,)|
Fc1ccc(cc1)S(=O)(=O)[C@]1(C[C@@H](C1)C(=O)NCC1CCOCC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r,wU:10.26,12.15,(-6.63,3.06,;-5.54,1.98,;-5.94,.49,;-4.85,-.6,;-3.37,-.2,;-2.97,1.29,;-4.06,2.37,;-2.28,-1.29,;-3.37,-2.38,;-1.19,-.2,;-1.19,-2.38,;-2.28,-3.47,;-1.19,-4.56,;-.1,-3.47,;-1.19,-6.1,;.14,-6.87,;-2.52,-6.87,;-2.52,-8.41,;-3.86,-9.18,;-3.86,-10.72,;-5.19,-11.49,;-6.52,-10.72,;-6.52,-9.18,;-5.19,-8.41,;-.1,-1.29,;1.39,-1.69,;2.48,-.6,;2.08,.89,;.59,1.29,;-.5,.2,;3.17,1.98,;4.26,3.06,;3.86,4.55,;4.95,5.64,;4.55,7.13,;3.06,7.53,;5.64,8.22,;7.12,7.82,;7.52,6.33,;6.43,5.24,;6.83,3.75,;2.08,3.06,;.99,4.15,;.99,1.98,;3.17,4.15,;4.26,.89,;5.34,-.2,;3.17,-.2,;5.34,1.98,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(C[C@@H](C1)C(=O)NCC1CCOCC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r,wU:10.26,wD:12.15,(-6.63,3.06,;-5.54,1.98,;-5.94,.49,;-4.85,-.6,;-3.37,-.2,;-2.97,1.29,;-4.06,2.37,;-2.28,-1.29,;-3.37,-2.38,;-1.19,-.2,;-1.19,-2.38,;-.1,-3.47,;-1.19,-4.56,;-2.28,-3.47,;-1.19,-6.1,;.14,-6.87,;-2.52,-6.87,;-2.52,-8.41,;-3.86,-9.18,;-3.86,-10.72,;-5.19,-11.49,;-6.52,-10.72,;-6.52,-9.18,;-5.19,-8.41,;-.1,-1.29,;1.39,-1.69,;2.48,-.6,;2.08,.89,;.59,1.29,;-.5,.2,;3.17,1.98,;4.26,3.06,;3.86,4.55,;4.95,5.64,;4.55,7.13,;3.06,7.53,;5.64,8.22,;7.12,7.82,;7.52,6.33,;6.43,5.24,;6.83,3.75,;2.08,3.06,;.99,4.15,;.99,1.98,;3.17,4.15,;4.26,.89,;5.34,-.2,;3.17,-.2,;5.34,1.98,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(C[C@@H](C1)C(=O)NCC1CCC(F)(F)CC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r,wU:10.28,wD:12.15,(-6.51,3.63,;-5.42,2.54,;-5.82,1.05,;-4.73,-.04,;-3.24,.36,;-2.84,1.85,;-3.93,2.94,;-2.15,-.73,;-3.24,-1.82,;-1.06,.36,;-1.06,-1.82,;.03,-2.91,;-1.06,-3.99,;-2.15,-2.91,;-1.06,-5.53,;.27,-6.3,;-2.4,-6.3,;-2.4,-7.84,;-3.73,-8.61,;-3.73,-10.15,;-5.06,-10.92,;-6.4,-10.15,;-7.21,-11.46,;-7.94,-10.21,;-6.4,-8.61,;-5.06,-7.84,;.03,-.73,;1.51,-1.13,;2.6,-.04,;2.2,1.45,;.72,1.85,;-.37,.76,;3.29,2.54,;4.38,3.63,;3.98,5.12,;5.07,6.2,;4.67,7.69,;3.19,8.09,;5.76,8.78,;7.25,8.38,;7.65,6.9,;6.56,5.81,;6.96,4.32,;2.2,3.63,;1.11,4.72,;1.11,2.54,;3.29,4.72,;4.38,1.45,;5.47,.36,;3.29,.36,;5.47,2.54,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(C[C@@H](C1)C(=O)NC1CCOCC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r,wU:10.25,wD:12.15,(-6.62,2.33,;-5.53,1.24,;-5.93,-.25,;-4.84,-1.34,;-3.36,-.94,;-2.96,.55,;-4.05,1.64,;-2.27,-2.03,;-3.36,-3.12,;-1.18,-.94,;-1.18,-3.12,;-.09,-4.21,;-1.18,-5.3,;-2.27,-4.21,;-1.18,-6.84,;-2.51,-7.61,;.16,-7.61,;.16,-9.15,;1.49,-9.92,;1.49,-11.46,;.16,-12.23,;-1.18,-11.46,;-1.18,-9.92,;-.09,-2.03,;1.4,-2.43,;2.49,-1.34,;2.09,.15,;.6,.55,;-.49,-.54,;3.18,1.24,;4.27,2.33,;3.87,3.81,;4.96,4.9,;4.56,6.39,;3.07,6.79,;5.65,7.48,;7.13,7.08,;7.53,5.59,;6.44,4.51,;6.84,3.02,;2.09,2.33,;1,3.42,;1,1.24,;3.18,3.42,;4.27,.15,;5.36,-.94,;3.18,-.94,;5.36,1.24,)|
CN(C)C(=O)[C@H]1C[C@@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:7.9,wD:5.4,(.67,-7.05,;-.67,-7.82,;-.67,-9.36,;-2,-7.05,;-3.33,-7.82,;-2,-5.51,;-.91,-4.42,;-2,-3.33,;-3.09,-4.42,;-.91,-2.24,;.58,-2.64,;1.67,-1.55,;1.27,-.06,;-.22,.34,;-1.31,-.75,;2.36,1.03,;3.45,2.11,;3.05,3.6,;4.14,4.69,;3.74,6.18,;2.25,6.58,;4.83,7.27,;6.31,6.87,;6.71,5.38,;5.62,4.29,;6.02,2.8,;1.27,2.11,;.18,3.2,;.18,1.03,;2.36,3.2,;3.45,-.06,;4.53,-1.15,;2.36,-1.15,;4.53,1.03,;-3.09,-2.24,;-2,-1.15,;-4.18,-3.33,;-4.18,-1.15,;-5.66,-1.55,;-6.75,-.46,;-6.36,1.03,;-7.44,2.11,;-4.87,1.42,;-3.78,.34,)|
FC1CN(C1)C(=O)[C@H]1C[C@@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:9.12,wD:7.7,(-5.99,-9.17,;-4.65,-8.4,;-3.17,-8.79,;-2.77,-7.31,;-4.25,-6.91,;-1.43,-6.54,;-.1,-7.31,;-1.43,-5,;-.34,-3.91,;-1.43,-2.82,;-2.52,-3.91,;-.34,-1.73,;1.14,-2.13,;2.23,-1.04,;1.83,.45,;.35,.85,;-.74,-.24,;2.92,1.54,;4.01,2.63,;3.61,4.11,;4.7,5.2,;4.3,6.69,;2.82,7.09,;5.39,7.78,;6.88,7.38,;7.28,5.89,;6.19,4.8,;6.59,3.32,;1.83,2.63,;.74,3.71,;.74,1.54,;2.92,3.71,;4.01,.45,;5.1,-.64,;2.92,-.64,;5.1,1.54,;-2.52,-1.73,;-3.61,-2.82,;-1.43,-.64,;-3.61,-.64,;-5.1,-1.04,;-6.19,.05,;-5.79,1.54,;-6.88,2.63,;-4.3,1.94,;-3.21,.85,)|
OC1CN(C1)C(=O)[C@H]1C[C@@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:9.12,wD:7.7,(-5.99,-9.17,;-4.65,-8.4,;-3.17,-8.79,;-2.77,-7.31,;-4.25,-6.91,;-1.43,-6.54,;-.1,-7.31,;-1.43,-5,;-.34,-3.91,;-1.43,-2.82,;-2.52,-3.91,;-.34,-1.73,;1.14,-2.13,;2.23,-1.04,;1.83,.45,;.35,.85,;-.74,-.24,;2.92,1.54,;4.01,2.63,;3.61,4.11,;4.7,5.2,;4.3,6.69,;2.82,7.09,;5.39,7.78,;6.88,7.38,;7.28,5.89,;6.19,4.8,;6.59,3.32,;1.83,2.63,;.74,3.71,;.74,1.54,;2.92,3.71,;4.01,.45,;5.1,-.64,;2.92,-.64,;5.1,1.54,;-2.52,-1.73,;-3.61,-2.82,;-1.43,-.64,;-3.61,-.64,;-5.1,-1.04,;-6.19,.05,;-5.79,1.54,;-6.88,2.63,;-4.3,1.94,;-3.21,.85,)|
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CC(=O)N1CCN(CC1)C(=O)[C@H]1C[C@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:13.16,11.11,(-6.24,-10.22,;-6.24,-8.68,;-7.57,-7.91,;-4.9,-7.91,;-3.57,-8.68,;-2.23,-7.91,;-2.23,-6.37,;-3.57,-5.6,;-4.9,-6.37,;-.9,-5.6,;.43,-6.37,;-.9,-4.06,;-1.99,-2.97,;-.9,-1.88,;.19,-2.97,;.19,-.8,;1.68,-1.19,;2.76,-.1,;2.37,1.38,;.88,1.78,;-.21,.69,;3.46,2.47,;4.54,3.56,;4.15,5.05,;5.23,6.14,;4.84,7.62,;3.35,8.02,;5.92,8.71,;7.41,8.32,;7.81,6.83,;6.72,5.74,;7.12,4.25,;2.37,3.56,;1.28,4.65,;1.28,2.47,;3.46,4.65,;4.54,1.38,;5.63,.29,;3.46,.29,;5.63,2.47,;-1.99,-.8,;-3.08,-1.88,;-.9,.29,;-3.08,.29,;-4.57,-.1,;-5.66,.98,;-5.26,2.47,;-6.35,3.56,;-3.77,2.87,;-2.68,1.78,)|
CC(=O)N1CCN(CC1)C(=O)[C@H]1C[C@@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:13.16,wD:11.11,(-6.24,-10.22,;-6.24,-8.68,;-7.57,-7.91,;-4.9,-7.91,;-3.57,-8.68,;-2.23,-7.91,;-2.23,-6.37,;-3.57,-5.6,;-4.9,-6.37,;-.9,-5.6,;.43,-6.37,;-.9,-4.06,;.19,-2.97,;-.9,-1.88,;-1.99,-2.97,;.19,-.8,;1.68,-1.19,;2.76,-.1,;2.37,1.38,;.88,1.78,;-.21,.69,;3.46,2.47,;4.54,3.56,;4.15,5.05,;5.23,6.14,;4.84,7.62,;3.35,8.02,;5.92,8.71,;7.41,8.32,;7.81,6.83,;6.72,5.74,;7.12,4.25,;2.37,3.56,;1.28,4.65,;1.28,2.47,;3.46,4.65,;4.54,1.38,;5.63,.29,;3.46,.29,;5.63,2.47,;-1.99,-.8,;-3.08,-1.88,;-.9,.29,;-3.08,.29,;-4.57,-.1,;-5.66,.98,;-5.26,2.47,;-6.35,3.56,;-3.77,2.87,;-2.68,1.78,)|
Fc1ccc(cc1)S(=O)(=O)[C@]1(C[C@@H](C1)C(=O)N1CCOCC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r,wU:10.24,12.15,(-6.31,2.84,;-5.22,1.75,;-5.62,.27,;-4.53,-.82,;-3.05,-.42,;-2.65,1.06,;-3.74,2.15,;-1.96,-1.51,;-3.05,-2.6,;-.87,-.42,;-.87,-2.6,;-1.96,-3.69,;-.87,-4.78,;.22,-3.69,;-.87,-6.32,;.47,-7.09,;-2.2,-7.09,;-2.2,-8.63,;-3.54,-9.4,;-4.87,-8.63,;-4.87,-7.09,;-3.54,-6.32,;.22,-1.51,;1.71,-1.91,;2.8,-.82,;2.4,.66,;.91,1.06,;-.18,-.03,;3.49,1.75,;4.58,2.84,;4.18,4.33,;5.27,5.42,;4.87,6.91,;3.38,7.31,;5.96,8,;7.44,7.6,;7.84,6.11,;6.75,5.02,;7.15,3.53,;2.4,2.84,;1.31,3.93,;1.31,1.75,;3.49,3.93,;4.58,.66,;5.67,-.42,;3.49,-.42,;5.67,1.75,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(C[C@@H](C1)C(=O)N1CCOCC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r,wU:10.24,wD:12.15,(-6.31,2.84,;-5.22,1.75,;-5.62,.27,;-4.53,-.82,;-3.05,-.42,;-2.65,1.06,;-3.74,2.15,;-1.96,-1.51,;-3.05,-2.6,;-.87,-.42,;-.87,-2.6,;.22,-3.69,;-.87,-4.78,;-1.96,-3.69,;-.87,-6.32,;.47,-7.09,;-2.2,-7.09,;-2.2,-8.63,;-3.54,-9.4,;-4.87,-8.63,;-4.87,-7.09,;-3.54,-6.32,;.22,-1.51,;1.71,-1.91,;2.8,-.82,;2.4,.66,;.91,1.06,;-.18,-.03,;3.49,1.75,;4.58,2.84,;4.18,4.33,;5.27,5.42,;4.87,6.91,;3.38,7.31,;5.96,8,;7.44,7.6,;7.84,6.11,;6.75,5.02,;7.15,3.53,;2.4,2.84,;1.31,3.93,;1.31,1.75,;3.49,3.93,;4.58,.66,;5.67,-.42,;3.49,-.42,;5.67,1.75,)|
CC(C)(O)CNC(=O)[C@H]1C[C@@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:10.12,wD:8.7,(-4.65,-9.23,;-3.32,-8.46,;-2.55,-9.8,;-4.09,-7.13,;-1.98,-7.69,;-1.98,-6.15,;-.65,-5.38,;.69,-6.15,;-.65,-3.84,;.44,-2.76,;-.65,-1.67,;-1.74,-2.76,;.44,-.58,;1.93,-.98,;3.02,.11,;2.62,1.6,;1.13,2,;.04,.91,;3.71,2.69,;4.8,3.78,;4.8,1.6,;5.89,.51,;3.71,.51,;5.89,2.69,;2.62,3.78,;1.53,4.87,;3.71,4.87,;1.53,2.69,;-1.74,-.58,;-2.83,-1.67,;-.65,.51,;-2.83,.51,;-4.31,.11,;-5.4,1.2,;-5,2.69,;-6.09,3.78,;-3.52,3.09,;-2.43,2,)|
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CC1(O)CCN(CC1)C(=O)[C@H]1C[C@@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:12.15,wD:10.10,(-5.83,-6.92,;-4.29,-6.87,;-5.1,-8.17,;-2.95,-7.64,;-1.62,-6.87,;-1.62,-5.33,;-2.95,-4.56,;-4.29,-5.33,;-.29,-4.56,;1.05,-5.33,;-.29,-3.02,;.8,-1.93,;-.29,-.84,;-1.38,-1.93,;.8,.25,;2.29,-.15,;3.38,.94,;2.98,2.43,;1.49,2.83,;.4,1.74,;4.07,3.52,;5.16,4.61,;5.16,2.43,;6.25,1.34,;4.07,1.34,;6.25,3.52,;2.98,4.61,;1.89,5.7,;4.07,5.7,;1.89,3.52,;-1.38,.25,;-2.47,-.84,;-.29,1.34,;-2.47,1.34,;-3.95,.94,;-5.04,2.03,;-4.64,3.52,;-5.73,4.61,;-3.16,3.92,;-2.07,2.83,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]1(C[C@@H](C1)C(=O)N1CCOCC1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:10.24,wD:12.15,(-5.77,4.09,;-4.68,3,;-5.08,1.51,;-3.99,.42,;-2.51,.82,;-2.11,2.31,;-3.2,3.4,;-1.42,-.27,;-2.51,-1.36,;-.33,.82,;-.33,-1.36,;.76,-2.45,;-.33,-3.53,;-1.42,-2.45,;-.33,-5.07,;1.01,-5.84,;-1.66,-5.84,;-1.66,-7.38,;-3,-8.15,;-4.33,-7.38,;-4.33,-5.84,;-3,-5.07,;.76,-.27,;2.25,-.67,;3.34,.42,;2.94,1.91,;1.45,2.31,;.36,1.22,;4.03,3,;5.12,4.09,;5.12,1.91,;6.2,.82,;4.03,.82,;6.2,3,;2.94,4.09,;1.85,5.18,;4.03,5.18,;1.85,3,)|
CC(C)NC1CC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |(.51,-7.3,;-.82,-8.07,;-.82,-9.61,;-2.16,-7.3,;-2.16,-5.76,;-1.07,-4.67,;-2.16,-3.58,;-3.25,-4.67,;-1.07,-2.49,;.42,-2.89,;1.51,-1.8,;1.11,-.32,;-.38,.08,;-1.47,-1.01,;2.2,.77,;3.29,1.86,;2.89,3.35,;3.98,4.44,;3.58,5.93,;2.09,6.32,;4.67,7.01,;6.16,6.62,;6.56,5.13,;5.47,4.04,;5.87,2.55,;3.29,-.32,;4.38,-1.41,;2.2,-1.41,;4.38,.77,;1.11,1.86,;.02,2.95,;.02,.77,;2.2,2.95,;-3.25,-2.49,;-4.33,-3.58,;-2.16,-1.41,;-4.33,-1.41,;-5.82,-1.8,;-6.91,-.71,;-6.51,.77,;-7.6,1.86,;-5.02,1.17,;-3.94,.08,)|
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COC(=O)NC1CC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |(-4.29,-10.08,;-2.96,-9.31,;-2.96,-7.77,;-4.29,-7,;-1.62,-7,;-1.62,-5.46,;-.53,-4.37,;-1.62,-3.28,;-2.71,-4.37,;-.53,-2.19,;.95,-2.59,;2.04,-1.5,;1.65,-.01,;.16,.39,;-.93,-.7,;2.73,1.08,;3.82,2.17,;3.42,3.65,;4.51,4.74,;4.11,6.23,;2.63,6.63,;5.2,7.32,;6.69,6.92,;7.09,5.43,;6,4.34,;6.4,2.86,;3.82,-.01,;4.91,-1.1,;2.73,-1.1,;4.91,1.08,;1.65,2.17,;.56,3.26,;.56,1.08,;2.73,3.26,;-2.71,-2.19,;-3.8,-3.28,;-1.62,-1.1,;-3.8,-1.1,;-5.29,-1.5,;-6.38,-.41,;-5.98,1.08,;-7.07,2.17,;-4.49,1.48,;-3.4,.39,)|
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Fc1ccc(cc1)S(=O)(=O)C1(CC(C1)NC(=O)N1CCOCC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |(-6.64,2.26,;-5.55,1.17,;-5.95,-.32,;-4.86,-1.41,;-3.38,-1.01,;-2.98,.48,;-4.07,1.57,;-2.29,-2.1,;-3.38,-3.19,;-1.2,-1.01,;-1.2,-3.19,;-.11,-4.28,;-1.2,-5.37,;-2.29,-4.28,;-1.2,-6.91,;.14,-7.68,;1.47,-6.91,;.14,-9.22,;1.47,-9.99,;1.47,-11.53,;.14,-12.3,;-1.2,-11.53,;-1.2,-9.99,;-.11,-2.1,;1.38,-2.5,;2.47,-1.41,;2.07,.08,;.58,.48,;-.51,-.61,;3.16,1.17,;4.25,2.26,;3.85,3.74,;4.94,4.83,;4.54,6.32,;3.05,6.72,;5.63,7.41,;7.12,7.01,;7.51,5.52,;6.43,4.43,;6.82,2.95,;2.07,2.26,;.98,3.34,;.98,1.17,;3.16,3.34,;4.25,.08,;5.34,-1.01,;3.16,-1.01,;5.34,1.17,)|
Fc1ccc(cc1)S(=O)(=O)C1(CC(C1)N1CCCC1=O)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |(-7.23,1.93,;-6.15,.84,;-6.54,-.64,;-5.45,-1.73,;-3.97,-1.33,;-3.57,.15,;-4.66,1.24,;-2.88,-2.42,;-3.97,-3.51,;-1.79,-1.33,;-1.79,-3.51,;-.7,-4.6,;-1.79,-5.69,;-2.88,-4.6,;-1.79,-7.23,;-3.04,-8.14,;-2.56,-9.6,;-1.02,-9.6,;-.54,-8.14,;.92,-7.66,;-.7,-2.42,;.79,-2.82,;1.88,-1.73,;1.48,-.25,;-.01,.15,;-1.1,-.94,;2.57,.84,;3.66,1.93,;3.26,3.42,;4.35,4.51,;3.95,6,;2.46,6.4,;5.04,7.09,;6.52,6.69,;6.92,5.2,;5.83,4.11,;6.23,2.62,;3.66,-.25,;4.74,-1.33,;2.57,-1.33,;4.74,.84,;1.48,1.93,;.39,3.02,;.39,.84,;2.57,3.02,)|
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Fc1ccc(cc1)S(=O)(=O)C1(Cc2ccccc2C1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(Cc2cccnc2C1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C1(Cc2ccc(cc2C1)C#N)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
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Fc1ccc(cc1)S(=O)(=O)C1(CC(C1)N1CCN(Cc2ccccc2)CC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |(-6.43,3.12,;-5.34,2.03,;-5.74,.55,;-4.65,-.54,;-3.16,-.14,;-2.76,1.34,;-3.85,2.43,;-2.07,-1.23,;-3.16,-2.32,;-.98,-.14,;-.98,-2.32,;.11,-3.41,;-.98,-4.5,;-2.07,-3.41,;-.98,-6.04,;.35,-6.81,;.35,-8.35,;-.98,-9.12,;-.98,-10.66,;-2.32,-11.43,;-2.32,-12.97,;-3.65,-13.74,;-4.98,-12.97,;-4.98,-11.43,;-3.65,-10.66,;-2.32,-8.35,;-2.32,-6.81,;.11,-1.23,;1.59,-1.63,;2.68,-.54,;2.29,.95,;.8,1.34,;-.29,.26,;3.37,2.03,;4.46,3.12,;4.06,4.61,;5.15,5.7,;4.75,7.19,;3.27,7.59,;5.84,8.28,;7.33,7.88,;7.73,6.39,;6.64,5.3,;7.04,3.81,;2.29,3.12,;1.2,4.21,;1.2,2.03,;3.37,4.21,;4.46,.95,;5.55,-.14,;3.37,-.14,;5.55,2.03,)|
CC(=O)N1CCN(CC1)C1CC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |(.18,-12.81,;-1.16,-12.04,;-2.49,-12.81,;-1.16,-10.5,;.18,-9.73,;.18,-8.19,;-1.16,-7.42,;-2.49,-8.19,;-2.49,-9.73,;-1.16,-5.88,;-.07,-4.79,;-1.16,-3.7,;-2.25,-4.79,;-.07,-2.61,;1.42,-3.01,;2.51,-1.92,;2.11,-.43,;.62,-.04,;-.47,-1.12,;3.2,.65,;4.29,1.74,;3.89,3.23,;4.98,4.32,;4.58,5.81,;3.09,6.21,;5.67,6.9,;7.16,6.5,;7.56,5.01,;6.47,3.92,;6.87,2.43,;2.11,1.74,;1.02,2.83,;1.02,.65,;3.2,2.83,;4.29,-.43,;5.38,-1.52,;3.2,-1.52,;5.38,.65,;-2.25,-2.61,;-3.33,-3.7,;-1.16,-1.52,;-3.33,-1.52,;-4.82,-1.92,;-5.91,-.83,;-5.51,.65,;-6.6,1.74,;-4.02,1.05,;-2.94,-.04,)|
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Fc1ccc(cc1)S(=O)(=O)C1(CCC(C1)N1CCN(Cc2ccccc2)CC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
CN1CCN(CC1)C1CCC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CC(=O)N1CCN(CC1)C1CCC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
Fc1ccc(cc1)S(=O)(=O)C1(CCC(C1)N1CCNCC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F
COCC(=O)N1CCN(CC1)C1CCC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CN(C)C(=O)N1CCN(CC1)C1CCC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CNC(=O)N1CCN(CC1)C1CCC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CS(=O)(=O)N1CCN(CC1)C1CCC(C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(F)(F)C(F)(F)F
CC(c1ccc(cc1)C1(CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
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CC(=O)N1CCC(CC1)C(=O)N[C@@H]1CC[C@](C1)(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
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OCC(=O)N[C@@H]1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@]1(CC[C@H](C1)NC(=O)Cc1cccnc1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
CC(=O)N1CCC(CC1)C(=O)N[C@@H]1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CCOC(=O)CC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F
C[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(O)=O
C[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(O)=O
CCOC(=O)CC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F |r|
CCOC(=O)[C@@H](C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F
CCOC(=O)[C@@H](C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1c(C)n(C)nc1OC
CCOC(=O)[C@H](C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1c(C)n(C)nc1OC
CCOC(=O)[C@H](C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(CC)nc1Cl
CCOC(=O)[C@@H](C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(CC)nc1Cl
CCOC(=O)[C@H](C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F
CCOC(=O)CC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1
CCOC(=O)CC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CCOC(=O)CC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1c(C)n(C)nc1OC |r|
CCOC(=O)CC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(CC)nc1Cl |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)C(F)(F)F |r|
CC(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)C(O)=O |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
COc1nn(C)c(C)c1S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1nn(C)c(C)c1S(=O)(=O)N1C[C@H](C[C@@H](C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1nn(C)c(C)c1S(=O)(=O)N1C[C@H](C[C@H](C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](C[C@@H](C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](C[C@H](C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
C[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)C(O)=O |r|
C[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)C(O)=O |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C#N)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(F)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)c(F)c1)C(F)(F)F |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
Cc1cc(ccc1F)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
COc1nn2CCCc2c1S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(OC(F)(F)F)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(OC(F)F)c1)C(F)(F)F |r|
COc1cccc(c1)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(Cl)c1)C(F)(F)F |r|
Cc1cccc(c1)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)S(C)(=O)=O)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cncc(c1)C(F)(F)F)C(F)(F)F |r|
COc1nn2CCCCc2c1S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(Br)c1)C(F)(F)F |r|
CCOc1nn(cc1S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C1CC1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1ccc(Cl)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1ccc2OCCc2c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1c(Cl)nc2sccn12)C(F)(F)F |r|
COc1ccccc1S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1ccc(Cl)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1ccc(Cl)cc1F)C(F)(F)F |r|
Cc1ccc(cc1Cl)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
Cc1c(Cl)cc(F)cc1S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1ccc(Cl)cn1)C(F)(F)F |r|
COc1cc(ccc1Cl)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1ccc(Cl)cc1S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1ccc(Cl)c(c1)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1ccc(C)cc1S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(C)ccc1S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC(F)F)cc1S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCC(F)F)n1)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cc(F)cc(c1)C(F)(F)F)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(F)(F)F |r|
COc1cc(ccn1)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
Cc1cc(c(F)cc1F)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
Cc1nn(cc1S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1c(Cl)nn2CCCCc12)C(F)(F)F |r|
Cc1cc(cc(C)c1F)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
Cc1cc(c(Cl)cc1F)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OC(F)F)n1)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)S(F)(F)(F)(F)F)C(F)(F)F |r|
CC(C)n1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](C[C@@H](C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
C[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1Cl)C1CC1)C(O)=O |r|
C[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F)C(O)=O |r|
CCOc1nn(cc1S(=O)(=O)N1C[C@H](C[C@@H](C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(F)F |r|
CCn1cc(c(OC(F)F)n1)S(=O)(=O)N1C[C@H](C[C@@H](C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC(F)F)cc1S(=O)(=O)N1C[C@H](C[C@@H](C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCC(F)F)n1)S(=O)(=O)N1C[C@H](C[C@@H](C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1nn2CCCc2c1S(=O)(=O)N1C[C@H](C[C@@H](C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1nn2CCCCc2c1S(=O)(=O)N1C[C@H](C[C@@H](C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
C[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1c(Cl)nn2CCCCc12)C(O)=O |r|
CCOc1sc(CC)nc1S(=O)(=O)N1C[C@H](C[C@@H](C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1sc(nc1S(=O)(=O)N1C[C@H](C[C@@H](C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C1CC1 |r|
CCc1nc(OC(C)C)c(s1)S(=O)(=O)N1C[C@H](C[C@@H](C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCc1nc(c(OCC(F)(F)F)s1)S(=O)(=O)N1C[C@H](C[C@@H](C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)n1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cn(nc1Cl)C1CC1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cncc(Br)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cncc(c1)C1CC1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(n1)C(F)(F)F)C(F)(F)F |r|
Cc1cncc(c1)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cncc(c1)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C1CC1)C(F)(F)F |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1sc(CC)nc1S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1sc(nc1S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C1CC1 |r|
CCOc1sc(nc1S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(F)(F)F |r|
CCc1nc(c(OC(C)C)s1)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCc1nc(c(OCC(F)(F)F)s1)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cc(ccc1F)C1CC1)C(F)(F)F |r|
C[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(O)=O |r|
C[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(O)=O |r|
C[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(C)c1)C(O)=O |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](C[C@@H](C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
C[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(OC(F)F)c1)C(O)=O |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](C[C@H](C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
C[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(OC(F)F)c1)C(O)=O |r|
C[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(C)c1)C(O)=O |r|
C[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(OC(F)(F)F)c1)C(O)=O |r|
C[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(OC(F)(F)F)c1)C(O)=O |r|
C[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(C)c1)C(O)=O |r|
C[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(C)c1)C(O)=O |r|
C[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C1CC1)C(O)=O |r|
C[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C1CC1)C(O)=O |r|
C[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cncc(c1)C(F)(F)F)C(O)=O |r|
C[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cncc(c1)C(F)(F)F)C(O)=O |r|
C[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccnc(c1)C(F)(F)F)C(O)=O |r|
C[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccnc(c1)C(F)(F)F)C(O)=O |r|
C[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccnc(c1)C1CC1)C(O)=O |r|
C[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccnc(c1)C1CC1)C(O)=O |r|
C[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1Cl)C(F)F)C(O)=O |r|
C[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1Cl)C(F)F)C(O)=O |r|
CC[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(O)=O
CC[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(O)=O
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](C[C@@H](C2CC2)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](C[C@H](C2CC2)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CC[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)C(O)=O |r|
CC[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)C(O)=O |r|
CC[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(C)c1)C(O)=O |r|
CC[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C1CC1)C(O)=O |r|
CC[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(C)c1)C(O)=O |r|
CC[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C1CC1)C(O)=O |r|
CC[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(CC)nc1Cl)C(O)=O |r|
CC[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(CC)nc1Cl)C(O)=O |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@H](C[C@@H](CC)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@H](C[C@H](CC)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(OC)c1)C(O)=O |r|
CC[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(CC)nc1OCCO)C(O)=O |r|
CC[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(OC)c1)C(O)=O |r|
CC[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(CC)nc1OCCO)C(O)=O |r|
CC[C@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccnc(c1)C(F)(F)F)C(O)=O |r|
CC[C@@H](C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccnc(c1)C(F)(F)F)C(O)=O |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](C[C@@H](C3CC3)C(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@H](C[C@H](C2CC2)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](C[C@H](C2CC2)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
Cc1cc(ccc1F)S(=O)(=O)N1C[C@H](C[C@H](C2CC2)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](C[C@H](C3CC3)C(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@H](C[C@@H](C2CC2)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](C[C@@H](C2CC2)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
Cc1cc(ccc1F)S(=O)(=O)N1C[C@H](C[C@@H](C2CC2)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@H](C[C@@H](C2CC2)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@H](C[C@H](C2CC2)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(O)=O |r|
CC(C)(C[C@@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)C(O)=O |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
Cc1cc(ccc1F)S(=O)(=O)N1C[C@@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)C(O)=O |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
Cc1cc(ccc1F)S(=O)(=O)N1C[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@@H](CC(C)(C)C(O)=O)Cc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(C[C@@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cncc(c1)C(F)(F)F)C(O)=O |r|
CC(C)(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cncc(c1)C(F)(F)F)C(O)=O |r|
CC(C)(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cncc(c1)C#N)C(O)=O |r|
CC(C)(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1Cl)C1CC1)C(O)=O |r|
Cc1nn(cc1S(=O)(=O)N1C[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(F)F |r|
CCOc1sc(CC)nc1S(=O)(=O)N1C[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1sc(nc1S(=O)(=O)N1C[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C1CC1 |r|
CCc1nc(c(OCC(F)(F)F)s1)S(=O)(=O)N1C[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCc1nc(c(OC(C)C)s1)S(=O)(=O)N1C[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)n1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(cc1S(=O)(=O)N1C[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(F)F |r|
CCn1cc(c(OC(F)F)n1)S(=O)(=O)N1C[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC(F)F)cc1S(=O)(=O)N1C[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCC(F)F)n1)S(=O)(=O)N1C[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1c(Cl)nn2CCCCc12)C(O)=O |r|
COc1nn2CCCCc2c1S(=O)(=O)N1C[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1nn2CCCc2c1S(=O)(=O)N1C[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CC3(CC3)C(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(F)(F)F
CC(C)(OC(=O)Nc1ccc2O[C@H](CC3(CC3)C(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(F)(F)F
Cc1cc(ccc1F)S(=O)(=O)N1C[C@H](CC2(CC2)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CC3(CC3)C(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C1CC1)C(F)(F)F |r|
Cc1cc(ccc1F)S(=O)(=O)N1C[C@@H](CC2(CC2)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@H](CC3(CC3)C(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C1CC1)C(F)(F)F |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CC2(CC2)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](CC2(CC2)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CC2(CC2)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@@H](CC2(CC2)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CC(O)C(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](C[C@](C)(O)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](C[C@@](C)(O)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CC(C)(OC(=O)Nc1ccc2O[C@@H](C[C@@](C)(CO)C(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(F)(F)F
CC(C)(OC(=O)Nc1ccc2O[C@@H](C[C@](C)(CO)C(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(F)(F)F
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](C[C@@](C)(O)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
C[C@@](O)(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(O)=O |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](C[C@](C)(O)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CC(O)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
C[C@](O)(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(O)=O |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CC(O)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CC(C)(CO)C(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CC(C)(CO)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CC(C)(CO)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
C[C@H](CC(O)=O)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F
C[C@@H](CC(O)=O)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@H](CC(O)=O)C1CC1
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@@H](CC(O)=O)C1CC1
CC(C)(OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)[C@@H](CC(O)=O)C1CC1)C(F)(F)F |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@@H](CC(O)=O)C1CC1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)[C@H](CC(O)=O)C1CC1)C(F)(F)F |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@H](CC(O)=O)C1CC1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)[C@H]1C[C@H]1C(O)=O)C(F)(F)F
CC(C)(OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)[C@@H]1C[C@@H]1C(O)=O)C(F)(F)F
CC(C)(OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)[C@@H]1C[C@H]1C(O)=O)C(F)(F)F
CC(C)(OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)[C@H]1C[C@@H]1C(O)=O)C(F)(F)F
Cc1ccc(cc1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@H]1C[C@H]1C(O)=O |r|
Cc1ccc(cc1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@@H]1C[C@@H]1C(O)=O |r|
Cc1ccc(cc1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@H]1C[C@@H]1C(O)=O |r|
Cc1ccc(cc1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@@H]1C[C@H]1C(O)=O |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@H]1C[C@@H]1C(O)=O |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@@H]1C[C@H]1C(O)=O |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@H]1C[C@H]1C(O)=O |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@@H]1C[C@@H]1C(O)=O |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@H]1C[C@H]1C(O)=O |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@@H]1C[C@@H]1C(O)=O |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@H]1C[C@@H]1C(O)=O |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@@H]1C[C@H]1C(O)=O |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)O[C@H](C(C)(C)C)C(F)(F)F)cc12
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)O[C@@H](C(C)(C)C)C(F)(F)F)cc12
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OCC3(CC3)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC3(CCC3)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)O[C@@H](C)C(C)(C)C)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)O[C@H](C)C(C)(C)C)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC3(CCCCC3)C(F)(F)F)cc12 |r|
CCC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)c(OC)c1)C(F)(F)F |r|
C[C@@H]1[C@H](CCC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1[C@@H](C)[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(Cl)n1)S(=O)(=O)N1[C@H](C)[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(Cl)n1)S(=O)(=O)N1[C@H](C)[C@@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(Cl)n1)S(=O)(=O)N1[C@@H](C)[C@@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
COc1cc(ccc1F)S(=O)(=O)N1[C@@H](C)[C@@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1[C@H](C)[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1cc(F)c2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)C(F)(F)F |r|
Cc1cc(ccc1F)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2c(F)cc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2c(F)cc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2c(F)cc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2c(F)cc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1cc(F)c2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
CC(C)(OC(=O)Nc1cc(F)c2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1cc(F)c2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C1CC1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1cc(F)c2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1ccnc(c1)C(F)(F)F)C(F)(F)F |r|
CC(C)(OC(=O)Nc1cc(F)c2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cncc(c1)C(F)(F)F)C(F)(F)F |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)c(C)c12
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CC(C)(C)C(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)c(C)c12
CCS(=O)(=O)c1ccc(nc1)[C@H](CO)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@@H]3CC[C@H](OC3)C(F)(F)F)Cc2c1 |r|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@@H]3CC[C@H](OC3)C(F)(F)F)Cc2c1 |r|
CC[C@@H]1N(C[C@H]2CC[C@H](OC2)C(F)(F)F)Cc2cc(cnc12)C(=O)N[C@@H](CO)c1ccc(cn1)S(=O)(=O)CC |r|
CCS(=O)(=O)c1ccc(nc1)[C@H](CO)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@H]3CC[C@@H](OC3)C(F)(F)F)Cc2c1 |r|
CC[C@@H]1N(C[C@@H]2CC[C@H](OC2)C(F)(F)F)Cc2cc(cnc12)C(=O)N[C@@H](CO)c1ccc(cn1)S(=O)(=O)CC |r|
CCS(=O)(=O)c1ccc(cc1)C(C)(CO)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)Cc2c1 |r,wU:31.35,wD:28.28,22.23,(12.26,-2.97,;10.91,-3.72,;9.59,-2.93,;8.8,-4.26,;10.38,-1.61,;8.27,-2.15,;8.2,-.53,;6.87,.24,;5.53,-.53,;5.53,-2.07,;6.87,-2.84,;4.2,.24,;4.2,-1.3,;4.2,1.78,;5.53,2.55,;2.87,-.53,;1.53,.24,;1.53,1.78,;.2,-.53,;.2,-2.07,;-1.13,-2.84,;-2.47,-2.07,;-3.93,-2.54,;-4.33,-4.03,;-5.82,-4.43,;-3.24,-5.12,;-4.84,-1.3,;-6.38,-1.3,;-7.15,.04,;-6.38,1.37,;-7.15,2.7,;-8.69,2.7,;-9.46,1.37,;-8.69,.04,;-9.46,4.04,;-8.69,5.37,;-11,4.04,;-10.23,5.37,;-3.93,-.05,;-2.47,-.53,;-1.13,.24,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@H]3CC[C@H](CC3)C(F)(F)F)Cc2c1 |r,wU:27.27,30.34,11.14,wD:21.22,(12.26,-2.97,;10.91,-3.72,;9.59,-2.93,;8.8,-4.26,;10.38,-1.61,;8.27,-2.15,;8.2,-.53,;6.87,.24,;5.53,-.53,;5.53,-2.07,;6.87,-2.84,;4.2,.24,;4.2,1.78,;5.53,2.55,;2.87,-.53,;1.53,.24,;1.53,1.78,;.2,-.53,;.2,-2.07,;-1.13,-2.84,;-2.47,-2.07,;-3.93,-2.54,;-4.33,-4.03,;-5.82,-4.43,;-3.24,-5.12,;-4.84,-1.3,;-6.38,-1.3,;-7.15,.04,;-8.69,.04,;-9.46,1.37,;-8.69,2.7,;-7.15,2.7,;-6.38,1.37,;-9.46,4.04,;-8.69,5.37,;-11,4.04,;-10.23,5.37,;-3.93,-.05,;-2.47,-.53,;-1.13,.24,)|
CCS(=O)(=O)c1ccc(cc1)C(C)(CO)NC(=O)c1cnc2[C@@H](C(C)C)N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)Cc2c1 |r,wU:31.35,22.23,wD:28.28,(12.26,-2.97,;10.91,-3.72,;9.59,-2.93,;8.8,-4.26,;10.38,-1.61,;8.27,-2.15,;8.2,-.53,;6.87,.24,;5.53,-.53,;5.53,-2.07,;6.87,-2.84,;4.2,.24,;4.2,-1.3,;4.2,1.78,;5.53,2.55,;2.87,-.53,;1.53,.24,;1.53,1.78,;.2,-.53,;.2,-2.07,;-1.13,-2.84,;-2.47,-2.07,;-3.93,-2.54,;-4.33,-4.03,;-5.82,-4.43,;-3.24,-5.12,;-4.84,-1.3,;-6.38,-1.3,;-7.15,.04,;-6.38,1.37,;-7.15,2.7,;-8.69,2.7,;-9.46,1.37,;-8.69,.04,;-9.46,4.04,;-8.69,5.37,;-11,4.04,;-10.23,5.37,;-3.93,-.05,;-2.47,-.53,;-1.13,.24,)|
CC[C@@H]1N(C[C@H]2CC[C@@H](OC2)C(F)(F)F)Cc2cc(cnc12)C(=O)N[C@@H](CO)c1ccc(cc1)S(=O)(=O)CC |r|
CC[C@@H]1N(C[C@@H]2CC[C@H](OC2)C(F)(F)F)Cc2cc(cnc12)C(=O)N[C@@H](CO)c1ccc(cc1)S(=O)(=O)CC |r|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1cnc2[C@@H](COC)N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)Cc2c1 |r,wU:30.34,11.14,21.22,wD:27.27,(12.26,-2.97,;10.91,-3.72,;9.59,-2.93,;8.8,-4.26,;10.38,-1.61,;8.27,-2.15,;8.2,-.53,;6.87,.24,;5.53,-.53,;5.53,-2.07,;6.87,-2.84,;4.2,.24,;4.2,1.78,;5.53,2.55,;2.87,-.53,;1.53,.24,;1.53,1.78,;.2,-.53,;.2,-2.07,;-1.13,-2.84,;-2.47,-2.07,;-3.93,-2.54,;-4.37,-4.17,;-5.83,-5.02,;-7.29,-4.17,;-4.84,-1.3,;-6.38,-1.3,;-7.15,.04,;-6.38,1.37,;-7.15,2.7,;-8.69,2.7,;-9.46,1.37,;-8.69,.04,;-9.46,4.04,;-8.69,5.37,;-11,4.04,;-10.23,5.37,;-3.93,-.05,;-2.47,-.53,;-1.13,.24,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1cnc2[C@H](COC)N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)Cc2c1 |r,wU:30.34,11.14,wD:27.27,21.22,(12.26,-2.97,;10.91,-3.72,;9.59,-2.93,;8.8,-4.26,;10.38,-1.61,;8.27,-2.15,;8.2,-.53,;6.87,.24,;5.53,-.53,;5.53,-2.07,;6.87,-2.84,;4.2,.24,;4.2,1.78,;5.53,2.55,;2.87,-.53,;1.53,.24,;1.53,1.78,;.2,-.53,;.2,-2.07,;-1.13,-2.84,;-2.47,-2.07,;-3.93,-2.54,;-4.37,-4.17,;-5.83,-5.02,;-7.29,-4.17,;-4.84,-1.3,;-6.38,-1.3,;-7.15,.04,;-6.38,1.37,;-7.15,2.7,;-8.69,2.7,;-9.46,1.37,;-8.69,.04,;-9.46,4.04,;-8.69,5.37,;-11,4.04,;-10.23,5.37,;-3.93,-.05,;-2.47,-.53,;-1.13,.24,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@@H]3CC[C@H](CO3)C(F)(F)F)Cc2c1 |r|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@H]3CC[C@@H](CO3)C(F)(F)F)Cc2c1 |r|
CC[C@@H]1N(C[C@H]2CC[C@@H](CC2)C(F)(F)F)Cc2cc(cnc12)C(=O)N[C@@H](CO)c1ccc(cn1)S(C)(=O)=O |r,wU:8.11,25.27,wD:5.4,2.1,(-5.83,-4.9,;-4.34,-4.5,;-3.94,-3.01,;-4.85,-1.77,;-6.39,-1.77,;-7.16,-.43,;-6.39,.9,;-7.16,2.23,;-8.7,2.23,;-9.47,.9,;-8.7,-.43,;-9.47,3.57,;-8.7,4.9,;-11.01,3.57,;-10.24,4.9,;-3.94,-.52,;-2.48,-1,;-1.14,-.23,;.19,-1,;.19,-2.54,;-1.14,-3.31,;-2.48,-2.54,;1.52,-.23,;1.52,1.31,;2.86,-1,;4.19,-.23,;4.19,1.31,;5.52,2.08,;5.52,-1,;6.86,-.23,;8.19,-1,;8.26,-2.62,;6.86,-3.31,;5.52,-2.54,;9.58,-3.4,;10.37,-2.08,;10.9,-4.19,;8.79,-4.73,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1cnc2[C@@H](CO)N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)Cc2c1 |r,wU:29.33,11.14,21.22,wD:26.26,(12.26,-2.97,;10.91,-3.72,;9.59,-2.93,;8.8,-4.26,;10.38,-1.61,;8.27,-2.15,;8.2,-.53,;6.87,.24,;5.53,-.53,;5.53,-2.07,;6.87,-2.84,;4.2,.24,;4.2,1.78,;5.53,2.55,;2.87,-.53,;1.53,.24,;1.53,1.78,;.2,-.53,;.2,-2.07,;-1.13,-2.84,;-2.47,-2.07,;-3.93,-2.54,;-4.33,-4.03,;-5.82,-4.43,;-4.84,-1.3,;-6.38,-1.3,;-7.15,.04,;-6.38,1.37,;-7.15,2.7,;-8.69,2.7,;-9.46,1.37,;-8.69,.04,;-9.46,4.04,;-8.69,5.37,;-11,4.04,;-10.23,5.37,;-3.93,-.05,;-2.47,-.53,;-1.13,.24,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@@H]3CC[C@@H](CO3)C(F)(F)F)Cc2c1 |r|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1cnc2[C@@H](Cc3ccccc3)N(CC(F)(F)F)Cc2c1 |r|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1cnc2[C@H](CO)N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)Cc2c1 |r,wU:29.33,11.14,wD:26.26,21.22,(12.26,-2.97,;10.91,-3.72,;9.59,-2.93,;8.8,-4.26,;10.38,-1.61,;8.27,-2.15,;8.2,-.53,;6.87,.24,;5.53,-.53,;5.53,-2.07,;6.87,-2.84,;4.2,.24,;4.2,1.78,;5.53,2.55,;2.87,-.53,;1.53,.24,;1.53,1.78,;.2,-.53,;.2,-2.07,;-1.13,-2.84,;-2.47,-2.07,;-3.93,-2.54,;-4.33,-4.03,;-5.82,-4.43,;-4.84,-1.3,;-6.38,-1.3,;-7.15,.04,;-6.38,1.37,;-7.15,2.7,;-8.69,2.7,;-9.46,1.37,;-8.69,.04,;-9.46,4.04,;-8.69,5.37,;-11,4.04,;-10.23,5.37,;-3.93,-.05,;-2.47,-.53,;-1.13,.24,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@H]3CC[C@H](CO3)C(F)(F)F)Cc2c1 |r|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1cnc2[C@H](Cc3ccccc3)N(CC(F)(F)F)Cc2c1 |r|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1cnc2C(N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)Cc2c1)C(F)(F)F |r,wU:27.31,11.14,wD:24.24,(12.26,-2.89,;10.91,-3.65,;9.59,-2.86,;8.8,-4.18,;10.38,-1.54,;8.27,-2.07,;8.2,-.45,;6.87,.32,;5.53,-.45,;5.53,-1.99,;6.87,-2.76,;4.2,.32,;4.2,1.86,;5.53,2.63,;2.87,-.45,;1.53,.32,;1.53,1.86,;.2,-.45,;.2,-1.99,;-1.13,-2.76,;-2.47,-1.99,;-3.93,-2.47,;-4.84,-1.22,;-6.38,-1.22,;-7.15,.11,;-6.38,1.44,;-7.15,2.78,;-8.69,2.78,;-9.46,1.44,;-8.69,.11,;-9.46,4.11,;-8.69,5.44,;-11,4.11,;-10.23,5.44,;-3.93,.02,;-2.47,-.45,;-1.13,.32,;-4.33,-3.96,;-5.82,-4.36,;-3.24,-5.05,;-4.73,-5.44,)|
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CCS(=O)(=O)c1ccc(nc1)[C@@H](CO)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)Cc2c1 |r,wU:30.34,wD:27.27,11.14,21.22,(12.26,-2.97,;10.91,-3.72,;9.59,-2.93,;8.8,-4.26,;10.38,-1.61,;8.27,-2.15,;8.2,-.53,;6.87,.24,;5.53,-.53,;5.53,-2.07,;6.87,-2.84,;4.2,.24,;4.2,1.78,;5.53,2.55,;2.87,-.53,;1.53,.24,;1.53,1.78,;.2,-.53,;.2,-2.07,;-1.13,-2.84,;-2.47,-2.07,;-3.93,-2.54,;-4.33,-4.03,;-5.82,-4.43,;-3.24,-5.12,;-4.84,-1.3,;-6.38,-1.3,;-7.15,.04,;-6.38,1.37,;-7.15,2.7,;-8.69,2.7,;-9.46,1.37,;-8.69,.04,;-9.46,4.04,;-8.69,5.37,;-11,4.04,;-10.23,5.37,;-3.93,-.05,;-2.47,-.53,;-1.13,.24,)|
CCS(=O)(=O)c1ccc(nc1)[C@H](CO)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)Cc2c1 |r,wU:30.34,11.14,wD:27.27,21.22,(12.26,-2.97,;10.91,-3.72,;9.59,-2.93,;8.8,-4.26,;10.38,-1.61,;8.27,-2.15,;8.2,-.53,;6.87,.24,;5.53,-.53,;5.53,-2.07,;6.87,-2.84,;4.2,.24,;4.2,1.78,;5.53,2.55,;2.87,-.53,;1.53,.24,;1.53,1.78,;.2,-.53,;.2,-2.07,;-1.13,-2.84,;-2.47,-2.07,;-3.93,-2.54,;-4.33,-4.03,;-5.82,-4.43,;-3.24,-5.12,;-4.84,-1.3,;-6.38,-1.3,;-7.15,.04,;-6.38,1.37,;-7.15,2.7,;-8.69,2.7,;-9.46,1.37,;-8.69,.04,;-9.46,4.04,;-8.69,5.37,;-11,4.04,;-10.23,5.37,;-3.93,-.05,;-2.47,-.53,;-1.13,.24,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)Cc2c1 |r,wU:11.14,30.34,wD:21.22,27.27,(10.77,-19.48,;9.58,-20.17,;8.39,-19.48,;7.7,-20.67,;9.08,-18.29,;7.2,-18.8,;6.16,-19.73,;4.83,-18.96,;4.83,-17.42,;6.16,-16.65,;7.49,-17.42,;3.49,-16.65,;3.49,-15.11,;4.83,-14.34,;2.16,-17.42,;.83,-16.65,;.83,-15.11,;-.51,-17.42,;-.51,-18.96,;-1.84,-19.73,;-3.18,-18.96,;-4.64,-19.44,;-5.04,-20.93,;-3.95,-22.02,;-6.53,-21.33,;-5.55,-18.19,;-7.09,-18.19,;-7.48,-16.71,;-6.4,-15.62,;-6.79,-14.13,;-8.28,-13.73,;-9.37,-14.82,;-8.97,-16.31,;-8.68,-12.24,;-7.59,-11.15,;-10.17,-11.85,;-9.08,-10.76,;-4.64,-16.95,;-3.18,-17.42,;-1.84,-16.65,)|
CCS(=O)(=O)c1ccc(cc1)[C@@H](CO)NC(=O)c1cnc2[C@H](C(C)C)N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)Cc2c1 |r,wU:27.27,wD:30.34,11.14,21.22,(12.26,-2.97,;10.91,-3.72,;9.59,-2.93,;8.8,-4.26,;10.38,-1.61,;8.27,-2.15,;8.2,-.53,;6.87,.24,;5.53,-.53,;5.53,-2.07,;6.87,-2.84,;4.2,.24,;4.2,1.78,;5.53,2.55,;2.87,-.53,;1.53,.24,;1.53,1.78,;.2,-.53,;.2,-2.07,;-1.13,-2.84,;-2.47,-2.07,;-3.93,-2.54,;-4.33,-4.03,;-5.82,-4.43,;-3.24,-5.12,;-4.84,-1.3,;-6.38,-1.3,;-7.15,.04,;-8.69,.04,;-9.46,1.37,;-8.69,2.7,;-7.15,2.7,;-6.38,1.37,;-9.46,4.04,;-8.69,5.37,;-11,4.04,;-10.23,5.37,;-3.93,-.05,;-2.47,-.53,;-1.13,.24,)|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CO)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CO)CN(c2c1)S(=O)(=O)c1cc(Br)cnc1Cl |r|
Cc1nn(cc1S(=O)(=O)N1C[C@H](CO)Oc2ccc(NC(=O)OC(C)(C)C)cc12)C(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CO)CN(c2c1)S(=O)(=O)c1cccc(Cl)c1 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CO)CN(c2c1)S(=O)(=O)c1cncc(Br)c1 |r|
Cn1cc(cn1)S(=O)(=O)N1C[C@H](CO)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
Cc1cccc(c1)S(=O)(=O)N1C[C@H](CO)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
Cc1cnc(Cl)c(c1)S(=O)(=O)N1C[C@H](CO)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CO)CN(c2c1)S(=O)(=O)c1cccc(c1)C#N |r|
Cc1c[nH]c(=O)c(c1)S(=O)(=O)N1C[C@H](CO)Oc2ccc(NC(=O)OC(C)(C)C)cc12
CC(C)(C)OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(C)(C)O
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(C)(C)O
CC(C)(OC(=O)Nc1ccc2O[C@@H](CN(c2c1)S(=O)(=O)c1ccc(F)c(F)c1)C(=O)C(F)(F)F)C(F)(F)F
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(=O)C(F)(F)F
CC(C)(OC(=O)Nc1ccc2O[C@@H](CN)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)OCc3ccccc3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)NC3CCOCC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CNC(=O)OCc3ccccc3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)OCc3ccccc3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
COC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CNC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)NC3CC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)NC3CCC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(C)NC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)NC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)Nc3ccsc3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CCNC(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNC(=O)NC3CCCCC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CN1CCN(C[C@H]2CN(c3cc(ccc3O2)N(C([O-])=O)C(C)(C)C(F)(F)F)S(=O)(=O)c2ccc(F)c(Cl)c2)S1(=O)=O
CNS(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)N3CCOCC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CCN(CC)S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CN(C)S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)N3CCCCC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)N3CCCC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC1CCCCN1S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC1CN(CC(C)O1)S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC1CCN(CC1)S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC1CN(CCO1)S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CN(C1CC1)S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CN(C1CCCC1)S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CN(CC(F)(F)F)S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CNS(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CNS(=O)(=O)N3CCCCC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(F)(F)F |r|
CC1CCCCN1S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC1CN(CCO1)S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CN(CC(F)(F)F)S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC(C)CN(C)S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC1CCN(C1)S(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CCNS(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC(C)NS(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CCNS(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)NS(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(C)NS(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CNS(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(F)c1 |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@H](CNS(=O)(=O)NC)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(C)n1)S(=O)(=O)N1C[C@H](CNS(=O)(=O)NC)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CNS(=O)(=O)NC)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCC(F)F)n1)S(=O)(=O)N1C[C@H](CNS(=O)(=O)NC)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC(F)F)cc1S(=O)(=O)N1C[C@H](CNS(=O)(=O)NC)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CNS(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CNS(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1c(OC)nn2CCCc12 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CSc3ccccn3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CSC3CCCC3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CSCc3ccccc3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CSC(C)(C)C)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
Cc1nc(SC[C@H]2CN(c3cc(NC(=O)OC(C)(C)C)ccc3O2)S(=O)(=O)c2cccc(c2)C(F)(F)F)[nH]c1C |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CSc3ccccc3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CSC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CS(=O)(=O)c3ccccn3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CS(=O)(=O)C(C)(C)C)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
Cc1nc([nH]c1C)S(=O)(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CS(=O)(=O)c3ccccc3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CS(=O)(=O)C3CCCC3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CS(=O)(=O)Cc3ccccc3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CS(C)(=O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CS(=O)(=O)NC3CC3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CS(=O)(=O)NCC(F)(F)F)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CS(=O)(=O)N3CCOCC3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CCNS(=O)(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CN(C)S(=O)(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@H](C)Oc2ccc(cc12)N(C([O-])=O)C(C)(C)C(F)(F)F
C[C@@H]1[C@H](CO)Oc2ccc(NC(=O)OCC(C)(C)C)cc2N1S(=O)(=O)c1cccc(c1)C#N
C[C@H]1COc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1ccc(F)cc1
C[C@@H]1COc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1ccc(F)cc1
CC(C)(OC(=O)Nc1ccc2OC[C@@H](CO)N(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
CC(C)(OC(=O)Nc1ccc2OC[C@H](CO)N(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CN3C(=O)COC3=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C#N
O=C(Nc1ccc2O[C@@H](CN3C(=O)COC3=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C#N)O[C@@H]1C[C@@H]2CC[C@H]1C2 |r|
CC(C)(C)COC(=O)Nc1ccc2O[C@@H](CN3C(=O)COC3=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C#N |r|
Cn1cc(cn1)S(=O)(=O)N1C[C@H](CN2C(=O)COC2=O)Oc2ccc(NC(=O)OC3C[C@@H]4CC[C@H]3C4)cc12 |r|
Cn1cc(cn1)S(=O)(=O)N1C[C@H](CN2C(=O)COC2=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
Cn1cc(cn1)S(=O)(=O)N1C[C@H](CN2C(=O)COC2=O)Oc2ccc(NC(=O)OCC(C)(C)C)cc12 |r|
Cn1cc(cn1)S(=O)(=O)N1C[C@H](CN2C(=O)COC2=O)Oc2ccc(NC(=O)OCC3CCCCO3)cc12 |r|
O=C(Nc1ccc2O[C@@H](CN3C(=O)COC3=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C#N)O[C@H]1CC2CCC1C2 |r|
Cn1cc(cn1)S(=O)(=O)N1C[C@H](CN2C(=O)COC2=O)Oc2ccc(NC(=O)O[C@H]3CC4CCC3C4)cc12 |r|
CN(C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C#N
CN(C)C[C@H]1CN(c2cc(NC(=O)OCC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C#N
CN(C)C[C@H]1CN(c2cc(NC(=O)OC3C[C@@H]4CC[C@H]3C4)ccc2O1)S(=O)(=O)c1cccc(c1)C#N |r|
CN(C)C[C@H]1CN(c2cc(NC(=O)O[C@@H]3C[C@@H]4CC[C@H]3C4)ccc2O1)S(=O)(=O)c1cccc(c1)C#N |r|
CN(C)C[C@H]1CN(c2cc(NC(=O)OCC(C)(C)C)ccc2O1)S(=O)(=O)c1cnn(C)c1 |r|
CN(C)C[C@H]1CN(c2cc(NC(=O)OC3CC4CCC3C4)ccc2O1)S(=O)(=O)c1cnn(C)c1 |r|
CN(C)C[C@H]1CN(c2cc(NC(=O)O[C@H]3CC4CCC3C4)ccc2O1)S(=O)(=O)c1cnn(C)c1 |r|
CN(C)C[C@H]1CN(c2cc(NC(=O)OC3CCOCC3)ccc2O1)S(=O)(=O)c1cccc(c1)C#N |r|
COC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F
COC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
COC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F |r|
COC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)c(OC)c1 |r|
COC(=O)C[C@@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
COC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F |r|
Cc1nn(cc1S(=O)(=O)N1C[C@H](CC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12)C(F)F
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(C)COC(=O)Nc1ccc2O[C@@H](CC(O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(Cl)c1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CC(O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(O)=O
CC(C)(C)OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(O)=O |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C)cc12)C(O)=O |r|
CC(C)(OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)C(O)=O)C(F)(F)F |r|
Cc1nn(cc1S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C)cc12)C(O)=O)C(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)C(O)=O |r|
Cc1nn(cc1S(=O)(=O)N1C[C@H](CC(=O)N2CCC2)Oc2ccc(NC(=O)OC(C)(C)C)cc12)C(F)F
CC(OC(=O)Nc1ccc2O[C@@H](CC(=O)N3CCC3)CN(c2c1)S(=O)(=O)c1cn(nc1C)C(F)F)C(C)(C)C
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(N)=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(N)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CNC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CNC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CN(C)C(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CN(C)C(=O)CC1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1
CNC(=O)C[C@@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CNC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CNC(=O)CC1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1
CC(C)(C)OC(=O)Nc1ccc2O[C@H](CC(=O)N3CCOC3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NCC3CCC3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NCCC(F)(F)F)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)CNC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NCc3cn[nH]c3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
Cn1cc(CNC(=O)C[C@H]2CN(c3cc(NC(=O)OC(C)(C)C)ccc3O2)S(=O)(=O)c2cccc(c2)C(F)(F)F)cn1 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NCc3cc[nH]n3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)n1cc(CNC(=O)C[C@H]2CN(c3cc(NC(=O)OC(C)(C)C)ccc3O2)S(=O)(=O)c2cccc(c2)C(F)(F)F)cn1 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NCc3cnn4ccccc34)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CCn1ccc(CNC(=O)C[C@H]2CN(c3cc(NC(=O)OC(C)(C)C)ccc3O2)S(=O)(=O)c2cccc(c2)C(F)(F)F)n1 |r|
Cn1ncc2CN(Cc12)C(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
Cn1ccc(CNC(=O)C[C@H]2CN(c3cc(NC(=O)OC(C)(C)C)ccc3O2)S(=O)(=O)c2cccc(c2)C(F)(F)F)n1 |r|
CCn1cc(CNC(=O)C[C@H]2CN(c3cc(NC(=O)OC(C)(C)C)ccc3O2)S(=O)(=O)c2cccc(c2)C(F)(F)F)cn1 |r|
CCn1ncc(CNC(=O)C[C@H]2CN(c3cc(NC(=O)OC(C)(C)C)ccc3O2)S(=O)(=O)c2cccc(c2)C(F)(F)F)c1C |r|
Cc1c(CNC(=O)C[C@H]2CN(c3cc(NC(=O)OC(C)(C)C)ccc3O2)S(=O)(=O)c2cccc(c2)C(F)(F)F)cnn1C |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NCc3cnn(Cc4ccccc4)c3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NCCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
COC(=O)CCNC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NCc3ccc(cc3)C(F)(F)F)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NCc3ccccc3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NCC3CC3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CCCNC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CCNC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)N3CCOC3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CNC(=O)C[C@H]1CN(c2cc(NC(=O)OCC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NCc3nn[nH]n3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NCCO)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)NC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC1CCN1C(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)N3CC(C3)C#N)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
COC1CN(C1)C(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)N3CCC3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)N3CCC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NCc3cc[nH]n3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
Cc1nn(cc1S(=O)(=O)N1C[C@H](CC(=O)N2CCC2)Oc2ccc(NC(=O)OCC(C)(C)C)cc12)C(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)C(N)=O |r|
CC(C)(OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)C(N)=O)C(F)(F)F |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C)cc12)C(N)=O |r|
COC(=O)CCNC(=O)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
Cc1nn(cc1S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C)cc12)C(N)=O)C(F)F |r|
CN(C)C(=O)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)C(=O)NCCC(O)=O |r|
CC(C)(C)OC(=O)Nc1ccc2OC(CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(C)(C)C#N
CC(C)(OC(=O)Nc1ccc2O[C@@H](CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(C)(C)C(O)=O)C(F)(F)F
Cn1c(n[nH]c1=O)C(C)(C)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NS(=O)(=O)C(F)(F)F)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
CC(C)(C)COC(=O)Nc1ccc2O[C@@H](CC(=O)NS(=O)(=O)C3CC3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
Cc1nn(cc1S(=O)(=O)N1C[C@H](CC(=O)NS(=O)(=O)C(F)(F)F)Oc2ccc(NC(=O)OCC(C)(C)C)cc12)C(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NS(=O)(=O)c3nccs3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NS(=O)(=O)c3ccncc3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NS(=O)(=O)C(C)(C)C)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NS(=O)(=O)c3ccc(cn3)C(F)(F)F)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)COC(=O)Nc1ccc2O[C@@H](CC(=O)NS(=O)(=O)C(F)(F)F)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NS(=O)(=O)c3ccccn3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NS(=O)(=O)c3cccnc3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NS(=O)(=O)c3cc(ccn3)C(F)(F)F)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NS(=O)(=O)c3cn[nH]c3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
Cc1ccnc(c1)S(=O)(=O)NC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
Cc1ccc(F)c(c1)S(=O)(=O)NC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NS(=O)(=O)c3ccccc3F)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NS(=O)(=O)c3ccccc3C(F)(F)F)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NS(=O)(=O)c3cccc(c3)C(F)(F)F)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NS(=O)(=O)c3cccc(F)c3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NS(=O)(=O)C3CC3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
Cc1ccc(cc1)S(=O)(=O)NC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)S(=O)(=O)NC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CCS(=O)(=O)NC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NS(C)(=O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
Cc1nn(cc1S(=O)(=O)N1C[C@H](CC(=O)NS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OCC(C)(C)C)cc12)C(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NS(=O)(=O)C3CCCC3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
Cc1ccccc1S(=O)(=O)NC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NS(=O)(=O)c3ccc(F)cc3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
Cc1ccc(C)c(c1)S(=O)(=O)NC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CCCc1ccc(cc1)S(=O)(=O)NC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
Cc1cccc(n1)S(=O)(=O)NC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)COC(=O)Nc1ccc2O[C@@H](CC(=O)NS(=O)(=O)C3CC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
CONC(=O)C[C@H]1CN(c2cc(NC(O)=O)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NOc3ccccc3C(F)(F)F)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NOCc3cccnc3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NOCc3ccc(cc3)C(F)(F)F)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NOCc3cccc(c3)C(F)(F)F)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NOc3ccc(F)cc3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NOC3CCCC3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CCONC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CC(=O)NOCc3ccccc3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
Cc1ccc(CONC(=O)C[C@H]2CN(c3cc(NC(=O)OC(C)(C)C)ccc3O2)S(=O)(=O)c2cccc(c2)C(F)(F)F)cc1 |r|
CC(C)ONC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CCCONC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)cc1)c1n[nH]c(=O)o1
CC(C)(OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)cc1)c1n[nH]c(=O)o1)C(F)(F)F |r|
Cc1nn(cc1S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C)cc12)c1n[nH]c(=O)o1)C(F)F |r|
Cc1nn(cc1S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)c1n[nH]c(=O)o1)C(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)c(Cl)c1)c1n[nH]c(=O)o1 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)c1n[nH]c(=O)o1 |r|
Cn1nc(C[C@H]2CN(c3cc(NC(=O)OC(C)(C)C)ccc3O2)S(=O)(=O)c2ccc(F)cc2)oc1=O |r|
Cc1nn(cc1S(=O)(=O)N1C[C@H](Cc2nn(C)c(=O)o2)Oc2ccc(NC(=O)OC(C)(C)C)cc12)C(F)F |r|
Cn1nc(C[C@H]2CN(c3cc(NC(=O)OC(C)(C)C)ccc3O2)S(=O)(=O)c2cccc(c2)C(F)(F)F)oc1=O |r|
Cn1c(n[nH]c1=O)[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1
CC(C)(C)OC(=O)Nc1ccc2OC(CC#N)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
CC(O)CC1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F
CC(C)(N)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F
CC(=O)NC(C)(C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F
CCC(=O)NCC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(O)C(=O)NCC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CCNC(=O)C3COC3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)C(=O)NCC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(=O)NCC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CCNC(=O)C3CC3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CCC(=O)NCC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NCC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(O)C(=O)NCC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CCNC(=O)C3CC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
CCC(=O)NCC[C@H]1CN(c2cc(NC(=O)OCC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NCC[C@H]1CN(c2cc(NC(=O)OCC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(C)COC(=O)Nc1ccc2O[C@@H](CCNC(=O)C3CC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(N)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC(C)(N)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@H](CCN3CCCC3=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCN3CCCC3=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
CC(=O)NC(C)(C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1
CC(=O)NC(C)(C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)c(F)c1 |r|
CC(=O)NC(C)(C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(=O)NC(C)(C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cnn(C(F)F)c1C |r|
CC(=O)NC(C)(C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC(C)(C)C[C@@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC(C)(C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F
CC(=O)NC(C)(C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC(C)(C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1 |r|
CC(=O)NC(C)(C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CC(C)(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1)NS(C)(=O)=O |r|
CC(=O)NC(C)(C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(F)c1 |r|
CC(C)(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1)NS(C)(=O)=O |r|
CC(C)(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(F)c1)NS(C)(=O)=O |r|
CC(C)(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(F)c1)NS(=O)(=O)C1CC1 |r|
CC(C)(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F)NS(C)(=O)=O |r|
CC(C)(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F)NS(=O)(=O)C1CC1 |r|
CC(C)(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(Cl)c1)NS(=O)(=O)C1CC1 |r|
CC(C)(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1)NS(=O)(=O)C1CC1 |r|
CC(C)(C[C@@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1)NS(=O)(=O)C1CC1 |r|
CC(C)(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F)NS(=O)(=O)C(F)(F)F |r|
CN(C)C(=O)C(=O)NC(C)(C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(=O)NC(C)(C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CC(C)(C)NC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1nc(OC)c(c1C)S(=O)(=O)N1C[C@H](CC(C)(C)NC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(cc1S(=O)(=O)N1C[C@H](CC(C)(C)NC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)C(F)F |r|
CCn1cc(c(OC(F)F)n1)S(=O)(=O)N1C[C@H](CC(C)(C)NC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(C)OC(=O)Nc1ccc2OC(CCO)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
CC(C)(C)OC(=O)Nc1ccc2OC(Cc3ncc[nH]3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
Cn1ccnc1CC1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CN3CCCC3=O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](Cn3cccn3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
Cc1nn(cc1S(=O)(=O)N1C[C@H](Cn2nccn2)Oc2ccc(NC(=O)OC(C)(C)C)cc12)C(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](Cn3cnnc3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](Cn3cncn3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
Cc1nn(cc1S(=O)(=O)N1C[C@H](Cn2ccnn2)Oc2ccc(NC(=O)OC(C)(C)C)cc12)C(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](Cn3ccnn3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](Cn3nccn3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](COc3ccccn3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](Cn3ccccc3=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](Cc3nc(=O)o[nH]3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
CC(C)(O)CC1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CN3CC(O)C3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CNC3(C)COC3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
CC1CCN1C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CN3CC(O)C3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CN3CCC3)CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
C[C@H]1CCc2ncc(NC(=O)OC(C)(C)C)cc2N1S(=O)(=O)c1ccc(F)cc1
CC(C)(C)OC(=O)Nc1cnc2C[C@@H](CN(c2c1)S(=O)(=O)c1ccc(F)cc1)NC(=O)OCc1ccccc1
CC(C)(C)OC(=O)NC1CN(c2cc(NC(=O)OCc3ccccc3)cnc2C1)S(=O)(=O)c1cccc(c1)C(F)(F)F
CC(C)(C)OC(=O)NC1CN(c2cc(NC(=O)OCc3ccccc3)cnc2C1)S(=O)(=O)c1cccc(c1)C#N
Cc1nn(cc1S(=O)(=O)N1CC(Cc2ncc(NC(=O)OCc3ccccc3)cc12)NC(=O)OC(C)(C)C)C(F)F
Fc1ccc(cc1)S(=O)(=O)N1C[C@H](Cc2ncc(NC(=O)OCc3ccccc3)cc12)N1CCCC1=O
CC(C)(C)COC(=O)Nc1cnc2C[C@@H](CN(c2c1)S(=O)(=O)c1ccc(F)cc1)N1CCCC1=O
CC(C)(C)COC(=O)Nc1cnc2C[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)cc1)N1CCCC1=O
CC(C)(C)OC(=O)Nc1cnc2CC(O)CN(c2c1)S(=O)(=O)c1ccc(F)cc1
Cc1nn(cc1S(=O)(=O)N1C[C@H](CO)Cc2ncc(NC(=O)OCC(C)(C)C)cc12)C(F)F
Cc1nn(cc1S(=O)(=O)N1C[C@@H](CO)Cc2ncc(NC(=O)OCC(C)(C)C)cc12)C(F)F
Cc1cccc(c1)S(=O)(=O)N1CC(CO)Cc2ncc(NC(=O)OC(C)(C)C)cc12
CC(C)(C)OC(=O)Nc1cnc2CC(CO)CN(c2c1)S(=O)(=O)c1ccc(F)c(F)c1
CC(C)(C)COC(=O)Nc1cnc2C[C@@H](CO)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(C)COC(=O)Nc1cnc2C[C@H](CO)CN(c2c1)S(=O)(=O)c1ccc(F)cc1 |r|
Cc1nn(cc1S(=O)(=O)N1C[C@H](CN2CC[C@@H](O)C2)Cc2ncc(NC([O-])=O)cc12)C(F)F
CC(C)(OC(=O)Nc1ccc2OC(CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(=O)C(F)(F)F)C(F)(F)F
CNS(=O)(=O)NC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(nc1OCCO)C(F)F |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@H](CC(C)(C)NC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)c(F)c1)[C@H](O)C(F)(F)F)C(F)(F)F
CC(C)(OC(=O)Nc1ccc2O[C@@H](CN(c2c1)S(=O)(=O)c1ccc(F)c(F)c1)[C@@H](O)C(F)(F)F)C(F)(F)F
CC(C)(OC(=O)Nc1ccc2O[C@@H](CN(c2c1)S(=O)(=O)c1ccc(F)c(F)c1)[C@H](O)C(F)(F)F)C(F)(F)F
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@H](O)C(F)(F)F |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@@H](O)C(F)(F)F |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12)[C@@H](O)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2OC(CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(O)C(F)(F)F)C(F)(F)F
CC(C)(OC(=O)Nc1ccc2O[C@@H](CN(c2c1)S(=O)(=O)c1ccc(F)cc1)[C@@H](N)C(F)(F)F)C(F)(F)F
CC(C)(OC(=O)Nc1ccc2O[C@@H](CN(c2c1)S(=O)(=O)c1ccc(F)cc1)[C@H](N)C(F)(F)F)C(F)(F)F
CC(C)(OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)cc1)[C@@H](N)C(F)(F)F)C(F)(F)F
CC(C)(OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)cc1)[C@H](N)C(F)(F)F)C(F)(F)F
CCS(=O)(=O)CC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F
CCS(=O)(=O)CC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F
CNS(=O)(=O)NC[C@@H]1Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N([C@@H]1C)S(=O)(=O)c1cn(nc1C)C(F)F
C[C@@H]1[C@H](CNCOC(O)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1ccc(F)c(F)c1
CC(=O)NC[C@H]1COc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1ccc(F)cc1
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](CC2(CC2)C(N)=O)Oc2ccc(cc12)N(C([O-])=O)C(C)(C)C(F)(F)F
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CC2(CC2)C(N)=O)Oc2ccc(cc12)N(C([O-])=O)C(C)(C)C(F)(F)F
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](C[C@H](C2CC2)C(N)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](C[C@@H](C2CC2)C(N)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](CC(C)(C)C(N)=O)Oc2ccc(cc12)N(C([O-])=O)C(C)(C)C(F)(F)F
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CC(C)(C)C(N)=O)Oc2ccc(cc12)N(C([O-])=O)C(C)(C)C(F)(F)F
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](CC(C)(C)C(N)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CC(C)(C)C(N)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CC(C)(C)C(N)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](C[C@@H](C2CC2)C(N)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@H](C[C@@H](C2CC2)C(N)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](C[C@H](C2CC2)C(N)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@H](C[C@H](C2CC2)C(N)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cncc(c1)C(F)(F)F)C(N)=O |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@H](CC(C)(C)C(N)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)N1C[C@H](CC(C)(C)C(N)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(OCC(=O)OC)n1)S(=O)(=O)N1C[C@H](CC(C)(C)C(N)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC#N)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(F)(F)F
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CC2(CC2)C#N)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](CC2(CC2)C#N)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CC(C)(C)C#N)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](CC(C)(C)C#N)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CC(C)(C[C@@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)C#N |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@@H](CC(C)(C)C#N)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
Cc1cc(ccc1F)S(=O)(=O)N1C[C@@H](CC(C)(C)C#N)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CC(C)(C)C#N)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
Cc1cc(ccc1F)S(=O)(=O)N1C[C@H](CC(C)(C)C#N)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@@H](CC(C)(C)C#N)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@H](CC(C)(C)C#N)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(=O)NS(=O)(=O)C3CC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)C(F)(F)F
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](C[C@H](C)C(=O)NS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](C[C@@H](C)C(=O)NS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CC(C)(C)S(=O)(=O)NC(=O)CC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F |r|
Cc1ccc(cc1)S(=O)(=O)NC(=O)CC[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCC(=O)NS(=O)(=O)C(F)(F)F)CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)C(F)(F)F |r|
CC(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(=O)NS(=O)(=O)C1CC1 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](C[C@@H](C)C(=O)NS(=O)(=O)C(C)(C)C)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](C[C@@H](C)C(=O)NS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](C[C@@H](C)C(=O)NS(=O)(=O)C(C)(C)C)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](C[C@H](C)C(=O)NS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](C[C@H](C)C(=O)NS(=O)(=O)C(C)(C)C)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](C[C@H](C)C(=O)NS(=O)(=O)C(C)(C)C)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CC3COC3)CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)C(F)(F)F
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CCc2n[nH]c(=O)[nH]2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CCc2n[nH]c(=O)n2C)Oc2ccc(cc12)N(C([O-])=O)C(C)(C)C(F)(F)F
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCc3noc(=O)[nH]3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(F)(F)F
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](CC(C)(C)c2noc(=O)[nH]2)Oc2ccc(cc12)N(C([O-])=O)C(C)(C)C(F)(F)F
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CC(C)(C)c2noc(=O)[nH]2)Oc2ccc(cc12)N(C([O-])=O)C(C)(C)C(F)(F)F
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCc3noc(=O)[nH]3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCc3noc(=O)[nH]3)CN(c2c1)S(=O)(=O)c1cccc(c1)C1CC1)C(F)(F)F |r|
CC(C)(C)OC(=O)Nc1ccc2O[C@@H](CCc3noc(=O)[nH]3)CN(c2c1)S(=O)(=O)c1cccc(c1)C1CC1 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CCc2noc(=O)[nH]2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CCc2noc(=O)[nH]2)Oc2ccc(NC(=O)OC(C)(C)C)cc12 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](CC(C)(C)c2noc(=O)[nH]2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@@H](CC(C)(C)c2noc(=O)[nH]2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CC(C)(C)c2noc(=O)[nH]2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CC(C)(C)c2noc(=O)[nH]2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CCc2n[nH]c(=O)o2)Oc2ccc(cc12)N(C([O-])=O)C(C)(C)C(F)(F)F
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CC(C)(C)c2n[nH]c(=O)o2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCc3n[nH]c(=O)o3)CN(c2c1)S(=O)(=O)c1cccc(c1)C1CC1)C(F)(F)F |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CC(C)(C)c2n[nH]c(=O)o2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(N(C([O-])=O)c1ccc2O[C@@H](CCc3nnn[nH]3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(F)(F)F
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCc3nnn[nH]3)CN(c2c1)S(=O)(=O)c1cccc(c1)C1CC1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCc3nnn[nH]3)CN(c2c1)S(=O)(=O)c1ccnc(c1)C(F)(F)F)C(F)(F)F |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CCc2nnn[nH]2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
Cc1c(ccc2O[C@@H](CO)CN(c12)S(=O)(=O)c1cccc(c1)C(F)(F)F)N(C([O-])=O)C(C)(C)C(F)(F)F
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](CS(=O)(=O)CC)Cc2ncc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CS(=O)(=O)CC)Cc2ncc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](CCC(O)=O)Cc2ncc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CCC(O)=O)Cc2ncc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CC(C)(OC(=O)Nc1ccc2CCCN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F
CCn1cc(c(Cl)n1)S(=O)(=O)N1CCCc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(OCCO)n1)S(=O)(=O)N1CCCc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCOc1nn(CC)cc1S(=O)(=O)N1CCCc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CC(C)(OC(=O)Nc1ccc2CCCN(c2c1)S(=O)(=O)c1ccnc(c1)C(F)(F)F)C(F)(F)F
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CNC(C)=O)Cc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
COc1cc(ccc1F)S(=O)(=O)N1C[C@@H](CNC(C)=O)Cc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CCC(O)=O)Cc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](CCC(O)=O)Cc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CC(C)(OC(=O)Nc1ccc2C[C@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cncc(c1)C(F)(F)F)C(F)(F)F |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@@H](CCC(O)=O)Cc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2C[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cncc(c1)C(F)(F)F)C(F)(F)F |r|
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CCC(O)=O)Cc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2C(=O)CCN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)C(F)(F)F
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3CCCCc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3CCCc23)c(F)c1
CC(C)(C)OC(=O)N1CCc2c(CC1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C(F)(F)F
OC(=O)c1ccc(cc1O)-c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CCCCc12
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3CC3)c3CCCCc23)c(F)c1
OC1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1
CC(C)(C)OC(=O)N1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3CC3)c3CCCC(=O)c23)c(F)c1
COC1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3CC3)c3CC(=O)CCc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3CC3)c3CCCCCc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3CCC3)c3CCCCc23)c(F)c1
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2Cl)c2CCCCc12
OC(=O)c1cc(F)c(cc1O)-c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CCCCc12
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3CCNCCc23)c(F)c1
OC(=O)c1ccc(-c2nn(Cc3c(Cl)cccc3C(F)(F)F)c3CCCCc23)c(F)c1
OC(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1
CN(C)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3CC3)c3CC(CCc23)C(=O)N2CCC2)c(F)c1
CNC(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1
CC(C)(C)OC(=O)N1CCCc2c1c(nn2C(=O)c1c(Cl)cccc1C1CC1)-c1ccc(cc1F)C(O)=O
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CCOCc12
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3CC3)c3COCCc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3COCCc23)c(F)c1
CC(=O)N1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1
COC(=O)N1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C#N
CS(=O)(=O)C1CN(C1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CCC1)C#N
CN1CCN(CC1=O)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CCC1)C#N
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(C(O)=O)c(C)c1)C(=O)c1c(Cl)cccc1C1CC1
COC(=O)N1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CC1(CC1)OC(=O)N1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CN(CCc23)C(=O)OCC2CC2)c(F)c1
CC(C)(C)OC(=O)N1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CN(C)C(=O)N1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CCN(C)C(=O)N1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CN(C(=O)N1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F)c1ccccc1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CN(CCc23)C(=O)N2CCCC2)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CN(CCc23)C(=O)N2CCOCC2)c(F)c1
CN1CCN(CC1)C(=O)N1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CC(C)(C)NC(=O)N1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CN1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CC(C)N1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CN(CC4CC4)CCc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CNCCc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3CC3)c3CNCCc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CC(CCc23)C(=O)N2CCC3(COC3)C2)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)c(F)ccc3C3CC3)c3CC(CCc23)C(=O)N2CC(C2)N2CC(F)C2)c(F)c1
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(C(O)=O)c(C)c1)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
Cc1cc(ccc1C(O)=O)-c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)N1CC2(C1)CCCO2
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CC(CCc23)C(=O)N2CC3(C2)CCCO3)c(F)c1
CN(C)[C@@H]1CCN(C1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |r|
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CC(CCc23)C(=O)N2CCC3(CCCO3)C2)c(F)c1
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)F
COC1(C)CN(C1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CC(CCc23)C(=O)N2CCC(C2)N2CCC2)c(F)c1
CN(C)C1CN(CC1(F)F)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
COC1(C)CN(C1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)F
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(C(O)=O)c(c1)C(F)(F)F)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)F)c3CC(CCc23)C(=O)N2CCC3(COC3)C2)c(F)c1
O[C@@H]1CN(C[C@@H]1F)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)F |r|
Cn1nc(c2CN(CCc12)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F)C(F)(F)F
CN(Cc1nccn1C)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CC(N(C)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F)c1ccn[nH]1
CN(Cc1ccn[nH]1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CN(Cc1ccon1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CC(C)n1cc(CN(C)C(=O)C2CCc3c(C2)n(nc3-c2ccc(cc2F)C(O)=O)C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)cn1
CN(Cc1csc(C)n1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CN(Cc1ccccn1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CN(Cc1cccnc1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CN(Cc1ccncc1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CN(CCn1cccn1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CN(CCn1ccnc1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CN(CCc1cnn(C)c1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CN(Cc1cnn(C)c1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
Cn1ncc2CN(Cc12)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CC(CCc23)C(=O)N2CCc3[nH]ncc3C2)c(F)c1
Cn1cc2CN(CCc2n1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CC(CCc23)C(=O)N2CCn3ncnc3C2)c(F)c1
Cc1nc2CN(Cc2[nH]1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CN(C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F)c1cnn(C)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CC(CCc23)C(=O)N2Cc3ncsc3C2)c(F)c1
Cc1nc2CN(Cc2s1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CC(CCc23)C(=O)N2CC[C@H](C2)C#N)c(F)c1 |r|
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CC(CCc23)C(=O)N2CCOCC2)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CC(CCc23)C(=O)N2CCOC3(CC3)C2)c(F)c1
CO[C@H]1CN(C[C@@H]1O)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |r|
CN(C)[C@H]1CN(C[C@@H]1O)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |r|
COCCN(C)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CN(C)CCNC(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
CN(C)CCN(C)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CC(CCc23)C(=O)N2CC3(COC3)C2)c(F)c1
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1C(F)(F)F)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CC(CCc23)C(=O)N2CC(C2)N2CC(F)C2)c(F)c1
CN(C)C1CN(C1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
OC1CN(C1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
OC1CCN(CC1)C(=O)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
OC(=O)c1ccc(-c2nn(C(=O)c3c(cccc3C3(CC3)C(F)(F)F)C(F)F)c3CC(CCc23)C(=O)N2CCC3(COC3)C2)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3CC3)c3CC(CCc23)NC2COC2)c(F)c1
CC(C)(C)OC(=O)NC1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3CC3)c3CC(CCc23)NCC(F)(F)F)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3CC3)c3CCCNc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CCCNc23)c(F)c1
CN1CCCc2c1c(nn2C(=O)c1c(Cl)cccc1C1CC1)-c1ccc(cc1F)C(O)=O
COC1CN(C1)C(=O)C1CNc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1
Cn1cc(COC2CCc3c(C2)n(nc3-c2ccc(cc2F)C(O)=O)C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)cn1
COC1CN(C1)C(=O)NC1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
COC1CN(C1)C(=O)N(C)C1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CC(CCc23)NC(=O)C2CCC2)c(F)c1
OCC1CCc2c(C1)n(nc2-c1ccc(cc1F)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CCCSc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CCCS(=O)c23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CCCS(=O)(=O)c23)c(F)c1
CN1CCCc2c(nn(C(=O)c3c(Cl)cccc3Cl)c12)-c1ccc(cc1F)C(O)=O
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)F)c3CCCOc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3CCCOc23)c(F)c1
CC(C)(OC(=O)Nc1ccc2OC(CN(c2c1)S(=O)(=O)c1ccc(F)c(F)c1)C(=O)C(F)(F)F)C(F)(F)F
CN1CCN(C[C@H]2CN(c3cc(NC(=O)OC(C)(C)C(F)(F)F)ccc3O2)S(=O)(=O)c2ccc(F)c(Cl)c2)S1(=O)=O |r|
CNS(=O)(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CCOc1nn(CC)cc1S(=O)(=O)N1C[C@H](C)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
C[C@H]1[C@@H](CO)Oc2ccc(NC(=O)OCC(C)(C)C)cc2N1S(=O)(=O)c1cccc(c1)C#N |r|
CC1CN(C1)C(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)(OC(=O)Nc1ccc2OC(CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(C)(C)C(O)=O)C(F)(F)F
Cn1c(n[nH]c1=O)C(C)(C)C1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)cc1
CONC(=O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
COc1nn(C)c(C)c1S(=O)(=O)N1C[C@H](CC(C)(C)NC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(O)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC1CCc2ncc(NC(=O)OC(C)(C)C)cc2N1S(=O)(=O)c1ccc(F)cc1
CC(C)(C)OC(=O)NC1CN(c2cc(NC(=O)OCc3ccccc3)cnc2C1)S(=O)(=O)c1ccc(F)cc1
Cc1nn(cc1S(=O)(=O)N1CC(CN2CC[C@@H](O)C2)Cc2ncc(NC(=O)OCC(C)(C)C)cc12)C(F)F |r|
CCn1cc(c(OCCO)n1)S(=O)(=O)C1C[C@H](CC(C)(C)NC(C)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2OC(CN(c2c1)S(=O)(=O)c1ccc(F)c(F)c1)C(O)C(F)(F)F)C(F)(F)F
C[C@H](NC(=O)OCc1ccccc1)[C@@H]1Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N([C@@H]1C)S(=O)(=O)c1ccc(F)c(F)c1 |r|
CC(=O)NCC1COc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1ccc(F)cc1
Cc1ccc(cc1)S(=O)(=O)N1C[C@@H](CC2(CC2)C(N)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
Cc1ccc(cc1)S(=O)(=O)N1C[C@H](CC2(CC2)C(N)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CCc2n[nH]c(=O)n2C)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CCc2n[nH]c(=O)o2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CC(C)(OC(=O)Nc1ccc2O[C@@H](CCc3nnn[nH]3)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(F)(F)F |r|
Cc1c(NC(=O)OC(C)(C)C(F)(F)F)ccc2O[C@@H](CO)CN(c12)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1CCC(=O)c2ncc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3[C@H](C(C)C)N(C[C@H]4CC[C@@H](CC4)C(F)(F)F)Cc3c2)nc1 |r,wU:26.29,wD:17.17,23.22,(11.55,4.09,;10.21,3.32,;8.88,4.09,;8.11,2.76,;9.65,5.43,;7.54,4.86,;7.5,6.43,;6.16,7.2,;4.83,6.43,;3.49,7.2,;2.16,6.43,;.83,7.2,;.83,8.74,;-.51,6.43,;-.51,4.89,;-1.84,4.12,;-3.17,4.89,;-4.64,4.41,;-5.04,2.93,;-6.52,2.53,;-3.95,1.84,;-5.54,5.66,;-7.08,5.66,;-7.85,6.99,;-7.08,8.33,;-7.85,9.66,;-9.39,9.66,;-10.16,8.33,;-9.39,6.99,;-10.16,10.99,;-9.39,12.33,;-11.7,10.99,;-10.93,12.33,;-4.64,6.91,;-3.17,6.43,;-1.84,7.2,;4.83,4.89,;6.16,4.12,)|
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CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3[C@@H](C(C)C)N(C[C@H]4CCc5nc(C)oc5C4)Cc3c2)nc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3[C@H](C(C)C)N(C[C@H]4CCc5nc(C)oc5C4)Cc3c2)nc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3[C@@H](C(C)C)N(C[C@@H]4CCc5nc(C)oc5C4)Cc3c2)nc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3[C@H](C(C)C)N(C[C@@H]4CCc5nc(C)oc5C4)Cc3c2)nc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3[C@H](C(C)C)N(CC4CCC(OC4)C(F)(F)F)Cc3c2)nc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3[C@@H](C(C)C)N(CC4CCC(OC4)C(F)(F)F)Cc3c2)nc1 |r|
CC[C@@H]1N(C[C@H]2CC[C@@H](CC2)C(F)(F)F)Cc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cn1)S(=O)(=O)CC |r,wU:25.27,8.11,wD:2.1,5.4,(-3.05,-10.32,;-1.56,-9.92,;-1.17,-8.43,;-2.07,-7.18,;-3.61,-7.18,;-4.38,-5.85,;-3.61,-4.52,;-4.38,-3.18,;-5.92,-3.18,;-6.69,-4.52,;-5.92,-5.85,;-6.69,-1.85,;-8.23,-1.85,;-5.92,-.51,;-5.15,-1.85,;-1.17,-5.94,;.3,-6.41,;1.63,-5.64,;2.97,-6.41,;2.97,-7.95,;1.63,-8.72,;.3,-7.95,;4.3,-5.64,;4.3,-4.1,;5.63,-6.41,;6.97,-5.64,;6.97,-4.1,;8.3,-3.33,;8.3,-6.41,;9.63,-5.64,;10.97,-6.41,;11.02,-7.98,;9.63,-8.72,;8.3,-7.95,;12.35,-8.75,;11.58,-10.08,;13.12,-7.42,;13.68,-9.52,;15.02,-8.75,)|
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CC[C@H]1N(C[C@H]2CC[C@@H](CC2)C(F)(F)F)Cc2cc(ccc12)C(=O)N[C@@H](CCO)c1ccc(cn1)S(=O)(=O)CC |r,wU:8.11,2.1,25.27,wD:5.4,(-6.52,-3.9,;-5.04,-3.5,;-4.64,-2.02,;-5.54,-.77,;-7.08,-.77,;-7.85,.56,;-7.08,1.9,;-7.85,3.23,;-9.39,3.23,;-10.16,1.9,;-9.39,.56,;-10.16,4.56,;-9.39,5.9,;-11.7,4.56,;-10.93,5.9,;-4.64,.48,;-3.17,,;-1.84,.77,;-.51,,;-.51,-1.54,;-1.84,-2.31,;-3.17,-1.54,;.83,.77,;.83,2.31,;2.16,,;3.49,.77,;3.49,2.31,;4.83,3.08,;4.83,4.62,;4.83,,;6.16,.77,;7.5,,;7.54,-1.57,;6.16,-2.31,;4.83,-1.54,;8.88,-2.34,;8.11,-3.67,;9.65,-1,;10.21,-3.11,;11.54,-2.34,)|
CC[C@@H]1N(C[C@H]2CC[C@@H](CC2)C(F)(F)F)Cc2cc(ccc12)C(=O)NCc1ccc(cn1)S(=O)(=O)CC |r,wU:8.11,wD:5.4,2.1,(-6.52,-3.87,;-5.04,-3.48,;-4.64,-1.99,;-5.54,-.74,;-7.08,-.74,;-7.85,.59,;-7.08,1.93,;-7.85,3.26,;-9.39,3.26,;-10.16,1.93,;-9.39,.59,;-10.16,4.59,;-9.39,5.93,;-11.7,4.59,;-10.93,5.93,;-4.64,.5,;-3.17,.03,;-1.84,.8,;-.51,.03,;-.51,-1.51,;-1.84,-2.28,;-3.17,-1.51,;.83,.8,;.83,2.34,;2.16,.03,;3.49,.8,;4.83,.03,;6.16,.8,;7.5,.03,;7.54,-1.54,;6.16,-2.28,;4.83,-1.51,;8.88,-2.31,;8.11,-3.64,;9.65,-.98,;10.21,-3.08,;11.54,-2.31,)|
CC[C@H]1N(C[C@H]2CC[C@@H](CC2)C(F)(F)F)Cc2cc(ccc12)C(=O)NCc1ccc(cn1)S(=O)(=O)CC |r,wU:8.11,2.1,wD:5.4,(-6.52,-3.87,;-5.04,-3.48,;-4.64,-1.99,;-5.54,-.74,;-7.08,-.74,;-7.85,.59,;-7.08,1.93,;-7.85,3.26,;-9.39,3.26,;-10.16,1.93,;-9.39,.59,;-10.16,4.59,;-9.39,5.93,;-11.7,4.59,;-10.93,5.93,;-4.64,.5,;-3.17,.03,;-1.84,.8,;-.51,.03,;-.51,-1.51,;-1.84,-2.28,;-3.17,-1.51,;.83,.8,;.83,2.34,;2.16,.03,;3.49,.8,;4.83,.03,;6.16,.8,;7.5,.03,;7.54,-1.54,;6.16,-2.28,;4.83,-1.51,;8.88,-2.31,;8.11,-3.64,;9.65,-.98,;10.21,-3.08,;11.54,-2.31,)|
CC[C@@H]1N(C[C@H]2CC[C@@H](CC2)C(F)(F)F)Cc2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)NC |r,wU:8.11,wD:5.4,2.1,(-7.19,-4.23,;-5.7,-3.83,;-5.3,-2.35,;-6.21,-1.1,;-7.75,-1.1,;-8.52,.23,;-7.75,1.57,;-8.52,2.9,;-10.06,2.9,;-10.83,1.57,;-10.06,.23,;-10.83,4.23,;-10.06,5.57,;-12.37,4.23,;-11.6,5.57,;-5.3,.14,;-3.84,-.33,;-2.51,.44,;-1.17,-.33,;-1.17,-1.87,;-2.51,-2.64,;-3.84,-1.87,;.16,.44,;.16,1.98,;1.49,-.33,;2.83,.44,;4.16,-.33,;4.16,-1.87,;5.5,-2.64,;6.83,-1.87,;6.83,-.33,;5.5,.44,;8.16,-2.64,;7.39,-3.98,;8.93,-3.98,;9.5,-1.87,;10.83,-2.64,)|
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CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3C(C(C)C)N(Cc4ccc(cc4)C(F)(F)F)C(=O)c3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3C(C(C)C)N(Cc4ccc(cc4)C(F)(F)F)C(=O)c3c2)nc1
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2C(C(C)C)N(Cc3ccc(cc3)C(F)(F)F)C(=O)c2c1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3[C@H](C(C)C)N(C[C@H]4CC[C@@H](CC4)C(F)(F)F)C(=O)c3c2)cc1 |r,wU:26.29,wD:17.17,23.22,(12.25,-32.16,;10.82,-32.98,;9.4,-32.16,;8.58,-33.58,;10.22,-30.73,;7.98,-31.33,;6.44,-31.99,;5.11,-31.22,;5.11,-29.68,;3.77,-28.91,;2.44,-29.68,;1.11,-28.91,;1.11,-27.37,;-.23,-29.68,;-.23,-31.22,;-1.56,-31.99,;-2.89,-31.22,;-4.36,-31.69,;-4.76,-33.18,;-3.67,-34.27,;-6.24,-33.58,;-5.26,-30.45,;-6.8,-30.45,;-7.57,-29.11,;-6.8,-27.78,;-7.57,-26.45,;-9.11,-26.45,;-9.88,-27.78,;-9.11,-29.11,;-9.88,-25.11,;-9.11,-23.78,;-11.42,-25.11,;-10.65,-23.78,;-4.36,-29.2,;-5.13,-27.87,;-2.89,-29.68,;-1.56,-28.91,;6.44,-28.91,;7.78,-29.68,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3c(c2)C(=O)N(CC2CCC(CC2)C(F)(F)F)C3(C)C)cc1 |(6.15,-28.35,;4.66,-28.75,;4.26,-30.24,;5.75,-30.64,;3.86,-31.72,;2.77,-29.84,;1.69,-30.93,;.2,-30.53,;-.2,-29.04,;-1.69,-28.64,;-2.78,-29.73,;-4.26,-29.33,;-4.66,-27.85,;-5.35,-30.42,;-4.88,-31.89,;-5.91,-33.03,;-7.41,-32.71,;-7.89,-31.25,;-6.86,-30.1,;-9.43,-31.25,;-10.2,-29.91,;-9.91,-32.71,;-11.39,-33.11,;-12.48,-32.02,;-13.97,-32.42,;-15.06,-31.33,;-14.66,-29.84,;-13.17,-29.44,;-12.08,-30.53,;-15.75,-28.75,;-15.35,-27.27,;-17.24,-29.15,;-16.84,-27.66,;-8.66,-33.62,;-9.75,-34.7,;-8.26,-35.1,;.89,-27.95,;2.38,-28.35,)|
CCC1(C)N(CC2CCC(CC2)C(F)(F)F)C(=O)c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC |(-6.17,-3.55,;-4.63,-3.55,;-3.86,-2.22,;-3.09,-3.55,;-5.11,-1.31,;-6.59,-1.71,;-7.68,-.62,;-7.28,.86,;-8.37,1.95,;-9.86,1.55,;-10.26,.07,;-9.17,-1.02,;-10.95,2.64,;-10.55,4.13,;-12.44,2.25,;-12.04,3.73,;-4.63,.15,;-5.4,1.48,;-3.09,.15,;-2.06,1.3,;-.55,.98,;-.08,-.49,;-1.11,-1.63,;-2.61,-1.31,;.54,2.06,;.14,3.55,;2.02,1.67,;3.11,2.76,;4.6,2.36,;5,.87,;6.49,.47,;7.58,1.56,;7.18,3.05,;5.69,3.45,;9.06,1.16,;10.55,.76,;8.66,-.33,;9.46,2.65,;10.95,3.05,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3[C@H](C(C)C)N(C[C@H]4CO[C@H](OC4)C(F)(F)F)Cc3c2)nc1 |r,wU:23.22,26.29,wD:17.17,(10.83,-9.4,;9.5,-8.63,;8.16,-9.4,;7.39,-10.73,;8.93,-10.73,;6.83,-8.63,;6.83,-7.09,;5.5,-6.32,;4.16,-7.09,;2.83,-6.32,;1.49,-7.09,;.16,-6.32,;.16,-4.78,;-1.17,-7.09,;-1.17,-8.63,;-2.51,-9.4,;-3.84,-8.63,;-5.3,-9.1,;-5.7,-10.59,;-7.19,-10.99,;-4.61,-11.68,;-6.21,-7.86,;-7.75,-7.86,;-8.52,-6.52,;-10.06,-6.52,;-10.83,-5.19,;-10.06,-3.85,;-8.52,-3.85,;-7.75,-5.19,;-10.83,-2.52,;-10.06,-1.19,;-12.37,-2.52,;-11.6,-1.19,;-5.3,-6.61,;-3.84,-7.09,;-2.51,-6.32,;4.16,-8.63,;5.5,-9.4,)|
CCN1C2C=CC(NC(=O)Cc3ccc(cc3)S(=O)(=O)CC)=CC2N=C1C(C)(C)Oc1ccc(F)cc1F |c:4,22,26|
CCN1C2C=CC(NC(=O)Cc3ccc(cc3)S(=O)(=O)CC)=CC2N=C1C(C)(C)Oc1ccc(Cl)c(F)c1 |c:4,22,26|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(OC(C)(C)c3ccc(Cl)cc3Cl)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(OC(C)(C)c3ccc(Cl)cc3Cl)c(F)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C#CC(C)(C)Oc2ccc(Cl)c(F)c2)cc1
OC(=O)c1ccc(N2C=C(C3C=CC=CC23)C(=O)c2c(Cl)cccc2Cl)c(F)c1 |c:8,11,13|
OC(=O)c1ccc(N2C=C(C3C=CC=C(F)C23)C(=O)c2c(Cl)cccc2Cl)c(F)c1 |c:8,11,t:13|
OC(=O)c1ccc(cc1)N1N=C(C2C=CC=NC12)C(=O)c1c(Cl)cccc1C1CC1 |c:11,14,16|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(OC3(CCOCC3)c3ccc(Cl)cc3Cl)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(OC3(CCOCC3)c3ccc(Cl)cc3Cl)c(F)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(OC(C)(C)c3ncc(Cl)cc3Cl)c(F)c2)cc1
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2c(Cl)cccc2C(F)(F)F)c2ccccc12
OC(=O)c1ccc(cc1O)-n1cc(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
OC(=O)c1ccc(c(F)c1)-n1cc(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2c(F)cccc2C(F)(F)F)c2cccc(F)c12
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2cccc(F)c12
OC(=O)c1ccc(c(F)c1)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2cccc(F)c12
OC(=O)c1ccc(c(F)c1)-n1cc(C(=O)c2c(F)cccc2C(F)(F)F)c2cccc(F)c12
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(OC(F)F)cc4)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(Cl)cc4)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(C#N)c(F)c4)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(nc4)C#N)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4cnc(nc4)C(F)(F)F)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccccc4)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4cccc(c4)C(F)(F)F)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4nnc(o4)C(F)(F)F)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ncc(Cl)cc4F)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(Cl)cn4)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(cn4)C(F)(F)F)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(cc4F)C#N)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(F)cc4)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(cc4)C#N)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(cc4)C(=O)C(F)(F)F)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(C[C@H]4CC[C@@H](CC4)C(F)(F)F)Cc3s2)cc1 |wU:25.28,wD:22.21,16.16,(-7.84,8.09,;-6.3,8.09,;-5.53,6.76,;-6.86,5.99,;-4.19,7.53,;-4.76,5.42,;-3.22,5.42,;-2.45,4.09,;-3.22,2.76,;-2.45,1.42,;-3.22,.09,;-4.76,.09,;-2.45,-1.25,;-.91,-1.25,;;1.46,-.48,;2.93,,;3.41,1.46,;4.91,1.78,;2.37,2.61,;3.83,-1.25,;5.37,-1.25,;6.14,-2.58,;5.37,-3.91,;6.14,-5.25,;7.68,-5.25,;8.45,-3.91,;7.68,-2.58,;8.45,-6.58,;9.22,-7.91,;7.12,-7.35,;9.79,-5.81,;2.93,-2.49,;1.46,-2.02,;,-2.49,;-4.76,2.76,;-5.53,4.09,)|
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(cc4)-c4ccn(C)c(=O)c4)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(cc4)-c4ccc(=O)n(C)c4)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(CC4CCN(CC(F)(F)F)CC4)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(c(C)n4)C(F)(F)F)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(C[C@H]4CC[C@@H](N(C)C4)C(F)(F)F)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(CC4CC[C@@H](CC4)c4nnc(C)o4)Cc3s2)cc1 |wU:25.28,wD:16.16,(-7.84,8.09,;-6.3,8.09,;-5.53,6.76,;-6.86,5.99,;-4.19,7.53,;-4.76,5.42,;-3.22,5.42,;-2.45,4.09,;-3.22,2.76,;-2.45,1.42,;-3.22,.09,;-4.76,.09,;-2.45,-1.25,;-.91,-1.25,;;1.46,-.48,;2.93,,;3.41,1.46,;4.91,1.78,;2.37,2.61,;3.83,-1.25,;5.37,-1.25,;6.14,-2.58,;5.37,-3.91,;6.14,-5.25,;7.68,-5.25,;8.45,-3.91,;7.68,-2.58,;8.45,-6.58,;7.83,-7.99,;8.97,-9.02,;10.31,-8.25,;11.71,-8.87,;9.99,-6.74,;2.93,-2.49,;1.46,-2.02,;,-2.49,;-4.76,2.76,;-5.53,4.09,)|
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc3s2)[C@H](C)c2cc(Br)ccc2F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc3s2)[C@@H](C)c2cc(Br)ccc2F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(CC4CC[C@@H](OC4)C(F)(F)F)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(CC4CC[C@H](OC4)C(F)(F)F)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(CC4CC[C@@H](CC4)C(F)F)Cc3s2)cc1 |wU:25.28,wD:16.16,(-7.84,8.09,;-6.3,8.09,;-5.53,6.76,;-6.86,5.99,;-4.19,7.53,;-4.76,5.42,;-3.22,5.42,;-2.45,4.09,;-3.22,2.76,;-2.45,1.42,;-3.22,.09,;-4.76,.09,;-2.45,-1.25,;-.91,-1.25,;;1.46,-.48,;2.93,,;3.41,1.46,;4.91,1.78,;2.37,2.61,;3.83,-1.25,;5.37,-1.25,;6.14,-2.58,;5.37,-3.91,;6.14,-5.25,;7.68,-5.25,;8.45,-3.91,;7.68,-2.58,;8.45,-6.58,;7.68,-7.91,;9.22,-7.91,;2.93,-2.49,;1.46,-2.02,;,-2.49,;-4.76,2.76,;-5.53,4.09,)|
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(CC4CC[C@@H](N(C)C4)C(F)(F)F)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(CC4CC[C@H](N(C)C4)C(F)(F)F)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(nc4OC)C(F)(F)F)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc3s2)C(C)c2c(F)cc(Cl)cc2F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc3s2)[C@H](C)c2ccc(cc2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc3s2)[C@@H](C)c2ccc(cc2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc3s2)[C@H](C)c2ccc(cc2F)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc3s2)[C@@H](C)c2ccc(cc2F)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc3s2)[C@H](C)c2ccc(Cl)cc2F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc3s2)[C@@H](C)c2ccc(Cl)cc2F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(cc4)-c4nnnn4C)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(C[C@@H]4CCN(CO4)C(=O)OC(C)(C)C)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(cc4)-c4nnn(C)n4)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(C[C@H]4CN(CCO4)C(=O)OC(C)(C)C)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(CC4CC[C@@H](CC4)C(=O)OC)Cc3s2)cc1 |wU:25.28,wD:16.16,(-7.84,8.09,;-6.3,8.09,;-5.53,6.76,;-6.86,5.99,;-4.19,7.53,;-4.76,5.42,;-3.22,5.42,;-2.45,4.09,;-3.22,2.76,;-2.45,1.42,;-3.22,.09,;-4.76,.09,;-2.45,-1.25,;-.91,-1.25,;;1.46,-.48,;2.93,,;3.41,1.46,;4.91,1.78,;2.37,2.61,;3.83,-1.25,;5.37,-1.25,;6.14,-2.58,;5.37,-3.91,;6.14,-5.25,;7.68,-5.25,;8.45,-3.91,;7.68,-2.58,;8.45,-6.58,;9.99,-6.58,;7.68,-7.91,;6.14,-7.91,;2.93,-2.49,;1.46,-2.02,;,-2.49,;-4.76,2.76,;-5.53,4.09,)|
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(cc4C#N)C(F)(F)F)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ncc(cc4F)C#N)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc3s2)[C@H](C)c2ccc(Cl)cn2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc3s2)[C@@H](C)c2ccc(Cl)cn2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc3s2)[C@@H](C)c2cc(C)c(cn2)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc3s2)[C@@H](C)c2ccc(C#N)c(C)n2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc3s2)[C@@H](C)c2ccc(C#N)c(OC)n2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc3s2)[C@@H](C)c2ncc(Cl)cc2F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(OC(F)F)cn4)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(cc4)C4CC4)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(cc4)C(C)=O)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)F)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(nc4)C(F)(F)F)Cc3s2)cc1
CCc1ccc(CN2Cc3sc(NC(=O)Cc4ccc(cc4)S(=O)(=O)CC)nc3[C@@H]2C(C)C)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(C)cc4)Cc3s2)cc1
CC(C)[C@@H]1N(Cc2ccc(Cl)cc2)Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12
CC(C)[C@@H]1N(Cc2ccc(OC(F)F)cc2)Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12
CC(C)[C@@H]1N(Cc2ccc(C#N)c(F)c2)Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12
CC(C)[C@@H]1N(Cc2ccc(cn2)C(F)(F)F)Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12
CC(C)[C@@H]1N(Cc2ccc(nc2)C(F)(F)F)Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12
CC(C)[C@@H]1N(Cc2ccc(Cl)c(C)n2)Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12
CC(C)[C@@H]1N(Cc2ccc(C#N)c(C)n2)Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12
CC(C)[C@@H]1N(Cc2ccc(C#N)c(Cl)c2)Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12
CC(C)[C@@H]1N(Cc2nnn(C)n2)Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12
CC(C)[C@@H]1N(Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12)[C@H](C)c1ccc(cc1Cl)C#N
CC(C)[C@@H]1N(Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12)[C@@H](C)c1ccc(C#N)c(F)c1
CC(C)[C@@H]1N(Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12)[C@H](C)c1ccc(C#N)c(F)c1
CC(C)[C@@H]1N(Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12)[C@H](C)c1ccc(nc1C)C(F)(F)F
CC(C)[C@@H]1N(Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12)[C@@H](C)c1ccc(cc1)C#N
CC(C)[C@@H]1N(Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12)[C@H](C)c1ccc(cc1)C#N
CC(C)[C@@H]1N(Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12)[C@H](C)c1ccc(cc1C)C#N
CC(C)[C@@H]1N(Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12)[C@H](C)c1ccc(cc1F)C#N
CC(C)[C@@H]1N(Cc2ccc(cc2)C#N)Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@H](C(C)C)N(Cc4ccc(Cl)cc4)Cc3s2)nc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@@H](C(C)C)N(Cc4ccc(OC(C)C)cc4)Cc3s2)nc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@@H](C(C)C)N(Cc4ccc(OC(F)(F)F)cc4Cl)Cc3s2)nc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3s2)nc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@@H](C(C)C)N(Cc4ccc(c(Cl)c4)C(F)(F)F)Cc3s2)nc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@@H](C(C)C)N(C[C@H]4CC[C@](C)(CC4)OC)Cc3s2)nc1 |wU:22.21,25.29,wD:16.16,25.25,(10.82,-11.15,;11.59,-9.81,;10.82,-8.48,;12.16,-7.71,;9.49,-9.25,;10.05,-7.14,;10.82,-5.81,;10.05,-4.48,;8.51,-4.48,;7.74,-3.14,;8.51,-1.81,;10.05,-1.81,;7.74,-.48,;6.2,-.48,;5.3,.77,;3.83,.29,;2.37,.77,;1.89,2.23,;2.92,3.38,;.39,2.55,;1.46,-.48,;-.08,-.48,;-.85,-1.81,;-.08,-3.14,;-.85,-4.48,;-2.39,-4.48,;-1.91,-5.94,;-3.16,-3.14,;-2.39,-1.81,;-3.16,-5.81,;-4.7,-5.81,;2.37,-1.72,;3.83,-1.25,;5.3,-1.72,;7.74,-5.81,;8.51,-7.14,)|
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@@H](C(C)C)N(Cc4ccc(cc4)-c4ccn(C)c(=O)c4)Cc3s2)nc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@@H](C(C)C)N(CC4CC[C@@](CC4)(OC)C(F)(F)F)Cc3s2)nc1 |wU:25.30,wD:16.16,25.28,(10.82,-11.15,;11.59,-9.81,;10.82,-8.48,;12.16,-7.71,;9.49,-9.25,;10.05,-7.14,;10.82,-5.81,;10.05,-4.48,;8.51,-4.48,;7.74,-3.14,;8.51,-1.81,;10.05,-1.81,;7.74,-.48,;6.2,-.48,;5.3,.77,;3.83,.29,;2.37,.77,;1.89,2.23,;2.92,3.38,;.39,2.55,;1.46,-.48,;-.08,-.48,;-.98,-1.72,;-.35,-3.13,;-1.26,-4.37,;-2.79,-4.21,;-3.42,-2.81,;-2.51,-1.56,;-2.32,-5.68,;-.78,-5.84,;-4.12,-4.98,;-5.46,-4.21,;-4.12,-6.52,;-5.59,-5.46,;2.37,-1.72,;3.83,-1.25,;5.3,-1.72,;7.74,-5.81,;8.51,-7.14,)|
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@@H](C(C)C)N(Cc4ccc(cc4)-c4nnn(C)n4)Cc3s2)nc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@@H](C(C)C)N(Cc4ccc(C#N)c(Cl)c4)Cc3s2)nc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3[C@@H](C(C)C)N(Cc4ccc(cc4)C#N)Cc3s2)nc1
CC(C)[C@@H]1N(Cc2ccc(Cl)cc2)Cc2sc(NS(=O)(=O)c3ccc(CC(O)=O)cc3)nc12
CC(C)[C@@H]1N(Cc2ccc(C#N)c(F)c2)Cc2sc(NS(=O)(=O)c3ccc(CC(O)=O)cc3)nc12
CC(C)[C@@H]1N(Cc2ccc(Cl)cc2)Cc2sc(NS(=O)(=O)c3cccc(c3)C(F)(F)F)nc12
CC(C)[C@@H]1N(Cc2ccc(Cl)cc2)Cc2sc(NC(=O)Cc3ccc(cc3)C#N)nc12
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3C(Cc4cccc(Br)c4)N(Cc4ccc(F)cc4)Cc3s2)cc1
CC(C)[C@@H]1N(Cc2ccc(Cl)cc2)Cc2sc(NC(=O)Cc3ccc(cc3)S(=O)(=O)NC3CC3)nc12
CC[C@H](C)[C@@H]1N(Cc2ccc(Cl)cc2)Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12
CC[C@H](C)C1N(Cc2ccc(C#N)c(F)c2)Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12
CC[C@H](C)C1N(Cc2ccc(Cl)cn2)Cc2sc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)nc12
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3c(CN(Cc4ccc(cn4)C#N)[C@@]3(C)C(C)C)s2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2nc3[C@H](C(C)C)N(Cc4ccc(Cl)cc4)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2nc3[C@H](C(C)C)N(Cc4ccc(cc4)C#N)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2nc3[C@H](C(C)C)N(Cc4ccc(cc4)-c4nnn(C)n4)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2nc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2nc3[C@H](C(C)C)N(CC4CCN(CO4)OC(C)(C)C)Cc3s2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2nc3[C@H](C(C)C)N(Cc4ccc(OC(F)F)cc4)Cc3s2)cc1
CC(C)[C@@H]1N(Cc2ccc(Cl)cn2)Cc2sc(nc12)C(=O)NCc1ccc(cc1)S(C)(=O)=O
CC(C)[C@@H]1N(Cc2ccc(OC(F)F)cc2)Cc2sc(nc12)C(=O)NCc1ccc(cc1)S(C)(=O)=O
COC(=O)c1ccc(CN2Cc3sc(nc3[C@@H]2C(C)C)C(=O)NCc2ccc(cc2)S(C)(=O)=O)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2nc3[C@H](C(C)C)N(Cc4ccc(Cl)cc4)Cc3s2)nc1
CCS(=O)(=O)c1ccc(CNC(=O)c2nc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3s2)nc1
CCS(=O)(=O)c1ccc(CNC(=O)c2nc3[C@H](C(C)C)N(Cc4ccc5OC(F)(F)Oc5c4)Cc3s2)nc1
CC(C)[C@@H]1N(Cc2ccc(cc2)C#N)Cc2sc(NC(=O)Cc3ccc(cc3F)S(C)(=O)=O)nc12
Cc1c(NC(=O)c2cccc(c2)C#N)cnc2n(C)cc(C3CCN(CC3)C(=O)C3CC4CC[C@@H]3C4)c12 |r|
Cc1c(NC(=O)c2cccc(c2)C#N)cnc2n(C)cc(C3CCN(CC3)C(=O)C3CC4CC[C@H]3C4)c12 |r|
COc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc(C3[C@H]4CC[C@@H]3CN(C4)C(=O)C(C)C)c2c1C(F)(F)F |r|
C[C@@H](C(=O)N1CC[C@H]([C@@H](C)C1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12)C(F)(F)F |r|
CC(C)C(=O)N1C[C@@H]2CC[C@H](C1)C2c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12 |r|
COc1ccc(cc1C#N)C(=O)Nc1cnc2n(C)cc(C3[C@H]4CC[C@@H]3CN(C4)C(=O)C3CCCC3)c2c1C |r|
c1cc(ccc1F)S(=O)(=O)[C@@]23CCN([C@@H]2CCc4c3ccc(c4)C(C(F)(F)F)(C(F)(F)F)F)C(=O)C5CCC(CC5)C(=O)O
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CCCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:3.2,wD:6.9,(-10.99,-.87,;-10.22,-2.2,;-10.99,-3.54,;-8.68,-2.2,;-7.91,-.87,;-6.37,-.87,;-5.6,-2.2,;-6.37,-3.54,;-7.91,-3.54,;-4.06,-2.2,;-3.29,-3.54,;-3.29,-.87,;-4.06,.46,;-3.29,1.8,;-1.75,1.8,;-.98,.46,;-1.75,-.87,;-.98,-2.2,;.56,-2.2,;1.33,-.87,;2.87,-.87,;3.64,.46,;2.87,1.8,;1.33,1.8,;.56,.46,;5.18,.46,;5.18,2,;6.72,.46,;8.26,.46,;6.72,-1.08,;6.72,2,;5.18,-1.08,;3.85,-1.85,;6.51,-1.85,;5.18,-2.62,;-.21,1.8,;1.2,2.42,;.11,3.3,;-.98,3.13,;-2.52,3.13,;-3.29,4.46,;-2.52,5.8,;-3.29,7.13,;-.98,5.8,;-.21,4.46,)|
OC(=O)[C@H]1CC[C@@](F)(CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:16.17,3.2,6.6,wD:6.10,15.38,(-6.98,10.68,;-7.74,9.34,;-9.28,9.33,;-6.97,8.01,;-5.43,8.01,;-4.65,6.68,;-5.42,5.35,;-5.68,3.83,;-6.96,5.34,;-7.73,6.67,;-3.97,4.83,;-3.7,3.31,;-2.79,5.82,;-2.91,7.36,;-1.48,7.94,;-.49,6.76,;-1.3,5.45,;-.57,4.1,;.97,4.05,;1.78,5.36,;3.32,5.31,;4.13,6.62,;3.4,7.97,;1.86,8.02,;1.05,6.71,;5.67,6.57,;5.72,8.11,;7.21,6.52,;8.75,6.47,;7.16,4.98,;7.26,8.06,;5.62,5.03,;4.27,4.3,;6.93,4.22,;5.58,3.49,;.18,8.15,;1.65,8.62,;.66,9.61,;-.68,9.42,;-2.22,9.31,;-3.08,10.58,;-2.41,11.97,;-3.28,13.24,;-.88,12.08,;-.01,10.81,)|
OC(=O)[C@H]1CC[C@@](F)(CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:16.17,3.2,6.6,wD:6.10,15.38,(-6.98,10.68,;-7.74,9.34,;-9.28,9.33,;-6.97,8.01,;-5.43,8.01,;-4.65,6.68,;-5.42,5.35,;-5.68,3.83,;-6.96,5.34,;-7.73,6.67,;-3.97,4.83,;-3.7,3.31,;-2.79,5.82,;-2.91,7.36,;-1.48,7.94,;-.49,6.76,;-1.3,5.45,;-.57,4.1,;.97,4.05,;1.78,5.36,;3.32,5.31,;4.13,6.62,;3.4,7.97,;1.86,8.02,;1.05,6.71,;5.67,6.57,;5.72,8.11,;7.21,6.52,;8.75,6.47,;7.16,4.98,;7.26,8.06,;5.62,5.03,;4.27,4.3,;6.93,4.22,;5.58,3.49,;.18,8.15,;.95,9.48,;1.65,8.62,;-.68,9.42,;-2.22,9.31,;-3.08,10.58,;-2.41,11.97,;-3.28,13.24,;-.88,12.08,;-.01,10.81,)|
CC[C@@]1(CC[C@@H](CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(O)=O |r,wU:14.15,2.47,wD:5.8,2.1,13.36,(-8.04,1.86,;-8.51,.4,;-7.47,-.74,;-6.3,.25,;-4.85,-.27,;-4.58,-1.79,;-5.75,-2.78,;-7.2,-2.26,;-3.13,-2.31,;-2.85,-3.82,;-1.95,-1.31,;-2.06,.22,;-.64,.8,;.36,-.37,;-.45,-1.68,;.27,-3.04,;1.81,-3.09,;2.62,-1.78,;4.16,-1.83,;4.97,-.52,;4.25,.84,;2.71,.89,;1.9,-.42,;6.51,-.56,;6.56,.97,;8.05,-.61,;9.59,-.66,;8.01,-2.15,;8.1,.93,;6.47,-2.1,;5.11,-2.83,;7.77,-2.91,;6.42,-3.64,;1.03,1.01,;1.65,2.42,;2.49,1.49,;.16,2.29,;-1.37,2.18,;-2.24,3.45,;-1.57,4.84,;-2.44,6.11,;-.03,4.95,;.83,3.67,;-9,-.96,;-9.57,-2.39,;-9.95,.25,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCNCC1 |r|
OC(=O)c1ccc(cc1)S(=O)(=O)N1CCC2(C1Cc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(=O)C12CCC(CC1)(CC2)C(=O)N1CC[C@]2([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@]2([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:6.9,14.37,wD:15.16,3.2,(-10.01,1.35,;-9.74,-.16,;-10.91,-1.16,;-8.29,-.68,;-8.01,-2.2,;-6.57,-2.72,;-5.39,-1.73,;-5.66,-.21,;-7.11,.31,;-3.94,-2.25,;-3.67,-3.76,;-2.76,-1.25,;-2.88,.28,;-1.45,.87,;-.46,-.31,;-1.27,-1.62,;-.54,-2.98,;1,-3.02,;1.81,-1.72,;3.35,-1.76,;4.16,-.46,;3.43,.9,;1.89,.95,;1.08,-.36,;5.7,-.5,;5.75,1.04,;7.24,-.55,;8.78,-.6,;7.19,-2.09,;7.29,.99,;5.65,-2.04,;4.29,-2.77,;6.96,-2.85,;5.6,-3.58,;.21,1.08,;1.68,1.55,;.69,2.54,;-.65,2.35,;-2.19,2.24,;-3.05,3.51,;-2.38,4.9,;-3.25,6.17,;-.85,5.01,;.02,3.74,)|
Fc1ccc(cc1)S(=O)(=O)[C@]12CCN([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCS(=O)(=O)CC1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCS(=O)(=O)CC1 |r|
OC(=O)C12CCC(CC1)(CC2)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCC(CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1 |r,wU:6.9,wD:3.2,(-10.01,1.35,;-9.74,-.16,;-10.91,-1.16,;-8.29,-.68,;-8.01,-2.2,;-6.57,-2.72,;-5.39,-1.73,;-5.66,-.21,;-7.11,.31,;-3.94,-2.25,;-3.67,-3.76,;-2.76,-1.25,;-2.88,.28,;-1.45,.87,;-.46,-.31,;-1.27,-1.62,;-.54,-2.98,;1,-3.02,;1.81,-1.72,;3.35,-1.76,;4.16,-.46,;3.43,.9,;1.89,.95,;1.08,-.36,;5.7,-.5,;5.75,1.04,;7.24,-.55,;8.78,-.6,;7.19,-2.09,;7.29,.99,;5.65,-2.04,;4.29,-2.77,;6.96,-2.85,;5.6,-3.58,;.21,1.08,;1.72,1.4,;.69,2.54,;-.65,2.35,;-2.19,2.24,;-3.05,3.51,;-2.38,4.9,;-3.25,6.17,;-.85,5.01,;.02,3.74,)|
OC(=O)C12CCC(CC1)(CC2)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1
FC(F)(F)C(F)(c1ccc2c(CCC3N(CCC23S(=O)(=O)c2ccc(Cl)cc2)C(=O)C2CCS(=O)(=O)CC2)c1)C(F)(F)F
CC(=O)N1CCC(CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1
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OC1(CCS(=O)(=O)CC1)C(=O)N1CCC2(C1COc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1
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OC(=O)c1ccc(cc1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(cc1)C(F)(F)F
CCc1ccc(cc1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccc(cc1)C(O)=O
OC(=O)C1CC2(C1)CC(C2)C(=O)N1CCC2(C1COc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(=O)C1CC2(C1)CC(C2)C(=O)N1CCC2(C1COc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
Cc1ccc(cc1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CC2(CC(C2)C(O)=O)C1
Cc1ccc(cc1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CC2(CC(C2)C(O)=O)C1
OC(=O)C1CC2(C1)CC(C2)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(cc1)C(F)(F)F |(8.51,4.91,;7.74,3.58,;8.51,2.24,;6.2,3.58,;5.11,4.66,;4.02,3.58,;5.11,2.49,;2.93,4.66,;1.84,3.58,;2.93,2.49,;.3,3.58,;-.47,4.91,;-.47,2.24,;.16,.83,;-.99,-.2,;-2.32,.57,;-2,2.08,;-3.14,3.11,;-4.61,2.63,;-4.93,1.13,;-6.39,.65,;-6.71,-.85,;-5.57,-1.88,;-4.1,-1.41,;-3.78,.1,;-8.18,-1.33,;-7.7,-2.79,;-9.64,-1.81,;-11.11,-2.28,;-10.12,-.34,;-9.17,-3.27,;-8.65,.14,;-7.62,1.28,;-10.16,.46,;-9.13,1.6,;-2.48,-.96,;-3.38,-2.2,;-1.85,-2.36,;-1.23,-1.86,;.17,-1.24,;1.42,-2.14,;1.26,-3.67,;-.15,-4.3,;-1.39,-3.39,;2.5,-4.58,;3.75,-5.48,;1.6,-5.82,;3.41,-3.33,)|
OC(=O)C1CC2(C1)CC(C2)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(cc1)C(F)(F)F |(8.51,4.91,;7.74,3.58,;8.51,2.24,;6.2,3.58,;5.11,4.66,;4.02,3.58,;5.11,2.49,;2.93,4.66,;1.84,3.58,;2.93,2.49,;.3,3.58,;-.47,4.91,;-.47,2.24,;.16,.83,;-.99,-.2,;-2.32,.57,;-2,2.08,;-3.14,3.11,;-4.61,2.63,;-4.93,1.13,;-6.39,.65,;-6.71,-.85,;-5.57,-1.88,;-4.1,-1.41,;-3.78,.1,;-8.18,-1.33,;-7.7,-2.79,;-9.64,-1.81,;-10.12,-.34,;-9.17,-3.27,;-11.11,-2.28,;-8.65,.14,;-7.62,1.28,;-10.16,.46,;-9.13,1.6,;-2.48,-.96,;-3.38,-2.2,;-1.85,-2.36,;-1.23,-1.86,;.17,-1.24,;1.42,-2.14,;1.26,-3.67,;-.15,-4.3,;-1.39,-3.39,;2.5,-4.58,;3.75,-5.48,;1.6,-5.82,;3.41,-3.33,)|
OC(=O)C1CC2(C1)CC(C2)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccn1
OC(=O)C1CC2(C1)CC(C2)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccn1
CCc1ccc(cc1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CC2(CC(C2)C(O)=O)C1 |(4.12,-4.44,;2.72,-5.07,;1.47,-4.17,;1.63,-2.63,;.39,-1.73,;-1.02,-2.36,;-1.18,-3.89,;.06,-4.79,;-2.27,-1.45,;-3.17,-2.7,;-1.64,-2.86,;-2.11,.08,;-.77,-.69,;.37,.34,;-.25,1.75,;-1.78,1.59,;-2.93,2.62,;-4.39,2.14,;-4.71,.64,;-6.18,.16,;-6.5,-1.35,;-5.35,-2.38,;-3.89,-1.9,;-3.57,-.39,;-7.96,-1.82,;-7.49,-3.29,;-9.43,-2.3,;-9.9,-.83,;-8.95,-3.76,;-10.89,-2.77,;-8.44,-.36,;-7.41,.79,;-9.95,-.04,;-8.92,1.11,;.52,3.08,;-.25,4.42,;2.06,3.08,;3.15,4.17,;4.23,3.08,;5.32,4.17,;6.41,3.08,;5.32,1.99,;7.95,3.08,;8.72,4.42,;8.72,1.75,;3.15,1.99,)|
CC1(CCS(=O)(=O)CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccn1
OC(=O)C1CC2(C1)CC(C2)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1
OC(=O)C1CC2(C1)CC(C2)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1
OC1(CCS(=O)(=O)CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccn1
Cc1ccc(cc1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCS(=O)(=O)C1 |w:33.38|
FC(F)(F)c1ccc(cc1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCS(=O)(=O)C1 |w:36.41|
CCc1ccc(cc1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCS(=O)(=O)C1 |w:34.39|
FC(F)(F)c1ccc(cc1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCS(=O)(=O)CC1
FC(F)(F)C(F)(c1ccc2c(CCC3N(CCC23S(=O)(=O)c2ccccn2)C(=O)C2CCS(=O)(=O)C2)c1)C(F)(F)F |w:27.31|
OC1(CCS(=O)(=O)CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1
CC1(CCS(=O)(=O)CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1
FC(F)(F)C(F)(c1ccc2c(CCC3N(CCC23S(=O)(=O)c2ccc(Cl)cc2)C(=O)C2CCS(=O)(=O)C2)c1)C(F)(F)F |w:28.32|
FC(F)(F)C(F)(c1ccc2c(CCC3N(CCC23S(=O)(=O)c2ccc(Cl)cc2)C(=O)C2CCS(=O)(=O)C2)c1)C(F)(F)F
CC(C)N1[C@@H](CCC1=O)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Cc1cccc(c1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)[C@H]1CC[C@@H](CC1)C(O)=O |r,wU:38.45,wD:35.38,(-4.63,3.09,;-3.1,3.2,;-2.43,4.59,;-.89,4.7,;-.02,3.43,;-.69,2.04,;-2.23,1.93,;.17,.77,;1.44,1.63,;.06,2.3,;-.5,-.62,;-1.49,.56,;-2.92,-.02,;-2.81,-1.56,;-1.31,-1.93,;-.58,-3.28,;.96,-3.33,;1.77,-2.02,;3.31,-2.07,;4.12,-.76,;3.39,.59,;1.85,.64,;1.04,-.67,;5.66,-.81,;5.61,-2.35,;7.2,-.86,;8.74,-.91,;7.15,-2.4,;7.25,.68,;5.71,.73,;7.06,1.46,;4.4,1.54,;5.75,2.27,;-3.98,-2.55,;-3.71,-4.07,;-5.43,-2.03,;-5.7,-.52,;-7.15,0,;-8.33,-.99,;-8.06,-2.51,;-6.61,-3.03,;-9.78,-.47,;-10.95,-1.46,;-10.05,1.05,)|
Cc1cccc(c1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C12CCC(CC1)(CC2)C(O)=O
Cc1cccc(c1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)[C@@H]1CCC(=O)N1Cc1ccc(cc1)C#N |r|
CN1[C@@H](CCC1=O)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(C)c1 |r|
Cc1cccc(c1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCS(=O)(=O)CC1
Cc1cccc(c1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1(C)CCS(=O)(=O)CC1
Cc1cccc(c1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1(O)CCC(CC1)C(O)=O |(-4.7,2.81,;-3.17,2.93,;-2.5,4.31,;-.96,4.43,;-.1,3.15,;-.77,1.77,;-2.3,1.65,;.1,.49,;1.37,1.36,;-.01,2.03,;-.57,-.89,;-1.56,.28,;-2.99,-.3,;-2.88,-1.84,;-1.38,-2.2,;-.65,-3.56,;.89,-3.61,;1.7,-2.3,;3.24,-2.35,;4.05,-1.04,;3.32,.32,;1.78,.37,;.97,-.94,;5.59,-1.09,;5.54,-2.63,;7.13,-1.14,;8.67,-1.18,;7.08,-2.67,;7.17,.4,;5.64,.45,;6.99,1.18,;4.33,1.26,;5.68,1.99,;-4.05,-2.83,;-3.78,-4.35,;-5.5,-2.31,;-5.76,-3.83,;-7.04,-2.32,;-7.82,-.98,;-7.05,.35,;-5.51,.36,;-4.74,-.97,;-7.83,1.68,;-9.37,1.68,;-7.06,3.02,)|
Cc1cccc(c1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)[C@@]1(C)CC[C@@H](CC1)C(O)=O |r,wU:39.46,35.39,wD:35.38,(-4.65,2.87,;-3.11,2.98,;-2.44,4.37,;-.91,4.48,;-.04,3.2,;-.71,1.82,;-2.25,1.7,;.15,.54,;1.43,1.41,;.04,2.08,;-.52,-.84,;-1.51,.33,;-2.94,-.25,;-2.82,-1.78,;-1.33,-2.15,;-.6,-3.51,;.94,-3.56,;1.75,-2.25,;3.29,-2.3,;4.1,-.99,;3.37,.37,;1.83,.42,;1.02,-.89,;5.64,-1.03,;5.59,-2.57,;7.18,-1.08,;8.72,-1.13,;7.13,-2.62,;7.23,.46,;5.69,.5,;7.04,1.23,;4.38,1.32,;5.74,2.04,;-4,-2.78,;-3.73,-4.29,;-5.45,-2.26,;-5.71,-3.77,;-4.68,-.92,;-5.46,.41,;-7,.4,;-7.76,-.93,;-6.99,-2.26,;-7.77,1.74,;-9.31,1.73,;-7.01,3.07,)|
Cc1cccc(c1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)CC(C)(C)O
Fc1cccc(c1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)[C@@H]1CCC(=O)N1Cc1ccc(cc1)C#N |r|
CN1[C@@H](CCC1=O)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1 |r|
FC(F)(F)C(F)(c1ccc2c(CCC3N(CCC23S(=O)(=O)c2cccc(Cl)c2)C(=O)C2CCS(=O)(=O)CC2)c1)C(F)(F)F
OC(=O)[C@H]1CC[C@@](O)(CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(Cl)c1 |r,wU:6.6,3.2,wD:6.10,(-9.31,1.73,;-7.77,1.74,;-7.01,3.07,;-7,.4,;-5.46,.41,;-4.68,-.92,;-5.45,-2.26,;-5.71,-3.77,;-6.99,-2.26,;-7.76,-.93,;-4,-2.78,;-3.73,-4.29,;-2.82,-1.78,;-2.94,-.25,;-1.51,.33,;-.52,-.84,;-1.33,-2.15,;-.6,-3.51,;.94,-3.56,;1.75,-2.25,;3.29,-2.3,;4.1,-.99,;3.37,.37,;1.83,.42,;1.02,-.89,;5.64,-1.03,;5.59,-2.57,;7.18,-1.08,;8.72,-1.13,;7.13,-2.62,;7.23,.46,;5.69,.5,;7.04,1.23,;4.38,1.32,;5.74,2.04,;.15,.54,;1.43,1.41,;.04,2.08,;-.71,1.82,;-.04,3.2,;-.91,4.48,;-2.44,4.37,;-3.11,2.98,;-4.65,2.87,;-2.25,1.7,)|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(Cl)c1 |r,wU:3.2,wD:6.9,(-10.95,-1.46,;-9.78,-.47,;-10.05,1.05,;-8.33,-.99,;-7.15,0,;-5.7,-.52,;-5.43,-2.03,;-6.61,-3.03,;-8.06,-2.51,;-3.98,-2.55,;-3.71,-4.07,;-2.81,-1.56,;-2.92,-.02,;-1.49,.56,;-.5,-.62,;-1.31,-1.93,;-.58,-3.28,;.96,-3.33,;1.77,-2.02,;3.31,-2.07,;4.12,-.76,;3.39,.59,;1.85,.64,;1.04,-.67,;5.66,-.81,;5.61,-2.35,;7.2,-.86,;8.74,-.91,;7.15,-2.4,;7.25,.68,;5.71,.73,;7.06,1.46,;4.4,1.54,;5.75,2.27,;.17,.77,;1.44,1.63,;.06,2.3,;-.69,2.04,;-.02,3.43,;-.89,4.7,;-2.43,4.59,;-3.1,3.2,;-4.63,3.09,;-2.23,1.93,)|
OC(=O)C12CCC(CC1)(CC2)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(Cl)c1
CN1[C@@H](CCC1=O)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(Cl)c1 |r|
FC(F)(F)C(F)(c1ccc2c(CCC3N(CCC23S(=O)(=O)c2cccc(Cl)c2)C(=O)[C@@H]2CCC(=O)N2Cc2ccc(cc2)C#N)c1)C(F)(F)F |r|
OC(=O)[C@H]1CC[C@@](F)(CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(Cl)c1 |r,wU:6.10,wD:6.6,3.2,(-7.02,3.08,;-7.78,1.74,;-9.32,1.73,;-7.01,.41,;-7.77,-.93,;-7,-2.26,;-5.46,-2.25,;-5.72,-3.77,;-4.69,-.92,;-5.47,.41,;-4.01,-2.77,;-3.74,-4.29,;-2.83,-1.78,;-2.95,-.24,;-1.52,.34,;-.53,-.84,;-1.34,-2.15,;-.61,-3.5,;.93,-3.55,;1.74,-2.24,;3.28,-2.29,;4.09,-.98,;3.36,.37,;1.82,.42,;1.01,-.89,;5.63,-1.03,;5.58,-2.57,;7.17,-1.08,;8.71,-1.13,;7.12,-2.62,;7.22,.46,;5.68,.51,;7.04,1.24,;4.37,1.32,;5.73,2.05,;.14,.55,;1.42,1.41,;.03,2.08,;-.72,1.82,;-.05,3.21,;-.92,4.48,;-2.45,4.37,;-3.12,2.98,;-4.66,2.87,;-2.26,1.71,)|
OC(=O)[C@@]1(F)CC[C@@H](CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(Cl)c1 |r,wU:3.2,wD:7.10,3.3,(-10.48,-.27,;-8.98,.05,;-8.51,1.52,;-7.94,-1.09,;-9.47,-1.31,;-6.77,-.09,;-5.32,-.62,;-5.04,-2.13,;-6.22,-3.13,;-7.67,-2.6,;-3.6,-2.65,;-3.32,-4.17,;-2.42,-1.66,;-2.53,-.12,;-1.11,.46,;-.11,-.72,;-.92,-2.03,;-.2,-3.38,;1.34,-3.43,;2.15,-2.12,;3.69,-2.17,;4.51,-.86,;3.78,.5,;2.24,.54,;1.43,-.76,;6.04,-.91,;6,-2.45,;7.58,-.96,;9.12,-1.01,;7.54,-2.5,;7.63,.58,;6.09,.63,;7.45,1.36,;4.78,1.44,;6.14,2.17,;.56,.67,;1.83,1.54,;.44,2.21,;-.31,1.94,;.36,3.33,;-.5,4.6,;-2.04,4.49,;-2.71,3.1,;-4.25,2.99,;-1.84,1.83,)|
Cc1cccc(c1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)[C@@]1(F)CC[C@@H](CC1)C(O)=O |r,wU:35.38,wD:35.39,39.46,(-4.66,2.87,;-3.12,2.98,;-2.45,4.37,;-.92,4.48,;-.05,3.21,;-.72,1.82,;-2.26,1.71,;.14,.55,;1.42,1.41,;.03,2.08,;-.53,-.84,;-1.52,.34,;-2.95,-.24,;-2.83,-1.78,;-1.34,-2.15,;-.61,-3.5,;.93,-3.55,;1.74,-2.24,;3.28,-2.29,;4.09,-.98,;3.36,.37,;1.82,.42,;1.01,-.89,;5.63,-1.03,;5.58,-2.57,;7.17,-1.08,;8.71,-1.13,;7.12,-2.62,;7.22,.46,;5.68,.51,;7.04,1.24,;4.37,1.32,;5.73,2.05,;-4.01,-2.77,;-3.74,-4.29,;-5.46,-2.25,;-5.72,-3.77,;-7,-2.26,;-7.77,-.93,;-7.01,.41,;-5.47,.41,;-4.69,-.92,;-7.78,1.74,;-7.02,3.08,;-9.32,1.73,)|
C[C@@]1(CC[C@@H](CC1)C(O)=O)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(Cl)c1 |r,wU:1.10,wD:4.7,1.0,(-5.72,-3.77,;-5.46,-2.25,;-7,-2.26,;-7.77,-.93,;-7.01,.41,;-5.47,.41,;-4.69,-.92,;-7.78,1.74,;-7.02,3.08,;-9.32,1.73,;-4.01,-2.77,;-3.74,-4.29,;-2.83,-1.78,;-2.95,-.24,;-1.52,.34,;-.53,-.84,;-1.34,-2.15,;-.61,-3.5,;.93,-3.55,;1.74,-2.24,;3.28,-2.29,;4.09,-.98,;3.36,.37,;1.82,.42,;1.01,-.89,;5.63,-1.03,;5.58,-2.57,;7.17,-1.08,;8.71,-1.13,;7.12,-2.62,;7.22,.46,;5.68,.51,;7.04,1.24,;4.37,1.32,;5.73,2.05,;.14,.55,;1.42,1.41,;.03,2.08,;-.72,1.82,;-.05,3.21,;-.92,4.48,;-2.45,4.37,;-3.12,2.98,;-4.66,2.87,;-2.26,1.71,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)[C@@H]1CCC(=O)N1Cc1ccc(cc1)C#N |r|
CN1[C@@H](CCC1=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(O)CC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CCN1[C@@H](CCC1=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(CN2[C@@H](CCC2=O)C(=O)N2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)Cc1ccnnc1 |r|
FC(F)(F)C(F)(c1ccc2c(CCC3N(CCC23S(=O)(=O)c2cccc(Cl)c2)C(=O)Cc2ccnnc2)c1)C(F)(F)F
CC(C)(O)[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:16.17,7.10,wD:15.38,4.3,(-10.74,.24,;-9.29,-.28,;-9.82,-1.73,;-8.77,1.17,;-7.85,-.8,;-7.57,-2.32,;-6.12,-2.84,;-4.95,-1.84,;-5.22,-.33,;-6.67,.19,;-3.5,-2.36,;-3.23,-3.88,;-2.32,-1.37,;-2.44,.17,;-1.01,.75,;-.02,-.43,;-.83,-1.74,;-.1,-3.09,;1.44,-3.14,;2.25,-1.83,;3.79,-1.88,;4.6,-.57,;3.87,.78,;2.34,.83,;1.52,-.48,;6.14,-.62,;6.09,-2.16,;7.68,-.67,;9.22,-.72,;7.63,-2.21,;7.73,.87,;6.19,.92,;7.55,1.65,;4.88,1.73,;6.24,2.46,;.66,.96,;1.93,1.82,;.54,2.49,;-.21,2.23,;-1.75,2.12,;-2.61,3.39,;-1.94,4.78,;-2.81,6.05,;-.41,4.89,;.46,3.62,)|
CC(C)(O)C12CCC(CC1)(CC2)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)c1cc([nH]n1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN1[C@@H](C[C@@H](F)C1=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN1[C@@H](C[C@H](F)C1=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN1[C@@H](CC(F)(F)C1=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN1[C@@H](C[C@H](F)C1=O)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1 |r|
CN1[C@@H](CC(F)(F)C1=O)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1 |r|
CN1[C@@H](C[C@H](F)C1=O)C(=O)N1CCC2(C1COc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1 |r|
CN1[C@@H](C[C@H](F)C1=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1 |r|
CN1[C@@H](C[C@H](F)C1=O)C(=O)N1CCC2(C1COc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN1[C@@H](C[C@H](F)C1=O)C(=O)N1CCC2(C1COc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1 |r|
CN1C(CCS1(=O)=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:8.8|
CN1CC(CC1=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:7.7|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCC(=O)N1CCC#N |r,w:33.38|
CN1C(=O)CCC1(C)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:8.8|
CC(C)N1[C@@H](C[C@H](F)C1=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
COCCN1[C@@H](C[C@H](F)C1=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN1[C@@H](C[C@H](O)C1=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C12CCC(CC1)(CC2)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1
OC(=O)[C@H]1CC[C@@](F)(CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1 |r,wU:3.2,6.6,wD:6.10,(-9.32,1.73,;-7.78,1.74,;-7.02,3.08,;-7.01,.41,;-5.47,.41,;-4.69,-.92,;-5.46,-2.25,;-5.72,-3.77,;-7,-2.26,;-7.77,-.93,;-4.01,-2.77,;-3.74,-4.29,;-2.83,-1.78,;-2.95,-.24,;-1.52,.34,;-.53,-.84,;-1.34,-2.15,;-.61,-3.5,;.93,-3.55,;1.74,-2.24,;3.28,-2.29,;4.09,-.98,;3.36,.37,;1.82,.42,;1.01,-.89,;5.63,-1.03,;5.58,-2.57,;7.17,-1.08,;8.71,-1.13,;7.12,-2.62,;7.22,.46,;5.68,.51,;7.04,1.24,;4.37,1.32,;5.73,2.05,;.14,.55,;1.42,1.41,;.03,2.08,;-.72,1.82,;-.05,3.21,;-.92,4.48,;-2.45,4.37,;-3.12,2.98,;-4.66,2.87,;-2.26,1.71,)|
C[C@@]1(CC[C@@H](CC1)C(O)=O)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1 |r,wU:4.7,1.0,wD:1.10,(-5.72,-3.77,;-5.46,-2.25,;-4.69,-.92,;-5.47,.41,;-7.01,.41,;-7.77,-.93,;-7,-2.26,;-7.78,1.74,;-9.32,1.73,;-7.02,3.08,;-4.01,-2.77,;-3.74,-4.29,;-2.83,-1.78,;-2.95,-.24,;-1.52,.34,;-.53,-.84,;-1.34,-2.15,;-.61,-3.5,;.93,-3.55,;1.74,-2.24,;3.28,-2.29,;4.09,-.98,;3.36,.37,;1.82,.42,;1.01,-.89,;5.63,-1.03,;5.58,-2.57,;7.17,-1.08,;8.71,-1.13,;7.12,-2.62,;7.22,.46,;5.68,.51,;7.04,1.24,;4.37,1.32,;5.73,2.05,;.14,.55,;1.42,1.41,;.03,2.08,;-.72,1.82,;-.05,3.21,;-.92,4.48,;-2.45,4.37,;-3.12,2.98,;-4.66,2.87,;-2.26,1.71,)|
Fc1cccc(c1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCS(=O)(=O)CC1
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OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1 |r,wU:3.2,wD:6.9,(-10.95,-1.46,;-9.78,-.47,;-10.05,1.05,;-8.33,-.99,;-7.15,0,;-5.7,-.52,;-5.43,-2.03,;-6.61,-3.03,;-8.06,-2.51,;-3.98,-2.55,;-3.71,-4.07,;-2.81,-1.56,;-2.92,-.02,;-1.49,.56,;-.5,-.62,;-1.31,-1.93,;-.58,-3.28,;.96,-3.33,;1.77,-2.02,;3.31,-2.07,;4.12,-.76,;3.39,.59,;1.85,.64,;1.04,-.67,;5.66,-.81,;5.61,-2.35,;7.2,-.86,;8.74,-.91,;7.15,-2.4,;7.25,.68,;5.71,.73,;7.06,1.46,;4.4,1.54,;5.75,2.27,;.17,.77,;1.44,1.63,;.06,2.3,;-.69,2.04,;-.02,3.43,;-.89,4.7,;-2.43,4.59,;-3.1,3.2,;-4.63,3.09,;-2.23,1.93,)|
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CC(C)(C)c1ccc2c(CCC3N(CCC23S(=O)(=O)c2cccc(F)c2)C(=O)C23CCC(CC2)(CC3)C(O)=O)c1
CC(C)(C)c1ccc2c(CCC3N(CCC23S(=O)(=O)c2cccc(F)c2)C(=O)C2CCS(=O)(=O)CC2)c1
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OC(=O)[C@@H]1CCC(=O)N1CC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC1(C)OCC(C)(CO1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CCCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1 |r,wU:6.9,wD:3.2,(-11,-4.27,;-10.23,-2.94,;-11,-1.6,;-8.69,-2.94,;-7.92,-4.27,;-6.38,-4.27,;-5.61,-2.94,;-6.38,-1.6,;-7.92,-1.6,;-4.07,-2.94,;-3.3,-4.27,;-3.3,-1.6,;-4.07,-.27,;-3.3,1.07,;-1.76,1.07,;-.99,-.27,;-1.76,-1.6,;-.99,-2.94,;.55,-2.94,;1.32,-1.6,;2.86,-1.6,;3.63,-.27,;2.86,1.07,;1.32,1.07,;.55,-.27,;5.17,-.27,;5.17,1.27,;6.71,-.27,;8.25,-.27,;6.71,-1.81,;6.71,1.27,;5.17,-1.81,;3.84,-2.58,;6.5,-2.58,;5.17,-3.35,;-.22,1.07,;1.11,1.84,;-.22,2.61,;-.99,2.4,;-2.53,2.4,;-3.3,3.73,;-2.53,5.07,;-.99,5.07,;-.22,6.4,;-.22,3.73,)|
OC(=O)C12CCC(CC1)(CC2)C(=O)N1CCCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1
Fc1cccc(c1)S(=O)(=O)C12CCCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCS(=O)(=O)CC1
C[C@@]1(CC[C@@H](CC1)C(O)=O)C(=O)N1CCCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1 |r,wU:1.10,wD:4.7,1.0,(-5.26,-4.7,;-5.53,-3.19,;-6.97,-3.71,;-8.15,-2.72,;-7.89,-1.21,;-6.44,-.68,;-5.26,-1.67,;-9.07,-.22,;-10.51,-.74,;-8.8,1.3,;-3.99,-3.19,;-3.22,-4.52,;-3.22,-1.85,;-3.99,-.52,;-3.22,.81,;-1.68,.81,;-.91,-.52,;-1.68,-1.85,;-.91,-3.19,;.63,-3.19,;1.4,-1.85,;2.94,-1.85,;3.71,-.52,;2.94,.81,;1.4,.81,;.63,-.52,;5.25,-.52,;5.25,1.02,;6.79,-.52,;8.33,-.52,;6.79,-2.06,;6.79,1.02,;5.25,-2.06,;3.92,-2.83,;6.59,-2.83,;5.25,-3.6,;-.14,.81,;1.2,1.58,;-.14,2.35,;-.91,2.15,;-2.45,2.15,;-3.22,3.48,;-2.45,4.82,;-.91,4.82,;-.14,6.15,;-.14,3.48,)|
Fc1ccc(cc1)S(=O)(=O)C12CCCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCS(=O)(=O)CC1
OC(=O)C12CCC(CC1)(CC2)C(=O)N1CCCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CCCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1 |r,wU:6.9,wD:3.2,(-10.99,-3.96,;-10.22,-2.62,;-10.99,-1.29,;-8.68,-2.62,;-7.91,-3.96,;-6.37,-3.96,;-5.6,-2.62,;-6.37,-1.29,;-7.91,-1.29,;-4.06,-2.62,;-3.29,-3.96,;-3.29,-1.29,;-4.06,.04,;-3.29,1.38,;-1.75,1.38,;-.98,.04,;-1.75,-1.29,;-.98,-2.62,;.56,-2.62,;1.33,-1.29,;2.87,-1.29,;3.64,.04,;2.87,1.38,;1.33,1.38,;.56,.04,;5.18,.04,;5.18,1.58,;6.72,.04,;8.26,.04,;6.72,-1.5,;6.72,1.58,;5.18,-1.5,;3.84,-2.27,;6.51,-2.27,;5.18,-3.04,;-.21,1.38,;1.12,2.15,;-.21,2.92,;-.98,2.71,;-2.52,2.71,;-3.29,4.05,;-2.52,5.38,;-.98,5.38,;-.21,4.05,)|
OC(=O)C12CCC(CC1)(CC2)C(=O)N1CCCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1
C[C@@]1(CC[C@@H](CC1)C(=O)N1CCCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1)C(O)=O |r,wU:4.7,1.0,wD:1.46,(-9.63,-3.36,;-8.27,-2.63,;-7.5,-3.97,;-5.96,-3.97,;-5.19,-2.63,;-5.96,-1.3,;-7.5,-1.3,;-3.65,-2.63,;-2.88,-3.97,;-2.88,-1.3,;-3.65,.03,;-2.88,1.37,;-1.34,1.37,;-.57,.03,;-1.34,-1.3,;-.57,-2.63,;.97,-2.63,;1.74,-1.3,;3.28,-1.3,;4.05,.03,;3.28,1.37,;1.74,1.37,;.97,.03,;5.59,.03,;5.59,1.57,;7.13,.03,;8.67,.03,;7.13,-1.51,;7.13,1.57,;5.59,-1.51,;4.26,-2.28,;6.93,-2.28,;5.59,-3.05,;.2,1.37,;1.54,2.14,;.2,2.91,;-.57,2.7,;-2.11,2.7,;-2.88,4.04,;-2.11,5.37,;-.57,5.37,;.2,4.04,;-9.63,-1.91,;-9.68,-.37,;-10.93,-2.73,)|
OC(=O)c1ccc(cc1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1
OC(=O)Cc1ccc(CC(=O)N2CCC3(C2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2cccc(F)c2)cc1
Fc1cccc(c1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)Cc1ccc(cc1)C#N
OC(=O)C1CCC(C1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1 |w:8.8,3.2|
OC(=O)c1cccc(CC(=O)N2CCC3(C2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2cccc(F)c2)c1
OC(=O)c1cncc(CC(=O)N2CCC3(C2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2cccc(F)c2)c1
OC(=O)C1CC2(C1)CC(C2)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1 |w:3.2,(8.74,1.34,;7.97,2.67,;8.74,4,;6.43,2.67,;5.34,3.76,;4.25,2.67,;5.34,1.58,;3.16,3.76,;2.08,2.67,;3.16,1.58,;.54,2.67,;-.23,4,;-.23,1.34,;.39,-.07,;-.75,-1.1,;-2.09,-.33,;-1.77,1.17,;-2.91,2.2,;-4.38,1.73,;-4.7,.22,;-6.16,-.25,;-6.48,-1.76,;-5.34,-2.79,;-3.87,-2.31,;-3.55,-.81,;-7.94,-2.24,;-7.47,-3.7,;-9.41,-2.71,;-10.87,-3.19,;-9.89,-1.25,;-8.93,-4.18,;-8.42,-.77,;-7.39,.37,;-9.93,-.45,;-8.9,.69,;-2.25,-1.86,;-3.15,-3.11,;-1.62,-3.27,;-1,-2.77,;-1.16,-4.3,;.08,-5.21,;1.49,-4.58,;1.65,-3.05,;3.06,-2.42,;.41,-2.14,)|
OC(=O)c1ccc(cc1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C1CCC(C1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:8.8,3.2|
OC(=O)c1cnc(cn1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1
Cc1cc(cc(c1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1)C(O)=O
OC(=O)C1CC2(C1)CC(C2)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:3.2,wU:16.18,wD:15.39,(8.82,1.61,;8.05,2.94,;8.82,4.28,;6.51,2.94,;5.42,4.03,;4.34,2.94,;5.42,1.85,;3.25,4.03,;2.16,2.94,;3.25,1.85,;.62,2.94,;-.15,4.28,;-.15,1.61,;.47,.2,;-.67,-.83,;-2,-.06,;-1.68,1.45,;-2.83,2.48,;-4.29,2,;-4.61,.5,;-6.08,.02,;-6.4,-1.49,;-5.25,-2.52,;-3.79,-2.04,;-3.47,-.54,;-7.86,-1.96,;-7.39,-3.43,;-9.33,-2.44,;-10.79,-2.91,;-9.8,-.97,;-8.85,-3.9,;-8.34,-.5,;-7.31,.65,;-9.84,-.18,;-8.81,.97,;-2.16,-1.59,;-3.07,-2.84,;-1.54,-3,;-.92,-2.5,;.49,-1.87,;1.73,-2.77,;1.57,-4.31,;2.82,-5.21,;.17,-4.93,;-1.08,-4.03,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccc(cc1)-c1nnco1 |r|
OCc1ccc(cc1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccc(cc1)-c1nn[nH]n1 |r|
NS(=O)(=O)c1ccc(cc1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)Cc1ccncc1 |r|
OC(=O)c1ccc(cc1)S(=O)(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)Cc1cncnc1 |r|
NS(=O)(=O)c1cc(ccc1Cl)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccc2C(=O)NCc2c1 |r|
NS(=O)(=O)c1cccc(c1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccc2NC(=O)Cc2c1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccc2[nH]cnc2c1 |r|
OC(=O)c1cc(cc(c1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(O)=O |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccc2NC(=O)COc2c1 |r|
OC(=O)C1CC2(C1)CC(C2)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1 |r,w:3.2,wU:16.18,wD:15.39,(8.93,1.43,;8.16,2.76,;8.93,4.09,;6.62,2.76,;5.53,3.85,;4.44,2.76,;5.53,1.67,;3.36,3.85,;2.27,2.76,;3.36,1.67,;.73,2.76,;-.04,4.09,;-.04,1.43,;.58,.02,;-.56,-1.01,;-1.9,-.24,;-1.58,1.27,;-2.72,2.3,;-4.18,1.82,;-4.5,.31,;-5.97,-.16,;-6.29,-1.67,;-5.14,-2.7,;-3.68,-2.22,;-3.36,-.72,;-7.75,-2.14,;-7.28,-3.61,;-9.22,-2.62,;-10.68,-3.09,;-9.69,-1.15,;-8.74,-4.08,;-8.23,-.68,;-7.2,.47,;-9.74,-.36,;-8.71,.79,;-2.06,-1.77,;-2.96,-3.02,;-1.43,-3.18,;-.81,-2.68,;.6,-2.05,;1.84,-2.96,;1.68,-4.49,;.27,-5.11,;-.97,-4.21,)|
OC(=O)c1ccc(cc1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccc2c(c1)C(=O)NS2(=O)=O |r|
OC(=O)c1cc(Cl)c(cc1Cl)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
NC(=O)c1ccc(cc1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
NC(=O)c1ccc(C(=O)N2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)c(F)c1 |r|
OC(=O)C1CCCC(C1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)c1cc(O)c(cc1O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCCCC1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccccc1 |r|
NC(=O)c1cccc(c1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Cn1ccc(cc1=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Cn1cc(ccc1=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
O[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:4.7,13.14,wD:12.35,1.0,(-9.96,.08,;-8.51,-.44,;-8.24,-1.96,;-6.79,-2.48,;-5.61,-1.49,;-5.88,.03,;-7.33,.55,;-4.16,-2.01,;-3.89,-3.52,;-2.99,-1.01,;-3.1,.52,;-1.67,1.1,;-.68,-.07,;-1.49,-1.38,;-.76,-2.74,;.78,-2.79,;1.59,-1.48,;3.13,-1.53,;3.94,-.22,;3.21,1.14,;1.67,1.19,;.86,-.12,;5.48,-.26,;5.53,1.28,;7.02,-.31,;8.56,-.36,;6.97,-1.85,;7.07,1.23,;5.43,-1.8,;4.07,-2.53,;6.74,-2.61,;5.38,-3.34,;-.01,1.31,;1.27,2.18,;-.12,2.85,;-.87,2.59,;-2.41,2.48,;-3.28,3.75,;-2.61,5.14,;-3.47,6.41,;-1.07,5.25,;-.2,3.98,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCC2(CC1)NC(=O)NC2=O |r,w:38.45,38.50,wU:14.14,wD:10.10,(-4.49,4.9,;-3.24,4,;-3.41,2.47,;-2.16,1.56,;-.75,2.19,;-.59,3.72,;-1.84,4.62,;.49,1.28,;1.4,2.53,;-.13,2.69,;.33,-.25,;-1,.52,;-2.15,-.51,;-1.52,-1.92,;.01,-1.76,;1.16,-2.79,;2.62,-2.31,;2.94,-.8,;4.41,-.33,;4.73,1.18,;3.58,2.21,;2.12,1.73,;1.8,.23,;6.19,1.65,;5.71,3.12,;7.66,2.13,;9.12,2.61,;8.13,.66,;7.18,3.59,;6.67,.19,;5.64,-.96,;8.17,-.13,;7.14,-1.28,;-2.29,-3.25,;-1.52,-4.58,;-3.83,-3.25,;-4.6,-4.58,;-6.14,-4.58,;-6.91,-3.25,;-6.14,-1.92,;-4.6,-1.92,;-7.81,-4.5,;-9.28,-4.02,;-10.53,-4.93,;-9.28,-2.48,;-7.81,-2.01,;-7.34,-.54,)|
OC(=O)C1CC2(C1)CC(C2)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C1CC2(C1)CC(C2)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)C12CCN(C1COc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCC2(CC1)NC(=O)NC2=O |(-4.49,4.9,;-3.24,4,;-3.41,2.47,;-2.16,1.56,;-.75,2.19,;-.59,3.72,;-1.84,4.62,;.49,1.28,;1.4,2.53,;-.13,2.69,;.33,-.25,;-1,.52,;-2.15,-.51,;-1.52,-1.92,;.01,-1.76,;1.16,-2.79,;2.62,-2.31,;2.94,-.8,;4.41,-.33,;4.73,1.18,;3.58,2.21,;2.12,1.73,;1.8,.23,;6.19,1.65,;5.71,3.12,;7.66,2.13,;9.12,2.61,;8.13,.66,;7.18,3.59,;6.67,.19,;5.64,-.96,;8.17,-.13,;7.14,-1.28,;-2.29,-3.25,;-1.52,-4.58,;-3.83,-3.25,;-4.6,-4.58,;-6.14,-4.58,;-6.91,-3.25,;-6.14,-1.92,;-4.6,-1.92,;-7.81,-4.5,;-9.28,-4.02,;-10.53,-4.93,;-9.28,-2.48,;-7.81,-2.01,;-7.34,-.54,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)[C@H]1CC[C@@H](CC1)c1nnn[nH]1 |r,wU:14.14,38.45,wD:10.10,35.38,(-2.52,5.85,;-1.66,4.58,;-2.33,3.19,;-1.46,1.92,;.07,2.03,;.74,3.42,;-.12,4.69,;.94,.76,;2.21,1.62,;.83,2.29,;.27,-.63,;-.72,.54,;-2.15,-.04,;-2.04,-1.57,;-.54,-1.94,;.19,-3.3,;1.73,-3.35,;2.54,-2.04,;4.08,-2.08,;4.89,-.78,;4.16,.58,;2.62,.63,;1.81,-.68,;6.43,-.82,;6.48,.72,;7.97,-.87,;9.51,-.92,;7.92,-2.41,;8.01,.67,;6.38,-2.36,;5.02,-3.09,;7.69,-3.17,;6.33,-3.9,;-3.21,-2.57,;-2.94,-4.08,;-4.66,-2.05,;-4.93,-.53,;-6.38,-.01,;-7.56,-1,;-7.29,-2.52,;-5.84,-3.04,;-9.01,-.48,;-10.28,-1.35,;-11.5,-.4,;-10.98,1.05,;-9.44,1,)|
CS(=O)(=O)c1ccc(cc1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)CC1CCS(=O)(=O)C1 |r,w:36.39|
CC(=O)N1CC(C1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CS(=O)(=O)N1CCC(CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)CC1CCS(=O)(=O)C1 |r|
CS(=O)(=O)N1CCC(CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1 |r|
Cc1cc(ccc1F)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCN(CC1)S(C)(=O)=O
CS(=O)(=O)N1CCC(CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccc(cc1)-n1cnnn1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccc(cc1)C#N |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)CC1CCS(=O)(=O)CC1 |r|
FC(F)(F)C(F)(c1ccc2c(OCC3N(CCC23S(=O)(=O)c2ccccc2)C(=O)CC2CCS(=O)(=O)CC2)c1)C(F)(F)F
CC(=O)N1CCC(CC1C(O)=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:8.9|
OC(=O)c1cc(ccc1Cl)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
COc1ccc(cc1C#N)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Oc1c(F)cc(cc1F)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)c1c(F)cc(cc1F)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCC(CO)(CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CC(CC(=O)N2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)C1 |r|
CS(=O)(=O)N1CC(CC(=O)N2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)C1 |r|
CS(=O)(=O)N1CCC(CC(=O)N2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)CC1 |r|
OC(=O)c1cc(ccc1O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccc(CC#N)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccc(C#N)c(F)c1 |r|
NC(=O)c1c(F)cc(cc1F)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC1CC(CCS1(=O)=O)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)c(C)c1
CC1CC(CCS1(=O)=O)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1
Cc1cc(ccc1F)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)[C@H]1CC[C@@H](CC1)C(O)=O |r,wU:36.39,wD:39.46,(-.14,6.13,;-.81,4.74,;.05,3.47,;-.62,2.08,;-2.15,1.97,;-3.02,3.24,;-2.35,4.63,;-3.22,5.9,;.25,.81,;1.52,1.67,;.13,2.34,;-.42,-.58,;-1.42,.59,;-2.84,.01,;-2.73,-1.52,;-1.23,-1.89,;-.51,-3.25,;1.03,-3.3,;1.85,-1.99,;3.38,-2.03,;4.2,-.73,;3.47,.63,;1.93,.68,;1.12,-.63,;5.73,-.77,;5.78,.77,;7.27,-.82,;8.81,-.87,;7.23,-2.36,;7.32,.72,;5.69,-2.31,;4.33,-3.04,;7,-3.12,;5.64,-3.85,;-3.91,-2.52,;-3.63,-4.03,;-5.35,-2,;-6.53,-2.99,;-7.98,-2.47,;-8.25,-.95,;-7.08,.04,;-5.63,-.48,;-9.7,-.43,;-10.88,-1.43,;-9.97,1.08,)|
CC(C)c1cc(ccc1F)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)[C@H]1CC[C@@H](CC1)C(O)=O |r,wU:38.41,wD:41.48,(1.48,5.69,;-.06,5.58,;-.93,6.85,;-.73,4.19,;.14,2.92,;-.53,1.53,;-2.07,1.42,;-2.94,2.69,;-2.27,4.08,;-3.13,5.35,;.33,.26,;1.61,1.13,;.22,1.8,;-.34,-1.13,;-1.33,.05,;-2.76,-.53,;-2.64,-2.07,;-1.15,-2.43,;-.42,-3.79,;1.12,-3.84,;1.93,-2.53,;3.47,-2.58,;4.28,-1.27,;3.55,.09,;2.01,.13,;1.2,-1.17,;5.82,-1.32,;5.87,.22,;7.36,-1.37,;8.9,-1.41,;7.31,-2.91,;7.41,.17,;5.77,-2.86,;4.41,-3.59,;7.08,-3.67,;5.72,-4.4,;-3.82,-3.06,;-3.55,-4.58,;-5.27,-2.54,;-6.45,-3.53,;-7.9,-3.01,;-8.17,-1.5,;-6.99,-.5,;-5.54,-1.03,;-9.62,-.98,;-10.79,-1.97,;-9.89,.54,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCS(=O)(=O)C1 |r,w:33.38|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCS(=O)(=O)C1 |r|
OC(=O)[C@@]1(O)CC[C@@H](CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:16.17,3.2,wD:15.38,7.10,3.3,(-8.47,1.84,;-8.94,.37,;-10.45,.04,;-7.91,-.77,;-9.43,-.99,;-6.73,.22,;-5.28,-.3,;-5.01,-1.81,;-6.18,-2.81,;-7.63,-2.29,;-3.56,-2.33,;-3.29,-3.85,;-2.38,-1.34,;-2.5,.2,;-1.07,.78,;-.08,-.4,;-.89,-1.71,;-.16,-3.06,;1.38,-3.11,;2.19,-1.8,;3.73,-1.85,;4.54,-.54,;3.81,.81,;2.27,.86,;1.46,-.45,;6.08,-.59,;6.13,.95,;7.62,-.64,;9.16,-.69,;7.57,-2.18,;7.67,.9,;6.03,-2.13,;4.68,-2.86,;7.34,-2.94,;5.99,-3.67,;.59,.99,;1.87,1.85,;.48,2.52,;-.27,2.26,;-1.81,2.15,;-2.67,3.42,;-2,4.81,;-2.87,6.08,;-.47,4.92,;.4,3.65,)|
CC(C)c1cc(ccc1F)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)[C@@]1(F)CC[C@@H](CC1)C(O)=O |r,wU:38.41,wD:42.49,38.42,(1.46,5.51,;-.08,5.39,;-.95,6.67,;-.75,4.01,;.12,2.73,;-.55,1.35,;-2.09,1.23,;-2.96,2.51,;-2.29,3.89,;-3.15,5.17,;.31,.07,;1.58,.94,;.2,1.61,;-.36,-1.31,;-1.35,-.14,;-2.78,-.72,;-2.67,-2.26,;-1.17,-2.62,;-.44,-3.98,;1.1,-4.03,;1.91,-2.72,;3.45,-2.77,;4.26,-1.46,;3.53,-.1,;1.99,-.05,;1.18,-1.36,;5.8,-1.51,;5.85,.03,;7.34,-1.55,;8.88,-1.6,;7.29,-3.09,;7.39,-.01,;5.75,-3.05,;4.39,-3.77,;7.06,-3.86,;5.7,-4.58,;-3.84,-3.25,;-3.57,-4.77,;-5.29,-2.73,;-5.55,-4.25,;-6.83,-2.73,;-7.61,-1.4,;-6.84,-.07,;-5.3,-.06,;-4.53,-1.39,;-7.62,1.26,;-9.16,1.26,;-6.85,2.6,)|
CC(C)c1cc(ccc1F)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1(O)CCS(=O)(=O)CC1
CC(C)c1cc(ccc1F)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C12CCC(CC1)(CC2)C(O)=O
OC(=O)[C@H]1CC[C@@](F)(CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)c(Cl)c1 |r,wU:6.10,wD:3.2,6.6,(-9.24,1.78,;-7.7,1.79,;-6.93,3.12,;-6.92,.46,;-7.69,-.88,;-6.91,-2.21,;-5.37,-2.21,;-5.64,-3.72,;-4.61,-.87,;-5.38,.46,;-3.93,-2.73,;-3.65,-4.24,;-2.75,-1.73,;-2.86,-.2,;-1.44,.38,;-.44,-.79,;-1.25,-2.1,;-.53,-3.46,;1.01,-3.51,;1.83,-2.2,;3.36,-2.24,;4.18,-.94,;3.45,.42,;1.91,.47,;1.1,-.84,;5.71,-.98,;5.76,.56,;7.25,-1.03,;8.79,-1.08,;7.21,-2.57,;7.3,.51,;5.67,-2.52,;4.31,-3.25,;6.98,-3.33,;5.62,-4.06,;.23,.6,;1.5,1.46,;.11,2.13,;-.64,1.87,;-2.17,1.76,;-3.04,3.03,;-2.37,4.42,;-3.24,5.69,;-.83,4.53,;-.16,5.92,;.03,3.26,)|
OC1(CCS(=O)(=O)CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)c(Cl)c1
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)c(Cl)c1 |r,wU:6.9,wD:3.2,(-10.88,-1.43,;-9.7,-.43,;-9.97,1.08,;-8.25,-.95,;-7.98,-2.47,;-6.53,-2.99,;-5.35,-2,;-5.63,-.48,;-7.08,.04,;-3.91,-2.52,;-3.63,-4.03,;-2.73,-1.52,;-2.84,.01,;-1.42,.59,;-.42,-.58,;-1.23,-1.89,;-.51,-3.25,;1.03,-3.3,;1.85,-1.99,;3.38,-2.03,;4.2,-.73,;3.47,.63,;1.93,.68,;1.12,-.63,;5.73,-.77,;5.78,.77,;7.27,-.82,;8.81,-.87,;7.23,-2.36,;7.32,.72,;5.69,-2.31,;4.33,-3.04,;7,-3.12,;5.64,-3.85,;.25,.81,;1.52,1.67,;.13,2.34,;-.62,2.08,;-2.15,1.97,;-3.02,3.24,;-2.35,4.63,;-3.22,5.9,;-.81,4.74,;-.14,6.13,;.05,3.47,)|
Cc1cc(ccc1F)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)[C@@]1(F)CC[C@@H](CC1)C(O)=O |r,wU:36.39,wD:40.47,36.40,(-.16,5.92,;-.83,4.53,;.03,3.26,;-.64,1.87,;-2.17,1.76,;-3.04,3.03,;-2.37,4.42,;-3.24,5.69,;.23,.6,;1.5,1.46,;.11,2.13,;-.44,-.79,;-1.44,.38,;-2.86,-.2,;-2.75,-1.73,;-1.25,-2.1,;-.53,-3.46,;1.01,-3.51,;1.83,-2.2,;3.36,-2.24,;4.18,-.94,;3.45,.42,;1.91,.47,;1.1,-.84,;5.71,-.98,;5.76,.56,;7.25,-1.03,;8.79,-1.08,;7.21,-2.57,;7.3,.51,;5.67,-2.52,;4.31,-3.25,;6.98,-3.33,;5.62,-4.06,;-3.93,-2.73,;-3.65,-4.24,;-5.37,-2.21,;-5.64,-3.72,;-6.91,-2.21,;-7.69,-.88,;-6.92,.46,;-5.38,.46,;-4.61,-.87,;-7.7,1.79,;-9.24,1.78,;-6.93,3.12,)|
OC(=O)C1CCC(C1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C1CCC(CC(=O)N2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)C1 |r,w:7.6,3.2|
CS(=O)(=O)N1CCC(F)(CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C12CC(C1)(C2)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CS(=O)(=O)NC1CC2(C1)CC(C2)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:5.4,wU:18.20,wD:17.41,(9.47,2.24,;8.13,1.47,;8.9,.13,;6.8,.7,;7.36,2.8,;5.82,2.8,;4.74,3.89,;3.65,2.8,;4.74,1.71,;2.56,3.89,;1.47,2.8,;2.56,1.71,;-.07,2.8,;-.84,4.14,;-.84,1.47,;-.21,.06,;-1.36,-.97,;-2.69,-.2,;-2.37,1.31,;-3.52,2.34,;-4.98,1.86,;-5.3,.35,;-6.77,-.12,;-7.09,-1.63,;-5.94,-2.66,;-4.48,-2.18,;-4.16,-.68,;-8.55,-2.1,;-8.08,-3.57,;-10.02,-2.58,;-11.48,-3.05,;-10.49,-1.11,;-9.54,-4.04,;-9.03,-.64,;-8,.51,;-10.53,-.32,;-9.5,.83,;-2.85,-1.73,;-3.76,-2.98,;-2.23,-3.14,;-1.61,-2.64,;-.2,-2.01,;1.04,-2.92,;.88,-4.45,;2.13,-5.35,;-.52,-5.07,;-1.77,-4.17,)|
OCC1(CCNCC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CS(=O)(=O)N1CCC(CO)(CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCOCC1 |r|
NC(=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CNC(=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
NC(=O)CC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ncc[nH]1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1nnn[nH]1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)Cc1nnn[nH]1 |r|
CCS(=O)(=O)c1ccc(CC(=O)N2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)cc1 |r|
CC(C)(C)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1(CCC1)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C#C |r|
CC#CC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CC1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CC(F)(F)C1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1(CCC1)C#N |r|
CC1(C)C(C(=O)N2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)C1(C)C |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)[C@H]1[C@H]2COC[C@@H]12 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCC1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)CC(F)(F)F |r|
CC1(CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
FC1CC(C1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:11.12,wD:10.33,(-9.63,-.11,;-8.18,-.63,;-7.53,-2.03,;-6.13,-1.37,;-6.79,.02,;-4.68,-1.89,;-4.41,-3.41,;-3.51,-.9,;-3.62,.64,;-2.19,1.22,;-1.2,.05,;-2.01,-1.26,;-1.28,-2.62,;.26,-2.67,;1.07,-1.36,;2.61,-1.41,;3.42,-.1,;2.69,1.26,;1.15,1.31,;.34,-0,;4.96,-.15,;5,1.39,;6.5,-.2,;8.04,-.24,;6.45,-1.73,;6.54,1.34,;4.91,-1.69,;3.55,-2.41,;6.22,-2.5,;4.86,-3.23,;-.53,1.43,;.74,2.3,;-.64,2.97,;-1.4,2.71,;-2.93,2.59,;-3.8,3.87,;-3.13,5.25,;-3.99,6.53,;-1.59,5.37,;-.73,4.09,)|
CC(O)(C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r,w:1.1|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1(CC1)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1COC1 |r|
OC(=O)C1(CCC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1(CCCC1)C(F)(F)F |r|
CC(C)(C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(C)(O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OCC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCC(F)(F)CC1 |r|
O[C@@H](C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CS(=O)(=O)CC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)S(=O)(=O)CC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)S(C)(=O)=O |r,w:1.0|
Fc1ccc(cc1)S(=O)(=O)CC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)CS(=O)(=O)c1ccccc1 |r|
CC(CS(=O)(=O)c1ccc(Cl)cc1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:1.0|
CC(C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)S(=O)(=O)c1ccc(cn1)C(F)(F)F |r,w:1.0|
CC(CC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)S(=O)(=O)c1ccc(Cl)cc1 |r,w:1.0|
CS(=O)(=O)CCC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)CS(=O)(=O)c1ccc(Cl)cc1 |r|
Cc1ccc(cc1)S(=O)(=O)CCC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
NC(C1CCS(=O)(=O)CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:1.0|
CC(=O)NC(C1CCS(=O)(=O)CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OCC(=O)NC(C1CCS(=O)(=O)CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:5.4|
NC1(CCC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:1.1|
O[C@H](C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
C[C@@](O)(C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CCC(C)(O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:2.3|
OC1(CCCCC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(C1CCOCC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:1.0|
OC1(CCC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC1(CCOCC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC1(CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(C)[C@H](O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
O[C@H](C1CCCCC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@](O)(C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CCNS(=O)(=O)CCC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC1(CCS(=O)(=O)CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
NC1(CCS(=O)(=O)CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CCC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C=C |r|
CCC(C)(O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C12CCC(CC1)(C2)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)[C@@H]1[C@H]2C[C@@H](C[C@@H]12)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CCC[C@@]1(CC[C@@H](CC1)C(O)=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:18.19,3.12,wD:17.40,6.9,3.2,(-1.4,-4.2,;-1.13,-2.68,;-2.32,-1.7,;-3.76,-2.23,;-2.99,-3.56,;-3.75,-4.9,;-5.29,-4.9,;-6.07,-3.57,;-5.3,-2.24,;-6.06,-6.24,;-7.6,-6.25,;-5.28,-7.57,;-4.04,-.72,;-5.48,-.19,;-2.86,.28,;-2.97,1.81,;-1.55,2.4,;-.55,1.22,;-1.36,-.09,;-.64,-1.44,;.9,-1.49,;1.71,-.18,;3.25,-.23,;4.07,1.08,;3.34,2.43,;1.8,2.48,;.99,1.17,;5.6,1.03,;5.56,-.51,;7.14,.98,;8.68,.93,;7.19,2.52,;7.1,-.56,;5.65,2.57,;7.01,3.3,;4.34,3.38,;5.7,4.11,;.12,2.61,;1.39,3.47,;0,4.14,;-.75,3.88,;-2.28,3.77,;-3.15,5.04,;-2.48,6.43,;-3.35,7.7,;-.94,6.54,;-.08,5.27,)|
COCC1(CCC(CC1)C(O)=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:3.2,wU:18.19,wD:17.40,(-1.4,-4.26,;-1.14,-2.74,;-2.32,-1.76,;-3.77,-2.29,;-2.99,-3.62,;-3.76,-4.96,;-5.3,-4.96,;-6.07,-3.63,;-5.31,-2.3,;-6.06,-6.3,;-7.6,-6.31,;-5.29,-7.63,;-4.04,-.77,;-5.49,-.25,;-2.86,.22,;-2.98,1.76,;-1.55,2.34,;-.56,1.16,;-1.37,-.15,;-.64,-1.5,;.9,-1.55,;1.71,-.24,;3.25,-.29,;4.06,1.02,;3.33,2.37,;1.79,2.42,;.98,1.11,;5.6,.97,;5.55,-.57,;7.14,.92,;8.68,.87,;7.19,2.46,;7.09,-.62,;5.65,2.51,;7.01,3.24,;4.34,3.32,;5.7,4.05,;.11,2.55,;1.39,3.41,;0,4.08,;-.75,3.82,;-2.29,3.71,;-3.15,4.98,;-2.48,6.37,;-3.35,7.64,;-.95,6.48,;-.08,5.21,)|
OC(=O)C1(O)CCC(CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:3.3,wU:16.17,wD:15.38,(-10.39,.27,;-9.44,-.94,;-10.01,-2.37,;-7.91,-.72,;-8.95,.42,;-7.64,-2.24,;-6.19,-2.76,;-5.01,-1.77,;-5.29,-.25,;-6.74,.27,;-3.57,-2.29,;-3.29,-3.8,;-2.39,-1.29,;-2.5,.24,;-1.08,.82,;-.08,-.35,;-.89,-1.66,;-.17,-3.02,;1.37,-3.07,;2.18,-1.76,;3.72,-1.81,;4.54,-.5,;3.81,.86,;2.27,.91,;1.46,-.4,;6.07,-.54,;6.03,-2.08,;7.61,-.59,;9.15,-.64,;7.66,.95,;7.57,-2.13,;6.12,.99,;7.48,1.72,;4.81,1.81,;6.17,2.53,;.59,1.03,;1.86,1.9,;.47,2.57,;-.28,2.31,;-1.81,2.19,;-2.68,3.47,;-2.01,4.85,;-2.88,6.13,;-.47,4.97,;.39,3.69,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCOC1 |r,w:33.38|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1(CCOCC1)C#N |r|
C[C@H]1C[C@H](C[C@@H](C)S1(=O)=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC1(CCNCC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@H]1C[C@H](C[C@@H](C)S1(=O)=O)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1 |r|
OCCN1[C@@H](C[C@H](F)C1=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
FC(F)(F)C(F)(c1ccc2c(CCC3N(CCC23S(=O)(=O)c2ccc(Cl)cc2)C(=O)c2ccc3cncn3c2)c1)C(F)(F)F
CC1(C)OC(=O)CC1C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:8.8|
CC(C)C1CC(CCO1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:3.2|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccc2cncn2c1 |r|
CO[C@H]1C[C@H](N(C)C1=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)[C@H]1CC[C@@](F)(CC1)C(=O)N1CCCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:6.6,3.2,wD:6.10,(-10.3,0,;-8.85,.53,;-8.59,2.05,;-7.67,-.46,;-6.23,.07,;-5.05,-.92,;-5.31,-2.44,;-5.05,-3.96,;-6.76,-2.97,;-7.94,-1.98,;-3.77,-2.44,;-3,-3.77,;-3,-1.11,;-3.77,.23,;-3,1.56,;-1.46,1.56,;-.69,.23,;-1.46,-1.11,;-.69,-2.44,;.85,-2.44,;1.62,-1.11,;3.16,-1.11,;3.93,.23,;3.16,1.56,;1.62,1.56,;.85,.23,;5.47,.23,;5.47,1.77,;7.01,.23,;8.55,.23,;7.01,-1.31,;7.01,1.77,;5.47,-1.31,;4.13,-2.08,;6.8,-2.08,;5.47,-2.85,;.08,1.56,;1.41,2.33,;.08,3.1,;-.69,2.89,;-2.23,2.89,;-3,4.23,;-2.23,5.56,;-3,6.89,;-.69,5.56,;.08,4.23,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)CN1CCS(=O)(=O)CC1 |r|
Cc1cc(ccc1F)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)[C@@]1(O)CC[C@@H](CC1)C(O)=O |r,wU:36.40,40.47,wD:36.39,(-.16,5.92,;-.83,4.53,;.03,3.26,;-.64,1.87,;-2.17,1.76,;-3.04,3.03,;-2.37,4.42,;-3.24,5.69,;.23,.6,;1.5,1.46,;.11,2.13,;-.44,-.79,;-1.44,.38,;-2.86,-.2,;-2.75,-1.73,;-1.25,-2.1,;-.53,-3.46,;1.01,-3.51,;1.83,-2.2,;3.36,-2.24,;4.18,-.94,;3.45,.42,;1.91,.47,;1.1,-.84,;5.71,-.98,;5.76,.56,;7.25,-1.03,;8.79,-1.08,;7.21,-2.57,;7.3,.51,;5.67,-2.52,;4.31,-3.25,;6.98,-3.33,;5.62,-4.06,;-3.93,-2.73,;-3.65,-4.24,;-5.37,-2.21,;-5.64,-3.72,;-4.61,-.87,;-5.38,.46,;-6.92,.46,;-7.69,-.88,;-6.91,-2.21,;-7.7,1.79,;-6.93,3.12,;-9.24,1.78,)|
OC(=O)[C@H]1CC[C@@](F)(CC1)C(=O)N1CCCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1 |r,wU:6.6,3.2,wD:6.10,(-10.32,-.69,;-8.87,-.16,;-8.61,1.35,;-7.69,-1.15,;-6.25,-.63,;-5.07,-1.62,;-5.34,-3.13,;-5.07,-4.65,;-6.78,-3.66,;-7.96,-2.67,;-3.8,-3.13,;-3.03,-4.47,;-3.03,-1.8,;-3.8,-.46,;-3.03,.87,;-1.49,.87,;-.72,-.46,;-1.49,-1.8,;-.72,-3.13,;.82,-3.13,;1.59,-1.8,;3.13,-1.8,;3.9,-.46,;3.13,.87,;1.59,.87,;.82,-.46,;5.44,-.46,;5.44,1.08,;6.98,-.46,;8.52,-.46,;6.98,-2,;6.98,1.08,;5.44,-2,;4.11,-2.77,;6.78,-2.77,;5.44,-3.54,;.05,.87,;1.39,1.64,;.05,2.41,;-.72,2.2,;-2.26,2.2,;-3.03,3.54,;-2.26,4.87,;-.72,4.87,;.05,6.2,;.05,3.54,)|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CCC2(C1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:6.9,wD:3.2,(-10.01,1.35,;-9.74,-.16,;-10.91,-1.16,;-8.29,-.68,;-8.01,-2.2,;-6.57,-2.72,;-5.39,-1.73,;-5.66,-.21,;-7.11,.31,;-3.94,-2.25,;-3.67,-3.76,;-2.76,-1.25,;-2.88,.28,;-1.45,.87,;-.46,-.31,;-1.27,-1.62,;-.54,-2.98,;1,-3.02,;1.81,-1.72,;3.35,-1.76,;4.16,-.46,;3.43,.9,;1.89,.95,;1.08,-.36,;5.7,-.5,;5.75,1.04,;7.24,-.55,;8.78,-.6,;7.19,-2.09,;7.29,.99,;5.65,-2.04,;4.29,-2.77,;6.96,-2.85,;5.6,-3.58,;.21,1.08,;1.49,1.94,;.1,2.61,;-.65,2.35,;-2.19,2.24,;-3.05,3.51,;-2.38,4.9,;-3.25,6.17,;-.85,5.01,;.02,3.74,)|
OC(=O)C12CCC(CC1)(CC2)C(=O)N1CCC2(C1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(=O)[C@H]1CC[C@@](F)(CC1)C(=O)N1CCC2(C1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:6.10,wD:3.2,6.6,(-6.97,3.38,;-7.73,2.04,;-9.27,2.04,;-6.96,.71,;-7.72,-.62,;-6.95,-1.95,;-5.41,-1.95,;-5.67,-3.47,;-4.64,-.61,;-5.42,.72,;-3.96,-2.47,;-3.69,-3.98,;-2.78,-1.47,;-2.9,.06,;-1.47,.64,;-.48,-.53,;-1.29,-1.84,;-.56,-3.2,;.98,-3.25,;1.79,-1.94,;3.33,-1.99,;4.14,-.68,;3.41,.68,;1.87,.73,;1.06,-.58,;5.68,-.73,;5.73,.81,;7.22,-.77,;8.76,-.82,;7.17,-2.31,;7.27,.77,;5.63,-2.26,;4.28,-2.99,;6.94,-3.08,;5.58,-3.8,;.19,.85,;1.47,1.72,;.08,2.39,;-.67,2.13,;-2.21,2.01,;-3.07,3.29,;-2.4,4.67,;-3.27,5.95,;-.87,4.79,;-0,3.51,)|
C[C@@]1(CC[C@@H](CC1)C(O)=O)C(=O)N1CCC2(C1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:1.10,wD:4.7,1.0,(-5.67,-3.47,;-5.41,-1.95,;-6.95,-1.95,;-7.72,-.62,;-6.96,.71,;-5.42,.72,;-4.64,-.61,;-7.73,2.04,;-6.97,3.38,;-9.27,2.04,;-3.96,-2.47,;-3.69,-3.98,;-2.78,-1.47,;-2.9,.06,;-1.47,.64,;-.48,-.53,;-1.29,-1.84,;-.56,-3.2,;.98,-3.25,;1.79,-1.94,;3.33,-1.99,;4.14,-.68,;3.41,.68,;1.87,.73,;1.06,-.58,;5.68,-.73,;5.73,.81,;7.22,-.77,;8.76,-.82,;7.17,-2.31,;7.27,.77,;5.63,-2.26,;4.28,-2.99,;6.94,-3.08,;5.58,-3.8,;.19,.85,;1.47,1.72,;.08,2.39,;-.67,2.13,;-2.21,2.01,;-3.07,3.29,;-2.4,4.67,;-3.27,5.95,;-.87,4.79,;-0,3.51,)|
CN1[C@@H](C[C@H](F)C1=O)C(=O)N1CCC2(C1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1 |r|
FC(F)(F)C(F)(c1ccc2c(NCC3N(CCC23S(=O)(=O)c2ccccc2)C(=O)C2CCS(=O)(=O)CC2)c1)C(F)(F)F
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CCC2(C1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1 |r,wU:3.2,wD:6.9,(-10.97,-1.49,;-9.8,-.49,;-10.07,1.02,;-8.35,-1.01,;-7.17,-.02,;-5.72,-.54,;-5.45,-2.06,;-6.63,-3.05,;-8.07,-2.53,;-4,-2.58,;-3.73,-4.09,;-2.82,-1.58,;-2.94,-.05,;-1.51,.53,;-.52,-.64,;-1.33,-1.95,;-.6,-3.31,;.94,-3.36,;1.75,-2.05,;3.29,-2.09,;4.1,-.79,;3.37,.57,;1.83,.62,;1.02,-.69,;5.64,-.83,;5.69,.71,;7.18,-.88,;8.72,-.93,;7.13,-2.42,;7.23,.66,;5.59,-2.37,;4.23,-3.1,;6.9,-3.18,;5.54,-3.91,;.15,.74,;1.43,1.61,;.04,2.28,;-.71,2.02,;-2.25,1.91,;-3.11,3.18,;-2.44,4.57,;-.91,4.68,;-.04,3.41,)|
Fc1ccc(cc1)S(=O)(=O)C12CCN(C1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCS(=O)(=O)CC1
Fc1cccc(c1)S(=O)(=O)C12CCN(C1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCS(=O)(=O)CC1
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CCC2(C1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1 |r,wU:3.2,wD:6.9,(-10.03,.74,;-9.76,-.78,;-10.94,-1.77,;-8.31,-1.3,;-7.13,-.31,;-5.68,-.83,;-5.41,-2.34,;-6.59,-3.34,;-8.04,-2.82,;-3.96,-2.86,;-3.69,-4.38,;-2.79,-1.87,;-2.9,-.33,;-1.47,.25,;-.48,-.93,;-1.29,-2.24,;-.56,-3.59,;.98,-3.64,;1.79,-2.33,;3.33,-2.38,;4.14,-1.07,;3.41,.29,;1.87,.33,;1.06,-.98,;5.68,-1.12,;5.73,.42,;7.22,-1.17,;8.76,-1.22,;7.17,-2.71,;7.26,.37,;5.63,-2.66,;4.27,-3.39,;6.94,-3.47,;5.58,-4.2,;.19,.46,;1.46,1.32,;.08,1.99,;-.68,1.73,;-2.21,1.62,;-3.08,2.89,;-2.41,4.28,;-.87,4.39,;-.2,5.78,;-.01,3.12,)|
OC(=O)[C@H]1CC[C@@](F)(CC1)C(=O)N1CCC2(C1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1 |r,wU:3.2,6.6,wD:6.10,(-7.04,3.04,;-7.8,1.7,;-9.34,1.7,;-7.03,.37,;-5.49,.38,;-4.71,-.95,;-5.48,-2.29,;-5.74,-3.81,;-7.02,-2.29,;-7.79,-.96,;-4.03,-2.81,;-3.76,-4.33,;-2.85,-1.82,;-2.97,-.28,;-1.54,.3,;-.55,-.87,;-1.36,-2.18,;-.63,-3.54,;.91,-3.59,;1.72,-2.28,;3.26,-2.33,;4.07,-1.02,;3.34,.34,;1.81,.39,;.99,-.92,;5.61,-1.07,;5.66,.47,;7.15,-1.11,;8.69,-1.16,;7.1,-2.65,;7.2,.42,;5.56,-2.61,;4.21,-3.33,;6.87,-3.42,;5.52,-4.14,;.12,.51,;1.4,1.38,;.01,2.05,;-.74,1.79,;-2.28,1.67,;-3.14,2.95,;-2.47,4.33,;-.94,4.45,;-.07,3.17,)|
OC(=O)[C@@]1(F)CC[C@@H](CC1)C(=O)N1CCC2(C1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1 |r,wU:3.2,wD:7.10,3.3,(-10.01,-2.67,;-9.44,-1.24,;-10.39,-.03,;-7.91,-1.02,;-8.95,.12,;-6.74,-.02,;-5.29,-.54,;-5.01,-2.06,;-6.19,-3.05,;-7.64,-2.53,;-3.57,-2.58,;-3.29,-4.1,;-2.39,-1.59,;-2.5,-.05,;-1.08,.53,;-.08,-.64,;-.89,-1.95,;-.17,-3.31,;1.37,-3.36,;2.18,-2.05,;3.72,-2.1,;4.53,-.79,;3.81,.57,;2.27,.62,;1.46,-.69,;6.07,-.84,;6.12,.7,;7.61,-.89,;9.15,-.93,;7.57,-2.42,;7.66,.65,;6.03,-2.38,;4.67,-3.1,;7.33,-3.19,;5.98,-3.92,;.59,.74,;1.86,1.61,;.47,2.28,;-.28,2.02,;-1.81,1.9,;-2.68,3.18,;-2.01,4.56,;-.47,4.68,;.39,3.4,)|
OC(=O)[C@H]1CC[C@@](F)(CC1)C(=O)N1CCC2(C1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1 |r,wU:3.2,6.6,wD:6.10,(-7,2.77,;-7.76,1.43,;-9.3,1.43,;-6.99,.1,;-5.45,.11,;-4.68,-1.23,;-5.44,-2.56,;-5.7,-4.08,;-6.98,-2.57,;-7.76,-1.24,;-3.99,-3.08,;-3.72,-4.6,;-2.81,-2.09,;-2.93,-.55,;-1.5,.03,;-.51,-1.15,;-1.32,-2.46,;-.59,-3.81,;.95,-3.86,;1.76,-2.55,;3.3,-2.6,;4.11,-1.29,;3.38,.07,;1.84,.11,;1.03,-1.2,;5.65,-1.34,;5.7,.2,;7.19,-1.39,;8.73,-1.44,;7.14,-2.93,;7.24,.15,;5.6,-2.88,;4.24,-3.61,;6.91,-3.69,;5.55,-4.42,;.16,.24,;1.44,1.11,;.05,1.78,;-.7,1.51,;-2.24,1.4,;-3.11,2.67,;-2.44,4.06,;-.9,4.17,;-.23,5.56,;-.03,2.9,)|
OC1(CCS(=O)(=O)CC1)C(=O)N1CCC2(C1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CCC2(C1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1 |r,wU:3.2,wD:6.9,(-10.01,1.35,;-9.74,-.16,;-10.91,-1.16,;-8.29,-.68,;-7.11,.31,;-5.66,-.21,;-5.39,-1.73,;-6.57,-2.72,;-8.01,-2.2,;-3.94,-2.25,;-3.67,-3.76,;-2.76,-1.25,;-2.88,.28,;-1.45,.87,;-.46,-.31,;-1.27,-1.62,;-.54,-2.98,;1,-3.02,;1.81,-1.72,;3.35,-1.76,;4.16,-.46,;3.43,.9,;1.89,.95,;1.08,-.36,;5.7,-.5,;5.75,1.04,;7.24,-.55,;8.78,-.6,;7.19,-2.09,;7.29,.99,;5.65,-2.04,;4.29,-2.77,;6.96,-2.85,;5.6,-3.58,;.21,1.08,;1.49,1.94,;.1,2.61,;-.65,2.35,;-2.19,2.24,;-3.05,3.51,;-2.38,4.9,;-3.25,6.17,;-.85,5.01,;.02,3.74,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)[C@@H]1CCCC(=O)N1 |r|
Cc1cc(ccc1F)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCc2cncn2C1 |w:34.39|
Cc1cc(ccc1F)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1(O)CCS(=O)(=O)CC1
CN1[C@@H](C[C@H](F)C1=O)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)c(C)c1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCc2cncn2C1 |r,w:33.38|
FC(F)(F)C(F)(c1ccc2c(CCC3N(CCC23S(=O)(=O)c2ccc(Cl)cc2)C(=O)C2CCc3cncn3C2)c1)C(F)(F)F |w:28.32|
FC(F)(F)C(F)(c1ccc2c(NCC3N(CCC23S(=O)(=O)c2ccc(Cl)cc2)C(=O)C2CCS(=O)(=O)CC2)c1)C(F)(F)F
Fc1ccc(cc1F)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCS(=O)(=O)CC1
CN1C(CCCC1=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
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Fc1ccc(cc1)S(=O)(=O)C12CCN(C1Cc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccc2OCC(=O)Nc2c1
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OC(=O)[C@H]1CC[C@@](F)(CC1)C(=O)N1CC2Oc3cc(ccc3C2(C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:3.2,6.6,wD:6.10,(-10.75,.83,;-9.96,-.49,;-10.71,-1.84,;-8.42,-.47,;-7.67,.88,;-6.13,.9,;-5.34,-.42,;-4.15,-1.39,;-6.09,-1.76,;-7.63,-1.79,;-4.18,.59,;-4.47,2.1,;-2.72,.08,;-2.27,-1.39,;-.73,-1.42,;.49,-2.35,;1.76,-1.47,;3.26,-1.82,;4.31,-.7,;3.86,.78,;2.36,1.13,;1.31,0,;-.23,.03,;-1.46,.96,;.28,1.49,;1.44,2.5,;-.01,3,;-.73,2.65,;-2.24,2.36,;-3.25,3.53,;-2.75,4.98,;-3.76,6.15,;-1.24,5.27,;-.23,4.11,;5.81,-1.05,;6.16,.45,;7.31,-1.4,;8.81,-1.75,;6.96,-2.9,;7.66,.1,;5.46,-2.55,;3.99,-2.99,;6.58,-3.6,;5.11,-4.04,)|
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1Oc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCS(=O)(=O)CC1
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CC2CCc3cc(ccc3C2(C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:6.9,wD:3.2,(-11.06,-1.4,;-9.75,-2.21,;-9.8,-3.75,;-8.4,-1.49,;-7.09,-2.3,;-5.73,-1.57,;-5.68,-.03,;-6.99,.78,;-8.35,.05,;-4.32,.7,;-4.28,2.24,;-3.02,-.11,;-2.9,-1.65,;-1.41,-2.02,;-.68,-3.37,;.86,-3.42,;1.67,-2.11,;3.21,-2.16,;4.02,-.85,;3.29,.51,;1.75,.55,;.94,-.76,;-.6,-.71,;-1.59,.47,;.07,.68,;1.35,1.55,;-.04,2.22,;-.79,1.95,;-2.33,1.84,;-3.19,3.11,;-2.52,4.5,;-3.39,5.77,;-.99,4.61,;-.12,3.34,;5.56,-.9,;5.51,-2.44,;7.1,-.95,;8.64,-1,;7.05,-2.49,;7.15,.59,;5.61,.64,;6.97,1.37,;4.3,1.45,;5.66,2.18,)|
OC(=O)C12CCC(CC1)(CC2)C(=O)N1CC2CCc3cc(ccc3C2(C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F
OC(=O)C1CCCC(C1)C(=O)N1CC2CCc3cc(ccc3C2(C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCS(=O)(=O)CC1
CC(C)(O)CC(=O)N1CC2CCc3cc(ccc3C2(C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F
OC(=O)c1cc(on1)C(=O)N1CC2CCc3cc(ccc3C2(C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F
OC(=O)c1cnc(cn1)C(=O)N1CC2CCc3cc(ccc3C2(C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F
OC(=O)c1c[nH]c(c1)C(=O)N1CC2CCc3cc(ccc3C2(C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F
OC(=O)c1cc([nH]n1)C(=O)N1CC2CCc3cc(ccc3C2(C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)CC1CC(=O)NC(=O)C1
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1cncs1
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1cc(=O)cco1
CCCCC(O)C(=O)N1CC2CCc3cc(ccc3C2(C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |w:4.4|
OC(C1CCCCC1)C(=O)N1CC2CCc3cc(ccc3C2(C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |w:1.0|
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccnnc1
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1cc2cnccc2[nH]1
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1coc2CCCC(=O)c12
Oc1cc(on1)C(=O)N1CC2CCc3cc(ccc3C2(C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1cnc[nH]1
Cn1nc2CCCCc2c1C(=O)N1CC2CCc3cc(ccc3C2(C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1c[nH]c2nccnc12
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)Cc1ccc2ncccc2c1
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1cnc(Cl)s1
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1=CCCC1 |t:39|
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1cc[nH]n1
OCC(O)C(=O)N1CC2CCc3cc(ccc3C2(C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |w:2.2|
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1cnc(s1)C1OCCO1
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccsc1
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccns1
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1Cc2cc(Cl)ccc2N1 |w:33.38|
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccno1
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccon1
Fc1ccc(cc1)S(=O)(=O)C12CN(CC1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1(CC1)C#N
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CC2CCc3cc(ccc3C2(C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:3.2,wD:6.9,(-11.06,-1.4,;-9.75,-2.21,;-9.8,-3.75,;-8.4,-1.49,;-8.35,.05,;-6.99,.78,;-5.68,-.03,;-5.73,-1.57,;-7.09,-2.3,;-4.32,.7,;-4.28,2.24,;-3.02,-.11,;-2.9,-1.65,;-1.41,-2.02,;-.68,-3.37,;.86,-3.42,;1.67,-2.11,;3.21,-2.16,;4.02,-.85,;3.29,.51,;1.75,.55,;.94,-.76,;-.6,-.71,;-1.59,.47,;.07,.68,;1.35,1.55,;-.04,2.22,;-.79,1.95,;-2.33,1.84,;-3.19,3.11,;-2.52,4.5,;-3.39,5.77,;-.99,4.61,;-.12,3.34,;5.56,-.9,;5.51,-2.44,;7.1,-.95,;8.64,-1,;7.05,-2.49,;7.15,.59,;5.61,.64,;6.97,1.37,;4.3,1.45,;5.66,2.18,)|
CN1[C@@H](CCC1=O)C(=O)N1CC2CCc3cc(ccc3C2(C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CCC2(C(COc3cc(ccc23)C(F)(C(F)(F)F)C(F)(F)F)C1)S(=O)(=O)c1ccc(F)cc1 |r,wU:3.2,wD:6.9,(-10.19,-4.7,;-8.65,-4.7,;-7.88,-6.04,;-7.88,-3.37,;-8.65,-2.04,;-7.88,-.7,;-6.34,-.7,;-5.57,-2.04,;-6.34,-3.37,;-5.57,.63,;-6.34,1.96,;-4.03,.63,;-3.26,1.96,;-1.72,1.96,;-.95,.63,;-1.72,-.7,;-.95,-2.04,;.59,-2.04,;1.36,-.7,;2.9,-.7,;3.67,.63,;2.9,1.96,;1.36,1.96,;.59,.63,;5.21,.63,;5.21,-.91,;6.75,.63,;8.29,.63,;6.75,-.91,;6.75,2.17,;5.21,2.17,;6.54,2.94,;3.88,2.94,;5.21,3.71,;-3.26,-.7,;-.18,1.96,;1.15,2.73,;-.18,3.5,;-.95,3.3,;-2.49,3.3,;-3.26,4.63,;-2.49,5.97,;-3.26,7.3,;-.95,5.97,;-.18,4.63,)|
OC(=O)C1CC2(C1)CC(C2)C(=O)N1CCC2(C(COc3cc(ccc23)C(F)(C(F)(F)F)C(F)(F)F)C1)S(=O)(=O)c1ccc(F)cc1 |w:3.2,(8.32,-4.4,;7.55,-3.06,;8.32,-1.73,;6.01,-3.06,;4.92,-1.97,;3.83,-3.06,;4.92,-4.15,;2.74,-4.15,;1.65,-3.06,;2.74,-1.97,;.11,-3.06,;-.66,-4.4,;-.66,-1.73,;-2.2,-1.73,;-2.97,-.39,;-2.2,.94,;-.66,.94,;.11,2.27,;-.66,3.61,;-2.2,3.61,;-2.97,4.94,;-4.51,4.94,;-5.28,3.61,;-4.51,2.27,;-2.97,2.27,;-5.28,6.27,;-3.94,7.04,;-6.05,7.61,;-6.82,8.94,;-4.71,8.38,;-7.38,6.84,;-6.61,5.5,;-7.95,6.27,;-6.61,3.96,;-7.95,4.73,;.11,-.39,;-3.74,.94,;-5.07,1.71,;-5.07,.17,;-4.51,-.39,;-3.74,-1.73,;-4.51,-3.06,;-6.05,-3.06,;-6.82,-4.4,;-6.82,-1.73,;-6.05,-.39,)|
Fc1ccc(cc1)S(=O)(=O)C12CCN(CC1COc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCS(=O)(=O)CC1
CC(C)(O)CC(=O)N1CCC2(C(COc3cc(ccc23)C(F)(C(F)(F)F)C(F)(F)F)C1)S(=O)(=O)c1ccc(F)cc1
CN1[C@@H](CCC1=O)C(=O)N1CCC2(C(COc3cc(ccc23)C(F)(C(F)(F)F)C(F)(F)F)C1)S(=O)(=O)c1ccc(F)cc1 |r|
CN1[C@@H](C[C@H](F)C1=O)C(=O)N1CCC2(C(COc3cc(ccc23)C(F)(C(F)(F)F)C(F)(F)F)C1)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C1CCCC(C1)C(=O)N1CCC2(C(COc3cc(ccc23)C(F)(C(F)(F)F)C(F)(F)F)C1)S(=O)(=O)c1ccc(F)cc1 |w:3.2|
OC(=O)C1CCC(C1)C(=O)N1CCC2(C(COc3cc(ccc23)C(F)(C(F)(F)F)C(F)(F)F)C1)S(=O)(=O)c1ccc(F)cc1 |w:3.2|
C[C@@]1(CC[C@@H](CC1)C(O)=O)C(=O)N1CCC2(C(COc3cc(ccc23)C(F)(C(F)(F)F)C(F)(F)F)C1)S(=O)(=O)c1ccc(F)cc1 |r,wU:1.0,4.7,wD:1.10,(-4.42,-1.57,;-5.86,-1.05,;-7.04,-.06,;-8.49,-.59,;-8.76,-2.1,;-7.58,-3.09,;-6.13,-2.56,;-10.2,-2.63,;-11.38,-1.64,;-10.47,-4.14,;-5.09,.29,;-5.86,1.62,;-3.55,.29,;-2.78,1.62,;-1.24,1.62,;-.47,.29,;-1.24,-1.05,;-.47,-2.38,;1.07,-2.38,;1.84,-1.05,;3.38,-1.05,;4.15,.29,;3.38,1.62,;1.84,1.62,;1.07,.29,;5.69,.29,;5.69,-1.25,;7.23,.29,;8.77,.29,;7.23,-1.25,;7.23,1.83,;5.69,1.83,;7.02,2.6,;4.35,2.6,;5.69,3.37,;-2.78,-1.05,;.3,1.62,;1.63,2.39,;.3,3.16,;-.47,2.95,;-2.01,2.95,;-2.78,4.29,;-2.01,5.62,;-2.78,6.95,;-.47,5.62,;.3,4.29,)|
OC(=O)[C@H]1CC[C@@](O)(CC1)C(=O)N1CCC2(C(COc3cc(ccc23)C(F)(C(F)(F)F)C(F)(F)F)C1)S(=O)(=O)c1ccc(F)cc1 |r,wU:6.6,3.2,wD:6.10,(-11.38,-1.64,;-10.2,-2.63,;-10.47,-4.14,;-8.76,-2.1,;-8.49,-.59,;-7.04,-.06,;-5.86,-1.05,;-4.42,-1.57,;-6.13,-2.56,;-7.58,-3.09,;-5.09,.29,;-5.86,1.62,;-3.55,.29,;-2.78,1.62,;-1.24,1.62,;-.47,.29,;-1.24,-1.05,;-.47,-2.38,;1.07,-2.38,;1.84,-1.05,;3.38,-1.05,;4.15,.29,;3.38,1.62,;1.84,1.62,;1.07,.29,;5.69,.29,;5.69,-1.25,;7.23,.29,;8.77,.29,;7.23,-1.25,;7.23,1.83,;5.69,1.83,;7.02,2.6,;4.35,2.6,;5.69,3.37,;-2.78,-1.05,;.3,1.62,;1.63,2.39,;.3,3.16,;-.47,2.95,;-2.01,2.95,;-2.78,4.29,;-2.01,5.62,;-2.78,6.95,;-.47,5.62,;.3,4.29,)|
CCNC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC1CN(CCC1C(O)=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC1CN(CCC1C(O)=O)C(=O)N1CCC2(C1COc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(=O)C1(O)CCN(CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCN(CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NC1CCOCC1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)Nc1ccncc1 |r|
CC(C)(O)CNC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(O)CCNC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(O)[C@H](F)CNC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)Nc1ccnnc1 |r|
OC(=O)[C@@H]1CCCN(C1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C1CCN(CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)[C@H]1CCCN(C1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C1CCN(CC1)S(=O)(=O)N1CCC2(C1Cc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
Fc1ccc(cc1)S(=O)(=O)C12CCN(C1Cc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NC1CCOCC1
CC(C)(O)CNC(=O)N1CCC2(C1Cc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(=O)C1CCN(CC1)C(=O)N1CCC2(C1Cc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CC(C)(O)CCNC(=O)N1CCC2(C1Cc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CC(C)(O)CNC(=O)N1CC2CCc3cc(ccc3C2(C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F
CC1CN(CCC1C(O)=O)C(=O)N1CC2CCc3cc(ccc3C2(C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F
COC(=O)C1CCN(CC1C)C(=O)N1CC2CCc3cc(ccc3C2(C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NC1CCS(=O)(=O)CC1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NCC1CCS(=O)(=O)CC1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1CCS(=O)(=O)CC1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NCC1CCS(=O)(=O)C1 |r,w:36.40|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NC1CCS(=O)(=O)C1 |r,w:35.39|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1CC(C1)N1CCS(=O)(=O)CC1 |r|
CC1CS(=O)(=O)CCN1C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:1.0|
CN(C1CCS(=O)(=O)C1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:1.1|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N(C1CC1)C1CCS(=O)(=O)C1 |r,w:35.43|
CC(=O)NC1CS(=O)(=O)CCC1NC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:12.12,4.3|
OC1CS(=O)(=O)CC1NC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:8.8,1.0|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NC1CCS(=O)(=O)C1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1CCNC2CS(=O)(=O)CC12 |r,w:39.43,44.48|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NCC1CCS(=O)(=O)C1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1C[C@@H]2C[C@H]1CS2(=O)=O |r,TLB:33:35:40.41:38|
CN(C1CCOCC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CS(=O)(=O)N1CCN(CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CS(=O)(=O)N1CCC(CC1)NC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CS(=O)(=O)C1CCC(CC1)NC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:17.18,wD:16.39,(-11.07,-5,;-9.9,-4,;-8.9,-5.18,;-10.89,-2.83,;-8.72,-3.01,;-7.27,-3.53,;-6.1,-2.54,;-6.37,-1.02,;-7.82,-.5,;-8.99,-1.49,;-5.19,-.03,;-3.74,-.55,;-3.47,-2.06,;-2.57,.45,;-2.68,1.98,;-1.26,2.56,;-.26,1.39,;-1.07,.08,;-.34,-1.28,;1.2,-1.33,;2.01,-.02,;3.55,-.06,;4.36,1.24,;3.63,2.6,;2.09,2.65,;1.28,1.34,;5.9,1.2,;5.94,2.74,;7.44,1.15,;8.97,1.1,;7.39,-.39,;7.48,2.69,;5.85,-.34,;4.49,-1.07,;7.16,-1.15,;5.8,-1.88,;.41,2.78,;1.68,3.64,;.3,4.31,;-.46,4.05,;-1.99,3.94,;-2.86,5.21,;-2.19,6.6,;-3.05,7.87,;-.65,6.71,;.21,5.44,)|
CN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(=O)[C@H]1CC[C@@H](CC1)C(O)=O |r,wU:39.46,wD:36.39,(1.65,-4.15,;.92,-2.79,;-.62,-2.74,;-1.35,-1.38,;-2.84,-1.02,;-2.96,.52,;-1.53,1.1,;-.54,-.07,;1,-.12,;1.81,1.19,;3.35,1.14,;4.08,-.22,;3.27,-1.53,;1.73,-1.48,;5.62,-.27,;5.67,1.27,;7.16,-.32,;8.7,-.36,;7.11,-1.85,;7.21,1.22,;5.57,-1.81,;4.21,-2.53,;6.88,-2.62,;5.52,-3.35,;.13,1.31,;1.41,2.18,;.02,2.85,;-.73,2.59,;-2.27,2.47,;-3.13,3.75,;-2.46,5.13,;-3.33,6.41,;-.93,5.25,;-.06,3.97,;-4.02,-2.01,;-3.75,-3.53,;-5.47,-1.49,;-5.74,.03,;-7.19,.55,;-8.37,-.45,;-8.09,-1.96,;-6.64,-2.48,;-9.82,.07,;-10.99,-.92,;-10.09,1.59,)|
CCN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(=O)[C@H]1CC[C@@H](CC1)C(O)=O |r,wU:40.47,wD:37.40,(3.11,-3.95,;1.57,-3.9,;.84,-2.54,;-.7,-2.5,;-1.43,-1.14,;-2.92,-.77,;-3.04,.76,;-1.61,1.35,;-.62,.17,;.92,.12,;1.73,1.43,;3.27,1.38,;4,.03,;3.19,-1.28,;1.65,-1.24,;5.54,-.02,;5.59,1.52,;7.08,-.07,;8.62,-.12,;7.03,-1.61,;7.13,1.47,;5.49,-1.56,;4.13,-2.29,;6.8,-2.37,;5.44,-3.1,;.05,1.56,;1.33,2.42,;-.06,3.09,;-.81,2.83,;-2.35,2.72,;-3.22,3.99,;-2.55,5.38,;-3.41,6.65,;-1.01,5.49,;-.14,4.22,;-4.1,-1.77,;-3.83,-3.28,;-5.55,-1.25,;-5.82,.27,;-7.27,.79,;-8.45,-.2,;-8.18,-1.72,;-6.73,-2.24,;-9.9,.32,;-11.07,-.67,;-10.17,1.83,)|
CN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(=O)C12CCC(CC1)(CC2)C(O)=O
CCN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(=O)C12CCC(CC1)(CC2)C(O)=O
CCCN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(=O)C12CCC(CC1)(CC2)C(O)=O
CCN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(=O)[C@H]1CC[C@@](C)(CC1)C(O)=O |r,wU:40.48,wD:37.40,40.44,(3.51,-3.96,;1.97,-3.91,;1.24,-2.55,;-.3,-2.5,;-1.02,-1.15,;-2.52,-.78,;-2.63,.76,;-1.21,1.34,;-.21,.16,;1.33,.12,;2.14,1.42,;3.68,1.38,;4.41,.02,;3.59,-1.29,;2.06,-1.24,;5.94,-.03,;5.99,1.51,;7.48,-.08,;9.02,-.13,;7.44,-1.62,;7.53,1.46,;5.9,-1.57,;4.54,-2.3,;7.21,-2.38,;5.85,-3.11,;.46,1.55,;1.73,2.42,;.34,3.09,;-.41,2.82,;-1.94,2.71,;-2.81,3.98,;-2.14,5.37,;-3.01,6.64,;-.6,5.48,;.26,4.21,;-3.7,-1.77,;-3.42,-3.29,;-5.14,-1.25,;-5.42,.26,;-6.87,.79,;-8.04,-.21,;-9.08,.93,;-7.77,-1.72,;-6.32,-2.25,;-9.57,-.43,;-10.52,.78,;-10.14,-1.86,)|
CN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(=O)[C@@]1(F)CC[C@@H](CC1)C(O)=O |r,wU:40.47,36.40,wD:36.39,(1.62,-4.36,;.89,-3.01,;-.65,-2.96,;-1.37,-1.6,;-2.87,-1.24,;-2.98,.3,;-1.56,.88,;-.56,-.29,;.98,-.34,;1.79,.97,;3.33,.92,;4.05,-.44,;3.24,-1.75,;1.7,-1.7,;5.59,-.49,;5.64,1.05,;7.13,-.53,;8.67,-.58,;7.09,-2.07,;7.18,1.01,;5.55,-2.02,;4.19,-2.75,;6.85,-2.84,;5.5,-3.56,;.11,1.09,;1.38,1.96,;-.01,2.63,;-.76,2.37,;-2.29,2.25,;-3.16,3.53,;-2.49,4.91,;-3.36,6.19,;-.95,5.03,;-.09,3.75,;-4.05,-2.23,;-3.77,-3.75,;-5.5,-1.71,;-5.76,-3.23,;-4.73,-.37,;-5.5,.96,;-7.04,.95,;-7.81,-.38,;-7.03,-1.71,;-7.82,2.28,;-9.36,2.28,;-7.05,3.62,)|
CN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(=O)[C@H]1CC[C@@](C)(CC1)C(O)=O |r,wU:39.47,wD:36.39,39.43,(2.06,-4.15,;1.33,-2.79,;-.21,-2.74,;-.93,-1.38,;-2.43,-1.02,;-2.54,.52,;-1.12,1.1,;-.12,-.08,;1.42,-.12,;2.23,1.19,;3.77,1.14,;4.49,-.22,;3.68,-1.53,;2.14,-1.48,;6.03,-.27,;6.08,1.27,;7.57,-.32,;9.11,-.36,;7.52,-1.85,;7.62,1.22,;5.99,-1.81,;4.63,-2.53,;7.29,-2.62,;5.94,-3.35,;.55,1.31,;1.82,2.18,;.43,2.85,;-.32,2.58,;-1.86,2.47,;-2.72,3.75,;-2.05,5.13,;-2.92,6.41,;-.52,5.25,;.35,3.97,;-3.61,-2.01,;-3.33,-3.53,;-5.06,-1.49,;-5.33,.03,;-6.78,.55,;-7.95,-.45,;-8.99,.69,;-7.68,-1.96,;-6.23,-2.48,;-9.48,-.67,;-10.43,.54,;-10.05,-2.1,)|
CCCN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(=O)[C@@]1(F)CC[C@@H](CC1)C(O)=O |r,wU:42.49,38.42,wD:38.41,(3.75,-5.66,;3.02,-4.31,;1.48,-4.26,;.75,-2.9,;-.79,-2.85,;-1.51,-1.5,;-3.01,-1.13,;-3.12,.41,;-1.7,.99,;-.7,-.19,;.84,-.24,;1.65,1.07,;3.19,1.02,;3.92,-.33,;3.1,-1.64,;1.57,-1.59,;5.45,-.38,;5.5,1.16,;6.99,-.43,;8.53,-.48,;6.95,-1.97,;7.04,1.11,;5.41,-1.92,;4.05,-2.65,;6.72,-2.73,;5.36,-3.46,;-.03,1.2,;1.24,2.06,;-.15,2.73,;-.9,2.47,;-2.43,2.36,;-3.3,3.63,;-2.63,5.02,;-3.5,6.29,;-1.09,5.13,;-.23,3.86,;-4.19,-2.12,;-3.91,-3.64,;-5.63,-1.6,;-5.9,-3.12,;-4.87,-.27,;-5.64,1.06,;-7.18,1.06,;-7.95,-.28,;-7.17,-1.61,;-7.96,2.39,;-9.5,2.38,;-7.19,3.73,)|
CCN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(=O)[C@@]1(F)CC[C@@H](CC1)C(O)=O |r,wU:41.48,37.41,wD:37.40,(3.08,-4.17,;1.54,-4.12,;.81,-2.76,;-.72,-2.72,;-1.45,-1.36,;-2.95,-.99,;-3.06,.54,;-1.64,1.13,;-.64,-.05,;.9,-.1,;1.71,1.21,;3.25,1.16,;3.98,-.19,;3.17,-1.5,;1.63,-1.45,;5.52,-.24,;5.56,1.3,;7.05,-.29,;8.59,-.34,;7.01,-1.83,;7.1,1.25,;5.47,-1.78,;4.11,-2.51,;6.78,-2.59,;5.42,-3.32,;.03,1.34,;1.3,2.2,;-.08,2.87,;-.84,2.61,;-2.37,2.5,;-3.24,3.77,;-2.57,5.16,;-3.43,6.43,;-1.03,5.27,;-.17,4,;-4.12,-1.99,;-3.85,-3.5,;-5.57,-1.46,;-5.84,-2.98,;-4.81,-.13,;-5.58,1.2,;-7.12,1.2,;-7.89,-.14,;-7.11,-1.47,;-7.9,2.53,;-9.44,2.52,;-7.13,3.86,)|
CCCN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(=O)[C@H]1CC[C@@H](CC1)C(O)=O |r,wU:41.48,wD:38.41,(3.77,-5.44,;3.04,-4.09,;1.5,-4.04,;.78,-2.68,;-.76,-2.63,;-1.49,-1.28,;-2.99,-.91,;-3.1,.63,;-1.67,1.21,;-.68,.03,;.86,-.02,;1.67,1.29,;3.21,1.24,;3.94,-.11,;3.13,-1.42,;1.59,-1.37,;5.48,-.16,;5.52,1.38,;7.02,-.21,;8.55,-.26,;6.97,-1.75,;7.06,1.33,;5.43,-1.7,;4.07,-2.43,;6.74,-2.51,;5.38,-3.24,;-.01,1.42,;1.26,2.28,;-.12,2.95,;-.88,2.69,;-2.41,2.58,;-3.28,3.85,;-2.61,5.24,;-3.47,6.51,;-1.07,5.35,;-.21,4.08,;-4.16,-1.9,;-3.89,-3.42,;-5.61,-1.38,;-5.89,.13,;-7.33,.65,;-8.51,-.34,;-8.24,-1.86,;-6.79,-2.38,;-9.96,.18,;-11.14,-.81,;-10.23,1.7,)|
CCN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(=O)[C@@]1(C)CC[C@@H](CC1)C(O)=O |r,wU:41.48,37.41,wD:37.40,(3.08,-4.17,;1.54,-4.12,;.81,-2.76,;-.72,-2.72,;-1.45,-1.36,;-2.95,-.99,;-3.06,.54,;-1.64,1.13,;-.64,-.05,;.9,-.1,;1.71,1.21,;3.25,1.16,;3.98,-.19,;3.17,-1.5,;1.63,-1.45,;5.52,-.24,;5.56,1.3,;7.05,-.29,;8.59,-.34,;7.01,-1.83,;7.1,1.25,;5.47,-1.78,;4.11,-2.51,;6.78,-2.59,;5.42,-3.32,;.03,1.34,;1.3,2.2,;-.08,2.87,;-.84,2.61,;-2.37,2.5,;-3.24,3.77,;-2.57,5.16,;-3.43,6.43,;-1.03,5.27,;-.17,4,;-4.12,-1.99,;-3.85,-3.5,;-5.57,-1.46,;-5.84,-2.98,;-4.81,-.13,;-5.58,1.2,;-7.12,1.2,;-7.89,-.14,;-7.11,-1.47,;-7.9,2.53,;-9.44,2.52,;-7.13,3.86,)|
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CN1[C@@H](C[C@H](F)C1=O)C(=O)N1CCC2(C1CN(C)c1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1 |r|
CCN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1)C(=O)C1CCS(=O)(=O)CC1
CN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1)C(=O)C1CCS(=O)(=O)CC1
CN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(=O)C1CCS(=O)(=O)CC1
CCN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(=O)C1CCS(=O)(=O)CC1
CN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1)C(=O)C1CCS(=O)(=O)CC1
CCN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1)C(=O)[C@@]1(F)CC[C@@H](CC1)C(O)=O |r,wU:36.40,40.47,wD:36.39,(3.02,-4.52,;1.48,-4.47,;.75,-3.11,;-.79,-3.06,;-1.51,-1.71,;-3.01,-1.34,;-3.12,.2,;-1.7,.78,;-.7,-.4,;.84,-.45,;1.65,.86,;3.19,.81,;3.92,-.54,;3.1,-1.85,;1.57,-1.8,;5.46,-.59,;5.5,.95,;6.99,-.64,;8.53,-.69,;6.95,-2.18,;7.04,.9,;5.41,-2.13,;4.05,-2.86,;6.72,-2.94,;5.36,-3.67,;-.03,.99,;1.24,1.85,;-.14,2.52,;-.9,2.26,;-2.43,2.15,;-3.3,3.42,;-2.63,4.81,;-1.09,4.92,;-.23,3.65,;-4.18,-2.33,;-3.91,-3.85,;-5.63,-1.81,;-5.9,-3.33,;-4.87,-.48,;-5.64,.85,;-7.18,.85,;-7.95,-.49,;-7.17,-1.82,;-7.96,2.18,;-9.5,2.17,;-7.19,3.52,)|
CN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1)C(=O)[C@@]1(F)CC[C@@H](CC1)C(O)=O |r,wU:35.39,39.46,wD:35.38,(1.56,-4.71,;.83,-3.35,;-.71,-3.31,;-1.43,-1.95,;-2.93,-1.58,;-3.04,-.05,;-1.62,.54,;-.62,-.64,;.92,-.69,;1.73,.62,;3.27,.57,;3.99,-.78,;3.18,-2.09,;1.64,-2.05,;5.53,-.83,;5.58,.71,;7.07,-.88,;8.61,-.93,;7.03,-2.42,;7.12,.66,;5.49,-2.37,;4.13,-3.1,;6.8,-3.18,;5.44,-3.91,;.05,.75,;1.32,1.61,;-.07,2.28,;-.82,2.02,;-2.35,1.91,;-3.22,3.18,;-2.55,4.57,;-1.01,4.68,;-.15,3.41,;-4.11,-2.58,;-3.83,-4.09,;-5.55,-2.06,;-5.82,-3.57,;-4.79,-.72,;-5.56,.61,;-7.1,.61,;-7.87,-.73,;-7.09,-2.06,;-7.88,1.94,;-9.42,1.93,;-7.11,3.27,)|
CN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1)C(=O)[C@@]1(F)CC[C@@H](CC1)C(O)=O |r,wU:36.40,40.47,wD:36.39,(1.6,-4.98,;.87,-3.63,;-.67,-3.58,;-1.4,-2.22,;-2.89,-1.85,;-3,-.32,;-1.58,.26,;-.58,-.91,;.95,-.96,;1.77,.35,;3.3,.3,;4.03,-1.06,;3.22,-2.37,;1.68,-2.32,;5.57,-1.11,;5.62,.43,;7.11,-1.15,;8.65,-1.2,;7.06,-2.69,;7.16,.39,;5.52,-2.64,;4.17,-3.37,;6.83,-3.46,;5.48,-4.18,;.09,.47,;1.36,1.34,;-.03,2.01,;-.78,1.75,;-2.32,1.63,;-3.18,2.91,;-2.51,4.29,;-.98,4.41,;-.31,5.79,;-.11,3.13,;-4.07,-2.85,;-3.79,-4.36,;-5.52,-2.33,;-5.78,-3.85,;-4.75,-.99,;-5.53,.34,;-7.07,.33,;-7.83,-1,;-7.06,-2.33,;-7.84,1.67,;-9.38,1.66,;-7.08,3,)|
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CN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1)C(=O)[C@@]1(F)CC[C@@H](CC1)C(O)=O |r,wU:36.40,40.47,wD:36.39,(1.62,-4.36,;.89,-3.01,;-.65,-2.96,;-1.37,-1.6,;-2.87,-1.24,;-2.98,.3,;-1.56,.88,;-.56,-.29,;.98,-.34,;1.79,.97,;3.33,.92,;4.05,-.44,;3.24,-1.75,;1.7,-1.7,;5.59,-.49,;5.64,1.05,;7.13,-.53,;8.67,-.58,;7.09,-2.07,;7.18,1.01,;5.55,-2.02,;4.19,-2.75,;6.85,-2.84,;5.5,-3.56,;.11,1.09,;1.38,1.96,;-.01,2.63,;-.76,2.37,;-2.29,2.25,;-3.16,3.53,;-2.49,4.91,;-3.36,6.19,;-.95,5.03,;-.09,3.75,;-4.05,-2.23,;-3.77,-3.75,;-5.49,-1.71,;-5.76,-3.23,;-4.73,-.37,;-5.5,.96,;-7.04,.95,;-7.81,-.38,;-7.03,-1.71,;-7.82,2.28,;-9.36,2.28,;-7.05,3.62,)|
CCN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1)C(=O)[C@H]1CC[C@@H](CC1)C(O)=O |r,wU:40.47,wD:37.40,(3.11,-3.95,;1.57,-3.9,;.84,-2.54,;-.7,-2.5,;-1.43,-1.14,;-2.92,-.77,;-3.04,.76,;-1.61,1.35,;-.62,.17,;.92,.12,;1.73,1.43,;3.27,1.38,;4,.03,;3.19,-1.28,;1.65,-1.24,;5.54,-.02,;5.59,1.52,;7.08,-.07,;8.62,-.12,;7.03,-1.61,;7.13,1.47,;5.49,-1.56,;4.13,-2.29,;6.8,-2.37,;5.44,-3.1,;.05,1.56,;1.33,2.42,;-.06,3.09,;-.81,2.83,;-2.35,2.72,;-3.22,3.99,;-2.55,5.38,;-3.41,6.65,;-1.01,5.49,;-.14,4.22,;-4.1,-1.77,;-3.83,-3.28,;-5.55,-1.25,;-5.82,.27,;-7.27,.79,;-8.45,-.2,;-8.18,-1.72,;-6.73,-2.24,;-9.9,.32,;-11.07,-.67,;-10.17,1.83,)|
CCN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1)C(=O)C1CCS(=O)(=O)CC1
NC(=O)CN1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(N)=O |r,w:1.0|
CNC(=O)CN1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN(CC(=O)N3CCOCC3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
CCOC(=O)Cc1csc(NC(=O)CN2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)n1 |r|
OC(=O)Cc1csc(NC(=O)CN2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)n1 |r|
CN(C)C(=O)CN1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
NC(=O)CCN1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)CN1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)CCCCCN1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)CCCN1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)CCN1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)CCCCN1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CCOC(=O)C(F)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(O)cc1 |r,w:5.5|
CCNC(=O)CN1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN(C3CCN(Cc4ccccc4)C3=O)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN(C3CCNC3=O)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
OC(=O)c1ccc2C(CCc2c1)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CNC(=O)CN1CCC2(C1COc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
NC(=O)CN1CCC2(C1COc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN(CC(=O)NCC(F)(F)F)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN(CC(=O)NC3CC3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
CNC(=O)CCN1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CNC(=O)C(N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)c1ccccc1 |r|
CNC(=O)C(C)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CNC(=O)C(F)(F)CN1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CCC(N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(=O)NC |r|
OC(=O)c1ccc(CN2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)c(F)c1 |r|
OC(=O)c1ccc(CN2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)c(Cl)c1 |r|
OC(=O)c1cccc(CN2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)c1 |r|
COc1cc(ccc1CN1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(O)=O |r|
OC(=O)c1ccc(CN2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)c(c1)C(O)=O |r|
CC(=O)N1CCC(CN2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)CC1 |r|
Cn1ncnc1CN1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN(Cc3ncc[nH]3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
Cn1ccnc1CN1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN(Cc3nnn[nH]3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
OC(=O)c1ccc(CN2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN(Cc3ccc(C#N)c(F)c3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
OC(=O)c1ccccc1CN1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)c1ccc(CN2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)cc1F |r|
OC(=O)c1ccc(CN2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)cc1Cl |r|
OC(=O)CN1C2CCc3cc(I)ccc3C2(CC1=O)S(=O)(=O)c1ccc(F)cc1
CN1CCC2(C1CN(C)c1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)c1ccccc1 |r|
OC(=O)c1ccc(cc1)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)c1ccccn1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)c1ccccc1F |r|
OC(=O)c1cccc(c1)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)c1cccnc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)c1ccnnc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)c1cccnn1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)c1cncnc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)c1cnccn1 |r|
CS(=O)(=O)c1ccc(cc1)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)c1ncccn1 |r|
CS(=O)(=O)c1cccc(c1)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Cn1nnc(n1)-c1ccc(cc1)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C1(CC1)c1ccc(cc1)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN(C)S(=O)(=O)c1cccc(c1)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN(C#N)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
CC(C)(C)OC(=O)N1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(=O)[C@H]1CC[C@@H](CC1)C(O)=O |r,wU:45.52,wD:42.45,(2.32,-4.99,;3.67,-4.27,;5.03,-3.54,;4.4,-5.62,;2.94,-2.91,;1.41,-2.86,;.59,-4.17,;.68,-1.5,;-.86,-1.46,;-1.59,-.1,;-3.09,.27,;-3.2,1.8,;-1.77,2.39,;-.78,1.21,;.76,1.16,;1.57,2.47,;3.11,2.42,;3.84,1.07,;3.03,-.24,;1.49,-.2,;5.38,1.02,;5.43,2.56,;6.92,.97,;8.46,.92,;6.87,-.57,;6.97,2.51,;5.33,-.52,;3.97,-1.25,;6.64,-1.33,;5.28,-2.06,;-.11,2.6,;1.16,3.46,;-.22,4.13,;-.97,3.87,;-2.51,3.76,;-3.38,5.03,;-2.71,6.42,;-3.57,7.69,;-1.17,6.53,;-.3,5.26,;-4.26,-.73,;-3.99,-2.24,;-5.71,-.21,;-5.98,1.31,;-7.43,1.83,;-8.61,.84,;-8.34,-.68,;-6.89,-1.2,;-10.06,1.36,;-11.23,.36,;-10.33,2.87,)|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CCC2(C1CCc1cc(CC(F)(F)F)ccc21)S(=O)(=O)c1ccc(Cl)cc1 |r,wU:6.9,wD:3.2,(8.24,-3.38,;6.75,-3.78,;6.35,-5.27,;5.66,-2.69,;6.06,-1.2,;4.97,-.11,;3.48,-.51,;3.09,-2,;4.17,-3.09,;2.4,.58,;2.79,2.07,;.91,.18,;.28,-1.23,;-1.25,-1.07,;-1.57,.44,;-.24,1.21,;-.24,2.75,;-1.57,3.52,;-2.9,2.75,;-4.24,3.52,;-5.57,2.75,;-6.9,3.52,;-8.24,2.75,;-9.57,1.98,;-9.01,4.08,;-7.47,1.42,;-5.57,1.21,;-4.24,.44,;-2.9,1.21,;-2.66,-.65,;-4.15,-1.05,;-3.06,-2.14,;-2.26,-2.14,;-3.35,-3.23,;-2.95,-4.71,;-1.46,-5.11,;-1.06,-6.6,;-.37,-4.02,;-.77,-2.54,)|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1 |r,wU:6.9,wD:3.2,(8.91,-3.76,;7.42,-4.16,;7.02,-5.65,;6.33,-3.07,;6.73,-1.59,;5.64,-.5,;4.15,-.9,;3.75,-2.38,;4.84,-3.47,;3.06,.19,;3.46,1.68,;1.57,-.21,;.95,-1.61,;-.58,-1.45,;-.9,.05,;.43,.82,;.43,2.36,;-.9,3.13,;-2.24,2.36,;-3.57,3.13,;-4.9,2.36,;-4.9,.82,;-3.57,.05,;-2.24,.82,;-6.24,3.13,;-6.24,1.59,;-6.24,4.67,;-7.57,5.44,;-4.9,5.44,;-4.9,3.9,;-7.57,2.36,;-8.91,3.13,;-7.57,.82,;-8.91,1.59,;-1.99,-1.03,;-3.48,-1.43,;-2.39,-2.52,;-1.59,-2.52,;-2.68,-3.61,;-2.28,-5.1,;-.8,-5.5,;-.4,-6.98,;.29,-4.41,;-.11,-2.92,)|
OC(=O)C12CCC(CC1)(CC2)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(cc1)C#N
CN(C)c1ccc(cc1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C12CCC(CC1)(CC2)C(O)=O
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(cc1)-c1cnoc1 |r,wU:3.2,wD:6.9,(-10.46,-1.47,;-9.29,-.47,;-9.56,1.04,;-7.84,-.99,;-6.66,0,;-5.21,-.52,;-4.94,-2.04,;-6.12,-3.03,;-7.57,-2.51,;-3.49,-2.56,;-3.22,-4.07,;-2.31,-1.56,;-2.43,-.03,;-1,.55,;-.01,-.62,;-.82,-1.93,;-.09,-3.29,;1.45,-3.34,;2.26,-2.03,;3.8,-2.07,;4.61,-.77,;3.88,.59,;2.34,.64,;1.53,-.67,;6.15,-.81,;6.2,.73,;7.69,-.86,;7.64,-2.4,;7.74,.68,;9.23,-.91,;6.1,-2.35,;4.74,-3.08,;7.41,-3.16,;6.05,-3.89,;.66,.77,;1.94,1.63,;.55,2.3,;-.2,2.04,;-1.74,1.93,;-2.61,3.2,;-1.94,4.59,;-.4,4.7,;.47,3.43,;-2.8,5.86,;-2.28,7.31,;-3.5,8.25,;-4.77,7.39,;-4.34,5.91,)|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(cc1)-c1cn[nH]c1 |r,wU:3.2,wD:6.9,(-10.57,-1.37,;-9.39,-.37,;-9.66,1.14,;-7.94,-.9,;-6.77,.1,;-5.32,-.42,;-5.04,-1.94,;-6.22,-2.93,;-7.67,-2.41,;-3.59,-2.46,;-3.32,-3.98,;-2.42,-1.47,;-2.53,.07,;-1.11,.65,;-.11,-.52,;-.92,-1.83,;-.19,-3.19,;1.34,-3.24,;2.16,-1.93,;3.7,-1.98,;4.51,-.67,;3.78,.69,;2.24,.74,;1.43,-.57,;6.05,-.72,;6.09,.82,;7.58,-.76,;7.54,-2.3,;7.63,.78,;9.12,-.81,;6,-2.26,;4.64,-2.98,;7.31,-3.07,;5.95,-3.79,;.56,.86,;1.83,1.73,;.45,2.4,;-.31,2.14,;-1.84,2.02,;-2.71,3.3,;-2.04,4.68,;-.5,4.8,;.36,3.52,;-2.9,5.96,;-2.38,7.41,;-3.6,8.35,;-4.87,7.48,;-4.44,6.01,)|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(c1)C1CC1 |r,wU:3.2,wD:6.9,(-10.9,-1.21,;-9.73,-.22,;-10,1.3,;-8.28,-.74,;-7.1,.25,;-5.65,-.27,;-5.38,-1.78,;-6.55,-2.78,;-8,-2.26,;-3.93,-2.3,;-3.66,-3.82,;-2.75,-1.31,;-2.87,.23,;-1.44,.81,;-.45,-.37,;-1.26,-1.68,;-.53,-3.03,;1.01,-3.08,;1.82,-1.77,;3.36,-1.82,;4.17,-.51,;3.44,.84,;1.9,.89,;1.09,-.42,;5.71,-.56,;5.76,.98,;7.25,-.61,;8.79,-.66,;7.2,-2.15,;7.3,.93,;5.66,-2.1,;4.31,-2.83,;6.97,-2.91,;5.61,-3.64,;.22,1.02,;1.5,1.88,;.11,2.55,;-.64,2.29,;.03,3.68,;-.84,4.95,;-2.37,4.84,;-3.04,3.45,;-2.18,2.18,;-4.58,3.34,;-5.85,2.47,;-5.97,4.01,)|
CC(C)c1cccc(c1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)[C@H]1CC[C@@H](CC1)C(O)=O |r,wU:40.47,wD:37.40,(-5.45,4.63,;-4.59,3.36,;-5.26,1.97,;-3.05,3.47,;-2.38,4.86,;-.85,4.97,;.02,3.7,;-.65,2.31,;-2.19,2.2,;.22,1.04,;1.49,1.9,;.1,2.57,;-.45,-.35,;-1.45,.83,;-2.87,.24,;-2.76,-1.29,;-1.27,-1.66,;-.54,-3.02,;1,-3.07,;1.81,-1.76,;3.35,-1.8,;4.16,-.5,;3.44,.86,;1.9,.91,;1.09,-.4,;5.7,-.54,;5.75,1,;7.24,-.59,;8.78,-.64,;7.19,-2.13,;7.29,.95,;5.65,-2.08,;4.3,-2.81,;6.96,-2.89,;5.61,-3.62,;-3.94,-2.29,;-3.66,-3.8,;-5.39,-1.77,;-5.66,-.25,;-7.11,.27,;-8.28,-.72,;-8.01,-2.24,;-6.56,-2.76,;-9.73,-.2,;-10.01,1.31,;-10.91,-1.2,)|
CC(C)(C)c1cccc(c1)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)[C@H]1CC[C@@H](CC1)C(O)=O |r,wU:38.41,wD:41.48,(-6.13,3.03,;-4.59,3.14,;-4.71,4.68,;-4.48,1.61,;-3.06,3.26,;-2.39,4.64,;-.85,4.76,;.01,3.48,;-.66,2.1,;-2.19,1.98,;.21,.82,;1.48,1.69,;.1,2.36,;-.46,-.56,;-1.46,.61,;-2.88,.03,;-2.77,-1.5,;-1.27,-1.87,;-.54,-3.23,;1,-3.28,;1.81,-1.97,;3.35,-2.02,;4.16,-.71,;3.43,.65,;1.89,.7,;1.08,-.61,;5.7,-.76,;5.74,.78,;7.24,-.8,;8.77,-.85,;7.19,-2.34,;7.28,.74,;5.65,-2.29,;4.29,-3.02,;6.96,-3.11,;5.6,-3.83,;-3.94,-2.5,;-3.67,-4.01,;-5.39,-1.98,;-6.57,-2.97,;-8.02,-2.45,;-8.29,-.93,;-7.11,.06,;-5.67,-.46,;-9.74,-.41,;-10.01,1.1,;-10.92,-1.41,)|
C[C@@]1(CC[C@@H](CC1)C(N)=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:16.17,4.7,1.0,wD:1.10,15.38,(-5.89,-3.47,;-5.63,-1.96,;-4.86,-.62,;-5.64,.71,;-7.18,.71,;-7.94,-.63,;-7.17,-1.96,;-7.95,2.04,;-9.49,2.03,;-7.19,3.37,;-4.18,-2.48,;-3.9,-3.99,;-3,-1.48,;-3.11,.05,;-1.69,.64,;-.69,-.54,;-1.51,-1.85,;-.78,-3.21,;.76,-3.25,;1.57,-1.95,;3.11,-1.99,;3.92,-.69,;3.2,.67,;1.66,.72,;.85,-.59,;5.46,-.73,;5.51,.81,;7,-.78,;8.54,-.83,;6.95,-2.32,;7.05,.76,;5.41,-2.27,;4.06,-3,;6.72,-3.08,;5.37,-3.81,;-.02,.85,;1.25,1.71,;-.14,2.38,;-.89,2.12,;-2.43,2.01,;-3.29,3.28,;-2.62,4.67,;-3.49,5.94,;-1.09,4.78,;-.22,3.51,)|
NC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:15.16,3.2,wD:14.37,6.9,(-10.91,-1.16,;-9.74,-.16,;-10.01,1.35,;-8.29,-.68,;-7.11,.31,;-5.66,-.21,;-5.39,-1.73,;-6.57,-2.72,;-8.01,-2.2,;-3.94,-2.25,;-3.67,-3.76,;-2.76,-1.25,;-2.88,.28,;-1.45,.87,;-.46,-.31,;-1.27,-1.62,;-.54,-2.98,;1,-3.02,;1.81,-1.72,;3.35,-1.76,;4.16,-.46,;3.43,.9,;1.89,.95,;1.08,-.36,;5.7,-.5,;5.75,1.04,;7.24,-.55,;8.78,-.6,;7.19,-2.09,;7.29,.99,;5.65,-2.04,;4.29,-2.77,;6.96,-2.85,;5.6,-3.58,;.21,1.08,;1.49,1.94,;.1,2.61,;-.65,2.35,;-2.19,2.24,;-3.05,3.51,;-2.38,4.9,;-3.25,6.17,;-.85,5.01,;.02,3.74,)|
NC(=O)C12CCC(CC1)(CC2)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)CNC(=O)CN1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1[C@H]2CC[C@@H]1C[C@H](C2)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,THB:11:9:3:6.5|
CC1(CCN(CC1)S(C)(=O)=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CS(=O)(=O)N1CC[C@H](CC(=O)N2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)C1 |r|
CC(=O)N1CC[C@H](CC(=O)N2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)C1 |r|
CS(=O)(=O)N1CC[C@@H](CC(=O)N2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)C1 |r|
CC(=O)N1CC[C@@H](CC(=O)N2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)C1 |r|
CNC(=O)N1CCC(O)(CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCC(O)(CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CS(=O)(=O)N1CCC(O)(CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CNC(=O)N1CCC(CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCN(CC1)C#N |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCN(CC1)C1COC1 |r|
OC1(CCN(CC1)C1COC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
FC(F)(F)C(F)(c1ccc2c(CCC3N(CCC23S(=O)(=O)c2ccc(Cl)cc2)C(=O)C2CCN(CC2)C2COC2)c1)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)[C@H]1C[C@@H]2CC[C@H](C1)N2C1COC1 |r,TLB:33:35:42:39.38|
C[C@H]1CN(CCN1CC(O)=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(CO)(CO)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC1(COP(O)(=O)OC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC1(COP(N)(=O)OC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:1.0|
CC1(COP(C)(=O)OC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)c1ccc(cc1F)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(C(O)=O)c1ccc(cc1Cl)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:1.0|
OC(C(O)=O)c1ccc(cc1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:1.0|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1(F)CCS(=O)(=O)CC1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1(F)CCOCC1 |r|
C[C@H]1CC(CC[C@H]1C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1)C(C)=O |r|
C[C@H]1CC(CC[C@H]1C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(O)=O |r|
C[C@@H]1CC(CC[C@H]1C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(O)=O |r|
C[C@H]1CC(O)CC[C@H]1C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1 |r,w:3.3|
C[C@H]1CC(C)(O)CC[C@H]1C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1 |r|
C[C@H]1CC(CC[C@H]1C(O)=O)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1cccc(F)c1 |r|
C[C@H]1CC(CC[C@H]1C(O)=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@@H]1CC(CC[C@H]1C(O)=O)C(=O)N1CCC2(C1COc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(c(Cl)cc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:15.16,3.2,wD:6.9,14.38,(-10.29,1.31,;-10.01,-.21,;-11.19,-1.2,;-8.56,-.73,;-7.39,.27,;-5.94,-.25,;-5.67,-1.77,;-6.84,-2.76,;-8.29,-2.24,;-4.22,-2.29,;-3.94,-3.81,;-3.04,-1.3,;-3.15,.24,;-1.73,.82,;-.73,-.36,;-1.54,-1.66,;-.82,-3.02,;.72,-3.07,;1.53,-1.76,;3.07,-1.81,;3.88,-.5,;3.16,.86,;3.97,2.17,;1.62,.91,;.81,-.4,;5.42,-.55,;5.47,.99,;6.96,-.6,;8.5,-.64,;6.91,-2.13,;7.01,.94,;5.38,-2.09,;4.02,-2.81,;6.68,-2.9,;5.33,-3.63,;-.06,1.03,;1.21,1.9,;-.18,2.57,;-.93,2.31,;-2.46,2.19,;-3.33,3.47,;-2.66,4.85,;-3.53,6.13,;-1.12,4.97,;-.26,3.69,)|
Cc1cc2c(CC[C@H]3N(CC[C@@]23S(=O)(=O)c2ccc(F)cc2)C(=O)[C@H]2CC[C@@H](CC2)C(O)=O)cc1C(F)(C(F)(F)F)C(F)(F)F |r,wU:7.7,27.33,wD:24.26,11.13,(3.97,2.17,;3.16,.86,;1.62,.91,;.81,-.4,;1.53,-1.76,;.72,-3.07,;-.82,-3.02,;-1.54,-1.66,;-3.04,-1.3,;-3.15,.24,;-1.73,.82,;-.73,-.36,;-.06,1.03,;1.21,1.9,;-.18,2.57,;-.93,2.31,;-2.46,2.19,;-3.33,3.47,;-2.66,4.85,;-3.53,6.13,;-1.12,4.97,;-.26,3.69,;-4.22,-2.29,;-3.94,-3.81,;-5.67,-1.77,;-5.94,-.25,;-7.39,.27,;-8.56,-.73,;-8.29,-2.24,;-6.84,-2.76,;-10.01,-.21,;-10.29,1.31,;-11.19,-1.2,;3.07,-1.81,;3.88,-.5,;5.42,-.55,;5.47,.99,;6.96,-.6,;8.5,-.64,;6.91,-2.13,;7.01,.94,;5.38,-2.09,;4.02,-2.81,;6.68,-2.9,;5.33,-3.63,)|
Cc1cc2c(CC[C@H]3N(CC[C@@]23S(=O)(=O)c2ccc(F)cc2)C(=O)[C@H]2CC[C@@H](CC2)C(O)=O)c(C)c1C(F)(C(F)(F)F)C(F)(F)F |r,wU:7.7,24.26,wD:27.33,11.13,(3.77,2.37,;2.96,1.06,;1.42,1.11,;.61,-.2,;1.34,-1.56,;.53,-2.87,;-1.01,-2.82,;-1.74,-1.46,;-3.23,-1.1,;-3.35,.44,;-1.92,1.02,;-.93,-.15,;-.26,1.23,;-.14,-.3,;1.13,.56,;-1.12,2.51,;-2.66,2.39,;-3.52,3.67,;-2.85,5.05,;-3.72,6.33,;-1.32,5.17,;-.45,3.89,;-4.41,-2.09,;-4.14,-3.61,;-5.86,-1.57,;-7.03,-2.56,;-8.48,-2.04,;-8.76,-.53,;-7.58,.47,;-6.13,-.05,;-10.21,-.01,;-10.48,1.51,;-11.38,-1,;2.88,-1.61,;3.61,-2.96,;3.69,-.3,;5.23,-.35,;5.28,1.19,;6.77,-.39,;8.31,-.44,;6.72,-1.93,;6.82,1.14,;5.18,-1.89,;3.83,-2.61,;6.49,-2.7,;5.13,-3.43,)|
COC(=O)C1(CCS(=O)(=O)CC1)NC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
FC(F)(F)C(F)(c1ccc2c(CC[C@@H]3N(CC[C@]23S(=O)(=O)c2ccccc2)C(=O)CN2CCS(=O)(=O)CC2)c1)C(F)(F)F |r|
CCN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1)C(=O)C1(O)CCS(=O)(=O)CC1
FC(F)(F)C(F)(c1ccc2c(CC[C@H]3N(CC[C@@]23S(=O)(=O)c2ccccc2)C(=O)CN2CCS(=O)(=O)CC2)c1)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1ccc2nncn2c1 |r|
FC(F)(F)C(F)(c1ccc2c(CCC3N(CCC23S(=O)(=O)c2ccc(Cl)cc2)C(=O)c2ccc3nncn3c2)c1)C(F)(F)F
CC(=O)N1CCN(CC(=O)N2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)CC1 |r|
OC1(CCS(=O)(=O)CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)c(F)c1
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)c(F)c1 |r,wU:6.9,wD:3.2,(-9.97,1.08,;-9.7,-.43,;-10.88,-1.43,;-8.25,-.95,;-7.98,-2.47,;-6.53,-2.99,;-5.35,-2,;-5.63,-.48,;-7.08,.04,;-3.91,-2.52,;-3.63,-4.03,;-2.73,-1.52,;-2.84,.01,;-1.42,.59,;-.42,-.58,;-1.23,-1.89,;-.51,-3.25,;1.03,-3.3,;1.85,-1.99,;3.38,-2.03,;4.2,-.73,;3.47,.63,;1.93,.68,;1.12,-.63,;5.73,-.77,;5.78,.77,;7.27,-.82,;8.81,-.87,;7.23,-2.36,;7.32,.72,;5.69,-2.31,;4.33,-3.04,;7,-3.12,;5.64,-3.85,;.25,.81,;1.52,1.67,;.13,2.34,;-.62,2.08,;-2.15,1.97,;-3.02,3.24,;-2.35,4.63,;-3.22,5.9,;-.81,4.74,;-.14,6.13,;.05,3.47,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)c1noc(=O)[nH]1 |r|
CN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1)C(=O)C1CCS(=O)(=O)CC1
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N(C1CC1)C1CCOCC1 |r|
CN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1)C(=O)C1(O)CCS(=O)(=O)CC1
FC(F)(F)C(F)(c1ccc2c(CCC3N(CCC23S(=O)(=O)c2ccc(Cl)cc2)C(=O)c2noc(=O)[nH]2)c1)C(F)(F)F
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1CCOCC1 |r|
C[C@H]1C[C@H](CC[C@@H]1C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(O)=O |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)[C@@H]1CCC(=O)N1CCC#N |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NC1CCOCC11NC(=O)NC1=O |r,w:46.51,41.46|
OC(=O)C1(CCS(=O)(=O)CC1)NC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
F[C@H]1C[C@H](N(CCC#N)C1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C12CCC(CC1)(CC2)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)c(Cl)c1
CC(C)C(N(C1CCS(=O)(=O)C1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(O)=O |r,w:5.4,3.2,3.51|
CN1[C@@H](CCCC1=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
F[C@H]1C[C@H](N(CC#N)C1)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N[C@@H]1CS(=O)(=O)C[C@H]1NC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1Cl)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCS(=O)(=O)CC1
OC1(CCS(=O)(=O)CC1)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)c(Cl)c1
OC(=O)C12CCC(CC1)(CC2)C(=O)N1CCC2(C1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1
CS(=O)(=O)N1CCN(CC(=O)N2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)CC1 |r|
CC(=O)NC1CS(=O)(=O)CCC1NC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(O)CN1[C@@H](C[C@H](F)C1=O)C(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN(CC(=O)N1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C1CCS(=O)(=O)C1 |r,w:1.41|
Cc1ccc(cc1F)S(=O)(=O)C12CCN(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)[C@H]1CC[C@@H](CC1)C(O)=O |r,wU:39.46,wD:36.39,(-3.22,5.9,;-2.35,4.63,;-3.02,3.24,;-2.15,1.97,;-.62,2.08,;.05,3.47,;-.81,4.74,;-.14,6.13,;.25,.81,;1.52,1.67,;.13,2.34,;-.42,-.58,;-1.42,.59,;-2.84,.01,;-2.73,-1.52,;-1.23,-1.89,;-.51,-3.25,;1.03,-3.3,;1.85,-1.99,;3.38,-2.03,;4.2,-.73,;3.47,.63,;1.93,.68,;1.12,-.63,;5.73,-.77,;5.78,.77,;7.27,-.82,;8.81,-.87,;7.23,-2.36,;7.32,.72,;5.69,-2.31,;4.33,-3.04,;7,-3.12,;5.64,-3.85,;-3.91,-2.52,;-3.63,-4.03,;-5.35,-2,;-5.63,-.48,;-7.08,.04,;-8.25,-.95,;-7.98,-2.47,;-6.53,-2.99,;-9.7,-.43,;-10.88,-1.43,;-9.97,1.08,)|
CN1CC2N(CCC2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1)C(=O)C12CCC(CC1)(CC2)C(O)=O
FC(F)(F)C(F)(c1ccc2c(CCC3N(CCC23S(=O)(=O)c2ccc(Cl)cc2)C(=O)[C@@H]2CCC(=O)N2CCC#N)c1)C(F)(F)F |r|
CN1[C@@H](C[C@H](O)C1=O)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1 |r|
CO[C@H]1C[C@H](N(C)C1=O)C(=O)N1CCC2(C1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CCN([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)C1CCN(CC1)C=O |r|
CC1(C)[C@H]2CC[C@]1(NC(=O)OCc1ccccc1)C(=N)\C2=C/C(=N)c1c(F)cccc1F |r|
CC1(C)[C@@H]2CC[C@@]1(NC(=O)OCc1ccccc1)c1nnc(cc21)-c1c(F)cccc1F |r|
CN(C(=O)OCc1ccccc1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r|
CC(=O)N(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)c1nnc(C)o1 |r|
CN(C(=O)OCc1ccccc1)[C@]12CC[C@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cc(C)no1 |r|
Cc1cc(no1)C(=O)N(CCO)C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r|
Cc1cc(no1)C(=O)N(CCF)C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1coc(C)n1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccnc(O)n1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1nnc(C)o1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cccc(O)n1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cnc(O)cn1 |r|
CCN(C(=O)OCc1ccccc1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r|
CC1(C)[C@H]2CC[C@]1(CN(CCC#N)C(=O)c1cccc(=O)[nH]1)c1nnc(cc21)-c1c(F)cccc1F |r,TLB:26:27:4.5:1,23:22:4.5:1|
CC1(C)[C@H]2CC[C@]1(CN(CCC#N)C(=O)c1c[nH]c(=O)cn1)c1nnc(cc21)-c1c(F)cccc1F |r|
CC1(C)[C@H]2CC[C@]1(CN(CC(F)F)C(=O)c1cccc(O)n1)c1nnc(cc21)-c1c(F)cccc1F |r|
CC1(C)[C@H]2CC[C@]1(CN(CC(F)F)C(=O)c1cnc(O)cn1)c1nnc(cc21)-c1c(F)cccc1F |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(O)nc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccnc(O)c1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cnc(O)nc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(O)nn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cnc(C)cn1 |r|
CCN(C[C@]12CC[C@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cnc(O)cn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cccnc1O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cncnc1O |r|
CC1(C)[C@@H]2CC[C@@]1(CN(CC(F)F)C(=O)c1c[nH]c(=O)cn1)c1nnc(cc21)-c1c(F)cccc1F |r|
CN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(=O)[nH]n1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cnn2cccnc12 |r|
CC1(C)[C@H]2CC[C@]1(CN(C1CC1)C(=O)c1ccc(=O)[nH]n1)c1nnc(cc21)-c1c(F)cccc1F |r|
CC1(CC1)N(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(=O)[nH]n1 |r|
CC1(C)[C@H]2CC[C@]1(CNC(=O)c1ccc(=O)[nH]n1)c1nnc(cc21)-c1c(F)cccc1F |r|
CC1(C)[C@H]2CC[C@]1(CN(C1CC1)C(=O)c1c[nH]c(=O)cn1)c1nnc(cc21)-c1c(F)cccc1F |r|
CC1(CC1)N(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1c[nH]c(=O)cn1 |r|
CN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1c[nH]c(=O)cn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cn[nH]c(=O)c1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)Cc1cnccn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cnc(NS(C)(=O)=O)cn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cnc(N)cn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1ccccc1F)C2(C)C)C(=O)c1c[nH]c(=O)cn1 |r|
CC1(C)[C@H]2CC[C@]1(CN(CC(F)F)C(=O)c1ccc(=O)[nH]n1)c1nnc(cc21)-c1c(F)cccc1F |r|
CC1(C)[C@H]2CC[C@]1(CN(CC(F)F)C(=O)c1ccc(=O)[nH]c1)c1nnc(cc21)-c1c(F)cccc1F |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1nnc[nH]1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1nnc(C)[nH]1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cnn[nH]1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1n[nH]c(=O)[nH]1 |r,THB:9:8:6.5:22,12:13:6.5:22|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cc(=O)[nH][nH]1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1c[nH]c(=O)[nH]1 |r,THB:9:8:6.5:22,12:13:6.5:22|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)C1(O)COC1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)C1CCCN1C(N)=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)Cc1nnn[nH]1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)C1(CC1)C(N)=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)CN1CCNC(=O)C1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)CCC1NC(=O)NC1=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)Cn1ccc(=O)[nH]c1=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)CC1NC(=O)c2ccccc12 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)CN1CCN(CC1)C(C)=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)CC1CCS(=O)(=O)C1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)C1CCCN(C1)C(N)=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)CC1Oc2ccccc2NC1=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)C1CCCN1S(C)(=O)=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(NC(C)=O)cc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc2[nH]c(C)nc2c1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(cc1)-c1ncccn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(NC(N)=O)cc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cccc(c1)-n1cnnc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(cc1)-c1nnn(C)n1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(cc1)S(=O)(=O)NC |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(Cn2nnnc2C)cc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(cc1)N1CCOCC1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(NS(C)(=O)=O)cc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc2[nH]nnc2c1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccncc1NC(C)=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(nc1)C#N |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cnc2[nH]cnc2c1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1c[nH]nc1-n1cnnn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1n[nH]c2cc(F)ccc12 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1c[nH]cn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cncnc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ncccn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(OCc2noc(C)n2)cc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cn[nH]c1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cc[nH]n1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cc(C)[nH]n1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cnccn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccnnc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cn(C)cn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cnn(C)c1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1nc2ccccc2c(=O)[nH]1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)C1CN(C1)C(C)=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)C1CN(C1)C(=O)C(C)C |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)C1CN(C1)S(C)(=O)=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1nn(C)cc1-c1ccno1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cc(n(C)n1)C(F)(F)F |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)CCN1CCN(CC1)C(N)=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cc(on1)-c1cn(C)nc1C |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cnc(nc1)-c1ccccc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(cc1)-c1noc(n1)C1CC1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cnn(c1)C1CCN(C1)C(C)=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cnn(c1)C1CCN(C)C1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)C1CN(CCN1C)C(C)=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)C1CN(C)CCN1C(C)=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)C1CN(CCO1)C(C)=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)CN1C(=O)CNC1=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(cc1)-c1ncn[nH]1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cocn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cn[nH]c1-c1ccccc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)C1CCN(CC1)C(N)=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)C1CCS(=O)(=O)C1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1c(C)n[nH]c1C |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(nc1)-n1ccnc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cc(CO)on1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1nc(N)n[nH]1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1nnc(CO)[nH]1 |r,THB:12:13:6.5:22,9:8:6.5:22|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1cnn(CC)c1C |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1c(C)noc1C |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1c(C)n[nH]c1C |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1ccc(cc1)C#N |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1c(C)nn(C)c1C |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1ccc(F)cc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)Cc1cccc(F)c1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1ccc(F)cc1F |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1cccc(F)c1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1ccccc1F |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1cnc(C)n1C |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1cn(C)c(C)n1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1cnn(CC)c1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)C1CC1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1ncn[nH]1 |r,THB:9:8:6.5:22,12:13:6.5:22|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1ccccc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1cn(C)cn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1cccnc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)Cc1ccc(F)cc1F |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1ccc(NC(C)=O)cc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1cn(nc1C)C(F)F |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1ccc(OC(F)F)cc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1ccc(NC(N)=O)cc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1c(F)cccc1F |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1cc(F)cc(F)c1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1ccc(F)c(F)c1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1ccc(NC(=O)NC)cc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1ccc(cc1)S(C)(=O)=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1ccc(cc1)S(=O)(=O)N(C)C |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)Cc1ccncc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)Cc1ccccn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1cc(F)ccc1F |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1ccccc1C#N |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1ccccc1S(C)(=O)=O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)Cc1cc(F)ccc1F |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1cccc(c1)C#N |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)c1cnoc1C |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)Cn1ccnn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)Cn1ccnc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)Cc1cncc(=O)[nH]1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cc(O)ccn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)Cc1ccon1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cn(C)nn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)Cc1ccccc1F |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)Cc1ccccc1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)Cn1cncn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(=O)n(C)n1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)Cc1n[nH]c(=O)[nH]1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)Cc1ccc(=O)[nH]n1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cnc(cn1)C(=O)OC |r|
CCN(C[C@@]12CC[C@@H](\C(=C\C(=N)c3c(F)cccc3F)C1=N)C2(C)C)C(=O)c1ncco1 |r|
CCN(C[C@@]12CC[C@@H](\C(=C\C(=N)c3c(F)cccc3F)C1=N)C2(C)C)C(=O)c1ncoc1C |r|
CCN(C[C@@]12CC[C@@H](\C(=C\C(=N)c3c(F)cccc3F)C1=N)C2(C)C)C(=O)c1cnc(C)o1 |r|
CCN(C[C@@]12CC[C@@H](\C(=C\C(=N)c3c(F)cccc3F)C1=N)C2(C)C)C(=O)c1coc(N)n1 |r|
CCN(C[C@@]12CC[C@@H](\C(=C\C(=N)c3c(F)cccc3F)C1=N)C2(C)C)C(=O)c1nc(C)c[nH]1 |r|
CCN(C[C@@]12CC[C@@H](\C(=C\C(=N)c3c(F)cccc3F)C1=N)C2(C)C)C(=O)CN1CCS(=O)(=O)CC1 |r|
CCN(C[C@@]12CC[C@@H](\C(=C\C(=N)c3c(F)cccc3F)C1=N)C2(C)C)C(=O)c1ncc(C)o1 |r|
CCN(C[C@@]12CC[C@@H](\C(=C\C(=N)c3c(F)cccc3F)C1=N)C2(C)C)C(=O)c1nc(C)co1 |r|
CCN(C[C@@]12CC[C@@H](\C(=C\C(=N)c3c(F)cccc3F)C1=N)C2(C)C)C(=O)c1coc(CS(C)(=O)=O)n1 |r|
CCN(C[C@@]12CC[C@@H](\C(=C\C(=N)c3c(F)cccc3F)C1=N)C2(C)C)C(=O)C(=N)\C=C/C(N)=N |r|
CCN(C[C@@]12CC[C@@H](\C(=C\C(=N)c3c(F)cccc3F)C1=N)C2(C)C)C(=O)c1nc(C)oc1C |r|
CCN(C[C@@]12CC[C@@H](\C(=C\C(=N)c3c(F)cccc3F)C1=N)C2(C)C)C(=O)c1coc(N)n1 |r,THB:21:20:6.5:22,9:8:6.5:22|
CCN(C[C@@]12CC[C@@H](\C(=C\C(=N)c3c(F)cccc3F)C1=N)C2(C)C)C(=O)c1nocc1C |r|
CCN(C[C@@]12CC[C@@H](\C(=C\C(=N)c3c(F)cccc3F)C1=N)C2(C)C)C(=O)C(=N)\C=C/C(=N)CC#N |r|
CCN(C[C@@]12CC[C@@H](\C(=C\C(=N)c3c(F)cccc3F)C1=N)C2(C)C)C(=O)CN1CCC(O)CC1 |r|
CCN(C[C@@]12CC[C@@H](\C(=C\C(=N)c3c(F)cccc3F)C1=N)C2(C)C)C(=O)c1cc(on1)C(C)(C)O |r|
CC1(C)[C@H]2CC[C@]1(CN(CC(F)F)C(=O)c1coc(CS(C)(=O)=O)n1)C(=N)\C2=C/C(=N)c1c(F)cccc1F |r|
CC(C)N(C[C@@]12CC[C@@H](\C(=C\C(=N)c3c(F)cccc3F)C1=N)C2(C)C)C(=O)c1coc(CS(C)(=O)=O)n1 |r|
CC1(C)[C@H]2CC[C@]1(CN(CC1CC1)C(=O)c1coc(CS(C)(=O)=O)n1)C(=N)\C2=C/C(=N)c1c(F)cccc1F |r|
CC1(C)[C@H]2CC[C@]1(CN(C1CC1)C(=O)c1coc(CS(C)(=O)=O)n1)C(=N)\C2=C/C(=N)c1c(F)cccc1F |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cnc(C)o1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1nc(C)co1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1coc(CO)n1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(CO)nn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(CS(C)(=O)=O)nn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cc(n[nH]1)C(C)(C)O |r,THB:12:13:6.5:22,9:8:6.5:22|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1coc(n1)C(C)(C)O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1nnccc1C |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ccc(nn1)C(C)(C)O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ncc(cn1)C(C)(C)O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ncc(O)cn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ncc(cn1)C#N |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cncc(CO)n1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)CN1CC(C1)C#N |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1coc(CC#N)n1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1nc(C)oc1C |r|
CCN(C(C)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ncco1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1cnc(cn1)C(C)(C)O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ncc(o1)C(C)(C)O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ncc(CS(C)(=O)=O)cn1 |r|
CCN([C@H](C)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ncco1 |r|
CCN([C@@H](C)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1ncco1 |r|
CCN([C@H](C)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1coc(n1)C(C)(C)O |r|
CCN([C@@H](C)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1coc(n1)C(C)(C)O |r|
CCN([C@H](C)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1nc(C)oc1C |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)CN1CC(O)C1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)c1nc(co1)C(C)(C)O |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)[C@@H](O)c1ncccn1 |r|
CCN(C[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(=O)[C@H](O)c1ncccn1 |r|
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(=O)OC(C)(C)C)C(=O)c1c(Cl)cccc1C1CC1 |t:20|
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:20|
COC(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(=O)OC(C)(C)C)C(=O)c1c(Cl)cccc1C1CC1 |t:15|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CCC1 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CC(F)C1 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CC(F)(F)C1 |c:6|
OC1CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:19|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CC(O)(C1)C1CC1 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CC(O)(C1)C(F)(F)F |c:6|
CC1(O)CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:20|
COC1(C)CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:21|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CC(C1)n1cccn1 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CC(C1)n1ccnc1 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CC(C1)n1cnnc1 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CC(C1)c1nnc[nH]1 |c:6|
NC1CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:19|
CC1(CN)CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:21|
CC(C)(O)C1CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:22|
CN(C)C1CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:21|
CN1CCCC11CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:24|
CN(C1CNC1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:20|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CC(C1)C(F)F |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CC(F)(C1)C#N |c:6|
OC[C@@H]1CCN1C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |r,t:20|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CC2(CCO2)C1 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CC2(C1)CCCO2 |c:6|
CN1CCC2CN(CC12)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:24|
COC[C@H]1CCCN1C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |r,t:22|
Cn1cnc(n1)C1CCCN1C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:26|
CNCC1CCCN1C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:22|
COC[C@@H]1CCCN1C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |r,t:22|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CCC[C@H]1CF |r,c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CCC[C@@H]1CF |r,c:6|
OC[C@@H]1CCCN1C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |r,t:21|
OC[C@H]1CCCN1C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |r,t:21|
CO[C@@H]1CCN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |r,t:21|
CO[C@H]1CCN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |r,t:21|
CC1(O)CCN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:21|
CN1CCN(CC11COC1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:25|
CN(C)[C@H]1CCN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |r,t:22|
CN(C)[C@@H]1CCN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |r,t:22|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CC2(C1)CCOC2 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CCC2(CCO2)C1 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CCC2(CCOC2)C1 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CC2COCC2C1 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CCC2(CCCO2)C1 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CC(C1)N1CC(F)C1 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CCC2(COC2)C1 |c:6|
CN1CCC11CCN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:24|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1C[C@@H]2COC[C@@H]2C1 |r,c:6|
CC(C)N1CC2(C1)CN(C2)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:25|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CC2(C1)CN(C2)c1ncccn1 |c:6|
CC(C)(C)OC(=O)N1CC2(C1)CN(C2)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:29|
CN1CCC(C1)OC(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:21|
CN1CCN(CC1=O)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:22|
CS(=O)(=O)C1CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:22|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CCc12)C(=O)N1CC2(COC2)C1 |c:6|
CN(C)[C@@H]1CCN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(ccc(F)c1Cl)C1CC1 |r,t:22|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)c(F)ccc2C2CC2)c2CC(CCc12)C(=O)N1CC(C1)N1CC(F)C1 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)c(F)ccc2C2CC2)c2CC(CCc12)C(=O)N1CC2(C1)CCOC2 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)c(F)ccc2C2CC2)c2CC(CCc12)C(=O)N1CCC2(CCN2)C1 |c:6|
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)c(F)ccc1C1CC1 |t:20|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)c(F)ccc2C2CC2)c2CC(CCc12)C(=O)N1CC2(C1)CCCO2 |c:6|
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(=O)OC(C)(C)C)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |t:20|
O[C@H]1CCC[C@H]1NC(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |r,t:21|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)N[C@H]1CCC[C@H]1F |r,c:6|
O[C@@H]1CCC[C@H]1NC(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |r,t:21|
O[C@@H]1CCC[C@@H]1NC(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |r,t:21|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)N[C@@H]1CNC[C@@H]1F |r,c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)N[C@H]1CNC[C@@H]1F |r,c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)N[C@@H]1COC[C@@H]1F |r,c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)N[C@H]1COC[C@@H]1F |r,c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)NCC1(F)CNC1 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)NCC1(F)CCNCC1 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)NC1CCNCC1(F)F |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)NC[C@]1(F)CCCNC1 |r,c:6|
CN(C)CC(F)(F)CNC(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |t:22|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)NC1CC1(F)F |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)Nc1ccn(CC(F)(F)F)n1 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)Nc1ccccc1F |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)Nc1ncccc1F |c:6|
CN(C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F)c1ccccn1 |t:15|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)Nc1ccccn1 |c:6|
CO[C@H]1CN(C[C@@H]1O)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |r,t:22|
CN(C)[C@H]1CN(C[C@@H]1O)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |r,t:23|
O[C@@H]1CN(C[C@@H]1F)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |r,t:21|
CN(C)C1CN(CC1(F)F)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |t:24|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)N1CCC(C1)N1CCC1 |c:6|
CN(C)[C@H]1CN(C[C@H]1F)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |r,t:23|
COC1(C)CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |t:21|
CN(C)[C@H]1CN(C[C@@H]1F)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |r,t:23|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)N1CC2(C1)CCCO2 |c:6|
CN(C)[C@@H]1CCN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |r,t:22|
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)F |t:20|
CN(Cc1cnn(C)c1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |t:23|
Cn1ncc2CN(Cc12)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |t:24|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)N1CCC2(COC2)C1 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)N1CC[C@H](C1)C#N |r,c:6|
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |t:20|
CN(Cc1cnccn1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |t:23|
OC1CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |t:19|
CC1(O)CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |t:20|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)F)c2CC(CCc12)C(=O)N1CCC2(COC2)C1 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)N1CC(C1)N1CC(F)C1 |c:6|
CC1(CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)N1CC2(C1)CCCO2)C(O)=O |c:4|
CN(C)[C@@H]1CCN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(C)(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |r,t:22|
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(C)(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |t:20|
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(C)(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)F |t:20|
COC1CN(C1)C(=O)C1(C)CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:21|
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(C)ccnc1N1CCC1 |t:20|
CN(C)[C@@H]1CCN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(=O)OC(C)(C)C)C(=O)c1c(Cl)cccc1C1(F)CCC1 |r,t:22|
COC(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(=O)OC(C)(C)C)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |t:15|
COC1(C)CCN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(=O)OC(C)(C)C)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |t:22|
COCCN(C)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |t:19|
CN(C)CCN(C)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |t:20|
CN(C)CCNC(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |t:19|
CC1(O)CCN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |t:21|
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(=O)OC(C)(C)C)C(=O)c1c(Cl)cccc1C1(F)CCC1 |t:20|
C[C@H]1C=C(CC[C@H]1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)N1CC(C)(O)C1 |r,c:2|
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=C[C@H](C)[C@@H](CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |r,t:20|
COC1CN(C1)C(=O)C1CCc2c(C1)n(nc2C1=CC[C@H]([C@@H](C)C1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |r,t:20|
C[C@H]1C=C(CC[C@H]1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)N1CC(O)C1 |r,c:2|
C[C@H]1CC(=CC[C@H]1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)N1CCC2(COC2)C1 |r,c:3|
C[C@H]1CC(=CC[C@H]1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)N1CCC(O)CC1 |r,c:3|
COC1CN(C1)C(=O)C1CCc2c(nn(C(=O)c3c(Cl)cccc3C3CC3)c2C1)N1CCC(CC1)C(=O)OC(C)(C)C
COC1CN(C1)C(=O)C1CCc2c(nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c2C1)N1CCC(CC1)C(=O)OC(C)(C)C
Cc1cccc2N(C(=O)\C(=C/c3c(Cl)cccc3C3CC3)c12)c1ccc(C(O)=O)c(O)c1
Cc1cccc2N(C(=O)\C(=C/c3c(Cl)cccc3C3CC3)c12)c1ccc(cc1)C(O)=O
Cc1cccc2N(C(=O)\C(=C\c3c(Cl)cccc3C3CC3)c12)c1ccc(cc1)C(O)=O
COc1cccc(Cl)c1\C=C1/C(=O)N(c2cccc(C)c12)c1ccc(C(O)=O)c(O)c1
Cc1cccc2N(C(=O)\C(=C/c3c(Cl)cccc3Cl)c12)c1ccc(C(O)=O)c(O)c1
Cc1cccc2N(C(=O)\C(=C/c3c(Cl)cccc3Cl)c12)c1ccc(cc1)C(O)=O
Cc1cccc2N(C(=O)\C(=C/c3c(Cl)cccc3C(F)(F)F)c12)c1ccc(C(O)=O)c(O)c1
Cc1cccc2N(C(=O)\C(=C/c3c(Cl)cccc3Br)c12)c1ccc(C(O)=O)c(O)c1
COc1cccc2N(C(=O)\C(=C/c3c(Cl)cccc3C3CC3)c12)c1ccc(C(O)=O)c(O)c1
Cc1cccc2N(C(=O)\C(=C/c3c(F)cccc3Cl)c12)c1ccc(C(O)=O)c(O)c1
Cc1cccc2N(C(=O)\C(=C/c3c(C)cccc3Cl)c12)c1ccc(C(O)=O)c(O)c1
COc1cccc2N(C(=O)\C(=C/c3c(Cl)cccc3Cl)c12)c1ccc(C(O)=O)c(O)c1
OC(=O)c1ccc(cc1O)N1C(=O)\C(=C/c2c(Cl)cccc2C2CC2)c2c1cccc2C1CC1
OC(=O)c1ccc(cc1)N1C(=O)\C(=C/c2c(Cl)cccc2C2CC2)c2c1cccc2-c1ccccc1
OC(=O)c1ccc(cc1O)N1C(=O)\C(=C/c2c(Cl)cccc2C2CC2)c2c1cccc2Cl
OC(=O)c1ccc(cc1)N1C(=O)\C(=C/c2c(Cl)cccc2Cl)c2c1cccc2F
OC(=O)c1ccc(cc1)N1C(=O)\C(=C\c2c(Cl)cccc2Cl)c2c1cccc2F
OC(=O)c1ccc(cc1)N1C(=O)\C(=C/c2c(Cl)cccc2C2CC2)c2c1cccc2F
OC(=O)c1ccc(cc1)N1C(=O)\C(=C\c2c(Cl)cccc2C2CC2)c2c1cccc2F
OC(=O)c1ccc(cc1)N1C(=O)\C(=C/c2c(F)cccc2Cl)c2c1cccc2F
OC(=O)c1ccc(cc1)N1C(=O)\C(=C\c2c(F)cccc2Cl)c2c1cccc2F
OC(=O)c1ccc(cc1)N1C(=O)\C(=C/c2c(F)cccc2F)c2c1cccc2F
OC(=O)c1ccc(cc1)N1C(=O)\C(=C\c2c(F)cccc2F)c2c1cccc2F
OC(=O)c1ccc(cc1)N1C(=O)\C(=C/c2c(Cl)cccc2C(F)(F)F)c2c1cccc2F
OC(=O)c1ccc(cc1)N1C(=O)\C(=C\c2c(Cl)cccc2C(F)(F)F)c2c1cccc2F
CCCc1cccc(Cl)c1\C=C1/C(=O)N(c2cccc(F)c12)c1ccc(cc1)C(O)=O
CCCc1cccc(Cl)c1\C=C1\C(=O)N(c2cccc(F)c12)c1ccc(cc1)C(O)=O
OC(=O)c1ccc(cc1O)N1C(=O)\C(=C/c2c(Cl)cccc2C2CC2)c2c1cccc2F
OC(=O)c1ccc(cc1O)N1C(=O)\C(=C\c2c(Cl)cccc2C2CC2)c2c1cccc2F
OC(=O)c1ccc(cc1O)N1C(=O)\C(=C/c2c(Cl)cccc2Cl)c2c1cccc2F
OC(=O)c1ccc(cc1O)N1C(=O)\C(=C\c2c(Cl)cccc2Cl)c2c1cccc2F
OC(=O)c1ccc(cc1)N1C(=O)\C(=C/c2c(Cl)cccc2Cl)c2c1cccc2Cl
Cc1cccc2N(C(=O)\C(=C/c3c(Cl)cccc3C3CC3)c12)c1ccc(C(O)=O)c(Cl)c1
Cc1cccc2N(C(=O)\C(=C/c3c(Cl)cccc3C3CC3)c12)c1ccc(C(O)=O)c(F)c1
OC(=O)c1ccc(cc1O)N1C(=O)\C(=C/c2c(Cl)cccc2C2CC2)c2c1cccc2C(F)(F)F
OC(=O)c1ccc(cc1O)N1C(=O)\C(=C/c2c(Cl)cccc2C2CC2)c2ccccc12
Cc1cccc2N(C(=O)\C(=C/c3c(Cl)cccc3C3CC3)c12)c1ccc(C(O)=O)c(OC(=O)C(C)(C)C)c1
Cc1cccc2N(C(=O)\C(=C/c3c(C)cccc3Cl)c12)c1ccc(cc1)C(O)=O
COc1cccc2N(C(=O)\C(=C/c3c(Cl)cccc3C3CC3)c12)c1ccc(cc1)C(O)=O
COc1cccc2N(C(=O)\C(=C/c3c(Cl)cccc3Cl)c12)c1ccc(cc1)C(O)=O
COc1cccc(Cl)c1\C=C1/C(=O)N(c2cccc(C)c12)c1ccc(cc1)C(O)=O
Cc1cccc2N(C(=O)\C(=C/c3c(Cl)cccc3C3CC3)c12)c1ccc(C(O)=O)c(N)c1
Cc1cccc2N(C(=O)\C(=C/c3c(Cl)cccc3C3CCC3)c12)c1ccc(cc1)C(O)=O
Cc1cccc2N(C(=O)\C(=C/c3c(Cl)cccc3C3CCC3)c12)c1ccc(C(O)=O)c(O)c1
CC(C)c1cccc(Cl)c1\C=C1/C(=O)N(c2cccc(C)c12)c1ccc(C(O)=O)c(O)c1
CCc1cccc(Cl)c1\C=C1/C(=O)N(c2cccc(C)c12)c1ccc(C(O)=O)c(O)c1
COC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CCCCc12 |c:7|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2COCCc12 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CCCc12 |c:6|
CC1(CC1)c1cccc(Cl)c1C(=O)n1nc(c2CCOCc12)C1=CCC(CC1)C(O)=O |t:26|
CC1(CC1)c1cccc(Cl)c1C(=O)n1nc(c2CCCc12)C1=CCC(CC1)C(O)=O |t:25|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CCC2)C#N)c2CCCc12 |c:6|
CCOC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CCC2)c2COCCc12 |c:8|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C#N)c2COCCc12 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CCC2)C#N)c2COCCc12 |c:6|
CC1CCCc2c1c(nn2C(=O)c1c(Cl)cccc1C1CC1)[C@@]1(CCC=CC1)C(O)=O |c:29|
CC1CCCc2c1c(nn2C(=O)c1c(Cl)cccc1C1CC1)C1=CCC(CC1)C(O)=O |t:26|
COC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2C[C@H](CCc12)C(O)=O |c:7|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC3(CCOC3=O)CCc12 |c:6|
OC[C@H]1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:13|
OCC1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)c(F)ccc1C1CC1 |t:13|
OCC1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1COC1 |t:13|
OCC1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |t:13|
C[C@H](O)[C@@H]1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:14|
CC(O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(=O)OC(C)(C)C)C(=O)c1c(Cl)cccc1C1CC1 |t:14|
C[C@@]1(CO)CCc2c(C1)n(nc2C1=CCC(CC1)C([O-])=O)C(=O)c1c(Cl)cccc1C1CC1 |t:14|
CC1(CO)CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:14|
O[C@H]1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:12|
OC1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:12|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(F)CCc12 |c:6|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CCCNc12 |c:6|
C[C@]1(CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CO)CCc12)C(O)=O |c:4|
CC1(CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CC(CO)CCc12)C(O)=O |c:4|
NC[C@H]1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:13|
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CCCOc12 |c:6|
OC(=O)C1CCN(CC1)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CCCCc12
O[C@@H]1CN(CCC1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CCCCc12
O[C@@H]1CN(CC[C@H]1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CCCCc12 |r|
O[C@@H]1CN(CCC1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CCCCc12
O[C@@H]1CN(CC[C@H]1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CCCCc12 |r|
CCOC(=O)[C@H]1CCN(C[C@H]1O)c1nn(C(=O)c2c(Cl)cccc2C2CC2)c2CCCCc12 |r|
Fc1ccc(cc1)S(=O)(=O)n1ncc2cnc(NC(=O)c3c(cccc3C(F)(F)F)C(F)(F)F)cc12
Cc1cccc(c1Cc1cn(-c2ccc(cc2)C(O)=O)c2ccccc12)C(F)(F)F
OC(=O)c1ccc(cc1)-n1cc(Cc2c(Cl)cccc2C(F)(F)F)c2ccccc12
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cncnc12
COc1cccc(F)c1C(=O)c1cn(-c2ccc(cc2)C(O)=O)c2ccccc12
COc1cccc(F)c1C(=O)c1cn(-c2ccc(cc2)C(O)=O)c2c(F)cccc12
OC(=O)c1ccc(cc1O)-n1cc(Cc2c(Cl)cccc2C(F)(F)F)c2ccccc12
Cc1cccc2c(cn(-c3ccc(cc3)C(O)=O)c12)C(=O)c1c(Cl)cccc1C(F)(F)F
OC(=O)c1ccc(nc1)-n1cc(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
Cc1cccc2c(cn(-c3ccc(cc3)C(O)=O)c12)C(=O)c1c(Cl)cccc1Cl
COc1cccc(F)c1C(=O)c1nn(-c2ccc(cc2)C(O)=O)c2ccccc12
Cc1cccc2c(cn(-c3ccc(cc3)C(O)=O)c12)C(=O)c1c(F)cccc1C(F)(F)F
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2c(F)cccc2OC(F)(F)F)c2cccc(F)c12
OC(=O)c1ccc(c(F)c1)-n1cc(C(=O)c2c(F)cccc2OC(F)(F)F)c2cccc(F)c12
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2c(F)cccc2OC(F)(F)F)c2ccccc12
OC(=O)c1ccc(cn1)-n1nc(C(=O)c2c(Cl)cccc2Cl)c2ccccc12
OC(=O)c1ccc(nc1)-n1nc(C(=O)c2c(Cl)cccc2Cl)c2ccccc12
OC(=O)c1ccc(nc1)-n1cc(Cc2c(Cl)cccc2C(F)(F)F)c2ccccc12
OC(=O)c1ccc(nc1)-n1cc(Cc2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
OC(=O)c1ccc(nc1)-n1cc(C(=O)c2c(Cl)cccc2C(F)(F)F)c2ccccc12
OC(=O)c1ccc(nc1)-n1cc(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccnc12
OC(=O)c1ccc(cn1)-n1nc(C(=O)c2c(Cl)cccc2C(F)(F)F)c2ccccc12
OC(=O)c1ccc(nc1)-n1nc(C(=O)c2c(Cl)cccc2C(F)(F)F)c2ccccc12
OC(=O)c1ccc(cc1)-n1cc(Cc2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
C[C@@H](C(=O)N1CC[C@H]([C@@H](C)C1)c1cn(C)c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc12)C(C)(C)C |r|
C[C@H](C1CCCC1)C(=O)N1CC[C@H]([C@@H](C)C1)c1cn(C)c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc12 |r|
C[C@H]1CN(CC[C@H]1c1cn(C)c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc12)C(=O)C1CCCC1 |r|
C[C@@H]1CN(CC[C@@H]1c1cn(C)c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc12)C(=O)C1CCCC1 |r|
CC(C)C(=O)N1CC[C@H]([C@@H](C)C1)c1cn(C)c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc12 |r|
Cn1cc(C2CCN(CC2)C(=O)c2ccns2)c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12
C[C@H](C1CCCC1)C(=O)N1CCC(CC1)c1cn(C)c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc12 |r|
Cn1cc(C2CCN(CC2)C(=O)C2CC2)c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12
CC(CC(=O)N1CCC(CC1)c1cn(C)c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc12)C(F)(F)F
C[C@@H](C(=O)N1CCC(CC1)c1cn(C)c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc12)C(C)(C)C |r|
Cn1cc(C2CCN(CC2)C(=O)C2CCC2)c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12
CC(C)CC(=O)N1CCC(CC1)c1cn(C)c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc12
Cn1cc(C2CCN(CC2)C(=O)CC2CC2)c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12
Cn1cc(C2CCN(CC2)C(=O)C2CCCCC2)c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12
Cc1cccc(F)c1C(=O)N1CCC(CC1)c1cn(C)c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc12
CC(C)[C@H](C)C(=O)N1CCC(CC1)c1cn(C)c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc12 |r|
Cn1cc(C2CCN(CC2)C(=O)C2CCCC2)c2cc(NS(=O)(=O)c3ccccc3F)ccc12
CC(C)C(=O)N1CC[C@H](CC1(C)C)c1cn(C)c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc12 |r|
Cn1cc([C@@H]2CCN(C(=O)C3CCCC3)C(C)(C)C2)c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12 |r|
C[C@H]1C[C@H](CCN1C(=O)C1CCCC1)c1cn(C)c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc12 |r|
C[C@H]1C[C@@H](CCN1C(=O)C1CCCC1)c1cn(C)c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc12 |r|
COc1cc(ccc1F)S(=O)(=O)Nc1ccc2n(C)cc(C3CCN(CC3)C(=O)C(C)C)c2c1
CC(C)C(=O)N1CCC(CC1)c1cn(C)c2ccc(NS(=O)(=O)c3ccc(F)c(O)c3)cc12
CC(C)C(=O)N1CCC(CC1)c1cn(C)c2ccc(NS(=O)(=O)c3ccc(F)c(O[C@@H]4CCOC4)c3)cc12 |r|
C[C@@H](C(=O)N1CCC(CC1)c1cn(C)c2ccc(NS(=O)(=O)c3ccc(C)cc3)cc12)C(C)(C)C |r|
C[C@@H](C(=O)N1CCC(CC1)c1cn(C)c2ccc(NS(=O)(=O)c3c(C)nn(C)c3C)cc12)C(C)(C)C |r|
CCOc1ccccc1S(=O)(=O)Nc1ccc2n(C)cc(C3CCN(CC3)C(=O)[C@H](C)C(C)(C)C)c2c1 |r|
C[C@@H](C(=O)N1CCC(CC1)c1cn(C)c2ccc(NS(=O)(=O)c3ccccc3F)cc12)C(C)(C)C |r|
C[C@@H](C(=O)N1CCC(CC1)c1cn(C)c2ccc(NS(=O)(=O)c3ccccc3)cc12)C(C)(C)C |r|
C[C@@H](C(=O)N1CCC(CC1)c1cn(C)c2ccc(NS(=O)(=O)c3c(C)noc3C)cc12)C(C)(C)C |r|
C[C@@H](C(=O)N1CCC(CC1)c1cn(C)c2ccc(NS(=O)(=O)c3ccc(F)cc3)cc12)C12CC(C1)C2 |r|
C[C@H](C1CCCC1)C(=O)N1CC[C@H]([C@@H](C)C1)c1cn(C)c2ccc(NS(=O)(=O)c3c(C)nn(C)c3C)cc12 |r|
CCOc1ccccc1S(=O)(=O)Nc1ccc2n(C)cc([C@@H]3CCN(C[C@@H]3C)C(=O)[C@H](C)C3CCCC3)c2c1 |r|
C[C@H](C1CCCC1)C(=O)N1CC[C@H]([C@@H](C)C1)c1cn(C)c2ccc(NS(=O)(=O)c3ccccc3F)cc12 |r|
C[C@H](C1CCCC1)C(=O)N1CC[C@H]([C@@H](C)C1)c1cn(C)c2ccc(NS(=O)(=O)c3cc(C)ccc3F)cc12 |r|
CCS(=O)(=O)c1ccc(nc1)CNC(=O)c2cc3c(nc2)[C@@H](N(C3)CC4CCC(CC4)C(F)(F)F)C(C)C
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4nccc(n4)C(F)(F)F)Cc3c2)nc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc3c2)S(=O)(=O)c2ccc(cc2)C#N)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc3c2)c2ncc([C@H](C)O)c(n2)C(F)(F)F)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc3c2)C(=O)OC(F)(F)F)nc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@@H](C(C)C)N(C[C@H]4CC[C@@H](CC4)C(F)(F)F)Cc3c2)cc1 |r,wU:17.17,26.29,wD:23.22,(11.42,-1.61,;9.88,-1.61,;9.11,-2.95,;10.45,-3.72,;8.34,-4.28,;7.78,-2.18,;6.44,-2.95,;5.11,-2.18,;5.11,-.64,;3.78,.13,;2.44,-.64,;1.11,.13,;1.11,1.67,;-.22,-.64,;-.22,-2.18,;-1.56,-2.95,;-2.89,-2.18,;-4.36,-2.65,;-4.83,-4.12,;-3.8,-5.26,;-6.34,-4.44,;-5.26,-1.41,;-6.8,-1.41,;-7.57,-.07,;-6.8,1.26,;-7.57,2.59,;-9.11,2.59,;-9.88,1.26,;-9.11,-.07,;-9.88,3.93,;-9.11,5.26,;-11.42,3.93,;-10.65,5.26,;-4.36,-.16,;-2.89,-.64,;-1.56,.13,;6.44,.13,;7.78,-.64,)|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCc1ccnn1C |r|
CC(C)[C@@H]1N(Cc2ccc(cc2)C(F)(F)F)Cc2cc(cnc12)C(=O)NCc1cnn(C)c1 |r|
CCS(=O)(=O)n1cc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc4ccc(cc4)C(F)(F)F)Cc3c2)cn1 |r|
CC1(O)CCN(CC1)C(=O)[C@H]1CC[C@]2([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@]12CC[C@@H]([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NCc1ccncc1 |r|
CC(=O)N1CCN(CC1)C(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1CCOCC1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@]12CC[C@H]([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1CCOCC1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@]12CC[C@H]([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)Nc1ccncc1 |r|
CC(=O)N1CCN(CC1)C(=O)[C@@H]1CC[C@]2([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NCc1ccncc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@]12CC[C@H]([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NCc1ccncc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)Nc1ccncc1 |r|
CC1(O)CCN(CC1)C(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NC1CCS(=O)(=O)C1 |r,w:36.39|
C[C@]1(O)CC[C@@H](CC1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:15.17,1.1,wD:14.37,11.11,5.8,1.0,(-12.06,-5.41,;-11.48,-3.98,;-12.99,-4.3,;-11.76,-2.46,;-10.58,-1.47,;-9.13,-1.99,;-8.86,-3.51,;-10.04,-4.5,;-7.96,-1,;-6.51,-1.52,;-6.23,-3.03,;-5.33,-.52,;-5.44,1.01,;-4.02,1.6,;-3.02,.42,;-3.84,-.89,;-3.11,-2.25,;-1.57,-2.3,;-.76,-.99,;.78,-1.03,;1.59,.27,;.87,1.63,;-.67,1.68,;-1.48,.37,;3.13,.23,;3.18,1.77,;4.67,.18,;6.21,.13,;4.62,-1.36,;4.72,1.72,;3.08,-1.31,;3.04,-2.85,;4.3,-2.26,;1.55,-1.26,;-2.35,1.81,;-3.74,2.48,;-1,2.53,;-1.68,3.19,;-2.55,4.47,;-1.88,5.85,;-.34,5.97,;.33,7.35,;.52,4.69,;-.15,3.31,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NC1CCS(=O)(=O)CC1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NCC1CCS(=O)(=O)C1 |r,w:36.40|
COC(=O)C1(CCS(=O)(=O)CC1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCN(CC1)C(=O)[C@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC1(O)CCN(CC1)C(=O)[C@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1CCOCC1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)Nc1ccncc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NCc1ccncc1 |r|
CC(C)(O)[C@H](F)CNC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(O)C(O)CNC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:4.4|
O[C@H]1C[C@@H](C1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:12.14,1.0,wD:11.34,8.8,3.5,(-12.95,-4.69,;-11.78,-3.7,;-11.65,-2.16,;-10.11,-2.29,;-10.24,-3.82,;-8.94,-1.3,;-7.49,-1.82,;-7.22,-3.33,;-6.31,-.82,;-6.43,.71,;-5,1.29,;-4.01,.12,;-4.82,-1.19,;-4.09,-2.55,;-2.55,-2.6,;-1.74,-1.29,;-.2,-1.33,;.61,-.03,;-.12,1.33,;-1.66,1.38,;-2.47,.07,;2.15,-.07,;2.2,1.47,;3.69,-.12,;5.23,-.17,;3.64,-1.66,;3.74,1.42,;2.1,-1.61,;2.05,-3.15,;3.32,-2.56,;.56,-1.56,;-3.34,1.51,;-4.72,2.18,;-1.98,2.23,;-2.67,2.89,;-3.53,4.17,;-2.86,5.55,;-1.33,5.67,;-.66,7.05,;-.46,4.39,;-1.13,3,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NC12CC(C1)C2 |r|
NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)Nc1ccnc2[nH]ncc12 |r|
C[C@@H](NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C1CC1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N[C@@H]1CCOC1 |r|
CC(C)(O)CNC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC1(CC1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N[C@H]1CCOC1 |r|
FC1CC1NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:3.4,1.0|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NC1(CC1)C#N |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NC1CC(F)(F)C1 |r|
O[C@H]1CC[C@@H](CC1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:14.16,1.0,wD:13.36,10.10,4.7,(-13.15,-5.09,;-11.97,-4.09,;-12.24,-2.58,;-11.07,-1.58,;-9.62,-2.1,;-9.35,-3.62,;-10.52,-4.61,;-8.44,-1.11,;-6.99,-1.63,;-6.72,-3.15,;-5.82,-.64,;-5.93,.9,;-4.5,1.48,;-3.51,.3,;-4.32,-1,;-3.59,-2.36,;-2.05,-2.41,;-1.24,-1.1,;.3,-1.15,;1.11,.16,;.38,1.52,;-1.16,1.57,;-1.97,.26,;2.65,.11,;2.69,1.65,;4.19,.06,;5.72,.02,;4.14,-1.48,;4.23,1.6,;2.6,-1.43,;2.55,-2.97,;3.82,-2.37,;1.06,-1.38,;-2.84,1.69,;-4.23,2.36,;-1.48,2.42,;-2.17,3.08,;-3.04,4.35,;-2.37,5.74,;-.83,5.85,;-.16,7.24,;.04,4.58,;-.63,3.19,)|
CNC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1CCc2[nH]ncc2C1 |r|
CC1N(CCNC1=O)C(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:1.0|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1CCS(=O)(=O)CC1 |r|
O[C@H]1C[C@H](C1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:12.14,wD:11.34,8.8,3.5,1.0,(-12.95,-4.69,;-11.78,-3.7,;-10.24,-3.82,;-10.11,-2.29,;-11.65,-2.16,;-8.94,-1.3,;-7.49,-1.82,;-7.22,-3.33,;-6.31,-.82,;-6.43,.71,;-5,1.29,;-4.01,.12,;-4.82,-1.19,;-4.09,-2.55,;-2.55,-2.6,;-1.74,-1.29,;-.2,-1.33,;.61,-.03,;-.12,1.33,;-1.66,1.38,;-2.47,.07,;2.15,-.07,;2.2,1.47,;3.69,-.12,;5.23,-.17,;3.64,-1.66,;3.74,1.42,;2.1,-1.61,;2.05,-3.15,;3.32,-2.56,;.56,-1.56,;-3.34,1.51,;-4.72,2.18,;-1.98,2.23,;-2.67,2.89,;-3.53,4.17,;-2.86,5.55,;-1.33,5.67,;-.66,7.05,;-.46,4.39,;-1.13,3,)|
CN(C)C(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1C[C@H](Cc2cccc(F)c2)NC(=O)C1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1CCNC(=O)C1 |r|
CC1(C)N(CCNC1=O)C(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN1CCN(CC1=O)C(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC1CN(CC(=O)N1)C(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:1.0|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1CC(=O)NC(=O)C1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NC1CC1(F)F |r,w:36.39|
C[C@H](NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C1CCC1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NCC1CCC1 |r|
C[C@H](CO)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
O[C@H](CNC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
C[C@@H](O)CNC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC[C@H](O)CNC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
O[C@@H]1CCC[C@H]1NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
O[C@@H](CNC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
C[C@H](O)CNC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
O[C@H]1CCC[C@@H]1NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@@H](CO)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@H](NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C1CC1 |r|
OCCNC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1CC(F)(F)C(F)(F)C1 |r|
OC[C@H]1CC(F)(F)CN1C(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1CCC(F)(F)C1 |r|
NC(=O)[C@H]1CC(F)(F)CN1C(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(O)C(C)(C)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NC1CCC(F)(F)C1 |r|
OC1(CNC(=O)[C@@H]2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)CCCCC1 |r|
OC1(CNC(=O)[C@@H]2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)CCCC1 |r|
OC1(CNC(=O)[C@@H]2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)CCC1 |r|
OC1(CNC(=O)[C@@H]2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)CC1 |r|
CN1CCC(O)(CNC(=O)[C@@H]2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)CC1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1CCC(=O)N1 |r|
OC1(CNC(=O)[C@@H]2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)CCOCC1 |r|
CS(=O)(=O)N1CCC(CC1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(I)ccc21)C(=O)N1CCOCC1 |r|
CC(=O)N1CCN(CC1)C(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(I)ccc21)S(=O)(=O)c1ccc(F)cc1 |r|
CS(=O)(=O)N1CCC(CC1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NCc1ccncc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1CCC2(CCNC2=O)CC1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1CCC2(CNC(=O)C2)CC1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1CCC2(CC(=O)N2)CC1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)N1CCC2(CNC2=O)CC1 |r|
OC(=O)C1CC(CNC(=O)[C@@H]2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)C1 |r,wU:14.15,wD:13.35,10.9,(-4.85,-15.42,;-6.38,-15.57,;-7.01,-16.97,;-7.28,-14.32,;-7.02,-12.8,;-8.54,-12.55,;-9.5,-11.25,;-8.71,-9.86,;-8.16,-8.35,;-9.69,-7.88,;-6.74,-7.53,;-6.85,-5.99,;-5.43,-5.41,;-4.43,-6.59,;-5.24,-7.89,;-4.51,-9.25,;-2.97,-9.3,;-2.16,-7.99,;-.62,-8.04,;.19,-6.73,;-.54,-5.37,;-2.08,-5.32,;-2.89,-6.63,;2.1,-7.18,;3.7,-7.61,;2.55,-9.04,;3.06,-10.62,;1.52,-10.34,;4.19,-9.41,;2.65,-5.23,;2.99,-3.57,;.99,-4.79,;4.28,-4.61,;-4.4,-4.8,;-4.36,-3.05,;-6.21,-4.43,;-2.7,-5.27,;-1.75,-4.05,;-.23,-4.26,;.47,-5.87,;2.02,-6.11,;-.59,-6.9,;-2.11,-6.69,;-8.79,-14.07,)|
OC(=O)[C@H]1CC[C@@H](C1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@H](CC(O)=O)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)[C@H]1C[C@@H](C1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:14.16,5.7,wD:13.36,10.10,3.2,(-12.48,-5.57,;-12.74,-4,;-14.24,-3.48,;-11.5,-2.95,;-9.97,-3.08,;-9.84,-1.55,;-11.37,-1.42,;-8.61,-.57,;-7.17,-1.22,;-6.97,-2.8,;-6.04,-.08,;-6.15,1.45,;-4.72,2.04,;-3.73,.86,;-4.54,-.45,;-3.81,-1.81,;-2.27,-1.85,;-1.46,-.54,;.08,-.59,;.89,.72,;.16,2.07,;-1.38,2.12,;-2.19,.81,;2.81,.24,;4.43,-.18,;3.22,-1.58,;3.64,-3.18,;2.14,-2.83,;4.79,-2.04,;3.35,2.2,;3.68,3.85,;1.74,2.66,;4.96,2.79,;-3.7,2.65,;-3.59,4.4,;-5.51,3.03,;-2,2.18,;-1.05,3.39,;.47,3.19,;1.17,1.57,;2.75,1.36,;.11,.54,;-1.41,.75,)|
OC(=O)C1CCN(C1)C(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)[C@@H]1C[C@@H](C1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:14.16,wD:13.36,10.10,5.7,3.2,(-12.48,-5.57,;-12.74,-4,;-14.24,-3.48,;-11.5,-2.95,;-11.37,-1.42,;-9.84,-1.55,;-9.97,-3.08,;-8.61,-.57,;-7.17,-1.22,;-6.97,-2.8,;-6.04,-.08,;-6.15,1.45,;-4.72,2.04,;-3.73,.86,;-4.54,-.45,;-3.81,-1.81,;-2.27,-1.85,;-1.46,-.54,;.08,-.59,;.89,.72,;.16,2.07,;-1.38,2.12,;-2.19,.81,;2.81,.24,;4.43,-.18,;3.22,-1.58,;3.64,-3.18,;2.14,-2.83,;4.79,-2.04,;3.35,2.2,;3.68,3.85,;1.74,2.66,;4.96,2.79,;-3.7,2.65,;-3.59,4.4,;-5.51,3.03,;-2,2.18,;-1.05,3.39,;.47,3.19,;1.17,1.57,;2.75,1.36,;.11,.54,;-1.41,.75,)|
OC(=O)C1CN(C1)C(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C12CC(C1)(C2)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)[C@H]1CC[C@H](C1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)[C@@H]1CC[C@H](C1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C1CCCC(C1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C1CCN(CC1)C(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)[C@H]1CC[C@@H](CC1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:16.18,3.2,wD:15.38,12.12,6.9,(-12.7,-5.91,;-12.98,-4.39,;-14.44,-3.86,;-11.78,-3.37,;-12.05,-1.86,;-10.88,-.86,;-9.43,-1.39,;-9.15,-2.9,;-10.33,-3.9,;-8.16,-.44,;-6.71,-1.11,;-6.39,-2.69,;-5.63,.08,;-5.74,1.62,;-4.31,2.2,;-3.32,1.02,;-4.13,-.29,;-3.4,-1.64,;-1.86,-1.69,;-1.05,-.38,;.49,-.43,;1.3,.88,;.57,2.24,;-.97,2.28,;-1.78,.97,;3.32,.44,;4.86,-.06,;3.67,-1.33,;4.06,-2.82,;2.78,-2.62,;5.14,-1.89,;4.05,2.28,;4.87,3.72,;3.46,3.78,;5.72,2.76,;-3.24,2.78,;-3.17,4.55,;-5,3.25,;-1.58,2.34,;-.64,3.56,;.89,3.35,;1.58,1.74,;2.92,1.63,;.52,.71,;-1,.91,)|
OC(=O)C12CCC(CC1)(CC2)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C1CCN(CC1)C(=O)[C@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@H]1CN(CC[C@@H]1C(O)=O)C(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)CNC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@H](NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(O)=O |r|
C[C@@H](CC(O)=O)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)CCNC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
N[C@H]1C[C@H](C1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:12.14,wD:11.34,8.8,3.5,1.0,(-11.73,-6.05,;-10.53,-5.03,;-8.99,-5.16,;-8.86,-3.62,;-10.4,-3.49,;-8.12,-2.24,;-8.3,-.68,;-9.84,-.18,;-6.79,-.12,;-6.9,1.42,;-5.47,2,;-4.48,.82,;-5.29,-.49,;-4.56,-1.84,;-3.02,-1.89,;-2.21,-.58,;-.67,-.63,;.14,.68,;-.59,2.04,;-2.13,2.08,;-2.94,.78,;2.14,.24,;3.83,-.16,;2.68,-1.53,;3.26,-3.1,;1.63,-2.8,;4.31,-1.88,;2.68,2.2,;3.06,3.82,;1.03,2.68,;4.33,2.68,;-4.46,2.61,;-4.39,4.35,;-6.3,2.97,;-2.74,2.14,;-1.8,3.36,;-.27,3.15,;.42,1.54,;1.97,1.32,;-.64,.51,;-2.16,.71,)|
N[C@H]1C[C@@H](C1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:12.14,1.0,wD:11.34,8.8,3.5,(-13.37,-4.25,;-12.15,-3.24,;-12.03,-1.7,;-10.49,-1.83,;-10.62,-3.36,;-9.24,-.88,;-7.8,-1.53,;-7.64,-3.11,;-6.69,-.36,;-6.8,1.17,;-5.38,1.76,;-4.38,.58,;-5.19,-.73,;-4.47,-2.09,;-2.93,-2.13,;-2.12,-.83,;-.58,-.87,;.23,.44,;-.49,1.79,;-2.03,1.84,;-2.84,.53,;2.28,.16,;3.83,-.39,;2.75,-1.63,;3.24,-3.25,;1.7,-2.93,;4.33,-2.15,;3.27,2.02,;4.21,3.42,;2.71,3.6,;4.93,2.03,;-4.35,2.36,;-4.25,4.1,;-6.18,2.73,;-2.65,1.9,;-1.71,3.11,;-.18,2.9,;.52,1.29,;2.01,1.4,;-.54,.26,;-2.07,.47,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)C(=O)NCC1CCNC1 |r|
N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
N[C@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
N[C@H]1CC[C@]2([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
N[C@@H]1CC[C@]2([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H](NC(=O)[C@@H]3CCC(=O)N3CCC#N)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
CC(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@]12CC[C@H](NC(=O)Cc3ccncc3)[C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H](NC(=O)Cc3ccncc3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
OC1(CCS(=O)(=O)CC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CS(=O)(=O)N1CCC(O)(CC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCC(CC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H](NC(=O)Cc3ccncc3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
OCC(=O)N[C@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCC(CC1)C(=O)N[C@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@]12CC[C@@H](NC(=O)Cc3ccncc3)[C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
NC(=O)[C@H]1CC[C@@H](CC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:16.18,3.2,wD:15.38,12.12,6.9,(-14.54,-4.38,;-13.01,-4.83,;-12.83,-6.41,;-11.77,-3.78,;-12.05,-2.26,;-10.87,-1.27,;-9.42,-1.79,;-9.15,-3.31,;-10.32,-4.3,;-8.38,-.6,;-9.12,.81,;-6.91,-1.22,;-5.62,-.32,;-5.73,1.21,;-4.31,1.79,;-3.31,.62,;-4.12,-.69,;-3.4,-2.05,;-1.86,-2.1,;-1.05,-.79,;.49,-.83,;1.3,.47,;.58,1.83,;-.96,1.88,;-1.77,.57,;3.33,.32,;3.51,-1.35,;3.74,2.29,;3.76,3.95,;5.12,3.2,;2.09,2.48,;5.15,-.09,;6.81,-.31,;6.28,1.17,;5.65,-1.65,;-3.28,2.42,;-3.17,4.16,;-5.09,2.8,;-1.58,1.94,;-.64,3.15,;.89,2.94,;1.59,1.33,;3.11,1.36,;.53,.3,;-1,.51,)|
OC1(CCOCC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN1[C@@H](C[C@@H](F)C1=O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OCC(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
NS(=O)(=O)N1CCC(CC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC1CC(CCS1(=O)=O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc3c2ccc(c3)C(C(F)(F)F)(C(F)(F)F)F)S(=O)(=O)c4ccc(cc4)F)O
C[C@@H](O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:16.18,3.2,wD:15.38,12.12,6.9,(-14.54,-4.38,;-13.01,-4.83,;-12.83,-6.41,;-11.77,-3.78,;-12.05,-2.26,;-10.87,-1.27,;-9.42,-1.79,;-9.15,-3.31,;-10.32,-4.3,;-8.38,-.6,;-9.12,.81,;-6.91,-1.22,;-5.62,-.32,;-5.73,1.21,;-4.31,1.79,;-3.31,.62,;-4.12,-.69,;-3.4,-2.05,;-1.86,-2.1,;-1.05,-.79,;.49,-.83,;1.3,.47,;.58,1.83,;-.96,1.88,;-1.77,.57,;3.33,.32,;3.51,-1.35,;3.74,2.29,;3.76,3.95,;5.12,3.2,;2.09,2.48,;5.15,-.09,;6.81,-.31,;6.28,1.17,;5.65,-1.65,;-3.28,2.42,;-3.17,4.16,;-5.09,2.8,;-1.58,1.94,;-.64,3.15,;.89,2.94,;1.59,1.33,;3.11,1.36,;.53,.3,;-1,.51,)|
OC(=O)C12CC(C1)(C2)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C1CC2(C1)CC(C2)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:10.11,3.2,wU:17.20,wD:16.40,13.14,(9.88,-4.21,;8.99,-2.9,;9.88,-1.58,;7.38,-2.9,;6.29,-1.81,;5.2,-2.9,;6.29,-3.98,;4.11,-1.81,;3.02,-2.9,;4.11,-3.98,;1.47,-3.14,;1.29,-4.73,;.76,-1.7,;-.83,-1.56,;-1.73,-2.81,;-3.2,-2.33,;-3.2,-.79,;-1.73,-.32,;-1.41,1.19,;-2.56,2.22,;-4.02,1.74,;-5.17,2.77,;-6.63,2.3,;-6.95,.79,;-5.81,-.24,;-4.34,.24,;-8.27,3.59,;-7.31,4.95,;-9.97,2.43,;-11.2,1.28,;-11.61,2.82,;-9.81,.79,;-9.2,5.22,;-10.19,6.62,;-10.87,5.2,;-8.51,6.73,;-4.39,-2.13,;-5.61,-3.38,;-3.26,-3.59,;-5.37,-.68,;-6.88,-1,;-7.91,.15,;-7.4,1.83,;-8.77,2.6,;-5.93,1.93,;-4.9,.79,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H](NC(=O)c3ccncc3F)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
Cc1ncn(C)c1C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Cc1nnsc1C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
NS(=O)(=O)CC(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H](NC(=O)C3CCS(=O)(=O)CC3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
CC1(COC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(CO)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC1(CC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC1(CCC(=O)N1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:1.0|
OC1(CCCCC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(C1CCOCC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:1.0|
O[C@@H](C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
O[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
NC(=O)c1c(F)cc(cc1F)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(Cc1ccncc1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:1.0|
Oc1ncccc1C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)c1ccc(cc1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H](NC(=O)C3CCC(=O)N3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r,w:15.17|
CC(C)(O)CC(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
O[C@H](CC(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(F)(F)F |r|
CC(=O)NC(CO)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:4.3|
CC(O)CC(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:1.0|
CS(=O)(=O)N1CC(O)(C1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN1[C@@H](C[C@@H](O)C1=O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(N1CCOCC1)C(=O)N[C@H]1CC[C@]2([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(O)[C@@H](O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Cn1nnnc1C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(O)Cn1nnnc1C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@@]1(O)C[C@@H](C1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:13.15,1.0,wD:12.35,9.9,4.6,1.1,(-13.25,-3.68,;-11.62,-3.61,;-11.96,-5.2,;-11.5,-2.08,;-9.96,-2.2,;-10.09,-3.74,;-8.96,-.99,;-9.91,.28,;-7.49,-1.61,;-6.16,-.74,;-6.27,.8,;-4.85,1.38,;-3.85,.2,;-4.66,-1.1,;-3.94,-2.46,;-2.4,-2.51,;-1.59,-1.2,;-.05,-1.25,;.76,.06,;.04,1.42,;-1.5,1.47,;-2.31,.16,;2.86,.12,;3,-1.51,;3.73,2.06,;4.36,3.57,;5.34,2.46,;2.95,3.48,;4.64,-.48,;6.26,-.96,;5.97,.54,;5.03,-2.06,;-3.82,2,;-3.67,3.74,;-5.62,2.37,;-2.12,1.52,;-1.18,2.74,;.35,2.53,;1.05,.92,;2.51,1.37,;-.01,-.11,;-1.54,.1,)|
C[C@]1(O)C[C@@H](C1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:13.15,1.1,wD:12.35,9.9,4.6,1.0,(-11.96,-5.2,;-11.62,-3.61,;-13.25,-3.68,;-11.5,-2.08,;-9.96,-2.2,;-10.09,-3.74,;-8.96,-.99,;-9.91,.28,;-7.49,-1.61,;-6.16,-.74,;-6.27,.8,;-4.85,1.38,;-3.85,.2,;-4.66,-1.1,;-3.94,-2.46,;-2.4,-2.51,;-1.59,-1.2,;-.05,-1.25,;.76,.06,;.04,1.42,;-1.5,1.47,;-2.31,.16,;2.86,.12,;3,-1.51,;3.73,2.06,;4.36,3.57,;5.34,2.46,;2.95,3.48,;4.64,-.48,;6.26,-.96,;5.97,.54,;5.03,-2.06,;-3.82,2,;-3.67,3.74,;-5.62,2.37,;-2.12,1.52,;-1.18,2.74,;.35,2.53,;1.05,.92,;2.51,1.37,;-.01,-.11,;-1.54,.1,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H](NC(=O)[C@@H]3CNC(=O)C3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H](NC(=O)[C@H]3CNC(=O)C3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H](NC(=O)[C@@H]3CC(=O)N3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H](NC(=O)C3CCNC(=O)C3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H](NC(=O)C3CCC(=O)NC3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
Cn1ccc(cc1=O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC1(CC(=O)N[C@@H]2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)CCS(=O)(=O)C1 |r,w:1.0|
CC(=O)NCC(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)NC(C)(C)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(C(O)=O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H](NC(=O)c3ccc(=O)[nH]c3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
Cn1cc(ccc1=O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H](NC(=O)c3cc[nH]c(=O)c3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
OC(=O)[C@H]1CC[C@@](O)(CC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:17.19,3.2,6.6,wD:13.13,6.10,16.39,(-14.46,-.42,;-13.69,-1.75,;-14.45,-3.08,;-12.15,-1.74,;-11.38,-.41,;-9.84,-.4,;-9.07,-1.73,;-8.07,-3.01,;-9.83,-3.07,;-11.37,-3.07,;-7.96,-.54,;-8.28,1.02,;-6.52,-1.2,;-5.27,-.26,;-5.38,1.27,;-3.95,1.85,;-2.96,.68,;-3.77,-.63,;-3.04,-1.99,;-1.5,-2.04,;-.69,-.73,;.85,-.77,;1.66,.53,;.93,1.89,;-.61,1.94,;-1.42,.63,;3.57,.08,;4.19,1.65,;5.34,-.14,;7,.14,;5.38,-1.95,;6.1,1.39,;4.29,-1.52,;4,-3.16,;6.19,-1.38,;3.42,-2.99,;-2.87,2.45,;-2.7,4.2,;-4.62,2.93,;-1.22,2,;-.28,3.21,;1.25,3,;1.83,1.58,;3.35,1.37,;.88,.36,;-.64,.57,)|
OC(=O)[C@H]1CC[C@@](F)(CC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:17.19,3.2,6.6,wD:16.39,13.13,6.10,(-14.86,-.93,;-13.86,-2.17,;-14.84,-3.42,;-12.23,-2.16,;-11.46,-.82,;-9.92,-.81,;-9.15,-2.14,;-8.14,-3.45,;-9.91,-3.48,;-11.45,-3.49,;-7.93,-1.06,;-8.31,.51,;-6.49,-1.73,;-5.35,-.68,;-5.46,.86,;-4.03,1.44,;-3.04,.27,;-3.85,-1.04,;-3.12,-2.4,;-1.58,-2.45,;-.77,-1.14,;.77,-1.19,;1.58,.12,;.85,1.48,;-.69,1.53,;-1.5,.22,;3.73,.27,;3.84,-1.36,;4.57,2.11,;5.33,3.63,;6.15,2.55,;3.89,3.65,;5.47,-.62,;7.03,-1.2,;6.84,.31,;5.82,-2.26,;-2.95,2.03,;-2.86,3.78,;-4.71,2.54,;-1.3,1.58,;-.36,2.8,;1.16,2.59,;1.86,.98,;3.39,1.44,;.8,-.05,;-.72,.16,)|
OC(=O)C12C3C4C1C1C2C3C41C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:18.24,wD:17.44,14.18,(7.74,6.28,;6.14,6.39,;5.56,7.89,;5.15,5.03,;4.09,3.44,;2.7,4.09,;3.75,5.68,;4.59,4.77,;5.99,4.12,;4.94,2.53,;3.54,3.18,;2.72,1.78,;3.81,.6,;1.14,2.12,;.2,.85,;.68,-.62,;-.57,-1.52,;-1.82,-.62,;-1.34,.85,;-2.37,1.99,;-3.88,1.67,;-4.35,.21,;-5.86,-.11,;-6.33,-1.58,;-5.3,-2.72,;-3.8,-2.4,;-3.32,-.94,;-8.38,-1.94,;-8.96,-.36,;-8.27,-3.94,;-7.94,-5.58,;-9.45,-5.15,;-6.64,-3.74,;-10.24,-1.93,;-11.94,-2.09,;-11.11,-3.39,;-11.15,-.54,;-1.42,-2.37,;-1.1,-4.09,;.44,-2.3,;-3.19,-2.31,;-3.81,-3.72,;-5.34,-3.88,;-6.4,-2.48,;-7.9,-2.89,;-5.62,-1.23,;-4.09,-1.07,)|
C[C@H]1C[C@@H](CC[C@H]1C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(O)=O |r|
OC1(CCNCC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(N)CC(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(N)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(N)[C@H](N)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(O)[C@@H](N)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(N1CCNCC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CS(=O)(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(O)COC(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(O)CNC(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC1(O)CN(C1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OCCNC(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CNC(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
O[C@H]1CN(C[C@H]1O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CNC(=O)CN(CC(=O)NC)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN(C)C(=O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN(C)C(=O)CN(CC(=O)N(C)C)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN(C)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H](NCc3ccccc3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
CC(C)(CO)CN[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H](Nc3ccccc3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
CN1C[C@H]2[C@@H](CC[C@]2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(=O)NCC(C)(C)O |r|
CN1C[C@H]2[C@@H](CC[C@]2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(=O)NC1CCN(CC1)S(C)(=O)=O |r|
CN1C[C@H]2[C@@H](CC[C@]2(c2ccc(cc12)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(=O)NCc1ccncc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H](NC(=O)Cc3ccncc3)[C@@H]1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
OC1(CCOCC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(O)CC(=O)N[C@@H]1CC[C@@]2([C@H]1CNc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(O)C(=O)NC[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(N)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(O)CN1C(C[C@@H](F)C1=O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(O)CN1N(CCC1=O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)OC1(CC(=O)N[C@@H]2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)CN(C1)C(C)=O |r|
OC(C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C1(O)CCOCC1 |r,w:1.0|
CC(C)(O)C(O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,w:4.4|
O[C@H]1C[C@H](C[C@H]1O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
O[C@H]1C[C@@H](C[C@H]1O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC[C@@]1(O)C[C@@H](C1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:14.16,2.1,wD:13.36,10.10,5.7,2.2,(-12.89,-5.05,;-12.33,-3.62,;-10.81,-3.38,;-11.29,-4.85,;-10.68,-1.85,;-9.14,-1.98,;-9.27,-3.51,;-7.97,-.98,;-8.24,.53,;-6.52,-1.5,;-5.34,-.51,;-5.45,1.03,;-4.03,1.61,;-3.03,.43,;-3.85,-.88,;-3.12,-2.23,;-1.58,-2.28,;-.77,-.97,;.77,-1.02,;1.58,.29,;.86,1.64,;-.68,1.69,;-1.49,.38,;3.12,.24,;3.07,-1.3,;3.17,1.78,;3.22,3.32,;4.71,1.73,;1.63,1.83,;4.66,.19,;6.2,.14,;5.61,1.41,;4.61,-1.35,;-2.36,1.82,;-3.75,2.49,;-1.01,2.55,;-1.69,3.21,;-2.56,4.48,;-1.89,5.87,;-.35,5.98,;.32,7.36,;.51,4.7,;-.16,3.32,)|
OC[C@]1(O)C[C@@H](C1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:14.16,2.2,wD:13.36,10.10,5.7,2.1,(-12.89,-5.05,;-12.33,-3.62,;-10.81,-3.38,;-11.29,-4.85,;-10.68,-1.85,;-9.14,-1.98,;-9.27,-3.51,;-7.97,-.98,;-8.24,.53,;-6.52,-1.5,;-5.34,-.51,;-5.45,1.03,;-4.03,1.61,;-3.03,.43,;-3.85,-.88,;-3.12,-2.23,;-1.58,-2.28,;-.77,-.97,;.77,-1.02,;1.58,.29,;.86,1.64,;-.68,1.69,;-1.49,.38,;3.12,.24,;3.07,-1.3,;3.17,1.78,;3.22,3.32,;4.71,1.73,;1.63,1.83,;4.66,.19,;6.2,.14,;5.61,1.41,;4.61,-1.35,;-2.36,1.82,;-3.75,2.49,;-1.01,2.55,;-1.69,3.21,;-2.56,4.48,;-1.89,5.87,;-.35,5.98,;.32,7.36,;.51,4.7,;-.16,3.32,)|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)N1CCC(C1=O)c1ccncc1 |r,w:36.43|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@H]([C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)N1CCOC1=O |r|
CC1(NC(=O)NC1=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(O)C[C@H]1NC(=O)N([C@@H]2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)C1=O |r|
CC(=O)N[C@H]1C[C@H](C1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:15.17,wD:14.37,11.11,6.8,4.3,(-15.05,-5.15,;-13.87,-4.16,;-14.14,-2.64,;-12.42,-4.68,;-11.24,-3.68,;-9.71,-3.81,;-9.58,-2.28,;-11.12,-2.15,;-8.4,-1.28,;-6.96,-1.81,;-6.68,-3.32,;-5.78,-.81,;-5.89,.72,;-4.47,1.31,;-3.47,.13,;-4.28,-1.18,;-3.56,-2.54,;-2.02,-2.58,;-1.21,-1.27,;.33,-1.32,;1.14,-.01,;.42,1.34,;-1.12,1.39,;-1.93,.08,;2.68,-.06,;4.22,-.11,;2.64,-1.6,;2.59,-3.14,;1.1,-1.55,;4.18,-1.65,;2.73,1.48,;2.78,3.02,;1.19,1.53,;4.27,1.43,;-2.8,1.52,;-4.19,2.19,;-1.45,2.25,;-2.13,2.9,;-3,4.18,;-2.33,5.56,;-.79,5.68,;-.12,7.06,;.07,4.4,;-.6,3.02,)|
CC(=O)N1CCC(O)(CC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(NC(=O)c1cn(cn1)C(=O)C(F)(F)F)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(NC(=O)C(C)(C)N)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N[C@H]1C[C@@H](C1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:15.17,4.3,wD:14.37,11.11,6.8,(-15.51,-4.45,;-14.33,-3.45,;-14.6,-1.94,;-12.88,-3.97,;-11.7,-2.98,;-11.58,-1.44,;-10.04,-1.57,;-10.17,-3.11,;-8.87,-.53,;-7.41,-1.25,;-7.26,-2.87,;-6.24,-.11,;-6.35,1.43,;-4.93,2.01,;-3.93,.84,;-4.74,-.47,;-4.02,-1.83,;-2.48,-1.88,;-1.67,-.57,;-.13,-.62,;.69,.69,;-.04,2.05,;-1.58,2.1,;-2.39,.79,;2.54,.23,;3.15,1.76,;4.31,.53,;6.03,.62,;4.74,-1.04,;5.06,2.08,;2.69,-1.54,;2.96,-3.2,;4.37,-1.44,;1.49,-2.77,;-3.88,2.6,;-3.74,4.32,;-5.66,2.98,;-2.2,2.15,;-1.25,3.37,;.27,3.16,;.85,1.74,;2.38,1.53,;-.09,.52,;-1.62,.73,)|
CC(=O)N1CCC(CNC(=O)[C@@H]2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)C1 |r|
OCC(=O)N[C@H]1C[C@@H](C1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:16.18,5.4,wD:15.38,12.12,7.9,(-16.86,-3.87,;-15.41,-4.39,;-14.23,-3.4,;-14.5,-1.88,;-12.78,-3.92,;-11.61,-2.92,;-11.48,-1.39,;-9.94,-1.52,;-10.07,-3.05,;-8.77,-.47,;-7.31,-1.21,;-7.09,-2.84,;-6.14,-.05,;-6.25,1.48,;-4.83,2.07,;-3.83,.89,;-4.65,-.42,;-3.92,-1.78,;-2.38,-1.82,;-1.57,-.52,;-.03,-.56,;.78,.75,;.06,2.1,;-1.48,2.15,;-2.29,.84,;2.65,.25,;3.21,1.88,;4.4,.47,;6.05,.48,;4.99,-1.06,;5.16,1.96,;2.84,-1.59,;3.06,-3.3,;4.56,-1.51,;1.58,-2.66,;-3.79,2.67,;-3.66,4.41,;-5.61,3.03,;-2.1,2.21,;-1.16,3.42,;.37,3.22,;.95,1.79,;2.48,1.58,;.01,.57,;-1.52,.78,)|
OCC(=O)N[C@H]1C[C@H](C1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:16.18,wD:15.38,12.12,7.9,5.4,(-16.86,-3.87,;-15.41,-4.39,;-14.23,-3.4,;-14.5,-1.88,;-12.78,-3.92,;-11.61,-2.92,;-10.07,-3.05,;-9.94,-1.52,;-11.48,-1.39,;-8.77,-.47,;-7.31,-1.21,;-7.09,-2.84,;-6.14,-.05,;-6.25,1.48,;-4.83,2.07,;-3.83,.89,;-4.65,-.42,;-3.92,-1.78,;-2.38,-1.82,;-1.57,-.52,;-.03,-.56,;.78,.75,;.06,2.1,;-1.48,2.15,;-2.29,.84,;2.65,.25,;3.21,1.88,;4.4,.47,;6.05,.48,;4.99,-1.06,;5.16,1.96,;2.84,-1.59,;3.06,-3.3,;4.56,-1.51,;1.58,-2.66,;-3.79,2.67,;-3.66,4.41,;-5.61,3.03,;-2.1,2.21,;-1.16,3.42,;.37,3.22,;.95,1.79,;2.48,1.58,;.01,.57,;-1.52,.78,)|
OCC(=O)N1CCC(CNC(=O)[C@@H]2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)C1 |r|
OCC(=O)N1CCC(O)(CC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(NC(=O)c1c[nH]cn1)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
[#6]-[#6](\[#7]=[#6](\[#7](-[#6])-[#6])-[#7](-[#6])-[#6])-[#6@@H]-1-[#6]-[#6][C@@]2([#6@H]-1-[#6]-[#6]-c1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(NC(=O)c1ccon1)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(NC(=O)c1ccncn1)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(NC(=O)c1ccncc1)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(NC(=O)C(C)(C)O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(NC(=O)[C@@H]1C[C@@H](F)C(=O)N1)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@@H](O)C(=O)NC(C)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@H](O)C(=O)NC(C)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@H](N)C(=O)NC(C)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(NS(=O)(=O)c1cnn(C)c1)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(NS(=O)(=O)c1nc[nH]n1)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CS(=O)(=O)N[C@H]1C[C@@H](C1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:16.18,5.4,wD:15.38,12.12,7.9,(-12.53,-7.32,;-11,-7.16,;-10.83,-8.69,;-9.47,-7,;-11.16,-5.6,;-9.96,-4.56,;-9.84,-3.03,;-8.3,-3.16,;-8.43,-4.69,;-7.59,-1.77,;-7.74,-.2,;-9.26,.31,;-6.22,.35,;-6.33,1.88,;-4.91,2.47,;-3.91,1.29,;-4.73,-.02,;-4,-1.38,;-2.46,-1.42,;-1.65,-.11,;-.11,-.16,;.7,1.15,;-.02,2.5,;-1.56,2.55,;-2.38,1.24,;2.74,.9,;4.29,.27,;3.2,-.94,;3.66,-2.6,;2.19,-2.29,;4.83,-1.46,;3.81,2.67,;4.83,4.06,;3.3,4.28,;5.55,2.61,;-3.86,3.06,;-3.79,4.79,;-5.66,3.42,;-2.18,2.61,;-1.24,3.82,;.29,3.62,;.98,2,;2.52,2.19,;-.07,.97,;-1.6,1.18,)|
CS(=O)(=O)N1CCC(CNC(=O)[C@@H]2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)C1 |r|
CS(=O)(=O)N1CC(O)(CNC(=O)[C@@H]2CC[C@@]3([C@H]2CCc2cc(ccc32)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)C1 |r|
NS(=O)(=O)N[C@@H]1C[C@@H](C1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:16.18,wD:15.38,12.12,7.9,5.4,(-13.36,-2.12,;-13.79,-3.6,;-15.27,-3.18,;-14.21,-5.08,;-12.29,-4.03,;-11.06,-3.02,;-10.93,-1.49,;-9.4,-1.62,;-9.52,-3.15,;-8.18,-.64,;-6.73,-1.29,;-6.51,-2.87,;-5.59,-.15,;-5.71,1.38,;-4.28,1.97,;-3.29,.79,;-4.1,-.52,;-3.37,-1.88,;-1.83,-1.92,;-1.02,-.62,;.52,-.66,;1.33,.65,;.6,2,;-.94,2.05,;-1.75,.74,;3.25,.19,;4.86,-.29,;3.7,-1.63,;4.16,-3.28,;2.63,-2.94,;5.33,-2.09,;3.85,2.13,;4.21,3.82,;2.15,2.58,;5.48,2.7,;-3.24,2.57,;-3.19,4.31,;-5.05,2.91,;-1.55,2.11,;-.61,3.32,;.92,3.12,;1.61,1.5,;3.15,1.3,;.55,.47,;-.97,.68,)|
NS(=O)(=O)N[C@@H]1C[C@@H](C1)NC(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:16.18,wD:15.38,12.12,7.9,5.4,(-13.59,-2.03,;-13.97,-3.52,;-15.46,-3.14,;-14.35,-5.01,;-12.45,-3.91,;-11.23,-2.9,;-11.1,-1.36,;-9.56,-1.49,;-9.69,-3.03,;-8.34,-.52,;-6.88,-1.17,;-6.63,-2.75,;-5.76,-.02,;-5.87,1.51,;-4.45,2.09,;-3.45,.92,;-4.27,-.39,;-3.54,-1.75,;-2,-1.8,;-1.19,-.49,;.35,-.54,;1.16,.77,;.44,2.13,;-1.1,2.18,;-1.92,.87,;3.2,.33,;3.54,2.2,;5.16,.37,;6.88,.42,;5.84,-1.2,;6.07,1.83,;3.37,-1.55,;3.72,-3.22,;4.98,-2.08,;2.17,-2.76,;-3.42,2.7,;-3.34,4.43,;-5.23,3.04,;-1.72,2.23,;-.78,3.45,;.75,3.24,;1.33,1.82,;2.84,1.48,;.39,.6,;-1.14,.81,)|
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CC(C)(OP(O)(O)=O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN1N(CCC1=O)C(=O)[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN1C[C@H](CC1=O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN1C[C@@H](CC1=O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OCCN1C[C@H](CC1=O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN1CCC(O)(CC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC1(CCN(CC1)C1COC1)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(O)CN1C[C@H](CC1=O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)(O)CN1C[C@@H](CC1=O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H](NC(=O)[C@@H]3CN(CCC#N)C(=O)C3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
OC(=O)CCN1C[C@H](CC1=O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OCCCN1C[C@H](CC1=O)C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@@]12CC[C@@H](NC(=O)C3(F)CCS(=O)(=O)CC3)[C@@H]1CCc1cc(ccc21)C(F)(C(F)(F)F)C(F)(F)F |r|
FC(F)(F)C(F)(c1ccc2c(CC[C@H]3[C@@H](CC[C@@]23S(=O)(=O)c2ccccc2)NC(=O)C2CCS(=O)(=O)CC2)c1)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)C12C(CNC(=O)Cc3ccncc3)C1CCc1cc(I)ccc21 |w:11.12|
OC(c1ccc2c(CCC3C(CNC(=O)Cc4ccncc4)C23S(=O)(=O)c2ccc(F)cc2)c1)(C(F)(F)F)C(F)(F)F |w:10.10|
Fc1ccc(cc1)S(=O)(=O)C12CC(NC(=O)Cc3ccncc3)C1CCc1cc(I)ccc21 |w:12.13|
CC(C)(O)C(=O)NCC1C2CCc3cc(I)ccc3C12S(=O)(=O)c1ccc(F)cc1 |w:8.7|
CCn1c(Cc2ccc(cc2)C(F)(F)F)cc2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCn1c(Cc2ccc(cc2)C(F)(F)F)cc2cc(ccc12)C(=O)NCc1ccc(cn1)S(=O)(=O)CC
CCn1c(Cc2ccc(cc2)C(F)(F)F)cc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cc1)S(=O)(=O)CC |r|
CCn1c(Cc2ccc(cc2)C(F)(F)F)cc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cn1)S(=O)(=O)CC |r|
CCn1c(Cc2ccc(cc2)C(F)(F)F)cc2cc(ccc12)C(=O)N[C@H](CO)c1ccc(cn1)S(=O)(=O)CC |r|
CCn1c(Cc2ccc3OC(F)(F)Oc3c2)cc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cn1)S(=O)(=O)CC |r|
CCn1c(Cc2ccc(OC(F)F)cc2)cc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cn1)S(=O)(=O)CC |r|
CCn1c(Cc2cccc(OC(F)F)c2)cc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cn1)S(=O)(=O)CC |r|
CCn1c(Cc2ccc(Cl)cc2)cc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cn1)S(=O)(=O)CC |r|
CCn1c(Cc2ccc(cn2)C(F)(F)F)cc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cc1)S(=O)(=O)CC |r|
CCn1c(CN2CCC(CC2)C(F)(F)F)cc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cc1)S(=O)(=O)CC |r|
CCn1c(CN2CCC(CC2)C(F)(F)F)cc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cn1)S(=O)(=O)CC
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(CN4CCC(CC4)C(F)(F)F)cc3c2)cc1
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(CN3CCC(CC3)C(F)(F)F)cc2c1
CCn1c(C[C@H]2CC[C@@H](CC2)C(F)(F)F)cc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cn1)S(=O)(=O)CC |wU:5.4,wD:8.11,25.27,(-5.85,6.52,;-7.36,6.2,;-7.84,4.74,;-6.93,3.49,;-5.39,3.49,;-4.62,2.16,;-3.08,2.16,;-2.31,.82,;-3.08,-.51,;-4.62,-.51,;-5.39,.82,;-2.31,-1.85,;-3.08,-3.18,;-1.54,-3.18,;-.77,-1.85,;-7.84,2.24,;-9.3,2.72,;-10.63,1.95,;-11.97,2.72,;-11.97,4.26,;-10.63,5.03,;-9.3,4.26,;-13.3,1.95,;-13.3,.41,;-14.63,2.72,;-15.97,1.95,;-17.3,2.72,;-18.64,1.95,;-15.97,.41,;-14.63,-.36,;-14.63,-1.9,;-15.97,-2.67,;-17.3,-1.9,;-17.3,-.36,;-15.97,-4.21,;-17.51,-4.21,;-14.43,-4.21,;-15.97,-5.75,;-17.3,-6.52,)|
CCn1c(C[C@H]2CC[C@@H](CC2)C(F)(F)F)cc2cc(ccc12)C(=O)NCc1ccc(cn1)S(=O)(=O)CC |wU:5.4,wD:8.11,(6.52,10.47,;5.01,10.15,;4.53,8.68,;5.44,7.44,;6.98,7.44,;7.75,6.1,;9.29,6.1,;10.06,4.77,;9.29,3.44,;7.75,3.44,;6.98,4.77,;10.06,2.1,;9.29,.77,;10.83,.77,;11.6,2.1,;4.53,6.19,;3.07,6.67,;1.74,5.9,;.4,6.67,;.4,8.21,;1.74,8.98,;3.07,8.21,;-.93,5.9,;-.93,4.36,;-2.26,6.67,;-3.6,5.9,;-4.93,6.67,;-6.27,5.9,;-7.6,6.67,;-7.6,8.21,;-6.27,8.98,;-4.93,8.21,;-8.93,8.98,;-8.16,10.31,;-9.7,7.64,;-10.27,9.75,;-11.6,8.98,)|
CCn1c(C[C@H]2CC[C@@H](CC2)C(F)(F)F)cc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cc1)S(=O)(=O)CC |wU:5.4,wD:8.11,25.27,(-5.85,6.52,;-7.36,6.2,;-7.84,4.74,;-6.93,3.49,;-5.39,3.49,;-4.62,2.16,;-3.08,2.16,;-2.31,.82,;-3.08,-.51,;-4.62,-.51,;-5.39,.82,;-2.31,-1.85,;-3.08,-3.18,;-1.54,-3.18,;-.77,-1.85,;-7.84,2.24,;-9.3,2.72,;-10.63,1.95,;-11.97,2.72,;-11.97,4.26,;-10.63,5.03,;-9.3,4.26,;-13.3,1.95,;-13.3,.41,;-14.63,2.72,;-15.97,1.95,;-17.3,2.72,;-18.64,1.95,;-15.97,.41,;-14.63,-.36,;-14.63,-1.9,;-15.97,-2.67,;-17.3,-1.9,;-17.3,-.36,;-15.97,-4.21,;-17.51,-4.21,;-14.43,-4.21,;-15.97,-5.75,;-17.3,-6.52,)|
CCn1c(C[C@H]2CC[C@@H](CC2)C(F)(F)F)cc2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC |wU:5.4,wD:8.11,(6.52,10.47,;5.01,10.15,;4.53,8.68,;5.44,7.44,;6.98,7.44,;7.75,6.1,;9.29,6.1,;10.06,4.77,;9.29,3.44,;7.75,3.44,;6.98,4.77,;10.06,2.1,;9.29,.77,;10.83,.77,;11.6,2.1,;4.53,6.19,;3.07,6.67,;1.74,5.9,;.4,6.67,;.4,8.21,;1.74,8.98,;3.07,8.21,;-.93,5.9,;-.93,4.36,;-2.26,6.67,;-3.6,5.9,;-4.93,6.67,;-6.27,5.9,;-7.6,6.67,;-7.6,8.21,;-6.27,8.98,;-4.93,8.21,;-8.93,8.98,;-8.16,10.31,;-9.7,7.64,;-10.27,9.75,;-11.6,8.98,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(Cc4ccc(cc4)C(F)(F)F)cc3c2)cc1
CCS(=O)(=O)c1ccc(nc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(Cc3ccc(cc3)C(F)(F)F)cc2c1
CCn1c(Cc2ccc(cc2)C(N)=O)cc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cn1)S(=O)(=O)CC
CCn1c(Cc2ccc(cc2)C#N)cc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cn1)S(=O)(=O)CC |r|
CCn1c(cc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cn1)S(=O)(=O)CC)C(=O)c1ccc(cn1)C(F)(F)F |r|
CCn1c(cc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cc1)S(=O)(=O)CC)C(O)c1ccc(cn1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3n(C4CC4)c(CC4CC[C@@H](CC4)C(F)(F)F)cc3c2)cc1 |r,wD:26.30,(5.51,-31.31,;4.18,-32.08,;2.84,-31.31,;2.07,-32.64,;3.61,-29.98,;1.51,-30.54,;.13,-31.28,;-1.21,-30.51,;-1.21,-28.97,;-2.54,-28.2,;-3.87,-28.97,;-5.21,-28.2,;-5.21,-26.66,;-6.54,-28.97,;-6.54,-30.51,;-7.88,-31.28,;-9.21,-30.51,;-10.67,-30.99,;-11.07,-32.47,;-12.16,-33.56,;-10.67,-33.96,;-11.58,-29.74,;-13.07,-30.14,;-13.84,-28.81,;-15.38,-28.81,;-16.15,-27.47,;-15.38,-26.14,;-13.84,-26.14,;-13.07,-27.47,;-16.15,-24.81,;-15.38,-23.47,;-17.69,-24.81,;-16.92,-23.47,;-10.67,-28.5,;-9.21,-28.97,;-7.88,-28.2,;.13,-28.2,;1.46,-28.97,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1cnc2n(C3CC3)c(C[C@H]3CC[C@@H](CC3)C(F)(F)F)cc2c1 |wU:27.28,wD:30.35,11.14,(-7.6,-7.11,;-6.27,-6.34,;-6.27,-4.8,;-7.81,-4.8,;-4.73,-4.8,;-6.27,-3.26,;-4.93,-2.49,;-4.93,-.95,;-6.27,-.18,;-7.6,-.95,;-7.6,-2.49,;-6.27,1.36,;-7.6,2.13,;-8.93,1.36,;-4.93,2.13,;-3.6,1.36,;-3.6,-.18,;-2.26,2.13,;-2.26,3.67,;-.93,4.44,;.4,3.67,;1.87,4.14,;2.34,5.61,;2.02,7.11,;3.49,6.64,;2.77,2.9,;4.31,2.9,;5.08,1.56,;6.62,1.56,;7.39,.23,;6.62,-1.1,;5.08,-1.1,;4.31,.23,;7.39,-2.44,;6.62,-3.77,;8.16,-3.77,;8.93,-2.44,;1.87,1.65,;.4,2.13,;-.93,1.36,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3n(CC(C)=C)c(Cc4ccc(cc4)C(F)(F)F)cc3c2)cc1
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(O[C@H]3CC[C@H](CC3)C(F)(F)F)nc2c1 |r,wU:27.28,30.35,11.14,(11.98,-30.44,;10.65,-31.21,;9.31,-30.44,;8.54,-31.77,;10.08,-29.11,;7.98,-29.67,;6.6,-30.41,;5.26,-29.64,;5.26,-28.1,;6.6,-27.33,;7.93,-28.1,;3.93,-27.33,;3.93,-25.79,;5.26,-25.02,;2.6,-28.1,;1.26,-27.33,;1.26,-25.79,;-.07,-28.1,;-.07,-29.64,;-1.4,-30.41,;-2.74,-29.64,;-4.2,-30.12,;-4.6,-31.61,;-5.69,-32.7,;-4.2,-33.09,;-5.11,-28.87,;-6.65,-28.87,;-7.42,-27.54,;-8.96,-27.54,;-9.73,-26.21,;-8.96,-24.87,;-7.42,-24.87,;-6.65,-26.21,;-9.73,-23.54,;-8.96,-22.2,;-11.27,-23.54,;-10.5,-22.2,;-4.2,-27.63,;-2.74,-28.1,;-1.4,-27.33,)|
CCn1c(O[C@H]2CC[C@@H](CC2)C(F)(F)F)nc2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC |wU:5.4,wD:8.11,(6.52,4.85,;5.01,4.53,;4.53,3.06,;5.44,1.82,;6.98,1.82,;7.75,.49,;9.29,.49,;10.06,-.85,;9.29,-2.18,;7.75,-2.18,;6.98,-.85,;10.06,-3.52,;9.29,-4.85,;10.83,-4.85,;11.6,-3.52,;4.53,.57,;3.07,1.05,;1.74,.28,;.4,1.05,;.4,2.59,;1.74,3.36,;3.07,2.59,;-.93,.28,;-.93,-1.26,;-2.26,1.05,;-3.6,.28,;-4.93,1.05,;-6.27,.28,;-7.6,1.05,;-7.6,2.59,;-6.27,3.36,;-4.93,2.59,;-8.93,3.36,;-8.16,4.69,;-9.7,2.03,;-10.27,4.13,;-11.6,3.36,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(O[C@H]4CC[C@@H](CC4)C(F)(F)F)nc3c2)cc1 |wU:23.23,wD:26.30,(-11.6,2.77,;-10.27,3.54,;-8.93,2.77,;-8.16,4.1,;-9.7,1.43,;-7.6,2,;-7.6,.46,;-6.27,-.31,;-4.93,.46,;-3.6,-.31,;-2.26,.46,;-.93,-.31,;-.93,-1.85,;.4,.46,;.4,2,;1.74,2.77,;3.07,2,;4.53,2.47,;5.01,3.94,;4.69,5.44,;6.16,4.97,;5.44,1.23,;6.98,1.23,;7.75,-.11,;9.29,-.11,;10.06,-1.44,;9.29,-2.78,;7.75,-2.78,;6.98,-1.44,;10.06,-4.11,;9.29,-5.44,;10.83,-5.44,;11.6,-4.11,;4.53,-.02,;3.07,.46,;1.74,-.31,;-4.93,2,;-6.27,2.77,)|
CCC(C)n1c(O[C@H]2CC[C@@H](CC2)C(F)(F)F)nc2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC |wU:7.6,wD:10.13,(2.47,4.76,;3.98,5.08,;5.01,3.94,;6.52,4.26,;4.53,2.47,;5.44,1.23,;6.98,1.23,;7.75,-.11,;9.29,-.11,;10.06,-1.44,;9.29,-2.78,;7.75,-2.78,;6.98,-1.44,;10.06,-4.11,;9.29,-5.44,;10.83,-5.44,;11.6,-4.11,;4.53,-.02,;3.07,.46,;1.74,-.31,;.4,.46,;.4,2,;1.74,2.77,;3.07,2,;-.93,-.31,;-.93,-1.85,;-2.26,.46,;-3.6,-.31,;-4.93,.46,;-6.27,-.31,;-7.6,.46,;-7.6,2,;-6.27,2.77,;-4.93,2,;-8.93,2.77,;-8.16,4.1,;-9.7,1.43,;-10.27,3.54,;-11.6,2.77,)|
CCC(C)n1c(O[C@H]2CC[C@H](CC2)C(F)(F)F)nc2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC |wU:10.13,7.6,(2.47,4.76,;3.98,5.08,;5.01,3.94,;6.52,4.26,;4.53,2.47,;5.44,1.23,;6.98,1.23,;7.75,-.11,;9.29,-.11,;10.06,-1.44,;9.29,-2.78,;7.75,-2.78,;6.98,-1.44,;10.06,-4.11,;9.29,-5.44,;10.83,-5.44,;11.6,-4.11,;4.53,-.02,;3.07,.46,;1.74,-.31,;.4,.46,;.4,2,;1.74,2.77,;3.07,2,;-.93,-.31,;-.93,-1.85,;-2.26,.46,;-3.6,-.31,;-4.93,.46,;-6.27,-.31,;-7.6,.46,;-7.6,2,;-6.27,2.77,;-4.93,2,;-8.93,2.77,;-8.16,4.1,;-9.7,1.43,;-10.27,3.54,;-11.6,2.77,)|
CCn1c(Oc2ccc(cc2)C(F)(F)F)nc2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(Oc4ccc(cc4)C(F)(F)F)nc3c2)cc1
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(Oc3ccc(cc3)C(F)(F)F)nc2c1
CCn1c(Oc2ccc(cc2)C(F)(F)F)nc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cc1)S(=O)(=O)CC
CCn1c(Oc2ccc(OC(F)(F)F)cc2)nc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cc1)S(=O)(=O)CC
CCn1c(Oc2ccc(cc2)C(F)(F)F)nc2cc(ccc12)C(=O)N[C@@H](CN(C)C)c1ccc(cc1)S(=O)(=O)CC
CCn1c(Oc2ccc(cc2)C(F)(F)F)nc2cc(ccc12)C(=O)N[C@@H](CN)c1ccc(cc1)S(=O)(=O)CC
CCn1c(OCC2CCC(F)(F)CC2)nc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cc1)S(=O)(=O)CC
CCn1c(OCC2CC(F)(F)C2)nc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cc1)S(=O)(=O)CC
CCn1c(OCc2ccc(cc2)C(F)(F)F)nc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cc1)S(=O)(=O)CC
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(OCc3ccc(cc3)C(F)(F)F)nc2c1
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(OCC3CCC(F)(F)CC3)nc2c1
CCn1c(OCC2CC2)nc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cc1)S(=O)(=O)CC
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(C[C@H]4CC[C@@H](CC4)C(F)(F)F)nc3c2)cc1 |wU:23.23,wD:26.30,(-11.6,8.98,;-10.27,9.75,;-8.93,8.98,;-8.16,10.31,;-9.7,7.64,;-7.6,8.21,;-7.6,6.67,;-6.27,5.9,;-4.93,6.67,;-3.6,5.9,;-2.26,6.67,;-.93,5.9,;-.93,4.36,;.4,6.67,;.4,8.21,;1.74,8.98,;3.07,8.21,;4.53,8.68,;5.01,10.15,;4.69,11.66,;6.16,11.18,;5.44,7.44,;6.98,7.44,;7.75,6.1,;9.29,6.1,;10.06,4.77,;9.29,3.44,;7.75,3.44,;6.98,4.77,;10.06,2.1,;9.29,.77,;10.83,.77,;11.6,2.1,;4.53,6.19,;3.07,6.67,;1.74,5.9,;-4.93,8.21,;-6.27,8.98,)|
CCC(C)n1c(C[C@H]2CC[C@@H](CC2)C(F)(F)F)nc2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC |wU:7.6,wD:10.13,(2.47,4.76,;3.98,5.08,;5.01,3.94,;6.52,4.26,;4.53,2.47,;5.44,1.23,;6.98,1.23,;7.75,-.11,;9.29,-.11,;10.06,-1.44,;9.29,-2.78,;7.75,-2.78,;6.98,-1.44,;10.06,-4.11,;9.29,-5.44,;10.83,-5.44,;11.6,-4.11,;4.53,-.02,;3.07,.46,;1.74,-.31,;.4,.46,;.4,2,;1.74,2.77,;3.07,2,;-.93,-.31,;-.93,-1.85,;-2.26,.46,;-3.6,-.31,;-4.93,.46,;-6.27,-.31,;-7.6,.46,;-7.6,2,;-6.27,2.77,;-4.93,2,;-8.93,2.77,;-8.16,4.1,;-9.7,1.43,;-10.27,3.54,;-11.6,2.77,)|
CCC(C)n1c(C[C@H]2CC[C@H](CC2)C(F)(F)F)nc2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC |wU:10.13,7.6,(2.47,4.76,;3.98,5.08,;5.01,3.94,;6.52,4.26,;4.53,2.47,;5.44,1.23,;6.98,1.23,;7.75,-.11,;9.29,-.11,;10.06,-1.44,;9.29,-2.78,;7.75,-2.78,;6.98,-1.44,;10.06,-4.11,;9.29,-5.44,;10.83,-5.44,;11.6,-4.11,;4.53,-.02,;3.07,.46,;1.74,-.31,;.4,.46,;.4,2,;1.74,2.77,;3.07,2,;-.93,-.31,;-.93,-1.85,;-2.26,.46,;-3.6,-.31,;-4.93,.46,;-6.27,-.31,;-7.6,.46,;-7.6,2,;-6.27,2.77,;-4.93,2,;-8.93,2.77,;-8.16,4.1,;-9.7,1.43,;-10.27,3.54,;-11.6,2.77,)|
CCn1c(C[C@H]2CC[C@@H](CC2)C(F)(F)F)nc2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC |wU:5.4,wD:8.11,(6.52,4.85,;5.01,4.53,;4.53,3.06,;5.44,1.82,;6.98,1.82,;7.75,.49,;9.29,.49,;10.06,-.85,;9.29,-2.18,;7.75,-2.18,;6.98,-.85,;10.06,-3.52,;9.29,-4.85,;10.83,-4.85,;11.6,-3.52,;4.53,.57,;3.07,1.05,;1.74,.28,;.4,1.05,;.4,2.59,;1.74,3.36,;3.07,2.59,;-.93,.28,;-.93,-1.26,;-2.26,1.05,;-3.6,.28,;-4.93,1.05,;-6.27,.28,;-7.6,1.05,;-7.6,2.59,;-6.27,3.36,;-4.93,2.59,;-8.93,3.36,;-8.16,4.69,;-9.7,2.03,;-10.27,4.13,;-11.6,3.36,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(C[C@H]3CC[C@@H](CC3)C(F)(F)F)nc2c1 |wU:27.28,wD:30.35,11.14,(-7.6,-7.11,;-6.27,-6.34,;-6.27,-4.8,;-7.81,-4.8,;-4.73,-4.8,;-6.27,-3.26,;-4.93,-2.49,;-4.93,-.95,;-6.27,-.18,;-7.6,-.95,;-7.6,-2.49,;-6.27,1.36,;-7.6,2.13,;-8.93,1.36,;-4.93,2.13,;-3.6,1.36,;-3.6,-.18,;-2.26,2.13,;-2.26,3.67,;-.93,4.44,;.4,3.67,;1.87,4.14,;2.34,5.61,;2.02,7.11,;3.49,6.64,;2.77,2.9,;4.31,2.9,;5.08,1.56,;6.62,1.56,;7.39,.23,;6.62,-1.1,;5.08,-1.1,;4.31,.23,;7.39,-2.44,;6.62,-3.77,;8.16,-3.77,;8.93,-2.44,;1.87,1.65,;.4,2.13,;-.93,1.36,)|
CCS(=O)(=O)c1ccc(cc1)[C@@H](CO)NC(=O)c1ccc2n(C3CC3)c(C[C@H]3CC[C@@H](CC3)C(F)(F)F)nc2c1 |wU:27.28,11.14,wD:30.35,(-7.6,-7.11,;-6.27,-6.34,;-6.27,-4.8,;-7.81,-4.8,;-4.73,-4.8,;-6.27,-3.26,;-4.93,-2.49,;-4.93,-.95,;-6.27,-.18,;-7.6,-.95,;-7.6,-2.49,;-6.27,1.36,;-7.6,2.13,;-8.93,1.36,;-4.93,2.13,;-3.6,1.36,;-3.6,-.18,;-2.26,2.13,;-2.26,3.67,;-.93,4.44,;.4,3.67,;1.87,4.14,;2.34,5.61,;2.02,7.11,;3.49,6.64,;2.77,2.9,;4.31,2.9,;5.08,1.56,;6.62,1.56,;7.39,.23,;6.62,-1.1,;5.08,-1.1,;4.31,.23,;7.39,-2.44,;6.62,-3.77,;8.16,-3.77,;8.93,-2.44,;1.87,1.65,;.4,2.13,;-.93,1.36,)|
CCn1c(C[C@H]2CC[C@@H](CC2)C(F)(F)F)nc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cc1)S(=O)(=O)CC |wU:5.4,wD:8.11,25.27,(3.85,6.52,;2.34,6.2,;1.87,4.74,;2.77,3.49,;4.31,3.49,;5.08,2.16,;6.62,2.16,;7.39,.82,;6.62,-.51,;5.08,-.51,;4.31,.82,;7.39,-1.85,;6.62,-3.18,;8.16,-3.18,;8.93,-1.85,;1.87,2.24,;.4,2.72,;-.93,1.95,;-2.26,2.72,;-2.26,4.26,;-.93,5.03,;.4,4.26,;-3.6,1.95,;-3.6,.41,;-4.93,2.72,;-6.27,1.95,;-7.6,2.72,;-8.93,1.95,;-6.27,.41,;-4.93,-.36,;-4.93,-1.9,;-6.27,-2.67,;-7.6,-1.9,;-7.6,-.36,;-6.27,-4.21,;-7.81,-4.21,;-4.73,-4.21,;-6.27,-5.75,;-7.6,-6.52,)|
CCn1c(C[C@H]2CC[C@@H](CC2)C(F)(F)F)nc2cc(ccc12)C(=O)N[C@H](CO)c1ccc(cc1)S(=O)(=O)CC |wU:5.4,25.27,wD:8.11,(3.85,6.52,;2.34,6.2,;1.87,4.74,;2.77,3.49,;4.31,3.49,;5.08,2.16,;6.62,2.16,;7.39,.82,;6.62,-.51,;5.08,-.51,;4.31,.82,;7.39,-1.85,;6.62,-3.18,;8.16,-3.18,;8.93,-1.85,;1.87,2.24,;.4,2.72,;-.93,1.95,;-2.26,2.72,;-2.26,4.26,;-.93,5.03,;.4,4.26,;-3.6,1.95,;-3.6,.41,;-4.93,2.72,;-6.27,1.95,;-7.6,2.72,;-8.93,1.95,;-6.27,.41,;-4.93,-.36,;-4.93,-1.9,;-6.27,-2.67,;-7.6,-1.9,;-7.6,-.36,;-6.27,-4.21,;-7.81,-4.21,;-4.73,-4.21,;-6.27,-5.75,;-7.6,-6.52,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](CCO)NC(=O)c1ccc2n(C3CC3)c(C[C@H]3CC[C@@H](CC3)C(F)(F)F)nc2c1 |wU:28.29,wD:31.36,11.15,(6.93,7.11,;5.6,6.34,;5.6,4.8,;7.14,4.8,;4.06,4.8,;5.6,3.26,;4.26,2.49,;4.26,.95,;5.6,.18,;6.93,.95,;6.93,2.49,;5.6,-1.36,;6.93,-2.13,;8.27,-1.36,;9.6,-2.13,;4.26,-2.13,;2.93,-1.36,;2.93,.18,;1.6,-2.13,;1.6,-3.67,;.26,-4.44,;-1.07,-3.67,;-2.53,-4.14,;-3.01,-5.61,;-2.69,-7.11,;-4.15,-6.64,;-3.44,-2.9,;-4.98,-2.9,;-5.75,-1.56,;-7.29,-1.56,;-8.06,-.23,;-7.29,1.1,;-5.75,1.1,;-4.98,-.23,;-8.06,2.44,;-7.29,3.77,;-8.83,3.77,;-9.6,2.44,;-2.53,-1.65,;-1.07,-2.13,;.26,-1.36,)|
CCC(C)n1c(C[C@H]2CC[C@@H](CC2)C(F)(F)F)nc2cc(ccc12)C(=O)NCc1ccc(nc1)S(=O)(=O)CC |wU:7.6,wD:10.13,(2.47,4.76,;3.98,5.08,;5.01,3.94,;6.52,4.26,;4.53,2.47,;5.44,1.23,;6.98,1.23,;7.75,-.11,;9.29,-.11,;10.06,-1.44,;9.29,-2.78,;7.75,-2.78,;6.98,-1.44,;10.06,-4.11,;9.29,-5.44,;10.83,-5.44,;11.6,-4.11,;4.53,-.02,;3.07,.46,;1.74,-.31,;.4,.46,;.4,2,;1.74,2.77,;3.07,2,;-.93,-.31,;-.93,-1.85,;-2.26,.46,;-3.6,-.31,;-4.93,.46,;-4.93,2,;-6.27,2.77,;-7.6,2,;-7.6,.46,;-6.27,-.31,;-8.93,2.77,;-8.16,4.1,;-9.7,1.43,;-10.27,3.54,;-11.6,2.77,)|
CCC(C)n1c(C[C@H]2CC[C@H](CC2)C(F)(F)F)nc2cc(ccc12)C(=O)NCc1ccc(nc1)S(=O)(=O)CC |wU:10.13,7.6,(2.47,4.76,;3.98,5.08,;5.01,3.94,;6.52,4.26,;4.53,2.47,;5.44,1.23,;6.98,1.23,;7.75,-.11,;9.29,-.11,;10.06,-1.44,;9.29,-2.78,;7.75,-2.78,;6.98,-1.44,;10.06,-4.11,;9.29,-5.44,;10.83,-5.44,;11.6,-4.11,;4.53,-.02,;3.07,.46,;1.74,-.31,;.4,.46,;.4,2,;1.74,2.77,;3.07,2,;-.93,-.31,;-.93,-1.85,;-2.26,.46,;-3.6,-.31,;-4.93,.46,;-4.93,2,;-6.27,2.77,;-7.6,2,;-7.6,.46,;-6.27,-.31,;-8.93,2.77,;-8.16,4.1,;-9.7,1.43,;-10.27,3.54,;-11.6,2.77,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(C[C@H]4CC[C@@H](CC4)C(F)(F)F)nc3c2)nc1 |wU:23.23,wD:26.30,(-11.6,8.98,;-10.27,9.75,;-8.93,8.98,;-8.16,10.31,;-9.7,7.64,;-7.6,8.21,;-7.6,6.67,;-6.27,5.9,;-4.93,6.67,;-3.6,5.9,;-2.26,6.67,;-.93,5.9,;-.93,4.36,;.4,6.67,;.4,8.21,;1.74,8.98,;3.07,8.21,;4.53,8.68,;5.01,10.15,;4.69,11.66,;6.16,11.18,;5.44,7.44,;6.98,7.44,;7.75,6.1,;9.29,6.1,;10.06,4.77,;9.29,3.44,;7.75,3.44,;6.98,4.77,;10.06,2.1,;9.29,.77,;10.83,.77,;11.6,2.1,;4.53,6.19,;3.07,6.67,;1.74,5.9,;-4.93,8.21,;-6.27,8.98,)|
CCS(=O)(=O)c1ccc(nc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(C[C@H]3CC[C@@H](CC3)C(F)(F)F)nc2c1 |wU:27.28,wD:30.35,11.14,(-7.6,-7.11,;-6.27,-6.34,;-6.27,-4.8,;-7.81,-4.8,;-4.73,-4.8,;-6.27,-3.26,;-4.93,-2.49,;-4.93,-.95,;-6.27,-.18,;-7.6,-.95,;-7.6,-2.49,;-6.27,1.36,;-7.6,2.13,;-8.93,1.36,;-4.93,2.13,;-3.6,1.36,;-3.6,-.18,;-2.26,2.13,;-2.26,3.67,;-.93,4.44,;.4,3.67,;1.87,4.14,;2.34,5.61,;2.02,7.11,;3.49,6.64,;2.77,2.9,;4.31,2.9,;5.08,1.56,;6.62,1.56,;7.39,.23,;6.62,-1.1,;5.08,-1.1,;4.31,.23,;7.39,-2.44,;6.62,-3.77,;8.16,-3.77,;8.93,-2.44,;1.87,1.65,;.4,2.13,;-.93,1.36,)|
CCS(=O)(=O)c1ccc(nc1)[C@@H](CO)NC(=O)c1ccc2n(C3CC3)c(C[C@H]3CC[C@@H](CC3)C(F)(F)F)nc2c1 |wU:27.28,11.14,wD:30.35,(-7.6,-7.11,;-6.27,-6.34,;-6.27,-4.8,;-7.81,-4.8,;-4.73,-4.8,;-6.27,-3.26,;-4.93,-2.49,;-4.93,-.95,;-6.27,-.18,;-7.6,-.95,;-7.6,-2.49,;-6.27,1.36,;-7.6,2.13,;-8.93,1.36,;-4.93,2.13,;-3.6,1.36,;-3.6,-.18,;-2.26,2.13,;-2.26,3.67,;-.93,4.44,;.4,3.67,;1.87,4.14,;2.34,5.61,;2.02,7.11,;3.49,6.64,;2.77,2.9,;4.31,2.9,;5.08,1.56,;6.62,1.56,;7.39,.23,;6.62,-1.1,;5.08,-1.1,;4.31,.23,;7.39,-2.44,;6.62,-3.77,;8.16,-3.77,;8.93,-2.44,;1.87,1.65,;.4,2.13,;-.93,1.36,)|
CS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(C[C@H]4CC[C@@H](CC4)C(F)(F)F)nc3c2)cc1 |wU:22.22,wD:25.29,(-10.93,3.54,;-9.6,2.77,;-8.83,4.1,;-10.37,1.43,;-8.27,2,;-8.27,.46,;-6.93,-.31,;-5.6,.46,;-4.26,-.31,;-2.93,.46,;-1.6,-.31,;-1.6,-1.85,;-.26,.46,;-.26,2,;1.07,2.77,;2.4,2,;3.87,2.47,;4.34,3.94,;4.02,5.44,;5.49,4.97,;4.77,1.23,;6.31,1.23,;7.08,-.11,;8.62,-.11,;9.39,-1.44,;8.62,-2.78,;7.08,-2.78,;6.31,-1.44,;9.39,-4.11,;8.62,-5.44,;10.16,-5.44,;10.93,-4.11,;3.87,-.02,;2.4,.46,;1.07,-.31,;-5.6,2,;-6.93,2.77,)|
CNS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(C[C@H]4CC[C@@H](CC4)C(F)(F)F)nc3c2)nc1 |wU:23.23,wD:26.30,(-11.6,2.77,;-10.27,3.54,;-8.93,2.77,;-8.16,4.1,;-9.7,1.43,;-7.6,2,;-7.6,.46,;-6.27,-.31,;-4.93,.46,;-3.6,-.31,;-2.26,.46,;-.93,-.31,;-.93,-1.85,;.4,.46,;.4,2,;1.74,2.77,;3.07,2,;4.53,2.47,;5.01,3.94,;4.69,5.44,;6.16,4.97,;5.44,1.23,;6.98,1.23,;7.75,-.11,;9.29,-.11,;10.06,-1.44,;9.29,-2.78,;7.75,-2.78,;6.98,-1.44,;10.06,-4.11,;9.29,-5.44,;10.83,-5.44,;11.6,-4.11,;4.53,-.02,;3.07,.46,;1.74,-.31,;-4.93,2,;-6.27,2.77,)|
CS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(C[C@H]3CC[C@@H](CC3)C(F)(F)F)nc2c1 |wU:26.27,wD:29.34,10.13,(-6.27,-6.73,;-6.27,-5.19,;-7.81,-5.19,;-4.73,-5.19,;-6.27,-3.65,;-4.93,-2.88,;-4.93,-1.34,;-6.27,-.57,;-7.6,-1.34,;-7.6,-2.88,;-6.27,.97,;-7.6,1.74,;-8.93,.97,;-4.93,1.74,;-3.6,.97,;-3.6,-.57,;-2.26,1.74,;-2.26,3.28,;-.93,4.05,;.4,3.28,;1.87,3.76,;2.34,5.22,;2.02,6.73,;3.49,6.25,;2.77,2.51,;4.31,2.51,;5.08,1.18,;6.62,1.18,;7.39,-.16,;6.62,-1.49,;5.08,-1.49,;4.31,-.16,;7.39,-2.82,;6.62,-4.16,;8.16,-4.16,;8.93,-2.82,;1.87,1.27,;.4,1.74,;-.93,.97,)|
CNS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(C[C@H]4CC[C@@H](CC4)C(F)(F)F)nc3c2)cc1 |wU:23.23,wD:26.30,(-11.6,2.77,;-10.27,3.54,;-8.93,2.77,;-8.16,4.1,;-9.7,1.43,;-7.6,2,;-7.6,.46,;-6.27,-.31,;-4.93,.46,;-3.6,-.31,;-2.26,.46,;-.93,-.31,;-.93,-1.85,;.4,.46,;.4,2,;1.74,2.77,;3.07,2,;4.53,2.47,;5.01,3.94,;4.69,5.44,;6.16,4.97,;5.44,1.23,;6.98,1.23,;7.75,-.11,;9.29,-.11,;10.06,-1.44,;9.29,-2.78,;7.75,-2.78,;6.98,-1.44,;10.06,-4.11,;9.29,-5.44,;10.83,-5.44,;11.6,-4.11,;4.53,-.02,;3.07,.46,;1.74,-.31,;-4.93,2,;-6.27,2.77,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C)c(Cc4ccc(cc4)C(F)(F)F)nc3c2)cc1
CCn1c(Cc2ccc(cc2)C(F)(F)F)nc2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(Cc4ccc(cc4)C(F)(F)F)nc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CC(F)(F)F)c(Cc4ccc(cc4)C(F)(F)F)nc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CCC4)c(Cc4ccc(cc4)C(F)(F)F)nc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CC(C)(C)C)c(Cc4ccc(cc4)C(F)(F)F)nc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C(C)C)c(Cc4ccc(cc4)C(F)(F)F)nc3c2)nc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CC(C)C)c(Cc4ccc(cc4)C(F)(F)F)nc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(c(Cc4ccc(cc4)C(F)(F)F)nc3c2)C(C)(C)C)nc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CC(C)C)c(Cc4ccc(cc4)C(F)(F)F)nc3c2)nc1
CCS(=O)(=O)c1ccc(cc1)[C@@H](C)NC(=O)c1ccc2n(CC(C)C)c(Cc3ccc(cc3)C(F)(F)F)nc2c1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(C[C@H]4CC[C@@H](CC4)OC)nc3c2)cc1 |wU:23.23,wD:26.30,(-11.6,7.64,;-10.27,8.41,;-8.93,7.64,;-8.16,8.98,;-9.7,6.31,;-7.6,6.87,;-7.6,5.33,;-6.27,4.56,;-4.93,5.33,;-3.6,4.56,;-2.26,5.33,;-.93,4.56,;-.93,3.02,;.4,5.33,;.4,6.87,;1.74,7.64,;3.07,6.87,;4.53,7.35,;5.01,8.82,;4.69,10.32,;6.16,9.85,;5.44,6.1,;6.98,6.1,;7.75,4.77,;9.29,4.77,;10.06,3.44,;9.29,2.1,;7.75,2.1,;6.98,3.44,;10.06,.77,;11.6,.77,;4.53,4.86,;3.07,5.33,;1.74,4.56,;-4.93,6.87,;-6.27,7.64,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(Cc3ccc(OC(F)(F)F)cc3)nc2c1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(Cc4ccc(OC(F)F)cc4)nc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(CC4CCN(CC4)C(=O)OC(C)(C)C)nc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(CC4CCN(CC(F)(F)F)CC4)nc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(Cc4ccc(nc4)C(F)(F)F)nc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(Cc4ccc(Cl)cn4)nc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CC(C)C)c(CN4CCC(CC4)C(F)(F)F)nc3c2)cc1
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(CN3CCC(CC3)C(F)(F)F)nc2c1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(nc3c2)C(C)c2ccc(cc2)C(F)(F)F)cc1
CCn1c(CC2CCC(OC2)C(F)(F)F)nc2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCn1c(CC2CCC(OC2)C(F)(F)F)nc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cc1)S(=O)(=O)CC
CCS(=O)(=O)c1ccc(CNC(=O)c2cc(Br)c3n(C)c(C[C@H]4CC[C@@H](CC4)C(F)(F)F)nc3c2)cc1 |wU:22.21,wD:25.28,(-11.6,3.33,;-10.27,4.1,;-8.93,3.33,;-8.16,4.67,;-9.7,2,;-7.6,2.56,;-7.6,1.02,;-6.27,.25,;-4.93,1.02,;-3.6,.25,;-2.26,1.02,;-.93,.25,;-.93,-1.29,;.4,1.02,;.4,2.56,;1.74,3.33,;1.74,4.87,;3.07,2.56,;4.53,3.04,;5.01,4.5,;5.44,1.79,;6.98,1.79,;7.75,.46,;9.29,.46,;10.06,-.87,;9.29,-2.21,;7.75,-2.21,;6.98,-.87,;10.06,-3.54,;9.29,-4.87,;10.83,-4.87,;11.6,-3.54,;4.53,.55,;3.07,1.02,;1.74,.25,;-4.93,2.56,;-6.27,3.33,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2cc(Br)c3n(C)c(Cc4ccc(cc4)C(F)(F)F)nc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2cc(OC)c3n(C)c(Cc4ccc(cc4)C(F)(F)F)nc3c2)cc1
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(nc2c1)C(=O)c1ccc(cc1)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(nc2c1)C(=O)N1CCC(CC1)C(F)(F)F
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(nc3c2)[C@@H](O)[C@H]2CC[C@@H](CC2)C(F)(F)F)cc1 |wU:27.30,wD:30.36,25.28,(-11.6,-.25,;-10.27,.52,;-8.93,-.25,;-8.16,1.08,;-9.7,-1.59,;-7.6,-1.02,;-7.6,-2.56,;-6.27,-3.33,;-4.93,-2.56,;-3.6,-3.33,;-2.26,-2.56,;-.93,-3.33,;-.93,-4.87,;.4,-2.56,;.4,-1.02,;1.74,-.25,;3.07,-1.02,;4.53,-.55,;5.01,.92,;4.69,2.42,;6.16,1.95,;5.44,-1.79,;4.53,-3.04,;3.07,-2.56,;1.74,-3.33,;6.98,-1.79,;7.75,-3.13,;7.75,-.46,;6.98,.87,;7.75,2.21,;9.29,2.21,;10.06,.87,;9.29,-.46,;10.06,3.54,;10.83,4.87,;9.29,4.87,;11.6,3.54,;-4.93,-1.02,;-6.27,-.25,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(nc3c2)C(=O)C2CCC(CC2)C(F)(F)F)cc1 |(-11.6,-.25,;-10.27,.52,;-8.93,-.25,;-8.16,1.08,;-9.7,-1.59,;-7.6,-1.02,;-7.6,-2.56,;-6.27,-3.33,;-4.93,-2.56,;-3.6,-3.33,;-2.26,-2.56,;-.93,-3.33,;-.93,-4.87,;.4,-2.56,;.4,-1.02,;1.74,-.25,;3.07,-1.02,;4.53,-.55,;5.01,.92,;4.69,2.42,;6.16,1.95,;5.44,-1.79,;4.53,-3.04,;3.07,-2.56,;1.74,-3.33,;6.98,-1.79,;7.75,-3.13,;7.75,-.46,;6.98,.87,;7.75,2.21,;9.29,2.21,;10.06,.87,;9.29,-.46,;10.06,3.54,;10.83,4.87,;9.29,4.87,;11.6,3.54,;-4.93,-1.02,;-6.27,-.25,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(nc3c2)C(=O)c2ccc(cc2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(cc1)[C@H](COC(N)=O)NC(=O)c1ccc2n(C3CC3)c(C[C@H]3CC[C@@H](CC3)C(F)(F)F)nc2c1 |wU:30.31,wD:33.38,11.17,(6.27,7.11,;4.93,6.34,;4.93,4.8,;6.47,4.8,;3.39,4.8,;4.93,3.26,;3.6,2.49,;3.6,.95,;4.93,.18,;6.27,.95,;6.27,2.49,;4.93,-1.36,;6.27,-2.13,;7.6,-1.36,;8.93,-2.13,;10.27,-1.36,;8.93,-3.67,;3.6,-2.13,;2.26,-1.36,;2.26,.18,;.93,-2.13,;.93,-3.67,;-.4,-4.44,;-1.74,-3.67,;-3.2,-4.14,;-3.68,-5.61,;-3.36,-7.11,;-4.82,-6.64,;-4.11,-2.9,;-5.65,-2.9,;-6.42,-1.56,;-7.96,-1.56,;-8.73,-.23,;-7.96,1.1,;-6.42,1.1,;-5.65,-.23,;-8.73,2.44,;-7.96,3.77,;-9.5,3.77,;-10.27,2.44,;-3.2,-1.65,;-1.74,-2.13,;-.4,-1.36,)|
CCS(=O)(=O)c1ccc(cc1)[C@@H](COC(N)=O)NC(=O)c1ccc2n(C3CC3)c(C[C@H]3CC[C@@H](CC3)C(F)(F)F)nc2c1 |wU:30.31,11.17,wD:33.38,(6.27,7.11,;4.93,6.34,;4.93,4.8,;6.47,4.8,;3.39,4.8,;4.93,3.26,;3.6,2.49,;3.6,.95,;4.93,.18,;6.27,.95,;6.27,2.49,;4.93,-1.36,;6.27,-2.13,;7.6,-1.36,;8.93,-2.13,;10.27,-1.36,;8.93,-3.67,;3.6,-2.13,;2.26,-1.36,;2.26,.18,;.93,-2.13,;.93,-3.67,;-.4,-4.44,;-1.74,-3.67,;-3.2,-4.14,;-3.68,-5.61,;-3.36,-7.11,;-4.82,-6.64,;-4.11,-2.9,;-5.65,-2.9,;-6.42,-1.56,;-7.96,-1.56,;-8.73,-.23,;-7.96,1.1,;-6.42,1.1,;-5.65,-.23,;-8.73,2.44,;-7.96,3.77,;-9.5,3.77,;-10.27,2.44,;-3.2,-1.65,;-1.74,-2.13,;-.4,-1.36,)|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3n(CC(C)C)c(Cc4ccc(cc4)C(F)(F)F)nc3c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3n(CC(C)C)c(CN4CCC(CC4)C(F)(F)F)nc3c2)cc1
CCS(=O)(=O)c1ccc(nc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(Oc3ccc(cc3)C(F)(F)F)nc2c1
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(CO[C@H]3CC[C@H](CC3)C(F)(F)F)nc2c1 |wU:31.36,28.29,wD:11.14,(-21.15,-7.11,;-19.82,-6.34,;-19.82,-4.8,;-21.36,-4.8,;-18.28,-4.8,;-19.82,-3.26,;-18.48,-2.49,;-18.48,-.95,;-19.82,-.18,;-21.15,-.95,;-21.15,-2.49,;-19.82,1.36,;-21.15,2.13,;-22.49,1.36,;-18.48,2.13,;-17.15,1.36,;-17.15,-.18,;-15.82,2.13,;-15.82,3.67,;-14.48,4.44,;-13.15,3.67,;-11.69,4.14,;-11.21,5.61,;-11.53,7.11,;-10.06,6.64,;-10.78,2.9,;-9.24,2.9,;-8.47,4.23,;-6.93,4.23,;-6.16,5.56,;-4.62,5.56,;-3.85,4.23,;-4.62,2.9,;-6.16,2.9,;-2.31,4.23,;-1.54,2.9,;-.77,4.23,;-1.54,5.56,;-11.69,1.65,;-13.15,2.13,;-14.48,1.36,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3n(C4CC4)c(C[C@H]4CC[C@@H](CC4)C(F)(F)F)nc3c2)cc1 |wU:23.23,wD:26.30,(-11.6,.25,;-10.27,-.52,;-8.93,.25,;-9.7,1.59,;-8.16,-1.08,;-7.6,1.02,;-6.27,.25,;-4.93,1.02,;-4.93,2.56,;-3.6,3.33,;-2.26,2.56,;-.93,3.33,;-.93,4.87,;.4,2.56,;.4,1.02,;1.74,.25,;3.07,1.02,;4.53,.55,;5.01,-.92,;6.16,-1.95,;4.69,-2.42,;5.44,1.79,;6.98,1.79,;7.75,.46,;9.29,.46,;10.06,-.87,;9.29,-2.21,;7.75,-2.21,;6.98,-.87,;10.06,-3.54,;9.29,-4.87,;10.83,-4.87,;11.6,-3.54,;4.53,3.04,;3.07,2.56,;1.74,3.33,;-6.27,3.33,;-7.6,2.56,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3n(C4CC4)c(CC4CCC(CC4)C(F)(F)F)nc3c2)cc1 |(-13.39,7.33,;-12.62,8.66,;-13.39,9.99,;-14.16,8.66,;-14.16,11.33,;-11.85,9.99,;-11.08,11.33,;-9.54,11.33,;-8.77,9.99,;-7.23,9.99,;-6.46,8.66,;-4.92,8.66,;-4.15,9.99,;-4.15,7.33,;-4.92,5.99,;-4.15,4.66,;-2.61,4.66,;-1.58,3.51,;-1.9,2.01,;-2.93,.86,;-1.58,.5,;-.17,4.14,;1.16,3.37,;2.5,4.14,;2.5,5.68,;3.83,6.45,;5.16,5.68,;5.16,4.14,;3.83,3.37,;6.5,6.45,;7.83,5.68,;6.5,7.99,;7.83,7.22,;-.33,5.67,;-1.84,5.99,;-2.61,7.33,;-9.54,8.66,;-11.08,8.66,)|
CS(=O)(=O)c1ccc(CNC(=O)c2cnc3n(C4CC4)c(Cc4ccc(cc4)C(F)(F)F)nc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3n(C4CC4)c(Cc4ccc(cc4)C(F)(F)F)nc3c2)cc1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2c(c1)N(CC1CCOCC1)CCS2(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c(c1)S(C)(=O)=NC
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2c(c1)N(CC1CCOCC1)CCS2=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2c(c1)N(CC1CCOCC1)C(=O)CS2=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2SCCN(CC3CCOCC3)c2c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c(c1)[S@](C)(=N)=O |r|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c(c1)[S@@](C)(=N)=O |r|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2SCCNc2c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2SCC(=O)Nc2c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(c(CO)c1)S(=O)CC1CCOCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(c(CO)c1)S(=O)CC1CCOCC1 |w:26.27|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(cc1)S(=O)CC1CCOCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(cc1)S(=O)CC1CCOCC1 |w:24.25|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(c(c1)C(=O)OC)S(=O)CC1CCOCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(SCC2CCOCC2)c(c1)C(=O)OC
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c(c1)S(=N)(=O)CC
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c(c1)S(C)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c(c1)[S@@](C)=O |r|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c(c1)[S@](C)=O |r|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(SCC2CCOCC2)c(CO)c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c(c1)S(=O)CC
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c(c1)S(C)(=O)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c(SC)c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(cc1)S(=N)(=O)CC1CCOCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2(F)CCOCC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2C3COCC23)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2(F)COC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OC2CCN(CC2)C(=O)OC(C)(C)C)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2(C)COC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OC[C@H]2[C@@H]3COC[C@H]23)c(c1)S(C)(=N)=O |r|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCN(CC2)C(=O)OC(C)(C)C)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCSCC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCCc2ccno2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCc2ccncc2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC(O)CO)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OC2CCOCC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCc2cc(C)nc(C)c2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCc2ccc(F)cc2F)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OC2CCNCC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OC2CCN(CC2)C(C)=O)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OC2CCN(CC2)S(C)(=O)=O)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCNCC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCN(CC2)C(C)=O)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCN(CC2)S(C)(=O)=O)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2CCOCC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N(C)CC2CCOCC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2COC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2(C)CCOCC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2CCC(=O)NC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2CNC(=O)C2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N[C@H](C)C2CCOCC2)c(c1)S(C)(=N)=O |r|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2CC(O)C2)c(c1)S(C)(=N)=O |(2.28,-4.62,;3.61,-3.85,;3.61,-2.31,;2.28,-1.54,;2.28,,;3.61,.77,;4.94,,;4.94,-1.54,;3.61,2.31,;4.94,3.08,;6.28,2.31,;7.61,3.08,;6.28,.77,;2.28,3.08,;2.28,4.62,;2.68,1.59,;.94,2.31,;.94,.77,;-.39,,;-1.72,.77,;-3.06,,;-3.06,-1.54,;-4.39,-2.31,;-5.88,-1.91,;-6.28,-3.4,;-7.61,-4.17,;-4.79,-3.8,;-1.72,2.31,;-.39,3.08,;-3.06,3.08,;-4.39,2.31,;-3.83,4.41,;-2.29,4.41,)|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2(F)CCOCC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CCN(CC2)C(C)=O)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCc2ccncc2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(CCN2CCOCC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c(c1)S(N)(=O)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2CCOCC2)c(c1)S(N)(=O)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(SCC2CCOCC2)cc1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2SCC(=O)N(CC3CCOCC3)c2c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2N(CC3CCOCC3)CCS(=O)c2c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2n(CC3CCOCC3)c(=O)sc2c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2N(CC3CCOCC3)C(C)(C)Sc2c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2N(CC3CCOCC3)C(C)(C)S(=O)c2c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2N(CC3CCOCC3)CS(=O)c2c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2N(CC3CCOCC3)CS(=N)(=O)c2c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCc2ccnc(OC)c2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCS(=O)(=O)CC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OC[C@H]2CNC(=O)O2)c(c1)S(C)(=N)=O |r|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(Oc2ccc(cc2)C#N)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N[C@@H](C)C2CCOCC2)c(c1)S(C)(=N)=O |r|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2CNC(=O)O2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NC2CCS(=O)(=O)CC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2CCN(CC2)C(C)=O)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NC2CCC(=O)NC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NC2CCS(=O)(=O)C2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CCSCC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCc2nonc2C)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2CN(C2)C(=O)OC)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCc2ccnc(C)c2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NC[C@H]2[C@@H]3COC[C@H]23)c(c1)S(C)(=N)=O |r|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2(O)CCOCC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2CCN(CC2)C(=O)OC)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2CCN(C2)C(=O)OC)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2CC3(COC3)C2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2CCNC(=O)C2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCc2c(C)noc2C)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2CSC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2CCN(C2)C(C)=O)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CCOC[C@H]2C)c(c1)S(C)(=N)=O |r|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NC[C@@H]2CNC(=O)O2)c(c1)S(C)(=N)=O |r|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NC[C@H]2CNC(=O)O2)c(c1)S(C)(=N)=O |r|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NC2CCNC(=O)C2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CCCC3(COC3)C2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CC3(CN(C3)C(=O)OC(C)(C)C)C2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CC3(COC3)C2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CCC3(COC3)C2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CC3(C2)CS(=O)(=O)C3)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CCC3(COC3)CC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2C[C@H]3C[C@@H]2CO3)c(c1)S(C)(=N)=O |r,TLB:19:20:26.25:23|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CC3CC2CO3)c(c1)S(C)(=N)=O |TLB:19:20:26.25:23|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCc2nn[nH]n2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CC3(CNC3)C2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CC3(CN(C3)C(C)=O)C2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CCOCC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2(CC)CCOCC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2(CCOCC2)OC)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2(CC)COC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCc2ccnc(OC)c2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CCC(O)CC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CC[C@H](O)C2)c(c1)S(C)(=N)=O |r|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CC[C@@H](O)C2)c(c1)S(C)(=N)=O |r|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CC(O)C2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCC2(COC2)N2CCCC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(NCc2ccncn2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CCCOCC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CCNCC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(N2CCS(=O)(=O)CC2)c(c1)S(C)(=N)=O
CC(C)CN(c1ccc(C)cc1C)S(=O)(=O)c1ccc(OCC2CCOCC2)c(c1)S(C)(=N)=O
COc1ccc(N(C(C)C)S(=O)(=O)c2ccc(OCC3CCOCC3)c(c2)S(C)(=N)=O)c(C)c1
COC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3cccnc23)c(F)c1
COC(=O)c1ccc(-c2cn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3cccnc23)c(F)c1
Cc1cccc(c1C(=O)n1nc(-c2ccc(cc2F)C(O)=O)c2ncccc12)C1(CC1)C(F)(F)F
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)F)c3cccnc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CF)CC3)c3cccnc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)c(F)ccc3C3(CC3)C(F)(F)F)c3cccnc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(cccc3C3(CC3)C(F)(F)F)C(F)F)c3cccnc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)c(F)ccc3C3(CC3)C(F)F)c3cccnc23)c(F)c1
Cc1c(F)ccc(c1C(=O)n1nc(-c2ccc(cc2F)C(O)=O)c2ncccc12)C1(CC1)C(F)(F)F
OC(=O)c1ccc(-c2cn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)F)c3cccnc23)c(F)c1
CCS(=O)(=O)c1ccc(CNC(=O)c2cc3CC(C)(C)OC4(CCN(CC4)[C@H](C)c4cnc(nc4)C(F)(F)F)c3s2)nc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cc3CC4(CC4)OC4(CCN(CC4)[C@H](C)c4cnc(nc4)C(F)(F)F)c3s2)nc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cc3CC4(CC4)OC4(CCN(CC4)C(C)c4ccc(cc4)C#N)c3s2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(10.67,-4.62,;9.34,-3.85,;8,-4.62,;7.23,-3.29,;8.77,-5.95,;6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;5.33,-7.7,;6.67,-6.93,)|
CCS(=O)(=O)c1ccc(CNC(=O)Nc2ccc(cc2)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)Nc2ccc(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1
CS(=O)(=O)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(8.77,-5.95,;8,-4.62,;9.34,-3.85,;7.23,-3.29,;6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;5.33,-7.7,;6.67,-6.93,)|
CNS(=O)(=O)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(10.67,-4.62,;9.34,-3.85,;8,-4.62,;7.23,-3.29,;8.77,-5.95,;6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;5.33,-7.7,;6.67,-6.93,)|
NS(=O)(=O)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(9.34,-3.85,;8,-4.62,;7.23,-3.29,;8.77,-5.95,;6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;5.33,-7.7,;6.67,-6.93,)|
CC(=O)NS(=O)(=O)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(10.67,-1.54,;9.34,-2.31,;8,-1.54,;9.34,-3.85,;8,-4.62,;7.23,-3.29,;8.77,-5.95,;6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;5.33,-7.7,;6.67,-6.93,)|
CS(=O)(=O)Nc1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(8.57,-6.72,;9.34,-5.39,;10.67,-6.16,;10.11,-4.06,;8,-4.62,;6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;5.33,-7.7,;6.67,-6.93,)|
CCS(=N)(=O)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(10.67,-4.62,;9.34,-3.85,;8,-4.62,;8.77,-5.95,;7.23,-3.29,;6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;5.33,-7.7,;6.67,-6.93,)|
CS(=O)(=O)NC(=O)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(11.44,-5.95,;10.67,-4.62,;12,-3.85,;9.9,-3.29,;9.34,-5.39,;8,-4.62,;8,-3.08,;6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;5.33,-7.7,;6.67,-6.93,)|
CCS(=O)(=O)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)nc1 |(10.67,-4.62,;9.34,-3.85,;8,-4.62,;7.23,-3.29,;8.77,-5.95,;6.67,-5.39,;6.67,-6.93,;5.33,-7.7,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;4,-5.39,;5.33,-4.62,)|
CS(=O)(=O)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)nc1 |(8.77,-5.95,;8,-4.62,;9.34,-3.85,;7.23,-3.29,;6.67,-5.39,;6.67,-6.93,;5.33,-7.7,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;4,-5.39,;5.33,-4.62,)|
CNS(=O)(=O)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)nc1 |(10.67,-4.62,;9.34,-3.85,;8,-4.62,;7.23,-3.29,;8.77,-5.95,;6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;5.33,-7.7,;6.67,-6.93,)|
OC(=O)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(8,-3.08,;8,-4.62,;9.34,-5.39,;6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;5.33,-7.7,;6.67,-6.93,)|
OC(=O)Cc1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(9.34,-6.93,;9.34,-5.39,;10.67,-4.62,;8,-4.62,;6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;5.33,-7.7,;6.67,-6.93,)|
OC(=O)Cc1ccc(CNC(=O)Nc2cc(Cl)c(c(c2)C#N)-c2ccccc2OC(F)(F)F)cc1 |(9.34,-13.09,;10.67,-12.32,;12,-13.09,;10.67,-10.78,;9.34,-10.01,;9.34,-8.47,;8,-7.7,;6.67,-8.47,;5.33,-7.7,;4,-8.47,;2.67,-7.7,;2.67,-6.16,;1.33,-8.47,;,-7.7,;,-6.16,;-1.33,-5.39,;-1.33,-3.85,;-2.67,-6.16,;-2.67,-7.7,;-1.33,-8.47,;-4,-8.47,;-5.33,-9.24,;-4,-5.39,;-4,-3.85,;-5.33,-3.08,;-6.67,-3.85,;-6.67,-5.39,;-5.33,-6.16,;-5.33,-7.7,;-6.67,-8.47,;-8,-9.24,;-7.44,-7.14,;-5.9,-9.8,;6.67,-10.01,;8,-10.78,)|
Cc1cc(NC(=O)NCc2ccc(CC(O)=O)cc2)cc(Cl)c1-c1ccccc1OC(F)(F)F |(-4,-8.47,;-2.67,-7.7,;-1.33,-8.47,;,-7.7,;1.33,-8.47,;2.67,-7.7,;2.67,-6.16,;4,-8.47,;5.33,-7.7,;6.67,-8.47,;8,-7.7,;9.34,-8.47,;9.34,-10.01,;10.67,-10.78,;10.67,-12.32,;9.34,-13.09,;12,-13.09,;8,-10.78,;6.67,-10.01,;,-6.16,;-1.33,-5.39,;-1.33,-3.85,;-2.67,-6.16,;-4,-5.39,;-4,-3.85,;-5.33,-3.08,;-6.67,-3.85,;-6.67,-5.39,;-5.33,-6.16,;-5.33,-7.7,;-6.67,-8.47,;-8,-9.24,;-7.44,-7.14,;-5.9,-9.8,)|
OC(=O)Cc1ccc(CNC(=O)Nc2ccc(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1
OC(=O)Cc1ccc(CNC(=O)Nc2cc(F)c(c(F)c2)-c2ccccc2OC(F)(F)F)cc1 |(9.34,-6.93,;9.34,-5.39,;10.67,-4.62,;8,-4.62,;6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;5.33,-7.7,;6.67,-6.93,)|
OC(=O)Cc1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)F)cc1 |(9.34,-6.93,;9.34,-5.39,;10.67,-4.62,;8,-4.62,;6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.82,-15.14,;-3.74,-14.56,;5.33,-7.7,;6.67,-6.93,)|
Cc1cc(NC(=O)NCc2ccc(CC(O)=O)cc2)cc(C)c1-c1ccccc1OC(F)F |(-4,-5.39,;-2.67,-4.62,;-1.33,-5.39,;,-4.62,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;8,-4.62,;9.34,-5.39,;9.34,-6.93,;10.67,-7.7,;10.67,-9.24,;9.34,-10.01,;12,-10.01,;8,-7.7,;6.67,-6.93,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;-2.67,-3.08,;-4,-2.31,;-5.33,-3.08,;-6.67,-2.31,;-6.67,-.77,;-5.33,,;-4,-.77,;-2.67,,;-2.67,1.54,;-1.33,2.31,;-4,2.31,)|
Cn1cc(cn1)-c1cc(NC(=O)NCc2ccc(CC(O)=O)cc2)ccc1-c1ccccc1OC(F)(F)F
Cn1cc(cn1)-c1cccc(OC(F)(F)F)c1-c1ccc(NC(=O)NCc2ccc(CC(O)=O)cc2)cc1
OC(=O)Cc1ccc(CNC(=O)Nc2ccc(cc2)-c2ccccc2)cc1
CC(C(O)=O)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(8,-3.08,;8,-4.62,;9.34,-5.39,;9.34,-6.93,;10.67,-4.62,;6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;5.33,-7.7,;6.67,-6.93,)|
OC(=O)C(F)(F)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(9.34,-2.31,;9.34,-3.85,;10.67,-4.62,;8,-4.62,;7.23,-3.29,;8.77,-5.95,;6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;5.33,-7.7,;6.67,-6.93,)|
OC(=O)COc1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(10.67,-3.08,;10.67,-4.62,;12,-5.39,;9.34,-5.39,;8,-4.62,;6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;5.33,-7.7,;6.67,-6.93,)|
CN(C(=O)NCc1ccc(CC(O)=O)cc1)c1cc(Cl)c(c(Cl)c1)-c1ccccc1OC(F)(F)F |(-1.33,-5.39,;-1.33,-6.93,;,-7.7,;,-9.24,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;8,-4.62,;9.34,-5.39,;9.34,-6.93,;10.67,-4.62,;6.67,-6.93,;5.33,-7.7,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,)|
CN(Cc1ccc(CC(O)=O)cc1)C(=O)Nc1cc(Cl)c(c(Cl)c1)-c1ccccc1OC(F)(F)F |(1.33,-5.39,;1.33,-6.93,;2.67,-7.7,;4,-6.93,;4,-5.39,;5.33,-4.62,;6.67,-5.39,;8,-4.62,;9.34,-5.39,;9.34,-6.93,;10.67,-4.62,;6.67,-6.93,;5.33,-7.7,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,)|
OC(=O)Cc1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)nc1 |(9.34,-6.93,;9.34,-5.39,;10.67,-4.62,;8,-4.62,;6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;5.33,-7.7,;6.67,-6.93,)|
CC(C(O)=O)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)nc1 |(8,-3.08,;8,-4.62,;9.34,-5.39,;9.34,-6.93,;10.67,-4.62,;6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;5.33,-7.7,;6.67,-6.93,)|
Cc1cc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)ccc1CC(O)=O |(5.33,-3.08,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-6.67,-10.01,;-8,-9.24,;-9.34,-10.01,;-9.34,-11.55,;-8,-12.32,;-6.67,-11.55,;-5.33,-12.32,;-5.33,-13.86,;-5.33,-15.4,;-6.87,-13.86,;-3.79,-13.86,;5.33,-7.7,;6.67,-6.93,;6.67,-5.39,;8,-4.62,;9.34,-5.39,;9.34,-6.93,;10.67,-4.62,)|
CCS(=O)(=O)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(10.4,1.23,;9.63,2.56,;8.09,2.56,;8.09,4.1,;8.09,1.02,;6.55,2.56,;5.78,3.9,;4.24,3.9,;3.47,2.56,;1.93,2.56,;1.15,1.23,;-.39,1.23,;-1.15,2.56,;-1.15,-.1,;-2.7,-.1,;-3.47,1.23,;-5.01,1.23,;-5.78,2.56,;-5.78,-.1,;-5.01,-1.44,;-5.78,-2.77,;-3.47,-1.44,;-7.32,-.1,;-8.09,1.23,;-9.63,1.23,;-10.4,-.1,;-9.63,-1.44,;-8.09,-1.44,;-7.32,-2.77,;-8.09,-4.1,;-9.63,-4.1,;-7.32,-5.44,;-8.86,-5.44,;4.24,1.23,;5.78,1.23,)|
CN1CC2(C1)CN(C2)C(=O)C1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:23|
COC1CN(C1)C(=O)[C@@]1(C)CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1CC1 |t:21|
COC1CN(C1)C(=O)[C@H]1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(C)ccnc1N1CCC1 |t:20|
CN(C)[C@@H]1CCN(C1)C(=O)[C@@H]1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(F)CCC1 |t:22|
CN(C)[C@@H]1CCN(C1)C(=O)[C@H]1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(F)CCC1 |t:22|
OC1CCN(C1)C(=O)[C@@H]1CCc2c(C1)n(nc2C1=CCC(CC1)C(O)=O)C(=O)c1c(Cl)cccc1C1(CC1)C(F)(F)F |t:20|
CCOC(=O)[C@@H]1CCC(=C[C@@H]1C)c1nn(C(=O)c2c(Cl)cccc2C2(CC2)C(F)(F)F)c2CC(CCc12)C(=O)N1CC(C)(O)C1 |r,c:8|
COC1CN(C1)C(=O)[C@H]1CCc2c(nn(C(=O)c3c(Cl)cccc3C3CC3)c2C1)N1CCC(CC1)C(O)=O
COC1CN(C1)C(=O)[C@H]1CCc2c(nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c2C1)N1CCC(CC1)C(O)=O
CC(F)(F)C(C)(C)OC(=O)Nc1ccc2OC(CN(c2c1)S(=O)(=O)c1ccc(F)c(F)c1)C(=O)C(F)(F)F
CC(C)(OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)cc1)C(C)(C)C(O)=O)C(F)(F)F
CC(C)(C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)NS(=O)(=O)C1CC1 |r|
CC(C)(C)OC(=O)Nc1cnc2CC(CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)NC(=O)OCc1ccccc1
CC(C)(OC(=O)Nc1ccc2O[C@H](CN(c2c1)S(=O)(=O)c1ccc(F)c(F)c1)[C@@H](O)C(F)(F)F)C(F)(F)F
C[C@@H]1[C@H](CNC(=O)Oc2ccccc2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc2N1S(=O)(=O)c1ccc(F)c(F)c1
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](C[C@H](C2CC2)C(N)=O)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](C[C@H](C)C(=O)NS(=O)(=O)C2CC2)Oc2ccc(NC(=O)OC(C)(C)C(F)(F)F)cc12
Cc1ccc(cc1)S(=O)(=O)NC(=O)CC[C@@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@@H](CS(=O)(=O)CC)Oc2ncc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCn1cc(c(Cl)n1)S(=O)(=O)N1C[C@H](CS(=O)(=O)CC)Oc2ncc(NC(=O)OC(C)(C)C(F)(F)F)cc12 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3[C@H](C(C)C)N(Cc3c2)c2nccc(n2)C(F)(F)F)nc1 |r|
CCOC(=O)c1cnc(nc1C(C)(C)C)N1Cc2cc(cnc2[C@@H]1C(C)C)C(=O)NCc1ccc(cc1)S(=O)(=O)CC |r|
CCS(=O)(=O)c1ccc(cc1)C(CO)NC(=O)c1ccc2n(C3CC3)c(CN3CCC(CC3)C(F)(F)F)cc2c1
CCn1c(CC2CCC(CC2)C(F)(F)F)cc2cc(ccc12)C(=O)N[C@H](CO)c1ccc(cn1)S(=O)(=O)CC |wD:25.27,(2.68,-5.16,;1.65,-4.01,;2.13,-2.55,;1.22,-1.3,;-.32,-1.3,;-1.09,.03,;-2.63,.03,;-3.4,1.36,;-2.63,2.7,;-1.09,2.7,;-.32,1.36,;-3.4,4.03,;-4.17,5.37,;-2.07,4.8,;-4.73,3.26,;2.13,-.06,;3.59,-.53,;4.92,.24,;6.26,-.53,;6.26,-2.07,;4.92,-2.84,;3.59,-2.07,;7.59,.24,;7.59,1.78,;8.93,-.53,;10.26,.24,;10.26,1.78,;11.59,2.55,;11.59,-.53,;11.59,-2.07,;12.93,-2.84,;14.26,-2.07,;14.26,-.53,;12.93,.24,;15.59,-2.84,;16.36,-1.51,;14.82,-4.18,;16.93,-3.61,;18.26,-2.84,)|
CCn1c(CC2CCC(CC2)C(F)(F)F)cc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cn1)S(=O)(=O)CC |wU:25.27,(2.68,-5.16,;1.65,-4.01,;2.13,-2.55,;1.22,-1.3,;-.32,-1.3,;-1.09,.03,;-2.63,.03,;-3.4,1.36,;-2.63,2.7,;-1.09,2.7,;-.32,1.36,;-3.4,4.03,;-4.17,5.37,;-2.07,4.8,;-4.73,3.26,;2.13,-.06,;3.59,-.53,;4.92,.24,;6.26,-.53,;6.26,-2.07,;4.92,-2.84,;3.59,-2.07,;7.59,.24,;7.59,1.78,;8.93,-.53,;10.26,.24,;10.26,1.78,;11.59,2.55,;11.59,-.53,;11.59,-2.07,;12.93,-2.84,;14.26,-2.07,;14.26,-.53,;12.93,.24,;15.59,-2.84,;16.36,-1.51,;14.82,-4.18,;16.93,-3.61,;18.26,-2.84,)|
CCn1c(Cc2ccc(NC=O)cc2)cc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cn1)S(=O)(=O)CC |r|
Cc1ccc(cc1)S(=O)(=O)n1c(cc2cc(Br)ccc12)C(O)c1ccc(cn1)C(F)(F)F
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3n(C4CC4)c(CC4CCC(CC4)C(F)(F)F)cc3c2)cc1 |(15.87,.24,;14.53,1.01,;13.2,.24,;12.43,1.57,;13.97,-1.1,;11.87,-.53,;10.53,.24,;9.2,-.53,;9.2,-2.07,;7.87,-2.84,;6.53,-2.07,;5.2,-2.84,;5.2,-4.38,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;-.27,-.06,;-.74,1.41,;-1.89,2.44,;-.42,2.91,;-1.17,-1.3,;-2.71,-1.3,;-3.48,-2.64,;-2.71,-3.97,;-3.48,-5.3,;-5.02,-5.3,;-5.79,-3.97,;-5.02,-2.64,;-5.79,-6.64,;-6.56,-7.97,;-7.13,-5.87,;-4.46,-7.41,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,;10.53,-2.84,;11.87,-2.07,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1cnc2n(C3CC3)c(CC3CCC(CC3)C(F)(F)F)cc2c1 |wD:11.14,(15.87,.24,;14.53,1.01,;13.2,.24,;12.43,1.57,;13.97,-1.1,;11.87,-.53,;10.53,.24,;9.2,-.53,;9.2,-2.07,;10.53,-2.84,;11.87,-2.07,;7.87,-2.84,;7.87,-4.38,;6.53,-5.15,;6.53,-2.07,;5.2,-2.84,;5.2,-4.38,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;-.27,-.06,;-.74,1.41,;-1.89,2.44,;-.42,2.91,;-1.17,-1.3,;-2.71,-1.3,;-3.48,-2.64,;-2.71,-3.97,;-3.48,-5.3,;-5.02,-5.3,;-5.79,-3.97,;-5.02,-2.64,;-5.79,-6.64,;-6.56,-7.97,;-7.13,-5.87,;-4.46,-7.41,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,)|
FC(F)(F)C1CCC(CC1)OC(=O)c1ccc2n(C3CC3)c(OC3CCC(CC3)C(F)(F)F)nc2c1 |(9.12,-27.52,;7.42,-28.51,;8.4,-30.22,;6.43,-26.8,;5.71,-29.5,;5.08,-31.4,;3.75,-32.17,;2.42,-31.4,;2.42,-29.86,;3.75,-29.09,;1.08,-32.17,;-.25,-31.4,;-.25,-29.86,;-1.58,-32.17,;-1.58,-33.71,;-2.92,-34.48,;-4.25,-33.71,;-5.72,-34.18,;-6.19,-35.65,;-7.34,-36.68,;-5.87,-37.15,;-6.62,-32.94,;-8.16,-32.94,;-8.93,-31.6,;-8.16,-30.27,;-8.93,-28.94,;-10.47,-28.94,;-11.24,-30.27,;-10.47,-31.6,;-11.24,-27.6,;-10.47,-26.27,;-12.78,-27.6,;-12.01,-26.27,;-5.72,-31.69,;-4.25,-32.17,;-2.92,-31.4,)|
CCn1c(OC2CCC(CC2)C(F)(F)F)nc2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC |(.29,2.55,;-.74,1.41,;-.27,-.06,;-1.17,-1.3,;-2.71,-1.3,;-3.48,-2.64,;-2.71,-3.97,;-3.48,-5.3,;-5.02,-5.3,;-5.79,-3.97,;-5.02,-2.64,;-5.79,-6.64,;-6.56,-7.97,;-7.13,-5.87,;-4.46,-7.41,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;5.2,-2.84,;5.2,-4.38,;6.53,-2.07,;7.87,-2.84,;9.2,-2.07,;9.2,-.53,;10.53,.24,;11.87,-.53,;11.87,-2.07,;10.53,-2.84,;13.2,.24,;12.43,1.57,;13.97,-1.1,;14.53,1.01,;15.87,.24,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(OC4CCC(CC4)C(F)(F)F)nc3c2)cc1 |(15.87,.24,;14.53,1.01,;13.2,.24,;12.43,1.57,;13.97,-1.1,;11.87,-.53,;10.53,.24,;9.2,-.53,;9.2,-2.07,;7.87,-2.84,;6.53,-2.07,;5.2,-2.84,;5.2,-4.38,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;-.27,-.06,;-.74,1.41,;-1.89,2.44,;-.42,2.91,;-1.17,-1.3,;-2.71,-1.3,;-3.48,-2.64,;-2.71,-3.97,;-3.48,-5.3,;-5.02,-5.3,;-5.79,-3.97,;-5.02,-2.64,;-5.79,-6.64,;-6.56,-7.97,;-7.13,-5.87,;-4.46,-7.41,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,;10.53,-2.84,;11.87,-2.07,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CC(C)C)c(O[C@H]4CC[C@@H](CC4)C(F)(F)F)nc3c2)cc1 |r,wU:27.30,wD:24.23,(14.53,6.69,;14.53,5.15,;13.2,4.38,;12.43,5.72,;13.97,3.05,;11.87,3.61,;11.87,2.07,;10.53,1.3,;9.2,2.07,;7.87,1.3,;6.53,2.07,;5.2,1.3,;5.2,-.24,;3.86,2.07,;3.86,3.61,;2.53,4.38,;1.2,3.61,;-.27,4.09,;-.74,5.55,;-2.25,5.87,;-3.28,4.73,;-2.73,7.34,;-1.17,2.84,;-2.71,2.84,;-3.48,1.51,;-5.02,1.51,;-5.79,.18,;-5.02,-1.16,;-3.48,-1.16,;-2.71,.18,;-5.79,-2.49,;-6.56,-3.83,;-7.13,-1.72,;-4.46,-3.26,;-.27,1.6,;1.2,2.07,;2.53,1.3,;9.2,3.61,;10.53,4.38,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CC(C)C)c(O[C@H]4CC[C@@H](CC4)C(F)(F)F)nc3c2)cc1 |r,wU:24.23,wD:27.30,(14.53,6.69,;14.53,5.15,;13.2,4.38,;12.43,5.72,;13.97,3.05,;11.87,3.61,;11.87,2.07,;10.53,1.3,;9.2,2.07,;7.87,1.3,;6.53,2.07,;5.2,1.3,;5.2,-.24,;3.86,2.07,;3.86,3.61,;2.53,4.38,;1.2,3.61,;-.27,4.09,;-.74,5.55,;-2.25,5.87,;-3.28,4.73,;-2.73,7.34,;-1.17,2.84,;-2.71,2.84,;-3.48,1.51,;-2.71,.18,;-3.48,-1.16,;-5.02,-1.16,;-5.79,.18,;-5.02,1.51,;-5.79,-2.49,;-6.56,-3.83,;-7.13,-1.72,;-4.46,-3.26,;-.27,1.6,;1.2,2.07,;2.53,1.3,;9.2,3.61,;10.53,4.38,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CC(C)C)c(CC4CCC(CC4)C(F)(F)F)nc3c2)cc1 |(14.53,6.69,;14.53,5.15,;13.2,4.38,;12.43,5.72,;13.97,3.05,;11.87,3.61,;11.87,2.07,;10.53,1.3,;9.2,2.07,;7.87,1.3,;6.53,2.07,;5.2,1.3,;5.2,-.24,;3.86,2.07,;3.86,3.61,;2.53,4.38,;1.2,3.61,;-.27,4.09,;-.74,5.55,;-2.25,5.87,;-3.28,4.73,;-2.73,7.34,;-1.17,2.84,;-2.71,2.84,;-3.48,1.51,;-2.71,.18,;-3.48,-1.16,;-5.02,-1.16,;-5.79,.18,;-5.02,1.51,;-5.79,-2.49,;-6.56,-3.83,;-7.13,-1.72,;-4.46,-3.26,;-.27,1.6,;1.2,2.07,;2.53,1.3,;9.2,3.61,;10.53,4.38,)|
CCn1c(CC2CCC(CC2)C(F)(F)F)nc2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC |(.29,2.55,;-.74,1.41,;-.27,-.06,;-1.17,-1.3,;-2.71,-1.3,;-3.48,-2.64,;-2.71,-3.97,;-3.48,-5.3,;-5.02,-5.3,;-5.79,-3.97,;-5.02,-2.64,;-5.79,-6.64,;-6.56,-7.97,;-7.13,-5.87,;-4.46,-7.41,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;5.2,-2.84,;5.2,-4.38,;6.53,-2.07,;7.87,-2.84,;9.2,-2.07,;9.2,-.53,;10.53,.24,;11.87,-.53,;11.87,-2.07,;10.53,-2.84,;13.2,.24,;12.43,1.57,;13.97,-1.1,;14.53,1.01,;15.87,.24,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(CC3CCC(CC3)C(F)(F)F)nc2c1 |wD:11.14,(15.87,.24,;14.53,1.01,;13.2,.24,;12.43,1.57,;13.97,-1.1,;11.87,-.53,;10.53,.24,;9.2,-.53,;9.2,-2.07,;10.53,-2.84,;11.87,-2.07,;7.87,-2.84,;7.87,-4.38,;6.53,-5.15,;6.53,-2.07,;5.2,-2.84,;5.2,-4.38,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;-.27,-.06,;-.74,1.41,;-1.89,2.44,;-.42,2.91,;-1.17,-1.3,;-2.71,-1.3,;-3.48,-2.64,;-2.71,-3.97,;-3.48,-5.3,;-5.02,-5.3,;-5.79,-3.97,;-5.02,-2.64,;-5.79,-6.64,;-6.56,-7.97,;-7.13,-5.87,;-4.46,-7.41,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,)|
CCS(=O)(=O)c1ccc(cc1)[C@@H](CO)NC(=O)c1ccc2n(C3CC3)c(CC3CCC(CC3)C(F)(F)F)nc2c1 |wU:11.14,(15.87,.24,;14.53,1.01,;13.2,.24,;12.43,1.57,;13.97,-1.1,;11.87,-.53,;10.53,.24,;9.2,-.53,;9.2,-2.07,;10.53,-2.84,;11.87,-2.07,;7.87,-2.84,;7.87,-4.38,;6.53,-5.15,;6.53,-2.07,;5.2,-2.84,;5.2,-4.38,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;-.27,-.06,;-.74,1.41,;-1.89,2.44,;-.42,2.91,;-1.17,-1.3,;-2.71,-1.3,;-3.48,-2.64,;-2.71,-3.97,;-3.48,-5.3,;-5.02,-5.3,;-5.79,-3.97,;-5.02,-2.64,;-5.79,-6.64,;-6.56,-7.97,;-7.13,-5.87,;-4.46,-7.41,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,)|
CCn1c(CC2CCC(CC2)C(F)(F)F)nc2cc(ccc12)C(=O)N[C@@H](CO)c1ccc(cc1)S(=O)(=O)CC |wD:25.27,(.29,2.55,;-.74,1.41,;-.27,-.06,;-1.17,-1.3,;-2.71,-1.3,;-3.48,-2.64,;-2.71,-3.97,;-3.48,-5.3,;-5.02,-5.3,;-5.79,-3.97,;-5.02,-2.64,;-5.79,-6.64,;-6.56,-7.97,;-7.13,-5.87,;-4.46,-7.41,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;5.2,-2.84,;5.2,-4.38,;6.53,-2.07,;7.87,-2.84,;7.87,-4.38,;6.53,-5.15,;9.2,-2.07,;9.2,-.53,;10.53,.24,;11.87,-.53,;11.87,-2.07,;10.53,-2.84,;13.2,.24,;12.43,1.57,;13.97,-1.1,;14.53,1.01,;15.87,.24,)|
CCn1c(CC2CCC(CC2)C(F)(F)F)nc2cc(ccc12)C(=O)N[C@H](CO)c1ccc(cc1)S(=O)(=O)CC |wU:25.27,(.29,2.55,;-.74,1.41,;-.27,-.06,;-1.17,-1.3,;-2.71,-1.3,;-3.48,-2.64,;-2.71,-3.97,;-3.48,-5.3,;-5.02,-5.3,;-5.79,-3.97,;-5.02,-2.64,;-5.79,-6.64,;-6.56,-7.97,;-7.13,-5.87,;-4.46,-7.41,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;5.2,-2.84,;5.2,-4.38,;6.53,-2.07,;7.87,-2.84,;7.87,-4.38,;6.53,-5.15,;9.2,-2.07,;9.2,-.53,;10.53,.24,;11.87,-.53,;11.87,-2.07,;10.53,-2.84,;13.2,.24,;12.43,1.57,;13.97,-1.1,;14.53,1.01,;15.87,.24,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](CCO)NC(=O)c1ccc2n(C3CC3)c(CC3CCC(CC3)C(F)(F)F)nc2c1 |wD:11.15,(15.87,.24,;14.53,1.01,;13.2,.24,;12.43,1.57,;13.97,-1.1,;11.87,-.53,;10.53,.24,;9.2,-.53,;9.2,-2.07,;10.53,-2.84,;11.87,-2.07,;7.87,-2.84,;7.87,-4.38,;9.2,-5.15,;9.2,-6.69,;6.53,-2.07,;5.2,-2.84,;5.2,-4.38,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;-.27,-.06,;-.74,1.41,;-1.89,2.44,;-.42,2.91,;-1.17,-1.3,;-2.71,-1.3,;-3.48,-2.64,;-2.71,-3.97,;-3.48,-5.3,;-5.02,-5.3,;-5.79,-3.97,;-5.02,-2.64,;-5.79,-6.64,;-6.56,-7.97,;-7.13,-5.87,;-4.46,-7.41,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CC(C)C)c(C[C@H]4CC[C@@H](CC4)C(F)(F)F)nc3c2)nc1 |r,wU:27.30,wD:24.23,(14.53,6.69,;14.53,5.15,;13.2,4.38,;12.43,5.72,;13.97,3.05,;11.87,3.61,;11.87,2.07,;10.53,1.3,;9.2,2.07,;7.87,1.3,;6.53,2.07,;5.2,1.3,;5.2,-.24,;3.86,2.07,;3.86,3.61,;2.53,4.38,;1.2,3.61,;-.27,4.09,;-.74,5.55,;-2.25,5.87,;-3.28,4.73,;-2.73,7.34,;-1.17,2.84,;-2.71,2.84,;-3.48,1.51,;-5.02,1.51,;-5.79,.18,;-5.02,-1.16,;-3.48,-1.16,;-2.71,.18,;-5.79,-2.49,;-6.56,-3.83,;-7.13,-1.72,;-4.46,-3.26,;-.27,1.6,;1.2,2.07,;2.53,1.3,;9.2,3.61,;10.53,4.38,)|
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CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(CC4CCC(CC4)C(F)(F)F)nc3c2)nc1 |(15.87,.24,;14.53,1.01,;13.2,.24,;12.43,1.57,;13.97,-1.1,;11.87,-.53,;11.87,-2.07,;10.53,-2.84,;9.2,-2.07,;7.87,-2.84,;6.53,-2.07,;5.2,-2.84,;5.2,-4.38,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;-.27,-.06,;-.74,1.41,;-1.89,2.44,;-.42,2.91,;-1.17,-1.3,;-2.71,-1.3,;-3.48,-2.64,;-2.71,-3.97,;-3.48,-5.3,;-5.02,-5.3,;-5.79,-3.97,;-5.02,-2.64,;-5.79,-6.64,;-6.56,-7.97,;-7.13,-5.87,;-4.46,-7.41,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,;9.2,-.53,;10.53,.24,)|
CCS(=O)(=O)c1ccc(nc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(CC3CCC(CC3)C(F)(F)F)nc2c1 |wD:11.14,(15.87,.24,;14.53,1.01,;13.2,.24,;12.43,1.57,;13.97,-1.1,;11.87,-.53,;11.87,-2.07,;10.53,-2.84,;9.2,-2.07,;9.2,-.53,;10.53,.24,;7.87,-2.84,;7.87,-4.38,;6.53,-5.15,;6.53,-2.07,;5.2,-2.84,;5.2,-4.38,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;-.27,-.06,;-.74,1.41,;-1.89,2.44,;-.42,2.91,;-1.17,-1.3,;-2.71,-1.3,;-3.48,-2.64,;-2.71,-3.97,;-3.48,-5.3,;-5.02,-5.3,;-5.79,-3.97,;-5.02,-2.64,;-5.79,-6.64,;-6.56,-7.97,;-7.13,-5.87,;-4.46,-7.41,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,)|
CCS(=O)(=O)c1ccc(nc1)[C@@H](CO)NC(=O)c1ccc2n(C3CC3)c(CC3CCC(CC3)C(F)(F)F)nc2c1 |wU:11.14,(15.87,.24,;14.53,1.01,;13.2,.24,;12.43,1.57,;13.97,-1.1,;11.87,-.53,;11.87,-2.07,;10.53,-2.84,;9.2,-2.07,;9.2,-.53,;10.53,.24,;7.87,-2.84,;7.87,-4.38,;6.53,-5.15,;6.53,-2.07,;5.2,-2.84,;5.2,-4.38,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;-.27,-.06,;-.74,1.41,;-1.89,2.44,;-.42,2.91,;-1.17,-1.3,;-2.71,-1.3,;-3.48,-2.64,;-2.71,-3.97,;-3.48,-5.3,;-5.02,-5.3,;-5.79,-3.97,;-5.02,-2.64,;-5.79,-6.64,;-6.56,-7.97,;-7.13,-5.87,;-4.46,-7.41,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,)|
CS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(CC4CCC(CC4)C(F)(F)F)nc3c2)cc1 |(13.97,-1.1,;13.2,.24,;14.53,1.01,;12.43,1.57,;11.87,-.53,;10.53,.24,;9.2,-.53,;9.2,-2.07,;7.87,-2.84,;6.53,-2.07,;5.2,-2.84,;5.2,-4.38,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;-.27,-.06,;-.74,1.41,;-1.89,2.44,;-.42,2.91,;-1.17,-1.3,;-2.71,-1.3,;-3.48,.03,;-5.02,.03,;-5.79,1.36,;-5.02,2.7,;-3.48,2.7,;-2.71,1.36,;-5.79,4.03,;-6.56,5.37,;-4.46,4.8,;-7.13,3.26,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,;10.53,-2.84,;11.87,-2.07,)|
CNS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(CC4CCC(CC4)C(F)(F)F)nc3c2)nc1 |(15.87,.24,;14.53,1.01,;13.2,.24,;12.43,1.57,;13.97,-1.1,;11.87,-.53,;11.87,-2.07,;10.53,-2.84,;9.2,-2.07,;7.87,-2.84,;6.53,-2.07,;5.2,-2.84,;5.2,-4.38,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;-.27,-.06,;-.74,1.41,;-1.89,2.44,;-.42,2.91,;-1.17,-1.3,;-2.71,-1.3,;-3.48,-2.64,;-2.71,-3.97,;-3.48,-5.3,;-5.02,-5.3,;-5.79,-3.97,;-5.02,-2.64,;-5.79,-6.64,;-6.56,-7.97,;-7.13,-5.87,;-4.46,-7.41,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,;9.2,-.53,;10.53,.24,)|
CS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(CC3CCC(CC3)C(F)(F)F)nc2c1 |wD:10.13,(13.97,-1.1,;13.2,.24,;14.53,1.01,;12.43,1.57,;11.87,-.53,;10.53,.24,;9.2,-.53,;9.2,-2.07,;10.53,-2.84,;11.87,-2.07,;7.87,-2.84,;7.87,-4.38,;6.53,-5.15,;6.53,-2.07,;5.2,-2.84,;5.2,-4.38,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;-.27,-.06,;-.74,1.41,;-1.89,2.44,;-.42,2.91,;-1.17,-1.3,;-2.71,-1.3,;-3.48,.03,;-5.02,.03,;-5.79,1.36,;-5.02,2.7,;-3.48,2.7,;-2.71,1.36,;-5.79,4.03,;-6.56,5.37,;-4.46,4.8,;-7.13,3.26,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,)|
CNS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(CC4CCC(CC4)C(F)(F)F)nc3c2)cc1 |(15.87,.24,;14.53,1.01,;13.2,.24,;12.43,1.57,;13.97,-1.1,;11.87,-.53,;10.53,.24,;9.2,-.53,;9.2,-2.07,;7.87,-2.84,;6.53,-2.07,;5.2,-2.84,;5.2,-4.38,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;-.27,-.06,;-.74,1.41,;-1.89,2.44,;-.42,2.91,;-1.17,-1.3,;-2.71,-1.3,;-3.48,-2.64,;-2.71,-3.97,;-3.48,-5.3,;-5.02,-5.3,;-5.79,-3.97,;-5.02,-2.64,;-5.79,-6.64,;-6.56,-7.97,;-7.13,-5.87,;-4.46,-7.41,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,;10.53,-2.84,;11.87,-2.07,)|
CCn1c(C[C@@H]2CC[C@@H](OC2)C(F)(F)F)nc2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC |r|
CCn1c(C[C@H]2CC[C@@H](OC2)C(F)(F)F)nc2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC |r|
CCn1c(C[C@@H]2CC[C@H](OC2)C(F)(F)F)nc2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC |r|
CCn1c(C[C@H]2CC[C@H](OC2)C(F)(F)F)nc2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC |r|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C)c(C[C@@H]3CC[C@@H](OC3)C(F)(F)F)nc2c1
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C)c(C[C@@H]3CC[C@H](OC3)C(F)(F)F)nc2c1
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C)c(C[C@H]3CC[C@@H](OC3)C(F)(F)F)nc2c1
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C)c(C[C@H]3CC[C@H](OC3)C(F)(F)F)nc2c1
CCS(=O)(=O)c1ccc(CNC(=O)c2cc(Br)c3n(C)c(CC4CCC(CC4)C(F)(F)F)nc3c2)cc1 |(11.46,-11.55,;10.12,-10.78,;10.12,-9.24,;8.58,-9.24,;11.66,-9.24,;10.12,-7.7,;11.46,-6.93,;11.46,-5.39,;10.12,-4.62,;10.12,-3.08,;8.79,-2.31,;8.79,-.77,;10.12,,;7.45,,;7.45,1.54,;6.12,2.31,;6.12,3.85,;4.79,1.54,;3.32,2.02,;2.85,3.48,;2.42,.77,;.88,.77,;.11,2.1,;-1.43,2.1,;-2.2,3.44,;-1.43,4.77,;.11,4.77,;.88,3.44,;-2.2,6.1,;-2.97,7.44,;-3.54,5.33,;-.87,6.87,;3.32,-.48,;4.79,,;6.12,-.77,;8.79,-5.39,;8.79,-6.93,)|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(nc3c2)C(O)[C@H]2CC[C@@H](CC2)C(F)(F)F)cc1 |r,wU:30.36,wD:27.29,(15.87,.24,;14.53,1.01,;13.2,.24,;12.43,1.57,;13.97,-1.1,;11.87,-.53,;10.53,.24,;9.2,-.53,;9.2,-2.07,;7.87,-2.84,;6.53,-2.07,;5.2,-2.84,;5.2,-4.38,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;-.27,-.06,;-.74,1.41,;-1.89,2.44,;-.42,2.91,;-1.17,-1.3,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,;-2.71,-1.3,;-3.48,.03,;-3.48,-2.64,;-5.02,-2.64,;-5.79,-3.97,;-5.02,-5.3,;-3.48,-5.3,;-2.71,-3.97,;-5.79,-6.64,;-6.56,-7.97,;-7.13,-5.87,;-4.46,-7.41,;10.53,-2.84,;11.87,-2.07,)|
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CCS(=O)(=O)c1ccc(cc1)[C@@H](COC(N)=O)NC(=O)c1ccc2n(C3CC3)c(CC3CCC(CC3)C(F)(F)F)nc2c1 |wU:11.17,(,-15.4,;1.33,-14.63,;1.33,-13.09,;2.87,-13.09,;-.21,-13.09,;1.33,-11.55,;2.67,-10.78,;2.67,-9.24,;1.33,-8.47,;,-9.24,;,-10.78,;1.33,-6.93,;,-6.16,;,-4.62,;-1.33,-3.85,;-2.67,-4.62,;-1.33,-2.31,;2.67,-6.16,;2.67,-4.62,;1.33,-3.85,;4,-3.85,;5.33,-4.62,;6.67,-3.85,;6.67,-2.31,;7.81,-1.28,;9.32,-1.6,;10.78,-1.12,;10.46,-2.63,;7.19,.13,;7.96,1.46,;7.19,2.79,;5.65,2.79,;4.88,4.13,;5.65,5.46,;7.19,5.46,;7.96,4.13,;4.88,6.8,;4.11,8.13,;6.21,7.57,;3.54,6.03,;5.65,-.03,;5.33,-1.54,;4,-2.31,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(CO[C@H]3CC[C@@H](CC3)C(F)(F)F)nc2c1 |wU:28.29,wD:11.14,31.36,(15.87,.24,;14.53,1.01,;13.2,.24,;12.43,1.57,;13.97,-1.1,;11.87,-.53,;10.53,.24,;9.2,-.53,;9.2,-2.07,;10.53,-2.84,;11.87,-2.07,;7.86,-2.84,;7.86,-4.38,;6.53,-5.15,;6.53,-2.07,;5.2,-2.84,;5.2,-4.38,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;-.27,-.06,;-.74,1.41,;-1.89,2.44,;-.42,2.91,;-1.17,-1.3,;-2.71,-1.3,;-3.48,-2.64,;-5.02,-2.64,;-5.79,-3.97,;-7.33,-3.97,;-8.1,-2.64,;-7.33,-1.3,;-5.79,-1.3,;-9.64,-2.64,;-11.18,-2.64,;-9.64,-1.1,;-9.64,-4.18,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,)|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(C3CC3)c(CO[C@H]3CC[C@@H](CC3)C(F)(F)F)nc2c1 |wU:31.36,wD:11.14,28.29,(15.87,.24,;14.53,1.01,;13.2,.24,;12.43,1.57,;13.97,-1.1,;11.87,-.53,;10.53,.24,;9.2,-.53,;9.2,-2.07,;10.53,-2.84,;11.87,-2.07,;7.86,-2.84,;7.86,-4.38,;6.53,-5.15,;6.53,-2.07,;5.2,-2.84,;5.2,-4.38,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;-.27,-.06,;-.74,1.41,;-1.89,2.44,;-.42,2.91,;-1.17,-1.3,;-2.71,-1.3,;-3.48,-2.64,;-5.02,-2.64,;-5.79,-1.3,;-7.33,-1.3,;-8.1,-2.64,;-7.33,-3.97,;-5.79,-3.97,;-9.64,-2.64,;-11.18,-2.64,;-9.64,-1.1,;-9.64,-4.18,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,)|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)cc1
CS(=O)(=O)c1ccc(CC(=O)Nc2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)cc1
OCCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)cc1
COCCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)cc1
CNS(=O)(=O)c1ccc(CC(=O)Nc2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)cc1
FC(F)(F)c1nc2cc(NC(=O)Cc3ccc(cc3)C#N)ccc2n1Cc1cccc2OC(F)(F)Oc12
CCOC(=O)Cc1ccc(CC(=O)Nc2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)cc1
OC(=O)Cc1ccc(CC(=O)Nc2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C2CC2)cc1
CS(=O)(=O)N1CCC(CC(=O)Nc2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)CC1
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)[C@@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C1CC1
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C1CCC1
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(C)(F)F
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)[C@H]1CCCO1
CCc1nc2cc(ccc2n1Cc1cccc2OC(F)(F)Oc12)C(=O)N[C@@H](CO)c1ccc(cc1)S(=O)(=O)CC
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)F
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C1(F)CC1
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C1(F)CCC1
CS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F
CS(=O)(=O)c1ccc(cc1)[C@@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F
CS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C1CC1
CS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C1CCC1
CS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)F
CS(=O)(=O)c1ccc(cc1)[C@@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)F
CS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C1(F)CC1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C2(F)CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(COC)nc3c2)cc1
CCc1nc2cc(ccc2n1Cc1cccc2OC(F)(F)Oc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(C)(C)C)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(C)C)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(C)nc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(CC(C)C)nc3c2)cc1
CS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C2CC2)cc1
CNS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C2CCC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(C)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)[C@H]2CCCO2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)[C@@H]2CCCO2)cc1
CS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C2(F)CC2)cc1
OCCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C2(F)CC2)cc1
CNS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C2(F)CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C2(F)CCC2)cc1
OCCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)F)cc1
OCCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)cc1
CNS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)cc1
OCCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C2CC2)cc1
CS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)[C@H](C)OC)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)[C@@H](C)OC)cc1
CS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)F)cc1
NS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)cc1
CCCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)cc1
COC(=O)CS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(C)(C)OC)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(OC)nc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)[C@H]2C[C@H]2C#N)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)[C@@H]2C[C@H]2C#N)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)[C@@H]2C[C@H]2C(=O)OC)cc1
CCS(=O)(=O)c1ccc(cc1)[C@H](COC)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)[C@H](COC)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C1CC1
CCS(=O)(=O)c1ccc(cc1)[C@H](COC)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C1(F)CC1
CCS(=O)(=O)c1ccc(nc1)[C@H](COC)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)nc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C2CC2)nc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C2CCC2)nc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(C)(F)F)nc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C2(F)CC2)nc1
CS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C2(F)CC2)nc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C2(F)CCC2)nc1
CS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)nc1
CS(=O)(=O)N1CCC(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)CC1
CS(=O)(=O)N1CCC(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C2CC2)CC1
CS(=O)(=O)N1CCC(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C2(F)CC2)CC1
COC(=O)CS(=O)(=O)N1CCC(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)CC1
CNC(=O)CS(=O)(=O)N1CCC(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)CC1
COC(=O)C(NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F)C1CCN(CC1)S(C)(=O)=O
CNS(=O)(=O)N1CCC(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)CC1
NC(=O)CS(=O)(=O)N1CCC(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)CC1
CNC(=O)CS(=O)(=O)N1CCC(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C2CC2)CC1
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4CCOc34)c(nc2c1)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OCOc34)c(nc2c1)C(F)(F)F
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cc(OC)cc(OC)c4)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4ccc(OC)c(c4)C#N)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4ccc(OC(F)(F)F)cc4)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4ccc(cc4)C#N)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4nnc5CCCn45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CC4CCCn5cc(C)nc45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc(OC)c4)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4ccnc(OC)c4)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc(c4)C#N)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cc(=O)[nH]c5ccccc45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(c(nc3c2)C(F)(F)F)C2(CC2)c2cccc(c2)C#N)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n([C@@H](C)c4cccc(c4)C#N)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n([C@H](C)c4cccc(c4)C#N)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cc(ccc4F)C#N)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5occc45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5CCOc45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5[nH]ncc45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OCOc45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc(c4)C(=O)OC)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cncc5[nH]ccc45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4CC(C)(C)Oc34)c(nc2c1)C1CC1
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4CCOc34)c(nc2c1)C1CC1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cc(OC)cc(OC)c4)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4ccc(OC(F)(F)F)cc4)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4ccc5OC(F)(F)Oc5c4)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4ccccc4OC(F)(F)F)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C[C@H]4CCN(C4)C(=O)OC(C)(C)C)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C[C@H]4CCCN4C(=O)OC(C)(C)C)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc(OC(F)(F)F)c4)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc(c4OC)C(F)(F)F)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cnn(CC(F)(F)F)c4)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc(c4)C#N)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc(OC(F)F)c4)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4ccn(CC(F)(F)F)n4)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cc(OC)cc(OC(F)(F)F)c4)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n([C@@H](C)c4cccc5OC(F)(F)Oc45)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4ccc(=O)n(CC(F)(F)F)c4)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5CC(C)(C)Oc45)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc(OC)c4OC)c(nc3c2)C2CC2)cc1
OC(=O)CC1CCC(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)CC1 |(5.2,-9,;6.53,-9.77,;6.53,-11.31,;7.87,-9,;7.87,-7.46,;9.2,-6.69,;9.2,-5.15,;7.87,-4.38,;7.87,-2.84,;6.53,-2.07,;5.2,-2.84,;5.2,-4.38,;3.86,-2.07,;3.86,-.53,;2.53,.24,;1.2,-.53,;-.27,-.06,;-.74,1.41,;.29,2.55,;1.79,2.23,;2.82,3.38,;2.35,4.84,;.84,5.16,;.07,6.49,;-1.44,6.17,;-1.6,7.71,;-2.98,6.17,;-1.6,4.64,;-.19,4.02,;-1.17,-1.3,;-.27,-2.55,;1.2,-2.07,;2.53,-2.84,;-2.71,-1.3,;-4.25,-1.3,;-2.71,-2.84,;-2.71,.24,;6.53,-5.15,;6.53,-6.69,)|
FC(F)(F)c1nc2cc(ccc2n1Cc1cccc2OC(F)(F)Oc12)C(=O)NCc1ccc2nn[nH]c2c1
OC[C@H](NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F)c1ccc(cc1)C#N
CCS(=O)(=O)c1ccc([C@H](CO)NC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)c(F)c1
COc1cc(Cn2c(nc3cc(ccc23)C(=O)NCc2ccc(cc2)S(=O)(=O)CCO)C(F)(F)F)cc(OC)c1
CCc1nc2cc(ccc2n1[C@@H](C)c1cccc2OC(F)(F)Oc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCc1nc2cc(ccc2n1[C@H](C)c1cccc2OC(F)(F)Oc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)c(O)c1
COC(=O)CS(=O)(=O)N1CCC(CNC(=O)c2ccc3n(Cc4cccc5[nH]ncc45)c(nc3c2)C(F)(F)F)CC1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cc(OC)cc(OC)c4)c(nc3c2)C(F)(F)F)nc1
FC(F)(F)c1nc2cc(ccc2n1Cc1cccc2OC(F)(F)Oc12)C(=O)NCc1ccc2c(c1)[nH]ccc2=O
CCS(=O)(=O)c1ccc(nc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F
CCS(=O)(=O)c1ccc(nc1)[C@@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F
CCS(=O)(=O)c1ccc(nc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)F
CCS(=O)(=O)c1ccc(nc1)[C@@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)F
CCS(=O)(=O)c1ccc(nc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C1CCC1
CCS(=O)(=O)c1ccc(nc1)[C@@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C1CCC1
CCS(=O)(=O)c1ccc(nc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C1CC1
CCS(=O)(=O)c1ccc(nc1)[C@@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C1CC1
CCS(=O)(=O)c1ccc(nc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C1(F)CC1
CCS(=O)(=O)c1ccc(nc1)[C@@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C1(F)CC1
CS(=O)(=O)c1ccc(nc1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc(OC)c4F)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5cnn(C)c45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4nc(C)cc(n4)C(F)(F)F)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5cn(C)nc45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5nc(C)n(C)c45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5n(C)ncc45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5cn[nH]c45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5nn(C)cc45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc(=O)n4CC(F)(F)F)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CC4CCN(CC4)C(=O)OC(C)(C)C)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccn(C)c4=O)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5ocnc45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OCCOc45)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n([C@H](C)c4cccc5OC(F)(F)Oc45)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4ccccc4)c(C)nc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5nonc45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5ncoc45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cc(O)cc(OC(F)(F)F)c4)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc(O)c4O)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CC4CCN(CC(F)(F)F)CC4)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C[C@H]4CCN(CC(F)(F)F)C4)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C[C@@H]4CCN(CC(F)(F)F)C4)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CC4CCN(CC4)c4ncc(F)cn4)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C[C@H]4CCN(C4)c4ncc(F)cn4)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C[C@H]4CCCN4c4ncc(F)cn4)c(nc3c2)C2CC2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)[n+]([O-])c1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)N(C)C)cc1
OCCS(=O)(=O)N1CCC(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)CC1
CS(=O)(=O)N1CCC(CC1)[C@@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F
CS(=O)(=O)N1CCC(CC1)[C@H](CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)[C@H](CC(O)=O)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)[C@H](COCC(O)=O)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)[C@H](CC(=O)NC)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)[C@H](CC(N)=O)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F
CNC(=O)CS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(cc1)C(O)C(=O)Nc1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)[C@H](O)C(=O)Nc1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(cc1)[C@@H](O)C(=O)Nc1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F |r|
CN1CCN(CCC1CNC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F)S(C)(=O)=O
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OCCc45)c(nc3c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(Cc4cccc5OC(F)(F)Oc45)c(nc3c2)C(=O)OC)cc1
CCS(=O)(=O)c1ccc(cc1)C(CO)(CO)NC(=O)c1ccc2n(Cc3cccc4OC(F)(F)Oc34)c(nc2c1)C(F)(F)F
OC(=O)Cc1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)F)cc1 |(10.4,1.93,;8.86,1.93,;8.09,3.26,;8.09,.59,;6.55,.59,;5.78,-.74,;4.24,-.74,;3.46,.59,;1.93,.59,;1.15,-.74,;-.39,-.74,;-1.15,.59,;-1.15,-2.07,;-2.7,-2.07,;-3.46,-3.41,;-5,-3.41,;-5.78,-4.74,;-5.78,-2.07,;-5,-.74,;-5.78,.59,;-3.46,-.74,;-7.32,-2.07,;-8.09,-3.41,;-9.63,-3.41,;-10.4,-2.07,;-9.63,-.74,;-8.09,-.74,;-7.32,.59,;-8.09,1.93,;-9.63,1.93,;-7.32,3.26,;4.24,1.93,;5.78,1.93,)|
Cc1cc(NC(=O)NCc2ccc(CC(O)=O)cc2)cc(C)c1-c1ccccc1OC(F)F |(-5.77,-4.74,;-5,-3.41,;-3.46,-3.41,;-2.7,-2.07,;-1.15,-2.07,;-.39,-.74,;-1.15,.59,;1.15,-.74,;1.92,.59,;3.46,.59,;4.24,-.74,;5.77,-.74,;6.55,.59,;8.08,.59,;8.85,1.93,;10.39,1.93,;8.08,3.26,;5.77,1.93,;4.24,1.93,;-3.46,-.74,;-5,-.74,;-5.78,.59,;-5.77,-2.07,;-7.31,-2.07,;-8.08,-3.41,;-9.62,-3.41,;-10.39,-2.07,;-9.62,-.74,;-8.08,-.74,;-7.31,.59,;-8.08,1.93,;-9.62,1.93,;-7.31,3.26,)|
OC(=O)Cc1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1F |(10.4,2.67,;8.86,2.67,;8.09,4,;8.09,1.33,;6.55,1.33,;5.78,2.67,;4.24,2.67,;3.47,1.33,;1.93,1.33,;1.15,,;-.39,,;-1.15,1.33,;-1.15,-1.33,;-2.7,-1.33,;-3.47,-2.67,;-5.01,-2.67,;-5.78,-4,;-5.78,-1.33,;-5.01,,;-5.78,1.33,;-3.47,,;-7.32,-1.33,;-8.09,-2.67,;-9.63,-2.67,;-10.4,-1.33,;-9.63,,;-8.09,,;-7.32,1.33,;-8.09,2.67,;-7.32,4,;-9.63,2.67,;-8.86,4,;4.24,,;5.78,,;6.55,-1.33,)|
OC(=O)Cc1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1Cl |(10.4,2.67,;8.86,2.67,;8.09,4,;8.09,1.33,;6.55,1.33,;5.78,2.67,;4.24,2.67,;3.46,1.33,;1.93,1.33,;1.15,,;-.38,,;-1.15,1.33,;-1.15,-1.33,;-2.7,-1.33,;-3.46,-2.67,;-5.01,-2.67,;-5.78,-4,;-5.78,-1.33,;-5.01,,;-5.78,1.33,;-3.46,,;-7.32,-1.33,;-8.09,-2.67,;-9.63,-2.67,;-10.4,-1.33,;-9.63,,;-8.09,,;-7.32,1.33,;-8.09,2.67,;-7.32,4,;-9.63,2.67,;-8.86,4,;4.24,,;5.78,,;6.55,-1.33,)|
Cc1cc(CC(O)=O)ccc1CNC(=O)Nc1cc(Cl)c(c(Cl)c1)-c1ccccc1OC(F)(F)F |(3.47,-1.33,;4.24,,;5.78,,;6.55,1.33,;8.09,1.33,;8.86,2.67,;10.4,2.67,;8.09,4,;5.78,2.67,;4.24,2.67,;3.47,1.33,;1.93,1.33,;1.16,,;-.38,,;-1.16,1.33,;-1.16,-1.33,;-2.7,-1.33,;-3.47,-2.67,;-5.01,-2.67,;-5.78,-4,;-5.78,-1.33,;-5.01,,;-5.78,1.33,;-3.47,,;-7.32,-1.33,;-8.09,-2.67,;-9.63,-2.67,;-10.4,-1.33,;-9.63,,;-8.09,,;-7.32,1.33,;-8.09,2.67,;-7.32,4,;-9.63,2.67,;-8.86,4,)|
OC(=O)Cc1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)c(F)c1 |(10.4,2.67,;8.86,2.67,;8.09,4,;8.09,1.33,;6.55,1.33,;5.78,2.67,;4.24,2.67,;3.46,1.33,;1.93,1.33,;1.15,,;-.38,,;-1.15,1.33,;-1.15,-1.33,;-2.7,-1.33,;-3.46,-2.67,;-5.01,-2.67,;-5.78,-4,;-5.78,-1.33,;-5.01,,;-5.78,1.33,;-3.46,,;-7.32,-1.33,;-8.09,-2.67,;-9.63,-2.67,;-10.4,-1.33,;-9.63,,;-8.09,,;-7.32,1.33,;-8.09,2.67,;-7.32,4,;-9.63,2.67,;-8.86,4,;4.24,,;3.46,-1.33,;5.78,,)|
OC(=O)CCc1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(10.78,4,;10.01,2.67,;10.78,1.33,;8.47,2.67,;7.7,1.33,;6.16,1.33,;5.39,,;3.85,,;3.08,1.33,;1.54,1.33,;.77,,;-.77,,;-1.54,1.33,;-1.54,-1.33,;-3.08,-1.33,;-3.85,-2.67,;-5.39,-2.67,;-6.16,-4,;-6.16,-1.33,;-5.39,,;-6.16,1.33,;-3.85,,;-7.7,-1.33,;-8.47,-2.67,;-10.01,-2.67,;-10.78,-1.33,;-10.01,,;-8.47,,;-7.7,1.33,;-8.47,2.67,;-7.7,4,;-10.01,2.67,;-9.24,4,;3.85,2.67,;5.39,2.67,)|
OC(C(O)=O)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(8.86,,;8.09,1.33,;8.86,2.67,;10.4,2.67,;8.09,4,;6.55,1.33,;5.78,2.67,;4.24,2.67,;3.46,1.33,;1.93,1.33,;1.15,,;-.38,,;-1.15,1.33,;-1.15,-1.33,;-2.7,-1.33,;-3.46,-2.67,;-5.01,-2.67,;-5.78,-4,;-5.78,-1.33,;-5.01,,;-5.78,1.33,;-3.46,,;-7.32,-1.33,;-8.09,-2.67,;-9.63,-2.67,;-10.4,-1.33,;-9.63,,;-8.09,,;-7.32,1.33,;-8.09,2.67,;-7.32,4,;-9.63,2.67,;-8.86,4,;4.24,,;5.78,,)|
OC(=O)C(F)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(10.4,2.67,;8.86,2.67,;8.09,4,;8.09,1.33,;8.86,,;6.55,1.33,;5.78,2.67,;4.24,2.67,;3.46,1.33,;1.93,1.33,;1.15,,;-.38,,;-1.15,1.33,;-1.15,-1.33,;-2.7,-1.33,;-3.46,-2.67,;-5.01,-2.67,;-5.78,-4,;-5.78,-1.33,;-5.01,,;-5.78,1.33,;-3.46,,;-7.32,-1.33,;-8.09,-2.67,;-9.63,-2.67,;-10.4,-1.33,;-9.63,,;-8.09,,;-7.32,1.33,;-8.09,2.67,;-7.32,4,;-9.63,2.67,;-8.86,4,;4.24,,;5.78,,)|
CCOC(=O)C1CN(Cc2ccncc2)CCN1Cc1ccc(cc1)-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCOC(=O)CC1CN(Cc2ccncc2)CCN1Cc1ccc(cc1)-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
OC(=O)C1CN(Cc2ccncc2)CCN1Cc1ccc(cc1)-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
OC(=O)CC1CN(Cc2ccncc2)CCN1Cc1ccc(cc1)-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCOC(=O)C1CN(Cc2ccc(cc2)-c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)CCN1Cc1ccncc1
CCOC(=O)CC1CN(Cc2ccc(cc2)-c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)CCN1Cc1ccncc1
OC(=O)C1CN(Cc2ccc(cc2)-c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)CCN1Cc1ccncc1
OC(=O)CC1CN(Cc2ccc(cc2)-c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)CCN1Cc1ccncc1
CC(C)NC(=O)C1CN(Cc2ccncc2)CCN1Cc1ccc(cc1)-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CC(C)NC(=O)C1CN(Cc2ccc(cc2)-c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)CCN1Cc1ccncc1
CC(C)OC(=O)CC1CN(Cc2ccc(cc2)-c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)CCN1Cc1ccncc1
OCCOC(=O)CC1CN(Cc2ccc(cc2)-c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)CCN1Cc1ccncc1
CCOCCOC(=O)CC1CN(Cc2ccc(cc2)-c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)CCN1Cc1ccncc1
NCCOC(=O)CC1CN(Cc2ccc(cc2)-c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)CCN1Cc1ccncc1
CCOC(=O)CC1CN(Cc2ccc(c(C)c2)-c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)CCN1Cc1ccncc1
CCOC(=O)C[C@H]1CN(Cc2ccc(c(C)c2)-c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)CCN1Cc1ccncc1
CCOC(=O)C[C@H]1CN(Cc2ccc(cc2)-c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)CCN1Cc1ccncc1
CCOC(=O)C[C@@H]1CN(Cc2ccc(cc2)-c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)CCN1Cc1ccncc1
Cc1cc(CN2CCN(Cc3ccncc3)[C@@H](CC(O)=O)C2)ccc1-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCOCCOC(=O)C[C@H]1CN(Cc2ccc(cc2)-c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)CCN1Cc1ccncc1
CCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(C[C@@H](C)C(F)(F)F)cc1OC |r,wU:9.8,wD:27.29,12.15,(4.2,-1.53,;2.67,-1.69,;1.76,-.45,;2.24,1.02,;.99,1.92,;.99,3.46,;-.34,4.23,;2.32,4.23,;2.32,5.77,;3.66,6.54,;3.66,8.08,;4.99,8.85,;6.33,8.08,;6.33,6.54,;4.99,5.77,;7.66,8.85,;7.66,7.31,;7.66,10.39,;8.99,8.08,;-.25,1.02,;-1.72,1.49,;.22,-.45,;-.68,-1.69,;-2.22,-1.53,;-3.12,-2.78,;-2.49,-4.18,;-3.4,-5.43,;-4.93,-5.27,;-5.56,-3.86,;-5.84,-6.51,;-6.74,-7.76,;-7.08,-5.61,;-4.59,-7.42,;-.96,-4.34,;-.06,-3.1,;1.47,-3.26,;2.1,-4.67,)|
CCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:12.15,(-2.05,-2.81,;-2.67,-1.41,;-1.77,-.16,;-2.25,1.3,;-1,2.21,;-1,3.75,;.33,4.52,;-2.33,4.52,;-2.33,6.06,;-3.67,6.83,;-5,6.06,;-6.33,6.83,;-6.33,8.37,;-5,9.14,;-3.67,8.37,;-7.67,9.14,;-8.7,8,;-6.64,10.28,;-9.17,9.46,;.25,1.3,;1.71,1.78,;-.23,-.16,;.68,-1.41,;.05,-2.81,;.95,-4.06,;2.49,-3.9,;3.39,-5.14,;4.92,-4.98,;5.08,-6.51,;4.76,-3.45,;6.45,-4.82,;7.99,-4.66,;6.62,-6.35,;6.29,-3.29,;3.11,-2.49,;2.21,-1.25,;2.83,.16,;4.37,.32,;4.99,1.73,;5.27,-.92,)|
CCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(C[C@H](C)C(F)(F)F)cc1OC |r,wU:9.8,27.29,wD:12.15,(4.2,-1.53,;2.67,-1.69,;1.76,-.45,;2.24,1.02,;.99,1.92,;.99,3.46,;-.34,4.23,;2.32,4.23,;2.32,5.77,;3.66,6.54,;3.66,8.08,;4.99,8.85,;6.33,8.08,;6.33,6.54,;4.99,5.77,;7.66,8.85,;8.69,7.71,;6.63,10,;9.17,9.17,;-.25,1.02,;-1.72,1.49,;.22,-.45,;-.68,-1.69,;-2.22,-1.53,;-3.12,-2.78,;-2.49,-4.18,;-3.4,-5.43,;-4.93,-5.27,;-5.56,-3.86,;-5.84,-6.51,;-6.74,-7.76,;-7.08,-5.61,;-4.59,-7.42,;-.96,-4.34,;-.06,-3.1,;1.47,-3.26,;2.1,-4.67,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(C)c1-c1ccc(C[C@H](C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,28.30,wD:9.9,13.16,(-1.71,-2.4,;-2.33,-1,;-1.43,.25,;-1.9,1.71,;-.66,2.62,;-.66,4.16,;.67,4.93,;-1.99,4.93,;-1.99,6.47,;-3.33,7.24,;-1.94,7.92,;-4.14,5.93,;-5.68,5.99,;-6.4,7.35,;-5.59,8.65,;-4.05,8.6,;-7.94,7.4,;-8.97,6.26,;-6.91,8.55,;-9.45,7.72,;.59,1.71,;2.05,2.19,;.11,.25,;1.02,-1,;.39,-2.4,;1.3,-3.65,;2.83,-3.49,;3.73,-4.73,;3.11,-6.14,;1.57,-6.3,;4.01,-7.39,;4.92,-8.63,;5.26,-6.48,;2.76,-8.29,;3.45,-2.08,;2.55,-.83,;3.17,.57,;4.71,.73,;5.33,2.14,;5.61,-.51,)|
CCn1nc(C(=O)NC[C@]2(O)CC[C@H](C[C@H]2NBr)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:9.9,15.16,13.18,(-2.19,-2.98,;-2.82,-1.57,;-1.91,-.33,;-2.39,1.14,;-1.14,2.04,;-1.14,3.58,;.19,4.35,;-2.48,4.35,;-2.48,5.89,;-3.81,6.66,;-2.43,7.34,;-4.53,8.02,;-6.07,8.08,;-6.89,6.77,;-6.17,5.41,;-4.63,5.36,;-3.9,4,;-4.72,2.69,;-8.43,6.83,;-9.46,5.68,;-7.4,7.97,;-9.94,7.15,;.1,1.14,;1.57,1.62,;-.37,-.33,;.53,-1.57,;-.1,-2.98,;.81,-4.22,;2.34,-4.06,;3.25,-5.31,;4.78,-5.15,;4.94,-6.68,;4.62,-3.62,;6.31,-4.99,;7.84,-4.83,;6.47,-6.52,;6.15,-3.46,;2.97,-2.66,;2.06,-1.41,;2.69,-0,;4.22,.16,;4.85,1.56,;5.13,-1.09,)|
CCn1nc(C(=O)NC[C@]2(O)CC[C@H](CC2NBr)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:9.9,13.18,(-2.19,-2.98,;-2.82,-1.57,;-1.91,-.33,;-2.39,1.14,;-1.14,2.04,;-1.14,3.58,;.19,4.35,;-2.48,4.35,;-2.48,5.89,;-3.81,6.66,;-2.43,7.34,;-4.53,8.02,;-6.07,8.08,;-6.89,6.77,;-6.17,5.41,;-4.63,5.36,;-3.9,4,;-4.72,2.69,;-8.43,6.83,;-9.46,5.68,;-7.4,7.97,;-9.94,7.15,;.1,1.14,;1.57,1.62,;-.37,-.33,;.53,-1.57,;-.1,-2.98,;.81,-4.22,;2.34,-4.06,;3.25,-5.31,;4.78,-5.15,;4.94,-6.68,;4.62,-3.62,;6.31,-4.99,;7.84,-4.83,;6.47,-6.52,;6.15,-3.46,;2.97,-2.66,;2.06,-1.41,;2.69,-0,;4.22,.16,;4.85,1.56,;5.13,-1.09,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2NBr)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.9,13.18,wD:9.8,(-2.19,-2.98,;-2.82,-1.57,;-1.91,-.33,;-2.39,1.14,;-1.14,2.04,;-1.14,3.58,;.19,4.35,;-2.48,4.35,;-2.48,5.89,;-3.81,6.66,;-2.43,7.34,;-4.53,8.02,;-6.07,8.08,;-6.89,6.77,;-6.17,5.41,;-4.63,5.36,;-3.9,4,;-4.72,2.69,;-8.43,6.83,;-9.46,5.68,;-7.4,7.97,;-9.94,7.15,;.1,1.14,;1.57,1.62,;-.37,-.33,;.53,-1.57,;-.1,-2.98,;.81,-4.22,;2.34,-4.06,;3.25,-5.31,;4.78,-5.15,;4.94,-6.68,;4.62,-3.62,;6.31,-4.99,;7.84,-4.83,;6.47,-6.52,;6.15,-3.46,;2.97,-2.66,;2.06,-1.41,;2.69,-0,;4.22,.16,;4.85,1.56,;5.13,-1.09,)|
CCn1nc(C(=O)NC[C@@H]2CC[C@H](CN2Br)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:12.16,(-2.02,-3.25,;-2.65,-1.84,;-1.74,-.6,;-2.22,.87,;-.97,1.77,;-.97,3.31,;-2.31,4.08,;.36,4.08,;.36,5.62,;1.7,6.39,;3.03,5.62,;4.36,6.39,;4.36,7.93,;3.03,8.7,;1.7,7.93,;.36,8.7,;5.7,8.7,;6.73,7.56,;4.67,9.85,;7.2,9.02,;.27,.87,;1.74,1.34,;-.2,-.6,;.7,-1.84,;.08,-3.25,;.98,-4.49,;2.51,-4.33,;3.42,-5.58,;2.79,-6.99,;4.2,-7.61,;1.39,-6.36,;2.17,-8.39,;1.54,-9.8,;3.57,-9.02,;.76,-7.77,;3.14,-2.93,;2.23,-1.68,;2.86,-.27,;4.39,-.11,;5.02,1.29,;5.3,-1.36,)|
CCn1nc(C(=O)NC[C@H]2CC[C@@H](CN2Br)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:12.16,wD:9.8,(-2.14,-2.89,;-2.77,-1.49,;-1.86,-.24,;-2.34,1.22,;-1.09,2.13,;-1.09,3.67,;.24,4.44,;-2.43,4.44,;-2.43,5.98,;-3.76,6.75,;-3.76,8.29,;-5.09,9.06,;-6.43,8.29,;-6.43,6.75,;-5.09,5.98,;-5.09,4.44,;-7.76,9.06,;-8.79,7.92,;-6.73,10.2,;-9.27,9.38,;.15,1.22,;1.62,1.7,;-.32,-.24,;.58,-1.49,;-.04,-2.89,;.86,-4.14,;2.39,-3.98,;3.3,-5.22,;4.83,-5.06,;4.99,-6.59,;4.67,-3.53,;6.36,-4.9,;7.89,-4.74,;6.52,-6.43,;6.2,-3.37,;3.02,-2.57,;2.11,-1.33,;2.74,.08,;4.27,.24,;4.9,1.65,;5.18,-1,)|
CCn1nc(C(=O)NC[C@@H]2CC[C@H](CN2Br)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:12.16,(-2.14,-2.89,;-2.77,-1.49,;-1.86,-.24,;-2.34,1.22,;-1.09,2.13,;-1.09,3.67,;.24,4.44,;-2.43,4.44,;-2.43,5.98,;-3.76,6.75,;-3.76,8.29,;-5.09,9.06,;-6.43,8.29,;-6.43,6.75,;-5.09,5.98,;-5.09,4.44,;-7.76,9.06,;-8.79,7.92,;-6.73,10.2,;-9.27,9.38,;.15,1.22,;1.62,1.7,;-.32,-.24,;.58,-1.49,;-.04,-2.89,;.86,-4.14,;2.39,-3.98,;3.3,-5.22,;4.83,-5.06,;4.99,-6.59,;4.67,-3.53,;6.36,-4.9,;7.89,-4.74,;6.52,-6.43,;6.2,-3.37,;3.02,-2.57,;2.11,-1.33,;2.74,.08,;4.27,.24,;4.9,1.65,;5.18,-1,)|
CCn1nc(C(=O)NC[C@H]2CC[C@H](CN2Br)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wD:9.8,12.16,(-1.9,-3.25,;-2.53,-1.85,;-1.62,-.6,;-2.1,.86,;-.85,1.77,;-.85,3.31,;-2.19,4.08,;.48,4.08,;.48,5.62,;1.81,6.39,;3.15,5.62,;4.48,6.39,;4.48,7.93,;3.15,8.7,;1.81,7.93,;.48,8.7,;5.81,8.7,;6.84,7.56,;4.78,9.84,;7.32,9.02,;.39,.86,;1.86,1.34,;-.08,-.6,;.82,-1.85,;.19,-3.25,;1.1,-4.5,;2.63,-4.34,;3.54,-5.58,;2.91,-6.99,;4.32,-7.62,;1.5,-6.36,;2.28,-8.4,;1.66,-9.8,;3.69,-9.02,;.88,-7.77,;3.26,-2.93,;2.35,-1.69,;2.98,-.28,;4.51,-.12,;5.14,1.29,;5.42,-1.36,)|
CCn1nc(C(=O)NC[C@@H]2CC[C@@H](CN2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,12.15,(-1.93,-2.82,;-2.56,-1.41,;-1.65,-.16,;-2.13,1.3,;-.88,2.21,;-.88,3.75,;.45,4.52,;-2.22,4.52,;-2.22,6.06,;-3.55,6.83,;-3.55,8.37,;-4.88,9.14,;-6.22,8.37,;-6.22,6.83,;-4.88,6.06,;-7.55,9.14,;-8.58,7.99,;-6.52,10.28,;-9.06,9.46,;.36,1.3,;1.83,1.78,;-.11,-.16,;.79,-1.41,;.17,-2.82,;1.07,-4.06,;2.6,-3.9,;3.51,-5.15,;5.04,-4.99,;5.2,-6.52,;4.88,-3.45,;6.57,-4.83,;8.1,-4.66,;6.73,-6.36,;6.41,-3.29,;3.23,-2.49,;2.33,-1.25,;2.95,.16,;4.48,.32,;5.11,1.73,;5.39,-.93,)|
CCn1nc(C(=O)NC[C@H]2CC[C@H](CN2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wD:9.8,12.15,(-1.93,-2.82,;-2.56,-1.41,;-1.65,-.16,;-2.13,1.3,;-.88,2.21,;-.88,3.75,;.45,4.52,;-2.22,4.52,;-2.22,6.06,;-3.55,6.83,;-3.55,8.37,;-4.88,9.14,;-6.22,8.37,;-6.22,6.83,;-4.88,6.06,;-7.55,9.14,;-8.58,7.99,;-6.52,10.28,;-9.06,9.46,;.36,1.3,;1.83,1.78,;-.11,-.16,;.79,-1.41,;.17,-2.82,;1.07,-4.06,;2.6,-3.9,;3.51,-5.15,;5.04,-4.99,;5.2,-6.52,;4.88,-3.45,;6.57,-4.83,;8.1,-4.66,;6.73,-6.36,;6.41,-3.29,;3.23,-2.49,;2.33,-1.25,;2.95,.16,;4.48,.32,;5.11,1.73,;5.39,-.93,)|
CCn1nc(C(=O)NC[C@@H]2CC[C@H](CO2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:12.15,(-1.93,-2.82,;-2.56,-1.41,;-1.65,-.16,;-2.13,1.3,;-.88,2.21,;-.88,3.75,;.45,4.52,;-2.22,4.52,;-2.22,6.06,;-3.55,6.83,;-3.55,8.37,;-4.88,9.14,;-6.22,8.37,;-6.22,6.83,;-4.88,6.06,;-7.55,9.14,;-8.58,7.99,;-6.52,10.28,;-9.06,9.46,;.36,1.3,;1.83,1.78,;-.11,-.16,;.79,-1.41,;.17,-2.82,;1.07,-4.06,;2.6,-3.9,;3.51,-5.15,;5.04,-4.99,;5.2,-6.52,;4.88,-3.45,;6.57,-4.83,;8.1,-4.66,;6.73,-6.36,;6.41,-3.29,;3.23,-2.49,;2.33,-1.25,;2.95,.16,;4.48,.32,;5.11,1.73,;5.39,-.93,)|
CCn1nc(C(=O)NC[C@H]2CC[C@@H](CO2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:12.15,wD:9.8,(-1.93,-2.82,;-2.56,-1.41,;-1.65,-.16,;-2.13,1.3,;-.88,2.21,;-.88,3.75,;.45,4.52,;-2.22,4.52,;-2.22,6.06,;-3.55,6.83,;-3.55,8.37,;-4.88,9.14,;-6.22,8.37,;-6.22,6.83,;-4.88,6.06,;-7.55,9.14,;-8.58,7.99,;-6.52,10.28,;-9.06,9.46,;.36,1.3,;1.83,1.78,;-.11,-.16,;.79,-1.41,;.17,-2.82,;1.07,-4.06,;2.6,-3.9,;3.51,-5.15,;5.04,-4.99,;5.2,-6.52,;4.88,-3.45,;6.57,-4.83,;8.1,-4.66,;6.73,-6.36,;6.41,-3.29,;3.23,-2.49,;2.33,-1.25,;2.95,.16,;4.48,.32,;5.11,1.73,;5.39,-.93,)|
CCn1nc(C(=O)NC[C@H]2CC[C@H](CO2)S(C)(=O)=O)c(Cl)c1-c1ccc(N[C@H](C)C(F)(F)F)cc1OC |r,wU:27.29,wD:9.8,12.15,(4.31,-1.54,;2.78,-1.7,;1.88,-.45,;2.35,1.01,;1.11,1.92,;1.11,3.46,;-.23,4.23,;2.44,4.23,;2.44,5.77,;3.78,6.54,;5.11,5.77,;6.44,6.54,;6.44,8.08,;5.11,8.85,;3.78,8.08,;7.78,8.85,;8.81,7.7,;6.75,9.99,;9.28,9.17,;-.14,1.01,;-1.6,1.49,;.34,-.45,;-.57,-1.7,;-2.1,-1.54,;-3,-2.78,;-2.38,-4.19,;-3.28,-5.44,;-4.81,-5.27,;-5.44,-3.87,;-5.72,-6.52,;-6.62,-7.77,;-6.97,-5.61,;-4.47,-7.43,;-.85,-4.35,;.06,-3.1,;1.59,-3.27,;2.22,-4.67,)|
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CCCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(N[C@H](C)C(F)(F)F)cc1OC |r,wU:10.9,28.30,wD:13.16,(4.96,-2,;4.05,-.76,;2.52,-.92,;1.62,.33,;2.09,1.79,;.85,2.7,;.85,4.24,;-.49,5.01,;2.18,5.01,;2.18,6.55,;3.51,7.32,;3.51,8.86,;4.85,9.63,;6.18,8.86,;6.18,7.32,;4.85,6.55,;7.51,9.63,;8.54,8.48,;6.48,10.77,;9.02,9.95,;-.4,1.79,;-1.86,2.27,;.08,.33,;-.83,-.92,;-2.36,-.76,;-3.27,-2,;-2.64,-3.41,;-3.55,-4.65,;-5.08,-4.49,;-5.7,-3.09,;-5.98,-5.74,;-6.89,-6.99,;-4.74,-6.64,;-7.23,-4.83,;-1.11,-3.57,;-.2,-2.32,;1.33,-2.48,;1.95,-3.89,)|
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CCn1nc(C(=O)NC[C@@]2(CC[C@@H](CC2)S(C)(=O)=O)C(N)=O)c(Cl)c1-c1ccc(N[C@H](C)C(F)(F)F)cc1OC |r,wU:9.8,30.32,12.15,wD:9.19,(3.43,-1.63,;1.89,-1.79,;.99,-.55,;1.47,.92,;.22,1.82,;.22,3.36,;-1.11,4.13,;1.55,4.13,;1.55,5.67,;2.89,6.44,;3.7,5.14,;5.24,5.19,;5.97,6.55,;5.15,7.86,;3.61,7.8,;7.5,6.6,;7.82,5.1,;7.18,8.11,;8.97,6.13,;1.5,7.12,;.23,6.26,;1.4,8.65,;-1.03,.92,;-2.49,1.39,;-.55,-.55,;-1.46,-1.79,;-2.99,-1.63,;-3.89,-2.88,;-3.27,-4.29,;-4.17,-5.53,;-5.7,-5.37,;-6.33,-3.96,;-6.61,-6.62,;-7.51,-7.86,;-7.85,-5.71,;-5.36,-7.52,;-1.73,-4.45,;-.83,-3.2,;.7,-3.36,;1.33,-4.77,)|
CCn1nc(C(=O)NC[C@]2(CC[C@@H](CC2)S(C)(=O)=O)C(N)=O)c(Cl)c1-c1ccc(N[C@H](C)C(F)(F)F)cc1OC |r,wU:30.32,9.19,12.15,wD:9.8,(3.43,-1.63,;1.89,-1.79,;.99,-.55,;1.47,.92,;.22,1.82,;.22,3.36,;-1.11,4.13,;1.55,4.13,;1.55,5.67,;2.89,6.44,;3.7,5.14,;5.24,5.19,;5.97,6.55,;5.15,7.86,;3.61,7.8,;7.5,6.6,;7.5,5.06,;7.5,8.14,;8.84,5.83,;1.5,7.12,;.23,6.26,;1.4,8.65,;-1.03,.92,;-2.49,1.39,;-.55,-.55,;-1.46,-1.79,;-2.99,-1.63,;-3.89,-2.88,;-3.27,-4.29,;-4.17,-5.53,;-5.7,-5.37,;-6.33,-3.96,;-6.61,-6.62,;-7.51,-7.86,;-7.85,-5.71,;-5.36,-7.52,;-1.73,-4.45,;-.83,-3.2,;.7,-3.36,;1.33,-4.77,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(C[C@@H](C)C(F)(F)F)cc1OC |r,wU:9.8,wD:9.9,28.30,13.16,(4.71,-1.61,;3.18,-1.77,;2.27,-.52,;2.75,.94,;1.5,1.85,;1.5,3.39,;2.84,4.16,;.17,4.16,;.17,5.7,;1.5,6.47,;1.4,4.93,;.78,7.83,;1.6,9.13,;3.14,9.08,;3.86,7.72,;3.04,6.41,;3.95,10.39,;4.27,8.88,;3.63,11.89,;5.42,9.91,;.26,.94,;-1.21,1.42,;.73,-.52,;-.17,-1.77,;-1.7,-1.61,;-2.61,-2.85,;-1.98,-4.26,;-2.89,-5.51,;-4.42,-5.35,;-5.04,-3.94,;-5.32,-6.59,;-6.23,-7.84,;-4.08,-7.5,;-6.57,-5.69,;-.45,-4.42,;.46,-3.18,;1.99,-3.34,;2.61,-4.74,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(C[C@H](C)C(F)(F)F)cc1OC |r,wU:9.8,28.30,wD:9.9,13.16,(4.02,-1.61,;2.49,-1.77,;1.59,-.52,;2.06,.94,;.82,1.85,;.82,3.39,;-.52,4.16,;2.15,4.16,;2.15,5.7,;3.49,6.47,;3.38,4.93,;2.76,7.83,;3.58,9.13,;5.12,9.08,;5.84,7.72,;5.02,6.41,;5.93,10.39,;6.96,9.24,;4.9,11.53,;7.44,10.71,;-.43,.94,;-1.89,1.42,;.05,-.52,;-.86,-1.77,;-2.39,-1.61,;-3.29,-2.85,;-2.67,-4.26,;-3.57,-5.51,;-5.1,-5.35,;-5.73,-3.94,;-6.01,-6.59,;-6.91,-7.84,;-7.26,-5.69,;-4.76,-7.5,;-1.14,-4.42,;-.23,-3.18,;1.3,-3.34,;1.93,-4.74,)|
CCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CCC(F)(F)F)cc1OC |r,wU:9.8,wD:12.15,(-.52,-3.4,;.56,-2.17,;-.06,-.77,;-1.57,-.45,;-1.73,1.09,;-3.06,1.86,;-3.06,3.4,;-4.4,1.09,;-5.73,1.86,;-7.07,1.09,;-7.07,-.45,;-8.4,-1.22,;-9.78,-.48,;-9.73,1.09,;-8.4,1.86,;-11.11,-1.25,;-12.16,-.09,;-10.06,-2.42,;-12.65,-1.58,;-.32,1.71,;-0,3.22,;.71,.57,;2.24,.73,;2.86,2.14,;4.4,2.3,;5.3,1.05,;6.83,1.21,;7.74,-.03,;7.11,-1.44,;6.48,-2.85,;8.52,-2.07,;5.7,-.81,;4.67,-.36,;3.12,-.57,;2.49,-1.97,;3.4,-3.22,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CCC(F)(F)F)cc1OC |r,wU:9.8,wD:9.9,13.16,(-.49,-3.4,;.58,-2.17,;-.04,-.77,;-1.55,-.45,;-1.71,1.09,;-3.04,1.86,;-3.04,3.4,;-4.38,1.09,;-5.71,1.86,;-7.04,1.09,;-7.04,2.63,;-7.04,-.45,;-8.38,-1.22,;-9.76,-.48,;-9.71,1.09,;-8.38,1.86,;-11.09,-1.25,;-12.14,-.09,;-10.04,-2.42,;-12.63,-1.58,;-.3,1.71,;.02,3.22,;.73,.57,;2.26,.73,;2.89,2.14,;4.42,2.3,;5.32,1.05,;6.85,1.21,;7.76,-.03,;9.29,.13,;10.82,.29,;9.13,1.66,;9.45,-1.41,;4.7,-.36,;3.14,-.57,;2.52,-1.97,;3.42,-3.22,)|
CCCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(C[C@H](C)C(F)(F)F)cc1OC |r,wU:10.9,29.31,wD:10.10,14.17,(4.79,-2.18,;3.89,-.93,;2.36,-1.09,;1.45,.15,;1.93,1.62,;.68,2.52,;.68,4.06,;-.65,4.83,;2.01,4.83,;2.01,6.37,;3.35,7.14,;3.24,5.61,;2.63,8.5,;3.44,9.81,;4.98,9.75,;5.7,8.39,;4.89,7.09,;5.8,11.06,;6.94,10.03,;4.65,12.09,;7.26,11.54,;-.56,1.62,;-2.03,2.09,;-.09,.15,;-.99,-1.09,;-2.53,-.93,;-3.43,-2.18,;-2.8,-3.59,;-3.71,-4.83,;-5.24,-4.67,;-5.87,-3.26,;-6.15,-5.92,;-7.05,-7.16,;-7.39,-5.01,;-4.9,-6.82,;-1.27,-3.75,;-.37,-2.5,;1.16,-2.66,;1.79,-4.07,)|
CCCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(C[C@H](C)C(F)(F)F)cc1OC |r,wU:10.9,28.30,wD:13.16,(4.97,-1.99,;4.06,-.75,;2.53,-.91,;1.63,.34,;2.1,1.8,;.86,2.71,;.86,4.25,;-.48,5.02,;2.19,5.02,;2.19,6.56,;3.52,7.33,;3.52,8.87,;4.86,9.64,;6.19,8.87,;6.19,7.33,;4.86,6.56,;7.52,9.64,;8.67,8.61,;6.38,10.67,;8.99,10.11,;-.39,1.8,;-1.86,2.28,;.09,.34,;-.82,-.91,;-2.35,-.75,;-3.26,-1.99,;-2.63,-3.4,;-3.54,-4.64,;-5.07,-4.48,;-5.69,-3.08,;-5.97,-5.73,;-6.88,-6.98,;-7.22,-4.82,;-4.73,-6.63,;-1.1,-3.56,;-.19,-2.31,;1.34,-2.47,;1.96,-3.88,)|
CCCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(C[C@@H](C)C(F)(F)F)cc1OC |r,wU:10.9,wD:10.10,29.31,14.17,(4.81,-2.19,;3.9,-.95,;2.37,-1.11,;1.46,.14,;1.94,1.6,;.69,2.51,;.69,4.05,;-.64,4.82,;2.03,4.82,;2.03,6.36,;3.36,7.13,;3.25,5.59,;2.64,8.49,;3.45,9.79,;4.99,9.74,;5.72,8.38,;4.9,7.07,;5.81,11.04,;6.95,10.01,;4.67,12.08,;7.27,11.52,;-.55,1.6,;-2.02,2.08,;-.08,.14,;-.98,-1.11,;-2.51,-.95,;-3.42,-2.19,;-2.79,-3.6,;-3.7,-4.85,;-5.23,-4.69,;-5.85,-3.28,;-6.13,-5.93,;-7.04,-7.18,;-7.38,-5.03,;-4.89,-6.84,;-1.26,-3.76,;-.35,-2.52,;1.18,-2.68,;1.8,-4.08,)|
CCCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(C[C@@H](C)C(F)(F)F)cc1OC |r,wU:10.9,wD:28.30,13.16,(4.97,-1.99,;4.06,-.75,;2.53,-.91,;1.63,.34,;2.1,1.8,;.86,2.71,;.86,4.25,;-.48,5.02,;2.19,5.02,;2.19,6.56,;3.52,7.33,;3.52,8.87,;4.86,9.64,;6.19,8.87,;6.19,7.33,;4.86,6.56,;7.52,9.64,;8.67,8.61,;6.38,10.67,;8.99,10.11,;-.39,1.8,;-1.86,2.28,;.09,.34,;-.82,-.91,;-2.35,-.75,;-3.26,-1.99,;-2.63,-3.4,;-3.54,-4.64,;-5.07,-4.48,;-5.69,-3.08,;-5.97,-5.73,;-6.88,-6.98,;-4.73,-6.63,;-7.22,-4.82,;-1.1,-3.56,;-.19,-2.31,;1.34,-2.47,;1.96,-3.88,)|
CCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC |r,wU:9.8,wD:12.15,(3.86,-.89,;2.33,-1.05,;1.43,.19,;1.9,1.66,;.66,2.56,;.66,4.1,;-.68,4.87,;1.99,4.87,;1.99,6.41,;3.32,7.18,;3.32,8.72,;4.66,9.49,;5.99,8.72,;5.99,7.18,;4.66,6.41,;7.32,9.49,;8.47,8.46,;6.18,10.52,;8.79,9.97,;-.59,1.66,;-2.05,2.13,;-.11,.19,;-1.02,-1.05,;-2.55,-.89,;-3.46,-2.14,;-2.83,-3.54,;-3.73,-4.79,;-3.11,-6.2,;-4.51,-6.82,;-1.7,-5.57,;-2.48,-7.6,;-1.86,-9.01,;-3.89,-8.23,;-1.07,-6.98,;-1.3,-3.7,;-.39,-2.46,;1.14,-2.62,;1.77,-4.03,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC |r,wU:9.8,wD:9.9,13.16,(3.71,-1.11,;2.18,-1.27,;1.27,-.02,;1.75,1.44,;.5,2.35,;.5,3.89,;-.83,4.66,;1.83,4.66,;1.83,6.2,;3.17,6.97,;3.06,5.43,;2.45,8.33,;3.26,9.63,;4.8,9.58,;5.52,8.22,;4.71,6.91,;5.62,10.88,;6.76,9.85,;4.47,11.91,;7.08,11.36,;-.74,1.44,;-2.21,1.92,;-.27,-.02,;-1.17,-1.27,;-2.71,-1.11,;-3.61,-2.35,;-2.98,-3.76,;-3.89,-5.01,;-3.26,-6.41,;-4.67,-7.04,;-1.86,-5.79,;-2.64,-7.82,;-2.01,-9.23,;-4.04,-8.45,;-1.23,-7.19,;-1.45,-3.92,;-.55,-2.68,;.98,-2.84,;1.61,-4.24,)|
CCn1nc(C(=O)NC[C@]2(O)CC[C@H](C[C@H]2O)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:9.9,15.16,13.17,(-2.15,-2.72,;-2.78,-1.31,;-1.87,-.06,;-2.35,1.4,;-1.1,2.31,;-1.1,3.85,;.23,4.62,;-2.44,4.62,;-2.44,6.16,;-3.77,6.93,;-2.39,7.6,;-4.49,8.29,;-6.03,8.34,;-6.85,7.03,;-6.12,5.67,;-4.59,5.62,;-3.86,4.26,;-8.39,7.09,;-8.86,8.55,;-7.91,5.62,;-9.89,7.41,;.14,1.4,;1.61,1.88,;-.33,-.06,;.57,-1.31,;-.05,-2.72,;.85,-3.96,;2.38,-3.8,;3.29,-5.05,;4.82,-4.89,;4.98,-6.42,;4.66,-3.35,;6.35,-4.73,;7.88,-4.56,;6.51,-6.26,;6.19,-3.19,;3.01,-2.39,;2.1,-1.15,;2.73,.26,;4.26,.42,;4.89,1.83,;5.17,-.83,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](C[C@@H]2O)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.9,15.16,13.17,wD:9.8,(-2.15,-2.72,;-2.78,-1.31,;-1.87,-.06,;-2.35,1.4,;-1.1,2.31,;-1.1,3.85,;.23,4.62,;-2.44,4.62,;-2.44,6.16,;-3.77,6.93,;-2.39,7.6,;-4.49,8.29,;-6.03,8.34,;-6.85,7.03,;-6.12,5.67,;-4.59,5.62,;-3.86,4.26,;-8.39,7.09,;-8.23,8.62,;-8.55,5.56,;-9.63,7.99,;.14,1.4,;1.61,1.88,;-.33,-.06,;.57,-1.31,;-.05,-2.72,;.85,-3.96,;2.38,-3.8,;3.29,-5.05,;4.82,-4.89,;4.98,-6.42,;4.66,-3.35,;6.35,-4.73,;7.88,-4.56,;6.51,-6.26,;6.19,-3.19,;3.01,-2.39,;2.1,-1.15,;2.73,.26,;4.26,.42,;4.89,1.83,;5.17,-.83,)|
CCn1nc(C(=O)NC[C@]2(O)CC[C@@H](C[C@H]2O)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,13.17,wD:9.9,15.16,(-2.15,-2.72,;-2.78,-1.31,;-1.87,-.06,;-2.35,1.4,;-1.1,2.31,;-1.1,3.85,;.23,4.62,;-2.44,4.62,;-2.44,6.16,;-3.77,6.93,;-2.39,7.6,;-4.49,8.29,;-6.03,8.34,;-6.85,7.03,;-6.12,5.67,;-4.59,5.62,;-3.86,4.26,;-8.39,7.09,;-8.39,8.63,;-8.39,5.55,;-9.72,7.86,;.14,1.4,;1.61,1.88,;-.33,-.06,;.57,-1.31,;-.05,-2.72,;.85,-3.96,;2.38,-3.8,;3.29,-5.05,;4.82,-4.89,;4.98,-6.42,;4.66,-3.35,;6.35,-4.73,;7.88,-4.56,;6.51,-6.26,;6.19,-3.19,;3.01,-2.39,;2.1,-1.15,;2.73,.26,;4.26,.42,;4.89,1.83,;5.17,-.83,)|
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CCn1nc(C(=O)NC[C@]2(O)CC[C@H](C[C@H]2O)S(C)(=O)=O)c(Cl)c1-c1ccc(C[C@H](C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,29.31,wD:9.9,15.16,13.17,(-1.75,-2.4,;-2.38,-1,;-1.47,.25,;-1.95,1.71,;-.7,2.62,;-.7,4.16,;.63,4.93,;-2.04,4.93,;-2.04,6.47,;-3.37,7.24,;-1.99,7.91,;-4.09,8.6,;-5.63,8.65,;-6.45,7.35,;-5.73,5.99,;-4.19,5.93,;-3.46,4.57,;-7.99,7.4,;-8.15,8.93,;-7.83,5.87,;-9.4,8.03,;.54,1.71,;2.01,2.19,;.07,.25,;.97,-1,;.34,-2.4,;1.25,-3.65,;2.78,-3.49,;3.69,-4.73,;3.06,-6.14,;1.53,-6.3,;3.97,-7.39,;4.87,-8.63,;2.72,-8.29,;5.21,-6.48,;3.41,-2.08,;2.5,-.84,;3.13,.57,;4.66,.73,;5.29,2.14,;5.57,-.51,)|
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CCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(C[C@H](C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,27.29,wD:12.15,(-1.6,-2.32,;-2.23,-.91,;-1.32,.34,;-1.8,1.8,;-.55,2.7,;-.55,4.24,;.78,5.01,;-1.89,5.01,;-1.89,6.55,;-3.22,7.32,;-4.56,6.55,;-5.89,7.32,;-5.89,8.86,;-4.56,9.63,;-3.22,8.86,;-7.22,9.63,;-7.06,11.17,;-7.38,8.1,;-8.47,10.54,;.69,1.8,;2.16,2.28,;.22,.34,;1.12,-.91,;.49,-2.32,;1.4,-3.56,;2.93,-3.4,;3.84,-4.65,;3.21,-6.06,;1.68,-6.22,;4.12,-7.3,;5.02,-8.55,;2.87,-8.21,;5.36,-6.4,;3.56,-2,;2.65,-.75,;3.28,.66,;4.81,.82,;5.44,2.22,;5.72,-.43,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(C[C@H](C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,28.30,wD:9.9,13.16,(-1.7,-2.42,;-2.32,-1.01,;-1.42,.23,;-1.9,1.7,;-.65,2.6,;-.65,4.14,;.68,4.91,;-1.98,4.91,;-1.98,6.45,;-3.32,7.22,;-1.93,7.9,;-4.13,5.92,;-5.67,5.97,;-6.4,7.33,;-5.58,8.64,;-4.04,8.58,;-7.93,7.39,;-7.61,8.89,;-8.25,5.88,;-9.08,8.42,;.6,1.7,;2.06,2.18,;.12,.23,;1.03,-1.01,;.4,-2.42,;1.3,-3.66,;2.84,-3.5,;3.74,-4.75,;3.11,-6.16,;1.58,-6.32,;4.02,-7.4,;4.93,-8.65,;2.77,-8.31,;5.27,-6.5,;3.46,-2.1,;2.56,-.85,;3.18,.56,;4.72,.72,;5.34,2.12,;5.62,-.53,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](C[C@@H]2O)S(C)(=O)=O)c(C)c1-c1ccc(C[C@H](C)C(F)(F)F)cc1OC(F)F |r,wU:9.9,29.31,15.16,13.17,wD:9.8,(-1.65,-2.53,;-2.27,-1.12,;-1.37,.12,;-1.85,1.59,;-.6,2.49,;-.6,4.03,;.73,4.8,;-1.93,4.8,;-1.93,6.34,;-3.27,7.11,;-1.88,7.79,;-3.99,8.47,;-5.53,8.52,;-6.34,7.22,;-5.62,5.86,;-4.08,5.8,;-3.36,4.45,;-7.88,7.27,;-7.56,8.78,;-8.2,5.77,;-9.03,8.3,;.65,1.59,;2.11,2.06,;.17,.12,;1.08,-1.12,;.45,-2.53,;1.35,-3.78,;2.89,-3.62,;3.79,-4.86,;3.16,-6.27,;1.63,-6.43,;4.07,-7.52,;4.98,-8.76,;2.82,-8.42,;5.32,-6.61,;3.51,-2.21,;2.61,-.96,;3.23,.44,;4.77,.6,;5.39,2.01,;5.67,-.64,)|
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CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(N)(=O)=O)c(Cl)c1-c1ccc(C[C@H](C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,28.30,wD:9.9,13.16,(.07,-2.33,;-.55,-.92,;.35,.32,;-.12,1.79,;1.12,2.69,;1.12,4.23,;2.46,5,;-.21,5,;-1.54,4.23,;-2.88,5,;-1.49,5.68,;-3.69,3.7,;-5.23,3.75,;-5.96,5.11,;-5.14,6.42,;-3.6,6.36,;-7.49,5.17,;-7.17,6.67,;-7.81,3.66,;-8.64,6.2,;2.37,1.79,;3.83,2.27,;1.89,.32,;2.8,-.92,;2.17,-2.33,;3.08,-3.57,;4.61,-3.41,;5.51,-4.66,;4.89,-6.07,;3.36,-6.23,;5.79,-7.31,;6.7,-8.56,;7.04,-6.41,;4.55,-8.22,;5.24,-2.01,;4.33,-.76,;4.96,.65,;6.49,.81,;7.11,2.21,;7.39,-.44,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(N)(=O)=O)c(C)c1-c1ccc(C[C@H](C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,28.30,wD:9.9,13.16,(-.33,-3.02,;-.95,-1.61,;-.05,-.37,;-.52,1.1,;.72,2,;.72,3.54,;2.06,4.31,;-.61,4.31,;-.61,5.85,;-1.94,6.62,;-.56,7.3,;-2.76,5.32,;-4.3,5.37,;-5.02,6.73,;-4.21,8.04,;-2.67,7.98,;-6.56,6.78,;-6.24,8.29,;-6.88,5.28,;-7.71,7.81,;1.97,1.1,;3.43,1.57,;1.49,-.37,;2.4,-1.61,;1.77,-3.02,;2.68,-4.27,;4.21,-4.11,;5.11,-5.35,;4.49,-6.76,;2.96,-6.92,;5.39,-8,;6.3,-9.25,;4.15,-8.91,;6.64,-7.1,;4.84,-2.7,;3.93,-1.45,;4.56,-.05,;6.09,.11,;6.71,1.52,;6.99,-1.13,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(N)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:9.9,13.16,(-.73,-3.32,;-1.36,-1.92,;-.45,-.67,;-.93,.79,;.32,1.7,;.32,3.24,;1.65,4.01,;-1.02,4.01,;-1.02,5.55,;-2.35,6.32,;-.97,6.99,;-3.17,5.01,;-4.71,5.07,;-5.43,6.43,;-4.61,7.73,;-3.07,7.68,;-6.97,6.48,;-6.65,7.99,;-7.29,4.97,;-8.11,7.51,;1.56,.79,;3.03,1.27,;1.09,-.67,;1.99,-1.92,;1.37,-3.32,;2.27,-4.57,;3.8,-4.41,;4.71,-5.66,;6.24,-5.49,;6.4,-7.03,;6.08,-3.96,;7.77,-5.33,;9.3,-5.17,;7.93,-6.87,;7.61,-3.8,;4.43,-3,;3.52,-1.76,;4.15,-.35,;5.68,-.19,;6.31,1.22,;6.59,-1.43,)|
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CCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CCCC(F)(F)F)cc1OC |r,wU:9.8,wD:12.15,(-1.04,-3.86,;-0,-2.72,;-.48,-1.25,;-1.95,-.78,;-1.95,.76,;-3.28,1.53,;-3.28,3.07,;-4.61,.76,;-5.95,1.53,;-7.28,.76,;-7.28,-.78,;-8.61,-1.55,;-9.99,-.81,;-9.95,.76,;-8.61,1.53,;-11.33,-1.58,;-9.97,-2.36,;-12.69,-.79,;-11.33,-3.15,;-.48,1.24,;-0,2.7,;.42,-.01,;1.96,-.01,;2.73,1.32,;4.27,1.32,;5.04,-.01,;6.58,-.01,;7.35,1.32,;8.89,1.32,;9.66,-.01,;10.43,-1.34,;8.33,-.78,;11,.76,;4.27,-1.34,;2.71,-1.39,;1.94,-2.72,;2.71,-4.06,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CCCC(F)(F)F)cc1OC |r,wU:9.8,wD:9.9,13.16,(-1.04,-3.86,;-0,-2.72,;-.48,-1.25,;-1.95,-.78,;-1.95,.76,;-3.28,1.53,;-3.28,3.07,;-4.61,.76,;-5.95,1.53,;-7.28,.76,;-7.28,2.3,;-7.28,-.78,;-8.61,-1.55,;-9.99,-.81,;-9.95,.76,;-8.61,1.53,;-11.33,-1.58,;-9.97,-2.36,;-12.69,-.79,;-11.33,-3.15,;-.48,1.24,;-0,2.7,;.42,-.01,;1.96,-.01,;2.73,1.32,;4.27,1.32,;5.04,-.01,;6.58,-.01,;7.35,1.32,;8.89,1.32,;9.66,-.01,;10.43,-1.34,;8.33,-.78,;11,.76,;4.27,-1.34,;2.71,-1.39,;1.94,-2.72,;2.71,-4.06,)|
CCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(C)c1-c1ccc(CCCC(F)(F)F)cc1OC |r,wU:9.8,wD:12.15,(-1.04,-3.86,;-0,-2.72,;-.48,-1.25,;-1.95,-.78,;-1.95,.76,;-3.28,1.53,;-3.28,3.07,;-4.61,.76,;-5.95,1.53,;-7.28,.76,;-7.28,-.78,;-8.61,-1.55,;-9.99,-.81,;-9.95,.76,;-8.61,1.53,;-11.33,-1.58,;-9.97,-2.36,;-12.69,-.79,;-11.33,-3.15,;-.47,1.28,;.01,2.74,;.42,-.01,;1.96,-.01,;2.73,1.32,;4.27,1.32,;5.04,-.01,;6.58,-.01,;7.35,1.32,;8.89,1.32,;9.66,-.01,;10.43,-1.34,;11,.76,;8.33,-.78,;4.27,-1.34,;2.71,-1.39,;1.94,-2.72,;2.71,-4.06,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(C)c1-c1ccc(CCCC(F)(F)F)cc1OC |r,wU:9.8,wD:9.9,13.16,(-1.04,-3.86,;-0,-2.72,;-.48,-1.25,;-1.95,-.78,;-1.95,.76,;-3.28,1.53,;-3.28,3.07,;-4.61,.76,;-5.95,1.53,;-7.28,.76,;-7.28,2.3,;-7.28,-.78,;-8.61,-1.55,;-9.99,-.81,;-9.95,.76,;-8.61,1.53,;-11.33,-1.58,;-9.97,-2.36,;-12.69,-.79,;-11.33,-3.15,;-.47,1.28,;.01,2.74,;.42,-.01,;1.96,-.01,;2.73,1.32,;4.27,1.32,;5.04,-.01,;6.58,-.01,;7.35,1.32,;8.89,1.32,;9.66,-.01,;10.43,-1.34,;8.33,-.78,;11,.76,;4.27,-1.34,;2.71,-1.39,;1.94,-2.72,;2.71,-4.06,)|
CCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C(F)(F)F)C(F)(F)F)cc1OC |r,wU:12.15,wD:9.8,(-3.68,2.45,;-3.36,.94,;-1.9,.47,;-1.42,-1,;.12,-1,;1.02,-2.24,;2.56,-2.08,;.4,-3.65,;1.3,-4.9,;.68,-6.3,;-.85,-6.47,;-1.48,-7.87,;-.58,-9.12,;.96,-8.96,;1.58,-7.55,;-1.2,-10.53,;.13,-11.29,;-1.2,-12.07,;-2.54,-9.76,;.6,.47,;2.06,.94,;-.65,1.37,;-.65,2.91,;-1.98,3.68,;-1.98,5.22,;-.65,5.99,;-.65,7.53,;.68,8.3,;2.02,7.53,;3.35,6.76,;1.25,6.2,;2.79,8.86,;.68,9.84,;2.02,10.61,;-.65,10.61,;.68,11.38,;.68,5.22,;.68,3.68,;2.02,2.91,;3.35,3.68,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C(F)(F)F)C(F)(F)F)cc1OC |r,wU:9.9,13.16,wD:9.8,(-3.75,2.53,;-3.43,1.03,;-1.96,.55,;-1.49,-.91,;.05,-.91,;.96,-2.16,;2.49,-2,;.33,-3.57,;1.24,-4.81,;.61,-6.22,;2.1,-6.59,;-.67,-5.36,;-2.05,-6.03,;-2.16,-7.57,;-.88,-8.43,;.5,-7.76,;-3.54,-8.24,;-2.21,-9.01,;-4.88,-7.47,;-3.54,-9.78,;.53,.55,;1.99,1.03,;-.72,1.46,;-.72,3,;-2.05,3.77,;-2.05,5.31,;-.72,6.08,;-.72,7.62,;.62,8.39,;1.95,7.62,;3.28,6.85,;2.72,8.95,;1.18,6.28,;.62,9.93,;1.95,10.7,;-.72,10.7,;.62,11.47,;.62,5.31,;.62,3.77,;1.95,3,;3.28,3.77,)|
CCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C(F)(F)F)C(F)(F)F)cc1OC(F)F |r,wU:12.15,wD:9.8,(-3.75,2.71,;-3.43,1.2,;-1.97,.73,;-1.49,-.74,;.05,-.74,;.95,-1.99,;2.48,-1.82,;.33,-3.39,;1.23,-4.64,;.61,-6.04,;-.93,-6.21,;-1.55,-7.61,;-.65,-8.86,;.88,-8.7,;1.51,-7.29,;-1.27,-10.27,;.06,-11.04,;-2.61,-9.5,;-1.27,-11.81,;.52,.73,;1.99,1.2,;-.72,1.63,;-.72,3.17,;-2.06,3.94,;-2.06,5.48,;-.72,6.25,;-.72,7.79,;.61,8.56,;1.94,7.79,;3.28,7.02,;2.71,9.12,;1.17,6.46,;.61,10.1,;1.94,10.87,;-.72,10.87,;.61,11.64,;.61,5.48,;.61,3.94,;1.94,3.17,;3.28,3.94,;4.61,3.17,;3.28,5.48,)|
CCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(C)c1-c1ccc(CC(C(F)(F)F)C(F)(F)F)cc1OC(F)F |r,wU:12.15,wD:9.8,(-3.75,2.71,;-3.43,1.2,;-1.97,.73,;-1.49,-.74,;.05,-.74,;.95,-1.99,;2.48,-1.82,;.33,-3.39,;1.23,-4.64,;.61,-6.04,;-.93,-6.21,;-1.55,-7.61,;-.65,-8.86,;.88,-8.7,;1.51,-7.29,;-1.27,-10.27,;.06,-11.04,;-2.61,-9.5,;-1.27,-11.81,;.52,.73,;1.99,1.2,;-.72,1.63,;-.72,3.17,;-2.06,3.94,;-2.06,5.48,;-.72,6.25,;-.72,7.79,;.61,8.56,;1.94,7.79,;3.28,7.02,;2.71,9.12,;1.17,6.46,;.61,10.1,;1.94,10.87,;-.72,10.87,;.61,11.64,;.61,5.48,;.61,3.94,;1.94,3.17,;3.28,3.94,;4.61,3.17,;3.28,5.48,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1C#N |r,wU:9.9,13.16,wD:9.8,(-5.23,1.38,;-4.91,-.12,;-3.44,-.6,;-2.97,-2.06,;-1.43,-2.06,;-.52,-3.31,;-1.15,-4.72,;1.01,-3.15,;1.91,-4.4,;3.44,-4.23,;3.02,-2.75,;3.34,-5.77,;4.61,-6.63,;6,-5.96,;6.11,-4.42,;4.83,-3.56,;7.27,-6.82,;7.44,-5.29,;7.11,-8.35,;8.68,-6.19,;-.95,-.6,;.51,-.12,;-2.2,.31,;-2.2,1.85,;-3.53,2.62,;-3.53,4.16,;-2.2,4.93,;-2.2,6.47,;-.87,7.24,;-.1,5.9,;-1.64,8.57,;.47,8.01,;1.8,8.78,;1.24,6.67,;-.3,9.34,;-.87,4.16,;-.87,2.62,;.47,1.85,;1.8,1.08,)|
CCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)CC(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:12.15,(-1.08,-3.12,;-.05,-1.98,;-.53,-.52,;-1.99,-.04,;-1.99,1.5,;-3.33,2.27,;-3.33,3.81,;-4.66,1.5,;-6,2.27,;-7.33,1.5,;-7.33,-.04,;-8.66,-.81,;-10.04,-.07,;-10,1.5,;-8.66,2.27,;-11.38,-.84,;-10.02,-1.62,;-12.74,-.05,;-11.38,-2.41,;-.53,1.98,;-.05,3.44,;.38,.73,;1.92,.73,;2.69,2.06,;4.23,2.06,;5,.73,;6.54,.73,;7.31,2.06,;7.31,3.6,;8.82,1.66,;5.77,1.98,;4.93,3.28,;4.09,4.57,;6.22,4.11,;3.64,2.44,;4.23,-.6,;2.66,-.65,;1.89,-1.98,;2.66,-3.32,;4.2,-3.32,;1.89,-4.65,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)CC(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:9.9,13.16,(-1.08,-3.12,;-.05,-1.98,;-.53,-.52,;-1.99,-.04,;-1.99,1.5,;-3.33,2.27,;-3.33,3.81,;-4.66,1.5,;-6,2.27,;-7.33,1.5,;-7.33,3.04,;-7.33,-.04,;-8.66,-.81,;-10.04,-.07,;-10,1.5,;-8.66,2.27,;-11.38,-.84,;-10.02,-1.62,;-12.74,-.05,;-11.38,-2.41,;-.53,1.98,;-.05,3.44,;.38,.73,;1.92,.73,;2.69,2.06,;4.23,2.06,;5,.73,;6.54,.73,;7.31,2.06,;7.31,3.6,;5.97,2.83,;5.77,1.98,;4.93,3.28,;4.09,4.57,;6.22,4.11,;3.64,2.44,;4.23,-.6,;2.66,-.65,;1.89,-1.98,;2.66,-3.32,;4.2,-3.32,;1.89,-4.65,)|
CCn1nc(C(=O)NC[C@@]2(CO)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:9.9,14.17,(3.4,.09,;1.87,-.07,;.96,1.18,;1.44,2.64,;.19,3.55,;.19,5.09,;-1.14,5.86,;1.53,5.86,;1.53,7.4,;2.86,8.17,;2.75,6.63,;4.03,5.77,;2.14,9.53,;2.95,10.83,;4.49,10.78,;5.21,9.42,;4.4,8.11,;5.31,12.08,;6.64,11.31,;3.97,12.85,;6.08,13.42,;-1.05,2.64,;-2.52,3.12,;-.58,1.18,;-1.48,-.07,;-3.02,.09,;-3.92,-1.15,;-3.29,-2.56,;-4.2,-3.81,;-3.57,-5.21,;-4.98,-5.84,;-2.17,-4.59,;-2.95,-6.62,;-2.32,-8.03,;-4.35,-7.25,;-1.54,-5.99,;-1.76,-2.72,;-.86,-1.48,;.67,-1.64,;1.3,-3.04,;2.83,-3.21,;.4,-4.29,)|
CCn1nc(C(=O)NC[C@@]2(CO)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)C(F)(F)F)cc1OC |r,wU:9.8,wD:9.9,14.17,(3.6,-1.55,;2.07,-1.71,;1.16,-.47,;1.64,1,;.39,1.9,;.39,3.44,;-.94,4.21,;1.73,4.21,;1.73,5.75,;3.06,6.52,;2.95,4.99,;4.23,4.13,;2.34,7.88,;3.15,9.19,;4.69,9.14,;5.41,7.78,;4.6,6.47,;5.51,10.44,;6.84,9.67,;4.17,11.21,;5.51,8.9,;-.85,1,;-2.32,1.48,;-.38,-.47,;-1.28,-1.71,;-2.81,-1.55,;-3.72,-2.8,;-3.09,-4.2,;-4,-5.45,;-5.53,-5.29,;-6.44,-6.53,;-6.16,-3.88,;-6.78,-2.47,;-4.75,-3.25,;-7.56,-4.51,;-1.56,-4.36,;-.66,-3.12,;.87,-3.28,;1.5,-4.69,)|
CCn1nc(C(=O)NC[C@@]2(CO)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(N[C@H](C)C(F)(F)F)cc1OC |r,wU:9.9,14.17,wD:9.8,29.31,(4.27,-1.43,;2.74,-1.59,;1.83,-.34,;2.31,1.12,;1.06,2.03,;1.06,3.57,;2.4,4.34,;-.27,4.34,;-.27,5.88,;1.06,6.65,;-.32,7.32,;-.43,8.86,;1.88,5.34,;3.42,5.4,;4.14,6.76,;3.32,8.06,;1.78,8.01,;5.68,6.81,;7.01,6.04,;4.34,7.58,;5.68,5.27,;-.18,1.12,;-1.65,1.6,;.29,-.34,;-.61,-1.59,;-2.15,-1.43,;-3.05,-2.67,;-2.42,-4.08,;-3.33,-5.33,;-4.86,-5.16,;-5.77,-6.41,;-5.49,-3.76,;-6.11,-2.35,;-6.89,-4.38,;-4.08,-3.13,;-.89,-4.24,;.01,-2.99,;1.54,-3.16,;2.17,-4.56,)|
CCn1nc(C(=O)NC[C@@]2(CC)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(N[C@H](C)C(F)(F)F)cc1OC |r,wU:9.8,wD:29.31,9.9,14.17,(3.59,-2.35,;2.06,-2.51,;1.15,-1.26,;1.63,.2,;.38,1.11,;.38,2.65,;-.95,3.42,;1.71,3.42,;1.71,4.96,;3.05,5.73,;2.94,4.19,;4.22,3.33,;2.33,7.09,;3.14,8.39,;4.68,8.34,;5.4,6.98,;4.59,5.67,;5.5,9.64,;6.83,8.87,;4.16,10.41,;5.5,8.1,;-.86,.2,;-2.33,.68,;-.39,-1.26,;-1.29,-2.51,;-2.83,-2.35,;-3.73,-3.6,;-3.1,-5,;-4.01,-6.25,;-5.54,-6.09,;-6.45,-7.33,;-6.17,-4.68,;-6.79,-3.27,;-4.76,-4.05,;-7.57,-5.31,;-1.57,-5.16,;-.67,-3.92,;.86,-4.08,;1.49,-5.48,)|
CCn1nc(C(=O)NC[C@]2(CC)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(N[C@H](C)C(F)(F)F)cc1OC |r,wU:9.8,14.17,wD:29.31,9.9,(4.26,-2.23,;2.73,-2.39,;1.82,-1.14,;2.3,.32,;1.05,1.23,;1.05,2.77,;2.38,3.54,;-.28,3.54,;-.28,5.08,;1.05,5.85,;-.33,6.52,;-.44,8.06,;1.87,4.54,;3.41,4.6,;4.13,5.96,;3.31,7.26,;1.77,7.21,;5.67,6.01,;7,5.24,;4.33,6.78,;5.67,4.47,;-.2,.32,;-1.66,.8,;.28,-1.14,;-.62,-2.39,;-2.16,-2.23,;-3.06,-3.47,;-2.43,-4.88,;-3.34,-6.12,;-4.87,-5.96,;-5.78,-7.21,;-5.5,-4.56,;-6.12,-3.15,;-6.9,-5.18,;-4.09,-3.93,;-.9,-5.04,;0,-3.79,;1.53,-3.95,;2.16,-5.36,)|
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Cn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:8.7,wD:8.8,12.15,(-2.64,-.96,;-1.74,.29,;-2.21,1.75,;-.97,2.66,;-.97,4.2,;.37,4.97,;-2.3,4.97,;-2.3,6.51,;-3.64,7.28,;-2.25,7.95,;-4.45,5.97,;-5.99,6.02,;-6.71,7.38,;-5.9,8.69,;-4.36,8.64,;-8.25,7.44,;-8.25,8.98,;-8.25,5.9,;-9.59,8.21,;.28,1.75,;1.74,2.23,;-.2,.29,;.71,-.96,;.08,-2.37,;.99,-3.61,;2.52,-3.45,;3.42,-4.7,;4.95,-4.54,;5.12,-6.07,;4.79,-3.01,;6.49,-4.38,;8.02,-4.21,;6.65,-5.91,;6.33,-2.84,;3.14,-2.04,;2.24,-.8,;2.87,.61,;4.4,.77,;5.02,2.18,;5.3,-.48,)|
Cn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:8.7,wD:11.14,(-1.84,-.49,;-.94,.76,;-1.41,2.23,;-.17,3.13,;-.17,4.67,;1.17,5.44,;-1.5,5.44,;-1.5,6.98,;-2.83,7.75,;-4.17,6.98,;-5.5,7.75,;-5.5,9.29,;-4.17,10.06,;-2.83,9.29,;-6.84,10.06,;-6.84,11.6,;-6.84,8.52,;-8.17,10.83,;1.08,2.23,;2.54,2.7,;.6,.76,;1.51,-.49,;.88,-1.89,;1.79,-3.14,;3.32,-2.98,;4.22,-4.22,;3.6,-5.63,;5,-6.26,;2.19,-5,;2.97,-7.04,;2.34,-8.44,;4.38,-7.66,;1.56,-6.41,;3.94,-1.57,;3.04,-.32,;3.67,1.08,;5.2,1.24,;5.82,2.65,;6.1,-0,)|
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Cn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CCCC(F)(F)F)cc1OC(F)F |r,wU:8.7,wD:8.8,12.15,(.4,-1.49,;-.37,-.16,;-1.87,.17,;-2.03,1.7,;-3.37,2.47,;-3.37,4.01,;-4.7,1.7,;-6.03,2.47,;-7.37,1.7,;-7.37,3.24,;-7.37,.16,;-8.7,-.61,;-10.08,.13,;-10.03,1.7,;-8.7,2.47,;-11.42,-.64,;-11.42,.93,;-11.42,-2.21,;-12.77,.14,;-.63,2.32,;-.23,3.81,;.4,1.18,;1.89,1.58,;2.29,3.06,;3.78,3.46,;4.87,2.37,;6.35,2.77,;7.44,1.68,;7.04,.2,;8.13,-.89,;9.22,-1.98,;9.22,.2,;7.04,-1.98,;4.47,.89,;2.97,.43,;2.57,-1.05,;3.66,-2.14,;5.14,-1.74,;3.26,-3.63,)|
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CCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1Cl |r,wU:9.8,wD:12.15,(3.93,-.5,;2.4,-.66,;1.49,.58,;1.97,2.05,;.72,2.95,;.72,4.49,;-.61,5.26,;2.06,5.26,;2.06,6.8,;3.39,7.57,;3.39,9.11,;4.72,9.88,;6.06,9.11,;6.06,7.57,;4.72,6.8,;7.39,9.88,;7.39,11.42,;7.39,8.34,;6.06,10.65,;-.52,2.05,;-1.99,2.52,;-.05,.58,;-.95,-.66,;-2.49,-.5,;-3.39,-1.75,;-2.76,-3.15,;-3.67,-4.4,;-3.04,-5.81,;-4.45,-6.43,;-1.64,-5.18,;-2.42,-7.21,;-1.79,-8.62,;-3.82,-7.84,;-1.01,-6.59,;-1.23,-3.31,;-.33,-2.07,;1.2,-2.23,)|
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CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1 |r,wU:9.8,wD:9.9,13.16,(1.72,-2.29,;2.35,-.88,;1.44,.37,;1.92,1.83,;.67,2.74,;.67,4.28,;-.66,5.05,;2.01,5.05,;2.01,6.59,;3.34,7.36,;3.23,5.82,;2.62,8.72,;3.43,10.02,;4.97,9.97,;5.7,8.61,;4.88,7.3,;5.79,11.27,;5.79,12.81,;5.79,9.73,;4.45,12.04,;-.57,1.83,;-2.04,2.31,;-.1,.37,;-1,-.88,;-.38,-2.29,;-1.28,-3.53,;-2.81,-3.37,;-3.72,-4.62,;-3.09,-6.02,;-4.5,-6.65,;-1.69,-5.4,;-2.47,-7.43,;-1.84,-8.84,;-3.87,-8.06,;-1.06,-6.8,;-3.44,-1.96,;-2.53,-.72,)|
CCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1 |r,wU:9.8,wD:12.15,(1.89,-2.04,;2.51,-.64,;1.61,.61,;2.08,2.07,;.84,2.98,;.84,4.52,;-.5,5.29,;2.17,5.29,;2.17,6.83,;3.51,7.6,;3.51,9.14,;4.84,9.91,;6.17,9.14,;6.17,7.6,;4.84,6.83,;7.51,9.91,;7.51,11.45,;7.51,8.37,;6.17,10.68,;-.41,2.07,;-1.87,2.55,;.07,.61,;-.84,-.64,;-.21,-2.04,;-1.12,-3.29,;-2.65,-3.13,;-3.55,-4.38,;-2.93,-5.78,;-4.33,-6.41,;-1.52,-5.16,;-2.3,-7.19,;-1.67,-8.6,;-3.71,-7.82,;-.89,-6.56,;-3.27,-1.72,;-2.37,-.48,)|
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CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CCC(F)(F)F)cc1C(F)(F)F |r,wU:9.8,wD:9.9,13.16,(0,-3.41,;.77,-2.08,;0,-.75,;-1.51,-.43,;-1.67,1.1,;-3,1.87,;-3,3.41,;-4.33,1.1,;-5.67,1.87,;-7,1.1,;-7,2.64,;-7,-.44,;-8.33,-1.21,;-9.72,-.46,;-9.67,1.1,;-8.33,1.87,;-11.05,-1.23,;-11.05,.34,;-11.05,-2.8,;-12.41,-.45,;-.26,1.73,;.14,3.22,;.77,.59,;2.26,.98,;2.66,2.47,;4.14,2.87,;5.23,1.78,;6.72,2.18,;7.81,1.09,;9.3,1.49,;10.78,1.89,;9.7,0,;8.9,2.98,;4.83,.29,;3.29,-.18,;2.88,-1.67,;2.46,-3.15,;4.36,-2.08,;1.39,-1.25,)|
CCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CCC(F)(F)F)cc1C(F)(F)F |r,wU:9.8,wD:12.15,(-.01,-3.41,;.76,-2.08,;-.01,-.75,;-1.52,-.43,;-1.68,1.1,;-3.02,1.87,;-3.02,3.41,;-4.35,1.1,;-5.68,1.87,;-7.02,1.1,;-7.02,-.44,;-8.35,-1.21,;-9.73,-.46,;-9.68,1.1,;-8.35,1.87,;-11.07,-1.23,;-11.07,.34,;-11.07,-2.8,;-12.42,-.45,;-.27,1.73,;.12,3.22,;.76,.59,;2.24,.98,;2.64,2.47,;4.13,2.87,;5.22,1.78,;6.71,2.18,;7.79,1.09,;9.28,1.49,;10.77,1.89,;9.68,0,;8.88,2.98,;4.82,.29,;3.28,-.18,;2.86,-1.67,;2.45,-3.15,;4.35,-2.08,;1.38,-1.25,)|
CCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(N[C@H](C)C(F)(F)F)cc1C(F)(F)F |r,wU:9.8,27.29,wD:12.15,(4.27,-.98,;2.74,-1.14,;1.83,.1,;2.31,1.57,;1.06,2.47,;1.06,4.01,;-.27,4.78,;2.4,4.78,;2.4,6.32,;3.73,7.09,;3.73,8.63,;5.07,9.4,;6.4,8.63,;6.4,7.09,;5.07,6.32,;7.73,9.4,;7.73,10.94,;7.73,7.86,;6.4,10.17,;-.18,1.57,;-1.65,2.04,;.29,.1,;-.61,-1.14,;-2.14,-.98,;-3.05,-2.23,;-2.42,-3.64,;-3.33,-4.88,;-4.86,-4.72,;-5.48,-3.31,;-5.76,-5.97,;-6.67,-7.21,;-7.01,-5.06,;-4.52,-6.87,;-.89,-3.8,;.02,-2.55,;1.55,-2.71,;3.08,-2.87,;1.39,-4.24,;1.71,-1.18,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CCC(F)(F)F)cc1Cl |r,wU:9.8,wD:9.9,13.16,(0,-3.41,;.77,-2.08,;0,-.75,;-1.51,-.43,;-1.67,1.1,;-3,1.87,;-3,3.41,;-4.33,1.1,;-5.67,1.87,;-7,1.1,;-7,2.64,;-7,-.44,;-8.33,-1.21,;-9.72,-.46,;-9.67,1.1,;-8.33,1.87,;-11.05,-1.23,;-11.05,.34,;-11.05,-2.8,;-12.41,-.45,;-.26,1.73,;.14,3.22,;.77,.59,;2.26,.98,;2.66,2.47,;4.14,2.87,;5.23,1.78,;6.72,2.18,;7.81,1.09,;9.3,1.49,;10.78,1.89,;9.7,0,;8.9,2.98,;4.83,.29,;3.35,-.1,;2.95,-1.59,)|
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COCCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)cc1OC |r,wU:11.10,wD:14.17,(6.62,.89,;5.09,.72,;4.47,-.68,;2.93,-.84,;2.03,.4,;2.5,1.87,;1.26,2.77,;1.26,4.31,;-.08,5.08,;2.59,5.08,;2.59,6.62,;3.93,7.39,;3.93,8.93,;5.26,9.7,;6.59,8.93,;6.59,7.39,;5.26,6.62,;7.93,9.7,;7.93,11.24,;7.93,8.16,;6.59,10.47,;.01,1.87,;-1.45,2.34,;.49,.4,;-.42,-.84,;-1.95,-.68,;-2.85,-1.93,;-2.23,-3.33,;-3.13,-4.58,;-4.66,-4.42,;-4.82,-5.95,;-4.5,-2.89,;-6.2,-4.26,;-7.73,-4.1,;-6.36,-5.79,;-6.03,-2.73,;-.7,-3.5,;.21,-2.25,;1.74,-2.41,;2.37,-3.82,)|
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C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC2CCCC2)cc1C(F)F)C(=O)NCC1(O)CC1 |r|
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CC(C)(O)CCNC(=O)c1nc(C(=O)N2CCC(F)(F)CC2)c(s1)-c1cnc(NC2CCCCC2)cc1C(F)(F)F
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CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)CC2)c(s1)-c1cnc(NC2CC(F)(F)C2)cc1C(F)(F)F
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)CC2)c(s1)-c1cnc(NC2CC3(C2)CC(F)(F)C3)cc1C(F)(F)F
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)CC2)c(s1)-c1cnc(NC2CCCC(F)(F)C2)cc1C(F)(F)F
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)CC2)c(s1)-c1cnc(NC2CC3(CCC3)C2)cc1C(F)(F)F
C[C@H]1CCN1C(=O)c1nc(sc1-c1cnc(NC2CCCCC2)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)CC2)c(s1)-c1cnc(NC2CCCCC2(F)F)cc1C(F)(F)F
C[C@H]1CCCCN1C(=O)c1nc(sc1-c1cnc(NC2CCCC2)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCCN1C(=O)c1nc(sc1-c1cnc(NC2CCCC2)cc1C(F)(F)F)C(=O)NC1CCS(=O)(=O)CC1 |r|
C[C@@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CCC(F)CC1)C(=O)NCC(C)(C)O)C(F)(F)F)C1CC1 |r|
C[C@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CCC(F)CC1)C(=O)NCC(C)(C)O)C(F)(F)F)C1CC1 |r|
C[C@H]1CCCCN1C(=O)c1nc(sc1-c1cnc(N[C@@H]2CCCCC2(F)F)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCCN1C(=O)c1nc(sc1-c1cnc(N[C@H]2CCCCC2(F)F)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
CC(Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CCCC[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F)C(F)(F)F |r|
C[C@H]1CCCCN1C(=O)c1nc(sc1-c1cnc(NC2CCCCC2)cc1C(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(N[C@@H]2CCCCC2(F)F)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(N[C@H]2CCCCC2(F)F)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCCC[C@@H]1C)C(=O)NCC(C)(C)O)C1CC1 |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC2CCCC2)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CCCC[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F)C1CC1 |r|
C[C@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F)C1CC1 |r|
C[C@H]1CCCCN1C(=O)c1nc(sc1-c1cnc(NC2CCCC2)cc1C(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC2CCCC2)cc1C(F)F)C(=O)NCC(C)(C)O |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NCC(C)(C)O)C1CC1 |r|
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1cnc(NC2CCCC2)cc1C(F)F)C(=O)NCC(C)(C)O |r|
C[C@@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CCCC[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F)C(F)(F)F |r|
CC(C)(O)CNC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1cnc(NC2CCCC2)cc1C(F)F |THB:11:13:19.18:15.16|
C[C@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CCCC[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F)C(F)(F)F |r|
C[C@@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F)C1CC1 |r|
C[C@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NCC1(O)CCC1)C(F)(F)F)C1CC1 |r|
C[C@@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NCC(C)(C)O)C1CC1 |r|
C[C@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)NCC(C)(C)O)C(F)(F)F)C1CC1 |r,THB:14:16:22.21:18.19|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
CC(C)(O)CNC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1cnc(NC2CCCC2)cc1C(F)(F)F |THB:11:13:19.18:15.16|
C[C@@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F)C(F)(F)F |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)NCC(C)(C)O)C1CC1 |r,THB:17:19:25.24:21.22|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C2CC2)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)CC2)c(s1)-c1cnc(NC2CCCCC2)cc1C#N
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)CC2)c(s1)-c1cnc(NC2CCCCC2)c(c1)C#N
Cc1c(cnc(NC2CCCCC2)c1C#N)-c1sc(nc1C(=O)N1CCC(F)CC1)C(=O)NCC(C)(C)O
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC2CCCC2)cc1C(F)F)C(=O)NC1CS(=O)(=O)C1 |r|
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)CC2)c(s1)-c1cnc(NC2CCCCC2)c(OC(F)F)c1
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)CC2)c(s1)-c1cnc(NC2CCCCC2)cc1C1CC1
Cc1c(F)c(NC2CCCCC2)ncc1-c1sc(nc1C(=O)N1CCC(F)CC1)C(=O)NCC(C)(C)O
Cc1cc(NC2CCCCC2)ncc1-c1sc(nc1C(=O)N1CCC(F)CC1)C(=O)NCC(C)(C)O
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)CC2)c(s1)-c1cnc(NC2CCCCC2)c(C#N)c1C(F)(F)F
CCOc1cc(NC2CCCCC2)ncc1-c1sc(nc1C(=O)N1CCC(F)CC1)C(=O)NCC(C)(C)O
CCc1cc(NC2CCCCC2)ncc1-c1sc(nc1C(=O)N1CCC(F)CC1)C(=O)NCC(C)(C)O
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC2CCCC2)cc1C(F)F)C(=O)NCC1(O)CCC1 |r|
C[C@H]1C[C@@H](C1)NC(=O)c1nc(C(=O)N2CCC[C@@H]2C)c(s1)-c1cnc(NC2CCCC2)cc1C(F)F |r,wU:17.19,3.5,wD:1.0,(-8.57,4.81,;-7.24,4.04,;-6.82,2.54,;-5.33,2.94,;-5.73,4.42,;-4,2.17,;-2.66,2.94,;-2.66,4.48,;-1.33,2.17,;-1.33,.63,;.14,.15,;.53,-1.34,;2.02,-1.74,;-.55,-2.43,;-2.09,-2.43,;-2.57,-3.89,;-1.32,-4.8,;-.08,-3.89,;1.25,-4.66,;1.04,1.4,;.14,2.64,;2.58,1.4,;3.35,.06,;4.89,.06,;5.66,1.4,;7.2,1.4,;7.97,.06,;7.49,-1.4,;8.74,-2.31,;9.99,-1.4,;9.51,.06,;4.89,2.73,;3.35,2.73,;2.58,4.06,;3.35,5.4,;1.04,4.06,)|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC2CCCC2)cc1C(F)F)C(=O)NCC1(O)COC1 |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC2CCCC2)cc1C(F)F)C(=O)N[C@H]1C[C@H](O)C1 |r,wU:1.0,31.34,wD:33.37,(.54,-4.66,;-.8,-3.89,;-2.04,-4.8,;-3.29,-3.89,;-2.81,-2.43,;-1.27,-2.43,;-.18,-1.34,;1.3,-1.74,;-.58,.15,;-2.05,.63,;-2.05,2.17,;-.58,2.64,;.32,1.4,;1.86,1.4,;2.63,.06,;4.17,.06,;4.94,1.4,;6.48,1.4,;7.25,.06,;6.78,-1.4,;8.02,-2.31,;9.27,-1.4,;8.79,.06,;4.17,2.73,;2.63,2.73,;1.86,4.06,;2.63,5.4,;.32,4.06,;-3.38,2.94,;-3.38,4.48,;-4.71,2.17,;-6.05,2.94,;-7.54,2.54,;-7.93,4.03,;-9.27,4.8,;-6.45,4.42,)|
C[C@H]1CCCCN1C(=O)c1nc(sc1-c1cnc(NC2CCCCC2)cc1C1CC1)C(=O)NC1CCS(=O)(=O)CC1 |r|
C[C@H]1CCCCN1C(=O)c1nc(sc1-c1cnc(NC2CCCCC2)cc1C1CC1)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC2(C)CCC2)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F)C(F)(F)F |r|
CC(C)(C)Nc1cc(c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)NCC(C)(C)O)C(F)(F)F |THB:16:18:24.23:20.21|
C[C@H]1CCCCN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCCN1C(=O)c1nc(sc1-c1cnc(NC2(C)CCC2)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)NCC(C)(C)O)C(F)(F)F)C(F)(F)F |r|
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
CC(C)(C)CNc1cc(c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)NCC(C)(C)O)C(F)(F)F |THB:17:19:25.24:21.22|
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1cnc(NCC(C)(C)C)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCCN1C(=O)c1nc(sc1-c1cnc(NCC(C)(C)C)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NCC(C)(C)C)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCCN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C2CC2)cc1C(F)F)C(=O)NCC(C)(C)O |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)NCC(C)(C)O)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCCC[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F |r|
CCC(C)(C)Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)NCC(C)(C)O |THB:20:22:28.27:24.25|
CCC(C)(C)Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)NCC(C)(C)O |r|
CCC(C)(C)Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCCC[C@@H]1C)C(=O)NCC(C)(C)O |r|
CCC(C)(C)Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NCC(C)(C)O |r|
CC(C)(O)CNC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1cnc(NC(C)(C)C2CC2)cc1C(F)F |THB:11:13:19.18:15.16|
CCC(C)(C)Nc1cc(c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)NCC(C)(C)O)C(F)(F)F |THB:17:19:25.24:21.22|
CC(C)(O)CNC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1cnc(NC2(CCC2)C(F)(F)F)cc1C(F)(F)F
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1cnc(NC2(CCC2)C(F)(F)F)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
CC[C@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)NCC(C)(C)O)C(F)(F)F)C(F)(F)F |r|
CC[C@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F)C(F)(F)F |r|
CCC(C)(C)Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC2(CCC2)C(F)(F)F)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C2CC2)cc1C(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C2CC2)cc1C(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C2CC2)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
CCC(C)(C)Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CCCC[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F |r|
CCC(C)(C)Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F |r|
C[C@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F)C(F)(F)F |r|
CC[C@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F)C(F)(F)F |r|
CC[C@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CCCC[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F)C(F)(F)F |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NCC(C)(C)C)cc1C(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCCN1C(=O)c1nc(sc1-c1cnc(NCC(C)(C)C)cc1C(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1cnc(NCC(C)(C)C)cc1C(F)F)C(=O)NCC(C)(C)O |r|
CC(C)(C)CNc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)NCC(C)(C)O |THB:20:22:28.27:24.25|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NCC2(CCC2)C(F)(F)F)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1cnc(NCC2(CCC2)C(F)(F)F)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
CC(C)(O)CNC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1cnc(NCC2(CCC2)C(F)(F)F)cc1C(F)(F)F
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NCC(C)(C)C(F)(F)F)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1cnc(NCC(C)(C)C(F)(F)F)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
CC(C)(O)CNC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1cnc(NCC(C)(C)C(F)(F)F)cc1C(F)(F)F
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC2(CCC2)C(F)(F)F)cc1C(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1cnc(NC2(CCC2)C(F)(F)F)cc1C(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NCC2(CC2)C(F)(F)F)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1cnc(NCC2(CC2)C(F)(F)F)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC2CCCC2(F)F)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
CC[C@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F)C1CC1 |r|
CC[C@@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F)C1CC1 |r|
CC[C@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)NCC(C)(C)O)C(F)(F)F)C1CC1 |r,THB:15:17:23.22:19.20|
CC[C@@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)NCC(C)(C)O)C(F)(F)F)C1CC1 |r,THB:15:17:23.22:19.20|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C(F)(F)F)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C)cc1C(F)F)C(=O)NCC1(O)CCC1 |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C)cc1C(F)(F)F)C(=O)NCC1(O)CCC1 |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)NCC(C)(C)O)C(F)(F)F |r|
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C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1cnc(NC(C2CC2)C2CC2)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC(C2CC2)C2CC2)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
CC(C)(O)CNC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1cnc(NC2(C)CCC2)cc1C(F)(F)F |THB:11:13:19.18:15.16|
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1cnc(NC2(C)CCC2)cc1C(F)(F)F)C(=O)NCC(C)(C)O |r|
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CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)N[C@H]1CC[C@H](O)C1)C(F)(F)F |r|
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CC[C@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)N[C@H]1COC[C@@H]1O)C(F)(F)F)C(F)(F)F |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N[C@@H]1C[C@H]1O)C(F)(F)F |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N[C@H]1C[C@@H]1O)C(F)(F)F |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N[C@@H]1COC[C@@H]1O)C(F)(F)F |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N[C@H]1COC[C@H]1O)C(F)(F)F |r|
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CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N[C@@H]1COC[C@@H]1O)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)NCC(C)(C)O)C1CC1 |r,THB:18:20:26.25:22.23|
CC[C@@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)NCC(C)(C)O)C1CC1 |r,THB:18:20:26.25:22.23|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N[C@H]1COC[C@H]1O)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NCC(C)(C)O)C1CC1 |r|
CC[C@@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NCC(C)(C)O)C1CC1 |r|
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CC(C)(O)CNC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1cnc(NC2(C)CCC2)cc1C(F)F |THB:11:13:19.18:15.16|
CC[C@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N[C@@H]1COC[C@H]1O)C(F)(F)F)C(F)(F)F |r|
C[C@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)NCC(C)(C)O)C(F)(F)F)C1CCC1 |r,THB:14:16:22.21:18.19|
C[C@@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)NCC(C)(C)O)C(F)(F)F)C1CCC1 |r,THB:14:16:22.21:18.19|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC2(C)CCC2)cc1C(F)F)C(=O)NCC(C)(C)O |r|
CC[C@H](Nc1cc(c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N[C@H]1COC[C@@H]1O)C(F)(F)F)C(F)(F)F |r|
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CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N[C@H]1C[C@H]1O)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N[C@@H]1C[C@H]1O)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N[C@H]1C[C@@H]1O)C(F)(F)F |r|
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CNC(=O)c1nc(C(=O)N2CCC[C@@H]2C)c(s1)-c1cnc(NC(C)(C)C)cc1C(F)(F)F |r|
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CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N1CC2CCC(C1)O2)C(F)(F)F |r,TLB:26:28:35:31.32|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N[C@H]1CC[C@H]1O)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N[C@@H]1CC[C@@H]1O)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NC1CN(C1)C(C)=O)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NC1CN(C1)S(C)(=O)=O)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N1CC2(COC2)C1)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N1CC2(CCO2)C1)C(F)(F)F |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NC1CCC1O)C(F)(F)F |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N[C@@H]1CC[C@H]1O)C(F)(F)F |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N[C@H]1CC[C@@H]1O)C(F)(F)F |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N[C@H]1CC[C@H]1O)C(F)(F)F |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N[C@@H]1CC[C@@H]1O)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N1CC2CC(C1)O2)C(F)(F)F |r,TLB:26:28:31:34|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N1CC(C1)S(C)(=O)=O)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NC1CCOCC1)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N1CCOCC1)C(F)(F)F |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C)cc1C(F)F)C(=O)N[C@H]1CCC[C@@H]1O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C)cc1C(F)F)C(=O)N[C@@H]1CCC[C@H]1O |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N[C@H]1CC[C@H](O)C1)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N[C@@H]1CC[C@@H](O)C1)C(F)(F)F |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C)cc1C(F)F)C(=O)N[C@H]1C[C@H](O)C1 |r,wU:30.32,1.0,wD:32.35,(-1.83,-4.66,;-2.6,-3.33,;-4.14,-3.33,;-4.62,-1.87,;-3.37,-.96,;-2.13,-1.87,;-.64,-1.47,;.45,-2.56,;-.24,.02,;-1.71,.5,;-1.71,2.04,;-.24,2.51,;.66,1.27,;2.2,1.27,;2.97,2.6,;4.51,2.6,;5.28,1.27,;6.82,1.27,;7.59,2.6,;8.36,3.93,;6.26,3.37,;8.93,1.83,;4.51,-.07,;2.96,-.15,;2.21,-1.49,;.67,-1.51,;2.99,-2.82,;-3.04,2.81,;-3.04,4.35,;-4.37,2.04,;-5.71,2.81,;-7.19,2.41,;-7.59,3.89,;-8.93,4.66,;-6.11,4.29,)|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C)cc1C(F)F)C(=O)N[C@H]1COC[C@@H]1O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C)cc1C(F)F)C(=O)N[C@@H]1COC[C@H]1O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C)cc1C(F)F)C(=O)N[C@@H]1CC[C@H]1O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C)cc1C(F)F)C(=O)N[C@H]1CC[C@@H]1O |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)N[C@@H]1CC[C@H]1O)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)N[C@H]1CC[C@@H]1O)C(F)(F)F |r|
CC[C@@H](CO)NC(=O)c1nc(C(=O)N2CCC[C@@H]2C)c(s1)-c1cnc(N[C@@H](C)C(F)(F)F)cc1C(F)F |r|
CC[C@H](CO)NC(=O)c1nc(C(=O)N2CCC[C@@H]2C)c(s1)-c1cnc(N[C@@H](C)C(F)(F)F)cc1C(F)F |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)NC1CN(C1)S(C)(=O)=O)C(F)(F)F |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)N[C@@H]1CC[C@@H](O)C1)C(F)(F)F |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)N[C@H]1CC[C@H](O)C1)C(F)(F)F |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C)cc1C(F)F)C(=O)NC1CCOCC1 |r|
CC(C)(C)Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)N[C@H]1CC[C@H](O)C1 |r,THB:19:21:27.26:23.24|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C)cc1C(F)F)C(=O)N[C@H]1CC[C@H](O)C1 |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)N[C@H]1CC[C@H](O)C1)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)N[C@H]1CC[C@H](O)C1)C(F)(F)F |r|
O[C@H]1COC[C@@H]1NC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1cnc(N[C@@H](C2CC2)C(F)(F)F)cc1C(F)F |r,THB:12:14:20.19:16.17|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)N[C@H]1CCC[C@@H]1O)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)N[C@H]1CCC[C@@H]1O)C(F)(F)F |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)N[C@@H]1CCC[C@H]1O)C(F)(F)F |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)NC1CCS(=O)(=O)CC1)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)NC1CCOCC1)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)N[C@H](C)CO)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)N[C@@H]1CC[C@@H](O)C1)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)N[C@@H]1CCC[C@H]1O)C(F)(F)F |r|
CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)NC1CCS(=O)(=O)CC1)C(F)(F)F |r|
C[C@H](CO)NC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1cnc(NC(C)(C)C)cc1C(F)F |r,THB:10:12:18.17:14.15|
C[C@H](CO)NC(=O)c1nc(C(=O)N2CC(F)(F)C[C@@H]2C)c(s1)-c1cnc(NC(C)(C)C)cc1C(F)F |r|
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C)cc1C(F)F)C(=O)N[C@H]1C[C@H](O)C1 |r,wU:32.34,1.0,wD:34.37,(-1.28,-4.88,;-2.05,-3.54,;-3.59,-3.54,;-4.07,-2.08,;-5.4,-1.31,;-5.4,-2.85,;-2.82,-1.17,;-1.58,-2.08,;-.24,-1.31,;1.09,-2.08,;-.24,.23,;-1.71,.71,;-1.71,2.25,;-.24,2.72,;.66,1.48,;2.2,1.48,;2.97,2.81,;4.51,2.81,;5.28,1.48,;6.82,1.48,;7.59,2.81,;8.93,2.04,;6.26,3.58,;8.36,4.14,;4.51,.14,;2.95,.1,;2.18,-1.24,;2.95,-2.57,;.64,-1.24,;-3.04,3.02,;-3.04,4.56,;-4.37,2.25,;-5.71,3.02,;-7.19,2.62,;-7.59,4.11,;-8.93,4.88,;-6.11,4.51,)|
CC(C)(C)Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)N[C@@H]1CC[C@@H](O)C1 |r|
C[C@H]1CC(F)(F)CN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C)cc1C(F)F)C(=O)NC1CCS(=O)(=O)CC1 |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C)cc1C(F)F)C(=O)N[C@@H]1CC[C@@H](O)C1 |r|
CC(C)(C)Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)NC1CCS(=O)(=O)CC1
CC(C)(C)Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)N[C@@H]1CCC[C@H]1O |r|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1cnc(NC(C)(C)C)cc1C(F)F)C(=O)NC1CCS(=O)(=O)CC1 |r|
FC(F)c1cc(N[C@@H](C2CC2)C(F)(F)F)ncc1-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)NC1CCS(=O)(=O)CC1 |r|
O[C@@H]1CC[C@H](C1)NC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1cnc(N[C@@H](C2CC2)C(F)(F)F)cc1C(F)F |r|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1C2CCC1CC2)C(=O)N[C@@H]1CC[C@@H](O)C1)C(F)(F)F |r|
O[C@@H]1CCC[C@H]1NC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1cnc(N[C@@H](C2CC2)C(F)(F)F)cc1C(F)F |r|
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O[C@H]1CC[C@@H](C1)NC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1cnc(N[C@@H](C2CC2)C(F)(F)F)cc1C(F)F |r|
O[C@@H]1COC[C@H]1NC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1cnc(N[C@@H](C2CC2)C(F)(F)F)cc1C(F)F |r|
O[C@@H]1CC[C@H]1NC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1cnc(N[C@@H](C2CC2)C(F)(F)F)cc1C(F)F |r|
O[C@H]1CC[C@@H]1NC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1cnc(N[C@@H](C2CC2)C(F)(F)F)cc1C(F)F |r|
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CC[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CC(F)(F)C[C@@H]1C)C(=O)N[C@H]1C[C@H](O)C1)C(F)(F)F |r,wU:2.2,33.36,wD:31.33,26.29,(6.48,5.16,;4.95,5.32,;4.04,4.08,;2.51,4.24,;1.6,2.99,;2.23,1.59,;1.33,.34,;1.95,-1.07,;1.05,-2.31,;3.48,-1.23,;-.21,.5,;-.83,1.91,;.07,3.15,;-1.11,-.74,;-.64,-2.21,;-1.88,-3.11,;-3.13,-2.21,;-2.65,-.74,;-3.56,.5,;-2.93,1.91,;-5.09,.34,;-5.86,-.99,;-7.36,-.67,;-7.86,-2.13,;-8.87,-1.01,;-7.53,.86,;-6.12,1.48,;-5.8,2.99,;-1.88,-4.65,;-3.22,-5.42,;-.55,-5.42,;-.55,-6.96,;-1.64,-8.05,;-.55,-9.14,;-.55,-10.68,;.54,-8.05,;4.67,2.67,;5.29,1.26,;6.07,3.3,;3.26,2.04,)|
C[C@H](Nc1cc(C(F)F)c(cn1)-c1sc(nc1C(=O)N1CCC[C@@H]1C)C(=O)N1CC(C1)S(C)(=O)=O)C(F)(F)F |r|
O[C@H]1CCC[C@@H]1NC(=O)c1nc(C(=O)N2C3CCC2CC3)c(s1)-c1cnc(N[C@@H](C2CC2)C(F)(F)F)cc1C(F)F |r,THB:12:14:20.19:16.17|
C[C@H]1CCCN1C(=O)c1nc(sc1-c1ccnc(NC2CCCCC2)c1C#N)C(=O)NCC(C)(C)O |r|
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CCS(=O)(=O)c1ccc2C(NCc2c1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc2C(N(Cc2c1)C=O)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)CC1(CC1)C#N)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc2C(N(Cc2c1)C(C)=O)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)C(F)(F)C1CC1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)C1(CC1)C#N)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)CC(C)(C)O)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
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CCS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)CCF)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)CC1CCC1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)C1CCO1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)CCC#N)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)CC1(CC1)OC)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)C1CCOC1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)C1CCCO1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)CC1(CC1)N(C)C)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)CC#N)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)C1(CO)CC1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
OC(c1ccc(NC(=O)C2NCc3cc(ccc23)S(=O)(=O)CC2CC2)cc1)(C(F)(F)F)C(F)(F)F
CC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)CC1CC1
OC(c1ccc(NC(=O)C2N(Cc3cc(ccc23)S(=O)(=O)CC2CC2)C=O)cc1)(C(F)(F)F)C(F)(F)F
COCC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)CC1CC1
CCOC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)CC1CC1
COC1(CC(=O)N2Cc3cc(ccc3C2C(=O)Nc2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)CC2CC2)CC1
OC(c1ccc(NC(=O)C2N(Cc3cc(ccc23)S(=O)(=O)CC2CC2)C(=O)CC2(O)CC2)cc1)(C(F)(F)F)C(F)(F)F
CC(C)(O)CC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)CC1CC1
OC(c1ccc(NC(=O)C2N(Cc3cc(ccc23)S(=O)(=O)CC2CC2)C(=O)C2CCCO2)cc1)(C(F)(F)F)C(F)(F)F
OC(c1ccc(NC(=O)C2N(Cc3cc(ccc23)S(=O)(=O)CC2CC2)C(=O)C2(CC2)C#N)cc1)(C(F)(F)F)C(F)(F)F
OC(c1ccc(NC(=O)C2N(Cc3cc(ccc23)S(=O)(=O)CC2CC2)C(=O)C2CCOC2)cc1)(C(F)(F)F)C(F)(F)F
NC(C1CC1)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)CC1CC1
COC1(CC1)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)CC1CC1
COC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)CC1CC1
OC(c1ccc(NC(=O)C2N(Cc3cc(ccc23)S(=O)(=O)CC2CC2)C(=O)C(F)(F)C2CC2)cc1)(C(F)(F)F)C(F)(F)F
CNS(=O)(=O)c1ccc2C(NCc2c1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CNS(=O)(=O)c1ccc2C(N(Cc2c1)C(C)=O)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CNS(=O)(=O)c1ccc2C(N(Cc2c1)C=O)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CC[C@@H](O)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)NC |r,w:14.15|
CNS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)OC)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCOC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)NC
CNS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)C1(CC1)OC)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CC[C@H](O)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)NC |r|
CNS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)COC)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CNS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)C1CCO1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CNS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)[C@H]1CCCO1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F |r|
CNS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)C1CCCO1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCC(OC)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)NC
CNS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)CO)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CNC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)NC
CS(=O)(=O)c1ccc2C(NCc2c1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
CS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)Cc1ccccc1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
COC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
COC1(CC1)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
CS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)C1(CC1)C#N)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CS(=O)(=O)c1ccc2C(N(Cc2c1)C=O)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)C1CCO1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CC(CF)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
CC[C@@H](O)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O |r|
CC(C)CC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
CS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)CC1CC1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)CC1(O)CC1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
C[C@H](F)CC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O |r|
COCC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
CS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)CCF)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCOC1(CC1)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
COC1(CC(=O)N2Cc3cc(ccc3C2C(=O)Nc2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O)CC1
C[C@@H](F)CC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O |r|
COC(C)(C)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
CC(C)OC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
CC(C)(O)CC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
CC(C)[C@@H](O)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O |r|
CC(C)[C@H](O)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O |r|
CC[C@H](O)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O |r,w:15.16|
CC(CO)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
CS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)CC1COC1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)CC1(CC1)C#N)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)C1(O)CC1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)CCC#N)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)C1C[C@H](O)C1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F |r,wD:17.19,(4.27,-4.57,;5.04,-3.23,;6.38,-4,;5.81,-1.9,;3.71,-2.46,;3.71,-.92,;2.37,-.15,;1.04,-.92,;-.42,-.45,;-1.33,-1.69,;-.42,-2.94,;1.04,-2.46,;2.37,-3.23,;-2.87,-1.69,;-3.64,-.36,;-3.64,-3.03,;-3.24,-4.52,;-4.73,-4.91,;-5.5,-6.25,;-5.13,-3.43,;-.9,1.02,;-2.41,1.34,;.13,2.16,;-.35,3.63,;.68,4.77,;.21,6.23,;-1.3,6.55,;-2.33,5.41,;-1.85,3.95,;-1.77,8.02,;-3.24,7.54,;-2.25,9.48,;-2.72,10.95,;-.78,9.96,;-3.71,9.01,;-.31,8.5,;.84,7.46,;.01,10,;1.16,8.97,)|
C[C@@H](O)CC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O |r|
C[C@H](O)CC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O |r|
COC1(CCCC1)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
CC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(c(F)c1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
CS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)C1(CC1)C#N)C(=O)Nc1ccc(cc1F)C(O)(C(F)(F)F)C(F)(F)F
CC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1F)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
CS(=O)(=O)c1ccc2C(N(Cc2c1)C=O)C(=O)Nc1ccc(c(F)c1)C(O)(C(F)(F)F)C(F)(F)F
CS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)C1(CC1)C#N)C(=O)Nc1ccc(c(F)c1)C(O)(C(F)(F)F)C(F)(F)F
COC1(CC1)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(c(F)c1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
COC1(CC1)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1F)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
CS(=O)(=O)c1ccc2C(N(Cc2c1)C=O)C(=O)Nc1ccc(cc1F)C(O)(C(F)(F)F)C(F)(F)F
CC1(COC1)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
CS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)C1COC1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CC1(CCO1)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
CS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)C1(F)CC1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCC(OC)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
COC1(CCC1)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
COC(C)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
CC1(CCO1)C(=O)N1Cc2cc(ccc2[C@@H]1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O |r|
CNC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
CCNC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
CS(=O)(=O)c1ccc2C(N(Cc2c1)C(N)=O)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)NC1CC1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)NC1CC1
OC(c1ccc(NC(=O)C2NCc3cc(ccc23)S(=O)(=O)C2CC2)cc1)(C(F)(F)F)C(F)(F)F
CC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)C1CC1
COC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)C1CC1
COC1(CC1)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)C1CC1
OC(c1ccc(NC(=O)C2N(Cc3cc(ccc23)S(=O)(=O)C2CC2)C=O)cc1)(C(F)(F)F)C(F)(F)F
OCC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)C1CC1
COCC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)C1CC1
OC(c1ccc(NC(=O)C2N(Cc3cc(ccc23)S(=O)(=O)C2CC2)C(=O)C2(CC2)C#N)cc1)(C(F)(F)F)C(F)(F)F
OC(c1ccc(NC(=O)C2N(Cc3cc(ccc23)S(=O)(=O)C2CC2)C(=O)[C@@H]2CCCO2)cc1)(C(F)(F)F)C(F)(F)F |r|
OC(c1ccc(NC(=O)C2N(Cc3cc(ccc23)S(=O)(=O)C2CC2)C(=O)[C@H]2CCCO2)cc1)(C(F)(F)F)C(F)(F)F |r|
CNC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)C1CC1
COCCS(=O)(=O)c1ccc2C(NCc2c1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
COCCS(=O)(=O)c1ccc2C(N(Cc2c1)C=O)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
COCCS(=O)(=O)c1ccc2C(N(Cc2c1)C(C)=O)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
COCCS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)C1(CC1)OC)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
COCCS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)OC)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
COCCS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)CO)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
COCCS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)COC)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CNC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)CCOC
OCCS(=O)(=O)c1ccc2C(NCc2c1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)CCO
COC1(CC1)C(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)CCO
OC(c1ccc(NC(=O)C2NCc3cc(ccc23)S(=O)(=O)CC2(CC2)C#N)cc1)(C(F)(F)F)C(F)(F)F
CC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)CC1(CC1)C#N
COC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)CC1(CC1)C#N
CC(C)CS(=O)(=O)c1ccc2C(N(Cc2c1)C(C)=O)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
OC(c1ccc(NC(=O)C2NCc3cc(ccc23)S(=O)(=O)CC2(O)CC2)cc1)(C(F)(F)F)C(F)(F)F
CC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)CC1(O)CC1
OC(c1ccc(NC(=O)C2N(Cc3cc(ccc23)S(=O)(=O)CC2(O)CC2)C=O)cc1)(C(F)(F)F)C(F)(F)F
OCC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)CC1(O)CC1
CC(O)CS(=O)(=O)c1ccc2C(N(Cc2c1)C(C)=O)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
OC(c1ccc(NC(=O)C2NCc3cc(ccc23)S(=O)(=O)CC2(F)CC2)cc1)(C(F)(F)F)C(F)(F)F
CC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)CC1(F)CC1
CCOC[C@H](NC(=O)c1cnc2[C@H](C(C)C)N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)Cc2c1)c1ccc(cc1)S(=O)(=O)CC |r,wU:4.4,21.24,wD:12.12,18.17,(6.93,4.75,;5.6,3.98,;5.6,2.44,;4.26,1.67,;4.26,.13,;2.93,-.64,;1.6,.13,;1.6,1.67,;.26,-.64,;.26,-2.18,;-1.07,-2.95,;-2.4,-2.18,;-3.87,-2.65,;-4.34,-4.12,;-5.85,-4.44,;-3.31,-5.26,;-4.77,-1.41,;-6.31,-1.41,;-7.08,-.07,;-6.31,1.26,;-7.08,2.59,;-8.62,2.59,;-9.39,1.26,;-8.62,-.07,;-9.39,3.93,;-8.62,5.26,;-10.93,3.93,;-10.16,5.26,;-3.87,-.16,;-2.4,-.64,;-1.07,.13,;5.6,-.64,;5.6,-2.18,;6.93,-2.95,;8.31,-2.2,;8.27,-.64,;6.93,.13,;9.65,-2.97,;8.88,-4.31,;10.42,-1.64,;10.98,-3.74,;12.31,-2.97,)|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(co1)C1(O)COC1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(CN)co1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(CNS(C)(=O)=O)co1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(CNCC(F)(F)F)co1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(CNC(N)=O)co1 |r,THB:8:7:4.5:1,11:12:4.5:1|
C[C@@](O)(CO)c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:24:25:18.17:34,21:20:18.17:34|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(co1)[C@H](O)C1CC1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(co1)[C@@H](O)C1CC1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(co1)[C@H](O)C(F)F |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(co1)[C@@H](O)C(F)F |r,THB:8:7:4.5:1,11:12:4.5:1|
CC(C)[C@@H](O)c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:24:25:18.17:34,21:20:18.17:34|
C[C@@H](c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(C)(=O)=O |r,THB:21:22:15.14:31,18:17:15.14:31|
C[C@H](c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(C)(=O)=O |r,THB:21:22:15.14:31,18:17:15.14:31|
CC(C)S(=O)(=O)Cc1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:26:27:20.19:36,23:22:20.19:36|
C[C@H](C(N)=O)c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:24:25:18.17:34,21:20:18.17:34|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(CC(=O)NCCO)co1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnn(CCC#N)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
C[C@H](O)Cn1cc(cn1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:23:24:17.16:33,20:19:17.16:33|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnn(CCS(C)(=O)=O)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
C[C@@H](O)Cn1cc(cn1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:23:24:17.16:33,20:19:17.16:33|
C[C@@H](NS(C)(=O)=O)c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:26:27:20.19:36,23:22:20.19:36|
Cc1oc(nc1CO)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:22:23:16.15:32,19:18:16.15:32|
Cc1oc(nc1CS(C)(=O)=O)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:25:26:19.18:35,22:21:19.18:35|
CCOC(=O)NCc1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:26:27:20.19:36,23:22:20.19:36|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(CS(N)(=O)=O)co1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC(C)(C#N)c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:24:25:18.17:34,21:20:18.17:34|
C[C@H](O)CNC(=O)Cc1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:27:28:21.20:37,24:23:21.20:37|
C[C@@H](O)CNC(=O)Cc1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:27:28:21.20:37,24:23:21.20:37|
CC(C)(c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(C)(=O)=O |r,THB:22:23:16.15:32,19:18:16.15:32|
C[C@](O)(C(F)F)c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:25:26:19.18:35,22:21:19.18:35|
C[C@@](O)(C(F)F)c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:25:26:19.18:35,22:21:19.18:35|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(co1)[C@@H](O)C(N)=O |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(co1)[C@H](O)CO |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(CNC(=O)CO)co1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(co1)[C@H](O)CCO |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(co1)[C@@H](O)CCO |r,THB:8:7:4.5:1,11:12:4.5:1|
CCS(=O)(=O)C(C)(C)c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:27:28:21.20:37,24:23:21.20:37|
CC(C)(c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)C1CC1 |r,THB:22:23:16.15:32,19:18:16.15:32|
C[C@H](NS(C)(=O)=O)c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:26:27:20.19:36,23:22:20.19:36|
C[C@@H](O)C(=O)NCc1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:26:27:20.19:36,23:22:20.19:36|
CN(Cc1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(C)(=O)=O |r,TLB:22:23:16.15:32,19:18:16.15:32|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(\C=C\C#N)co1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(CCC#N)co1 |r,THB:8:7:4.5:1,11:12:4.5:1|
C[C@H](NCC(F)(F)F)c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:27:28:21.20:37,24:23:21.20:37|
C[C@H](N)c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:22:23:16.15:32,19:18:16.15:32|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(co1)[C@H](O)C(N)=O |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(co1)[C@@H](O)CO |r,TLB:8:7:4.5:1,11:12:4.5:1|
C[C@@H](N)c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:22:23:16.15:32,19:18:16.15:32|
C[C@@H](NCC(F)(F)F)c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:27:28:21.20:37,24:23:21.20:37|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1ccc(NCCO)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CCS(=O)(=O)CCn1cc(cn1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:26:27:20.19:36,23:22:20.19:36|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1ccc(NS(C)(=O)=O)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CCOC(=O)Nc1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:25:26:19.18:35,22:21:19.18:35|
CC[C@@H](O)Cn1cc(cn1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:24:25:18.17:34,21:20:18.17:34|
CC[C@H](O)Cn1cc(cn1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:24:25:18.17:34,21:20:18.17:34|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1ccn(CCS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CCS(=O)(=O)CCn1ccc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:26:27:20.19:36,23:22:20.19:36|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(CNCC(N)=O)co1 |r,THB:8:7:4.5:1,11:12:4.5:1|
Cc1oc(nc1[C@@H](O)C(F)(F)F)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:26:27:20.19:36,23:22:20.19:36|
Cc1oc(nc1[C@H](O)C(F)(F)F)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:26:27:20.19:36,23:22:20.19:36|
C[C@H](O)Cc1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:23:24:17.16:33,20:19:17.16:33|
C[C@@H](O)Cc1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:23:24:17.16:33,20:19:17.16:33|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1ccc(CS(C)(=O)=O)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
C[C@H](O)Cn1cc(cn1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:23:24:17.16:33,20:19:17.16:33|
C[C@@H](O)Cn1cc(cn1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:23:24:17.16:33,20:19:17.16:33|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnn(CCS(C)(=O)=O)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CCS(=O)(=O)[C@@H](C)c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:26:27:20.19:36,23:22:20.19:36|
CCS(=O)(=O)[C@H](C)c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:26:27:20.19:36,23:22:20.19:36|
C[C@@H](c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)C1CC1 |r,THB:21:22:15.14:31,18:17:15.14:31|
C[C@H](c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(=O)(=O)C1CC1 |r,THB:21:22:15.14:31,18:17:15.14:31|
C[C@H](C#N)c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:23:24:17.16:33,20:19:17.16:33|
C[C@@H](C#N)c1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:23:24:17.16:33,20:19:17.16:33|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1ccn(CCC#N)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1ccn(CCS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
C[C@H](O)Cn1ccc(n1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:23:24:17.16:33,20:19:17.16:33|
C[C@@H](O)Cn1ccc(n1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:23:24:17.16:33,20:19:17.16:33|
CC(C)(O)Cn1ccc(n1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:24:25:18.17:34,21:20:18.17:34|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnn(CCC#N)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnn(c1)C1(CC#N)COC1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1ccnc(NS(C)(=O)=O)c1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1ccc(N=S(C)(N)=O)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC[C@H](O)Cn1cc(cn1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:24:25:18.17:34,21:20:18.17:34|
CC[C@@H](O)Cn1cc(cn1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:24:25:18.17:34,21:20:18.17:34|
CC(C)(O)Cn1cc(cn1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:24:25:18.17:34,21:20:18.17:34|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnn(CCS(N)(=O)=O)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnn(CCNS(C)(=O)=O)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnn(CCC(N)=O)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnn(CCS(N)(=O)=O)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnn(CCO)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CS(=O)(=O)Nc1ncc(cn1)-c1cncc(n1)[C@]12CC[C@H](C1)c1cc(nnc21)-c1c(F)cccc1F |r|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1ccc(nc1)S(N)(=O)=O |r,THB:8:7:4.5:1,11:12:4.5:1|
CC(C)(O)c1ccnc(c1)-c1cncc(n1)[C@]12CC[C@H](C1)c1cc(nnc21)-c1c(F)cccc1F |r|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnn(CCO)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
C[C@H](Cn1cc(cn1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)NS(C)(=O)=O |r,TLB:22:23:16.15:32,19:18:16.15:32|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnn(C[C@@H](O)CO)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(C[S@@](C)(=N)=O)co1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(C[S@](C)(=N)=O)co1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
COCCn1cc(cn1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:23:24:17.16:33,20:19:17.16:33|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cc(ccn1)S(N)(=O)=O |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(CS(C)(=O)=O)c(Cl)o1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(CCS(C)(=O)=O)co1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1ccn(C[C@@H](O)CO)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(CO)c(CO)o1 |r,THB:8:7:4.5:1,11:12:4.5:1|
C[C@@H](Cc1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C#N |r,TLB:22:23:16.15:32,19:18:16.15:32|
C[C@H](Cc1coc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C#N |r,TLB:22:23:16.15:32,19:18:16.15:32|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1ccnc(NS(C)(=O)=O)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1ccn(C[C@H](O)CO)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1ccn(CCNS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1ccn(CCO)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC[C@@H](O)Cn1ccc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:24:25:18.17:34,21:20:18.17:34|
CC[C@H](O)Cn1ccc(n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:24:25:18.17:34,21:20:18.17:34|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnn(C[C@@H](O)C(F)(F)F)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnn(C[C@@H](O)CO)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1ccn(C[C@@H](O)C(F)(F)F)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cc(NS(C)(=O)=O)ccn1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnn(C[C@H](O)CO)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(CCS(C)(=O)=O)c(Cl)o1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnc(NS(C)(=O)=O)nc1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1ccn(C[C@H](O)C(F)(F)F)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
Cc1oc(nc1CNS(C)(=O)=O)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:26:27:20.19:36,23:22:20.19:36|
C[C@H](O)Cn1cc(nn1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:23:24:17.16:33,20:19:17.16:33|
C[C@@H](O)Cn1cc(nn1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:23:24:17.16:33,20:19:17.16:33|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1ccnc(NS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cccc(NS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1ccc(NS(C)(=O)=O)cn1 |r,THB:8:7:4.5:1,11:12:4.5:1|
C[C@H](O)Cn1nc(cc1C)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:24:25:18.17:34,21:20:18.17:34|
C[C@@H](O)Cn1nc(cc1C)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:24:25:18.17:34,21:20:18.17:34|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnn(c1)[C@@H]1C[C@H](O)C1 |r,wU:3.13,32.37,34.40,wD:6.24,THB:8:7:4.5:1,11:12:4.5:1,(-6.1,2.53,;-4.61,2.13,;-6.1,1.73,;-4.22,3.62,;-5.55,2.85,;-5.55,1.31,;-4.22,.54,;-2.88,1.31,;-1.55,.54,;-.21,1.31,;-.21,2.85,;-1.55,3.62,;-2.88,2.85,;1.12,3.62,;2.45,2.85,;2.45,1.31,;3.79,3.62,;3.79,5.16,;2.45,5.93,;1.12,5.16,;-.21,5.93,;-4.22,-1,;-5.55,-1.77,;-5.55,-3.31,;-4.22,-4.08,;-2.88,-3.31,;-2.88,-1.77,;-1.55,-4.08,;-1.39,-5.61,;.12,-5.93,;.89,-4.6,;-.14,-3.45,;2.42,-4.44,;3.65,-5.36,;4.58,-4.13,;6.1,-3.91,;3.35,-3.21,)|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnn(c1)C(CO)CO |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnn(c1)[C@H]1C[C@H](O)C1 |r,wU:3.13,32.37,wD:6.24,34.40,THB:8:7:4.5:1,11:12:4.5:1,(-6.1,2.53,;-4.61,2.13,;-6.1,1.73,;-4.22,3.62,;-5.55,2.85,;-5.55,1.31,;-4.22,.54,;-2.88,1.31,;-1.55,.54,;-.21,1.31,;-.21,2.85,;-1.55,3.62,;-2.88,2.85,;1.12,3.62,;2.45,2.85,;2.45,1.31,;3.79,3.62,;3.79,5.16,;2.45,5.93,;1.12,5.16,;-.21,5.93,;-4.22,-1,;-5.55,-1.77,;-5.55,-3.31,;-4.22,-4.08,;-2.88,-3.31,;-2.88,-1.77,;-1.55,-4.08,;-1.39,-5.61,;.12,-5.93,;.89,-4.6,;-.14,-3.45,;2.42,-4.44,;3.35,-3.21,;4.58,-4.13,;6.1,-3.91,;3.65,-5.36,)|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1nc(CCC(N)=O)co1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnn(CC#N)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnn(CCC(N)=O)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1ccc(NCCS(C)(=O)=O)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
C[C@H](O)C(=O)Nc1ccc(cn1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:26:27:20.19:36,23:22:20.19:36|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1ccc(CNS(C)(=O)=O)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1ccc(nc1)N1CC(O)C1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1ccc(NS(C)(=O)=O)nn1 |r,THB:8:7:4.5:1,11:12:4.5:1|
Cc1cc(cc(NS(C)(=O)=O)n1)-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:26:27:20.19:36,23:22:20.19:36|
Cc1cc(cc(NS(C)(=O)=O)n1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:26:27:20.19:36,23:22:20.19:36|
Cc1cc(cnc1NS(C)(=O)=O)-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:26:27:20.19:36,23:22:20.19:36|
Cc1cc(cnc1NS(C)(=O)=O)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:26:27:20.19:36,23:22:20.19:36|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnc(NS(C)(=O)=O)nc1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
C[C@H](Cn1cc(cn1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(N)=O |r,TLB:22:23:16.15:32,19:18:16.15:32|
C[C@@H](Cn1cc(cn1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C(N)=O |r,TLB:22:23:16.15:32,19:18:16.15:32|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnn(CC(N)=O)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnn(CC(=O)NCCO)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
Cc1n[nH]cc1-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:20:21:14.13:30,17:16:14.13:30|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnn(CS(C)(=O)=O)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cn(C[C@@H](O)CO)nn1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnn(C[C@@H](O)CO)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnn(C[C@H](O)CO)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnn(CCC(=O)NCCO)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnc(CC(N)=O)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
Cc1nc(NS(C)(=O)=O)ccc1-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:26:27:20.19:36,23:22:20.19:36|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-n1cnc(CC(N)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cc(CO)n[nH]1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1ccc(CNS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
Cc1cc(nn1C[C@@H](O)CO)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:25:26:19.18:35,22:21:19.18:35|
Cc1cc(nn1C[C@H](O)CO)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:25:26:19.18:35,22:21:19.18:35|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(n1)[C@@H](O)CO |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnc(NCCS(C)(=O)=O)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnc(CC(N)=O)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-n1cnc(n1)[C@H](O)CO |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-n1cnc(n1)[C@@H](O)CO |r,THB:8:7:4.5:1,11:12:4.5:1|
Cc1cc(NS(C)(=O)=O)ncc1-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:26:27:20.19:36,23:22:20.19:36|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnn(C[C@@H](O)CO)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnn(C[C@H](O)CO)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cn(C[C@H](O)CO)nn1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cn(C[C@@H](O)CO)nn1 |r,THB:8:7:4.5:1,11:12:4.5:1|
Cc1c(cnn1C[C@@H](O)CO)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:25:26:19.18:35,22:21:19.18:35|
Cc1nn(C[C@@H](O)CO)cc1-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:25:26:19.18:35,22:21:19.18:35|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(NS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CCC(N)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CCS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnc(NCC(N)=O)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnc(NCC(N)=O)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnn(CS(C)(=O)=O)c1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnn(C[C@H](O)CO)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnn(C[C@@H](O)CO)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnn(CCC(N)=O)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnn(C[C@@H](O)CO)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnn(C[C@H](O)CO)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-n1cnc(CCC(N)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-n1cnc(CCS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(n1)C(CO)CO |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-n1cnc(CNS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-n1cnc(n1)C(CO)CO |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-n1ccc(CNS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnc(NCCS(C)(=O)=O)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnc(NCCS(C)(=O)=O)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
C[C@@H](O)CNc1ncc(cn1)-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:25:26:19.18:35,22:21:19.18:35|
C[C@@H](O)CNc1ncc(cn1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:25:26:19.18:35,22:21:19.18:35|
C[C@@](O)(CO)Cn1cc(cn1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:25:26:19.18:35,22:21:19.18:35|
C[C@](O)(CO)Cn1cc(cn1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:25:26:19.18:35,22:21:19.18:35|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnn(CS(C)(=O)=O)c1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnc(NS(C)(=O)=O)cn1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CCS(=O)(=O)Nc1ncc(cn1)-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:26:27:20.19:36,23:22:20.19:36|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnc(NC[C@H](O)CO)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnc(NC[C@@H](O)CO)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnc(NCC(N)=O)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
Cc1nc(NS(C)(=O)=O)ncc1-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:26:27:20.19:36,23:22:20.19:36|
Cc1nc(NS(C)(=O)=O)ncc1-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:26:27:20.19:36,23:22:20.19:36|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnc(NCC(O)CO)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CCO)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1ccc(CCC(N)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-n1ccc(CCC(N)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC(C)S(=O)(=O)Nc1ncc(cn1)-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:27:28:21.20:37,24:23:21.20:37|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CCNS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnc(NC[C@H](O)CO)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnc(NC[C@@H](O)CO)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
C[C@H](O)CNc1ncc(cn1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:25:26:19.18:35,22:21:19.18:35|
Cc1nc(NS(C)(=O)=O)ncc1-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:26:27:20.19:36,23:22:20.19:36|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnn(CC(N)=O)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnn(C[C@@H](O)C(N)=O)c1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnn(C[C@H](O)C(N)=O)c1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cn(C[C@H](O)CO)nn1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cn(C[C@@H](O)CO)nn1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1ncnn1C[C@@H](O)CO |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1ncnn1C[C@H](O)CO |r,TLB:8:7:4.5:1,11:12:4.5:1|
C[C@H](O)Cn1cc(cn1)-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:23:24:17.16:33,20:19:17.16:33|
C[C@@H](O)Cn1cc(cn1)-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:23:24:17.16:33,20:19:17.16:33|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1ccn(CCC(N)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CNS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnn(c1)C1COC1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnn(c1)C(CO)CO |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CCS(=O)(=O)Nc1ncc(cn1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:26:27:20.19:36,23:22:20.19:36|
CC(C)S(=O)(=O)Nc1ncc(cn1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:27:28:21.20:37,24:23:21.20:37|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnc2[nH]c(=O)[nH]c2c1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1nnc(CS(=O)(=O)C2CC2)[nH]1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cn(C[C@@H](O)CO)cn1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-n1cnc(CCS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1ccn(C[C@H](O)CO)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1ccn(C[C@@H](O)CO)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
C[C@H](O)CNc1ncc(cn1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:25:26:19.18:35,22:21:19.18:35|
C[C@H](O)CNc1ncc(cn1)-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:25:26:19.18:35,22:21:19.18:35|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(Nc2cnn(C[C@@H](O)CO)c2)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(Nc2cnn(C[C@H](O)CO)c2)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnc(CCC(N)=O)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnc(CCC(N)=O)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC(C)S(=O)(=O)Nc1ncc(cn1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:27:28:21.20:37,24:23:21.20:37|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnc(CS(C)(=O)=O)nc1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnc(CS(C)(=O)=O)nc1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnc(CS(C)(=O)=O)nc1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CCC#N)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CCS(=O)(=O)Cc1nnc([nH]1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:25:26:19.18:35,22:21:19.18:35|
CC(C)S(=O)(=O)Cc1n[nH]c(n1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:26:27:20.19:36,23:22:20.19:36|
CCS(=O)(=O)Nc1ncc(cn1)-c1cncc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:26:27:20.19:36,23:22:20.19:36|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1ncnn1CS(C)(=O)=O |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1ncnn1C[C@@H](O)CO |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cn(C[C@H](O)CO)cn1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1noc(CCS(C)(=O)=O)n1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1noc(C=C)n1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1ncn(CCS(C)(=O)=O)n1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1ncn(CCS(C)(=O)=O)n1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1ncnn1CCS(C)(=O)=O |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnc(NC(N)=O)nc1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(C[C@@H](O)CO)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(n1)[C@@H]1CCS(=O)(=O)C1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(n1)[C@H]1CCS(=O)(=O)C1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnc(NS(=O)(=O)C2CC2)nc1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CCS(=O)(=O)[C@@H](C)c1nnc([nH]1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:26:27:20.19:36,23:22:20.19:36|
CCS(=O)(=O)[C@H](C)c1nnc([nH]1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,THB:26:27:20.19:36,23:22:20.19:36|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CNC(=O)CO)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1ncnn1CS(C)(=O)=O |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnc(nc1)[C@@H](O)CO |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnc(nc1)[C@@H](O)CO |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cncc(n1)-c1cnc(nc1)[C@H](O)CO |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1nnc(CCS(C)(=O)=O)o1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnc(nc1)[C@H](O)CO |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnc(nc1)[C@@H](O)CO |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnc(nc1)[C@H](O)CO |r,THB:8:7:4.5:1,11:12:4.5:1|
C[C@@H](Cc1ncn(n1)-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(C)(=O)=O |r,TLB:22:23:16.15:32,19:18:16.15:32|
C[C@H](Cc1ncn(n1)-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)S(C)(=O)=O |r,TLB:22:23:16.15:32,19:18:16.15:32|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cn(CCS(C)(=O)=O)cn1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cncn1CCS(C)(=O)=O |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CCS(=O)(=O)C2COC2)n1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CS(=O)(=O)CC2CC2)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnc(CCS(C)(=O)=O)nc1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnc(CCS(C)(=O)=O)nc1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CNC(=O)CCc1ncn(n1)-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:25:26:19.18:35,22:21:19.18:35|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(C[C@H](O)CO)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CCS(=O)(=O)CC2CC2)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(n1)C1(O)COC1 |r,THB:8:7:4.5:1,11:12:4.5:1|
Cc1cc(nc(c1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)-c1cnc(NS(C)(=O)=O)nc1 |r,TLB:15:16:9.8:25,12:11:9.8:25|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)S(C)(=O)=O |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cn(CS(C)(=O)=O)cn1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1ncn(CS(C)(=O)=O)n1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CC2CS(=O)(=O)C2)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(n1)C1CS(=O)(=O)C1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC(C)S(=O)(=O)CCc1ncn(n1)-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:27:28:21.20:37,24:23:21.20:37|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CCS(=O)(=O)C2CC2)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CS(=O)c1ncn(n1)-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:22:23:16.15:32,19:18:16.15:32|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(n1)S(C)(=O)=O |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1ncn(C[C@H](O)CO)n1 |r,TLB:8:7:4.5:1,11:12:4.5:1|
C[C@H](CS(C)(=O)=O)c1ncn(n1)-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:26:27:20.19:36,23:22:20.19:36|
C[C@@H](CS(C)(=O)=O)c1ncn(n1)-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:26:27:20.19:36,23:22:20.19:36|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(n1)[C@@H](O)CCO |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(n1)[C@H](O)CCO |r,TLB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1nccc(n1)-n1cnc(CCS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-n1cnc(C=C)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CC[S@](C)(=N)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CC[S@@](C)(=N)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(c1)-n1cnc(CCS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CCCS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(c(Cl)c21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CCS(C)(=O)=O)n1 |r,wU:3.14,wD:6.25,TLB:8:7:4.5:1,11:13:4.5:1,(-5.59,2.53,;-4.1,2.13,;-5.59,1.73,;-4.5,3.62,;-5.83,2.85,;-5.83,1.31,;-4.5,.54,;-3.16,1.31,;-1.83,.54,;-.5,1.31,;-.5,2.85,;-1.83,3.62,;-1.83,5.16,;-3.16,2.85,;.84,3.62,;2.17,2.85,;2.17,1.31,;3.51,3.62,;3.51,5.16,;2.17,5.93,;.84,5.16,;-.5,5.93,;-4.5,-1,;-5.83,-1.77,;-5.83,-3.31,;-4.5,-4.08,;-3.16,-3.31,;-3.16,-1.77,;-1.83,-4.08,;-1.67,-5.61,;-.16,-5.93,;.61,-4.6,;2.14,-4.44,;2.77,-3.03,;4.3,-2.87,;5.83,-2.71,;4.14,-1.34,;4.46,-4.4,;-.42,-3.45,)|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cc(Cl)cc1F)c1ccnc(n1)-n1cnc(CCS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cc(Cl)cc(n1)-n1cnc(CCS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(n1)C1(CS(C)(=O)=O)CC1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(CCc2ncn(n2)-c2nccc(n2)[C@@]23CC[C@@H](c4cc(nnc24)-c2c(F)cccc2F)C3(C)C)COC1 |r,TLB:23:24:17.16:33,20:19:17.16:33|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)N1CCN(CCS(C)(=O)=O)CC1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cc(O)cc1F)c1ccnc(n1)-n1cnc(CCS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1ccn(CCS(C)(=O)=O)c(=O)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
Cc1nnc([nH]1)-c1cc(nc(c1)S(C)(=O)=O)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:24:25:18.17:34,21:20:18.17:34|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-n1cnc(n1)C(F)F |r,THB:8:7:4.5:1,11:12:4.5:1|
Cc1cc(nc(c1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)-n1cnc(CCS(C)(=O)=O)n1 |r,TLB:15:16:9.8:25,12:11:9.8:25|
Cc1cc(nc(c1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)-n1cnc(CC2CS(=O)(=O)C2)n1 |r,TLB:15:16:9.8:25,12:11:9.8:25|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-n1cnc(CC2CS(=O)(=O)C2)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
Cc1cc(nc(c1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)-c1cnn(CCC(N)=O)c1 |r,TLB:15:16:9.8:25,12:11:9.8:25|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(n1)C(F)F |r,THB:8:7:4.5:1,11:12:4.5:1|
COc1cc(nc(n1)-n1cnc(CCS(C)(=O)=O)n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:27:28:21.20:37,24:23:21.20:37|
Cc1cc(nc(n1)-n1cnc(CC2CS(=O)(=O)C2)n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:27:28:21.20:37,24:23:21.20:37|
CNS(=O)(=O)c1ncn(n1)-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:24:25:18.17:34,21:20:18.17:34|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)ccc(Cl)c1F)c1ccnc(n1)-n1cnc(CCS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)ccc(O)c1F)c1ccnc(n1)-n1cnc(CCS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnc(nc1)C(O)=O |r,THB:8:7:4.5:1,11:12:4.5:1|
Cc1ccc(nc1-n1cnc(CCS(C)(=O)=O)n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:26:27:20.19:36,23:22:20.19:36|
Cc1ccc(F)c(c1F)-c1cc2[C@@H]3CC[C@@](c2nn1)(c1cccc(n1)-n1cnc(CCS(C)(=O)=O)n1)C3(C)C |r,TLB:17:16:13.14:36,10:11:13.14:36|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CC#N)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC(C)(Cc1ncn(n1)-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)C#N |r,TLB:23:24:17.16:33,20:19:17.16:33|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1ccn(CC(N)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
COCCc1cn(nc1CCS(C)(=O)=O)-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:29:30:23.22:39,26:25:23.22:39|
COCCc1nn(cc1CCS(C)(=O)=O)-c1nccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:29:30:23.22:39,26:25:23.22:39|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cc(nc(c1)-n1cnc(CCS(C)(=O)=O)n1)-n1ccc(CCS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CS(=O)(=O)C2COC2)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1ccc(CCS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnn(C[S@](C)(=N)=O)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnn(C[S@@](C)(=N)=O)c1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC(=O)NCCS(=O)(=O)Cc1ncn(n1)-c1cccc(n1)[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C |r,TLB:29:30:23.22:39,26:25:23.22:39|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1n[nH]c(CCS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-n1cnc(CS(=O)(=O)C[C@H]2CCC(=O)N2)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-n1cnc(CS(=O)(=O)C[C@@H]2CCC(=O)N2)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1nc(ncc1Br)-n1cnc(CCS(C)(=O)=O)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
Cc1cnc(nc1[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)-n1cnc(CCS(C)(=O)=O)n1 |r,TLB:15:16:9.8:25,12:11:9.8:25|
COc1cnc(nc1[C@@]12CC[C@@H](c3cc(nnc13)-c1c(F)cccc1F)C2(C)C)-n1cnc(CCS(C)(=O)=O)n1 |r,TLB:16:17:10.9:26,13:12:10.9:26|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(CCCC#N)n1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1ccc(nn1)C1(O)COC1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1ccc(NS(C)(=O)=O)nn1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnc(nc1)C1(O)COC1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnc(nc1)C1(O)COC1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)N1CCN(CCS(C)(=O)=O)C(=O)C1 |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnc(N)c(c1)C#N |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-c1cnc(NS(C)(=O)=O)c(c1)C#N |r,TLB:8:7:1:4.5,11:12:1:4.5|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnc(N)c(c1)C#N |r,THB:8:7:4.5:1,11:12:4.5:1|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1cccc(n1)-c1cnc(NS(C)(=O)=O)c(c1)C#N |r,TLB:8:7:1:4.5,11:12:1:4.5|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1cnc(n1)S(N)(=O)=O |r,TLB:8:7:1:4.5,11:12:1:4.5|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1ccc(n1)S(N)(=O)=O |r,TLB:8:7:1:4.5,11:12:1:4.5|
CC1(C)[C@H]2CC[C@@]1(c1nnc(cc21)-c1c(F)cccc1F)c1ccnc(n1)-n1ccc(n1)C(F)F |r,TLB:8:7:1:4.5,11:12:1:4.5|
CCS(=O)(=O)c1ccc(CNC(=O)c2cc3C[C@H](C)OC4(CCN(CC4)[C@H](C)c4cnc(nc4)C(F)(F)F)c3s2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cc3C[C@H](C)OC4(CCN(Cc5ccc(cc5F)-c5ncon5)CC4)c3s2)nc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cc3CC(C)OC4(CCN(CC4)C(C)c4ccc(nc4)C(F)(F)F)c3s2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2cc3CC(C)OC4(CCN(CC4)C(C)c4ccc(nc4)C(F)(F)F)c3s2)nc1
CCS(=O)(=O)c1ccc(CNC(=O)c2cc3C[C@H](C)OC4(CCN(CC4)C(C)c4cnc(s4)C(F)(F)F)c3s2)nc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cc3CCOC4(CCN(CC4)[C@@H](C)c4ccc(cc4)C#N)c3s2)cc1 |r|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)NS(=O)=O)c(Cl)c1-c1cnc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:9.9,13.16,(-1.2,-3.71,;-1.82,-2.3,;-.92,-1.05,;-1.39,.41,;-.15,1.32,;-.15,2.86,;1.19,3.63,;-1.48,3.63,;-1.48,5.17,;-2.82,5.94,;-2.71,4.4,;-4.35,5.88,;-5.17,7.19,;-4.45,8.55,;-2.91,8.6,;-2.09,7.3,;-5.26,9.85,;-4.54,11.21,;-5.36,12.52,;-3,11.27,;1.1,.41,;2.56,.89,;.62,-1.05,;1.53,-2.3,;.9,-3.71,;1.81,-4.95,;3.34,-4.79,;4.24,-6.04,;5.77,-5.88,;5.93,-7.41,;5.61,-4.34,;7.31,-5.72,;8.84,-5.55,;7.47,-7.25,;7.14,-4.18,;3.96,-3.38,;3.06,-2.14,;3.68,-.73,;5.22,-.57,;5.84,.84,;6.12,-1.82,)|
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CCn1nc(C(=O)NC[C@@]2(O)CC[C@H](C)C[C@@H]2O)c(Cl)c1-c1cnc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.9,16.17,13.13,wD:9.8,(-1.48,-2.48,;-2.11,-1.07,;-1.21,.17,;-1.68,1.64,;-.44,2.54,;-.44,4.08,;.9,4.85,;-1.77,4.85,;-1.77,6.39,;-3.1,7.16,;-3,5.63,;-2.38,8.52,;-3.2,9.83,;-4.73,9.77,;-5.55,11.08,;-5.46,8.41,;-4.64,7.11,;-5.36,5.75,;.81,1.64,;2.28,2.11,;.33,.17,;1.24,-1.07,;.61,-2.48,;1.52,-3.73,;3.05,-3.57,;3.96,-4.81,;3.33,-6.22,;4.74,-6.84,;1.92,-5.59,;2.7,-7.63,;2.08,-9.03,;4.11,-8.25,;1.3,-7,;3.68,-2.16,;2.77,-.91,;3.4,.49,;4.93,.65,;5.56,2.06,;5.83,-.59,)|
CCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)C(C)=O)c(Cl)c1-c1cnc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:12.15,(.07,-1.73,;-.55,-.32,;.35,.93,;-.12,2.39,;1.12,3.3,;1.12,4.84,;2.45,5.61,;-.21,5.61,;-.21,7.15,;-1.55,7.92,;-2.88,7.15,;-4.21,7.92,;-4.21,9.46,;-2.88,10.23,;-1.55,9.46,;-5.55,10.23,;-5.55,11.77,;-6.88,9.46,;2.37,2.39,;3.83,2.87,;1.89,.93,;2.8,-.32,;2.17,-1.73,;3.08,-2.97,;4.61,-2.81,;5.51,-4.06,;7.04,-3.9,;7.2,-5.43,;6.88,-2.36,;8.58,-3.73,;10.11,-3.57,;8.74,-5.27,;8.41,-2.2,;5.23,-1.4,;4.33,-.16,;4.95,1.25,;6.49,1.41,;7.11,2.82,;7.39,.16,)|
CCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(=O)(=O)NC(=O)NC)c(Cl)c1-c1cnc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:12.15,(-1.95,-2.6,;-2.57,-1.19,;-1.67,.05,;-2.14,1.52,;-.9,2.42,;-.9,3.96,;.44,4.73,;-2.23,4.73,;-2.23,6.27,;-3.57,7.04,;-4.9,6.27,;-6.23,7.04,;-6.23,8.58,;-4.9,9.35,;-3.57,8.58,;-7.57,9.35,;-8.9,8.58,;-7.57,10.89,;-7.57,7.81,;-8.9,7.04,;-8.9,5.5,;-10.23,7.81,;-11.57,7.04,;.35,1.52,;1.81,1.99,;-.13,.05,;.78,-1.19,;.15,-2.6,;1.06,-3.85,;2.59,-3.69,;3.49,-4.93,;5.02,-4.77,;5.19,-6.3,;4.86,-3.24,;6.56,-4.61,;8.09,-4.45,;6.72,-6.14,;6.4,-3.08,;3.21,-2.28,;2.31,-1.03,;2.94,.37,;4.47,.53,;5.09,1.94,;5.37,-.71,)|
CCn1nc(C(=O)NC[C@H]2CC[C@@H](CC2)NCS(=O)(=O)NO)c(Cl)c1-c1cnc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:12.15,(1,-4.05,;.37,-2.64,;1.28,-1.39,;.8,.07,;2.05,.98,;2.05,2.52,;3.38,3.29,;.71,3.29,;.71,4.83,;-.62,5.6,;-1.95,4.83,;-3.29,5.6,;-3.29,7.14,;-1.95,7.91,;-.62,7.14,;-4.62,7.91,;-5.95,7.14,;-7.29,7.91,;-8.06,6.57,;-6.52,9.24,;-8.62,8.68,;-9.96,7.91,;3.29,.07,;4.76,.55,;2.82,-1.39,;3.72,-2.64,;3.1,-4.05,;4,-5.29,;5.53,-5.13,;6.44,-6.38,;7.97,-6.22,;8.13,-7.75,;7.81,-4.69,;9.5,-6.06,;11.03,-5.89,;9.66,-7.59,;9.34,-4.52,;6.16,-3.72,;5.25,-2.48,;5.88,-1.07,;7.41,-.91,;8.04,.5,;8.32,-2.16,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@H](C)CC2)c(C)c1-c1cnc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:9.9,13.13,(-2.16,-2.8,;-2.79,-1.39,;-1.88,-.15,;-2.36,1.32,;-1.11,2.22,;-1.11,3.76,;.22,4.53,;-2.44,4.53,;-2.44,6.07,;-3.78,6.84,;-3.67,5.31,;-5.32,6.79,;-6.13,8.1,;-5.41,9.46,;-6.23,10.76,;-3.87,9.51,;-3.06,8.2,;.13,1.32,;1.6,1.8,;-.34,-.15,;.56,-1.39,;-.06,-2.8,;.84,-4.04,;2.37,-3.88,;3.28,-5.13,;4.81,-4.97,;4.97,-6.5,;4.65,-3.44,;6.34,-4.81,;7.87,-4.65,;6.5,-6.34,;6.18,-3.28,;3,-2.48,;2.1,-1.23,;2.72,.18,;4.25,.34,;4.88,1.74,;5.16,-.91,)|
CCn1nc(C(=O)NC[C@H]2CC[C@H](C)CC2)c(Cl)c1-c1cnc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:12.12,(-1.95,-2.6,;-2.57,-1.19,;-1.67,.05,;-2.14,1.52,;-.9,2.42,;-.9,3.96,;.44,4.73,;-2.23,4.73,;-2.23,6.27,;-3.57,7.04,;-4.9,6.27,;-6.23,7.04,;-6.23,8.58,;-7.57,9.35,;-4.9,9.35,;-3.57,8.58,;.35,1.52,;1.81,1.99,;-.13,.05,;.78,-1.19,;.15,-2.6,;1.06,-3.85,;2.59,-3.69,;3.49,-4.93,;5.02,-4.77,;5.19,-6.3,;4.86,-3.24,;6.56,-4.61,;8.09,-4.45,;6.72,-6.14,;6.4,-3.08,;3.21,-2.28,;2.31,-1.03,;2.94,.37,;4.47,.53,;5.09,1.94,;5.37,-.71,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@H](C)CC2)c(Cl)c1-c1cnc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:9.9,13.13,(-1.48,-2.3,;-2.11,-.9,;-1.2,.35,;-1.68,1.81,;-.43,2.72,;-.43,4.26,;.9,5.03,;-1.76,5.03,;-1.76,6.57,;-3.1,7.34,;-2.99,5.8,;-4.64,7.29,;-5.45,8.59,;-4.73,9.95,;-5.55,11.26,;-3.19,10.01,;-2.37,8.7,;.82,1.81,;2.28,2.29,;.34,.35,;1.25,-.9,;.62,-2.3,;1.52,-3.55,;3.06,-3.39,;3.96,-4.63,;3.33,-6.04,;4.74,-6.67,;1.93,-5.41,;2.71,-7.45,;2.08,-8.85,;4.12,-8.07,;1.3,-6.82,;3.68,-1.98,;2.78,-.74,;3.4,.67,;4.93,.83,;5.56,2.24,;5.84,-.41,)|
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CCn1nc(C(=O)NC[C@@]2(O)CC[C@H](C)C[C@@H]2O)c(Cl)c1-c1ccc(CC(C)(C)C(F)(F)F)nc1OC(F)F |r,wU:9.9,16.17,13.13,wD:9.8,(-2.08,-2.67,;-2.7,-1.27,;-1.8,-.02,;-2.27,1.44,;-1.03,2.35,;-1.03,3.89,;.31,4.66,;-2.36,4.66,;-2.36,6.2,;-3.7,6.97,;-2.31,7.64,;-4.42,8.33,;-5.96,8.38,;-6.77,7.08,;-8.31,7.13,;-6.05,5.72,;-4.51,5.66,;-3.79,4.3,;.22,1.44,;1.68,1.92,;-.26,-.02,;.65,-1.27,;.02,-2.67,;.93,-3.92,;2.46,-3.76,;3.36,-5.01,;4.89,-4.84,;5.06,-6.38,;4.73,-3.31,;6.43,-4.68,;7.96,-4.52,;6.59,-6.22,;6.26,-3.15,;3.08,-2.35,;2.18,-1.11,;2.81,.3,;4.34,.46,;4.96,1.87,;5.24,-.79,)|
CCn1nc(C(=O)NC[C@H]2CC[C@H](C)CC2)c(C)c1-c1ccc(CC(C)(C)C(F)(F)F)nc1OC(F)F |r,wU:9.8,wD:12.12,(-1.95,-2.58,;-2.58,-1.17,;-1.68,.08,;-2.15,1.54,;-.91,2.45,;-.91,3.99,;.43,4.76,;-2.24,4.76,;-2.24,6.3,;-3.57,7.07,;-4.91,6.3,;-6.24,7.07,;-6.24,8.61,;-7.57,9.38,;-4.91,9.38,;-3.57,8.61,;.34,1.54,;1.81,2.02,;-.14,.08,;.77,-1.17,;.14,-2.58,;1.05,-3.82,;2.58,-3.66,;3.49,-4.91,;5.02,-4.75,;5.18,-6.28,;4.86,-3.22,;6.55,-4.59,;8.08,-4.42,;6.71,-6.12,;6.39,-3.05,;3.21,-2.26,;2.3,-1.01,;2.93,.4,;4.46,.56,;5.09,1.97,;5.36,-.69,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@H](C)CC2)c(C)c1-c1ccc(CC(C)(C)C(F)(F)F)nc1OC(F)F |r,wU:9.8,wD:9.9,13.13,(-1.35,-2.04,;-1.97,-.63,;-1.07,.61,;-1.55,2.08,;-.3,2.98,;-.3,4.52,;1.03,5.29,;-1.63,5.29,;-1.63,6.83,;-2.97,7.6,;-1.58,8.28,;-3.78,6.3,;-5.32,6.35,;-6.05,7.71,;-7.58,7.76,;-5.23,9.02,;-3.69,8.96,;.95,2.08,;2.41,2.55,;.47,.61,;1.38,-.63,;.75,-2.04,;1.65,-3.29,;3.19,-3.13,;4.09,-4.37,;3.46,-5.78,;4.87,-6.4,;2.06,-5.15,;2.84,-7.19,;2.21,-8.59,;4.25,-7.81,;1.43,-6.56,;3.81,-1.72,;2.91,-.47,;3.53,.93,;5.07,1.09,;5.69,2.5,;5.97,-.15,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@H](C)C[C@@H]2O)c(C)c1-c1ccc(CC(C)(C)C(F)(F)F)nc1OC(F)F |r,wU:9.9,16.17,13.13,wD:9.8,(-2.08,-2.67,;-2.7,-1.27,;-1.8,-.02,;-2.27,1.44,;-1.03,2.35,;-1.03,3.89,;.31,4.66,;-2.36,4.66,;-2.36,6.2,;-3.7,6.97,;-2.31,7.64,;-4.42,8.33,;-5.96,8.38,;-6.77,7.08,;-8.31,7.13,;-6.05,5.72,;-4.51,5.66,;-3.79,4.3,;.22,1.44,;1.68,1.92,;-.26,-.02,;.65,-1.27,;.02,-2.67,;.93,-3.92,;2.46,-3.76,;3.36,-5.01,;4.89,-4.84,;5.06,-6.38,;4.73,-3.31,;6.43,-4.68,;7.96,-4.52,;6.59,-6.22,;6.26,-3.15,;3.08,-2.35,;2.18,-1.11,;2.81,.3,;4.34,.46,;4.96,1.87,;5.24,-.79,)|
CCn1nc(C(=O)NC[C@H]2CC[C@H](C)CC2)c(Cl)c1-c1ncc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:12.12,(-1.95,-2.58,;-2.58,-1.17,;-1.68,.08,;-2.15,1.54,;-.91,2.45,;-.91,3.99,;.43,4.76,;-2.24,4.76,;-2.24,6.3,;-3.57,7.07,;-4.91,6.3,;-6.24,7.07,;-6.24,8.61,;-7.57,9.38,;-4.91,9.38,;-3.57,8.61,;.34,1.54,;1.81,2.02,;-.14,.08,;.77,-1.17,;.14,-2.58,;1.05,-3.82,;2.58,-3.66,;3.49,-4.91,;5.02,-4.75,;5.18,-6.28,;4.86,-3.22,;6.55,-4.59,;8.08,-4.42,;6.71,-6.12,;6.39,-3.05,;3.21,-2.26,;2.3,-1.01,;2.93,.4,;4.46,.56,;5.09,1.97,;5.36,-.69,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@H](C)CC2)c(Cl)c1-c1ncc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:9.9,13.13,(-2.03,-2.54,;-2.66,-1.13,;-1.75,.12,;-2.23,1.58,;-.98,2.49,;-.98,4.03,;.35,4.8,;-2.31,4.8,;-2.31,6.34,;-3.65,7.11,;-2.26,7.78,;-4.46,5.8,;-6,5.85,;-6.73,7.21,;-8.27,7.27,;-5.91,8.52,;-4.37,8.47,;.26,1.58,;1.73,2.06,;-.21,.12,;.69,-1.13,;.07,-2.54,;.97,-3.78,;2.5,-3.62,;3.41,-4.87,;4.94,-4.71,;5.1,-6.24,;4.78,-3.17,;6.47,-4.54,;8,-4.38,;6.63,-6.08,;6.31,-3.01,;3.13,-2.21,;2.23,-.97,;2.85,.44,;4.38,.6,;5.01,2.01,;5.29,-.65,)|
CCn1nc(C(=O)NC[C@H]2CC[C@H](C)CC2)c(Cl)c1-c1cnc(CC(C)(C)C(F)(F)F)cc1C(C)(F)F |r,wU:9.8,wD:12.12,(6.37,-1.38,;4.83,-1.54,;3.93,-.3,;4.4,1.17,;3.16,2.07,;3.16,3.61,;4.49,4.38,;1.83,4.38,;1.83,5.92,;.49,6.69,;-.84,5.92,;-2.18,6.69,;-2.18,8.23,;-3.51,9,;-.84,9,;.49,8.23,;1.91,1.17,;.45,1.64,;2.39,-.3,;1.48,-1.54,;-.05,-1.38,;-.95,-2.63,;-.33,-4.04,;-1.23,-5.28,;-2.76,-5.12,;-2.92,-6.65,;-2.6,-3.59,;-4.29,-4.96,;-5.83,-4.8,;-4.46,-6.49,;-4.13,-3.43,;1.2,-4.2,;2.11,-2.95,;3.64,-3.11,;3.48,-4.64,;5.17,-3.27,;3.8,-1.58,)|
CCc1cc(CC(C)(C)C(F)(F)F)ncc1-c1c(Cl)c(nn1CC)C(=O)NC[C@@]1(O)CC[C@H](C)CC1 |r,wU:28.29,wD:28.30,32.34,(1.69,-4.18,;1.07,-2.77,;-.47,-2.61,;-1.37,-3.85,;-2.9,-3.69,;-3.81,-4.94,;-3.18,-6.34,;-4.59,-6.97,;-1.77,-5.72,;-2.55,-7.75,;-1.93,-9.16,;-3.96,-8.38,;-1.15,-7.13,;-3.53,-2.29,;-2.62,-1.04,;-1.09,-1.2,;-.19,.05,;-.66,1.51,;-2.13,1.99,;.58,2.42,;1.83,1.51,;1.35,.05,;2.26,-1.2,;3.79,-1.04,;.58,3.96,;-.75,4.73,;1.92,4.73,;1.92,6.27,;3.25,7.04,;3.14,5.5,;2.53,8.39,;3.34,9.7,;4.88,9.65,;5.7,10.95,;5.61,8.29,;4.79,6.98,)|
CCc1cc(C[C@@H](C)C(F)(F)F)ncc1-c1c(Cl)c(nn1CC)C(=O)NC[C@@]1(O)CC[C@H](C)CC1 |r,wU:27.28,wD:27.29,6.6,31.33,(2.01,-4.78,;1.38,-3.37,;-.15,-3.21,;-1.05,-4.45,;-2.59,-4.29,;-3.49,-5.54,;-5.02,-5.38,;-5.65,-3.97,;-5.93,-6.62,;-6.83,-7.87,;-7.17,-5.72,;-4.68,-7.53,;-3.21,-2.89,;-2.31,-1.64,;-.78,-1.8,;.13,-.56,;-.35,.91,;-1.81,1.38,;.9,1.81,;2.15,.91,;1.67,-.56,;2.57,-1.8,;4.11,-1.64,;.9,3.35,;-.43,4.12,;2.23,4.12,;2.23,5.66,;3.57,6.43,;3.46,4.9,;2.84,7.79,;3.66,9.1,;5.2,9.05,;6.01,10.35,;5.92,7.69,;5.11,6.38,)|
CCc1cc(C[C@@H](C)C(F)(F)F)ncc1-c1c(Cl)c(nn1CC)C(=O)NC[C@H]1CC[C@H](C)CC1 |r,wU:27.28,wD:6.6,30.32,(2.18,-4.55,;1.55,-3.14,;.02,-2.98,;-.89,-4.23,;-2.42,-4.07,;-3.32,-5.31,;-4.85,-5.15,;-5.48,-3.75,;-5.76,-6.4,;-6.67,-7.64,;-7.01,-5.49,;-4.51,-7.3,;-3.04,-2.66,;-2.14,-1.41,;-.61,-1.58,;.3,-.33,;-.18,1.13,;-1.64,1.61,;1.07,2.04,;2.31,1.13,;1.84,-.33,;2.74,-1.58,;4.27,-1.41,;1.07,3.58,;-.27,4.35,;2.4,4.35,;2.4,5.89,;3.74,6.66,;3.74,8.2,;5.07,8.97,;6.4,8.2,;7.74,8.97,;6.4,6.66,;5.07,5.89,)|
CCc1cc(C[C@@H](C)C(F)(F)F)ncc1-c1c(C)c(nn1CC)C(=O)NC[C@H]1CC[C@H](C)CC1 |r,wU:27.28,wD:6.6,30.32,(2.18,-4.55,;1.55,-3.14,;.02,-2.98,;-.89,-4.23,;-2.42,-4.07,;-3.32,-5.31,;-4.85,-5.15,;-5.48,-3.75,;-5.76,-6.4,;-6.67,-7.64,;-7.01,-5.49,;-4.51,-7.3,;-3.04,-2.66,;-2.14,-1.41,;-.61,-1.58,;.3,-.33,;-.18,1.13,;-1.64,1.61,;1.07,2.04,;2.31,1.13,;1.84,-.33,;2.74,-1.58,;4.27,-1.41,;1.07,3.58,;-.27,4.35,;2.4,4.35,;2.4,5.89,;3.74,6.66,;3.74,8.2,;5.07,8.97,;6.4,8.2,;7.74,8.97,;6.4,6.66,;5.07,5.89,)|
CCc1cc(CCC(C)(C)C)ncc1-c1c(Cl)c(nn1CC)C(=O)NC[C@@]1(O)CC[C@H](C)CC1 |r,wU:26.27,wD:26.28,30.32,(3.69,-3.52,;2.79,-2.27,;3.41,-.86,;4.94,-.7,;5.57,.7,;7.1,.86,;7.73,2.27,;9.26,2.38,;10.8,2.48,;10.03,3.77,;10.03,1.1,;4.66,1.95,;3.13,1.79,;2.51,.38,;.98,.22,;-.06,1.36,;.27,2.87,;-1.46,.74,;-1.3,-.79,;.21,-1.11,;.83,-2.52,;-.07,-3.77,;-2.8,1.51,;-2.8,3.05,;-4.13,.74,;-5.46,1.51,;-6.8,.74,;-6.8,2.28,;-6.8,-.8,;-8.13,-1.57,;-9.51,-.83,;-10.85,-1.6,;-9.46,.74,;-8.13,1.51,)|
CCn1nc(C(=O)NC[C@H]2CC[C@H](C)CC2)c(Cl)c1-c1cnc(CC(C)C(F)(F)F)cc1OC |r,wU:9.8,wD:12.12,(4.17,-1.53,;2.63,-1.69,;1.73,-.45,;2.2,1.02,;.96,1.92,;.96,3.46,;-.37,4.23,;2.29,4.23,;2.29,5.77,;3.63,6.54,;3.63,8.08,;4.96,8.85,;6.29,8.08,;7.63,8.85,;6.29,6.54,;4.96,5.77,;-.29,1.02,;-1.75,1.49,;.19,-.45,;-.72,-1.69,;-2.25,-1.53,;-3.15,-2.78,;-2.53,-4.18,;-3.43,-5.43,;-4.96,-5.27,;-5.59,-3.86,;-5.87,-6.51,;-6.77,-7.76,;-7.11,-5.61,;-4.62,-7.42,;-.99,-4.34,;-.09,-3.1,;1.44,-3.26,;2.07,-4.67,)|
CCn1nc(C(=O)NC[C@H]2CC[C@H](C)CC2)c(Cl)c1-c1cnc(C[C@@H](C)C(F)(F)F)cc1OC |r,wU:9.8,wD:24.26,12.12,(4.17,-1.53,;2.63,-1.69,;1.73,-.45,;2.2,1.02,;.96,1.92,;.96,3.46,;-.37,4.23,;2.29,4.23,;2.29,5.77,;3.63,6.54,;3.63,8.08,;4.96,8.85,;6.29,8.08,;7.63,8.85,;6.29,6.54,;4.96,5.77,;-.29,1.02,;-1.75,1.49,;.19,-.45,;-.72,-1.69,;-2.25,-1.53,;-3.15,-2.78,;-2.53,-4.18,;-3.43,-5.43,;-4.96,-5.27,;-5.59,-3.86,;-5.87,-6.51,;-6.77,-7.76,;-7.11,-5.61,;-4.62,-7.42,;-.99,-4.34,;-.09,-3.1,;1.44,-3.26,;2.07,-4.67,)|
CCn1nc(C(=O)NC[C@H]2CC[C@H](C)CC2)c(Cl)c1-c1cnc(C[C@H](C)C(F)(F)F)cc1OC |r,wU:9.8,24.26,wD:12.12,(4.17,-1.53,;2.63,-1.69,;1.73,-.45,;2.2,1.02,;.96,1.92,;.96,3.46,;-.37,4.23,;2.29,4.23,;2.29,5.77,;3.63,6.54,;3.63,8.08,;4.96,8.85,;6.29,8.08,;7.63,8.85,;6.29,6.54,;4.96,5.77,;-.29,1.02,;-1.75,1.49,;.19,-.45,;-.72,-1.69,;-2.25,-1.53,;-3.15,-2.78,;-2.53,-4.18,;-3.43,-5.43,;-4.96,-5.27,;-5.59,-3.86,;-5.87,-6.51,;-6.77,-7.76,;-7.11,-5.61,;-4.62,-7.42,;-.99,-4.34,;-.09,-3.1,;1.44,-3.26,;2.07,-4.67,)|
CCn1nc(C(=O)NC[C@@]2(O)CC[C@H](C)CC2)c(Cl)c1-c1cnc(O[C@H](C)C(F)(F)F)cc1OC |r,wU:9.8,25.27,wD:9.9,13.13,(3.98,-1.23,;2.45,-1.39,;1.55,-.15,;2.02,1.32,;.78,2.22,;.78,3.76,;-.56,4.53,;2.11,4.53,;2.11,6.07,;3.44,6.84,;3.34,5.31,;2.72,8.2,;3.54,9.51,;5.08,9.46,;5.89,10.76,;5.8,8.1,;4.98,6.79,;-.47,1.32,;-1.93,1.79,;.01,-.15,;-.9,-1.39,;-2.43,-1.23,;-3.34,-2.48,;-2.71,-3.88,;-3.61,-5.13,;-5.15,-4.97,;-5.77,-3.56,;-6.05,-6.21,;-6.96,-7.46,;-7.3,-5.31,;-4.81,-7.12,;-1.18,-4.05,;-.27,-2.8,;1.26,-2.96,;1.89,-4.37,)|
CCn1nc(C(=O)NC[C@H]2CC[C@H](C)CC2)c(Cl)c1-c1cnc(O[C@@H](C)C(F)(F)F)cc1OC |r,wU:9.8,wD:24.26,12.12,(4.15,-1.02,;2.62,-1.18,;1.71,.07,;2.19,1.53,;.94,2.44,;.94,3.98,;-.39,4.75,;2.28,4.75,;2.28,6.29,;3.61,7.06,;3.61,8.6,;4.94,9.37,;6.28,8.6,;7.61,9.37,;6.28,7.06,;4.94,6.29,;-.3,1.53,;-1.77,2.01,;.17,.07,;-.73,-1.18,;-2.26,-1.02,;-3.17,-2.26,;-2.54,-3.67,;-3.45,-4.92,;-4.98,-4.75,;-5.61,-3.35,;-5.88,-6,;-6.79,-7.25,;-7.13,-5.1,;-4.64,-6.91,;-1.01,-3.83,;-.11,-2.58,;1.43,-2.75,;2.05,-4.15,)|
CCn1nc(C(=O)NC[C@H]2CC[C@H](C)CC2)c(Cl)c1-c1cnc(O[C@H](C)C(F)(F)F)cc1OC |r,wU:9.8,24.26,wD:12.12,(4.15,-1.02,;2.62,-1.18,;1.71,.07,;2.19,1.53,;.94,2.44,;.94,3.98,;-.39,4.75,;2.28,4.75,;2.28,6.29,;3.61,7.06,;3.61,8.6,;4.94,9.37,;6.28,8.6,;7.61,9.37,;6.28,7.06,;4.94,6.29,;-.3,1.53,;-1.77,2.01,;.17,.07,;-.73,-1.18,;-2.26,-1.02,;-3.17,-2.26,;-2.54,-3.67,;-3.45,-4.92,;-4.98,-4.75,;-5.61,-3.35,;-5.88,-6,;-6.79,-7.25,;-7.13,-5.1,;-4.64,-6.91,;-1.01,-3.83,;-.11,-2.58,;1.43,-2.75,;2.05,-4.15,)|
CC1(C)Cc2cc(NC(=O)c3cnn4cccnc34)c(cc2O1)N1CCN(CCN)CC1
CC1(C)Cc2cc(NC(=O)c3cnn4cccnc34)c(cc2O1)N1CCN(CCNS(C)(=O)=O)CC1
CC(=O)NCCN1CCN(CC1)c1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2cccnc12
CN(C)CCN1CCN(CC1)c1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2cccnc12
Cc1ccc(=O)[nH]c1CN1CCN(CC1)c1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2cccnc12
CC1(C)Cc2cc(NC(=O)c3cnn4cccnc34)c(cc2O1)N1CCN(C[C@@H]2CCCC(=O)N2)CC1 |r|
Cc1nc[nH]c1CN1CCN(CC1)c1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2cccnc12
CCc1nc[nH]c1CN1CCN(CC1)c1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2cccnc12
CC1(C)Cc2cc(NC(=O)c3cnn4cccnc34)c(cc2O1)N1CCN(Cc2[nH]cnc2Cl)CC1
Cc1ncsc1CN1CCN(CC1)c1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2cccnc12
Cc1oncc1CN1CCN(CC1)c1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2cccnc12
CC1(C)Cc2cc(NC(=O)c3cnn4cccnc34)c(cc2O1)N1CCN(CC1)C1COC1
Cc1nocc1CN1CCN(CC1)c1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2cccnc12
CCc1oc(=O)[nH]c1CN1CCN(CC1)c1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2cccnc12
Cc1noc(C)c1CN1CCN(CC1)c1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2cccnc12
CC[C@@H]1CC(=O)NN1C1CCN(CC1)c1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2cccnc12 |r|
CC1(C)Cc2cc(NC(=O)c3cnn4cccnc34)c(O[C@H]3CN(CC(N)=O)C[C@@H]3N)cc2O1 |r|
COc1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2ccc(Cl)nc12
CCN1C[C@H](COc2cc3OC(C)(C)Cc3cc2NC(=O)c2cnn3cccnc23)CC1=O |r|
CN1C[C@H](COc2cc3OC(C)(C)Cc3cc2NC(=O)c2cnn3cccnc23)CC1=O |r|
CC1(C)Cc2cc(NC(=O)c3cnn4cccnc34)c(OC[C@@H]3Cc4ccccc4[C@H]3N)cc2O1 |r|
CC1(C)Cc2cc(NC(=O)c3cnn4cccnc34)c(OC[C@H]3C[C@@H]4NCCO[C@H]4C3)cc2O1 |r|
COc1cc2OC(C)(C)Cc2cc1CC(=O)c1cnn2ccc(nc12)C1CCNC1=O
COc1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2ccc(nc12)N1C[C@@H](N)CC(F)(F)C1 |r|
COc1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2ccc(nc12)N(C)C1CC1
COc1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2ccc(nc12)N1CCC[C@@H](N)C1 |r|
COc1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2ccc(N[C@@H]3CCCNC3)nc12 |r|
COc1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2ccc(N)nc12
COc1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2ccc(nc12)N1CCNCC1
COc1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2ccc(NCCN)nc12
COc1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2ccc(nc12)N(C)C
CC1(C)Cc2cc3NC(=O)c4cnn5ccc(NCCN6CCN(CC6)c3cc2O1)nc45
O=C(Nc1cc2CCC(=O)Nc2cc1N1CCOCC1)c1cnn2cccnc12
OCCN1C(=O)CCc2cc(NC(=O)c3cnn4cccnc34)c(cc12)N1CCOCC1
OCCCN1C(=O)CCc2cc(NC(=O)c3cnn4cccnc34)c(cc12)N1CCOCC1
CC1(C)Cc2cc(NC(=O)c3cnn4ccc(=O)[nH]c34)c(cc2O1)N1CCOCC1
C[C@@]1(CCC#N)COc2cc(N3CCOCC3)c(NC(=O)c3cnn4cccnc34)cc2C1 |r|
Cn1cc(COc2cc3C(=O)N(C[C@@H](F)C(C)(C)O)Cc3cc2NC(=O)c2cnn3cccnc23)cn1 |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(O[C@@H]3C[C@H](F)C3)cc2C1=O |r,wU:26.27,28.30,wD:4.4,(-7.2,.34,;-7.24,1.88,;-8.73,1.48,;-8.01,3.22,;-5.7,1.88,;-4.93,3.22,;-4.93,.55,;-3.39,.55,;-2.49,1.79,;-1.02,1.32,;.31,2.09,;1.64,1.32,;2.98,2.09,;2.98,3.63,;1.64,4.4,;4.31,4.4,;4.47,5.93,;5.98,6.25,;6.75,4.92,;8.25,4.6,;8.73,3.13,;7.7,1.99,;6.19,2.31,;5.72,3.77,;1.64,-.22,;2.98,-.99,;2.98,-2.53,;1.89,-3.62,;2.98,-4.71,;2.98,-6.25,;4.07,-3.62,;.31,-.99,;-1.02,-.22,;-2.49,-.7,;-2.96,-2.16,)|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(O[C@H]3CCNC3)cc2C1=O |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(O[C@@H]3C[C@H](Cl)C3)cc2C1=O |r,wU:26.27,28.30,wD:4.4,(-7.2,.34,;-7.24,1.88,;-8.73,1.48,;-8.01,3.22,;-5.7,1.88,;-4.93,3.22,;-4.93,.55,;-3.39,.55,;-2.49,1.79,;-1.02,1.32,;.31,2.09,;1.64,1.32,;2.98,2.09,;2.98,3.63,;1.64,4.4,;4.31,4.4,;4.47,5.93,;5.98,6.25,;6.75,4.92,;8.25,4.6,;8.73,3.13,;7.7,1.99,;6.19,2.31,;5.72,3.77,;1.64,-.22,;2.98,-.99,;2.98,-2.53,;1.89,-3.62,;2.98,-4.71,;2.98,-6.25,;4.07,-3.62,;.31,-.99,;-1.02,-.22,;-2.49,-.7,;-2.96,-2.16,)|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(OCC(F)F)cc2C1=O |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(O[C@H]3CC[C@@H](O)C3)cc2C1=O |r|
CC(C)Oc1cc2C(=O)N(Cc2cc1NC(=O)c1cnn2cccnc12)[C@H]1CCOC1 |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(OC3CCNCC3)cc2C1=O |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(OC[C@@H]3CNC(=O)C3)cc2C1=O |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(OC3CNC3)cc2C1=O |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(OC3CC3)cc2C1=O |r|
CC(C)Oc1cc2C(=O)N(C[C@@H](F)C(C)(C)O)Cc2cc1NC(=O)c1cnn2cccnc12 |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(OCC3COC3)cc2C1=O |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(OC3CCCC3)cc2C1=O |r|
CC(C)Oc1cc2C(=O)N(C[C@@H](F)C(C)(C)O)Cc2cc1NC(=O)c1cnn2cc(C)cnc12 |r|
CCOc1cc2C(=O)N(C[C@@H](F)C(C)(C)O)Cc2cc1NC(=O)c1cnn2cccnc12 |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(O[C@@H]3CCOC3)cc2C1=O |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(OC3CCOCC3)cc2C1=O |r|
COc1cc2C(=O)N(C[C@@H](F)C(C)(C)O)Cc2cc1NC(=O)c1cnn2cccnc12 |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(OC3COC3)cc2C1=O |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(OC(F)F)cc2C1=O |r|
Cn1cc(Oc2cc3C(=O)N(C[C@@H](F)C(C)(C)O)Cc3cc2NC(=O)c2cnn3cccnc23)cn1 |r|
CC(C)(C)Oc1cc2C(=O)N(C[C@@H](F)C(C)(C)O)Cc2cc1NC(=O)c1cnn2cccnc12 |r|
CNc1cc2C(=O)N(C[C@@H](F)C(C)(C)O)Cc2cc1NC(=O)c1cnn2cccnc12 |r|
O=C(Nc1cc2CN(CC3CCOCC3)C(=O)c2cc1N1CCOCC1)c1cnn2cccnc12
O=C(Nc1cc2CN(CCN3CCCC3)C(=O)c2cc1N1CCOCC1)c1cnn2cccnc12
O=C(Nc1cc2CN(C3CC4(COC4)C3)C(=O)c2cc1N1CCOCC1)c1cnn2cccnc12
CC(C)N1Cc2cc(NC(=O)c3cnn4cccnc34)c(cc2C1=O)N(C)C
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(cc2C1=O)N1CCC(CC(F)F)CC1 |r|
CC(C)N1Cc2cc(NC(=O)c3cnn4cccnc34)c(cc2C1=O)C1CC1
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(cc2C1=O)C#N |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(cc2C1=O)N1CCN2CCC[C@@H]2C1 |r|
CO[C@@H]1C[C@H]2CN(CCN2C1)c1cc2C(=O)N(C[C@@H](F)C(C)(C)O)Cc2cc1NC(=O)c1cnn2cccnc12 |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4ccc(Cl)nc34)c(cc2C1=O)N1CCOCC1 |r|
CCc1oncc1CN1CCN(CC1)c1cc2C(=O)N(C[C@@H](F)C(C)(C)O)Cc2cc1NC(=O)c1cnn2cccnc12 |r|
CCc1nocc1CN1CCN(CC1)c1cc2C(=O)N(C[C@@H](F)C(C)(C)O)Cc2cc1NC(=O)c1cnn2cccnc12 |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(cc2C1=O)N1CCN(CC1)C1COC1 |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(cc2C1=O)N1CCN(CCn2ccnc2)CC1 |r|
CO[C@@H]1C[C@@H]2CN(CCN2C1)c1cc2C(=O)N(C[C@@H](F)C(C)(C)O)Cc2cc1NC(=O)c1cnn2cccnc12 |r|
CO[C@H]1C[C@@H]2CN(CCN2C1)c1cc2C(=O)N(C[C@@H](F)C(C)(C)O)Cc2cc1NC(=O)c1cnn2cccnc12 |r|
CC(F)(F)CN1CCN(CC1)c1cc2C(=O)N(C[C@@H](F)C(C)(C)O)Cc2cc1NC(=O)c1cnn2cccnc12 |r|
C[C@H]1C[C@@H]2CN(CCN2C1)c1cc2C(=O)N(C[C@@H](F)C(C)(C)O)Cc2cc1NC(=O)c1cnn2cccnc12 |r|
COCCN1CCN(CC1)c1cc2C(=O)N(C[C@@H](F)C(C)(C)O)Cc2cc1NC(=O)c1cnn2cccnc12 |r|
CC(C)N1CCN(CC1)c1cc2C(=O)N(C[C@@H](F)C(C)(C)O)Cc2cc1NC(=O)c1cnn2cccnc12 |r|
CN(C)c1cc2C(=O)N(C[C@@H](F)C(C)(C)O)Cc2cc1NC(=O)c1cnn2ccc(NC(C)=O)nc12 |r|
CN(C)c1cc2C(=O)N(C[C@@H](F)C(C)(C)O)Cc2cc1NC(=O)c1cnn2ccc(nc12)C(=O)NC1CC1 |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cc(O)cnc34)c(cc2C1=O)N1CCOCC1 |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(OCC(F)(F)F)cc2C1=O |r|
Cc1ccc(nc1)-c1cc2OC(C)(C)Cc2cc1NC(=O)c1cnn2cccnc12
Cc1ccc(nc1)-c1cc2C(=O)N(C[C@@H](F)C(C)(C)O)Cc2cc1NC(=O)c1cnn2cccnc12 |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(cc2C1=O)C1COC1 |r|
CC(C)(O)[C@H](F)CN1Cc2cc(NC(=O)c3cnn4cccnc34)c(cc2C1=O)C(C)(C)O |r|
CC(C)N1Cc2cc(NC(=O)c3cnn4cccnc34)c(N(C)C)c(CO)c2C1=O
Cn1ccc2cc(NC(=O)c3cnn4cccnc34)c(cc2c1=O)N1CCOCC1
O=C(Nc1cc2SCCOc2cc1N1CCOCC1)c1cnn2cccnc12
CC1(C)Cc2cc(NC(=O)c3cnn4cccnc34)c(cc2[S@]1=O)N1CCOCC1 |r|
CN(C)c1cc2[C@H](O)C(C)(C)Cc2cc1NC(=O)c1cnn2cccnc12 |r|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(OC)(C(F)(F)F)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(OC3CCCCC3)c(c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(C3=CCC(=O)CC3)c(c2)C(F)(F)F)cc1 |t:17|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C2CCCCC2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(C3=CCC(O)CC3)c(c2)C(F)(F)F)cc1 |t:17|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3c(CCCC3(O)c3ccc(OC)cc3)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3C(=O)C(C)(CCc3n2)c2ccc(OC)nc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3C(=O)C(C)(CCc3n2)c2nccn3ccnc23)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3C(=O)C(C)(CCc3n2)c2cc(C)nc(C)n2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3C(=O)C(C)(CCc3n2)c2nccn3cc(C)nc23)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3C(=O)C(C)(CCc3n2)c2ccc(OC)nn2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3C(=O)C(C)(CCc3n2)c2nccn3cccc23)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3C(=O)C(C)(CCc3n2)c2nc(C)cn3ccnc23)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(C)c3C(=O)C(C)(CCc3n2)c2cccc(OC)n2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(C)c3C(=O)C(C)(CCc3n2)c2nccc(OC)n2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(C)c3C(=O)C(C)(CCc3n2)c2cc(OC)ccn2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(C)c3C(=O)C(C)(CCc3n2)c2nccn3ccnc23)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(C)c3C(=O)C(C)(CCc3n2)c2cc(C)nc(C)n2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(C)c3C(=O)C(C)(CCc3n2)c2nc(C)cc(C)n2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(C)c3C(=O)C(C)(CCc3n2)c2ccc(OC)nn2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(C)c3C(=O)C(C)(CCc3n2)c2ccc(C)nn2)cc1
COc1ccc(nn1)C1(C)CCc2nc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)cc(C)c2C1=O
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(C)c3C(=O)C(C)(CCc3n2)c2ccc3OCOc3c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(C)c3C(=O)C(C)(CCc3n2)c2ccc3n(C)cnc3c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3C(=O)C(C)(CCc3n2)n2nc(C)cc2C)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(C)c3C(=O)C(C)(CCc3n2)n2cccn2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3C(=O)C(C)(CCc3n2)c2nccn3c(C)cnc23)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3C(=O)C(C)(CCc3n2)c2ccnc(n2)C(C)C)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3C(=O)C(C)(CCc3n2)c2ncc(OC)cn2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(C)c3C(=O)C(C)(CCc3n2)c2ncc(OC)cn2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3C(=O)C(C)(CCc3n2)c2ccc(nn2)C(C)C)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(C)c3C(=O)C(C)(CCc3n2)c2cccnc2O)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(C)c3C(=O)C(C)(CCc3n2)c2ncccc2O)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(C)c3C(=O)C(C)(CCc3n2)c2c(C)ccnc2O)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3C(=O)C(c4ncccc4O)C(C)(C)Cc3n2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(C)c3C(=O)C(C)(CCc3n2)c2ccc(O)cn2)cc1
Cc1cc(NC(=O)Cc2ccc(cc2)S(C)(=O)=O)nc2CCC(C)(C(=O)c12)c1ncccc1O
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3C(=O)C(c4ccc(O)cn4)C(C)(C)Cc3n2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3C(=O)C(C(C)Cc3n2)c2ncccc2O)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3C(=O)C(C)(CCc3n2)c2ncc(Cl)n3ccnc23)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc3CCC(C)(C(=O)c3cn2)c2cc(C)nc(C)n2)cc1
CCc1nc(C)cc(n1)C1(C)CCc2nc(NC(=O)Cc3ccc(cc3)S(=O)(=O)CC)ccc2C1=O
CCc1cc(nc(CC)n1)C1(C)CCc2nc(NC(=O)Cc3ccc(cc3)S(=O)(=O)CC)ccc2C1=O
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(C)c3C(=O)C(C)(CCc3n2)c2cc(C)nc(OC)n2)cc1
CCc1cc(CN2CC3(C2)CN(C3)C(=O)OC(C)(C)C)ccc1-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCc1cc(CN2CC3(C2)CN(C3)S(C)(=O)=O)ccc1-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCc1cc(CN2CC3(C2)CCS(=O)(=O)CC3)ccc1-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCc1cc(CN2CCC3(CN(C3)S(C)(=O)=O)CC2)ccc1-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCc1cc(CN2CCCC3(CN(C3)S(C)(=O)=O)C2)ccc1-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCc1cc(CN2CC3(C2)CCN(C3)S(C)(=O)=O)ccc1-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CC(C)c1c(F)c(CN2CC3(C2)CN(C3)S(C)(=O)=O)cc(F)c1-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CC(C)c1c(F)c(CN2CC3(C2)CN(C3)S(C)(=O)=O)c(F)cc1-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCc1cc(CN2CCC(CS(C)(=O)=O)CC2)ccc1-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCc1cc(CN2CCC(CC2)S(C)(=O)=O)ccc1-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CC(C)c1cc(CN2CCC3(CS(=O)(=O)C3)C2)ccc1-c1ccc(cc1C)C(O)(C(F)(F)F)C(F)(F)F
CC(C)c1cc(CN2CC3(C2)CS(=O)(=O)C3)ccc1-c1ccc(cc1C)C(O)(C(F)(F)F)C(F)(F)F
CCC(C)c1cc(CN2CC3(C2)CN(C3)S(C)(=O)=O)ccc1-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CC(C)c1cc(CN2CC3(C2)CN(C3)S(C)(=O)=O)c(F)c(F)c1-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CC(C)c1cc(CN2CC3(C2)CN(C3)S(C)(=O)=O)cc(F)c1-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCc1cc(CN2CCC3(CS(=O)(=O)C3)C2)ccc1-c1ccc(cc1C)C(O)(C(F)(F)F)C(F)(F)F
CCc1cc(CN2CCC3(CS(=O)(=O)C3)C2)ccc1-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCc1cc(CN2CC3(C2)CS(=O)(=O)C3)ccc1-c1ccc(cc1C)C(O)(C(F)(F)F)C(F)(F)F
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Cc1cc(ccc1-c1c(F)cc(CN2CC3(C2)CN(C3)S(C)(=O)=O)c(F)c1C1CC1)C(O)(C(F)(F)F)C(F)(F)F |(-5.85,.95,;-5.08,-.38,;-5.85,-1.72,;-5.08,-3.05,;-3.54,-3.05,;-2.77,-1.72,;-3.54,-.38,;-2.77,.95,;-3.54,2.28,;-5.08,2.28,;-2.77,3.62,;-1.23,3.62,;-.46,4.95,;1.08,4.95,;2.17,3.86,;3.26,4.95,;2.17,6.04,;4.35,6.04,;5.44,4.95,;4.35,3.86,;6.98,4.95,;8.52,4.95,;6.98,3.41,;6.98,6.49,;-.46,2.28,;1.08,2.28,;-1.23,.95,;-.46,-.38,;-.46,-1.92,;.87,-1.15,;-5.85,-4.39,;-6.62,-5.72,;-7.18,-3.62,;-6.41,-2.28,;-7.95,-4.95,;-8.52,-2.85,;-4.52,-5.16,;-3.75,-3.82,;-5.29,-6.49,;-3.18,-5.93,)|
CCc1cc(ccc1-c1c(F)cc(CN2CC3(C2)CN(C3)S(C)(=O)=O)c(F)c1C1CC1)C(O)(C(F)(F)F)C(F)(F)F |(-7.39,.95,;-5.85,.95,;-5.08,-.38,;-5.85,-1.72,;-5.08,-3.05,;-3.54,-3.05,;-2.77,-1.72,;-3.54,-.38,;-2.77,.95,;-3.54,2.28,;-5.08,2.28,;-2.77,3.62,;-1.23,3.62,;-.46,4.95,;1.08,4.95,;2.17,3.86,;3.26,4.95,;2.17,6.04,;4.35,6.04,;5.44,4.95,;4.35,3.86,;6.98,4.95,;8.52,4.95,;6.98,3.41,;6.98,6.49,;-.46,2.28,;1.08,2.28,;-1.23,.95,;-.46,-.38,;-.46,-1.92,;.87,-1.15,;-5.85,-4.39,;-6.62,-5.72,;-7.18,-3.62,;-6.41,-2.28,;-7.95,-4.95,;-8.52,-2.85,;-4.52,-5.16,;-3.75,-3.82,;-5.29,-6.49,;-3.18,-5.93,)|
CS(=O)(=O)N1CC2(CN(Cc3cc(F)c(-c4ccc(cc4F)C(O)(C(F)(F)F)C(F)(F)F)c(C4CC4)c3F)C2)C1 |(-8.52,4.95,;-6.98,4.95,;-6.98,6.49,;-6.98,3.41,;-5.44,4.95,;-4.35,3.86,;-3.26,4.95,;-2.17,3.86,;-1.08,4.95,;.46,4.95,;1.23,3.62,;2.77,3.62,;3.54,2.28,;5.08,2.28,;2.77,.95,;3.54,-.38,;2.77,-1.72,;3.54,-3.05,;5.08,-3.05,;5.85,-1.72,;5.08,-.38,;5.85,.95,;5.85,-4.39,;6.62,-5.72,;7.18,-3.62,;6.41,-2.28,;7.95,-4.95,;8.52,-2.85,;4.52,-5.16,;3.75,-3.82,;5.29,-6.49,;3.18,-5.93,;1.23,.95,;.46,-.38,;-.87,-1.15,;.46,-1.93,;.46,2.28,;-1.08,2.28,;-2.17,6.04,;-4.35,6.04,)|
CS(=O)(=O)N1CC2(CN(Cc3cc(F)c(-c4ccc(cc4Cl)C(O)(C(F)(F)F)C(F)(F)F)c(C4CC4)c3F)C2)C1 |(-8.52,4.95,;-6.98,4.95,;-6.98,6.49,;-6.98,3.41,;-5.44,4.95,;-4.35,3.86,;-3.26,4.95,;-2.17,3.86,;-1.08,4.95,;.46,4.95,;1.23,3.62,;2.77,3.62,;3.54,2.28,;5.08,2.28,;2.77,.95,;3.54,-.38,;2.77,-1.72,;3.54,-3.05,;5.08,-3.05,;5.85,-1.72,;5.08,-.38,;5.85,.95,;5.85,-4.39,;6.62,-5.72,;7.18,-3.62,;6.41,-2.28,;7.95,-4.95,;8.52,-2.85,;4.52,-5.16,;3.75,-3.82,;5.29,-6.49,;3.18,-5.93,;1.23,.95,;.46,-.38,;-.87,-1.15,;.46,-1.93,;.46,2.28,;-1.08,2.28,;-2.17,6.04,;-4.35,6.04,)|
[H][C@]12CCc3c(OC)nc(OC)nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2C |r,t:18|
COc1cc(ccn1)-c1nc(OC)c2CC[C@@H]3[C@@H](C)C(=O)C(=C[C@@]3(C)c2n1)C#N |r,c:22|
COc1nc(nc2c1CC[C@@H]1[C@@H](C)C(=O)C(=C[C@@]21C)C#N)-c1ccnc(C)c1 |r,c:16|
COc1nc(nc2c1CC[C@@H]1[C@@H](C)C(=O)C(=C[C@@]21C)C#N)-c1ccncc1C |r,c:16|
[H][C@]12CCc3c(OC)nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2C)-c1ccncc1 |r,t:16|
COc1nc(nc2c1CC[C@@H]1[C@@H](C)C(=O)C(=C[C@@]21C)C#N)-c1ccnc(F)c1 |r,c:16|
COc1nc(nc2c1CC[C@@H]1[C@@H](C)C(=O)C(=C[C@@]21C)C#N)-c1cccnc1 |r,c:16|
COc1nc(Nc2ccncc2)nc2c1CC[C@@H]1[C@@H](C)C(=O)C(=C[C@@]21C)C#N |r,c:24|
COc1nc(nc2c1CC[C@@H]1[C@@H](C)C(=O)C(=C[C@@]21C)C#N)-c1ccnc2ccccc12 |r,c:16|
COc1nc(CCNC=O)nc2c1CC[C@@H]1[C@@H](C)C(=O)C(=C[C@@]21C)C#N |r,c:21|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)CC(C#N)=C1O)-c1ccncc1)-c1ccccc1 |r,c:18|
[H][C@]12CCc3c(nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2C)-c1ccncc1)-c1ccccc1 |r,t:14|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)[C@@H]2O[C@]2(C#N)C1=O)-c1ccncc1)-c1ccccc1 |r|
[H][C@]12CCc3c(nc(nc3[C@]1(C)C=C(C(N)=O)C(=O)[C@@H]2C)-c1ccncc1)-c1ccccc1 |r,t:14|
C[C@@H]1[C@H]2CCc3c(O)nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccncc1 |r,t:16|
C[C@@H]1[C@H]2CCc3c(OS(=O)(=O)c4ccc(C)cc4)nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccncc1 |r,t:27|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccccc1)-c1ccccc1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccc(cc1)C(F)(F)F)-c1ccccc1 |r,t:15|
[H][C@]12CCc3c(nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2C)-c1ccncc1)-c1ccc(CO)cc1 |r,t:14|
C[C@@H]1[C@H]2CCc3c(ncnc3[C@]2(C)C=C(C#N)C1=O)-c1ccccc1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)C1CCCCC1)-c1ccccc1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccncc1)-c1ccc(cc1)C(F)(F)F |r,t:15|
[H][C@]12CCc3c(nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2C)-c1ccncc1)-c1cccnc1 |r,t:14|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccncc1)-c1cccc(c1)C(F)(F)F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccncc1)-c1ccc(C)cc1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccncc1)-c1ccc(Cl)cc1 |r,t:15|
[H][C@]12CCc3c(nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2C)-c1ccncc1)-c1ccncc1 |r,t:14|
COc1ccc(cc1)-c1nc(nc2c1CC[C@@H]1[C@@H](C)C(=O)C(=C[C@@]21C)C#N)-c1ccncc1 |r,c:23|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccncc1)-c1ccc(Cl)c(Cl)c1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1ccccc1 |r,t:15|
COc1cc(ccn1)-c1nc(-c2ccccc2)c2CC[C@@H]3[C@@H](C)C(=O)C(=C[C@@]3(C)c2n1)C#N |r,c:27|
C[C@@H]1[C@H]2CCc3c(nc(N)nc3[C@]2(C)C=C(C#N)C1=O)-c1ccccc1 |r,t:16|
C[C@@H]1[C@H]2CCc3c(nc(NC(=O)C4CCCCC4)nc3[C@]2(C)C=C(C#N)C1=O)-c1ccccc1 |r,t:25|
[H][C@]12CCc3c(Cc4ccccc4)nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2C)-c1ccncc1 |r,t:22|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1ccccc1F |r,t:15|
CC1=C2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1ccccc1F |r,c:1,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1cccc(F)c1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1ccc(F)cc1 |r,t:15|
CC(C)Oc1nc(nc2c1CC[C@@H]1[C@@H](C)C(=O)C(=C[C@@]21C)C#N)-c1ccnc2ccccc12 |r,c:18|
CC(C)c1nc(nc2c1CC[C@@H]1[C@@H](C)C(=O)C(=C[C@@]21C)C#N)-c1ccnc2ccccc12 |r,c:17|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc(C)c1)-c1ccccc1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)C1CCN(CC1)C(=O)OC(C)(C)C)-c1ccccc1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)C1CCNCC1)-c1ccccc1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)C1CCN(CC1)C(C)=O)-c1ccccc1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)C1=CCCN(C1)C(=O)OC(C)(C)C)-c1ccccc1 |r,t:15,22|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)C1=CCCNC1)-c1ccccc1 |r,t:15,22|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)C1=CCCN(C1)C(C)=O)-c1ccccc1 |r,t:15,22|
[H][C@]12CCc3c(nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2C)-c1ccnc(C)c1)-c1ccc(F)cc1 |r,t:14|
[H][C@]12CCc3c(nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2C)-c1ccnc(C)c1)-c1ccccc1F |r,t:14|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1ccc(F)cc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc(c1)C1CC1)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc(c1)C(F)(F)F)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)CC(C#N)=C1O)-c1ccncc1C)-c1ccccc1F |r,c:18|
[H][C@]12CCc3c(nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2C)-c1ccncc1C)-c1ccccc1F |r,t:14|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccncc1F)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cncc(C)c1)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cnc2ccccc2c1)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccc2ncccc2c1)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc(NC(C)=O)c1)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cccc2cccnc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cc(C)nc2c(F)cccc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc(c1)N1CCOCC1)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc(c1)-c1ccccc1)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cncc2ccccc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cnn2ccccc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2c(C)cccc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cc(C)nc2ccccc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1sc(C)nc1C)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1noc(C)n1)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cn(C)c2ncccc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccc(C)cc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ncnc2ccccc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1nccc2ccccc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2cc(F)ccc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2c(F)cccc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cc(C)ncn1)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnnc1)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2CCCc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccccc1F)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc(CO)c1)-c1ccccc1F |r,t:15|
[H][C@]12CCc3c(nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2C)-c1ccnc(CF)c1)-c1ccccc1F |r,t:14|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cccc2ncccc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cc(C)nc2ccc(F)cc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cccc2cnccc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1c(C)noc1C)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccc(C)nc1)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccc(F)cc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2c(F)cc(F)cc12)-c1ccccc1F |r,t:15|
[H][C@]12CCc3c(nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2C)N1CCN(C)CC1)-c1ccccc1F |r,t:14|
[H][C@]12CCc3c(nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2C)N1CCOCC1)-c1ccccc1F |r,t:14|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)C1CC1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(OC4CCC4)nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12 |r,t:21|
C[C@@H]1[C@H]2CCc3c(OCC4CCC4)nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12 |r,t:22|
C[C@@H]1[C@H]2CCc3c(OC4CCCCC4)nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12 |r,t:23|
C[C@@H]1[C@H]2CCc3c(OC4CCCC4)nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12 |r,t:22|
C[C@@H]1[C@H]2CCc3c(NS(C)(=O)=O)nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12 |r,t:20|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)N(C)C |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1c(C)noc1C |r,wU:1.0,wD:2.2,11.13,t:15,(-2.52,-5.78,;-2.52,-4.24,;-1.18,-3.47,;.15,-4.24,;1.48,-3.47,;1.48,-1.93,;2.82,-1.16,;2.82,.38,;1.48,1.15,;.15,.38,;.15,-1.16,;-1.18,-1.93,;-1.18,-.39,;-2.52,-1.16,;-3.85,-1.93,;-5.19,-1.16,;-6.52,-.39,;-3.85,-3.47,;-5.19,-4.24,;1.48,2.69,;.15,3.46,;.15,5,;1.48,5.78,;2.82,5,;4.15,5.77,;5.48,5,;5.48,3.46,;4.15,2.69,;2.82,3.46,;4.15,-1.93,;4.15,-3.47,;2.82,-4.24,;5.61,-3.94,;6.52,-2.7,;5.61,-1.45,;6.38,-.12,)|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1ccc(cc1)C(=O)N(C)Cc1ccccc1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1ccco1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1cc2ccccc2o1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1ccc(C)o1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1nc(C)no1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1noc(C)n1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1nccs1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cc(C)nc2ccccc12)-c1cccc(F)c1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cc(C)nc2ccccc12)-c1ccc(F)cc1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(OC4CCC4)nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cc(C)nc2ccccc12 |r,t:21|
C[C@@H]1[C@H]2CCc3c(OC4CCCC4)nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cc(C)nc2ccccc12 |r,t:22|
C[C@@H]1[C@H]2CCc3c(OC4CCC4)nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ncnc2ccccc12 |r,t:21|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ncnc2ccccc12)-c1cccc(F)c1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ncnc2ccccc12)-c1ccc(F)cc1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cc(CF)nc2ccccc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cc(C=O)nc2ccccc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cc(COC(C)=O)nc2ccccc12)-c1ccccc1F |r,t:15|
CC1(C)[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1ccccc1F |r,t:16|
Cc1cc(-c2nc(c3CC[C@@H]4C(C)(C)C(=O)C(=C[C@@]4(C)c3n2)C#N)-c2ccccc2F)c2ccccc2n1 |r,c:16|
C[C@@H]1[C@H]2CCc3c(OC4CCCC4)nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cc(CF)nc2ccccc12 |r,t:22|
C[C@@H]1[C@H]2CCc3c(OC4CCCC4)nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2c(F)cccc12 |r,t:22|
CC1(C)[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cc(CF)nc2ccccc12)-c1ccccc1F |r,t:16|
CC(C)c1cc(-c2nc(c3CC[C@@H]4[C@@H](C)C(=O)C(=C[C@@]4(C)c3n2)C#N)-c2ccccc2F)c2ccccc2n1 |r,c:17|
CCC[C@]1(C)[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1ccccc1F |r,t:18|
CC1(C)[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc(c1)C1CC1)-c1ccccc1F |r,t:16|
CC[C@]1(C)[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1ccccc1F |r,t:17|
CC1(C)[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2c(F)cccc12)-c1ccccc1F |r,t:16|
CC1=C2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2c(F)cccc12)-c1ccccc1F |r,c:1,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)[C@@H]2O[C@]2(C#N)C1=O)-c1ccnc2cc(F)ccc12)-c1ccccc1F |r|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)[C@@H]2O[C@]2(C#N)C1=O)-c1ccnc(c1)C1CC1)-c1ccccc1F |r|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)[C@@H]2O[C@]2(C#N)C1=O)-c1ccnc2ccccc12)-c1ccccc1F |r|
CC1(C)[C@H]2CCc3c(nc(nc3[C@]2(C)[C@@H]2O[C@]2(C#N)C1=O)-c1ccnc2ccccc12)-c1ccccc1F |r|
COc1nc(nc2c1CC[C@@H]1[C@@H](C)C(=O)C=C[C@@]21C)-c1ccncc1 |r,c:16|
COC(=O)[C@]1(C)[C@H]2CCc3c(OC)nc(nc3[C@]2(C)C=CC1=O)-c1ccncc1 |r,c:21|
C[C@@]1(CCCO)[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc(c1)C1CC1)-c1ccccc1F |r,t:19|
CCC[C@]1(C)[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc(c1)C1CC1)-c1ccccc1F |r,t:18|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)N1CCCC1 |r,t:15|
[H][C@]12CCc3c(nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2C)N1CCN(CC1)C(C)=O)-c1ccccc1F |r,t:14|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccc(nc1)C1CC1)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccc(nc1)-c1ccccc1)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccc(CCS(C)(=O)=O)nc1)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc(CS(C)(=O)=O)c1)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc(CCS(C)(=O)=O)c1)-c1ccccc1F |r,t:15|
[H][C@]12CCc3c(nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2CC=C)-c1ccnc(c1)C1CC1)-c1ccccc1F |r,t:14|
[H][C@]12CCc3c(nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2CCC)-c1ccnc(c1)C1CC1)-c1ccccc1F |r,t:14|
[H][C@]12CCc3c(nc(nc3[C@@]1(C=C(C#N)C(=O)[C@@H]2C)c1ccccc1)-c1ccnc(c1)C1CC1)-c1ccccc1F |r,t:13|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@@]2(C=C(C#N)C1=O)c1ccccc1)-c1ccnc2ccccc12)-c1ccccc1F |r,t:14|
CC1(C)[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cccc2ncccc12)-c1ccccc1F |r,t:16|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc(CCC(O)=O)c1)-c1ccccc1F |r,t:15|
CCOC(=O)CCc1cc(ccn1)-c1nc(c2CC[C@@H]3[C@@H](C)C(=O)C(=C[C@@]3(C)c2n1)C#N)-c1ccccc1F |r,c:25|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc(CCC(=O)N(C)C)c1)-c1ccccc1F |r,t:15|
CCS(=O)(=O)CCc1cc(ccn1)-c1nc(c2CC[C@@H]3[C@@H](C)C(=O)C(=C[C@@]3(C)c2n1)C#N)-c1ccccc1F |r,c:25|
CCS(=O)(=O)Cc1cc(ccn1)-c1nc(c2CC[C@@H]3[C@@H](C)C(=O)C(=C[C@@]3(C)c2n1)C#N)-c1ccccc1F |r,c:24|
CCC[C@@]12C=C(C#N)C(=O)C[C@H]1CCc1c(nc(nc21)-c1ccnc(CF)c1)-c1ccccc1F |r,t:4|
CCC[C@@]12C=C(C#N)C(=O)C[C@H]1CCc1c(nc(nc21)-c1ccnc2ccccc12)-c1ccccc1F |r,t:4|
C[C@@]1(CC2CC2)[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1ccccc1F |r,t:20|
CCC[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1ccccc1F |r,t:17|
CCC[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cccc2ncccc12)-c1ccccc1F |r,t:17|
CC(C)c1cccc(c1)-c1nc(nc2c1CC[C@@H]1[C@@H](C)C(=O)C(=C[C@@]21C)C#N)-c1ccnc2ccccc12 |r,c:24|
CC(C)c1ccc(cc1)-c1nc(nc2c1CC[C@@H]1[C@@H](C)C(=O)C(=C[C@@]21C)C#N)-c1ccnc2ccccc12 |r,c:24|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1cccc(c1)-c1ccccc1 |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1ccc(cc1)-c1ccccc1 |r,t:15|
CC(C)CC[C@@]12C=C(C#N)C(=O)C[C@H]1CCc1c(nc(nc21)-c1ccnc2ccccc12)-c1ccccc1F |r,t:6|
CC(C)CC[C@@]12C=C(C#N)C(=O)C[C@H]1CCc1c(nc(nc21)-c1ccnc(CF)c1)-c1ccccc1F |r,t:6|
CC(=C)C[C@]1(C)[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1ccccc1F |r,t:19|
CCC[C@@]12C=C(C#N)C(=O)C[C@H]1CCc1c(nc(nc21)-c1ccnc(c1)C1CC1)-c1ccccc1F |r,t:4|
CCC[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(CCC)C=C(C#N)C1=O)-c1ccnc(c1)C1CC1)-c1ccccc1F |r,t:19|
[H][C@]12CCc3c(nc(nc3[C@]1(CCC)C=C(C#N)C(=O)[C@@H]2C)-c1ccnc(c1)C1CC1)-c1ccccc1F |r,t:16|
C[C@@H]1[C@H]2Cc3c(nc(nc3-c3ccccc3F)-c3ccnc4ccccc34)[C@]2(C)C=C(C#N)C1=O |r,t:34|
[H][C@]12Cc3c(nc(nc3-c3ccccc3F)-c3ccnc(CF)c3)[C@]1(C)C=C(C#N)C(=O)[C@@H]2C |r,t:30|
C[C@@H]1[C@H]2Cc3c(nc(nc3-c3ccccc3F)-c3cc(C)nc4c(F)cccc34)[C@]2(C)C=C(C#N)C1=O |r,t:36|
C[C@@H]1[C@H]2Cc3c(nc(nc3-c3ccccc3F)-c3cccc4ncccc34)[C@]2(C)C=C(C#N)C1=O |r,t:34|
[H][C@]12Cc3c(nc(nc3-c3ccccc3F)-c3ccnc(c3)C3CC3)[C@]1(C)C=C(C#N)C(=O)[C@@H]2C |r,t:32|
C[C@H]1[C@@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc2ccccc12)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc(CCC(N)=O)c1)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc(CCNC(C)=O)c1)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccncc1-c1ccccc1)-c1ccccc1F |r,t:15|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccncc1C1CC1)-c1ccccc1F |r,t:15|
CC[C@]1(C)[C@H]2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccnc(c1)C1CC1)-c1ccccc1F |r,t:17|
[H][C@]12CCCc3c(nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2C)-c1ccnc(C)c1)-c1ccccc1 |r,t:15|
C[C@@H]1[C@H]2CCCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1cccc2ncccc12)-c1ccccc1 |r,t:16|
[H][C@]12CCc3c(nc(nc3[C@]1(C)C=C(C(N)=O)C(=O)[C@@H]2C)-c1ccnc(C)c1)-c1ccc(F)cc1 |r,t:14|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)CC(C(N)=O)C1=O)-c1ccnc(C)c1)-c1ccc(F)cc1 |r|
C[C@@H]1[C@H]2CCc3c(nc(nc3[C@]2(C)CC(C#N)C1=O)-c1ccnc2ccccc12)-c1ccccc1F |r|
[H][C@]12CCc3c(nc(nc3[C@]1(C)CC(C#N)C(=O)[C@@H]2C)-c1ccnc(C)c1)-c1ccc(F)cc1 |r|
CCc1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(C#N)n1-c1ccc(CC(C)C(F)(F)F)cc1OC |r,wU:9.8,wD:9.9,13.16,(5.07,-1.9,;3.54,-2.06,;2.63,-.81,;3.11,.65,;1.86,1.56,;1.86,3.1,;3.19,3.87,;.53,3.87,;.53,5.41,;1.86,6.18,;1.75,4.64,;1.14,7.54,;1.95,8.84,;3.49,8.79,;4.22,7.43,;3.4,6.12,;4.31,10.09,;5.08,11.43,;3.59,11.45,;5.85,10.04,;.62,.65,;-.85,1.13,;-2.31,1.6,;1.09,-.81,;.19,-2.06,;-1.35,-1.9,;-2.25,-3.14,;-1.62,-4.55,;-2.53,-5.8,;-4.06,-5.64,;-4.69,-4.23,;-4.97,-6.88,;-5.87,-8.13,;-3.72,-7.79,;-6.21,-5.98,;-.09,-4.71,;.81,-3.47,;2.34,-3.63,;2.97,-5.03,)|
CCc1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)n1-c1ncc(CC(C)(C)C(F)(F)F)cc1OC(F)F |r,wU:9.8,wD:12.15,(-1.02,-2.56,;-1.65,-1.15,;-.74,.09,;-1.22,1.56,;.03,2.46,;.03,4,;1.36,4.77,;-1.3,4.77,;-1.3,6.31,;-2.64,7.08,;-3.97,6.31,;-5.3,7.08,;-5.3,8.62,;-3.97,9.39,;-2.64,8.62,;-6.64,9.39,;-7.97,10.16,;-8,8.67,;-6.58,10.93,;1.28,1.56,;2.74,2.03,;.8,.09,;1.7,-1.15,;1.08,-2.56,;1.98,-3.81,;3.52,-3.65,;4.42,-4.89,;3.79,-6.3,;5.2,-6.92,;2.39,-5.67,;3.17,-7.7,;2.54,-9.11,;4.57,-8.33,;1.76,-7.08,;4.14,-2.24,;3.24,-.99,;3.86,.41,;5.39,.57,;6.02,1.98,;6.3,-.67,)|
CCc1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(Cl)n1-c1ccc(N[C@H](C)C(F)(F)F)cc1OC |r,wU:9.8,27.29,wD:12.15,(4.42,-1.69,;2.89,-1.85,;1.98,-.6,;2.46,.86,;1.21,1.77,;1.21,3.31,;-.12,4.08,;2.55,4.08,;2.55,5.62,;3.88,6.39,;3.88,7.93,;5.21,8.7,;6.55,7.93,;6.55,6.39,;5.21,5.62,;7.88,8.7,;8.65,10.03,;7.16,10.06,;9.42,8.64,;-.03,.86,;-1.5,1.34,;.44,-.6,;-.46,-1.85,;-1.99,-1.69,;-2.9,-2.93,;-2.27,-4.34,;-3.18,-5.59,;-4.71,-5.42,;-5.34,-4.02,;-5.62,-6.67,;-6.52,-7.92,;-6.86,-5.76,;-4.37,-7.58,;-.74,-4.5,;.16,-3.25,;1.69,-3.42,;2.32,-4.82,)|
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CCc1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)n1-c1ccc(CC(C)C)cc1OC |r,wU:9.8,wD:9.9,13.16,(-.15,-3.26,;.94,-2.17,;.46,-.71,;-1,-.23,;-1,1.31,;-2.34,2.08,;-2.34,3.62,;-3.67,1.31,;-5,2.08,;-6.34,1.31,;-6.34,2.85,;-6.34,-.23,;-7.67,-1,;-9.05,-.26,;-9.01,1.31,;-7.67,2.08,;-10.39,-1.03,;-11.63,-1.93,;-10.28,-2.57,;-11.77,-.35,;.46,1.78,;.94,3.25,;1.37,.54,;3.41,.54,;4.18,1.87,;5.72,1.87,;6.49,.54,;8.03,.54,;8.8,1.87,;8.03,3.21,;10.34,1.87,;5.72,-.8,;4.15,-.84,;3.38,-2.18,;4.15,-3.51,)|
CCc1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(C#N)n1-c1ccc(CCC(F)(F)F)cc1F |r,wU:9.8,wD:12.15,(-1.07,-4,;.02,-2.91,;-.45,-1.45,;-1.92,-.97,;-1.92,.57,;-3.25,1.34,;-3.25,2.88,;-4.59,.57,;-5.92,1.34,;-7.25,.57,;-7.25,-.97,;-8.59,-1.74,;-9.97,-1,;-9.92,.57,;-8.59,1.34,;-11.3,-1.77,;-12.64,-2.54,;-11.36,-3.31,;-12.61,-.95,;-.45,1.05,;.02,2.51,;.42,4,;.45,-.2,;2.49,-.2,;3.26,1.13,;4.8,1.13,;5.57,-.2,;7.11,-.2,;7.88,-1.53,;9.42,-1.53,;10.96,-1.53,;9.42,-3.07,;9.42,.01,;4.8,-1.53,;3.26,-1.53,;2.49,-2.87,)|
CCc1nc(C(=O)NC[C@H]2CC[C@@H](CC2)S(C)(=O)=O)c(C(N)=O)n1-c1ccc(CCC(F)(F)F)cc1F |r,wU:9.8,wD:12.15,(-1.07,-3.83,;.02,-2.74,;-.45,-1.27,;-1.92,-.8,;-1.92,.74,;-3.25,1.51,;-3.25,3.05,;-4.59,.74,;-5.92,1.51,;-7.25,.74,;-7.25,-.8,;-8.59,-1.57,;-9.97,-.83,;-9.92,.74,;-8.59,1.51,;-11.3,-1.6,;-12.55,-2.5,;-11.19,-3.13,;-12.69,-.92,;-.45,1.22,;.02,2.68,;-1.01,3.83,;1.53,3,;.45,-.03,;2.49,-.03,;3.26,1.31,;4.8,1.31,;5.57,-.03,;7.11,-.03,;7.88,-1.36,;9.42,-1.36,;10.96,-1.36,;9.42,-2.9,;9.42,.18,;4.8,-1.36,;3.26,-1.36,;2.49,-2.7,)|
CCc1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(C#N)n1-c1ccc(CCC(F)(F)F)cc1F |r,wU:9.8,wD:9.9,13.16,(-1.07,-4.14,;.02,-3.05,;-.45,-1.58,;-1.92,-1.11,;-1.92,.43,;-3.25,1.2,;-3.25,2.74,;-4.59,.43,;-5.92,1.2,;-7.25,.43,;-7.25,1.97,;-7.25,-1.11,;-8.59,-1.88,;-9.97,-1.14,;-9.92,.43,;-8.59,1.2,;-11.3,-1.91,;-12.55,-2.81,;-11.19,-3.44,;-12.69,-1.23,;-.45,.91,;.02,2.37,;.5,4.14,;.45,-.34,;2.49,-.34,;3.26,.99,;4.8,.99,;5.57,-.34,;7.11,-.34,;7.88,-1.67,;9.42,-1.67,;10.96,-1.67,;9.42,-3.21,;9.42,-.13,;4.8,-1.67,;3.26,-1.67,;2.49,-3.01,)|
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CCc1nc(C(=O)NC[C@@]2(O)CC[C@@H](CC2)S(C)(=O)=O)c(Cl)n1-c1ccc(CCCC(F)(F)F)cc1F |r,wU:9.8,wD:9.9,13.16,(-1.35,-4.04,;-.26,-2.95,;-.73,-1.49,;-2.2,-1.01,;-2.2,.53,;-3.53,1.3,;-3.53,2.84,;-4.87,.53,;-6.2,1.3,;-7.53,.53,;-7.53,2.07,;-7.53,-1.01,;-8.87,-1.78,;-10.25,-1.04,;-10.2,.53,;-8.87,1.3,;-11.58,-1.81,;-12.61,-2.96,;-11.16,-3.29,;-13.08,-1.44,;-.73,1,;-.26,2.47,;.17,-.24,;2.21,-.24,;2.98,1.09,;4.52,1.09,;5.29,-.24,;6.83,-.24,;7.6,1.09,;9.14,1.09,;9.91,-.24,;10.68,-1.58,;8.58,-1.01,;11.25,.53,;4.52,-1.58,;2.98,-1.58,;2.21,-2.91,)|
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CCN(C[C@H]1CC[C@@H](CC1)C(F)(F)F)c1ncnc(NC[C@@H]2CCN(CC(N)=O)C[C@H]2O)c1F |r,wU:21.21,4.3,wD:30.32,7.10,(4.53,-5.75,;3.2,-4.98,;3.2,-3.44,;4.54,-2.68,;4.57,-1.14,;3.23,-.37,;3.23,1.17,;4.57,1.99,;5.9,1.17,;5.9,-.37,;4.57,3.53,;4.57,5.07,;3.03,3.53,;6.11,3.53,;1.86,-2.67,;1.86,-1.13,;.53,-.36,;-.8,-1.13,;-.8,-2.67,;-2.11,-3.48,;-3.44,-2.7,;-3.44,-1.16,;-2.1,-.39,;-2.1,1.15,;-3.44,1.92,;-3.44,3.46,;-4.78,4.21,;-6.11,3.42,;-4.8,5.75,;-4.77,1.15,;-4.77,-.39,;-6.1,-1.16,;.53,-3.44,;.56,-4.98,)|
CCN(C[C@H]1CC[C@H](CC1)C(F)(F)F)c1ncnc(NC[C@@H]2CCN(CC(N)=O)C[C@H]2O)c1F |r,wU:21.21,4.3,7.10,wD:30.32,(4.53,-5.75,;3.2,-4.98,;3.2,-3.44,;4.54,-2.68,;4.57,-1.14,;3.23,-.37,;3.23,1.17,;4.57,1.99,;5.9,1.17,;5.9,-.37,;4.57,3.53,;4.57,5.07,;3.03,3.53,;6.11,3.53,;1.86,-2.67,;1.86,-1.13,;.53,-.36,;-.8,-1.13,;-.8,-2.67,;-2.11,-3.48,;-3.44,-2.7,;-3.44,-1.16,;-2.1,-.39,;-2.1,1.15,;-3.44,1.92,;-3.44,3.46,;-4.78,4.21,;-6.11,3.42,;-4.8,5.75,;-4.77,1.15,;-4.77,-.39,;-6.1,-1.16,;.53,-3.44,;.56,-4.98,)|
NC(=O)CN1CC[C@@H](CNc2ncnc(N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)C3CC3)c2F)[C@H](O)C1 |r,wU:7.7,17.16,wD:32.35,20.23,(-6.11,3.7,;-4.78,4.49,;-4.8,6.03,;-3.44,3.74,;-3.44,2.2,;-2.1,1.43,;-2.1,-.11,;-3.44,-.88,;-3.44,-2.42,;-2.11,-3.2,;-.8,-2.39,;-.8,-.85,;.53,-.08,;1.86,-.85,;1.86,-2.39,;3.2,-3.16,;4.54,-2.4,;4.57,-.86,;3.23,-.09,;3.23,1.45,;4.57,2.27,;5.9,1.45,;5.9,-.09,;4.57,3.81,;4.57,5.35,;3.03,3.81,;6.11,3.81,;3.2,-4.7,;2.43,-6.03,;3.97,-6.03,;.53,-3.16,;.56,-4.7,;-4.77,-.11,;-6.1,-.88,;-4.77,1.43,)|
NC(=O)CN1CC[C@@H](CNc2ncnc(N(C[C@H]3CC[C@H](CC3)C(F)(F)F)C3CC3)c2F)[C@H](O)C1 |r,wU:7.7,17.16,20.23,wD:32.35,(-6.11,3.7,;-4.78,4.49,;-4.8,6.03,;-3.44,3.74,;-3.44,2.2,;-2.1,1.43,;-2.1,-.11,;-3.44,-.88,;-3.44,-2.42,;-2.11,-3.2,;-.8,-2.39,;-.8,-.85,;.53,-.08,;1.86,-.85,;1.86,-2.39,;3.2,-3.16,;4.54,-2.4,;4.57,-.86,;3.23,-.09,;3.23,1.45,;4.57,2.27,;5.9,1.45,;5.9,-.09,;4.57,3.81,;4.57,5.35,;3.03,3.81,;6.11,3.81,;3.2,-4.7,;2.43,-6.03,;3.97,-6.03,;.53,-3.16,;.56,-4.7,;-4.77,-.11,;-6.1,-.88,;-4.77,1.43,)|
NC(=O)CN1CC[C@@H](CNc2ncnc(N(C[C@H]3CC[C@@H](CC3)C(F)(F)F)C3CCC3)c2F)[C@H](O)C1 |r,wU:7.7,17.16,wD:33.36,20.23,(-6.11,4.13,;-4.78,4.91,;-4.8,6.45,;-3.44,4.16,;-3.44,2.62,;-2.1,1.85,;-2.1,.31,;-3.44,-.46,;-3.44,-2,;-2.11,-2.78,;-.8,-1.97,;-.8,-.43,;.53,.34,;1.86,-.43,;1.86,-1.97,;3.2,-2.74,;4.54,-1.98,;4.57,-.44,;3.23,.33,;3.23,1.87,;4.57,2.69,;5.9,1.87,;5.9,.33,;4.57,4.23,;4.57,5.77,;3.03,4.23,;6.11,4.23,;3.2,-4.28,;2.11,-5.37,;3.2,-6.45,;4.29,-5.37,;.53,-2.74,;.56,-4.28,;-4.77,.31,;-6.1,-.46,;-4.77,1.85,)|
CCN(CC1CC[C@]2(COC2)CC1)c1ncnc(NC[C@@H]2CCN(CC(N)=O)C[C@H]2O)c1F |r|
CCN(C[C@@]1(F)CC[C@@H](CC1)C(F)(F)F)c1ncnc(NC[C@@H]2CCN(CC(N)=O)C[C@H]2O)c1F |r,wU:22.22,4.5,wD:31.33,4.4,8.11,(4.53,-5.75,;3.2,-4.98,;3.2,-3.44,;4.54,-2.68,;4.57,-1.14,;4.57,.4,;3.23,-.37,;3.23,1.17,;4.57,1.99,;5.9,1.17,;5.9,-.37,;4.57,3.53,;4.57,5.07,;6.11,3.53,;3.03,3.53,;1.86,-2.67,;1.86,-1.13,;.53,-.36,;-.8,-1.13,;-.8,-2.67,;-2.11,-3.48,;-3.44,-2.7,;-3.44,-1.16,;-2.1,-.39,;-2.1,1.15,;-3.44,1.92,;-3.44,3.46,;-4.78,4.21,;-6.11,3.42,;-4.8,5.75,;-4.77,1.15,;-4.77,-.39,;-6.1,-1.16,;.53,-3.44,;.56,-4.98,)|
CCN(C[C@]1(F)CC[C@@H](CC1)C(F)(F)F)c1ncnc(NC[C@@H]2CCN(CC(N)=O)C[C@H]2O)c1F |r,wU:22.22,4.10,8.11,wD:31.33,4.4,(4.53,-5.75,;3.2,-4.98,;3.2,-3.44,;4.54,-2.68,;4.57,-1.14,;4.57,.4,;5.9,-.37,;5.9,1.17,;4.57,1.99,;3.23,1.17,;3.23,-.37,;4.57,3.53,;4.57,5.07,;6.11,3.53,;3.03,3.53,;1.86,-2.67,;1.86,-1.13,;.53,-.36,;-.8,-1.13,;-.8,-2.67,;-2.11,-3.48,;-3.44,-2.7,;-3.44,-1.16,;-2.1,-.39,;-2.1,1.15,;-3.44,1.92,;-3.44,3.46,;-4.78,4.21,;-6.11,3.42,;-4.8,5.75,;-4.77,1.15,;-4.77,-.39,;-6.1,-1.16,;.53,-3.44,;.56,-4.98,)|
NC(=O)CN1CCC(CNc2ncnc(N3CCOC[C@@H]3C3CC[C@@H](CC3)C(F)(F)F)c2F)CC1 |r,wU:20.21,24.28,(-6.11,3.42,;-4.78,4.21,;-4.8,5.75,;-3.44,3.46,;-3.44,1.92,;-4.77,1.15,;-4.77,-.39,;-3.44,-1.16,;-3.44,-2.7,;-2.11,-3.48,;-.8,-2.67,;-.8,-1.13,;.53,-.36,;1.86,-1.13,;1.86,-2.67,;3.2,-3.44,;3.2,-4.98,;4.53,-5.75,;5.87,-4.98,;5.87,-3.44,;4.54,-2.68,;4.57,-1.14,;5.9,-.37,;5.9,1.17,;4.57,1.99,;3.23,1.17,;3.23,-.37,;4.57,3.53,;4.57,5.07,;6.11,3.53,;3.03,3.53,;.53,-3.44,;.56,-4.98,;-2.1,-.39,;-2.1,1.15,)|
CCN(C[C@H]1CC[C@@H](CC1)C(F)(F)F)c1ncnc(NC[C@@]2(O)CCN(CC(N)=O)C[C@@H]2O)c1F |r,wU:21.22,31.33,4.3,wD:21.21,7.10,(4.57,-5.77,;3.23,-5,;3.23,-3.46,;4.57,-2.69,;4.57,-1.15,;3.23,-.38,;3.23,1.16,;4.6,2.03,;5.9,1.16,;5.9,-.38,;4.62,3.57,;4.64,5.11,;3.08,3.59,;6.16,3.55,;1.9,-2.69,;1.9,-1.16,;.56,-.39,;-.77,-1.16,;-.77,-2.69,;-2.1,-3.46,;-3.44,-2.69,;-3.44,-1.15,;-4.77,-1.92,;-2.1,-.38,;-2.1,1.15,;-3.44,1.92,;-3.44,3.46,;-2.1,4.23,;-.77,3.46,;-2.1,5.77,;-4.77,1.15,;-4.77,-.38,;-6.1,-1.15,;.56,-3.46,;.56,-5,)|
CCN(C[C@H]1CC[C@H](CC1)C(F)(F)F)c1ncnc(NC[C@@]2(O)CCN(CC(N)=O)C[C@@H]2O)c1F |r,wU:21.22,31.33,4.3,7.10,wD:21.21,(4.57,-5.77,;3.23,-5,;3.23,-3.46,;4.57,-2.69,;4.57,-1.15,;3.23,-.38,;3.23,1.16,;4.6,2.03,;5.9,1.16,;5.9,-.38,;4.62,3.57,;4.64,5.11,;3.08,3.59,;6.16,3.55,;1.9,-2.69,;1.9,-1.16,;.56,-.39,;-.77,-1.16,;-.77,-2.69,;-2.1,-3.46,;-3.44,-2.69,;-3.44,-1.15,;-4.77,-1.92,;-2.1,-.38,;-2.1,1.15,;-3.44,1.92,;-3.44,3.46,;-2.1,4.23,;-.77,3.46,;-2.1,5.77,;-4.77,1.15,;-4.77,-.38,;-6.1,-1.15,;.56,-3.46,;.56,-5,)|
CCN(C[C@H]1CC[C@@H](CC1)C(F)(F)F)c1ncnc2n(CC3(O)CCN(CC(N)=O)C[C@H]3O)ccc12 |r,wU:4.3,wD:31.33,7.10,(4.76,-5.39,;3.43,-4.62,;3.43,-3.08,;4.76,-2.31,;4.79,-.77,;3.45,0,;3.45,1.54,;4.75,2.42,;6.12,1.54,;6.12,0,;4.73,3.96,;4.71,5.5,;3.19,3.94,;6.27,3.98,;2.09,-2.31,;2.09,-.77,;.76,0,;-.57,-.77,;-.57,-2.31,;-1.72,-3.34,;-3.22,-3,;-3.99,-1.67,;-4.76,-.34,;-3.22,-.34,;-3.99,1,;-5.53,1,;-6.26,2.35,;-5.49,3.69,;-3.95,3.69,;-6.26,5.02,;-6.3,-.34,;-5.53,-1.67,;-6.26,-3.03,;-1.09,-4.75,;.44,-4.59,;.76,-3.08,)|
CCN(C[C@H]1CC[C@H](CC1)C(F)(F)F)c1ncnc2n(CC3(O)CCN(CC(N)=O)C[C@H]3O)ccc12 |r,wU:4.3,7.10,wD:31.33,(4.76,-5.39,;3.43,-4.62,;3.43,-3.08,;4.76,-2.31,;4.79,-.77,;3.45,0,;3.45,1.54,;4.75,2.42,;6.12,1.54,;6.12,0,;4.73,3.96,;4.71,5.5,;3.19,3.94,;6.27,3.98,;2.09,-2.31,;2.09,-.77,;.76,0,;-.57,-.77,;-.57,-2.31,;-1.72,-3.34,;-3.22,-3,;-3.99,-1.67,;-4.76,-.34,;-3.22,-.34,;-3.99,1,;-5.53,1,;-6.26,2.35,;-5.49,3.69,;-3.95,3.69,;-6.26,5.02,;-6.3,-.34,;-5.53,-1.67,;-6.26,-3.03,;-1.09,-4.75,;.44,-4.59,;.76,-3.08,)|
Cc1cc(CN2CCN(Cc3ccncc3)[C@@H](CC([O-])=O)C2)ccc1-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
Cc1nc(-c2ccc(F)cc2-c2ccncc2C)c2c(n1)[C@]1(C)C=C(C#N)C(=O)[C@H](C)[C@H]1CC2
CCC[C@H]1C(=O)C(C#N)=C[C@@]2(C)c3nc(-c4ccncc4C4CC4)nc(-c4ccccc4F)c3CC[C@H]12
CS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2ccc(cc2F)C(O)(C(F)(F)F)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2ccc(cc2F)C(O)(C(F)(F)F)C(F)(F)F)cc1
OC(c1ccc(c(F)c1)-c1ccc(NC(=O)Cc2ccc(cc2)[N+]([O-])=O)cc1)(C(F)(F)F)C(F)(F)F
OC(c1ccc(c(F)c1)-c1ccc(NC(=O)Cc2ccccc2[N+]([O-])=O)cc1)(C(F)(F)F)C(F)(F)F
Nc1ccc(CC(=O)Nc2ccc(cc2)-c2ccc(cc2F)C(O)(C(F)(F)F)C(F)(F)F)cc1
Nc1cccc(CC(=O)Nc2ccc(-c3ccc(C(O)(C(F)(F)F)C(F)(F)F)cc3F)cc2)c1
CCCCC(=O)Nc1ccc(cc1)-c1ccc(cc1F)C(O)(C(F)(F)F)C(F)(F)F
c1ccc(cc1)S(=O)(=O)[N@@](CC(F)(F)F)c2ccc(cc2)C(C(F)(F)F)(C(F)(F)F)O
C[C@H](N)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C=O
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2ccccc12
Cc1c(cc(cc1NC(=O)c2cnc(nc2)C)Cl)CN3CCN([C@H](C3)C)C(=O)C4CCCC4
Cc1ccc(c(c1)C)NC(=O)[C@H]2CN(C[C@@H]2c3nnc(n3C4CC4)C5CC(C5)CC(C)C)C(=O)C
COc1ccc2[C@H](N(CCc2n1)C(=O)[C@@H]1C[C@@H](C1)C(O)=O)C(=O)Nc1cc2CCC(C)(C)c2c(F)c1 |r,wU:14.15,16.20,wD:6.23,(-.09,7.06,;1.24,6.29,;1.24,4.75,;-.09,3.98,;-.08,2.44,;1.24,1.67,;1.24,.13,;2.58,-.64,;3.91,.13,;3.91,1.67,;2.58,2.44,;2.58,3.99,;2.58,-2.18,;1.24,-2.95,;3.91,-2.95,;3.91,-4.49,;5.48,-4.49,;5.48,-2.95,;6.57,-5.57,;8.05,-5.18,;6.17,-7.06,;-.09,-.64,;-.09,-2.18,;-1.42,.13,;-2.76,-.64,;-2.76,-2.18,;-4.09,-2.94,;-4.41,-4.45,;-5.94,-4.61,;-6.57,-3.2,;-7.66,-2.11,;-8.05,-3.6,;-5.42,-2.17,;-5.42,-.64,;-6.76,.13,;-4.1,.14,)|
CCS(=O)(=O)c1ccc(CC(=O)Nc2cnc3[C@H](C(C)C)N(C[C@H]4CC[C@@H](CC4)C(F)(F)F)Cc3c2)nc1 |r,wU:17.17,23.22,wD:26.29,(11.49,2.96,;10.16,2.19,;8.83,2.96,;8.06,4.29,;9.6,4.29,;7.49,2.19,;7.5,.66,;6.17,-.12,;4.83,.65,;3.49,-.12,;2.16,.65,;2.16,2.19,;.83,-.12,;-.51,.65,;-.51,2.2,;-1.84,2.96,;-3.17,2.19,;-4.63,2.67,;-5.03,4.16,;-6.52,4.56,;-3.94,5.25,;-5.54,1.42,;-7.08,1.42,;-7.85,.09,;-7.08,-1.24,;-7.85,-2.58,;-9.39,-2.58,;-10.16,-1.24,;-9.39,.09,;-10.16,-3.91,;-9.39,-5.25,;-11.49,-3.14,;-11.49,-4.68,;-4.63,.18,;-3.17,.65,;-1.84,-.12,;4.83,2.19,;6.16,2.96,)|
Cc1c(cn2ccnc2c1CN3CCN([C@H](C3)C)C(=O)C4CCCC4)NC(=O)c5cnc(nc5)C
Cc1noc(C)c1C(O)c1cc2cc(CC(=O)N[C@@H](c3ccccc3)c3ccc(C)cc3C)ccc2o1 |r|
Cc1noc(C)c1COc1ccc(CC(=O)NC(c2ccccc2)c2ccc(C)cc2C)cc1
C[C@@H]1CC[C@@]2(CC[C@@]3(C(=CC[C@H]4[C@]3(CC[C@@H]5[C@@]4(CC[C@@H](C5(C)C)O)C)C)[C@@H]2[C@H]1C)C)C(=O)O
c1ccc(cc1)S(=O)(=O)[N@@](CC(F)(F)F)c2ccc(cc2)C(C(F)(F)F)(C(F)(F)F)O
c1cc(ccc1CN2CCN(CC2)Cc3ccncc3)c4ccc(cc4F)C(C(F)(F)F)(C(F)(F)F)O
c1cc(ccc1c2c(c3ccc(cc3s2)O)C(=O)c4ccc(cc4)OCCN5CCCC5)O
CCOc1ccc2nc(NS(=O)(=O)c3ccc4N(CC)C(=O)c5cccc3c45)sc2c1
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)NCc1cc2cc(F)ccc2[nH]1
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)Nc1cccc2ccncc12
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)Nc1ccc(cc1)N1CCOCC1
O=C1Nc2ccc(c3cccc1c23)S(=O)(=O)Nc1ccc(cc1)N1CCOCC1
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)NCCN1CCOCC1
O=C1Nc2ccc(c3cccc1c23)S(=O)(=O)Nc1ccc(Oc2ccccc2)cc1
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)Nc1ccc(cc1)\N=N\c1ccccc1
COc1ccc(NC(=O)c2ccc(NS(=O)(=O)c3ccc4NC(=O)c5cccc3c45)cc2)cc1
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)Nc1cccc(NC(=O)OC(C)(C)C)c1
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)Nc1ccc(cc1)C(C)=O
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)NC1CCN(CC1)C(C)=O
CCN1c2ccc(c3c2c(ccc3)C1=O)S(=O)(=O)NCC4CCN(CC4)C(=O)C
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)Nc1cccc(c1)C(C)=O
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)Nc1ccc(NC(C)=O)cc1
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)Nc1ccccc1C(C)(C)C
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)Nc1ccc(OC)c(OC)c1
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)N(C(=O)c1ccncc1)c1ccc(OC)cc1
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)NCc1nc(C)cc(n1)C(F)(F)F
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)NCc1cc(Cl)ccc1Cl
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)Nc1cccc(c1)S(N)(=O)=O
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)Nc1ccc2ccccc2c1
CCCCCOC(=O)c1c(C)oc2cc(NS(=O)(=O)c3ccc4NC(=O)c5cccc3c45)ccc12
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)Nc1ccc2N(CCc2c1)C(C)=O
O=C1Nc2ccc(c3cccc1c23)S(=O)(=O)Nc1ccc(cc1)-c1ccccc1
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)Nc1ccccc1C(=O)c1ccccc1
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)Nc1cccc(c1)C(C)(C)C
CCN1C(=O)c2cccc3c(ccc1c23)S(=O)(=O)NCc1ccc(OC)cc1
Oc1cccc(\C=N\NC(=O)CSc2nnc(COc3ccc(Cl)cc3)n2CC=C)c1
COc1ccc(cc1)-c1nnc(SCC(=O)NCCc2ccc(cc2)S(N)(=O)=O)nc1-c1ccc(OC)cc1
C[C@@H](Sc1nnc(CNc2cccc(c2)C(F)(F)F)n1-c1ccccc1)C(=O)Nc1ccc(cc1)C(C)=O |r|
CC(N1C(=O)S\C(=C/c2cc(C)n(c2C)-c2ccc(cc2)S(N)(=O)=O)C1=O)c1ccccc1C#N
NS(=O)(=O)c1ccc(cc1)N1NC(\C(=C/c2ccc(o2)-c2ccc(cc2)S(N)(=O)=O)C1=O)C(F)(F)F
NC(=O)c1ccc(NC(=O)c2cccc(COc3ccc(Cl)cc3)c2)cc1
NS(=O)(=O)c1ccc(NC(=O)c2ccc(COc3ccccc3Cl)o2)cc1
COc1ccc(\C=N\c2ccc(cc2C)-c2ccc(\N=C\c3ccc(OC)c(O)c3)c(C)c2)cc1O
COc1cc(\C=C2\N=C(SCC(=O)Nc3ccc(cc3)S(N)(=O)=O)N(C2=O)c2ccccc2)cc(OC)c1OC |t:7|
CCC(C)(C)C1CCc2nc3sc(C(=O)Nc4ccc(cc4)S(N)(=O)=O)c(N)c3cc2C1
NS(=O)(=O)c1ccc(NC(=O)CSc2nnc(CCCN3C(=O)c4cccc5cccc(C3=O)c45)n2CC=C)cc1
CCCC1CC(=O)Oc2cc(OCC(=O)Nc3ccc(cc3)S(N)(=O)=O)c(Cl)cc12
CC(C)CN(Cc1ccc(s1)-c1cccc(c1)S(C)(=O)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(s1)-c1ccc(cc1)S(C)(=O)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)-c1ccc(NS(C)(=O)=O)cc1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)-c1ccc(cc1)S(N)(=O)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)-c1ccc(cc1)C(N)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)-c1ccc(CNC(C)=O)cc1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)-c1ccc(CC(N)=O)cc1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)-c1cccc(CC(N)=O)c1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)-c1ccc(cc1)S(C)(=O)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(s1)-c1ccccc1NS(C)(=O)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(s1)-c1cccc(NS(C)(=O)=O)c1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(s1)-c1ccc(NS(C)(=O)=O)cc1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(s1)-c1ccc(cc1)C(N)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(s1)-c1ccc(cc1)C(=O)N(C)C)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(s1)-c1ccc(CN)cc1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(s1)-c1ccc(=O)[nH]c1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(s1)-c1ccc(N)nc1)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(s1)-c1c(C)noc1C)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1cnc(s1)-c1ccc(cc1)S(C)(=O)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1cccc(c1)-c1ccc(cc1)S(C)(=O)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)-c1ccc(nc1)S(C)(=O)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)-c1ccc(cn1)S(C)(=O)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1cnc(cn1)-c1ccc(cc1)S(C)(=O)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(s1)-c1ccc(nc1)C#N)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(s1)-c1cncnc1)S(=O)(=O)Cc1ccccc1
OC(c1ccc2n(CC(F)(F)F)c(=O)c3ccccc3c2c1)(C(F)(F)F)C(F)(F)F
CCCCn1c2ccc(CC)cc2c2ccccc2c1=O
CCCCn1c2cc(OC)c(cc2c2ccccc2c1=O)C(O)(C(F)(F)F)C(F)(F)F
OC(c1ccc2n(CC3CC3)c(=O)c3ccccc3c2c1)(C(F)(F)F)C(F)(F)F
CCCCn1c2ccc(cc2c2ccccc2c1=O)C(C)(C)C
CCCCn1c2ccc(cc2c2ccccc2c1=O)C(C)C
CCCCCCc1ccc2n(CCCC)c(=O)c3ccccc3c2c1
CCCCn1c2ccccc2c2ccccc2c1=O
CCCCn1c2ccc(C)cc2c2ccccc2c1=O
CCCCn1c2c(OC)cc(cc2c2ccccc2c1=O)C(O)(C(F)(F)F)C(F)(F)F
OC(c1ccc2[nH]c(=O)c3ccccc3c2c1)(C(F)(F)F)C(F)(F)F
Cn1c2ccc(cc2c2ccccc2c1=O)C(O)(C(F)(F)F)C(F)(F)F
CCn1c2ccc(cc2c2ccccc2c1=O)C(O)(C(F)(F)F)C(F)(F)F
CCCCCCCCCn1c2ccc(cc2c2ccccc2c1=O)C(O)(C(F)(F)F)C(F)(F)F
CCCCn1c2ccc(CO)cc2c2ccccc2c1=O
CCCCn1c2ccc(cc2c2cc(OC)ccc2c1=O)C(O)(C(F)(F)F)C(F)(F)F
CCCCn1c2ccc(cc2c2cc(C)ccc2c1=O)C(O)(C(F)(F)F)C(F)(F)F
CCCCn1c2ccc(cc2c2cc(Cl)ccc2c1=O)C(O)(C(F)(F)F)C(F)(F)F
CCCCn1c2ccc(cc2c2cc(ccc2c1=O)C(F)(F)F)C(O)(C(F)(F)F)C(F)(F)F
CCCCn1c2ccc(cc2c2ccccc2c1=O)C(O)(C(F)(F)F)C(F)(F)F
CCCCn1c2ccc(cc2c2cc(O)ccc2c1=O)C(O)(C(F)(F)F)C(F)(F)F
CCCn1c2ccc(cc2c2ccccc2c1=O)C(O)(C(F)(F)F)C(F)(F)F
CCCCCCn1c2ccc(cc2c2ccccc2c1=O)C(O)(C(F)(F)F)C(F)(F)F
CCCCn1c2ccc(cc2c2c(OC)cccc2c1=O)C(O)(C(F)(F)F)C(F)(F)F
OC(c1ccc2n(CC3CCCCC3)c(=O)c3ccccc3c2c1)(C(F)(F)F)C(F)(F)F
CC(C)n1c2ccc(cc2c2ccccc2c1=O)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)CC(=O)Nc2nc(c(s2)C(=O)c3ccccc3Cl)c4cccc(c4)Cl
CCS(=O)(=O)c1ccc(cc1)CC(=O)Nc2nc(c(s2)C(=O)c3ccccc3)c4ccccc4
CC1=C(C(CCC1)(C)C)/C=C/C(=C/C=C/C(=C/C(=O)O)/C)/C
CC(C)CN(Cc1ccccc1)S(=O)(=O)Cc1ccc(cc1)-c1ccc(cc1)S(C)(=O)=O
CC(C)CN(CCc1ccccc1)S(=O)(=O)c1ccc(cc1)-c1ccc(cc1)S(C)(=O)=O
C[C@@H]1[C@H]([C@H](C[C@@H](O1)O[C@@H]2[C@H](O[C@H](C[C@@H]2O)O[C@@H]3[C@H](O[C@H](C[C@@H]3O)O[C@H]4CC[C@]5([C@@H](C4)CC[C@@H]6[C@@H]5C[C@H]([C@]7([C@@]6(CC[C@@H]7C8=CC(=O)OC8)O)C)O)C)C)C)O)O
C[C@H](CCCC(C)(C)O)[C@H]1CC[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C |t:15|
C[C@@H]([C@H]1CC[C@@H]2[C@@]1(CC[C@H]3[C@H]2CC=C4[C@@]3(CC[C@@H](C4)O)C)C)[C@@H](CCC(C)C)O
CC(C)CCC[C@@](C)(O)[C@H]1CC[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C |r,t:15|
CC(C)CN(Cc1ccccc1C(F)(F)F)S(=O)(=O)c1ccc(OC2CCN(CC2)S(C)(=O)=O)cn1
CC(C)CN(Cc1ccc(cc1)F)S(=O)(=O)c2ccc(nc2)NC3CCN(CC3)S(=O)(=O)C
CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(cc1)N1CCOCC1
CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(cc1)N1CCC(O)CC1
CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(cc1)N1CCN(C)CC1
CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(cc1)N1CCN(CC1)C(C)=O
CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(cc1)N1CCN(CC1)S(=O)(=O)N(C)C
CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(cc1)N1CCN(CC1)S(C)(=O)=O
CC(C)CN(CCc1ccccc1)S(=O)(=O)c1ccc(cc1)N1CCN(CC1)S(C)(=O)=O
CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(cc1F)N1CCN(CC1)S(C)(=O)=O
CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(N2CCN(CC2)S(C)(=O)=O)c(F)c1
CC(C)CN(CCc1ccccc1)S(=O)(=O)c1ccc(cc1F)N1CCN(CC1)S(C)(=O)=O
CC(C)CN(CCc1ccccc1)S(=O)(=O)c1ccc(N2CCN(CC2)S(C)(=O)=O)c(F)c1
CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(cn1)N1CCN(CC1)S(C)(=O)=O
CC(C)CN(CCc1ccccc1)S(=O)(=O)c1ccc(cn1)N1CCN(CC1)S(C)(=O)=O
CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(nc1)N1CCN(CC1)S(C)(=O)=O
CC(C)CN(CCc1ccccc1)S(=O)(=O)c1ccc(nc1)N1CCN(CC1)S(C)(=O)=O
CC(C)CN(Cc1ccccc1Cl)S(=O)(=O)c1ccc(cc1)N1CCN(CC1)S(C)(=O)=O
CC(C)CN(Cc1cccc(Cl)c1)S(=O)(=O)c1ccc(cc1)N1CCN(CC1)S(C)(=O)=O
CC(C)CN(Cc1ccc(Cl)cc1)S(=O)(=O)c1ccc(cc1)N1CCN(CC1)S(C)(=O)=O
CC(C)CN(Cc1ccccc1C(F)(F)F)S(=O)(=O)c1ccc(cc1)N1CCN(CC1)S(C)(=O)=O
CC(C)CN(Cc1ccccc1C(F)(F)F)S(=O)(=O)c1ccc(cc1)N1CCN(CC1)C(C)=O
CC(C)CN(Cc1ccccc1C(F)(F)F)S(=O)(=O)c1ccc(NC2CCN(CC2)S(C)(=O)=O)cc1
CC(C)CN(c1ccccc1C(F)(F)F)S(=O)(=O)c1ccc(NC2CCN(CC2)S(C)(=O)=O)cc1
CC(C)CN(Cc1ccccc1C(F)(F)F)S(=O)(=O)c1ccc(OC2CCN(CC2)S(C)(=O)=O)cc1
CC(C)CN(Cc1ccccc1C(F)(F)F)S(=O)(=O)c1ccc(cc1)C(=O)C1CCN(CC1)S(C)(=O)=O
CC(C)CN(Cc1ccccc1C(F)(F)F)S(=O)(=O)c1ccc(cc1)C(O)C1CCN(CC1)S(C)(=O)=O
[#6]-[#6](-[#6])-[#6]-[#7](-[#6]-c1ccccc1C(F)(F)F)S(=O)(=O)c1ccc(\[#6]=[#6]-2/[#6]-[#6]-[#7](-[#6]-[#6]-2)S([#6])(=O)=O)cc1
CC(C)CN(c1ccccc1F)S(=O)(=O)c1ccc(OC2CCN(CC2)S(C)(=O)=O)cc1
CC(C)CN(c1cccc(F)c1)S(=O)(=O)c1ccc(OC2CCN(CC2)S(C)(=O)=O)cc1
CC(C)CN(c1ccc(F)cc1)S(=O)(=O)c1ccc(OC2CCN(CC2)S(C)(=O)=O)cc1
CC(C)CN(c1ccccc1C#N)S(=O)(=O)c1ccc(OC2CCN(CC2)S(C)(=O)=O)cc1
CC(C)CN(c1cccc(c1)C#N)S(=O)(=O)c1ccc(OC2CCN(CC2)S(C)(=O)=O)cc1
CC(C)CN(c1ccc(cc1)C#N)S(=O)(=O)c1ccc(OC2CCN(CC2)S(C)(=O)=O)cc1
CC(C)CN(c1ccccn1)S(=O)(=O)c1ccc(OC2CCN(CC2)S(C)(=O)=O)cc1
CC(C)CN(c1cccnc1)S(=O)(=O)c1ccc(OC2CCN(CC2)S(C)(=O)=O)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(-c3ccccc3)c(c2)C(C)C)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(Oc3ccc(Cl)cc3C(F)(F)F)s2)-c2cccc(c2)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(c(s2)C(=O)c2ccccc2Cl)-c2cccc(Cl)c2)cc1
Cc1ccc(NC(=O)C[C@H](CCC(O)=O)c2nnn([C@@H]3C[C@H](CC(C)(C)C)C3)c2C(F)(F)F)c(C)c1 |r,wU:19.18,21.21,wD:9.9,(20.75,-24.44,;19.84,-23.19,;18.31,-23.35,;17.41,-22.1,;18.04,-20.7,;17.13,-19.46,;15.6,-19.62,;14.7,-18.37,;14.97,-21.02,;13.44,-21.18,;12.81,-22.59,;13.72,-23.83,;13.09,-25.24,;11.56,-25.4,;13.99,-26.49,;12.54,-19.93,;13.02,-18.47,;11.77,-17.56,;10.53,-18.47,;9.05,-18,;8.35,-16.63,;6.98,-17.33,;5.52,-16.85,;5.2,-15.34,;3.73,-14.87,;6.34,-14.31,;4.79,-13.84,;7.68,-18.7,;11,-19.93,;10.09,-21.18,;8.56,-21.02,;10.72,-22.59,;9.31,-22.51,;19.56,-20.54,;20.18,-19.13,;20.47,-21.78,)|
Cc1ccc(NC(=O)C[C@H](CCC(O)=O)c2noc([C@@H]3C[C@H](CC(C)(C)C)C3)c2C2CC2)c(Cl)c1 |r,wU:19.18,21.21,wD:9.9,(16.24,-21,;15.33,-19.75,;13.8,-19.91,;12.9,-18.67,;13.53,-17.27,;12.62,-16.02,;11.09,-16.18,;10.19,-14.93,;10.46,-17.58,;8.93,-17.74,;8.3,-19.15,;9.21,-20.4,;8.58,-21.8,;7.05,-21.97,;9.48,-23.05,;8.03,-16.5,;8.51,-15.03,;7.26,-14.12,;6.02,-15.03,;4.54,-14.56,;3.84,-13.19,;2.47,-13.89,;1.01,-13.41,;.68,-11.91,;-.79,-11.43,;1.83,-10.88,;.28,-10.41,;3.17,-15.26,;6.49,-16.5,;5.58,-17.74,;4.17,-18.37,;5.41,-19.28,;15.05,-17.1,;15.67,-15.69,;15.96,-18.34,)|
CC(C)C[C@H]1C[C@H](C1)c1onc([C@@H](CC(O)=O)CC(=O)Nc2cc(C)ccc2Cl)c1C1CC1 |r,wU:6.8,4.3,wD:12.13,(20.31,-3.58,;21.78,-4.06,;22.92,-3.03,;22.1,-5.56,;23.56,-6.04,;24.94,-5.34,;25.64,-6.71,;24.26,-7.41,;27.11,-7.19,;28.35,-6.28,;29.6,-7.19,;29.12,-8.65,;30.02,-9.9,;29.4,-11.3,;30.3,-12.55,;29.67,-13.96,;31.83,-12.39,;31.56,-9.74,;32.18,-8.33,;31.28,-7.08,;33.72,-8.17,;34.62,-9.42,;33.99,-10.82,;34.89,-12.06,;34.26,-13.47,;36.42,-11.91,;37.05,-10.49,;36.14,-9.25,;36.77,-7.84,;27.58,-8.65,;26.67,-9.9,;25.26,-10.52,;26.51,-11.43,)|
CC(C)C[C@H]1C[C@H](C1)c1onc([C@@H](CC(O)=O)CC(=O)Nc2ccc(C)cc2Cl)c1C1CC1 |r,wU:6.8,4.3,wD:12.13,(.09,-.42,;1.56,-.89,;2.7,.14,;1.88,-2.4,;3.34,-2.87,;4.71,-2.17,;5.41,-3.55,;4.04,-4.25,;6.89,-4.02,;8.13,-3.11,;9.38,-4.02,;8.9,-5.48,;9.8,-6.73,;9.17,-8.14,;10.08,-9.38,;9.45,-10.79,;11.61,-9.23,;11.33,-6.57,;11.96,-5.17,;11.06,-3.92,;13.49,-5.01,;14.4,-6.25,;13.77,-7.65,;14.67,-8.9,;16.2,-8.74,;17.11,-9.99,;16.83,-7.32,;15.92,-6.08,;16.54,-4.67,;7.36,-5.48,;6.45,-6.73,;5.04,-7.36,;6.28,-8.26,)|
Cc1noc(C)c1CN(CC(O)=O)c1ccc(CC(=O)NC(c2ccccc2)c2ccc(C)cc2)cc1
Cc1ccc([C@@H](NC(=O)Cc2ccc3oc(cc3c2)C(N2CC(N)C2)c2ccncc2)c2ccccc2)c(C)c1 |r|
CC(C)CCC(NC(=O)Cc1ccc2oc(cc2c1)C(O)c1c(C)noc1C)c1ncc(C)cc1C
Cc1noc(C)c1COc1ccc(CC(=O)NC(c2ccc(Cl)cc2)c2ccc(Cl)cc2C)cc1
Cc1noc(C)c1C(O)c1cc2cc(CC(=O)NC(c3ccccc3)c3ccc(C)cc3C)ccc2o1
Cc1ccc(C(NC(=O)Cc2ccc(OCC(O)c3cccnc3C)cc2)c2ccccc2)c(C)c1
CC(C)CN(c1ccc(C)cc1C)S(=O)(=O)c1ccc(OCc2ccncc2)cc1
Fc1cccc(c1C(=O)Nc1ccc2cnn(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(F)(F)F
OC[C@H]1CN(c2cc(NC(=O)c3c(F)cccc3Cl)ccc2O1)S(=O)(=O)c1cccc(c1)C#N |r|
Fc1ccc(cc1)S(=O)(=O)N1CCCc2ccc(NC(=O)c3c(F)cccc3Cl)cc12
CC(C)C(C)N(c1ccc(cn1)C(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)cc1
CC(C)CN(c1ccc(Cl)cc1)S(=O)(=O)c1ccc(OCc2c(C)noc2C)cc1
OC(c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3n(CCc4ccc(Cl)cc4Cl)ccc3c2)cc1
CCCN(Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1)Cc1ccc(OC2CCCC2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(cs2)-c2cc(Cl)ccc2Cl)cc1
[Na+].OCCNC(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1)C([O-])=O
OC(=O)c1ccc(cc1O)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
[Na+].[O-]C(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cccnc23)c(F)c1
Cc1c(cc(-c2cn(c3ccccc23)S(=O)(=O)N2CCCCC2)n1CC1CCCCC1)S(N)(=O)=O
Cc1c(cc(-c2cc(cc(c2)C(C)(C)C)C(C)(C)C)n1CC1CCCCC1)S(=O)(=O)NCCO
Cc1c(cc(-c2cc(cc(c2)C(C)(C)C)C(C)(C)C)n1CC1CCCCC1)S(N)(=O)=O
CO[C@@H]1Cc2ccccc2CN([C@@H]1Cc1ccccc1)S(=O)(=O)c1cccc2cccnc12 |r|
FC(F)(F)Oc1ccccc1S(=O)(=O)N1Cc2cncnc2-n2ccnc2[C@H]1Cc1ccccc1 |r|
Fc1ccc(OC(F)(F)F)c(c1)S(=O)(=O)N1Cc2nccnc2-n2ccnc2[C@H]1Cc1ccccc1 |r|
COc1ccccc1S(=O)(=O)N1Cc2ccccc2COCC1Cc1ccccc1
CC1=C(C(CCC1)(C)C)/C=C/C(=C\C=C\C(=C\C(=O)O)\C)/C
C/C(=C\c1ccc(cc1)C(=O)O)/c2ccc3c(c2)C(CCC3(C)C)(C)C
CN1c2cc3c(cc2N=C(c2ccc(cc2)C(O)=O)c2ccc4ccccc4c12)C(C)(C)CCC3(C)C |t:9|
[H][C@@]1(C[C@H](O)[C@H](O)[C@@H](C)O1)O[C@H]1[C@@H](O)C[C@H](O[C@@]2([H])[C@@H](O)C[C@]([H])(O[C@H]3CC[C@@]4(C)[C@]([H])(CC[C@]5([H])[C@]4([H])C[C@@H](O)[C@]4(C)[C@H](CC[C@]54O)C(=O)OC)C3)O[C@@H]2C)O[C@@H]1C |r|
[H][C@@]1(C[C@H](O)[C@H](O)[C@@H](C)O1)O[C@H]1[C@@H](O)C[C@H](O[C@@]2([H])[C@@H](O)C[C@]([H])(O[C@H]3CC[C@@]4(C)[C@]([H])(CC[C@]5([H])[C@]4([H])C[C@@H](O)[C@]4(C)[C@H](CC[C@]54O)C4=CC(=O)O\C4=C/c4ccccc4O)C3)O[C@@H]2C)O[C@@H]1C |r,t:52|
[H][C@@]1(C[C@H](O)[C@]([H])(O[C@H]2C[C@H](O)[C@H](O[C@@]3([H])C[C@H](O)[C@H](O)[C@@H](C)O3)[C@@H](C)O2)[C@@H](C)O1)O[C@H]1CC[C@@]2(C)[C@]([H])(CC[C@]3([H])[C@]2([H])C[C@@H](O)[C@]2(C)[C@H](CC[C@]32O)C(CO)CCO)C1 |r|
Cc1cc(ccc1-c1ccc(CN2CCN(Cc3ccncc3)CC2)cc1)C(O)(C(F)(F)F)C(F)(F)F
Cc1cc(CN2CCN(Cc3ccncc3)CC2)ccc1-c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CC(N1CCN(Cc2ccc(cc2)-c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)CC1)c1ccncc1
CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(Cl)c1C |r,wU:30.34,wD:28.29,(19.83,-3.9,;18.5,-4.68,;18.5,-6.22,;19.84,-6.98,;19.83,-5.44,;17.17,-6.99,;15.83,-6.22,;15.06,-4.88,;16.6,-4.88,;14.51,-7,;14.51,-8.55,;13.17,-9.32,;11.84,-8.55,;10.51,-9.32,;10.34,-10.85,;8.84,-11.17,;8.07,-9.83,;9.1,-8.69,;8.78,-7.18,;7.32,-6.7,;7,-5.19,;5.54,-4.71,;4.39,-5.73,;4.71,-7.24,;6.17,-7.73,;8.21,-12.57,;9.11,-13.82,;6.68,-12.73,;6.05,-14.14,;4.62,-14.69,;5.17,-16.13,;6.61,-15.58,;4.54,-17.54,;3.01,-17.7,;5.45,-18.79,;11.84,-7.01,;10.51,-6.24,;13.17,-6.24,;13.17,-4.7,)|
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CCS(=O)(=O)CC3)c2ccccc12
Cc1c(cc(-c2ccc(c3ccccc23)S(=O)(=O)NC(C)(C)C)n1CC1CCCCC1)C(=O)N1CC2(C1)CCS(=O)(=O)CC2
CC(C)n1ccc[n+]1-c1ccc(cc1C(C)(C)C)-c1cc(C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(C)n1CC1CCCCC1 |r,wU:26.30,wD:24.25,(26.41,-32.77,;25.78,-34.18,;24.25,-34.33,;26.68,-35.43,;28.22,-35.43,;28.7,-36.9,;27.45,-37.8,;26.2,-36.89,;24.74,-37.37,;23.58,-36.33,;22.12,-36.8,;21.8,-38.3,;22.95,-39.34,;24.41,-38.87,;25.55,-39.9,;25.23,-41.4,;27.02,-39.43,;26.64,-40.98,;20.35,-38.78,;19.87,-40.24,;18.33,-40.24,;17.42,-41.49,;18.04,-42.9,;15.89,-41.33,;14.98,-42.57,;13.46,-42.81,;13.7,-44.33,;15.22,-44.09,;12.79,-45.58,;11.26,-45.42,;13.42,-46.99,;17.86,-38.78,;16.39,-38.31,;19.1,-37.87,;19.09,-36.33,;17.76,-35.56,;17.75,-34.02,;16.43,-33.25,;15.09,-34.01,;15.09,-35.56,;16.42,-36.33,)|
Cc1c(cc(-c2cc(c3OCCC4(CC4)c3c2)C(C)(C)C)n1CC1CCCCC1)C(=O)NC1CCOCC1
CC(=O)N1CCN(Cc2ccc(cc2)-c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)CC1
CC(=O)Nc1nc(C)c(s1)S(=O)(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCC(=O)Nc1ccc2nn(nc2c1)-c1ccc(CC)cc1
Cc1ccsc1C(=O)Nc1nc2c(C)cc(C)cc2s1
Cc1cccc(c1)C(=O)Nc1cc(no1)-c1ccccc1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(C(O)CN2CCOCC2)c(CO)c1
OC(=O)c1ccc(cc1)-c1nn(c2ccccc12)S(=O)(=O)c1ccccc1C(F)(F)F
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(Oc3ccccc3)c2)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(Oc3cccc(OC(F)(F)F)c3)c2)-n2ccc(C)n2)cc1
CCCN(Cc1ccccc1)Cc2ccc(cc2)NC(=O)Cc3ccc(cc3)S(=O)(=O)CC
O=S(=O)(N1Cc2ccccc2COCC1Cc1ccccc1)c1cccc2cccnc12
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N(C([2H])([2H])C([2H])([2H])[2H])C([2H])([2H])C([2H])([2H])[2H])-c1cc(ccc1Cl)C(=O)NCC(C)(C)O
[H][C@@]12C[C@]1([H])C[C@@H](C2)Oc1cc(ccc1N(C)C(=O)c1c(F)cccc1Cl)-c1cc(ccc1Cl)C(N)=O |r|
OC(c1ccc(CN2CCCc3cc(ccc23)-c2cn[nH]c2)cc1)(C(F)(F)F)C(F)(F)F
NC(=O)c1ccc2N(Cc3ccc(cc3)C(O)(C(F)(F)F)C(F)(F)F)CCc2c1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cccc(c2)-c2cc(Cl)ccc2Cl)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)F)cc1 |(.3,-24.38,;1.64,-23.61,;2.96,-24.38,;3.73,-25.71,;2.19,-25.7,;4.3,-23.61,;5.64,-24.38,;6.98,-23.61,;6.97,-22.06,;8.3,-21.28,;9.64,-22.05,;9.64,-23.59,;10.97,-21.27,;12.31,-22.04,;12.31,-23.58,;13.64,-24.34,;13.65,-25.88,;14.97,-23.57,;14.96,-22.02,;16.29,-21.24,;13.63,-21.26,;16.31,-24.33,;16.31,-25.87,;17.65,-26.63,;18.98,-25.86,;18.97,-24.31,;17.63,-23.55,;17.62,-22.01,;18.95,-21.23,;18.93,-19.69,;20.29,-21.99,;5.64,-21.3,;4.31,-22.07,)|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1
CC(C)CN(Cc1ccc(cc1)N1CCN(CC1)NS(C)(=O)=O)S(=O)(=O)Cc1ccccc1
CC(C)CN(Cc1ccc(cc1)N1CCN(CS(C)(=O)=O)CC1)S(=O)(=O)Cc1ccccc1
CN(C)CCN(Cc1ccc(cc1)N1CCN(CC1)C(C)=O)S(=O)(=O)Cc1ccccc1
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCC2(CC1)N(C)C(=O)N(C)C2=O |r|
Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2nc(Cl)c(Cc3ccccc3)c(Cl)c2c1
OC(c1cncs1)(c1ccncc1)c1ccc2nc(Cl)c(Cc3ccc(Cl)cc3)c(Cl)c2c1
Cn1cncc1C(O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(C#N)c(Cc3ccc(cc3)-n3cccn3)c(C#N)c2c1
COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cnnn1C)c1sc(C)nc1C
CC(CCO)N(C)C(=O)CCCN1c2ccccc2N(Cc2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)S1(=O)=O
COc1cccc(CN(C)C(=O)CCCN2c3ccccc3N(Cc3ccc(cc3)C(O)(C(F)(F)F)C(F)(F)F)S2(=O)=O)c1
CN(Cc1ccccc1C)C(=O)CCCN1c2ccccc2N(Cc2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)S1(=O)=O
OC(c1ccc(CN2c3ccccc3N(CCCC(=O)N3CCCC3)S2(=O)=O)cc1)(C(F)(F)F)C(F)(F)F
CC(C)C(=O)N1CCC(CN2c3ccccc3N(Cc3ccc(cc3)C(O)(C(F)(F)F)C(F)(F)F)S2(=O)=O)CC1
CCC(=O)N1CCCC(CN2c3ccccc3N(Cc3ccc(cc3)C(O)(C(F)(F)F)C(F)(F)F)S2(=O)=O)C1
CCC(CC)c1ccc(CN2c3ccccc3N(CCCC(=O)N3CCCC3)S2(=O)=O)cc1
CC(C)c1ccc(CN2c3ccccc3N(CCCC(=O)N3CCCC3)S2(=O)=O)cc1
OC(c1ccc(CN2c3ccccc3N(CCCC(=O)N3CCCC3)S2(=O)=O)cc1)C(F)(F)F
O=C(CCCN1c2ccccc2N(Cc2ccccc2)S1(=O)=O)N1CCCC1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2ccc(C)cc2C)c(F)c1
CC(=O)N1CCN(CC1)c1ccc(CN(C2CCC2)S(=O)(=O)c2ccc(OC(F)F)cc2)c(F)c1
CCCC[Si]1(CCCC)c2ccccc2-c2cc(ccc12)C(O)(C(F)(F)F)C(F)(F)F
C[Si]1(C)c2ccccc2-c2cc(ccc12)C(O)(C(F)(F)F)C(F)(F)F
CC[Si]1(CC)c2ccccc2-c2cc(ccc12)C(O)(C(F)(F)F)C(F)(F)F
CCCC[Si]1(C)c2ccccc2-c2cc(ccc12)C(O)(C(F)(F)F)C(F)(F)F
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1OCC(F)(F)F)-c1cc(ccc1Cl)C(N)=O
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1OCC(F)(F)F)-c1cc(nn1C(C)C)C(N)=O
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1OCC(F)(F)F)-c1cn(C)nc1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1OCC(F)(F)F)-c1cnn(C)c1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1OCC(F)(F)F)-c1cc(CC(N)=O)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1OCC(F)(F)F)-c1cc(NC(C)=O)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1OCC1CCC1)-c1cc(NC(C)=O)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1OCC(C)C)-c1cc(NC(C)=O)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1OC1CC2CC2C1)-c1cc(NC(C)=O)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(C)=O)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CCCC1)-c1cc(NC(C)=O)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CCCCC1)-c1cc(NC(C)=O)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1-c1ccccc1)-c1cc(NC(C)=O)nn1C(C)C
CC(C)n1nc(NC(C)=O)cc1-c1ccc(N(C)C(=O)c2c(F)cccc2Cl)c(c1)N1CC2CC2C1
[2H]C([2H])([2H])N(C(=O)c1c(Cl)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(C)=O)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(C)cccc1F)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(C)=O)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ncc(cc1N1CC2CC2C1)-c1cc(NC(C)=O)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC=O)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(=O)CC)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(=O)C2CC2)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(=O)[C@H]2C[C@H](O)C2)nn1C(C)C |r,wU:33.36,wD:35.39,(.26,3.23,;1.33,3.85,;.26,4.46,;1.32,4.88,;2.66,3.08,;2.67,1.54,;3.73,.93,;1.33,.77,;1.33,-.77,;2.4,-1.39,;,-1.54,;-1.33,-.77,;-1.33,.77,;,1.54,;,2.77,;4,3.86,;5.33,3.09,;6.66,3.86,;6.66,5.4,;5.33,6.17,;4,5.4,;2.66,6.17,;1.44,5.49,;.22,6.2,;.22,7.6,;1.43,8.27,;2.65,7.56,;8,6.17,;8.14,7.69,;9.64,8.01,;10.27,9.42,;11.8,9.58,;12.53,8.58,;12.43,10.98,;11.85,12.37,;13.29,12.93,;13.79,14.05,;13.85,11.49,;10.42,6.68,;9.39,5.53,;9.7,4.03,;10.87,3.64,;8.78,3.21,)|
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(=O)CO)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(=O)CN(C)C)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(=O)NC)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(=O)N2CC3(COC3)C2)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(=O)N2CC(O)C2)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(=O)NCCO)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(=O)OC(C)C)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(C)=O)nn1C1CCCC1
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(C)=O)nn1C1CCC1
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(C)=O)nn1CC(C)(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(C)=O)nn1C1COC1
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(C)=O)nn1CC1CC1
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(C)=O)nn1C(C)C1CC1
CC(C)n1nc(NC(C)=O)cc1-c1cnc(N(C)C(=O)c2c(F)cccc2Cl)c(c1)N1CCCCC1
CC(C)c1nc(NC(C)=O)sc1-c1cnc(N(C)C(=O)c2c(F)cccc2Cl)c(c1)N1CCCCC1
CC(C)n1nc(NC(C)=O)nc1-c1cnc(N(C)C(=O)c2c(F)cccc2Cl)c(c1)N1CCCCC1
CC(C)n1cc(NC(C)=O)nc1-c1cnc(N(C)C(=O)c2c(F)cccc2Cl)c(c1)N1CCCCC1
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(=O)C(C)C)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(=O)[C@@H]2C[C@H](O)C2)nn1C(C)C |r,wU:33.36,35.39,(.26,3.23,;1.33,3.85,;.26,4.46,;1.32,4.88,;2.66,3.08,;2.67,1.54,;3.73,.93,;1.33,.77,;1.33,-.77,;2.4,-1.39,;,-1.54,;-1.33,-.77,;-1.33,.77,;,1.54,;,2.77,;4,3.86,;5.33,3.09,;6.66,3.86,;6.66,5.4,;5.33,6.17,;4,5.4,;2.66,6.17,;1.44,5.49,;.22,6.2,;.22,7.6,;1.43,8.27,;2.65,7.56,;8,6.17,;8.14,7.69,;9.64,8.01,;10.27,9.42,;11.8,9.58,;12.53,8.58,;12.43,10.98,;13.85,11.49,;13.29,12.93,;13.79,14.05,;11.85,12.37,;10.42,6.68,;9.39,5.53,;9.7,4.03,;10.87,3.64,;8.78,3.21,)|
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(=O)NC(CO)CO)nn1C(C)C
[2H]C([2H])([2H])N(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CC2CC2C1)-c1cc(NC(=O)OC2(C)CC2)nn1C(C)C
OC(=O)c1ccc(cc1O)-c1nc(C(=O)c2c(Cl)cccc2C2CC2)n2cccnc12
OC(=O)C1(O)CCN(CC1)c1nc(C(=O)c2c(Cl)cccc2C(F)(F)F)n2ccccc12
O[C@H]1CN(CC[C@@H]1C(O)=O)c1nc(C(=O)c2c(Cl)cccc2C(F)(F)F)n2ccccc12 |r|
O[C@@H]1CN(CC[C@H]1C(O)=O)c1nc(C(=O)c2c(Cl)cccc2C(F)(F)F)n2ccccc12 |r|
OC(=O)c1ccc(-c2nc(C(=O)c3c(Cl)cccc3C(F)(F)F)n3CCCCc23)c(F)c1
OC(=O)c1ccc(-c2nc(C(=O)c3ccccc3C(F)(F)F)n3CCCCc23)c(F)c1
OC(=O)c1ccc(-c2nc(C(=O)c3c(F)cccc3Cl)n3CCCCc23)c(F)c1
OC(=O)c1ccc(-c2nc(C(=O)c3c(Cl)cccc3Cl)n3CCCCc23)c(F)c1
OC(=O)c1ccc(-c2nc(C(=O)c3c(Cl)cccc3C#N)n3CCCCc23)c(F)c1
COc1cccc(Cl)c1C(=O)c1nc(c2CCCCn12)-c1ccc(cc1F)C(O)=O
OC(=O)c1ccc(-c2nc(C(=O)c3c(Cl)cccc3C3CC3)n3CCCCc23)c(F)c1
OC(=O)c1ccc(-c2nc(C(=O)c3c(cccc3C(F)(F)F)C#N)n3CCCCc23)c(F)c1
COc1cccc(c1C(=O)c1nc(c2CCCCn12)-c1ccc(cc1F)C(O)=O)C(F)(F)F
OC(=O)c1ccc(cc1)-c1nc(C(=O)c2c(Cl)cccc2C(F)(F)F)n2ccccc12
OC(=O)c1ccc(cc1)-c1nc(C(=O)c2c(Cl)cccc2C(F)(F)F)n2CCCCc12
OC(=O)c1ccc(cc1)-c1nc(C(=O)c2c(Cl)cccc2C(F)(F)F)n2cccnc12
OC(=O)c1ccc(cc1)-c1nc(C(=O)c2c(Cl)cccc2C(F)(F)F)n2ccncc12
OC(=O)c1ccc(cc1)-n1nc(C(=O)c2c(Cl)cccc2C(F)(F)F)c2CCCCc12
OC(=O)c1ccc(cc1)-c1cn2ccnc(-c3c(Cl)cccc3C(F)(F)F)c2n1 |(9.49,.73,;8.8,-.29,;9.34,-1.4,;7.27,-.19,;6.59,1.2,;5.05,1.3,;4.2,.03,;4.87,-1.36,;6.41,-1.46,;2.66,.02,;1.76,1.24,;.3,.77,;-1.03,1.55,;-2.38,.77,;-2.38,-.77,;-1.03,-1.55,;-1.02,-3.09,;-2.36,-3.86,;-3.43,-3.24,;-2.37,-5.4,;-1.04,-6.17,;.3,-5.41,;.31,-3.87,;1.64,-3.1,;1.65,-1.87,;2.71,-3.72,;2.71,-2.49,;.3,-.77,;1.76,-1.24,)|
OC(=O)c1ccc(cc1)-c1cn2CCOC(c2n1)c1c(Cl)cccc1C(F)(F)F
OC(=O)c1ccc(cc1O)-c1nc(C(=O)c2c(Cl)cccc2C(F)(F)F)n2ccccc12
OC(=O)c1ccc(-c2nc(C(=O)c3c(Cl)cccc3C(F)(F)F)n3ccccc23)c(F)c1
OC(=O)C1CCC(=CC1)c1nc(C(=O)c2c(Cl)cccc2C(F)(F)F)n2ccccc12 |c:6|
OC(=O)[C@H]1CC[C@@H](CC1)c1nc(C(=O)c2c(Cl)cccc2C(F)(F)F)n2ccccc12 |r,wU:6.9,wD:3.2,(3.2,7.95,;3.96,6.98,;5.18,7.15,;3.38,5.55,;1.86,5.34,;1.29,3.91,;2.23,2.7,;3.76,2.91,;4.33,4.34,;1.76,1.24,;2.66,.02,;1.76,-1.24,;2.24,-2.7,;1.42,-3.62,;3.75,-3.01,;4.77,-1.86,;4.39,-.69,;6.28,-2.16,;6.77,-3.63,;5.75,-4.78,;4.24,-4.47,;3.22,-5.62,;2.01,-5.37,;3.61,-6.79,;2.4,-6.54,;.3,-.77,;-1.03,-1.55,;-2.38,-.77,;-2.38,.77,;-1.03,1.55,;.3,.77,)|
OC(=O)[C@H]1CC[C@H](CC1)c1nc(C(=O)c2c(Cl)cccc2C(F)(F)F)n2ccccc12 |r,wU:6.9,3.2,(3.2,7.95,;3.96,6.98,;5.18,7.15,;3.38,5.55,;4.33,4.34,;3.76,2.91,;2.23,2.7,;1.29,3.91,;1.86,5.34,;1.76,1.24,;2.66,.02,;1.76,-1.24,;2.24,-2.7,;1.42,-3.62,;3.75,-3.01,;4.77,-1.86,;4.39,-.69,;6.28,-2.16,;6.77,-3.63,;5.75,-4.78,;4.24,-4.47,;3.22,-5.62,;2.01,-5.37,;3.61,-6.79,;2.4,-6.54,;.3,-.77,;-1.03,-1.55,;-2.38,-.77,;-2.38,.77,;-1.03,1.55,;.3,.77,)|
OC(=O)C1CCN(CC1)c1nc(C(=O)c2c(Cl)cccc2C(F)(F)F)n2ccccc12
CN(C(=O)c1c(F)cccc1Cl)c1ncc(cc1OCC(F)(F)F)-c1cc(ccc1Cl)C(N)=O
CN(C(=O)c1c(F)cccc1Cl)c1ncc(cc1OCC1CCC1)-c1cc(ccc1Cl)C(N)=O
CCNc1cc(ccc1N(C)C(=O)c1c(F)cccc1Cl)-c1cc(ccc1Cl)C(N)=O
CCN(CC)c1cc(ccc1N(C)C(=O)c1c(F)cccc1Cl)-c1cc(ccc1Cl)C(N)=O
CN(C(=O)c1c(F)cccc1Cl)c1ccc(cc1N1CCCCC1)-c1cc(ccc1Cl)C(N)=O
Cn1ccc2c(cccc12)S(=O)(=O)N(CC(F)(F)F)c1ccc(cc1)-c1cc(ccc1Cl)C(N)=O
NC(=O)c1ccc(Cl)c(c1)-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl
Cc1ccc(cc1-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl)C(N)=O
NC(=O)c1cc(c(Cl)cc1F)-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl
CNC(=O)c1ccc(Cl)c(c1)-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl
CCNC(=O)c1ccc(Cl)c(c1)-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl
Fc1cccc(Cl)c1C(=O)N1CCCc2cc(ccc12)-c1cc(ccc1Cl)C(=O)NC1CCCC1
OCCNC(=O)c1ccc(Cl)c(c1)-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl
NC(=O)c1ccc(Cl)c(c1)-c1ccc2N(CCCCc2c1)C(=O)c1c(F)cccc1Cl
CC1(C)CN(C(=O)c2c(F)cccc2Cl)c2ccc(cc2C1)-c1cc(ccc1Cl)C(N)=O
CC1(C)CCN(C(=O)c2c(F)cccc2Cl)c2ccc(cc12)-c1cc(ccc1Cl)C(N)=O
CN1CCN(C(=O)c2c(F)cccc2Cl)c2ccc(cc12)-c1cc(ccc1Cl)C(N)=O
CN(C(=O)c1c(F)cccc1Cl)c1ccc(cc1Br)-c1cc(ccc1Cl)C(N)=O
CCc1cc(ccc1N(C)C(=O)c1c(F)cccc1Cl)-c1cc(ccc1Cl)C(N)=O
CN(C(=O)c1c(F)cccc1Cl)c1ccc(cc1C(F)(F)F)-c1cc(ccc1Cl)C(N)=O
COc1cc(ccc1N(C)C(=O)c1c(F)cccc1Cl)-c1cc(ccc1Cl)C(N)=O
CCOc1cc(ccc1N(C)C(=O)c1c(F)cccc1Cl)-c1cc(ccc1Cl)C(N)=O
CC(C)Oc1cc(ccc1N(C)C(=O)c1c(F)cccc1Cl)-c1cc(ccc1Cl)C(N)=O
CCCOc1cc(ccc1N(C)C(=O)c1c(F)cccc1Cl)-c1cc(ccc1Cl)C(N)=O
CCCCOc1cc(ccc1N(C)C(=O)c1c(F)cccc1Cl)-c1cc(ccc1Cl)C(N)=O
CN(C(=O)c1c(F)cccc1Cl)c1ccc(cc1OCC(F)(F)F)-c1cc(ccc1Cl)C(N)=O
CN(C(=O)c1c(F)cccc1Cl)c1ccc(cc1)-c1cc(ccc1Cl)C(N)=O
CCN(C(=O)c1c(F)cccc1Cl)c1ccc(cc1)-c1cc(ccc1Cl)C(N)=O
CN(C(=O)c1c(F)cccc1Cl)c1ccc(cc1F)-c1cc(ccc1Cl)C(N)=O
CN(C(=O)c1c(F)cccc1Cl)c1ccc(cc1Cl)-c1cc(ccc1Cl)C(N)=O
CN(C(=O)c1c(F)cccc1Cl)c1ccc(cc1C)-c1cc(ccc1Cl)C(N)=O
CCN(C(=O)c1c(F)cccc1Cl)c1ccc(cc1OC)-c1cc(ccc1Cl)C(N)=O
COCCNC(=O)c1ccc(Cl)c(c1)-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl
Fc1cccc(Cl)c1C(=O)N1CCCc2cc(ccc12)-c1cc(ccc1Cl)C(=O)NCCN1CCOCC1
NC(=O)c1cccc(c1)-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl
COc1ccc(cc1-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl)C(N)=O
NC(=O)c1ccc(F)c(c1)-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl
NC(=O)c1cc(F)cc(c1)-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl
NC(=O)c1cc(ccc1F)-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl
NC(=O)c1cc(c(F)cc1F)-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl
CN(C)C(=O)c1ccc(Cl)c(c1)-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl
OCC(O)CNC(=O)c1ccc(Cl)c(c1)-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl
NC(=O)c1ccc(Cl)c(c1)-c1ccc2N(CCc2c1)C(=O)c1c(F)cccc1Cl
CC1CCc2cc(ccc2N1C(=O)c1c(F)cccc1Cl)-c1cc(ccc1Cl)C(N)=O
NC(=O)c1ccc(Cl)c(c1)-c1ccc2N(CCC(F)(F)c2c1)C(=O)c1c(F)cccc1Cl
NC(=O)c1ccc(Cl)c(c1)-c1ccc2N(CCOc2c1)C(=O)c1c(F)cccc1Cl
CCN(C(=O)c1c(F)cccc1Cl)c1ccc(cc1C(F)(F)F)-c1cc(ccc1Cl)C(N)=O
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(Oc3ccccc3C(F)(F)F)s2)-c2cccc(CN(C)C)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(Oc3ccc(cc3Cl)C(F)(F)F)s2)-c2cccc(c2)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(Oc3ccccc3Cl)s2)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(Oc3ccccc3C(F)(F)F)s2)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(Oc3ccccc3OC)s2)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(Oc3ccc(Cl)cc3)s2)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(Oc3ccc(cc3)C(F)(F)F)s2)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(Oc3ccc(OC)cc3)s2)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(Oc3ccccc3)s2)-c2ccc(Cl)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(Oc3ccccc3)s2)-c2cccc(Cl)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(Oc3ccccc3C(F)(F)F)s2)-c2cccc(Cl)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(Oc3ccccc3C(F)(F)F)s2)-c2cccc(c2)C#N)cc1
CCc1sc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)nc1-c1cc(Cl)ccc1Cl
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(C)s2)-c2cc(Cl)ccc2Cl)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)-c2ccccc2)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)-c2ccccc2)-c2cc(Cl)ccc2Cl)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(Cl)c2)-c2ccc(Cl)cc2OC(F)(F)F)cc1
CS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(Cl)c2)-c2ccc(Cl)cc2OC(F)(F)F)cc1
Cc1cc(NC(=O)Cc2ccc(cc2)S(C)(=O)=O)ccc1-c1ccc(Cl)cc1OC(F)(F)F
CS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(F)c2)-c2ccc(Cl)cc2OC(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccc(F)cc2C#N)cc1 |(-3.74,3.7,;-2.67,3.08,;-2.67,1.54,;-3.73,.92,;-3.74,2.16,;-1.33,.77,;,1.54,;1.33,.77,;1.33,-.77,;2.67,-1.54,;2.66,-3.08,;1.6,-3.7,;4,-3.86,;3.99,-5.4,;5.33,-6.17,;5.32,-7.71,;6.39,-8.33,;3.98,-8.48,;2.65,-7.7,;1.58,-8.32,;2.66,-6.16,;3.98,-10.02,;2.64,-10.78,;2.63,-12.32,;3.96,-13.1,;3.96,-14.33,;5.3,-12.34,;5.31,-10.8,;6.65,-10.03,;7.72,-9.42,;,-1.54,;-1.33,-.77,)|
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2C#N)cc1 |(-3.74,3.7,;-2.67,3.08,;-2.67,1.54,;-3.73,.92,;-3.74,2.16,;-1.33,.77,;,1.54,;1.33,.77,;1.33,-.77,;2.67,-1.54,;2.66,-3.08,;1.6,-3.7,;4,-3.86,;3.99,-5.4,;5.33,-6.17,;5.32,-7.71,;6.39,-8.33,;3.98,-8.48,;2.65,-7.7,;1.58,-8.32,;2.66,-6.16,;3.98,-10.02,;2.64,-10.78,;2.63,-12.32,;3.96,-13.1,;5.3,-12.34,;5.31,-10.8,;6.65,-10.03,;7.72,-9.42,;,-1.54,;-1.33,-.77,)|
NS(=O)(=O)c1ccc(CC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(-3.74,2.16,;-2.67,1.54,;-2.67,2.77,;-3.73,.92,;-1.33,.77,;,1.54,;1.33,.77,;1.33,-.77,;2.67,-1.54,;2.66,-3.08,;1.6,-3.7,;4,-3.86,;3.99,-5.4,;5.33,-6.17,;5.32,-7.71,;6.39,-8.33,;3.98,-8.48,;2.65,-7.7,;1.58,-8.32,;2.66,-6.16,;3.98,-10.02,;2.64,-10.78,;2.63,-12.32,;3.96,-13.1,;5.3,-12.34,;5.31,-10.8,;6.65,-10.03,;7.98,-10.81,;9.05,-10.21,;7.97,-12.05,;9.04,-11.44,;,-1.54,;-1.33,-.77,)|
CS(=O)(=O)c1ccc(CC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(-3.74,2.16,;-2.67,1.54,;-2.67,2.77,;-3.73,.92,;-1.33,.77,;,1.54,;1.33,.77,;1.33,-.77,;2.67,-1.54,;2.66,-3.08,;1.6,-3.7,;4,-3.86,;3.99,-5.4,;5.33,-6.17,;5.32,-7.71,;6.39,-8.33,;3.98,-8.48,;2.65,-7.7,;1.58,-8.32,;2.66,-6.16,;3.98,-10.02,;2.64,-10.78,;2.63,-12.32,;3.96,-13.1,;5.3,-12.34,;5.31,-10.8,;6.65,-10.03,;7.98,-10.81,;9.05,-10.21,;7.97,-12.05,;9.04,-11.44,;,-1.54,;-1.33,-.77,)|
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(-3.74,3.7,;-2.67,3.08,;-2.67,1.54,;-3.73,.92,;-3.74,2.16,;-1.33,.77,;,1.54,;1.33,.77,;1.33,-.77,;2.67,-1.54,;2.66,-3.08,;1.6,-3.7,;4,-3.86,;3.99,-5.4,;5.33,-6.17,;5.32,-7.71,;6.39,-8.33,;3.98,-8.48,;2.65,-7.7,;1.58,-8.32,;2.66,-6.16,;3.98,-10.02,;2.64,-10.78,;2.63,-12.32,;3.96,-13.1,;5.3,-12.34,;5.31,-10.8,;6.65,-10.03,;7.98,-10.81,;9.05,-10.21,;7.97,-12.05,;9.04,-11.44,;,-1.54,;-1.33,-.77,)|
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(C)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(-3.74,3.7,;-2.67,3.08,;-2.67,1.54,;-3.73,.92,;-3.74,2.16,;-1.33,.77,;,1.54,;1.33,.77,;1.33,-.77,;2.67,-1.54,;2.66,-3.08,;1.6,-3.7,;4,-3.86,;3.99,-5.4,;2.66,-6.16,;2.65,-7.7,;1.58,-8.32,;3.98,-8.48,;5.32,-7.71,;6.39,-8.33,;5.33,-6.17,;3.98,-10.02,;2.64,-10.78,;2.63,-12.32,;3.96,-13.1,;5.3,-12.34,;5.31,-10.8,;6.65,-10.03,;7.98,-10.81,;9.05,-10.21,;7.97,-12.05,;9.04,-11.44,;,-1.54,;-1.33,-.77,)|
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(Cl)c(c(c2)C#N)-c2ccccc2OC(F)(F)F)cc1 |(-3.74,3.7,;-2.67,3.08,;-2.67,1.54,;-3.73,.92,;-3.74,2.16,;-1.33,.77,;,1.54,;1.33,.77,;1.33,-.77,;2.67,-1.54,;2.66,-3.08,;1.6,-3.7,;4,-3.86,;3.99,-5.4,;5.33,-6.17,;5.32,-7.71,;6.39,-8.33,;3.98,-8.48,;2.65,-7.7,;2.66,-6.16,;1.32,-8.47,;.25,-9.08,;3.98,-10.02,;2.64,-10.78,;2.63,-12.32,;3.96,-13.1,;5.3,-12.34,;5.31,-10.8,;6.65,-10.03,;7.98,-10.81,;9.05,-10.21,;7.97,-12.05,;9.04,-11.44,;,-1.54,;-1.33,-.77,)|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(-c3ccccc3OC(F)(F)F)c(c2)-c2cncnc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(c2)-c2ccno2)-c2ccccc2OC(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(c2)C(O)=O)-c2ccccc2OC(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(c2)C(C)=O)-c2ccccc2OC(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(-c3ccccc3OC(F)(F)F)c(c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(C)c2)-c2ccccc2OC(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(nc2)-c2ccccc2OC(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2ccccc2OC(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(-c3cccn3C)c(Cl)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(Cl)c2)-c2ncccc2C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(Cl)c2)-c2ccccc2CN(C)C)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(Cl)c2)-c2ccccc2OC(C)C)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(Cl)c2)-c2ccccc2C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(Cl)c2)-c2ccccc2Cl)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(Cl)c2)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2cc(Cl)ccc2Cl)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cccc(n2)-c2cc(Cl)ccc2Cl)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nnc(s2)-c2cc(Cl)ccc2Cl)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(s2)-c2cc(Cl)ccc2Cl)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ncc(s2)-c2cc(Cl)ccc2Cl)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cc(Cl)ccc2Cl)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2csc(n2)-c2cc(Cl)ccc2Cl)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(co2)-c2cc(Cl)ccc2Cl)cc1
Fc1cccc(F)c1C(=O)Nc1ccc2CCCN(c2c1)S(=O)(=O)c1cccs1
CS(=O)(=O)N1CCCc2ccc(NC(=O)c3c(F)cccc3F)cc12
Fc1cccc(F)c1C(=O)Nc1ccc2CCCN(c2c1)S(=O)(=O)c1ccccc1
Cc1ccc(cc1)S(=O)(=O)N1CCCc2ccc(NC(=O)c3c(F)cccc3F)cc12
Fc1ccc(cc1)S(=O)(=O)N1CCCc2ccc(NC(=O)c3c(F)cccc3F)cc12
Fc1ccc(cc1)S(=O)(=O)N1CCc2ccc(NC(=O)c3c(F)cccc3F)cc12
Fc1ccc(cc1)S(=O)(=O)N1CCCCc2ccc(NC(=O)c3c(F)cccc3F)cc12
Fc1ccc(cc1)S(=O)(=O)N1CCc2cc(NC(=O)c3c(F)cccc3F)ccc12
Fc1ccc(cc1)S(=O)(=O)N1CCCc2cc(NC(=O)c3c(F)cccc3F)ccc12
Fc1ccc(cc1)S(=O)(=O)N1CCCCc2cc(NC(=O)c3c(F)cccc3F)ccc12
CC(=O)Nc1ccc2CCCN(c2c1)S(=O)(=O)c1ccc(F)cc1
Fc1ccc(cc1)S(=O)(=O)N1CCCc2ccc(NC(=O)C3CC3)cc12
Fc1ccc(cc1)S(=O)(=O)N1CCCc2ccc(NC(=O)c3ccccc3)cc12
Fc1ccc(cc1)C(=O)Nc1ccc2CCCN(c2c1)S(=O)(=O)c1ccc(F)cc1
Fc1ccc(cc1)S(=O)(=O)N1CCCc2ccc(NC(=O)c3cccc(F)c3)cc12
Fc1ccc(cc1)S(=O)(=O)N1CCCc2ccc(NC(=O)c3ccccc3F)cc12
Cc1ccccc1C(=O)Nc1ccc2CCCN(c2c1)S(=O)(=O)c1ccc(F)cc1
Fc1ccc(cc1)S(=O)(=O)N1CCCc2ccc(NC(=O)c3ccccc3Cl)cc12
Fc1ccc(cc1)S(=O)(=O)N1CCCc2ccc(NC(=O)c3ccno3)cc12
Fc1ccc(cc1)S(=O)(=O)N1CCCc2ccc(NC(=O)c3ccncc3)cc12
Fc1ccc(cc1)S(=O)(=O)N1CCCc2ccc(NC(=O)c3cnccn3)cc12
Fc1ccc(cc1)S(=O)(=O)N1CCCc2ccc(NS(=O)(=O)c3ccccc3)cc12
Fc1cccc(F)c1C(=O)Nc1ccc2CCCN(C(=O)c3ccccc3)c2c1
C[Si](C)(O)c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1ccccc1
CCn1c(SCC(=O)Nc2cccc3ccccc23)nnc1C1Cc2ccccc2C1
CCn1c(OCC(=O)Nc2cccc3ccccc23)nnc1C1Cc2ccccc2C1
CCn1c(CCC(=O)Nc2cccc3ccccc23)nnc1C1Cc2ccccc2C1
CCn1c(nnc1C1Cc2ccccc2C1)C(C)CC(=O)Nc1cccc2ccccc12
CCn1c(CC(C)C(=O)Nc2cccc3ccccc23)nnc1C1Cc2ccccc2C1
CCn1c(nnc1C1Cc2ccccc2C1)C(O)CC(=O)Nc1cccc2ccccc12
CCn1c(CCC(=O)Nc2cccc3ccccc23)nnc1C1CCCCC1
CCn1c(CCC(=O)Nc2cccc3ccccc23)nnc1CC1CCCCC1
CCn1c(nnc1CCC(=O)Nc2cccc3c2cccc3)CCC4CCCCC4
CCn1c(CCC(C)C)nnc1CCC(=O)Nc1cccc2ccccc12
CCn1c(CCC(=O)Nc2cccc3ccccc23)nnc1CCC(C)(C)C
CCn1c(CCC(=O)Nc2cccc3ccccc23)nnc1CCc1ccccc1
CCn1c(CCC2CCCCC2)nnc1CCC(=O)Nc1cccc(Cl)c1C
CCn1c(CCC2CCCCC2)nnc1CCC(=O)Nc1ccc(C)cc1C
CCn1c(CCC2CCCCC2)nnc1CCC(=O)Nc1cc(C)cc(C)c1
Cc1ccc(NC(=O)CCc2nnc(CCC3CCCCC3)n2C2CC2)c(C)c1
Cc1ccc(NC(=O)CCc2nnc(CCC3CCCCC3)n2C2CCC2)c(C)c1
Cc1ccc(NC(=O)CCc2nnc(CCC3CCCCC3)n2C2CC2(F)F)c(C)c1
CCC(C)CCc1nnc(CCC(=O)Nc2ccc(C)cc2C)n1C1CC1
CC(C)CCCc1nnc(CCC(=O)Nc2ccc(C)cc2C)n1C1CC1
Cc1ccc(NC(=O)CCc2nnc(CCCC(C)(C)C)n2C2CC2)c(C)c1
CC(C)Cc1ccc(cc1)-c1nnc(CCC(=O)Nc2ccc(C)cc2C)n1C1CC1
CC(C)Cc1cc(no1)-c1nnc(CCC(=O)Nc2ccc(C)cc2C)n1C1CC1
CC(C)C[C@H]1C[C@@H](C1)c1nnc(CCC(=O)Nc2ccc(C)cc2C)n1C1CC1 |r,wU:4.3,wD:6.8,(9.15,-15.02,;8.56,-13.94,;7.33,-13.91,;9.36,-12.63,;8.62,-11.28,;7.15,-10.85,;7.6,-9.42,;9.06,-9.8,;6.98,-8.01,;7.75,-6.68,;6.72,-5.53,;5.33,-6.17,;4,-5.4,;4,-3.86,;2.66,-3.08,;1.6,-3.7,;2.67,-1.54,;1.33,-.77,;,-1.54,;-1.33,-.77,;-1.33,.77,;-2.4,1.39,;,1.54,;1.33,.77,;2.4,1.39,;5.47,-7.69,;4.32,-8.72,;2.91,-9.1,;4.04,-10.15,)|
CC(C)C[C@H]1C[C@H](C1)c1nnc(CCC(=O)Nc2ccc(C)cc2C)n1C1CC1 |r,wD:4.3,6.8,(9.15,-15.02,;8.56,-13.94,;7.33,-13.91,;9.36,-12.63,;8.62,-11.28,;9.06,-9.8,;7.6,-9.42,;7.15,-10.85,;6.98,-8.01,;7.75,-6.68,;6.72,-5.53,;5.33,-6.17,;4,-5.4,;4,-3.86,;2.66,-3.08,;1.6,-3.7,;2.67,-1.54,;1.33,-.77,;,-1.54,;-1.33,-.77,;-1.33,.77,;-2.4,1.39,;,1.54,;1.33,.77,;2.4,1.39,;5.47,-7.69,;4.32,-8.72,;2.91,-9.1,;4.04,-10.15,)|
CC(C)C[C@H]1C[C@H](C1)c1nnc([C@H]2CCN(C)C[C@@H]2C(=O)Nc2ccc(C)cc2C)n1C1CC1 |r,wU:18.20,4.3,6.8,wD:12.12,(-12.25,.44,;-11.01,.47,;-10.37,-.59,;-10.27,1.82,;-8.74,1.85,;-7.67,2.96,;-6.62,1.89,;-7.63,.79,;-5.09,2.05,;-4.31,3.38,;-2.81,3.06,;-2.67,1.54,;-1.33,.77,;-1.33,-.77,;,-1.54,;1.33,-.77,;2.4,-1.39,;1.33,.77,;,1.54,;-0,3.08,;1.06,3.7,;-1.34,3.85,;-1.34,5.39,;-.01,6.16,;-.01,7.7,;-1.34,8.47,;-1.34,9.7,;-2.68,7.7,;-2.68,6.16,;-3.74,5.54,;-4.06,.91,;-4.37,-.6,;-4,-2.01,;-5.47,-1.56,)|
CC(C)C[C@H]1C[C@H](C1)c1nnc([C@H]2C[C@H](O)C[C@@H]2C(=O)Nc2ccc(C)cc2C)n1C1CC1 |r,wU:4.3,6.8,12.12,wD:17.19,14.15,(2.36,7.33,;2.68,6.14,;1.81,5.27,;4.17,5.74,;4.56,4.26,;5.9,3.48,;5.11,2.21,;3.79,2.92,;5.62,.75,;7.1,.32,;7.14,-1.22,;5.7,-1.71,;5.38,-3.22,;6.42,-4.36,;5.65,-5.7,;6.15,-6.82,;4.14,-5.38,;4,-3.86,;2.66,-3.08,;2.67,-1.85,;1.33,-3.85,;-.01,-3.08,;0,-1.54,;-1.33,-.76,;-2.67,-1.53,;-3.73,-.91,;-2.67,-3.07,;-1.34,-3.84,;-1.35,-5.07,;4.75,-.52,;3.21,-.57,;1.93,-1.26,;2.03,.28,)|
CNS(=O)(=O)c1cccc(c1)-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl
NS(=O)(=O)c1cccc(c1)-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl
NC(=O)c1ccccc1-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl
Fc1cc(cc(c1)-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl)C(=O)N1CCOCC1
Fc1ccc(cc1-c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl)C(=O)N1CCCC1
Cc1cc(ccc1-c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1cccc(Cl)c1)C1(CC1)C(O)=O
Cc1cc(ccc1-c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1cccc2n(C)ccc12)C1(CC1)C(O)=O
Cc1cc(CO)ccc1-c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1cccc(Cl)c1
Cc1cc(CO)ccc1-c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1cccc2n(C)ccc12
Cc1cc2nccn2cc1-c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1cccc(Cl)c1
Cc1cc2nccn2cc1-c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1cccc2n(C)ccc12
Cc1cc(O)ccc1-c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1cccc(Cl)c1
Cc1cc(O)ccc1-c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1cccc2n(C)ccc12
CNC(=O)c1ccc(F)c(c1)-c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1cccc(Cl)c1
CNC(=O)c1ccc(F)c(c1)-c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1cccc2n(C)ccc12
CNC(=O)c1cccc(c1)-c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1cccc(Cl)c1
CNC(=O)c1cccc(c1)-c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1cccc2n(C)ccc12
NC(=O)c1cccc(c1)-c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1cccc(Cl)c1
Cn1ccc2c(cccc12)S(=O)(=O)N(CC(F)(F)F)c1ccc(cc1)-c1cccc(c1)C(N)=O
NC(=O)c1ccc(Cl)c(c1)-c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1cccc(Cl)c1
OC(c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1cccc(Cl)c1)(C(F)(F)F)C(F)(F)F
Cn1ccc2c(cccc12)S(=O)(=O)N(CC(F)(F)F)c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
Cc1ccc(cc1C)S(=O)(=O)N(CC(F)(F)F)c1ccc2N(CCCc2c1)C(=O)c1c(F)cccc1Cl
Cn1ccc2c1cccc2S(=O)(=O)N(CC(F)(F)F)c3ccc4c(c3)CCCN4C(=O)c5cccs5
Cc1ccc(cc1C)S(=O)(=O)N(CC(F)(F)F)c1ccc2N(CCCc2c1)C(=O)c1cccs1
Cc1ccc(cc1C)S(=O)(=O)Nc1ccc2N(CCCc2c1)C(=O)c1cccs1
Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc1ccc(F)cc1F)c1cccc(c1)C(F)(F)F
Cc1ccc(cc1)S(=O)(=O)N(CC(O)=O)c1cccc(c1)C(F)(F)F
Cc1csc(NC(=O)CN(c2cccc(c2)C(F)(F)F)S(=O)(=O)c2ccc(C)cc2)n1
Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc1ccc(OCc2ccccc2)cc1)c1cccc(c1)C(F)(F)F
Cc1ccc(cc1)S(=O)(=O)N(CC(=O)NCc1ccc(F)cc1)c1cccc(c1)C(F)(F)F
CC(=O)N1CCN(CC1)C(=O)CN(c1cccc(c1)C(F)(F)F)S(=O)(=O)c1ccc(C)cc1
Cc1ccc(cc1)S(=O)(=O)N(CC(=O)NCc1ccc(O)cc1)c1cccc(c1)C(F)(F)F
Cc1ccc(cc1)S(=O)(=O)N(CC(=O)NCc1ccncc1)c1cccc(c1)C(F)(F)F
COC(=O)c1ccc(CNC(=O)CN(c2cccc(c2)C(F)(F)F)S(=O)(=O)c2ccc(C)cc2)cc1
Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc1ccc(F)cc1)c1cccc(c1)C(F)(F)F
COC(=O)c1ccc(NC(=O)CN(c2cccc(c2)C(F)(F)F)S(=O)(=O)c2ccc(C)cc2)cc1
Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc1ccc(cc1)C#N)c1cccc(c1)C(F)(F)F
Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc1ccc(cc1)C(N)=O)c1cccc(c1)C(F)(F)F
CC(=O)c1ccc(NC(=O)CN(c2cccc(c2)C(F)(F)F)S(=O)(=O)c2ccc(C)cc2)cc1
Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc1ccc(O)cc1)c1cccc(c1)C(F)(F)F
COc1ccc(NC(=O)CN(c2cccc(c2)C(F)(F)F)S(=O)(=O)c2ccc(C)cc2)cc1OC
Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)c1cccc(c1)C(F)(F)F
Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc1ccc(cc1)C#N)c1ccc(cc1)C(F)(F)F
Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc1ccc(cc1)C#N)c1ccc(cc1)C#N
Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc1ccc(cc1)C#N)c1ccc(F)cc1
Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc1ccc(cc1)C#N)c1ccc(Cl)c(Cl)c1
Cc1ccc(cc1)N(CC(=O)Nc1ccc(cc1)C#N)S(=O)(=O)c1ccc(F)cc1
Cc1ccc(cc1)N(CC(=O)Nc1ccc(cc1)C#N)S(=O)(=O)Cc1ccc(F)cc1
Cc1ccc(cc1)N(CC(=O)Nc1ccc(cc1)C#N)S(=O)(=O)Cc1ccccc1
COC(=O)c1ccccc1NC(=O)CN(c1cccc(c1)C(F)(F)F)S(=O)(=O)c1ccc(C)cc1
COC(=O)c1cccc(NC(=O)CN(c2cccc(c2)C(F)(F)F)S(=O)(=O)c2ccc(C)cc2)c1
Cc1ccc(cc1)S(=O)(=O)N(CC(=O)NC1CCCCC1)c1cccc(c1)C(F)(F)F
Cc1ccc(CNC(=O)CN(c2cccc(c2)C(F)(F)F)S(=O)(=O)c2ccc(C)cc2)cc1
OC(=O)c1ccc(cc1)-n1nc(Sc2c(Cl)cccc2Cl)c2cc(ccc12)C(=O)N1CC(F)(F)C1
CN(C)C(=O)c1ccc2c(Oc3c(Cl)cccc3Cl)nn(-c3ccc(cc3)C(O)=O)c2c1
OC(=O)c1cc(F)c(c(F)c1)-n1nc(Oc2c(Cl)cccc2Cl)c2ccccc12 |(5.25,-19.06,;6.29,-20.19,;7.81,-19.94,;5.75,-21.64,;6.74,-22.82,;6.19,-24.27,;7.17,-25.45,;4.68,-24.52,;3.69,-23.34,;2.18,-23.59,;4.24,-21.89,;4.14,-25.97,;4.99,-27.25,;4.04,-28.45,;4.44,-29.94,;5.93,-30.32,;6.35,-31.81,;5.27,-32.91,;7.84,-32.19,;8.92,-31.09,;8.5,-29.61,;7.01,-29.22,;6.61,-27.74,;2.58,-27.92,;1.22,-28.63,;-.08,-27.81,;-.02,-26.27,;1.36,-25.56,;2.65,-26.38,)|
OC(=O)[C@H]1CC[C@H](CC1)n1nc(Oc2c(Cl)cccc2Cl)c2ccccc12 |r,wU:3.2,6.9,(26.9,-35.1,;25.39,-35.4,;24.38,-34.25,;24.91,-36.86,;25.92,-38.02,;25.43,-39.47,;23.92,-39.78,;22.9,-38.63,;23.4,-37.16,;23.43,-41.24,;24.32,-42.49,;23.4,-43.73,;23.86,-45.2,;25.37,-45.54,;26.41,-44.4,;25.95,-42.93,;27.91,-44.74,;28.38,-46.21,;27.33,-47.34,;25.83,-47.01,;24.78,-48.14,;21.94,-43.24,;20.61,-44,;19.28,-43.22,;19.29,-41.68,;20.63,-40.92,;21.96,-41.7,)|
CN(Cc1ccccc1)C(=O)c1ccc2n(nc(Sc3c(Cl)cccc3Cl)c2c1)-c1ccc(cc1)C(O)=O
OC(=O)c1ccc(cc1)-n1nc(Cc2c(Cl)cccc2Cl)c2ccccc12
CN(C)C(=O)c1ccc2n(nc(Oc3c(C)cccc3Cl)c2c1)-c1ccc(cc1)C(O)=O
OC(=O)[C@H]1CC[C@@H](CC1)n1nc(Oc2c(Cl)cccc2Cl)c2ccccc12 |r,wU:3.2,wD:6.9,(37.03,-35.92,;35.52,-36.23,;34.5,-35.07,;35.03,-37.68,;36.05,-38.84,;35.56,-40.3,;34.05,-40.6,;33.03,-39.45,;33.52,-37.99,;33.55,-42.06,;34.45,-43.32,;33.53,-44.55,;33.99,-46.02,;35.49,-46.36,;36.54,-45.23,;36.07,-43.76,;38.04,-45.57,;38.5,-47.03,;37.46,-48.16,;35.95,-47.83,;34.91,-48.96,;32.07,-44.07,;30.73,-44.82,;29.4,-44.04,;29.42,-42.5,;30.76,-41.74,;32.08,-42.53,)|
CN(C)C(=O)c1ccc2n(nc(Oc3c(Cl)cccc3Cl)c2c1)-c1ccc(cc1)C(O)=O
CN(C)C(=O)c1ccc2c(nn(C(=O)c3c(Cl)cccc3Cl)c2c1)-c1ccc(cc1)C(O)=O
CCN(C)C(=O)c1ccc2n(nc(Sc3c(Cl)cccc3Cl)c2c1)-c1ccc(cc1)C(O)=O
CS(=O)(=O)c1ccc2n(nc(Oc3c(Cl)cccc3Cl)c2c1)-c1ccc(cc1)C(O)=O
OC(=O)c1ccc(cc1)-n1nc(Oc2c(Cl)cccc2Cl)c2cccnc12
OC(=O)c1ccc(cn1)-n1nc(Oc2c(Cl)cccc2Cl)c2ccccc12
CCc1nn(C)c(CC)c1Oc1nn(-c2ccc(cc2)C(O)=O)c2ccccc12
CN(C)C(=O)c1ccc2n(nc(Oc3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1)C(O)=O
OC(=O)c1ccc(cc1)-n1nc(Oc2c(Cl)cccc2Cl)c2ccccc12
OC(=O)c1ccc(cc1)-n1nc(c2ccccc12)S(=O)(=O)c1c(Cl)cccc1Cl
CN(C)C(=O)c1ccc2n(nc([S+]([O-])c3c(Cl)cccc3Cl)c2c1)-c1ccc(cc1)C(O)=O
OC(=O)c1ccc(cc1)-n1nc([S+]([O-])c2c(Cl)cccc2Cl)c2ccccc12
OC(=O)c1ccc(cc1)-n1nc(Sc2c(Cl)cccc2Cl)c2ccccc12
CN(c1nn(-c2ccc(cc2)C(O)=O)c2ccccc12)c1c(Cl)cccc1Cl
OC(=O)c1ccc(cc1)-n1nc(Nc2c(Cl)cccc2Cl)c2ccccc12
Cc1noc(C)c1[C@H](O)c1cc2cc(CC(=O)N[C@@H](c3ccccc3)c3ccc(C)cc3C)ccc2o1 |r|
CN(C)C(=O)c1ccc2n(nc(Sc3ccccc3)c2c1)-c1ccc(cc1)C(O)=O
CN(C)C(=O)c1ccc2n(nc(Sc3c(F)cccc3Cl)c2c1)-c1ccc(cc1)C(O)=O
CN(C)C(=O)c1ccc2n(nc(Sc3cccc(Cl)c3Cl)c2c1)-c1ccc(cc1)C(O)=O
CN(C)C(=O)c1ccc2n(nc(Sc3ccc(Cl)cc3Cl)c2c1)-c1ccc(cc1)C(O)=O
CN(C)C(=O)c1ccc2n(nc(Sc3cc(Cl)ccc3Cl)c2c1)-c1ccc(cc1)C(O)=O
CN(CCO)C(=O)c1ccc2n(nc(Sc3c(Cl)cccc3Cl)c2c1)-c1ccc(cc1)C(O)=O
OC(=O)c1ccc(cc1)-n1nc(Sc2c(Cl)cccc2Cl)c2cc(ccc12)C(=O)N1CCCC1
OC(=O)c1ccc(cc1)-n1nc(Sc2c(Cl)cccc2Cl)c2cc(ccc12)C(=O)N1CCOCC1
Cc1cccc2c(Oc3c(Cl)cccc3Cl)nn(-c3ccc(cc3)C(O)=O)c12
OC(=O)c1ccc(cc1)-n1nc(Oc2c(Cl)cccc2Cl)c2cc(ccc12)C#N
OC(=O)c1ccc(c(F)c1)-n1nc(Oc2c(Cl)cccc2Cl)c2ccccc12
CN(C)C(=O)c1ccc2n(nc(Nc3c(Cl)cccc3Cl)c2c1)-c1ccc(cc1)C(O)=O
Cc1cc(ccc1-n1nc(Oc2c(Cl)cccc2Cl)c2ccccc12)C(O)=O
Cc1cccc2n(nc(Oc3c(Cl)cccc3Cl)c12)-c1ccc(cc1)C(O)=O
CN(C)C(=O)c1ccc2n(nc(c2c1)S(=O)(=O)c1c(Cl)cccc1Cl)-c1ccc(cc1)C(O)=O
CN(C)C(=O)c1ccc2n(nc(Sc3c(Cl)cccc3Cl)c2c1)-c1ccc(cc1)C(O)=O
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2Cl)c2ccccc12
CN(C)C(=O)c1ccc2n(nc(Sc3c(C)cccc3C)c2c1)-c1ccc(cc1)C(O)=O
CN(C)C(=O)c1ccc2n(nc(Sc3c(C)cc(C)cc3C)c2c1)-c1ccc(cc1)C(O)=O
CNC(=O)c1ccc2n(nc(Sc3c(Cl)cccc3Cl)c2c1)-c1ccc(cc1)C(O)=O
OC(=O)c1ccc(cc1)-n1nc(Sc2c(Cl)cccc2Cl)c2cc(ccc12)C(=O)N1CCC1
CN1CCN(CC1)C(=O)c1ccc2n(nc(Sc3c(Cl)cccc3Cl)c2c1)-c1ccc(cc1)C(O)=O
OC(=O)c1ccc(cc1)-n1nc(Oc2c(Cl)cccc2Cl)c2cccc(F)c12
OC(=O)c1ccc(cc1)-n1nc(Oc2c(Cl)cccc2Cl)c2ncccc12
Clc1cccc(Cl)c1Oc1n[nH]c2ccccc12
CN(C)C(=O)c1ccc2n(nc(Sc3ccccc3C)c2c1)-c1ccc(cc1)C(O)=O
OC(=O)c1ccc(cc1)-n1nc(Oc2c(Cl)cccc2Cl)c2c(F)cccc12
OC(=O)c1ccc(nc1)-n1nc(Oc2c(Cl)cccc2Cl)c2ccccc12
CCCC1=N[C@@H](CCCCN2C[C@H](Cc3ccccc3)N(CCCC3CCCC3)C2=S)CN1 |r,t:3|
C\C=C\C1=N[C@@H](CCCCN2C[C@H](Cc3ccccc3)N(CCc3ccccc3)C2=S)CN1 |r,t:3|
CCCC1=N[C@@H](CCCCN2C[C@H](Cc3ccccc3)N(CC3CCC(C)CC3)C2=S)CN1 |r,wD:12.12,5.5,t:3,(13.24,-47.1,;14.22,-45.9,;15.74,-46.15,;16.71,-44.95,;18.24,-45.04,;18.8,-43.59,;20.29,-43.2,;21.37,-44.29,;22.86,-43.89,;23.95,-44.98,;25.44,-44.59,;25.99,-43.15,;27.53,-43.23,;28.5,-42.03,;27.94,-40.59,;28.91,-39.4,;28.36,-37.96,;26.84,-37.72,;25.87,-38.93,;26.43,-40.36,;27.93,-44.72,;29.36,-45.28,;30.7,-44.51,;32.03,-45.29,;33.36,-44.53,;33.37,-42.99,;34.71,-42.22,;32.04,-42.21,;30.69,-42.97,;26.63,-45.56,;26.55,-47.09,;17.61,-42.63,;16.31,-43.46,)|
Fc1ccc(CC2=N[C@@H](CCCCN3C[C@H](Cc4ccccc4)N(CCc4ccccc4)C3=S)CN2)cc1 |r,t:6|
Cc1cccc(CC2=N[C@@H](CCCCN3C[C@H](Cc4ccccc4)N(CCc4ccccc4)C3=S)CN2)c1 |r,t:7|
S=C1N(CCCC[C@H]2CNC(CCC3CCCC3)=N2)C[C@H](Cc2ccccc2)N1CCc1ccccc1 |r,c:18|
C=CCC1=N[C@@H](CCCCN2C[C@H](Cc3ccccc3)N(CCc3ccccc3)C2=S)CN1 |r,t:3|
CC(CC1=N[C@@H](CCCCN2C[C@H](Cc3ccccc3)N(CCc3ccccc3)C2=S)CN1)c1ccccc1 |r,t:3|
Fc1cccc(CC2=N[C@@H](CCCCN3C[C@H](Cc4ccccc4)N(CCc4ccccc4)C3=S)CN2)c1 |r,t:7|
CCCC1=N[C@@H](CCCCN2C[C@H](Cc3ccccc3)N(CCC3C4CC5CC(C4)CC3C5)C2=S)CN1 |r,wU:12.12,wD:5.5,t:3,TLB:22:23:25:29.28.27,THB:27:26:23:29.28.30,27:28:23:25.26.32,30:31:25:29.28.27,30:28:25:23.32.31,(22.13,-39.35,;20.66,-39.83,;20.34,-41.33,;18.87,-41.81,;17.63,-40.9,;16.38,-41.81,;14.92,-41.33,;14.6,-39.82,;13.13,-39.35,;12.82,-37.84,;11.35,-37.36,;10.88,-35.9,;9.34,-35.89,;8.44,-34.64,;9.19,-33.3,;10.72,-33.28,;11.47,-31.93,;10.67,-30.61,;9.12,-30.64,;8.39,-31.99,;8.86,-37.36,;7.4,-37.83,;6.26,-36.8,;4.79,-37.27,;4.17,-38.66,;4.53,-40.17,;3.3,-38.92,;1.82,-38.87,;1.4,-37.5,;2.59,-38.59,;2.04,-36.13,;3.56,-36.21,;3.85,-37.62,;10.11,-38.26,;10.11,-39.8,;16.85,-43.27,;18.39,-43.27,)|
CCCC1=N[C@@H](CCCCN2C[C@H](Cc3ccccc3)N(CCC3CC4CCC3C4)C2=S)CN1 |r,t:3,THB:22:23:29:26.27|
CCCC1=N[C@@H](CCCCN2C[C@H](N(CCc3ccccc3)C2=S)C(C)(C)C)CN1 |r,t:3|
CCCC[C@H]1CN(CCCC[C@H]2CNC(CCC)=N2)C(=S)N1CCc1ccccc1 |r,c:17|
COc1cccc(CC2=N[C@@H](CCCCN3C[C@H](Cc4ccccc4)N(CCc4ccccc4)C3=S)CN2)c1 |r,t:8|
S=C1N(CCCC[C@H]2CNC(CC3CCCCC3)=N2)C[C@H](Cc2ccccc2)N1CCc1ccccc1 |r,c:18|
COc1nc2ccc(cc2c(Cl)c1-c1cnc(nc1)C#N)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F
Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2nc(Cl)c(cc2c1)-c1ccccc1
Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2nc(Cl)c(-c3ccccc3)c(Cl)c2c1
COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cncn1C)c1ccc(Cl)cc1
COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C#N)C(O)(c1cncn1C)c1ccc(Cl)cc1
COc1nc2ccc(cc2c(Cl)c1Cc1ccc(F)cc1)C(O)(c1cncn1C)c1ccc(Cl)cc1
COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F
COc1nc2ccc(cc2c(Cl)c1Cc1ccc(F)cc1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F
CCN(CC)c1nc2ccc(cc2c(Cl)c1-c1ccccc1)C(O)(c1cncn1C)c1ccncc1
CN(CCO)c1nc2ccc(cc2c(Cl)c1-c1ccccc1)C(O)(c1cncn1C)c1ccncc1
CN(C)c1c(c(Cl)nc2ccc(cc12)C(O)(c1cncn1C)c1ccncc1)-c1ccccc1
CN(C)c1nc2ccc(cc2c(Cl)c1-c1ccccc1)C(O)(c1cncn1C)c1ccncc1
COc1c(-c2ccccc2)c(nc2ccc(cc12)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F)C(F)(F)F
COc1nc2ccc(cc2c(Cl)c1Cc1ccccc1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F
COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F
COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cncn1C)c1ccc(Cl)cc1
COc1nc2ccc(cc2c(Cl)c1-c1ccccc1)C(O)(c1cncn1C)c1ccncc1
Cn1cncc1C(O)(c1ccncc1)c1ccc2nc(Cl)c(-c3ccccc3)c(Cl)c2c1
Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2nc(c(-c3ccccc3)c(c2c1)C(F)(F)F)C(F)(F)F
Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2nc(C#N)c(-c3ccccc3)c(C#N)c2c1
Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2nc(C#N)c(-c3ccccc3)c(Cl)c2c1
COc1nc2ccc(cc2c(Cl)c1-c1ccccc1)C(O)(c1cncn1C)c1ccc(Cl)cc1
Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2ncc(-c3ccccc3)c(Cl)c2c1
COc1nc2ccc(cc2c(Cl)c1-c1ccc(cc1)S(C)(=O)=O)C(O)(c1cncn1C)c1ccc(nc1)C(F)(F)F
CNc1c(c(Cl)nc2ccc(cc12)C(O)(c1cncn1C)c1ccncc1)-c1ccccc1
Cn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2nc(c(-c3ccccc3)c(Cl)c2c1)C(F)(F)F
COc1nc2ccc(cc2c(OC)c1-c1ccccc1)C(O)(c1cncn1C)c1ccc(Cl)cc1
Cn1cncc1C(O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(N3CCC3)c(-c3ccccc3)c(Cl)c2c1
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CC2)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12)C(F)(F)F |r|
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12 |r,wU:27.28,wD:29.33,(8.76,1.15,;7.67,.06,;6.19,.46,;7.28,1.55,;8.07,-1.42,;6.98,-2.51,;6.59,-4,;8.07,-3.6,;5.5,-2.11,;5.1,-.63,;3.61,-.23,;2.52,-1.32,;1.03,-.92,;.56,.55,;-.98,.55,;-1.46,-.92,;-.21,-1.82,;-.21,-3.36,;-1.55,-4.13,;-2.88,-3.36,;-4.21,-4.13,;-4.21,-5.67,;-2.88,-6.44,;-1.55,-5.67,;-2.07,1.64,;-1.67,3.12,;-3.56,1.24,;-4.65,2.33,;-6.19,2.33,;-6.19,3.87,;-4.65,3.87,;-7.28,4.96,;-6.88,6.44,;-8.76,4.56,;2.92,-2.8,;1.83,-3.89,;2.23,-5.38,;3.72,-5.78,;4.81,-4.69,;4.41,-3.2,)|
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CCOCC2)c2ccccc12
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C2CCCCC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
CC(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(C(F)F)c1Cl |r,wU:26.27,wD:28.32,(47.02,-5.86,;46.22,-7.17,;46.96,-8.52,;44.68,-7.14,;43.87,-8.45,;45.2,-9.21,;43.87,-9.98,;42.33,-8.41,;41.52,-9.73,;39.98,-9.68,;39.25,-8.32,;37.71,-8.28,;36.84,-7,;35.37,-7.44,;35.32,-8.98,;36.78,-9.49,;37.21,-10.97,;36.14,-12.09,;34.65,-11.72,;33.59,-12.83,;34.02,-14.31,;35.52,-14.68,;36.59,-13.56,;34.02,-6.67,;34.02,-5.13,;32.69,-7.44,;31.35,-6.67,;29.86,-7.07,;29.46,-5.59,;30.95,-5.19,;28.13,-4.81,;26.79,-5.59,;28.12,-3.27,;40.06,-7.01,;39.32,-5.66,;40.13,-4.35,;37.78,-5.62,;41.59,-7.06,;42.39,-5.75,)|
CC(C)(C)NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O |r,wU:32.35,wD:34.40,(3.57,-7.2,;4.66,-6.11,;6.15,-6.51,;5.06,-7.6,;4.26,-4.62,;5.35,-3.53,;6.84,-3.93,;4.95,-2.05,;3.46,-1.65,;3.07,-.16,;4.16,.93,;5.64,.53,;6.04,-.96,;6.73,1.62,;6.33,3.11,;7.82,.53,;8.22,2.02,;1.58,.24,;1.1,1.7,;-.44,1.7,;-.91,.24,;.33,-.67,;.33,-2.21,;-1,-2.98,;-2.33,-2.21,;-3.67,-2.98,;-3.67,-4.52,;-2.33,-5.29,;-1,-4.52,;-1.53,2.79,;-1.13,4.28,;-3.01,2.39,;-4.1,3.48,;-5.64,3.48,;-5.64,5.02,;-4.1,5.02,;-6.73,6.11,;-8.22,5.71,;-6.33,7.6,)|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CC(F)(F)C2)C(=O)NCC(C)(C)O)c2ccccc12)C(F)(F)F |r|
CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c(Cl)c1C(F)F)S(=O)(=O)NC(C)(C)C
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2-c2cccc(F)c2)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2CCCCc12 |r,wU:27.28,wD:29.33,(8.76,1.15,;7.67,.06,;6.19,.46,;7.28,1.55,;8.07,-1.42,;6.98,-2.51,;6.59,-4,;8.07,-3.6,;5.5,-2.11,;5.1,-.63,;3.61,-.23,;2.52,-1.32,;1.03,-.92,;.56,.55,;-.98,.55,;-1.46,-.92,;-.21,-1.82,;-.21,-3.36,;-1.55,-4.13,;-2.88,-3.36,;-4.21,-4.13,;-4.21,-5.67,;-2.88,-6.44,;-1.55,-5.67,;-2.07,1.64,;-1.67,3.12,;-3.56,1.24,;-4.65,2.33,;-6.19,2.33,;-6.19,3.87,;-4.65,3.87,;-7.28,4.96,;-6.88,6.44,;-8.76,4.56,;2.92,-2.8,;1.83,-3.89,;2.23,-5.38,;3.72,-5.78,;4.81,-4.69,;4.41,-3.2,)|
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(Cl)c1Cl |r,wU:27.28,wD:29.33,(8.76,1.15,;7.67,.06,;6.19,.46,;7.28,1.55,;8.07,-1.42,;6.98,-2.51,;6.59,-4,;8.07,-3.6,;5.5,-2.11,;5.1,-.63,;3.61,-.23,;2.52,-1.32,;1.03,-.92,;.56,.55,;-.98,.55,;-1.46,-.92,;-.21,-1.82,;-.21,-3.36,;-1.55,-4.13,;-2.88,-3.36,;-4.21,-4.13,;-4.21,-5.67,;-2.88,-6.44,;-1.55,-5.67,;-2.07,1.64,;-1.67,3.12,;-3.56,1.24,;-4.65,2.33,;-6.19,2.33,;-6.19,3.87,;-4.65,3.87,;-7.28,4.96,;-6.88,6.44,;-8.76,4.56,;2.92,-2.8,;1.83,-3.89,;4.41,-3.2,;4.81,-4.69,)|
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12)C(F)(F)F |r,wU:25.26,wD:27.31,1.0,(22.5,-20.14,;21.77,-18.79,;20.23,-18.76,;19.42,-20.07,;20.75,-20.84,;19.42,-21.61,;17.88,-20.04,;17.07,-21.36,;15.53,-21.3,;14.8,-19.95,;13.26,-19.91,;12.39,-18.63,;10.92,-19.07,;10.87,-20.61,;12.33,-21.12,;12.76,-22.6,;11.69,-23.72,;10.2,-23.35,;9.14,-24.46,;9.57,-25.94,;11.07,-26.31,;12.14,-25.19,;9.57,-18.3,;9.57,-16.75,;8.23,-19.07,;6.9,-18.3,;5.41,-18.7,;5.01,-17.21,;6.5,-16.81,;3.67,-16.44,;2.34,-17.21,;3.67,-14.9,;15.6,-18.64,;14.87,-17.3,;15.67,-15.99,;17.21,-16.03,;17.94,-17.38,;17.14,-18.68,;22.57,-17.48,;24.11,-17.52,;21.84,-16.13,;23.33,-16.14,)|
CC(C)(O)CNC(=O)c1nc(CC2CCCCC2)c(s1)-c1ccc(c2ccccc12)S(=O)(=O)NC1(CC1)C#N
CC(C)(C)NS(=O)(=O)c1ncc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12
CC(C)(C)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O |r,wU:29.32,wD:31.37,(4.46,-5.78,;5.55,-4.69,;7.04,-5.09,;5.95,-6.18,;5.15,-3.2,;3.66,-2.8,;3.27,-1.32,;4.35,-.23,;5.84,-.63,;6.24,-2.11,;6.93,.46,;8.02,-.63,;8.02,1.55,;6.53,1.95,;1.78,-.92,;1.3,.55,;-.24,.55,;-.71,-.92,;.53,-1.82,;.53,-3.36,;-.8,-4.13,;-2.14,-3.36,;-3.47,-4.13,;-3.47,-5.67,;-2.14,-6.44,;-.8,-5.67,;-1.33,1.64,;-.93,3.12,;-2.81,1.24,;-3.9,2.33,;-5.44,2.33,;-5.44,3.87,;-3.9,3.87,;-6.53,4.96,;-6.13,6.44,;-8.02,4.56,)|
CC(C)(C)c1cc(cc(c1)C(O)(C(F)(F)F)C(F)(F)F)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O |r,wU:35.37,wD:37.42,(39.13,-12.67,;39.93,-11.36,;41.47,-11.4,;40.7,-12.68,;39.21,-10.01,;37.67,-9.96,;36.93,-8.6,;37.74,-7.3,;39.28,-7.33,;40.01,-8.69,;40.07,-6.02,;40.84,-4.68,;41.61,-6.06,;42.36,-7.41,;42.42,-4.74,;43.1,-5.65,;39.34,-4.66,;40.14,-3.35,;37.8,-4.62,;38.55,-3.32,;35.4,-8.56,;34.53,-7.28,;33.05,-7.72,;33.01,-9.26,;34.46,-9.77,;34.89,-11.25,;33.83,-12.37,;32.34,-12,;31.28,-13.11,;31.71,-14.59,;33.21,-14.96,;34.28,-13.84,;31.71,-6.95,;31.71,-5.41,;30.38,-7.72,;29.04,-6.95,;27.55,-7.36,;27.15,-5.87,;28.64,-5.47,;25.82,-5.09,;24.48,-5.87,;25.82,-3.55,)|
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(Cl)c1 |r,wU:27.28,wD:29.33,(72.21,-6.55,;70.87,-5.78,;70.87,-7.32,;71.68,-4.47,;69.33,-5.75,;68.52,-7.06,;69.86,-7.83,;68.52,-8.6,;66.99,-7.03,;66.18,-8.34,;64.64,-8.29,;63.9,-6.94,;62.37,-6.89,;61.5,-5.62,;60.02,-6.06,;59.98,-7.59,;61.43,-8.11,;61.86,-9.59,;60.8,-10.71,;59.3,-10.34,;58.25,-11.45,;58.67,-12.92,;60.17,-13.29,;61.25,-12.18,;58.68,-5.28,;58.68,-3.74,;57.34,-6.05,;56,-5.29,;54.52,-5.69,;54.12,-4.2,;55.61,-3.8,;52.78,-3.43,;51.45,-4.2,;52.78,-1.88,;64.71,-5.63,;63.98,-4.28,;66.24,-5.67,)|
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(C)(C)C)C(=O)NC2CCS(=O)(=O)CC2)c2ccccc12
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2COC(C)(C)C)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)N2CC3(C2)CS(=O)(=O)C3)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1cc(cc(c1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O)C(F)(F)F |r,wU:31.33,wD:33.38,1.0,(90.63,-20.79,;91.43,-19.48,;90.7,-18.12,;89.16,-18.08,;87.82,-17.31,;89.15,-16.54,;88.35,-19.4,;86.82,-19.36,;86.02,-20.67,;86.74,-22.02,;88.28,-22.07,;89.1,-20.76,;89.01,-23.42,;90.34,-22.64,;90.35,-24.18,;88.21,-24.74,;84.48,-20.63,;83.61,-19.35,;82.13,-19.79,;82.09,-21.33,;83.54,-21.84,;83.97,-23.32,;82.91,-24.43,;81.42,-24.07,;80.36,-25.18,;80.78,-26.65,;82.28,-27.02,;83.36,-25.91,;80.79,-19.02,;80.79,-17.48,;79.45,-19.79,;78.12,-19.02,;76.63,-19.42,;76.23,-17.93,;77.72,-17.54,;74.9,-17.16,;73.56,-17.94,;74.9,-15.62,;92.97,-19.51,;93.71,-20.87,;93.78,-18.2,;94.5,-19.51,)|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12)C(F)(F)F |r,wU:23.24,wD:25.29,1.0,(47.78,-20.49,;47.05,-19.14,;45.51,-19.11,;44.7,-20.42,;46.03,-21.19,;44.7,-21.96,;43.16,-20.39,;42.35,-21.7,;40.81,-21.65,;40.08,-20.3,;38.54,-20.25,;37.67,-18.98,;36.2,-19.42,;36.15,-20.96,;37.6,-21.47,;38.04,-22.95,;36.97,-24.07,;35.43,-24.1,;35.47,-25.64,;37.01,-25.61,;34.85,-18.65,;34.85,-17.1,;33.51,-19.41,;32.18,-18.65,;30.69,-19.05,;30.29,-17.56,;31.78,-17.16,;28.95,-16.79,;27.62,-17.56,;28.95,-15.24,;40.88,-18.99,;40.15,-17.65,;40.95,-16.34,;42.49,-16.38,;43.22,-17.73,;42.42,-19.03,;47.85,-17.83,;49.38,-17.87,;47.12,-16.48,;48.6,-16.49,)|
C[C@H](NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O)C(F)(F)F |r,wU:32.38,wD:1.0,30.33,(6.28,-4.61,;6.02,-3.09,;4.57,-2.57,;3.39,-3.56,;3.66,-5.07,;1.94,-3.03,;1.67,-1.51,;.23,-.99,;-.95,-1.98,;-.69,-3.49,;.76,-4.02,;-1.86,-4.48,;-3.04,-3.49,;-1.09,-5.82,;-2.63,-5.82,;-.04,.53,;1.03,1.64,;.31,3,;-1.21,2.73,;-1.42,1.2,;-2.78,.48,;-4.09,1.3,;-5.45,.57,;-6.76,1.39,;-6.7,2.93,;-5.34,3.65,;-4.04,2.84,;.98,4.38,;.12,5.66,;2.52,4.49,;3.38,3.21,;3.09,1.7,;4.6,1.41,;4.89,2.92,;5.46,.13,;6.99,.24,;4.78,-1.25,;7.2,-2.1,;8.38,-1.11,;8.19,-3.28,;6.21,-.92,)|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2Cc2ccc(F)cc2)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NC(=O)c1cc(cc(c1)C(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O)C(F)(F)F |r,wU:30.32,wD:32.37,1.0,(85.01,-7.33,;85.81,-6.01,;85.08,-4.66,;83.54,-4.62,;82.8,-3.27,;82.73,-5.94,;81.2,-5.9,;80.4,-7.21,;81.13,-8.56,;82.66,-8.61,;83.48,-7.3,;83.39,-9.95,;84.72,-9.18,;84.73,-10.72,;82.59,-11.27,;78.86,-7.17,;77.99,-5.89,;76.51,-6.33,;76.47,-7.87,;77.92,-8.38,;78.35,-9.86,;77.29,-10.97,;75.8,-10.6,;74.74,-11.71,;75.17,-13.19,;76.66,-13.56,;77.74,-12.44,;75.17,-5.56,;75.17,-4.02,;73.83,-6.33,;72.5,-5.56,;71.01,-5.96,;70.61,-4.47,;72.1,-4.08,;69.28,-3.7,;67.94,-4.48,;69.28,-2.16,;87.35,-6.05,;88.09,-7.41,;88.16,-4.74,;88.89,-6.05,)|
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CS(=O)(=O)C3)c(Cl)c1Cl
CCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12 |r,wU:28.29,wD:30.34,(9.88,-3.89,;9.88,-2.35,;8.54,-1.58,;8.54,-3.12,;9.88,-.81,;7.21,-.81,;7.21,.73,;8.75,.73,;7.21,2.27,;5.67,.73,;4.9,-.6,;3.36,-.6,;2.59,.73,;1.05,.73,;.14,1.98,;-1.32,1.5,;-1.32,-.04,;.14,-.52,;.54,-2,;-.55,-3.09,;-2.03,-2.69,;-3.12,-3.78,;-2.72,-5.27,;-1.24,-5.67,;-.15,-4.58,;-2.65,2.27,;-2.65,3.81,;-3.99,1.5,;-5.32,2.27,;-6.81,1.87,;-7.21,3.36,;-5.72,3.76,;-8.54,4.13,;-8.54,5.67,;-9.88,3.36,;3.36,2.06,;2.59,3.4,;3.36,4.73,;4.9,4.73,;5.67,3.4,;4.9,2.06,)|
C[C@H](NC(=O)c1cc(cc(c1)C1(CC1)C#N)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O)C(F)(F)F |r,wU:31.34,wD:33.39,1.0,(43.37,-21.19,;44.17,-19.88,;43.43,-18.52,;41.89,-18.49,;41.15,-17.13,;41.09,-19.8,;39.55,-19.76,;38.75,-21.07,;39.48,-22.42,;41.02,-22.48,;41.83,-21.16,;41.74,-23.82,;43.07,-23.04,;43.08,-24.58,;40.94,-25.14,;40.14,-26.46,;37.22,-21.03,;36.34,-19.75,;34.87,-20.19,;34.82,-21.73,;36.27,-22.24,;36.71,-23.72,;35.64,-24.84,;34.16,-24.47,;33.1,-25.58,;33.52,-27.05,;35.02,-27.42,;36.09,-26.31,;33.52,-19.42,;33.52,-17.88,;32.19,-20.19,;30.85,-19.42,;29.37,-19.82,;28.97,-18.34,;30.46,-17.94,;27.63,-17.56,;26.3,-18.34,;27.63,-16.02,;45.71,-19.92,;46.45,-21.27,;46.51,-18.6,;47.24,-19.91,)|
CC(C)(CCO)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12 |r,wU:29.30,wD:31.35,(8.54,-3.12,;8.54,-1.58,;9.88,-.81,;9.88,-2.35,;9.88,-3.89,;8.54,-4.66,;7.21,-.81,;7.21,.73,;8.75,.73,;7.21,2.27,;5.67,.73,;4.9,-.6,;3.36,-.6,;2.59,.73,;1.05,.73,;.14,1.98,;-1.32,1.5,;-1.32,-.04,;.14,-.52,;.54,-2,;-.55,-3.09,;-2.03,-2.69,;-3.12,-3.78,;-2.72,-5.27,;-1.24,-5.67,;-.15,-4.58,;-2.65,2.27,;-2.65,3.81,;-3.99,1.5,;-5.32,2.27,;-6.81,1.87,;-7.21,3.36,;-5.72,3.76,;-8.54,4.13,;-8.54,5.67,;-9.88,3.36,;3.36,2.06,;2.59,3.4,;3.36,4.73,;4.9,4.73,;5.67,3.4,;4.9,2.06,)|
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c(c1)C(F)(F)F |r,wU:27.28,wD:29.33,(72.21,-6.55,;70.88,-5.78,;70.87,-7.32,;71.68,-4.47,;69.34,-5.75,;68.53,-7.06,;69.86,-7.83,;68.53,-8.6,;66.99,-7.03,;66.18,-8.34,;64.64,-8.29,;63.91,-6.94,;62.37,-6.89,;61.5,-5.62,;60.03,-6.06,;59.98,-7.59,;61.43,-8.11,;61.87,-9.59,;60.8,-10.71,;59.31,-10.34,;58.25,-11.45,;58.68,-12.92,;60.18,-13.3,;61.25,-12.18,;58.68,-5.28,;58.68,-3.74,;57.34,-6.05,;56.01,-5.29,;54.52,-5.69,;54.12,-4.2,;55.61,-3.8,;52.78,-3.43,;51.45,-4.2,;52.78,-1.88,;64.71,-5.63,;66.25,-5.67,;63.99,-4.28,;62.45,-4.23,;64.79,-2.97,;63.21,-2.94,)|
Cc1c(OC(F)F)c(ccc1S(=O)(=O)NC(C)(C)C)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O |r,wU:34.36,wD:36.41,(4.81,-4.68,;4.41,-3.19,;2.92,-2.79,;1.83,-3.88,;2.23,-5.37,;3.72,-5.77,;1.14,-6.46,;2.52,-1.3,;3.61,-.21,;5.1,-.61,;5.5,-2.1,;6.98,-2.5,;6.59,-3.99,;8.07,-3.59,;8.07,-1.41,;7.67,.08,;6.19,.48,;7.28,1.57,;8.76,1.17,;1.03,-.9,;.56,.56,;-.98,.56,;-1.46,-.9,;-.21,-1.81,;-.21,-3.35,;-1.55,-4.12,;-2.88,-3.35,;-4.21,-4.12,;-4.21,-5.66,;-2.88,-6.43,;-1.55,-5.66,;-2.07,1.65,;-1.67,3.14,;-3.56,1.25,;-4.65,2.34,;-6.19,2.34,;-6.19,3.88,;-4.65,3.88,;-7.28,4.97,;-6.88,6.46,;-8.76,4.57,)|
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC3(C2)CS(=O)(=O)C3)c2ccccc12
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCCN2CCOCC2)c2ccccc12
CC(C)(C)NS(=O)(=O)c1ncc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12 |r,wU:27.28,wD:29.33,(6.19,.46,;7.67,.06,;8.76,1.15,;7.28,1.55,;8.07,-1.42,;6.98,-2.51,;6.59,-4,;8.07,-3.6,;5.5,-2.11,;5.1,-.63,;3.61,-.23,;2.52,-1.32,;1.03,-.92,;.56,.55,;-.98,.55,;-1.46,-.92,;-.21,-1.82,;-.21,-3.36,;-1.55,-4.13,;-2.88,-3.36,;-4.21,-4.13,;-4.21,-5.67,;-2.88,-6.44,;-1.55,-5.67,;-2.07,1.64,;-1.67,3.12,;-3.56,1.24,;-4.65,2.33,;-6.19,2.33,;-6.19,3.87,;-4.65,3.87,;-7.28,4.96,;-6.88,6.44,;-8.76,4.56,;2.92,-2.8,;1.83,-3.89,;2.23,-5.38,;3.72,-5.78,;4.81,-4.69,;4.41,-3.2,)|
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC2CS(=O)(=O)C2)c2ccccc12
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CC2)C(=O)NCC(C)(C)O)c2ccccc12)C(F)(F)F |r|
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC(C)(C)C(N)=O)c2ccccc12
CCS(=O)(=O)c1ccc(CNC(=O)c2nc(CC3CCCCC3)c(s2)-c2ccc(c3ccccc23)S(=O)(=O)NC(C)(C)C)cc1
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NC23CC(C2)(C3)C(O)=O)c2ccccc12
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CC(C2)C(C)(C)C(O)=O)c2ccccc12
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N2CCC(C)(C2)C(O)=O)c2ccccc12
CC[C@H](NC(=O)c1cc(cc(c1)C1(C)CC1)-c1sc(nc1CC1CCCCC1)C(=O)N[C@H]1C[C@@H](C1)C(O)=O)C(F)(F)F |r,wU:31.34,wD:33.39,2.1,(68.28,-22.54,;67.54,-21.19,;68.34,-19.87,;67.61,-18.52,;66.07,-18.48,;65.33,-17.12,;65.26,-19.79,;63.73,-19.76,;62.93,-21.06,;63.65,-22.42,;65.19,-22.47,;66.01,-21.15,;65.92,-23.81,;65.12,-25.13,;67.25,-23.04,;67.26,-24.58,;61.39,-21.02,;60.52,-19.74,;59.04,-20.18,;59,-21.72,;60.45,-22.23,;60.88,-23.71,;59.82,-24.83,;58.33,-24.46,;57.27,-25.57,;57.69,-27.04,;59.19,-27.42,;60.27,-26.3,;57.7,-19.41,;57.7,-17.87,;56.36,-20.18,;55.03,-19.42,;53.54,-19.82,;53.14,-18.33,;54.63,-17.93,;51.81,-17.56,;50.47,-18.33,;51.81,-16.02,;69.88,-19.91,;70.62,-21.26,;70.69,-18.59,;71.41,-19.9,)|
CC(C)(CCF)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)N[C@H]2C[C@@H](C2)C(O)=O)c2ccccc12 |r,wU:29.30,wD:31.35,(7.11,-2.53,;7.51,-1.04,;8.6,-2.13,;8.6,.05,;10.08,-.35,;11.17,.74,;6.02,-.64,;4.93,-1.73,;4.53,-3.22,;6.02,-2.82,;3.44,-1.33,;3.04,.16,;1.56,.56,;.47,-.53,;-1.02,-.13,;-1.93,1.11,;-3.39,.64,;-3.39,-.9,;-1.93,-1.38,;-1.53,-2.87,;-2.62,-3.96,;-4.1,-3.56,;-5.19,-4.65,;-4.79,-6.13,;-3.31,-6.53,;-2.22,-5.44,;-4.48,1.73,;-4.08,3.21,;-5.97,1.33,;-7.06,2.42,;-8.6,2.42,;-8.6,3.96,;-7.06,3.96,;-9.68,5.04,;-11.17,4.65,;-9.29,6.53,;.87,-2.02,;-.22,-3.11,;.18,-4.6,;1.66,-4.99,;2.75,-3.91,;2.35,-2.42,)|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c(c1)C(F)F)C(F)(F)F |r|
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(=O)NCC2CS(=O)(=O)C2)c2ccccc12
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCCCC2)C(N)=O)c2ccccc12
CC(C)CCC[C@@H](C)[C@H]1CC[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C |t:14|
C\C(=C/c1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)c1c(F)cccc1Cl |r|
OC(=O)CC[C@H]1CN(c2cc(\C=C\c3c(Cl)cccc3C(F)(F)F)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
[H][C@@]1([#6]-[#6][C@@]2([H])[#6]-3=[#6](-[#6]-[#6][C@]12[#6])[C@@]1([#6])[#6]-[#6]-[#6@H](-[#8])-[#6][C@]1([H])[#6]-[#6]-3)[#6@H](-[#6])-[#6]-[#6]\[#6]=[#6](/[#6])-[#6] |r,c:6|
C[C@H]1CN(c2nc(COc3c(F)cccc3Cl)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
[H][C@@]1([#6]-[#6][C@@]2([H])[C@]3([H])[#6]-[#6]=[#6]4-[#6]-[#6@@H](-[#8])-[#6]-[#6][C@]4([#6])[C@@]3([H])[#6]-[#6][C@]12[#6])[#6@H](-[#6])-[#6]-[#6]\[#6]=[#6](\[#6])-[#6] |r,t:9|
CCS(=O)(=O)c1ccc(cc1)CC(=O)Nc2cc(c(nc2)O[C@@H](C)c3ccccc3)Cl
C[C@@H](Oc1ccc(NC(C)=O)cc1Cl)c1ccccc1 |r|
CC(=O)Nc1ccc(OC2CC2)c(Cl)c1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cnc(OCc3ccccc3)c(Cl)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cnc(O[C@H](C)c3ccccc3)c(Cl)c2)cc1 |r|
C[C@H](Oc1ccc(NC(C)=O)cc1Cl)c1ccccc1 |r|
CCS(=O)(=O)c1ccc(CC(N)=O)cc1
CC(Oc1ccc(NC(C)=O)cc1Cl)C(F)(F)F
CC(C)Oc1ccc(NC(C)=O)cc1Cl
C[C@H](Oc1ncc(NC(=O)Cc2ccncc2)cc1Cl)c1ccccc1 |r|
C[C@H](Oc1ncc(NC(C)=O)cc1Cl)c1ccccc1 |r|
CCOc1ncc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1Cl
CCOc1ccc(cc1Cl)NC(=O)C
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)C(=O)c2ccccc2C)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(-c3ccc(CC(C)C)c(c3)C#N)c(c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)C(=O)c2ccccc2C2CCCC2)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(-c3cccc(c3)C#N)c(c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(C(C)C)c(c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)C(=O)c2ccccc2CC(C)C)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(-c3ccc(CC4CCN(CC4)C(=O)C(C)(C)C)c(c3)C#N)c(c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(-c3ccc(CC4CCN(CC4)C(C)=O)c(c3)C#N)c(c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)C(=O)c2ccccc2C(C)C)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(-c3ccc(CC4CCCCC4)c(c3)C#N)c(c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(-c3ccccc3)c(c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(Cl)c2)-c2ccc(CC3CCN(CC3)C(=O)C(C)(C)C)cc2C(F)(F)F)cc1
COc1cc(O)c(C(CC(=O)N2CC(C)CC(C)C2)c2ccccc2OC)c(OC)c1
COc1ccc(cc1)C(CC(=O)N1CC(C)CC(C)C1)c1c(O)cc(OC)cc1OC
COc1cc(O)c(C(CC(=O)N2CC(C)CC(C)C2)c2ccc3OCOc3c2)c(OC)c1
CC1CC(C)CN(C1)C(=O)CC(c1ccc(C)cc1)c1c(O)ccc2ccccc12
CC1CC(C)CN(C1)C(=O)CC(c1ccc2OCOc2c1)c1c(O)ccc2ccccc12
CC1CC(C)CN(C1)C(=O)CC(c1ccc2OCOc2c1)c1c(O)cccc1Oc1ccccc1
CC1CC(C)CN(C1)C(=O)CC(c1ccc2OCOc2c1)c1cc(C)ccc1O
CC1CC(C)CN(C1)C(=O)CC(c1ccc2OCOc2c1)c1c(C)cccc1O
CCCOc1ccc(O)c(c1)C(CC(=O)N1CC(C)CC(C)C1)c1ccc2OCOc2c1
CCOc1ccc(O)c(c1)C(CC(=O)N1CC(C)CC(C)C1)c1ccc2OCOc2c1
CCc1ccc(O)c(c1)C(CC(=O)N1CC(C)CC(C)C1)c1ccc2OCOc2c1
COc1cc(O)c(C(CC(=O)N2CCCC(C2)C(F)(F)F)c2ccc3OCOc3c2)c(OC)c1
COc1cc(O)c(C(CC(=O)N2CCC(CC2)c2ccccc2)c2ccc3OCOc3c2)c(OC)c1
CCn1c2ccc(C)cc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCn1c2ccccc2c3c1ccc(c3)C(=O)NCc4ccc(cc4)S(=O)(=O)CC
CCn1c2ccccc2c2cc(NC(=O)Cc3ccc(cc3)S(=O)(=O)CC)ccc12
CCn1c2ccccc2c2cc(ccc12)C(=O)NCc1ccc(cn1)S(=O)(=O)CC
CCn1c2ccccc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)NC
CCn1c2ccccc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(C)(=O)=O
CCn1c2ccc(Cl)cc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCn1c2ccc(F)cc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CC4CCC4)c4ccccc4c3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CC(C)C)c4ccccc4c3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CC4CC4)c4ccccc4c3c2)cc1
CCn1c2ccccc2c2cc(NC(=O)NCc3ccc(cc3)S(=O)(=O)CC)ccc12
CCCn1c2ccccc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C)c4ccccc4c3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3[nH]c4ccccc4c3c2)cc1
CCn1c2CCCc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCn1c2CCCCc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
COc1cc(O)c(C(CC(=O)N2C[C@@H](C)C[C@@H](C)C2)c2ccc3OCOc3c2)c(OC)c1 |r|
COc1ccc(cc1)C(CC(=O)N1C[C@@H](C)C[C@@H](C)C1)c1c(O)cc(OC)cc1OC |r|
COc1ccc(cc1)C(CC(=O)N1CCCC(C)C1)c1c(O)cc(OC)cc1OC
COc1cccc(c1)C(CC(=O)N1C[C@@H](C)C[C@@H](C)C1)c1c(O)cc(OC)cc1OC |r|
COc1cc(O)c(C(CC(=O)N2C[C@@H](C)C[C@@H](C)C2)c2ccc(C)cc2)c(OC)c1 |r|
COc1cc(O)c(C(CC(=O)N2C[C@@H](C)C[C@@H](C)C2)c2ccc(Cl)cc2)c(OC)c1 |r|
COc1cc(O)c(C(CC(=O)N2C[C@@H](C)C[C@@H](C)C2)c2ccc(cc2)C(F)(F)F)c(OC)c1 |r|
COc1cc(OC)c(C(CC(=O)N2CCCC(C)C2)c2ccc3OCOc3c2)c(OC)c1
CC1CCCN(C1)C(=O)CC(c1ccc2OCOc2c1)c1cc(ccc1O)-c1ccccc1
COc1ccc(C(CC(=O)N2CCCC(C)C2)c2ccc3OCOc3c2)c(O)c1
COc1cccc(O)c1C(CC(=O)N1CCCC(C)C1)c1ccc2OCOc2c1
COc1cc(O)c(C(CC(=O)N2C[C@H](C)O[C@H](C)C2)c2ccc3OCOc3c2)c(OC)c1 |r|
COc1cc(O)c(C(CC(=O)N2CCCC(C)(C)C2)c2ccc3OCOc3c2)c(OC)c1
COc1cc(O)c(C(CC(=O)N2CCC(C)CC2)c2ccc3OCOc3c2)c(OC)c1
COc1cc(O)c(C(CC(=O)N2CCCCC2C)c2ccc3OCOc3c2)c(OC)c1
COc1cc(O)c(C(CC(=O)Nc2ccc(C)cc2)c2ccc3OCOc3c2)c(OC)c1
CCCCNC(=O)CC(c1ccc2OCOc2c1)c1c(O)cc(OC)cc1OC
CCN(CC)C(=O)CC(c1ccc2OCOc2c1)c1c(O)cc(OC)cc1OC
COc1cc(O)c(C(CC(=O)N2CCCCCC2)c2ccc3OCOc3c2)c(OC)c1
COc1cc(O)c(C(CC(=O)N2CCCCC2)c2ccc3OCOc3c2)c(OC)c1
COc1cc(O)c(C(CC(=O)N2CCCC2)c2ccc3OCOc3c2)c(OC)c1
COc1cc(O)c(C(CC(=O)N2CCCC(C)C2)c2ccc3OCOc3c2)c(OC)c1
CCn1c2ccccc2c2cc(NC(=O)CNC(=O)Cc3ccc(cc3)S(=O)(=O)CC)ccc12
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CC4CCCCC4)c4ccccc4c3c2)cc1
CCn1ccc2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCn1c2ccccc2c2cc(NC(=O)CC(C)CC(=O)Nc3ccc(C#N)c(Cl)c3)ccc12
CCCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CC)c4ccccc4c3c2)cc1
CCn1c2ccc(cc2c2ncccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C(C)C)c4ccccc4c3c2)cc1
CCn1c(C)c(C)c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
OC(c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1cccnc1)(C(F)(F)F)C(F)(F)F
Cc1ccc(cc1)S(=O)(=O)N(CC(F)(F)F)c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
OC(c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1ccc(cc1)C#N)(C(F)(F)F)C(F)(F)F
OC(c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1cccc(c1)C#N)(C(F)(F)F)C(F)(F)F
OC(c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1ccccc1C#N)(C(F)(F)F)C(F)(F)F
OC(c1ccc(cc1)N(CC(F)(F)F)C(=O)c1ccccc1)(C(F)(F)F)C(F)(F)F
CC(=O)NCCN(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1
CCN(c1cccc(c1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1
OC(c1ccc2N(CCc2c1)S(=O)(=O)c1ccccc1)(C(F)(F)F)C(F)(F)F
NS(=O)(=O)c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1ccccc1
CS(=O)(=O)CCN(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1
COC(c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1ccccc1)(C(F)(F)F)C(F)(F)F
OC(c1ccc(cc1)N(Cc1ccccc1)S(=O)(=O)c1ccccc1)(C(F)(F)F)C(F)(F)F
OC(c1ccc(cc1)N(CCC(F)(F)F)S(=O)(=O)c1ccccc1)(C(F)(F)F)C(F)(F)F
CCN(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1
COCCN(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1
OCCN(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1
OC(c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)Cc1ccccc1)(C(F)(F)F)C(F)(F)F
OC(c1ccc(NC(=O)c2ccc(cc2)C(F)(F)F)cc1)(C(F)(F)F)C(F)(F)F
OC(c1ccc(NC(=O)c2ccccc2)cc1)(C(F)(F)F)C(F)(F)F
NC(=O)c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1ccccc1
OC(=O)c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1ccccc1
OCc1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1ccccc1
OC(=O)CCN(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1
OC(c1ccc(NS(=O)(=O)c2ccccc2)cc1)(C(F)(F)F)C(F)(F)F
OC(c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)C1CC1)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(c(s2)C(=O)c2cccc(F)c2)-c2cccc(Cl)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(c(s2)C(=O)c2cccc(F)c2)-c2cccc(c2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(c(s2)C(=O)c2ccccc2F)-c2cccc(Cl)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(c(s2)C(=O)c2cccc(Cl)c2)-c2cccc(Cl)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(c(s2)C(=O)c2ccccc2)-c2cccc(c2)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(c(s2)C(=O)c2ccccc2)-c2cccc(Cl)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(c(s2)C(=O)c2ccccc2)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)C(=O)c2cccc(F)c2)-c2cccc(Cl)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)C(=O)c2ccccc2F)-c2cccc(Cl)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)C(=O)c2ccc(Cl)cc2)-c2cccc(Cl)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)C(=O)c2cccc(Cl)c2)-c2cccc(Cl)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)C(=O)c2ccccc2)-c2cccc(c2)C(O)=O)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)C(=O)c2ccccc2)-c2cccc(CN(C)C)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)C(=O)c2ccccc2)-c2cccc(c2)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)C(=O)c2ccccc2)-c2ccc(Cl)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)C(=O)c2ccccc2)-c2cccc(Cl)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)C(=O)c2ccccc2)-c2ccccc2Cl)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)C(=O)C2CCCCC2)-c2ccccc2)cc1
CCC(=O)c1sc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)nc1-c1ccccc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)C(C)=O)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)C(=O)OC)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(Oc3ccccc3)s2)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(Cc3ccccc3)s2)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)C(C)C)-c2ccccc2)cc1
CCc1sc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)nc1-c1ccccc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(C)s2)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(cs2)-c2c(Cl)cccc2Cl)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(cs2)-c2ccc(Cl)cc2Cl)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(cs2)-c2cccc(Cl)c2Cl)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(cs2)-c2ccc(Cl)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(cs2)-c2cccc(Cl)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(cs2)-c2ccccc2Cl)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(cs2)-c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(cs2)C2CCCCC2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(C)cs2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2nccs2)cc1
CN(C)S(=O)(=O)c1ccc(CC(=O)Nc2nc(cs2)-c2cc(Cl)ccc2Cl)cc1
CNS(=O)(=O)c1ccc(CC(=O)Nc2nc(cs2)-c2cc(Cl)ccc2Cl)cc1
Clc1ccc(Cl)c(c1)-c1csc(NC(=O)Cc2ccc(cc2)S(=O)(=O)C2CCCCC2)n1
CC(C)S(=O)(=O)c1ccc(CC(=O)Nc2nc(cs2)-c2cc(Cl)ccc2Cl)cc1
CCCS(=O)(=O)c1ccc(CC(=O)Nc2nc(cs2)-c2cc(Cl)ccc2Cl)cc1
CS(=O)(=O)c1ccc(CC(=O)Nc2nc(cs2)-c2cc(Cl)ccc2Cl)cc1
Clc1ccc(Cl)c(c1)-c1csc(NC(=O)Cc2ccc(cc2)C#N)n1
Clc1ccc(CC(=O)Nc2nc(cs2)-c2cc(Cl)ccc2Cl)cc1
Clc1ccc(Cl)c(c1)-c1csc(NC(=O)Cc2ccccc2)n1
Clc1ccc(Cl)c(c1)-c1csc(NC(=O)CC2CCCCC2)n1
CC(C)CC(=O)Nc1nc(cs1)-c1cc(Cl)ccc1Cl
CCC(=O)Nc1nc(cs1)-c1cc(Cl)ccc1Cl
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3n(CCc4ccc(Cl)c(Cl)c4)ccc3c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3n(CCc4cccc(c4)C(F)(F)F)ccc3c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3n(CCc4ccccc4C(F)(F)F)ccc3c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3n(CCc4ccc(OC(C)C)cc4)ccc3c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3n(CCc4ccc(cc4)C#N)ccc3c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3n(CCc4ccc(Cl)cc4)ccc3c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3n(CCc4ccc(F)cc4)ccc3c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3n(CCc4ccccc4)ccc3c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc3n(CCc4ccc(cc4)C(F)(F)F)ccc3c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(NCCc3ccc(cc3)C(F)(F)F)c(Cl)c2)cc1
CCCN(CCc1ccc(cc1)C(F)(F)F)c1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(NCCc3ccc(cc3)C(F)(F)F)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CNCc3ccc(cc3)C(F)(F)F)cc2)cc1
CCCN(Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1)Cc1ccc(cc1)-c1ccccc1
CCCN(Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1)Cc1ccc(cc1)C(F)(F)F
CCCN(Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1)Cc1ccc(cc1)C(C)(C)C
CCCN(Cc1ccc(CC)cc1)Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CCCN(Cc1ccc(C)cc1)Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CC1(C)CCC(C)(C)c2cc(ccc12)C(=O)Nc1ccccc1
C[Si]1(C)CC[Si](C)(C)c2cc(ccc12)C(=O)Nc1ccccc1
Cc1cc(cc2c1[nH]c(=O)c1ccccc21)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cccnc2OCc2ccc(cc2)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cccnc2OCc2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2ccc(cc2Cl)C#N)cc1
CCS(=O)(=O)c1ccc(cc1)C(NC(C)=O)C(=O)Nc1cc(cs1)-c1cc(cnc1OCC(F)(F)F)C#N
CCS(=O)(=O)c1ccc(cc1)[C@@H](NC(C)=O)C(=O)Nc1cc(cs1)-c1cccnc1OCc1ccc(OC(F)(F)F)cc1 |r|
CCS(=O)(=O)c1ccc(cc1)[C@H](NC(C)=O)C(=O)Nc1cc(cs1)-c1cccnc1OCc1ccc(OC(F)(F)F)cc1 |r|
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cccnc2OC)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cc(cnc2OC)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cccnc2Oc2ccc(cc2)C#N)cc1
CCS(=O)(=O)c1ccc(cc1)C(N)C(=O)Nc1cc(cs1)-c1cc(cc(F)c1OC)C#N
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cc(cnc2OCC(F)(F)F)C#N)cc1
CCS(=O)(=O)c1ccc(cc1)C(NC(C)=O)C(=O)Nc1cc(cs1)-c1cc(cnc1OC)C#N
CCS(=O)(=O)c1ccc(cc1)C(NC(C)=O)C(=O)Nc1cc(cs1)-c1cccnc1OCc1ccccc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cc(ccc2OC)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cncnc2OC)cc1
CNS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cc(cnc2OC)C#N)cc1
CCOc1ncccc1-c1csc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)c1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cccnc2OC\C=C\c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cccnc2OCc2ccc(cc2)C(=O)OC)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cccnc2OCc2cccc(c2)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cccnc2OCc2ccc(OC(F)(F)F)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cc(cc(F)c2OC)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cccnc2OCC(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cccnc2OCCCc2ccccc2)cc1
CC[S+]([O-])c1ccc(CC(=O)Nc2cc(cs2)-c2cc(cnc2OC)C#N)cc1
CCS(=N)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cc(ccc2OC)C#N)cc1
CCS(=O)(=O)N1CCC(CC(=O)Nc2cc(cs2)-c2cc(cnc2OC)C#N)CC1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cccc(Cl)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cc(Cl)cc(c2)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cc(ccc2Cl)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cccnc2Oc2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cccnc2OCCc2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(cs2)-c2cccnc2Oc2ccc(OC(F)(F)F)cc2)cc1
CCCOc1ncccc1-c1csc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)c1
CCS(=O)(=O)c1ccc(cc1)C(NC(C)=O)C(=O)Nc1cc(cs1)-c1cccnc1Oc1ccc(cc1)C#N
CCS(=O)(=O)c1ccc(cc1)C(NC(C)=O)C(=O)Nc1cc(cs1)-c1cc(cc(F)c1OC)C#N
CCS(=O)(=O)c1ccc(cc1)C(NC(C)=O)C(=O)Nc1cc(cs1)-c1cccnc1OCc1ccc(OC(F)(F)F)cc1
CCC(=O)Nc1ccc(cc1)-c1c[nH]c2ncnc(N[C@H](C)c3ccccc3)c12 |r|
CN(C)CCn1cc(-c2cccc(O)c2)c2c(N)ncnc12
CCn1cncc1C(O)(c1ccc(Cl)cc1)c1ccc2nc(Cl)c(-c3ccccc3)c(Cl)c2c1
COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(C1CCN(CC1)C(C)=O)c1ccccc1
Cn1cncc1C(O)(c1ccnc(F)c1)c1ccc2nc(Cl)c(-c3ccccc3)c(Cl)c2c1
Cn1cncc1C(O)(c1ccc2nc(Cl)c(-c3ccccc3)c(Cl)c2c1)c1ccnc2ccccc12
Cc1ncc(n1C)C(O)(c1ccc(Cl)cc1)c1ccc2nc(Cl)c(-c3ccccc3)c(Cl)c2c1
Cn1cncc1C(O)(c1cccnc1)c1ccc2nc(Cl)c(-c3ccccc3)c(Cl)c2c1
Cn1ccnc1C(O)(c1ccnc(F)c1)c1ccc2nc(Cl)c(-c3ccccc3)c(Cl)c2c1
OC(c1ccccc1)(c1cccnc1)c1ccc2nc(Cl)c(-c3ccccc3)c(Cl)c2c1
Cn1cncc1C(O)(c1ccnc(c1)C(F)(F)F)c1ccc2nc(Cl)c(-c3ccccc3)c(Cl)c2c1
CNC(c1cncn1C)(c1ccc(Cl)cc1)c1ccc2nc(OC)c(Cc3ccc(cc3)-n3cccn3)c(Cl)c2c1
COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cnnn1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cnnn1C)c1cnnn1C
COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)c1cnnn1C
COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(O)(C1CCN(CC1)C(C)=O)c1cncn1C
OC(c1ccccc1)(c1ccncc1)c1ccc2nc(Cl)c(-c3ccccc3)c(Cl)c2c1
Cc1cc(ccn1)C(O)(c1cncn1C)c1ccc2nc(Cl)c(-c3ccccc3)c(Cl)c2c1
Cn1cncc1C(O)(c1ccc(nc1)C(F)(F)F)c1ccc2nc(Cl)c(-c3ccccc3)c(Cl)c2c1
Cc1nc(C)c(s1)C(O)(c1cncn1C)c1ccc2nc(Cl)c(-c3ccccc3)c(Cl)c2c1
COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)-n1cccn1)C(N)(c1cncn1C)c1ccc(Cl)cc1
Cn1cncc1C(O)(c1ccc2nc(Cl)c(-c3ccccc3)c(Cl)c2c1)c1ccccn1
OC(c1ccc2N(Cc3ccc(F)cc3)CCSc2c1)(C(F)(F)F)C(F)(F)F
OC(c1ccc2N(CCSc2c1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
CC(C)(O)[C@H](F)CNC(=O)C[C@@H]1CCc2cc(ccc2N1S(=O)(=O)c1ccc(F)cc1)C(O)(C(F)(F)F)C(F)(F)F |r|
OC(c1ccc2N(CCSc2c1)S(O)(O)c1ccc(Cl)nc1)(C(F)(F)F)C(F)(F)F
COc1ccc(cc1)S(O)(O)N1CCSc2cc(ccc12)C(O)(C(F)(F)F)C(F)(F)F
OC(c1ccc2N(CCSc2c1)S(=O)(=O)c1ccc(Cl)cc1)(C(F)(F)F)C(F)(F)F
OC(c1ccc2N(CCSc2c1)S(=O)(=O)c1cccc(F)c1)(C(F)(F)F)C(F)(F)F
OC(c1ccc2N(CCSc2c1)S(=O)(=O)c1ccccc1)(C(F)(F)F)C(F)(F)F
CC1(C)CCN(c2ccc(cc12)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CC1CCN(c2ccc(cc12)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CN1CCN(c2ccc(cc12)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(c1ccc2N(CCNc2c1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
OC(c1ccc2N(CC(CC(=O)N3CCOCC3)Sc2c1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
CC(C)(O)CNC(=O)CC1CN(c2ccc(cc2S1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CC(C)(CNC(=O)C[C@H]1CN(c2ccc(cc2S1)C(C(F)(F)F)(C(F)(F)F)O)S(=O)(=O)c3ccc(cc3)F)O
CC(C)(O)CC(=O)NCC1CN(c2ccc(cc2S1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CC(C)(O)CNC(=O)CC1CSc2cc(ccc2N1S(=O)(=O)c1ccc(F)cc1)C(O)(C(F)(F)F)C(F)(F)F
CC(C)(O)CNC(=O)C[C@@H]1CCc2cc(ccc2N1S(=O)(=O)c1ccc(F)cc1)C(O)(C(F)(F)F)C(F)(F)F |r|
CC(C)(O)CNC(=O)CC1CN(c2ccc(cc2C1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(c1ccc2N(CC(CC(=O)Nc3nncs3)Sc2c1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
NC(=O)CC1CN(c2ccc(cc2S1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(=O)CC1CN(c2ccc(cc2S1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CNC(=O)CC1CN(c2ccc(cc2S1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
COC(=O)CC1CN(c2ccc(cc2S1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(c1ccc2N(CCSc2c1)S(O)(O)c1cccnc1)(C(F)(F)F)C(F)(F)F
OC(c1ccc2N(CCSc2c1)S(=O)(=O)c1ccccc1F)(C(F)(F)F)C(F)(F)F
OC(c1ccc2N(CCCc2c1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
OC(c1ccc2N(CCOc2c1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
OC(c1ccc2N(CC(CC(=O)Nc3ccncc3)Sc2c1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
CC(C)(O)CNC(=O)C[C@H]1CCc2cc(ccc2N1S(=O)(=O)c1ccc(F)cc1)C(O)(C(F)(F)F)C(F)(F)F |r|
OC(c1ccc2N(CCSc2c1)C(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
CC(C)(O)CNC(=O)CC1CCc2cc(ccc2N1S(=O)(=O)c1ccc(F)cc1)C(O)(C(F)(F)F)C(F)(F)F
OC1CN(C1)C(=O)CC1CN(c2ccc(cc2S1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CC(C)(O)CNC(=O)C[C@@H]1CN(c2ccc(cc2S1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
COc1ccc2[C@@H](N(CCc2c1)C(=O)CC(C)(O)CC(O)=O)C(=O)Nc1cc(F)c(c(F)c1)[Si](C)(C)C |r|
COc1ccc2[C@@H](N(CCc2c1)C(=O)\C=C\C(O)=O)C(=O)Nc1cc(F)c(c(F)c1)[Si](C)(C)C |r|
COc1ccc2[C@@H](N(CCc2c1)C(=O)CC1SC(=O)NC1=O)C(=O)Nc1cc(F)c(c(F)c1)[Si](C)(C)C |r|
COc1ccc2[C@@H](N(CCc2c1)C(=O)CC(C)(C)CC(O)=O)C(=O)Nc1cc(F)c(c(F)c1)[Si](C)(C)C |r|
COc1ccc2[C@@H](N(CCc2c1)C(=O)CC(C)CC(O)=O)C(=O)Nc1cc(F)c(c(F)c1)[Si](C)(C)C |r|
COc1ccc2[C@@H](N(CCc2c1)C(=O)CCCCC(O)=O)C(=O)Nc1cc(F)c(c(F)c1)[Si](C)(C)C |r|
COc1ccc2[C@@H](N(CCc2c1)C(=O)\C=C/C(O)=O)C(=O)Nc1cc(F)c(c(F)c1)[Si](C)(C)C |r|
COc1ccc2[C@@H](N(CCc2c1)C(=O)CCC(O)=O)C(=O)Nc1cc(F)c(c(F)c1)[Si](C)(C)C |r|
COc1ccc2[C@@H](N(CCc2c1)C(=O)c1cc(O)no1)C(=O)Nc1cc(F)c(c(F)c1)[Si](C)(C)C |r|
COc1ccc(cc1)[C@@H](N(C)C(=O)c1cc(O)no1)C(=O)Nc1cc(F)c(c(F)c1)[Si](C)(C)C |r|
COc1ccc2c(c1)CCN(C(=O)CN(C)CC(=O)O)[C@H]2C(=O)Nc3cc(F)c([Si](C)(C)C)c(F)c3
COc1ccc2[C@@H](N(CCc2c1)C(=O)CCCC(N)=O)C(=O)Nc1cc(F)c(c(F)c1)[Si](C)(C)C |r|
COc1ccc(cc1)[C@@H](N(C)C(=O)CCC(O)=O)C(=O)Nc1cc(F)c(c(F)c1)[Si](C)(C)C |r|
COc1ccc2[C@@H](N(CCc2c1)C(=O)CCCC(O)=O)C(=O)Nc1cc(F)c(c(F)c1)[Si](C)(C)C |r|
COc1ccc2[C@@H](N(CCc2c1)C(=O)COCC(O)=O)C(=O)Nc1cc(F)c(c(F)c1)[Si](C)(C)C |r|
COc1ccc2[C@@H](N(CCOc2c1)C(=O)c1cc(O)no1)C(=O)Nc1cc(F)c(c(F)c1)[Si](C)(C)C |r|
COc1ccc(cc1)C(N(C)C(=O)c1ccc(O)nc1)C(=O)Nc1ccc(cc1)C(C)C
COc1ccc(cc1)C(N(C)C(=O)c1ccc(=O)[nH]c1)C(=O)Nc1ccc(cc1)C(C)(C)C
COc1ccc(cc1)C(NC(=O)c1ccc(=O)[nH]c1)C(=O)Nc1ccc(cc1)C(C)(C)C
COc1ccc(cc1)C(N(C)C(=O)c1cc(O)no1)C(=O)Nc1cc(F)c(c(F)c1)[Si](C)(C)C
COc1ccc(cc1)C(N(C)C(=O)c1ccc(=O)[nH]c1)C(=O)Nc1ccc2c(CCC2(C)C)c1
COc1ccc(cc1)C(CN(C)C(=O)c1ccc(=O)[nH]c1)C(=O)Nc1ccc(cc1)C(C)(C)C
COc1ccc(cc1)C(N(C)C(=O)c1ccno1)C(=O)Nc1ccc(cc1)[Si](C)(C)C
COc1ccc(cc1)C(N(C)C(=O)c1ccco1)C(=O)Nc1ccc(cc1)[Si](C)(C)C
COc1ccc(cc1)C(N(C)C(=O)c1ccco1)C(=O)Nc1ccc(cc1)C(C)(C)C
COc1ccc(cc1)C(N(C)C(=O)c1ccc(=O)[nH]c1)C(=O)N(C)c1ccc(cc1)C(C)(C)C
COc1ccc(cc1)C(N(C)C(=O)c1ccc(O)nc1)C(=O)Nc1ccc(cc1)[Si](C)(C)C
CCCN(C(C(=O)Nc1ccc(cc1)C(C)(C)C)c1ccc(OC)cc1)C(=O)c1ccc(=O)[nH]c1
COc1ccc(C(N(C)C(=O)c2ccc(=O)[nH]c2)C(=O)Nc2ccc(cc2)C(C)(C)C)c(C)c1
COc1ccc(cc1)C(N(C)C(=O)c1cc(O)no1)C(=O)Nc1ccc(cc1)[Si](C)(C)C
COc1ccc(cc1)C(N(C)C(=O)c1ccno1)C(=O)Nc1ccc(cc1)C(C)(C)C
COc1ccc(cc1)C(N(C)C(=O)c1cc(O)no1)C(=O)Nc1ccc(cc1)C(C)(C)C
COc3ccc([C@@H](C(=O)Nc1cc(F)c([Si](C)(C)C)c(F)c1)N(C)C(=O)c2cc(O)no2)cc3
COc1ccc(cc1)C(N(C)C(=O)c1ccc(=O)[nH]c1)C(=O)Nc1ccc(C)cc1
COc1ccc(CC(N(C)C(=O)c2ccc(=O)[nH]c2)C(=O)Nc2ccc(cc2)C(C)(C)C)cc1
COc1ccc(cc1)C(CC(=O)Nc1ccc(cc1)C(C)(C)C)N(C)C(=O)c1ccc(=O)[nH]c1
COc1ccc(cc1)C(N(C)C(=O)c1ccc(=O)[nH]c1)C(=O)Nc1ccc(c(Cl)c1)C(C)(C)C
CC(CC(=O)Nc1ccc(C#N)c(Cl)c1)CC(=O)Nc1ccc2n(CC3CC3)c(=O)n(CC3CC3)c(=O)c2c1
CCC1Oc2cc(NC(=O)CC(C)CC(=O)Nc3ccc(C#N)c(Cl)c3)ccc2N(CC)C1=O
CCn1ccc2cc(NC(=O)CC(C)CC(=O)Nc3ccc(C#N)c(Cl)c3)ccc12
CCn1c2ccccc2c2cc(NC(=O)CC(C)CC(=O)Nc3ccccc3)ccc12
CCn1c2ccccc2c2cc(NC(=O)CCCCC(=O)Nc3ccc(cc3)C#N)ccc12
CCn1c2ccccc2c2cc(NC(=O)CC(C)CC(=O)Nc3cccc(c3)C#N)ccc12
CCn1c2ccccc2c2cc(NC(=O)CC(C)CC(=O)Nc3ccc(cc3)C#N)ccc12
CCn1c2ccc(NC(=O)CC(C)CC(=O)Nc3ccc(C#N)c(Cl)c3)cc2oc1=O
CCn1c2CCCCc2c2cc(NC(=O)CC(C)CC(=O)Nc3ccc(cc3)C#N)ccc12
CCn1c2ccccc2c2cc(NC(=O)CC(C)CC(=O)Nc3ccc(C#N)c(c3)C(F)(F)F)ccc12
CCn1c2ccccc2c2cc(ccc12)N(C)C(=O)CC(C)CC(=O)N(C)c1ccc(cc1)C#N
CCn1c2ccccc2c2cc(NC(=O)CN(C)CC(=O)Nc3ccc(cc3)C#N)ccc12
CCn1c2ccccc2c2cc(NC(=O)CC(C)(C)CC(=O)Nc3ccc(cc3)C#N)ccc12
CCn1c2ccccc2c2cc(NC(=O)CCC(=O)Nc3ccc(cc3)C#N)ccc12
CCn1c(=O)n(CC2CC2)c2ccc(NC(=O)CC(C)CC(=O)Nc3ccc(C#N)c(Cl)c3)cc2c1=O
CCn1c2ccc(NC(=O)CC(C)CC(=O)Nc3ccc(C#N)c(Cl)c3)cc2c(=O)n(CC2CC2)c1=O
CCN1C(=O)C(C)Oc2cc(NC(=O)CC(C)CC(=O)Nc3ccc(C#N)c(Cl)c3)ccc12
CCN1C(=O)COc2cc(NC(=O)CC(C)CC(=O)Nc3ccc(C#N)c(Cl)c3)ccc12
CCn1c2ccccc2c2cc(NC(=O)CC(C)CC(=O)Nc3ccccc3C#N)ccc12
CCN1c2ccc(cc2C(=O)N(C1=O)CC)NC(=O)C[C@H](C)CC(=O)Nc3ccc(c(c3)Cl)C#N
CC(CC(=O)Nc1ccc(cc1)C#N)CC(=O)Nc1ccc2[nH]c3CCCCc3c2c1
CCn1c2ccccc2c2cc(NC(=O)CC(C)CC(=O)Nc3ccc(F)cc3)ccc12
CCn1c2ccccc2c2cc(NC(=O)COCC(=O)Nc3ccc(cc3)C#N)ccc12
CCn1c2ccccc2c2cc(NC(=O)CCCC(=O)Nc3ccc(cc3)C#N)ccc12
[H][C@@]12CC(C(O)[C@@]1(C)CC[C@]1([H])c3cc(c(O)cc3CC[C@@]21[H])-c1cccc2c3ccccc3oc12)C(O)=O |r|
[H][C@@]12CC(=C[C@@]1(C)CC[C@]1([H])c3cc(C(=O)c4ccccc4)c(O)cc3CC[C@@]21[H])C(O)=O |r,c:3|
[H][C@@]12CC(=C[C@@]1(C)CC[C@]1([H])c3cc(c(OC)cc3CC[C@@]21[H])C12CC3CC(CC(C3)C1)C2)C(O)=O |r,c:3,TLB:13:23:26:30.29.28,THB:24:25:28:32.23.31,24:23:26.25.30:28,31:23:26:30.29.28,31:29:26:32.24.23|
[H][C@@]12CC(=C[C@@]1(C)CC[C@]1([H])c3cc(c(O)cc3CC[C@@]21[H])C12CC3CC(CC(C3)C1)C2)C(O)=O |r,c:3,TLB:13:22:25:29.28.27,THB:23:24:27:31.22.30,23:22:25.24.29:27,30:22:25:29.28.27,30:28:25:31.23.22|
COc1ccccc1C(=O)c1sc(N)nc1-c1ccc(Cl)c(c1)C(F)(F)F
Nc1nc(c(s1)C(=O)c1ccccc1Cl)-c1cc(cc(c1)C(F)(F)F)C(F)(F)F
Nc1nc(c(s1)C(=O)c1ccccc1Cl)-c1cc(Br)cc(c1)C(F)(F)F
Nc1nc(c(s1)C(=O)c1ccccc1C(F)(F)F)-c1cccc(c1)C(F)(F)F
Nc1nc(c(s1)C(=O)c1ccccc1Br)-c1cccc(c1)C(F)(F)F
Nc1nc(c(s1)C(=O)c1c(F)cccc1C(F)(F)F)-c1cccc(c1)C(F)(F)F
Nc1nc(c(s1)C(=O)c1c(F)cccc1Cl)-c1cccc(c1)C(F)(F)F
COc1ccccc1C(=O)c1sc(N)nc1-c1cc(Br)cc(c1)C(F)(F)F
Nc1nc(c(s1)C(=O)c1ccccc1Cl)-c1ccc(Cl)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(CC(=O)Nc2nc(c(s2)C(=O)c2ccccc2Cl)-c2ccccc2Cl)cc1
Nc1nc(c(s1)C(=O)c1ccccc1Cl)-c1cccc(Cl)c1
COc1ccccc1C(=O)c1sc(N)nc1-c1cccc(c1)C(F)(F)F
Nc1nc(c(s1)C(=O)c1ccccc1Cl)-c1cccc(c1)C(F)(F)F
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c(CC#N)c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c(c1)[S+](C)[O-]
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c(CC(O)=O)c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)cc1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c(CO)c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c(c1)S(C)(=N)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c(CC(N)=O)c1
C[Si](C)(O)c1ccc(cc1)N(CCc1ccccc1)S(=O)(=O)c1ccccc1
CC(C)(O)c1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1ccccc1
CCN(c1ccc(cc1)[Si](C)(C)O)S(=O)(=O)c1ccccc1
COC(=O)CN(c1ccc(cc1)C(C)(C)O)S(=O)(=O)c1ccccc1
C[Si](C)(O)c1ccc(cc1)N(Cc1ccccc1)S(=O)(=O)c1ccccc1
CCCCN(c1ccc(cc1)[Si](C)(C)O)S(=O)(=O)c1ccccc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)Nc2cccnc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)N(C)C)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)Nc2ccccc2F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)Nc2cc(ccn2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)N2CCc3ccccc23)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(F)c2)C(C)(C)C(=O)Nc2ccc(F)cc2)cc1
CCOC(=O)C(C)(C)c1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)Nc2ccncc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)Nc2ccccc2C)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)N2Cc3ccccc3C2)cc1
CCS(=O)(=O)c1ccc(cc1)CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)Nc3ccccc3
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)Nc2cc(F)ccn2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(F)c2)C(C)(C)C(=O)Nc2cc(ccn2)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)N2CCC2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)N2CC3(CCC3)C2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)N2CCCCC2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)Nc2cccc(F)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)Nc2ccc(F)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)Nc2ccc(F)cc2F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)N(C)c2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(c(F)c2)C(C)(C)C(=O)Nc2ccc(F)cc2F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)Nc2cccc(n2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)Nc2cc(Cl)ccn2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)Nc2cc(ccn2)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)Nc2ccccn2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C(=O)Nc2ncccc2F)cc1
Cc1c(ccc2c1c(cn2C)C3CCN(CC3)C(=O)C4CCCC4)NC(=O)c5cccc(c5)C#N
COc1c(NC(=O)c2cccc(c2)C#N)cnc2n(C)cc(C3CCN(CC3)C(=O)C(C)C)c12
Cc1c(NC(=O)c2cccc(c2)C#N)cnc2n(C)cc(C3CCN(CC3)C(=O)C3CCC3)c12
Cn1cc(C2CCN(CC2)C(=O)C2CCCC2)c2cc(NC(=O)c3cc(ccn3)C#N)ncc12
Cn1cc(C2CCN(CC2)C(=O)C2CCCC2)c2cc(NC(=O)c3cc(ccn3)C#N)ccc12
Cc1c(NC(=O)c2cccc(c2)C#N)cnc2n(C)cc(C3CCN(CC3)C(=O)C3CCOC3)c12
Cn1cc(c2c1ccc(c2)NC(=O)c3cc(ccn3)C#N)C4CCN(CC4)C(=O)C5CCCCC5
CC(C)C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12
Cn1cc(C2CCN(CC2)C(=O)C2CCCC2)c2cc(NC(=O)c3cccc(c3)C#N)ccc12
CC(C)C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C(C)C)c12
Cc1noc(C)c1C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12
CC(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12
Cn1cc(C2CCN(CC2)C(=O)C2CCCC2)c2nc(NC(=O)c3cc(ccn3)C#N)ccc12
O=C(Nc1ccc2[nH]cc(C3CCN(CC3)C(=O)C3CCCC3)c2c1)c1cccc(c1)C#N
CC(C)C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3ccc(F)c(c3)C#N)c(C)c12
CCC(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3cccc(c3)C#N)c(C)c12
CC(C)C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3ccc(C)c(c3)C#N)c(C)c12
Cc1c(NC(=O)c2cccc(c2)C#N)cnc2n(C)cc(C3CCN(CC3)C(=O)C3CCCCC3)c12
Cc1c(NC(=O)c2cccc(c2)C#N)cnc2n(C)cc(C3CCN(CC3)C(=O)CC3CC3)c12
Cc1c(NC(=O)c2cccc(c2)C#N)cnc2n(C)cc(C3CCN(CC3)C(=O)C3CC3)c12
Cc1c(NC(=O)c2cccc(c2)C#N)cnc2n(C)cc(C3CCN(CC3)C(=O)C3CCCC3)c12
Cn1cc(C2CCN(CC2)C(=O)C2CCCC2)c2cc(NC(=O)c3cc(ccn3)C#N)cnc12
Cn1cc(C2CCN(CC2)C(=O)C2CCCC2)c2cc(NC(=O)c3ccccc3)ccc12
CC(C)C(=O)N1CCC(CC1)c1cn(C)c2ncc(NC(=O)c3ccc(Cl)c(c3)C#N)c(C)c12
Cn1cc(C2CCN(CC2)C(=O)C2CCCC2)c2cc(NC(=O)c3cccc(c3)C#N)cnc12
Cn1cc(C2CCN(CC2)C(=O)C2CCCC2)c2nc(NC(=O)c3cc(ccn3)C#N)ncc12
CCn1cc(C2CCN(CC2)C(=O)C2CCCC2)c2cc(NC(=O)c3cc(ccn3)C#N)ccc12
CC(C)Oc1cc(Br)cc(c1)-c1ccsc1C(=O)c1ccccc1Cl
Nc1cc(c(s1)C(=O)c1ccccc1Cl)-c1cccc(c1)C(F)(F)F
FC(F)(F)c1cc(Br)cc(c1)-c1ncsc1C(=O)c1ccccc1Cl
COc1ccccc1C(=O)c1sccc1-c1cccc(c1)C(F)(F)F
COc1ccccc1C(=O)c1sc(N)cc1-c1cc(Cl)cc(Cl)c1
Clc1cc(ccn1)-c1ccsc1C(=O)c1ccccc1Cl
COc1ccccc1C(=O)c1sc(N)cc1-c1cccc(c1)C(F)(F)F
FC(F)(F)c1cccc(c1)-c1ncsc1C(=O)c1ccccc1Cl
FC(F)(F)c1cccc(c1)-c1ccsc1C(=O)c1ccccc1Cl
FC(F)(F)c1cccc(c1)-c1ccccc1C(=O)c1ccccc1Cl
Nc1ccc(C(=O)c2ccccc2Cl)c(c1)-c1cccc(c1)C(F)(F)F
Clc1ccccc1C(=O)c1sccc1-c1cccc2ccccc12
COc1ccccc1C(=O)c1sccc1-c1cccc(Cl)c1
COc1ccccc1C(=O)c1sccc1-c1ccnc(Cl)c1
Nc1cc(c(s1)C(=O)c1ccccc1Cl)-c1cc(Cl)cc(Cl)c1
COc1ccccc1C(=O)c1sc(N)cc1-c1cccc(Cl)c1
COc1ccccc1C(=O)c1sc(N)cc1-c1ccnc(Cl)c1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cccc(c2)-c2cccc(Cl)c2)cc1
CCS(=O)(=O)c1ccc(cc1)C(NC(=O)CC(C)C)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)C(NC(=O)Cc1ccccc1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)C(NC(=O)Cc1ccncn1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)C(NC(=O)c1ccccc1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)C(NC(=O)CCc1ccccc1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)C(NC(=O)Cc1ccccn1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)[C@H](C(=O)Nc2ccc(cc2)C(C(F)(F)F)(C(F)(F)F)O)NC(=O)C
CCS(=O)(=O)c1ccc(cc1)[C@H](NC(C)=O)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C(F)(F)F)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(cc1)C(NC(C)=O)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)C(NC(=O)OC)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)(C)OC)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)[C@H](O)C(F)(F)F)cc1 |r|
CCS(=O)(=O)c1ccc(cc1)C(NC(=O)NC)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)C(NS(C)(=O)=O)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)C(NC(=O)Cc1ccnnc1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
COc1ccc(cc1)C(NC(=O)c1ccc(O)nc1)C(=O)Nc1ccc(cc1)C(C)C
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2cccc(Cl)c2)cc1
CCS(=O)(=O)c1ccc(cc1)C(NC(=O)CC(C)(C)O)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C#N)(C(F)(F)F)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(cc1)C(NC(=O)Cc1cccnn1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)C(C)C)cc1
CCS(=O)(=O)c1ccc(cc1)C(N)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
Cc1c(nc(-c2ccc(Cl)o2)n1-c1c(Cl)ccc(N2CC(C2)C(O)=O)c1Cl)C(F)(F)F |(18.17,-25.5,;17.85,-27.01,;18.88,-28.15,;18.11,-29.48,;16.6,-29.16,;15.46,-30.2,;15.63,-31.73,;14.22,-32.36,;13.19,-31.22,;11.66,-31.39,;13.95,-29.89,;16.43,-27.63,;15.1,-26.86,;15.11,-25.32,;16.45,-24.56,;13.78,-24.55,;12.44,-25.32,;12.45,-26.87,;11.12,-27.65,;9.63,-27.25,;9.24,-28.74,;10.73,-29.13,;7.91,-29.51,;6.57,-28.75,;7.91,-31.05,;13.78,-27.63,;12.44,-28.39,;20.42,-28.15,;21.19,-29.48,;21.18,-26.81,;21.96,-28.15,)|
Cc1c(nc(-c2ccc(Cl)o2)n1-c1c(Cl)ccc(N2CC(C2)c2nnn[nH]2)c1Cl)C(F)(F)F |(61.88,-24.53,;61.56,-26.04,;62.59,-27.18,;61.82,-28.51,;60.31,-28.19,;59.17,-29.23,;59.34,-30.76,;57.93,-31.39,;56.9,-30.25,;55.37,-30.42,;57.66,-28.92,;60.14,-26.66,;58.81,-25.89,;58.82,-24.35,;60.16,-23.59,;57.49,-23.58,;56.15,-24.35,;56.16,-25.9,;54.83,-26.67,;53.34,-26.28,;52.95,-27.77,;54.44,-28.16,;51.62,-28.54,;51.14,-30.01,;49.6,-30.01,;49.13,-28.54,;50.37,-27.63,;57.49,-26.66,;56.15,-27.42,;64.13,-27.18,;64.9,-28.51,;64.89,-25.84,;65.67,-27.18,)|
Cc1c(nc(-c2ccc(Cl)o2)n1-c1c(Cl)ccc(NCC(C)(C)C(O)=O)c1Cl)C1(CC1)C(F)(F)F |(39.4,-36.32,;39.08,-37.83,;40.11,-38.98,;39.34,-40.31,;37.83,-39.99,;36.69,-41.03,;36.85,-42.56,;35.45,-43.19,;34.42,-42.05,;32.89,-42.21,;35.18,-40.71,;37.67,-38.46,;36.33,-37.69,;36.34,-36.15,;37.68,-35.38,;35.01,-35.37,;33.67,-36.15,;33.68,-37.7,;32.34,-38.47,;31.01,-37.7,;29.67,-38.48,;29.68,-40.02,;28.34,-39.24,;28.34,-37.71,;27.01,-38.48,;28.34,-36.17,;35.01,-38.45,;33.66,-39.21,;41.64,-38.97,;41.64,-37.43,;42.97,-38.19,;42.42,-40.31,;43.96,-40.3,;41.65,-41.64,;43.18,-41.64,)|
CC(C)Cc1nc(-c2ccco2)n(c1C)-c1c(Cl)cccc1Cl |(52.04,-6.79,;50.5,-6.79,;49.74,-8.13,;49.73,-5.46,;48.19,-5.46,;47.42,-6.8,;45.92,-6.48,;44.78,-7.52,;44.94,-9.05,;43.54,-9.68,;42.5,-8.54,;43.27,-7.2,;45.75,-4.95,;47.16,-4.32,;47.49,-2.81,;44.42,-4.18,;44.42,-2.63,;45.76,-1.87,;43.09,-1.86,;41.76,-2.63,;41.76,-4.18,;43.1,-4.95,;41.75,-5.7,)|
Cc1c(nc(-c2ccc(Cl)o2)n1-c1c(Cl)ccc(N2CC(C2)C(N)=O)c1Cl)C(F)(F)F |(37.14,-25.15,;36.82,-26.66,;37.85,-27.8,;37.08,-29.13,;35.57,-28.81,;34.43,-29.85,;34.6,-31.38,;33.19,-32.01,;32.16,-30.87,;30.63,-31.04,;32.92,-29.54,;35.4,-27.28,;34.07,-26.51,;34.08,-24.97,;35.42,-24.21,;32.75,-24.2,;31.41,-24.97,;31.42,-26.52,;30.09,-27.29,;28.6,-26.9,;28.21,-28.39,;29.7,-28.78,;26.88,-29.16,;25.54,-28.4,;26.88,-30.7,;32.75,-27.28,;31.41,-28.04,;39.39,-27.8,;40.16,-29.13,;40.15,-26.46,;40.93,-27.8,)|
CC(C)Cc1nc(-c2ccc(Cl)o2)n(c1C)-c1c(Cl)ccc(N2CC(C2)C(O)=O)c1Cl |(67.2,-18.88,;67.96,-17.55,;69.5,-17.55,;67.19,-16.22,;65.66,-16.22,;64.89,-17.55,;63.38,-17.23,;62.24,-18.27,;62.4,-19.8,;61,-20.43,;59.96,-19.29,;58.43,-19.46,;60.73,-17.96,;63.21,-15.7,;64.63,-15.08,;64.95,-13.57,;61.88,-14.93,;61.89,-13.39,;63.22,-12.63,;60.55,-12.62,;59.22,-13.39,;59.22,-14.94,;57.89,-15.71,;56.41,-15.32,;56.01,-16.81,;57.5,-17.2,;54.68,-17.58,;53.35,-16.82,;54.69,-19.12,;60.56,-15.7,;59.21,-16.46,)|
Cc1c(nc(-c2ccc(Cl)o2)n1-c1c(Cl)cccc1Cl)C(F)(F)F |(14.42,-15.48,;14.1,-16.99,;15.13,-18.13,;14.36,-19.47,;12.86,-19.15,;11.71,-20.19,;11.88,-21.72,;10.47,-22.35,;9.44,-21.21,;7.91,-21.37,;10.21,-19.87,;12.69,-17.62,;11.35,-16.85,;11.36,-15.3,;12.7,-14.54,;10.03,-14.53,;8.69,-15.31,;8.7,-16.85,;10.03,-17.62,;8.69,-18.37,;16.67,-18.13,;17.44,-19.46,;17.44,-16.79,;18.21,-18.13,)|
C[C@@H](C(=O)OC(C)C)N(c1c(cccc1Cl)Cl)C(=O)c2ccco2
Cc1c(nc(C2CC2)n1-c1c(Cl)ccc(N2CC3(CC(C3)C(O)=O)C2)c1Cl)C1(CC1)C(F)(F)F |(63.47,-36.06,;63.15,-37.56,;64.18,-38.71,;63.41,-40.04,;61.9,-39.72,;60.76,-40.76,;59.26,-41.08,;60.29,-42.22,;61.73,-38.19,;60.4,-37.42,;60.41,-35.88,;61.75,-35.11,;59.08,-35.11,;57.74,-35.88,;57.75,-37.43,;56.41,-38.2,;54.93,-37.8,;54.54,-39.29,;53.04,-38.89,;52.64,-40.38,;54.13,-40.78,;51.3,-41.15,;49.97,-40.37,;51.3,-42.69,;56.03,-39.69,;59.08,-38.19,;57.73,-38.94,;65.71,-38.7,;65.71,-37.16,;67.04,-37.93,;66.49,-40.03,;68.03,-40.03,;65.72,-41.37,;67.25,-41.36,)|
CC(C)Cc1cn(c(n1)-c1cnco1)-c1c(cccc1C#N)C#N |(32.6,-18.35,;31.06,-18.35,;30.29,-19.68,;30.29,-17.02,;28.75,-17.02,;27.72,-15.88,;26.3,-16.5,;26.47,-18.03,;27.98,-18.35,;25.33,-19.07,;25.5,-20.6,;24.09,-21.23,;23.06,-20.09,;23.82,-18.76,;24.97,-15.73,;23.65,-16.5,;22.32,-15.74,;22.31,-14.19,;23.65,-13.42,;24.98,-14.19,;26.32,-13.43,;27.65,-12.66,;22.31,-17.26,;20.96,-18.01,)|
Cc1c(Cc2ccccc2)nc(-c2ccco2)n1-c1c(Cl)cccc1Cl |(60.91,-1.41,;60.59,-2.91,;61.62,-4.06,;63.16,-4.06,;63.93,-5.39,;63.16,-6.72,;63.92,-8.05,;65.47,-8.04,;66.24,-6.71,;65.46,-5.38,;60.85,-5.39,;59.34,-5.07,;58.21,-6.11,;58.37,-7.64,;56.96,-8.27,;55.93,-7.13,;56.7,-5.79,;59.17,-3.54,;57.84,-2.77,;57.85,-1.23,;59.19,-.46,;56.51,-.45,;55.19,-1.23,;55.19,-2.78,;56.52,-3.54,;55.18,-4.3,)|
Cc1c(nc(-c2ccc(Cl)o2)n1-c1c(Cl)ccc(N2CC(CC(O)=O)C2)c1Cl)C(F)(F)F |(18.43,-36.34,;18.11,-37.85,;19.14,-38.99,;18.37,-40.33,;16.86,-40.01,;15.72,-41.05,;15.88,-42.58,;14.48,-43.21,;13.45,-42.07,;11.91,-42.23,;14.21,-40.73,;16.69,-38.48,;15.36,-37.71,;15.37,-36.16,;16.7,-35.4,;14.04,-35.39,;12.7,-36.16,;12.7,-37.71,;11.37,-38.49,;9.89,-38.09,;9.5,-39.58,;8.16,-40.36,;6.83,-39.59,;6.82,-38.05,;5.5,-40.36,;10.98,-39.97,;14.04,-38.48,;12.69,-39.23,;20.67,-38.99,;21.45,-40.32,;21.44,-37.65,;22.21,-38.99,)|
CCOC(=O)C(C)N(C(=O)c1cccs1)c1c(C)cccc1Cl
N#Cc1cccc(C#N)c1-n1cc(nc1-c1cnco1)C1CC1 |(36.26,-17.73,;37.6,-16.97,;38.94,-16.22,;37.61,-15.46,;37.6,-13.91,;38.94,-13.14,;40.27,-13.91,;41.61,-13.14,;42.95,-12.37,;40.27,-15.45,;41.6,-16.22,;43.02,-15.59,;44.05,-16.74,;43.28,-18.07,;41.77,-17.75,;40.62,-18.79,;40.79,-20.32,;39.39,-20.96,;38.35,-19.81,;39.12,-18.47,;45.59,-16.73,;46.91,-17.5,;46.91,-15.96,)|
[H][C@@]12CNc3cc(ccc3[C@@]1(CCN2C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:16.18,wD:19.25,1.0,10.28,(14.49,-6.66,;13.16,-7.44,;13.16,-5.88,;11.82,-5.1,;10.48,-5.88,;9.14,-5.12,;7.81,-5.89,;7.81,-7.43,;9.15,-8.2,;10.48,-7.44,;11.81,-8.21,;12.13,-9.73,;13.67,-9.9,;14.31,-8.49,;15.82,-8.17,;16.3,-6.71,;16.84,-9.32,;18.34,-9.01,;19.36,-10.15,;18.88,-11.62,;17.37,-11.93,;16.35,-10.79,;19.91,-12.77,;19.42,-14.24,;21.41,-12.46,;10.71,-9.29,;9.61,-10.38,;9.22,-8.89,;11.1,-10.78,;10,-11.86,;10.38,-13.35,;11.87,-13.76,;12.26,-15.25,;12.97,-12.67,;12.58,-11.19,;6.48,-5.12,;5.14,-4.35,;5.15,-5.89,;3.81,-5.12,;5.15,-7.43,;3.8,-6.65,;6.48,-3.58,;7.81,-2.81,;5.15,-2.81,;6.47,-2.04,)|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)Cc1ccccc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:16.18,wD:19.25,1.0,10.28,(38.9,-47.28,;37.57,-48.06,;37.57,-46.51,;36.22,-45.72,;34.88,-46.5,;33.55,-45.74,;32.22,-46.51,;32.22,-48.05,;33.55,-48.82,;34.88,-48.06,;36.22,-48.83,;36.53,-50.35,;38.08,-50.52,;38.72,-49.11,;40.23,-48.8,;40.71,-47.34,;41.25,-49.95,;42.74,-49.63,;43.77,-50.78,;43.29,-52.25,;41.78,-52.56,;40.75,-51.41,;44.31,-53.4,;43.83,-54.86,;45.82,-53.08,;35.12,-49.92,;34.02,-51.01,;33.62,-49.51,;35.5,-51.41,;34.4,-52.49,;32.93,-52.07,;31.83,-53.15,;32.21,-54.64,;33.71,-55.05,;34.8,-53.97,;30.89,-45.74,;29.55,-44.97,;29.55,-46.51,;28.22,-45.74,;29.55,-48.05,;28.21,-47.27,;30.89,-44.2,;32.22,-43.43,;29.55,-43.43,;30.88,-42.66,)|
[H][C@@]12COc3cc(ccc3[C@@]1(CCN2C(=O)C1(O)CCS(=O)(=O)CC1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CN(C)c3cc(ccc3[C@@]1(CCN2C(=O)C1(O)CCS(=O)(=O)CC1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CNc3cc(ccc3[C@@]1(CCN2C(=O)C1(O)CCS(=O)(=O)CC1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12COc3cc(ccc3[C@@]1(CCN2C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:16.18,wD:19.25,1.0,10.28,(38.73,-26.8,;37.4,-27.58,;37.4,-26.03,;36.05,-25.25,;34.71,-26.03,;33.38,-25.26,;32.05,-26.03,;32.05,-27.58,;33.38,-28.35,;34.71,-27.58,;36.05,-28.35,;36.36,-29.88,;37.91,-30.05,;38.55,-28.63,;40.06,-28.32,;40.54,-26.86,;41.08,-29.47,;42.57,-29.15,;43.6,-30.3,;43.12,-31.77,;41.61,-32.08,;40.58,-30.93,;44.14,-32.92,;43.66,-34.38,;45.65,-32.6,;34.95,-29.44,;33.85,-30.53,;33.45,-29.03,;35.33,-30.93,;34.23,-32.01,;34.62,-33.49,;36.11,-33.91,;36.49,-35.4,;37.21,-32.82,;36.81,-31.33,;30.72,-25.26,;29.38,-24.49,;29.38,-26.03,;28.05,-25.26,;29.38,-27.57,;28.04,-26.79,;30.72,-23.72,;32.05,-22.95,;29.38,-22.95,;30.71,-22.18,)|
[H][C@@]12CN(C)c3cc(ccc3[C@@]1(CCN2C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:17.19,wD:20.26,1.0,11.29,(37.5,-6.4,;36.17,-7.18,;36.17,-5.63,;34.82,-4.84,;34.82,-3.3,;33.48,-5.62,;32.15,-4.86,;30.82,-5.63,;30.82,-7.18,;32.15,-7.95,;33.48,-7.18,;34.82,-7.95,;35.13,-9.47,;36.68,-9.65,;37.32,-8.23,;38.83,-7.92,;39.31,-6.46,;39.85,-9.07,;41.34,-8.75,;42.37,-9.9,;41.89,-11.37,;40.38,-11.68,;39.35,-10.53,;42.91,-12.52,;42.43,-13.98,;44.42,-12.2,;33.72,-9.04,;32.62,-10.13,;32.22,-8.63,;34.1,-10.53,;33,-11.6,;33.39,-13.09,;34.88,-13.5,;35.26,-14.99,;35.98,-12.42,;35.58,-10.93,;29.49,-4.86,;28.15,-4.09,;28.15,-5.63,;26.82,-4.86,;28.15,-7.17,;26.81,-6.39,;29.49,-3.32,;30.82,-2.55,;28.15,-2.55,;29.48,-1.78,)|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1cccc(C)c1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:16.18,wD:19.25,1.0,10.28,(65.64,-25.66,;64.32,-26.44,;64.32,-24.89,;62.97,-24.1,;61.63,-24.88,;60.3,-24.12,;58.97,-24.89,;58.97,-26.43,;60.3,-27.2,;61.63,-26.44,;62.97,-27.21,;63.28,-28.73,;64.83,-28.9,;65.47,-27.49,;66.97,-27.18,;67.46,-25.71,;68,-28.33,;69.49,-28.01,;70.52,-29.15,;70.04,-30.63,;68.53,-30.94,;67.5,-29.79,;71.06,-31.77,;70.58,-33.24,;72.57,-31.46,;61.86,-28.3,;60.77,-29.38,;60.37,-27.89,;62.25,-29.79,;61.15,-30.86,;61.54,-32.35,;63.02,-32.76,;64.12,-31.67,;65.61,-32.08,;63.73,-30.19,;57.63,-24.12,;56.29,-23.35,;56.3,-24.89,;54.97,-24.12,;56.3,-26.43,;54.96,-25.65,;57.63,-22.58,;58.97,-21.81,;56.3,-21.81,;57.62,-21.04,)|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1cccc(F)c1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:16.18,wD:19.25,1.0,10.28,(15.64,-25.66,;14.31,-26.44,;14.32,-24.88,;12.97,-24.1,;11.63,-24.88,;10.29,-24.12,;8.96,-24.89,;8.96,-26.43,;10.3,-27.2,;11.63,-26.44,;12.96,-27.21,;13.28,-28.73,;14.82,-28.9,;15.46,-27.49,;16.97,-27.17,;17.45,-25.71,;17.99,-28.33,;19.49,-28.01,;20.51,-29.15,;20.03,-30.62,;18.52,-30.94,;17.5,-29.79,;21.06,-31.77,;20.57,-33.24,;22.56,-31.46,;11.86,-28.29,;10.76,-29.38,;10.37,-27.89,;12.25,-29.78,;11.15,-30.86,;11.54,-32.35,;13.02,-32.76,;14.12,-31.67,;15.61,-32.08,;13.73,-30.19,;7.63,-24.12,;6.29,-23.35,;6.3,-24.89,;4.96,-24.12,;6.3,-26.43,;4.95,-25.65,;7.63,-22.58,;8.96,-21.81,;6.3,-21.81,;7.62,-21.04,)|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1ccc(C)cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:16.18,wD:19.25,1.0,10.28,(64.23,-6.6,;62.9,-7.39,;62.9,-5.83,;61.56,-5.05,;60.21,-5.83,;58.88,-5.06,;57.55,-5.83,;57.55,-7.38,;58.88,-8.15,;60.21,-7.38,;61.55,-8.15,;61.86,-9.68,;63.41,-9.85,;64.05,-8.43,;65.56,-8.12,;66.04,-6.66,;66.58,-9.27,;68.07,-8.96,;69.1,-10.1,;68.62,-11.57,;67.11,-11.88,;66.09,-10.73,;69.64,-12.72,;69.16,-14.18,;71.15,-12.41,;60.45,-9.24,;59.35,-10.33,;58.96,-8.83,;60.83,-10.73,;59.74,-11.81,;60.12,-13.3,;61.61,-13.71,;62,-15.2,;62.71,-12.62,;62.32,-11.13,;56.22,-5.06,;54.88,-4.29,;54.88,-5.83,;53.55,-5.06,;54.88,-7.37,;53.54,-6.6,;56.22,-3.52,;57.55,-2.75,;54.88,-2.75,;56.21,-1.98,)|
[H][C@@]12CN(CCC)c3cc(ccc3[C@@]1(CCN2C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:19.21,wD:22.28,1.0,13.31,(13.85,-27.45,;12.52,-28.23,;12.53,-26.67,;11.18,-25.89,;11.18,-24.35,;12.51,-23.58,;12.51,-22.04,;9.84,-26.67,;8.5,-25.91,;7.18,-26.68,;7.17,-28.22,;8.51,-28.99,;9.84,-28.22,;11.17,-29,;11.49,-30.52,;13.03,-30.69,;13.67,-29.28,;15.18,-28.96,;15.67,-27.5,;16.21,-30.11,;17.7,-29.8,;18.73,-30.94,;18.24,-32.41,;16.73,-32.72,;15.71,-31.57,;19.27,-33.56,;18.79,-35.02,;20.78,-33.25,;10.07,-30.08,;8.98,-31.17,;8.58,-29.68,;10.46,-31.57,;9.36,-32.65,;9.75,-34.14,;11.23,-34.55,;11.62,-36.04,;12.33,-33.46,;11.94,-31.98,;5.84,-25.91,;4.5,-25.14,;4.51,-26.68,;3.17,-25.91,;4.51,-28.22,;3.17,-27.44,;5.84,-24.37,;7.18,-23.6,;4.51,-23.6,;5.83,-22.83,)|
[H][C@@]12CN(CC)c3cc(ccc3[C@@]1(CCN2C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:18.20,wD:21.27,1.0,12.30,(63.95,-6.23,;62.62,-7.01,;62.62,-5.46,;61.28,-4.67,;61.28,-3.13,;62.61,-2.36,;59.93,-5.45,;58.6,-4.69,;57.27,-5.46,;57.27,-7,;58.6,-7.77,;59.93,-7.01,;61.27,-7.78,;61.58,-9.3,;63.13,-9.47,;63.77,-8.06,;65.28,-7.75,;65.76,-6.29,;66.3,-8.9,;67.79,-8.58,;68.82,-9.73,;68.34,-11.2,;66.83,-11.51,;65.81,-10.36,;69.36,-12.35,;68.88,-13.81,;70.87,-12.03,;60.17,-8.87,;59.07,-9.96,;58.68,-8.46,;60.55,-10.36,;59.46,-11.43,;59.84,-12.92,;61.33,-13.33,;61.72,-14.82,;62.43,-12.24,;62.04,-10.76,;55.94,-4.69,;54.6,-3.92,;54.6,-5.46,;53.27,-4.69,;54.6,-7,;53.26,-6.22,;55.94,-3.15,;57.27,-2.38,;54.6,-2.38,;55.93,-1.61,)|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:16.18,19.25,wD:1.0,10.28,(65.23,-46.28,;63.9,-47.07,;63.9,-45.51,;62.56,-44.73,;61.22,-45.51,;59.88,-44.74,;58.55,-45.51,;58.55,-47.06,;59.89,-47.83,;61.22,-47.06,;62.55,-47.83,;62.87,-49.36,;64.41,-49.53,;65.05,-48.11,;66.56,-47.8,;67.04,-46.34,;67.58,-48.95,;67.09,-50.41,;68.11,-51.56,;69.62,-51.25,;70.1,-49.78,;69.08,-48.64,;70.65,-52.4,;70.16,-53.86,;72.15,-52.09,;61.45,-48.92,;60.35,-50.01,;59.96,-48.51,;61.84,-50.41,;60.74,-51.49,;61.12,-52.98,;62.61,-53.39,;63,-54.88,;63.71,-52.3,;63.32,-50.81,;57.22,-44.74,;55.88,-43.97,;55.89,-45.51,;54.55,-44.74,;55.89,-47.05,;54.54,-46.28,;57.22,-43.2,;58.55,-42.43,;55.89,-42.43,;57.21,-41.66,)|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1cccc(Cl)c1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:16.18,wD:19.25,1.0,10.28,(39.24,-25.54,;37.91,-26.32,;37.91,-24.77,;36.57,-23.98,;35.23,-24.76,;33.89,-24,;32.56,-24.77,;32.56,-26.32,;33.89,-27.09,;35.22,-26.32,;36.56,-27.09,;36.87,-28.61,;38.42,-28.79,;39.06,-27.37,;40.57,-27.06,;41.05,-25.6,;41.59,-28.21,;43.09,-27.89,;44.11,-29.04,;43.63,-30.51,;42.12,-30.82,;41.1,-29.67,;44.65,-31.66,;44.17,-33.12,;46.16,-31.34,;35.46,-28.18,;34.36,-29.27,;33.97,-27.77,;35.84,-29.67,;34.75,-30.74,;35.13,-32.23,;36.62,-32.65,;37.72,-31.56,;39.2,-31.96,;37.33,-30.07,;31.23,-24,;29.89,-23.23,;29.89,-24.77,;28.56,-24,;29.89,-26.31,;28.55,-25.53,;31.23,-22.46,;32.56,-21.69,;29.89,-21.69,;31.22,-20.92,)|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1ccc(Cl)cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:16.18,wD:19.25,1.0,10.28,(39.12,-6.49,;37.79,-7.27,;37.79,-5.71,;36.45,-4.93,;35.11,-5.71,;33.77,-4.95,;32.44,-5.72,;32.44,-7.26,;33.78,-8.03,;35.11,-7.26,;36.44,-8.04,;36.76,-9.56,;38.3,-9.73,;38.94,-8.31,;40.45,-8,;40.93,-6.54,;41.47,-9.15,;42.97,-8.84,;43.99,-9.98,;43.51,-11.45,;42,-11.76,;40.98,-10.61,;44.54,-12.6,;44.05,-14.06,;46.04,-12.29,;35.34,-9.12,;34.24,-10.21,;33.85,-8.72,;35.73,-10.61,;34.63,-11.69,;35.01,-13.18,;36.5,-13.59,;36.89,-15.08,;37.6,-12.5,;37.21,-11.02,;31.11,-4.95,;29.77,-4.18,;29.78,-5.72,;28.44,-4.95,;29.78,-7.26,;28.43,-6.48,;31.11,-3.41,;32.44,-2.64,;29.78,-2.64,;31.1,-1.87,)|
OC(=O)c1ccc(cc1Cl)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
OC(=O)c1ccc(-c2cn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cccnc23)c(F)c1
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12 |c:6|
OC(=O)c1ccc(cc1)-c1nn(Cc2c(Cl)cccc2Cl)c2ccccc12
OC(=O)c1ccc(cc1F)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
Nc1cc(ccc1C(O)=O)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
COc1cc(ccc1C(O)=O)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cccc(F)c23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cccc(F)c23)c(Cl)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cnccc23)c(F)c1
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cncnc23)c(F)c1
O[C@H]1CN(CC[C@H]1C(O)=O)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12 |r|
CC(C)Oc1cccc(Cl)c1C(=O)n1nc(-c2ccc(cc2)C(O)=O)c2ccccc12
OC(=O)c1ccc(cc1)-c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cccnc23)c(F)c1
OC(=O)c1ccc(cc1)-c1nn(c2ccccc12)S(=O)(=O)c1c(Cl)cccc1Cl
OC(=O)C1CCC(=CC1)c1nn(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccnc12 |c:6|
C[C@H]1CN(CCN1C(=O)C1CCCC1)C1CCc2ccc(NC(=O)c3cccc(c3)C#N)cc12 |r|
Cc1ncc(cc1F)C(=O)Nc1cccc2C(CCc12)N1CC2CCC(C1)N2C(=O)C1CCCC1
Cc1ncc(cc1F)C(=O)Nc1ccc2CCC(N3CC4CCC(C3)N4C(=O)C3CCCC3)c2c1
O=C(Nc1ccc2CCC(N3CC4CCC(C3)N4C(=O)C3CCCC3)c2c1)Nc1cccc(c1)C#N
O=C(Nc1cccc2C(CCc12)N1CC2CCC(C1)N2C(=O)C1CCCCC1)c1cccc(c1)C#N
O=C(CC1CCC1)N1C2CCC1CN(C2)C1CCc2c1cccc2NC(=O)c1cccc(c1)C#N
Cc1ccc(cn1)C(=O)Nc1cccc2C(CCc12)N1CC2CCC(C1)N2C(=O)C1CCCC1
O=C(Nc1cccc(c1)C#N)Nc1cccc2C(CCc12)N1CC2CCC(C1)N2C(=O)C1CCCC1
O=C(Nc1ccc2CCC(N3CCN(CC3)C(=O)C3CCCC3)c2c1)c1cccc(c1)C#N
O=C(Nc1cccc2C(CCc12)N1CCN(CC1)C(=O)C1CCCC1)c1cccc(c1)C#N
O=C(C1CCCC1)N1C2CCC1CN(C2)C1CCc2ccc(NC(=O)c3cccc(c3)C#N)cc12
O=C(Nc1ccc2CCC(N3CC4CCC(C3)N4C(=O)C3CCCCC3)c2c1)c1cccc(c1)C#N
O=C(Nc1ccc2CC[C@H](N3CC4CCC(C3)N4C(=O)C3CCCCC3)c2c1)c1cccc(c1)C#N |r|
O=C(Nc1cccc(CN2CCN(CC2)C(=O)C2CCCC2)c1)c1cccc(c1)C#N
O=C(Nc1ccc2CCN(C3CCN(CC3)C(=O)C3CCCC3)c2c1)c1cccc(c1)C#N
O=C(Nc1ccc2ccn(C3CCN(CC3)C(=O)C3CCCC3)c2c1)c1cccc(c1)C#N
O=C(Nc1cccc2N(CCc12)C1CCN(CC1)C(=O)C1CCCC1)c1cccc(c1)C#N
C[C@H]1CN(C[C@@H](C)N1C(=O)C1CCCC1)C1CCc2ccc(NC(=O)c3cccc(c3)C#N)cc12 |r|
C[C@H]1CN(CCN1C(=O)C1CCCC1)C1CCc2c1cccc2NC(=O)c1cccc(c1)C#N |r|
C[C@H]1CN(C[C@@H](C)N1C(=O)C1CCCC1)C1CCc2c1cccc2NC(=O)c1cccc(c1)C#N |r|
O=C(Nc1ccc2CCC(N3CC4CCC(C3)N4C(=O)C3CCC3)c2c1)c1cccc(c1)C#N
O=C(CC1CCC1)N1C2CCC1CN(C2)C1CCc2ccc(NC(=O)c3cccc(c3)C#N)cc12
Cc1ccc(cn1)C(=O)Nc1ccc2CCC(N3CC4CCC(C3)N4C(=O)C3CCCC3)c2c1
O=C(Nc1cccc2C(CCc12)N1CC2CCC(C1)N2C(=O)C1CCC1)c1cccc(c1)C#N
O=C(CC1CCOCC1)Nc1cccc2C(CCc12)N1CC2CCC(C1)N2C(=O)C1CCCC1
O=C(C1CCCC1)N1C2CCC1CN(C2)C1CCc2c1cccc2NC(=O)c1cccc(c1)C#N
O=C(CC1CCOCC1)Nc1ccc2CCC(N3CC4CCC(C3)N4C(=O)C3CCCC3)c2c1
C[C@@H]1CN(CCN1C(=O)C1CCCC1)C1CCc2ccc(NC(=O)c3cccc(c3)C#N)cc12 |r|
C[C@@H]1CN(CCN1C(=O)C1CCCC1)C1CCc2c1cccc2NC(=O)c1cccc(c1)C#N |r|
Cn1cc(C2CCN(CC2)C(=O)C2CCCC2)c2cccc(NC(=O)c3cccc(c3)C#N)c12
OC(=O)[C@H]1CC[C@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:14.17,wD:6.9,3.2,(.2,-10.82,;-.7,-9.58,;-2.23,-9.74,;-.07,-8.17,;1.46,-8.01,;2.08,-6.6,;1.18,-5.36,;-.35,-5.52,;-.98,-6.92,;1.8,-3.95,;3.34,-3.79,;.9,-2.7,;-.64,-2.7,;-1.12,-1.24,;.13,-.33,;1.38,-1.24,;-.9,.81,;-.43,2.28,;-1.46,3.42,;-2.96,3.1,;-3.44,1.64,;-2.41,.49,;-3.99,4.24,;-5.02,5.39,;-5.14,3.21,;-6.28,2.18,;-6.17,4.36,;-4.11,2.07,;-2.85,5.28,;-1.7,6.31,;-1.82,4.13,;-3.88,6.42,;1.16,.81,;2.3,-.22,;.02,1.84,;2.19,1.96,;1.71,3.42,;2.74,4.56,;4.25,4.24,;5.28,5.39,;4.73,2.78,;3.7,1.64,)|
COC(=O)N1CCC(C1)(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)c(c1)C1CC1 |r,wU:14.17,3.2,wD:6.9,(2.94,11.52,;3.42,10.06,;4.92,9.74,;2.39,8.91,;2.86,7.45,;1.83,6.3,;.32,6.62,;-.15,8.09,;.88,9.23,;-.71,5.48,;-2.21,5.8,;-.23,4.01,;1.23,3.54,;1.23,2,;-.23,1.52,;-1.14,2.77,;.4,.12,;-.51,-1.13,;.12,-2.54,;1.65,-2.7,;2.55,-1.45,;1.93,-.05,;2.28,-4.11,;2.9,-5.51,;3.68,-3.48,;5.09,-2.85,;4.31,-4.89,;3.06,-2.07,;.87,-4.73,;-.54,-5.36,;.24,-3.32,;1.5,-6.14,;-1.56,.75,;-2.33,2.09,;-.79,-.58,;-2.9,-.02,;-4.23,.75,;-5.56,-.02,;-5.56,-1.56,;-6.9,-2.33,;-4.23,-2.33,;-2.9,-1.56,;-4.23,-3.87,;-3.46,-5.2,;-5,-5.2,)|
CCc1cc(ccc1F)S(=O)(=O)[C@]1(CCN(C1)C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:12.30,22.27,wD:19.20,(3.42,7.12,;2.39,5.97,;2.86,4.51,;1.83,3.36,;2.31,1.9,;3.82,1.58,;4.85,2.72,;4.37,4.19,;5.4,5.33,;1.28,.75,;2.42,-.28,;.14,1.78,;.25,-.39,;-1,-1.3,;-.52,-2.76,;1.02,-2.76,;1.5,-1.3,;1.92,-4.01,;3.46,-3.85,;1.3,-5.41,;-.23,-5.57,;-.86,-6.98,;.05,-8.23,;1.58,-8.07,;2.2,-6.66,;-.58,-9.63,;.32,-10.88,;-2.11,-9.79,;-.78,.75,;-.31,2.22,;-1.34,3.36,;-2.84,3.04,;-3.32,1.58,;-2.29,.43,;-3.87,4.19,;-4.9,5.33,;-5.02,3.16,;-6.16,2.13,;-6.05,4.3,;-3.99,2.01,;-2.73,5.22,;-1.58,6.25,;-1.7,4.07,;-3.76,6.36,)|
COc1ccc(cc1)S(=O)(=O)[C@]1(CCN(C1)C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:11.29,21.26,wD:18.19,(4.86,6.61,;5.33,5.15,;4.3,4,;2.8,4.32,;1.76,3.18,;2.24,1.72,;3.75,1.4,;4.78,2.54,;1.21,.57,;2.35,-.46,;.07,1.6,;.18,-.57,;-1.07,-1.48,;-.59,-2.94,;.95,-2.94,;1.43,-1.48,;1.85,-4.19,;3.39,-4.03,;1.23,-5.6,;-.3,-5.76,;-.93,-7.16,;-.02,-8.41,;1.51,-8.25,;2.13,-6.84,;-.65,-9.82,;.25,-11.06,;-2.18,-9.98,;-.85,.57,;-.37,2.04,;-1.41,3.18,;-2.91,2.86,;-3.39,1.4,;-2.36,.25,;-3.94,4,;-4.97,5.15,;-2.8,5.04,;-1.77,3.89,;-3.83,6.18,;-1.65,6.07,;-5.09,2.97,;-6.23,1.94,;-6.12,4.12,;-4.06,1.83,)|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(Cl)cc1 |r,wU:14.17,3.2,wD:6.9,(-2.42,-10.14,;-.89,-9.98,;.01,-11.22,;-.27,-8.57,;-1.17,-7.33,;-.54,-5.92,;.99,-5.76,;1.89,-7,;1.27,-8.41,;1.61,-4.35,;3.15,-4.19,;.71,-3.11,;-.83,-3.11,;-1.31,-1.64,;-.06,-.74,;1.18,-1.64,;-.82,.61,;-2.36,.62,;-3.11,1.96,;-2.33,3.29,;-.79,3.27,;-.03,1.93,;-3.09,4.63,;-3.84,5.97,;-4.43,3.88,;-5.77,3.12,;-5.18,5.22,;-3.67,2.53,;-1.74,5.39,;-.4,6.14,;-.99,4.05,;-2.5,6.73,;.69,.61,;.52,2.14,;2.04,-.15,;1.45,1.95,;.67,3.27,;1.42,4.61,;2.96,4.63,;3.72,5.97,;3.75,3.31,;2.99,1.96,)|
Cc1ccc(cc1)S(=O)(=O)[C@]1(CCN(C1)C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:10.28,20.25,wD:17.18,(3.72,5.97,;2.96,4.63,;1.42,4.61,;.67,3.27,;1.45,1.95,;2.99,1.96,;3.75,3.31,;.69,.61,;.52,2.14,;2.04,-.15,;-.06,-.74,;-1.31,-1.64,;-.83,-3.11,;.71,-3.11,;1.18,-1.64,;1.61,-4.35,;3.15,-4.19,;.99,-5.76,;-.54,-5.92,;-1.17,-7.33,;-.27,-8.57,;1.27,-8.41,;1.89,-7,;-.89,-9.98,;-2.42,-10.14,;.01,-11.22,;-.82,.61,;-2.36,.62,;-3.11,1.96,;-2.33,3.29,;-.79,3.27,;-.03,1.93,;-3.09,4.63,;-3.84,5.97,;-4.43,3.88,;-5.77,3.12,;-5.18,5.22,;-3.67,2.53,;-1.74,5.39,;-.4,6.14,;-.99,4.05,;-2.5,6.73,)|
OC(=O)C1CCN(CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
c1cc(ccc1[C@@]2(CCN(C2)C(=O)C3CCC(CC3)C(=O)O)S(=O)(=O)c4ccc(cc4)F)C(C(F)(F)F)(C(F)(F)F)F
CC(=O)N1CCN(CC1)C(=O)N1CC[C@@](C1)(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCN(CC1)C(=O)N2CC[C@](C2)(c3ccc(cc3)C(C(F)(F)F)(C(F)(F)F)O)S(=O)(=O)c4ccc(cc4)F
CS(=O)(=O)N1CCC(CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CCNC(=O)N1CCC(C1)(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
CC(=O)N1CCC(C1)(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1
OC(c1ccc(cc1)[C@@]1(CCNC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F |r|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:14.17,3.2,wD:6.9,(-2.42,-10.14,;-.89,-9.98,;.01,-11.22,;-.27,-8.57,;-1.17,-7.33,;-.54,-5.92,;.99,-5.76,;1.89,-7,;1.27,-8.41,;1.61,-4.35,;3.15,-4.19,;.71,-3.11,;-.83,-3.11,;-1.31,-1.64,;-.06,-.74,;1.18,-1.64,;-.82,.61,;-2.36,.62,;-3.11,1.96,;-2.33,3.29,;-.79,3.27,;-.03,1.93,;-3.09,4.63,;-3.84,5.97,;-4.43,3.88,;-5.77,3.12,;-5.18,5.22,;-3.67,2.53,;-1.74,5.39,;-.4,6.14,;-.99,4.05,;-2.5,6.73,;.69,.61,;.52,2.14,;2.04,-.15,;1.45,1.95,;.67,3.27,;1.42,4.61,;2.96,4.63,;3.72,5.97,;3.75,3.31,;2.99,1.96,)|
CCc1ccc(cc1)S(=O)(=O)[C@]1(CCN(C1)C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:11.29,21.26,wD:18.19,(1.07,7.43,;.18,6.18,;.82,4.78,;-.07,3.52,;.57,2.12,;2.1,1.98,;3,3.23,;2.35,4.63,;2.74,.58,;4.15,1.22,;3.39,-.82,;1.34,-.06,;.1,-.97,;.57,-2.43,;2.11,-2.43,;2.59,-.97,;3.02,-3.68,;4.55,-3.52,;2.39,-5.09,;.86,-5.25,;.24,-6.65,;1.14,-7.9,;2.67,-7.74,;3.3,-6.33,;.51,-9.31,;-1.02,-9.47,;1.42,-10.55,;-.06,.58,;-1.31,-.31,;-2.71,.33,;-2.86,1.86,;-1.6,2.75,;-.2,2.11,;-4.26,2.5,;-4.9,1.1,;-3.62,3.9,;-2.97,5.3,;-2.21,3.26,;-5.02,4.54,;-5.66,3.14,;-5.96,4.65,;-6.3,1.74,;-7.06,3.78,)|
CC(=O)N1CCC(CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCN(CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Cc1cc(ccc1F)S(=O)(=O)[C@]1(CCN(C1)C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:11.29,21.26,wD:18.19,(2.32,6.24,;2.8,4.77,;1.77,3.63,;2.25,2.16,;3.75,1.84,;4.78,2.99,;4.31,4.45,;5.34,5.6,;1.22,1.02,;2.36,-.01,;.07,2.05,;.18,-.12,;-1.06,-1.03,;-.59,-2.49,;.95,-2.49,;1.43,-1.03,;1.86,-3.74,;3.39,-3.58,;1.23,-5.15,;-.3,-5.31,;-.92,-6.71,;-.02,-7.96,;1.51,-7.8,;2.14,-6.39,;-.65,-9.37,;.26,-10.61,;-2.18,-9.53,;-.85,1.02,;-.37,2.48,;-1.4,3.63,;-2.91,3.31,;-3.38,1.84,;-2.35,.7,;-3.94,4.45,;-4.97,5.6,;-5.08,3.42,;-6.23,2.39,;-6.11,4.57,;-4.05,2.28,;-2.79,5.48,;-1.65,6.51,;-1.76,4.34,;-3.82,6.63,)|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccccc1 |r,wU:6.9,wD:14.17,3.2,(67.73,-20.71,;66.4,-21.49,;66.4,-23.03,;65.06,-20.73,;65.05,-19.18,;63.71,-18.42,;62.39,-19.2,;62.39,-20.75,;63.73,-21.5,;61.05,-18.44,;61.03,-16.9,;59.72,-19.22,;58.47,-18.32,;57.23,-19.22,;57.7,-20.69,;59.24,-20.69,;56.16,-20.68,;55.37,-22.01,;53.84,-22,;53.08,-20.65,;53.85,-19.33,;55.39,-19.34,;51.54,-20.64,;50.76,-21.97,;51.55,-19.1,;52.89,-18.34,;50.22,-18.32,;51.55,-17.55,;50.21,-19.86,;49.44,-18.52,;49.1,-20.94,;48.67,-19.84,;57.69,-22.23,;56.92,-23.56,;56.15,-22.22,;59.02,-23.01,;59.01,-24.54,;60.34,-25.32,;61.68,-24.55,;61.68,-23.01,;60.35,-22.24,)|
CS(=O)(=O)N1CCC(CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(c1ccc(cc1)[C@]1(CCNC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F |r|
OC(c1ccc(cc1)C1(CCN(C1)C(=O)C1CCCC1)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F
CC(=O)N1CCC(CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)C(O)(C1CN(C1)C(C)=O)c1ccc(nc1)C(F)(F)F
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)n1cccn1)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)C(O)(C1CN(C1)C(C)=O)c1cnnn1C
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)C(O)(c1cnc(C)n1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1CC(F)(F)F)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1CC1CCC(F)(F)CC1)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1OC(C)C)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1CN1CC(C1)C(F)(F)F)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1CN1CCC(F)CC1)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)C(O)(c1cnnn1C)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1OCc1nccs1)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)C(O)(c1cnnn1C)c1cc(C)nc(C)c1
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)C(O)(c1cncn1C)c1ccnc(c1)C(F)(F)F
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)C(O)(C1CCOCC1)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)C(O)(c1cnnn1C)c1ccc(C)nc1C
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)C(O)(c1cnnn1C)c1ccnc(c1)C(F)(F)F
COc1nc2ccc(cc2c(Cl)c1CN1CCC(CC1)C(F)(F)F)C(O)(C1CN(C1)C(C)=O)c1cnc(C)n1C
COc1nc2ccc(cc2c(Cl)c1CC1CCS(=O)(=O)CC1)C(O)(c1cnnn1C)c1ccc(C)nc1C
C[C@H]1CN(Cc2c(C)c(NC(=O)c3ccc(C)nc3)cn3ncnc23)CCN1C(=O)C1CCCC1 |r|
C[C@H]1C[C@@H](CCN1C(=O)CC(C(F)(F)F)C(F)(F)F)Oc1c(C)c(NC(=O)c2ccc(C)nc2)cn2ncnc12 |r|
C[C@H]1C[C@H](CCN1C(=O)CC(C(F)(F)F)C(F)(F)F)Oc1c(C)c(NC(=O)c2ccc(C)nc2)cn2ncnc12 |r|
C[C@H]1CN(Cc2c(C)c(NC(=O)c3ccc(C)nc3)cc3nnc(C)n23)CCN1C(=O)C1CCCC1 |r|
C[C@H]1CN(Cc2c(C)c(NC(=O)c3ccc(C)nc3)cn3nc(C)nc23)CCN1C(=O)C1CCCC1 |r|
C[C@H]1CN(Cc2c(C)c(NC(=O)c3ccc(C)nc3)cn3ncnc23)CCN1C(=O)C1CCC(F)(F)C1 |r|
CC(C)CC(=O)N1CCN(Cc2c(C)c(NC(=O)c3ccc(C)nc3)cn3ncnc23)C[C@@H]1C |r|
C[C@H]1CN(Cc2c(C)c(NC(=O)c3ccc(C)nc3)cn3ncnc23)CCN1C(=O)CC(C(F)(F)F)C(F)(F)F |r|
C[C@H]1CN(Cc2cc(F)cc(NC(=O)c3ccc(C)nc3)c2C)CCN1C(=O)C1CCCC1 |r|
C[C@H]1CN(Cc2c(C)c(NC(=O)c3ccc(C)nc3)cn3ncnc23)CCN1C(=O)c1ccccc1 |r|
C[C@H]1CN(Cc2c(C)c(NC(=O)c3ccc(C)nc3)cn3ncnc23)CCN1C(=O)CCC(F)(F)F |r|
C[C@H]1CN(Cc2c(C)c(NC(=O)c3ccc(C)nc3)cc3nncn23)CCN1C(=O)C1CCCC1 |r|
CC(C)C(=O)N1CCN(Cc2c(C)c(NC(=O)c3ccc(C)nc3)cn3ncnc23)C[C@@H]1C |r|
C[C@H]1CN(Cc2c(C)c(NC(=O)c3ccc(C)nc3)cn3ncnc23)CCN1C(=O)C1CCOCC1 |r|
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2cccnc12
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2cccc(Cl)c12
Cc1cccc(Cl)c1C(=O)c1cn(-c2ccc(cc2)C(O)=O)c2c(F)cccc12
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2ccccc12
OC(=O)c1ccc(c(Cl)c1)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2ccccc12
OC(=O)c1ccc(cc1)-n1nc(C(=O)c2c(Cl)cccc2Cl)c2ccccc12
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2c(F)cccc2Cl)c2ccccc12
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2c(F)cccc12
COc1cccc2c(cn(-c3ccc(cc3)C(O)=O)c12)C(=O)c1c(Cl)cccc1Cl
Cc1cccc2c(cn(-c3ccc(cc3F)C(O)=O)c12)C(=O)c1ccccc1Cl
OC(=O)c1ccc(c(F)c1)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2ccccc12
OC(=O)c1ccc(c(c1)C(F)(F)F)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2ccccc12
OC(=O)c1ccc(cc1F)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2ccccc12
OC(=O)c1ccc(c(F)c1F)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2ccccc12
OC(=O)c1cc(F)c(c(F)c1)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2ccccc12 |(10.56,-42.93,;9.05,-43.26,;8.01,-42.12,;8.59,-44.73,;9.62,-45.87,;9.16,-47.33,;10.19,-48.47,;7.65,-47.65,;6.62,-46.53,;5.11,-46.86,;7.08,-45.06,;7.18,-49.12,;8.1,-50.36,;7.2,-51.62,;7.68,-53.08,;6.66,-54.23,;9.19,-53.39,;10.2,-52.24,;9.71,-50.78,;11.7,-52.54,;12.2,-54.01,;11.17,-55.16,;9.66,-54.85,;8.64,-56,;5.73,-51.15,;4.39,-51.93,;3.05,-51.16,;3.05,-49.61,;4.38,-48.84,;5.72,-49.61,)|
OC(=O)c1cc(Cl)c(c(Cl)c1)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2ccccc12 |(22.37,-42.13,;20.87,-42.46,;19.83,-41.32,;20.4,-43.93,;21.44,-45.07,;20.97,-46.53,;22.01,-47.68,;19.46,-46.85,;18.43,-45.73,;16.93,-46.06,;18.89,-44.26,;19,-48.32,;19.91,-49.56,;19.01,-50.82,;19.5,-52.28,;18.47,-53.43,;21,-52.59,;22.01,-51.44,;21.52,-49.98,;23.52,-51.75,;24.01,-53.21,;22.99,-54.36,;21.48,-54.05,;20.45,-55.2,;17.54,-50.35,;16.2,-51.13,;14.87,-50.36,;14.87,-48.81,;16.2,-48.04,;17.53,-48.81,)|
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2c(F)cccc2F)c2ccccc12
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2c(Cl)cc(Cl)cc2Cl)c2ccccc12
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2ccccc2Cl)c2ccccc12
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2ccc(F)cc12
Cc1cccc(Cl)c1C(=O)c1cn(-c2ccc(cc2F)C(O)=O)c2ncccc12
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccc(F)c12
OC(=O)c1ccc(c(F)c1)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2cccnc12
Cc1cccc(Cl)c1C(=O)c1cn(-c2ccc(cc2F)C(O)=O)c2ccccc12
Cc1cccc(Cl)c1C(=O)c1cn(-c2ccc(cc2)C(O)=O)c2cccc(F)c12
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2c(Cl)cccc2C(F)(F)F)c2c(F)cccc12
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccnc12
OC(=O)c1ccc(cc1C(F)(F)F)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2ccccc12
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2c(F)cc(F)cc2Cl)c2ccccc12
OC(=O)c1ccc(c(F)c1)-n1cc(C(=O)c2c(Cl)cccc2C(F)(F)F)c2c(F)cccc12
Cc1c(C(=O)c2c(Cl)cccc2Cl)c2ccccc2n1-c1ccc(cc1)C(O)=O
Cc1cc(ccc1-n1cc(C(=O)c2c(Cl)cccc2Cl)c2ccccc12)C(O)=O
Cc1cc(ccc1C(O)=O)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2ccccc12
Cc1cccc(Cl)c1C(=O)c1cn(-c2ccc(cc2)C(O)=O)c2ccccc12
Cc1cccc(Cl)c1C(=O)c1cn(-c2ccc(cc2F)C(O)=O)c2cccc(F)c12
OC(=O)c1ccc(c(F)c1)-n1cc(C(=O)c2c(Cl)cccc2C(F)(F)F)c2cccnc12
OC(=O)c1ccc(cc1O)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2ccccc12
OC(=O)c1ccc(cc1)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2cc(F)ccc12
OC(=O)c1ccc(c(F)c1)-n1cc(C(=O)c2c(Cl)cccc2Cl)c2c(F)cccc12
CCOc1cc(F)cc(c1)-c1ccc2CC(CC(O)=O)N(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
OC(=O)CCCC1Cc2ccc(cc2N1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1cc(F)cc(OC(F)F)c1
OC1CCN(CC1)C(=O)CC1Cc2ccc(cc2N1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1cc(F)cc(OC(F)F)c1
OC(=O)c1cc2ccc(cc2n1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1cc(F)cc(OC(F)F)c1
CC(C)(C[C@H]1CN(c2cc(ccc2O1)-c1cc(F)cc(OC(F)F)c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(O)=O |r|
OC(=O)CC1Cc2ccc(cc2N1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1cc(F)cc(OC(F)F)c1
OC(=O)C[C@@H]1Cc2ccc(cc2N1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1cc(F)cc(OC(F)F)c1 |r|
OC(=O)CCC1Cc2ccc(cc2N1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1cc(F)cc(OC(F)F)c1
OC(=O)C1CN(C1)C(=O)CC1Cc2ccc(cc2N1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1cc(F)cc(OC(F)F)c1
FC(F)Oc1cc(F)cc(c1)-c1ccc2CC(CC(=O)N3CCS(=O)(=O)CC3)N(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
Fc1cccc(Cl)c1COc1ccc2CCN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
FC(F)Oc1cc(F)cc(c1)-c1ccc2CCN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
FC(F)Oc1cc(F)cc(c1)-c1ccc2cnn(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
FC(F)Oc1cc(F)cc(c1)-c1ccc2ncn(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
OC(=O)Cc1cc2ccc(cc2n1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1cc(F)cc(OC(F)F)c1
OC(=O)Cc1cn(c2cc(ccc12)-c1cc(F)cc(OC(F)F)c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
OC(=O)CCc1cn(c2cc(ccc12)-c1cc(F)cc(OC(F)F)c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
OC(=O)CC1CN(c2cc(ccc12)-c1cc(F)cc(OC(F)F)c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
OC(=O)CCCC1CN(c2cc(ccc12)-c1cc(F)cc(OC(F)F)c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
FC(F)Oc1cc(F)cc(c1)-c1ccc2CC(CC(=O)N3CC(=O)C3)N(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
FC(F)Oc1cc(F)cc(c1)-c1ccc2CC(CC(=O)N3CCC(=O)C3)N(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
FC(F)Oc1cc(F)cc(c1)-c1ccc2CC(CC(=O)N3CCOCC3)N(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
OC(=O)CC1Cc2ccc(cc2N1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1ccc2OC(F)(F)Oc2c1
OC(=O)CC1Cc2ccc(cc2N1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1ccc2OCOc2c1
OC(=O)CC1Cc2ccc(cc2N1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1ccc2OCCc2c1
OC(=O)CC1Cc2ccc(cc2N1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1cc(F)cc(Cl)c1
OC(=O)CC1Cc2ccc(cc2N1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1cc(F)cc(c1)C(F)(F)F
CC(C)Oc1cc(F)cc(c1)-c1ccc2CC(CC(O)=O)N(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
OC1CN(C1)C(=O)CC1Cc2ccc(cc2N1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1cc(F)cc(OC(F)F)c1
COc1cc(F)cc(c1)-c1ccc2CC(CC(O)=O)N(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
OC(=O)CCc1cc2ccc(cc2n1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1cc(F)cc(OC(F)F)c1
FC(F)Oc1cc(F)cc(c1)-c1ccc2CC(CC(=O)N3CC4(COC4)C3)N(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
OC(=O)CCCc1cn(c2cc(ccc12)-c1cc(F)cc(OC(F)F)c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
FC(F)Oc1cc(F)cc(c1)-c1ccc2CC(CC(=O)N3CCC(=O)CC3)N(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
OC(=O)CC1Cc2ccc(cc2N1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1cccc(OC(F)(F)F)c1
FC(F)Oc1cc(F)cc(c1)-c1ccc2ccn(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
OC(=O)C1CCN(CC1)C(=O)CC1Cc2ccc(cc2N1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1cc(F)cc(OC(F)F)c1
OC(=O)CCCc1cc2ccc(cc2n1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1cc(F)cc(OC(F)F)c1
OC(=O)CCC1CN(c2cc(ccc12)-c1cc(F)cc(OC(F)F)c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
OC(=O)CC1Cc2ccc(cc2N1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1cc(F)cc(F)c1
OC(=O)C[C@H]1Cc2ccc(cc2N1S(=O)(=O)c1cccc(c1)C(F)(F)F)-c1cc(F)cc(OC(F)F)c1 |r|
CC(=O)N1CCc2c(ccc(n2)OC)[C@@H]1C(=O)Nc3ccc(cc3)OCc4ccccc4OC
COc1ccc2C(N(CCc2n1)C(C)=O)C(=O)Nc1ccc(OCc2ccccc2)cc1
CCOc1ccccc1CN1CCc2cc(NC(=O)[C@@H]3N(CCc4nc(OC)ccc34)C(=O)CCCC(O)=O)ccc12 |r|
CC1(CCc2c1c(cc(c2)NC(=O)[C@H]3c4ccc(nc4CCN3C(=O)CCCC(=O)O)OC)F)C
COc1ccc2C(N(CCc2n1)C(C)=O)C(=O)Nc1ccc(OCc2ccccc2Cl)cc1
CCOc1ccccc1CN1CCc2cc(NC(=O)[C@@H]3N(CCc4nc(OC)ccc34)C(C)=O)ccc12 |r|
COc1ccc2C(N(CCc2n1)C(C)=O)C(=O)Nc1ccc2N(Cc3ccccc3OC(F)(F)F)CCc2c1
COc1ccccc1COc1ccc(cc1)C(=O)NCc1ccc(cc1)S(N)(=O)=O
COc1ccc2C(N(CCc2n1)C(C)=O)C(=O)Nc1ccc2N(Cc3ccccc3OC)CCc2c1
COc1ccc2[C@H](N(CCc2n1)C(C)=O)C(=O)Nc1ccc(OCc2ccccc2OC)cc1 |r|
OC(=O)c1ccc(NCc2c(noc2-c2ccccc2)-c2c(Cl)cccc2C(F)(F)F)cc1 |(17.9,-10.08,;17.57,-8.58,;18.7,-7.54,;16.1,-8.11,;14.96,-9.15,;13.5,-8.68,;13.17,-7.18,;11.71,-6.71,;10.57,-7.75,;9.11,-7.28,;7.86,-8.2,;6.61,-7.29,;7.07,-5.82,;8.62,-5.81,;9.51,-4.57,;11.05,-4.73,;11.94,-3.48,;11.31,-2.07,;9.77,-1.93,;8.88,-3.17,;7.88,-9.78,;9.25,-10.55,;10.61,-9.73,;9.28,-12.12,;7.92,-12.93,;6.54,-12.16,;6.52,-10.58,;5.15,-9.81,;5.13,-8.27,;3.83,-10.59,;3.81,-9.03,;14.3,-6.14,;15.77,-6.6,)|
OC(=O)Cc1ccc(NC(=O)c2c(noc2-c2ccccc2)-c2c(Cl)cccc2C(F)(F)F)cc1 |(69.68,-30.44,;70.44,-29.1,;71.98,-29.09,;69.67,-27.77,;68.13,-27.78,;67.37,-29.1,;65.84,-29.11,;65.08,-27.79,;63.56,-27.79,;62.8,-29.12,;63.57,-30.43,;61.28,-29.12,;60,-30,;58.78,-29.05,;59.29,-27.59,;60.84,-27.64,;61.79,-26.41,;63.32,-26.61,;64.26,-25.39,;63.68,-23.95,;62.13,-23.75,;61.19,-24.97,;60.02,-31.54,;61.37,-32.29,;62.69,-31.5,;61.39,-33.83,;60.05,-34.62,;58.72,-33.86,;58.7,-32.32,;57.36,-31.57,;57.34,-30.05,;56.04,-32.34,;56.03,-30.8,;65.83,-26.47,;67.35,-26.45,)|
Cc1cc2n(nc(-c3ccc(cc3)C(O)=O)c2s1)C(=O)c1c(Cl)cccc1Cl
OC(=O)c1ccc(NCc2c(noc2-c2cccc(O)c2)-c2c(Cl)cccc2C(F)(F)F)cc1 |(68.2,-47.19,;67.04,-48.22,;67.34,-49.73,;65.57,-47.72,;64.41,-48.75,;62.95,-48.26,;62.65,-46.74,;61.18,-46.24,;60.02,-47.27,;58.56,-46.78,;57.3,-47.67,;56.06,-46.75,;56.54,-45.28,;58.1,-45.3,;59.01,-44.06,;60.54,-44.24,;61.46,-43.01,;60.85,-41.6,;59.32,-41.43,;58.7,-40.02,;58.41,-42.66,;57.28,-49.21,;58.61,-49.99,;59.94,-49.23,;58.59,-51.52,;57.25,-52.28,;55.92,-51.5,;55.94,-49.96,;54.62,-49.18,;54.64,-47.64,;53.28,-49.93,;53.28,-48.4,;63.8,-45.72,;65.26,-46.2,)|
OC(=O)c1ccc(NCc2c(noc2-c2cc[nH]c2)-c2c(Cl)cccc2C(F)(F)F)cc1 |(18.26,-45.22,;17.1,-46.24,;17.4,-47.75,;15.63,-45.74,;14.47,-46.77,;13.01,-46.28,;12.71,-44.76,;11.24,-44.26,;10.08,-45.29,;8.62,-44.8,;7.36,-45.69,;6.12,-44.77,;6.6,-43.3,;8.16,-43.32,;9.08,-42.08,;10.62,-42.1,;11.11,-40.65,;9.88,-39.73,;8.62,-40.62,;7.34,-47.23,;8.67,-48.01,;10,-47.25,;8.65,-49.54,;7.31,-50.3,;5.98,-49.52,;6,-47.98,;4.68,-47.2,;4.7,-45.66,;3.34,-47.95,;3.34,-46.42,;13.86,-43.74,;15.32,-44.22,)|
OC(=O)c1ccc(NCc2c(noc2-c2cccs2)-c2c(Cl)cccc2C(F)(F)F)cc1 |(66.05,-26.26,;64.89,-27.29,;65.19,-28.8,;63.42,-26.79,;62.26,-27.81,;60.8,-27.32,;60.5,-25.81,;59.03,-25.31,;57.87,-26.33,;56.41,-25.84,;55.15,-26.74,;53.91,-25.81,;54.39,-24.34,;55.95,-24.36,;56.86,-23.13,;58.4,-23.14,;58.89,-21.69,;57.66,-20.77,;56.4,-21.66,;55.13,-28.28,;56.46,-29.05,;57.79,-28.29,;56.44,-30.59,;55.1,-31.34,;53.77,-30.56,;53.79,-29.03,;52.47,-28.24,;52.49,-26.7,;51.13,-28.99,;51.13,-27.46,;61.65,-24.78,;63.11,-25.27,)|
OC(=O)c1ccc(NCc2c(noc2-c2ccco2)-c2c(Cl)cccc2C(F)(F)F)cc1 |(42.15,-26.31,;40.99,-27.34,;41.3,-28.85,;39.53,-26.84,;38.36,-27.87,;36.9,-27.38,;36.6,-25.86,;35.14,-25.36,;33.98,-26.39,;32.51,-25.9,;31.26,-26.79,;30.01,-25.87,;30.49,-24.4,;32.05,-24.41,;32.97,-23.18,;34.5,-23.2,;34.99,-21.74,;33.76,-20.82,;32.51,-21.71,;31.24,-28.33,;32.56,-29.1,;33.9,-28.35,;32.55,-30.64,;31.2,-31.4,;29.88,-30.62,;29.89,-29.08,;28.57,-28.29,;28.59,-26.76,;27.23,-29.04,;27.24,-27.52,;37.75,-24.84,;39.22,-25.32,)|
OC(=O)c1ccc(CNc2c(noc2-c2ccccc2)-c2c(Cl)cccc2C(F)(F)F)cc1 |(66.19,-9.77,;65.87,-8.26,;67.02,-7.23,;64.41,-7.78,;63.26,-8.81,;61.8,-8.33,;61.49,-6.82,;60.03,-6.34,;58.88,-7.37,;57.42,-6.89,;56.17,-7.79,;54.93,-6.88,;55.39,-5.41,;56.95,-5.42,;57.85,-4.18,;59.39,-4.35,;60.29,-3.11,;59.67,-1.7,;58.14,-1.54,;57.23,-2.78,;56.19,-9.38,;57.56,-10.14,;58.92,-9.33,;57.58,-11.72,;56.22,-12.53,;54.84,-11.75,;54.83,-10.18,;53.49,-9.42,;53.47,-7.88,;52.16,-10.2,;52.15,-8.65,;62.63,-5.8,;64.09,-6.27,)|
OC(=O)c1ccc(cc1)C(=O)Nc1c(noc1-c1ccccc1)-c1c(Cl)cccc1C(F)(F)F |(41.67,-9.99,;41.39,-8.48,;42.56,-7.48,;39.94,-7.97,;38.77,-8.97,;37.32,-8.46,;37.04,-6.95,;38.2,-5.95,;39.65,-6.45,;35.59,-6.44,;35.31,-4.92,;34.42,-7.44,;32.97,-6.93,;31.7,-7.81,;30.47,-6.86,;30.97,-5.41,;32.53,-5.45,;33.46,-4.23,;34.99,-4.43,;35.92,-3.21,;35.33,-1.79,;33.8,-1.59,;32.87,-2.81,;31.72,-9.39,;33.09,-10.15,;34.45,-9.34,;33.11,-11.73,;31.75,-12.54,;30.37,-11.76,;30.35,-10.19,;29.02,-9.43,;29,-7.89,;27.69,-10.21,;27.67,-8.66,)|
Cc1onc(c1C(=O)Nc1ccc(cc1)C(O)=O)-c1c(Cl)cccc1C(F)(F)F |(46.52,-5.01,;45.65,-6.29,;44.1,-6.33,;43.68,-7.8,;44.95,-8.67,;46.17,-7.74,;47.7,-7.74,;48.47,-9.07,;48.47,-6.4,;50.01,-6.4,;50.78,-7.74,;52.32,-7.74,;53.09,-6.4,;52.31,-5.06,;50.77,-5.07,;54.63,-6.39,;55.4,-7.73,;55.39,-5.06,;44.97,-10.22,;46.32,-10.94,;47.63,-10.13,;46.37,-12.48,;45.04,-13.29,;43.69,-12.55,;43.65,-11.01,;42.31,-10.27,;42.28,-8.73,;40.99,-11.07,;40.96,-9.5,)|
OC(=O)c1ccc(NC(=O)c2c(noc2-c2ccccc2)-c2c(Cl)cccc2C(F)(F)F)cc1 |(74.24,-7.9,;73.47,-6.57,;74.24,-5.23,;71.93,-6.57,;71.16,-7.9,;69.62,-7.9,;68.85,-6.57,;67.31,-6.57,;66.54,-7.9,;67.31,-9.24,;65.01,-7.9,;63.79,-8.85,;62.52,-7.98,;62.94,-6.49,;64.49,-6.45,;65.35,-5.17,;66.88,-5.29,;67.75,-4.02,;67.08,-2.63,;65.53,-2.52,;64.67,-3.79,;63.83,-10.38,;65.18,-11.1,;66.48,-10.28,;65.23,-12.63,;63.91,-13.45,;62.56,-12.72,;62.51,-11.18,;61.16,-10.45,;61.12,-8.91,;59.84,-11.25,;59.82,-9.68,;69.61,-5.24,;71.15,-5.23,)|
CC(C)(C)OC(=O)c1ccc(NC(=O)c2c(noc2-c2ccccc2)-c2c(Cl)cccc2C(F)(F)F)cc1 |(42.68,-30.58,;41.91,-29.25,;42.68,-27.91,;43.44,-29.24,;40.37,-29.25,;39.6,-27.92,;40.36,-26.58,;38.06,-27.92,;37.29,-29.26,;35.75,-29.26,;34.98,-27.92,;33.44,-27.92,;32.67,-29.26,;33.44,-30.59,;31.14,-29.26,;29.9,-30.19,;28.64,-29.29,;29.09,-27.81,;30.64,-27.79,;31.53,-26.53,;33.07,-26.67,;33.96,-25.4,;33.31,-24,;31.76,-23.86,;30.88,-25.13,;29.92,-31.72,;31.26,-32.47,;32.58,-31.68,;31.28,-34.01,;29.95,-34.8,;28.61,-34.05,;28.59,-32.51,;27.25,-31.75,;27.23,-30.21,;25.92,-32.53,;25.91,-30.98,;35.74,-26.59,;37.28,-26.58,)|
OC(=O)c1cccc(NC(=O)c2c(noc2-c2ccccc2)-c2c(Cl)cccc2C(F)(F)F)c1 |(17.09,-50.46,;17.85,-49.12,;19.39,-49.12,;17.08,-47.8,;17.84,-46.47,;17.07,-45.15,;15.55,-45.15,;14.8,-46.48,;13.27,-46.48,;12.52,-47.8,;13.28,-49.12,;10.99,-47.81,;9.73,-48.7,;8.49,-47.78,;8.96,-46.31,;10.52,-46.33,;11.46,-45.08,;12.99,-45.26,;13.91,-44.02,;13.29,-42.58,;11.74,-42.42,;10.82,-43.66,;9.75,-50.24,;11.09,-51,;12.42,-50.21,;11.11,-52.54,;9.78,-53.33,;8.44,-52.58,;8.42,-51.03,;7.09,-50.28,;7.07,-48.75,;5.77,-51.06,;5.75,-49.52,;15.56,-47.8,)|
OC(=O)c1ccc(NCc2c(noc2-c2cccc3ccccc23)-c2c(Cl)cccc2C(F)(F)F)cc1 |(43.87,-46.35,;42.71,-47.38,;43.02,-48.89,;41.25,-46.88,;40.08,-47.91,;38.62,-47.41,;38.32,-45.9,;36.85,-45.4,;35.69,-46.42,;34.23,-45.93,;32.97,-46.83,;31.72,-45.9,;32.2,-44.43,;33.77,-44.45,;34.68,-43.22,;36.21,-43.4,;37.13,-42.17,;36.52,-40.75,;34.98,-40.58,;34.37,-39.19,;32.86,-39.02,;31.95,-40.25,;32.57,-41.65,;34.07,-41.81,;32.95,-48.37,;34.27,-49.15,;35.61,-48.39,;34.26,-50.68,;32.91,-51.44,;31.59,-50.66,;31.61,-49.12,;30.28,-48.33,;30.3,-46.8,;28.94,-49.08,;28.95,-47.56,;39.47,-44.87,;40.94,-45.36,)|
OC(=O)c1ccc(cc1)S(=O)(=O)Nc1c(noc1-c1ccccc1)-c1c(Cl)cccc1C(F)(F)F |(19.75,-25.52,;18.61,-26.56,;18.95,-28.06,;17.15,-26.1,;16.01,-27.14,;14.54,-26.67,;14.22,-25.17,;15.35,-24.13,;16.81,-24.59,;12.75,-24.69,;11.73,-23.52,;13.26,-23.23,;11.62,-25.74,;10.15,-25.27,;8.91,-26.18,;7.65,-25.29,;8.11,-23.81,;9.66,-23.8,;10.56,-22.56,;12.09,-22.71,;12.98,-21.47,;12.35,-20.06,;10.81,-19.91,;9.92,-21.16,;8.93,-27.77,;10.3,-28.53,;11.66,-27.72,;10.33,-30.1,;8.97,-30.92,;7.59,-30.14,;7.57,-28.57,;6.23,-27.81,;6.22,-26.27,;4.91,-28.59,;4.89,-27.04,)|
OC(=O)c1ccc(NC(=O)c2c(noc2-c2ccccc2)-c2c(Cl)cccc2C(F)(F)F)cc1F |(43.04,-48.33,;42.27,-47,;43.03,-45.67,;40.73,-47.01,;39.96,-45.68,;38.43,-45.69,;37.68,-47.01,;36.15,-47.01,;35.39,-48.34,;36.15,-49.66,;33.87,-48.34,;32.63,-49.27,;31.37,-48.37,;31.8,-46.89,;33.36,-46.87,;34.26,-45.6,;35.8,-45.74,;36.69,-44.48,;36.04,-43.06,;34.48,-42.93,;33.6,-44.2,;32.65,-50.81,;34,-51.57,;35.32,-50.77,;34.02,-53.1,;32.69,-53.9,;31.35,-53.14,;31.33,-51.6,;29.99,-50.85,;29.97,-49.32,;28.68,-51.63,;28.66,-50.08,;38.44,-48.34,;39.97,-48.33,;40.74,-49.66,)|
OC(=O)c1c(noc1-c1ccccc1)-c1c(Cl)cccc1C(F)(F)F |(11.48,-32.82,;10.15,-32.04,;8.82,-32.8,;10.16,-30.51,;9.15,-29.34,;9.95,-28.03,;11.45,-28.37,;11.58,-29.91,;12.91,-30.71,;12.87,-32.25,;14.2,-33.04,;15.55,-32.3,;15.57,-30.74,;14.25,-29.95,;7.61,-29.33,;6.84,-30.65,;7.6,-31.98,;5.31,-30.64,;4.55,-29.29,;5.33,-27.97,;6.86,-27.99,;7.65,-26.67,;9.18,-26.68,;6.89,-25.33,;8.41,-25.33,)|
OC(=O)c1ccc(CNC(=O)c2c(noc2-c2ccccc2)-c2c(Cl)cccc2C(F)(F)F)cc1 |(66.78,-52.93,;67.54,-51.6,;69.08,-51.59,;66.77,-50.26,;65.23,-50.27,;64.45,-48.94,;65.22,-47.61,;64.45,-46.28,;62.92,-46.28,;62.17,-47.6,;62.93,-48.92,;60.65,-47.6,;59.37,-48.52,;58.15,-47.59,;58.62,-46.13,;60.18,-46.14,;61.09,-44.89,;62.63,-45.05,;63.55,-43.8,;62.92,-42.4,;61.37,-42.22,;60.46,-43.47,;59.41,-50.06,;60.74,-50.81,;62.07,-50.02,;60.77,-52.34,;59.44,-53.14,;58.09,-52.38,;58.08,-50.84,;56.73,-50.09,;56.72,-48.56,;55.43,-50.86,;55.41,-49.32,;66.76,-47.59,;67.53,-48.92,)|
OC(=O)[C@]1(F)CC[C@@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:15.18,3.3,wD:7.10,3.2,(2.91,-8.62,;1.52,-7.95,;.25,-8.81,;1.42,-6.41,;.2,-7.36,;.51,-5.16,;1.14,-3.76,;2.67,-3.6,;3.57,-4.84,;2.95,-6.25,;3.3,-2.19,;4.83,-2.03,;2.39,-.94,;.85,-.94,;.37,.52,;1.62,1.43,;2.87,.52,;.09,1.27,;-.54,-.14,;-2.07,-.3,;-2.97,.94,;-2.35,2.35,;-.82,2.51,;-4.51,.78,;-4.34,-.75,;-4.67,2.31,;-4.83,3.85,;-3.14,2.48,;-6.2,2.15,;-6.04,.62,;-7.57,.46,;-7.07,1.77,;-5.88,-.91,;2.65,2.57,;3.8,1.54,;3.68,3.72,;1.51,3.6,;.04,3.13,;-1.1,4.16,;-.78,5.66,;-1.93,6.69,;.68,6.14,;1.83,5.11,)|
Fc1ccc(cc1)S(=O)(=O)[C@]1(CCN(C1)C(=O)[C@H]1CC[C@@H](CC1)c1nnn[nH]1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:17.18,wD:10.31,20.25,(5.4,-2.16,;3.86,-2.16,;3.09,-3.5,;1.55,-3.5,;.78,-2.16,;1.55,-.83,;3.09,-.83,;-.76,-2.16,;-.76,-3.7,;-2.1,-2.93,;-1.53,-.83,;-2.44,.42,;-1.53,1.66,;-.07,1.19,;-.07,-.35,;.7,2.52,;-.07,3.86,;2.24,2.52,;3.01,3.86,;4.55,3.86,;5.32,2.52,;4.55,1.19,;3.01,1.19,;6.86,2.52,;7.77,3.77,;9.23,3.29,;9.23,1.75,;7.77,1.28,;-3.07,-.83,;-3.84,.51,;-5.38,.51,;-6.15,-.83,;-5.38,-2.16,;-3.84,-2.16,;-7.69,-.83,;-9.23,-.83,;-7.69,.71,;-9.03,1.48,;-6.36,1.48,;-8.09,2.2,;-7.69,-2.37,;-6.36,-3.14,;-9.03,-3.14,;-7.29,-3.86,)|
C[C@@]1(CC[C@@H](CC1)C(O)=O)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:1.10,wD:15.18,4.7,(17.83,-28.31,;16.5,-27.54,;15.16,-26.78,;15.15,-25.23,;16.49,-24.46,;17.83,-25.23,;17.83,-26.76,;16.48,-22.92,;15.15,-22.15,;17.82,-22.14,;16.51,-29.09,;17.88,-29.78,;15.22,-29.93,;13.78,-29.38,;12.82,-30.58,;13.66,-31.87,;15.14,-31.47,;12.11,-31.87,;11.34,-33.2,;9.81,-33.2,;9.04,-31.88,;9.8,-30.55,;11.34,-30.54,;7.5,-31.88,;5.96,-31.87,;6.73,-30.55,;5.19,-30.56,;7.49,-29.21,;5.94,-29.21,;6.74,-33.22,;5.2,-33.22,;7.51,-34.55,;5.95,-34.54,;14.42,-33.2,;14.41,-34.74,;13.08,-33.97,;15.96,-33.21,;16.72,-34.54,;18.26,-34.55,;19.04,-33.21,;20.58,-33.21,;18.26,-31.87,;16.72,-31.88,)|
Fc1ccc(cc1)S(=O)(=O)[C@]1(CCN(C1)C(=O)C1CCS(=O)(=O)CC1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
C[C@@]1(CC[C@@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(O)=O |r,wU:12.15,1.43,wD:4.7,1.0,(.2,-7.36,;1.42,-6.41,;.51,-5.16,;1.14,-3.76,;2.67,-3.6,;3.57,-4.84,;2.95,-6.25,;3.3,-2.19,;4.83,-2.03,;2.39,-.94,;.85,-.94,;.37,.52,;1.62,1.43,;2.87,.52,;.09,1.27,;-.54,-.14,;-2.07,-.3,;-2.97,.94,;-2.35,2.35,;-.82,2.51,;-4.51,.78,;-4.34,-.75,;-4.67,2.31,;-4.83,3.85,;-3.14,2.48,;-6.2,2.15,;-6.04,.62,;-7.57,.46,;-7.07,1.77,;-5.88,-.91,;2.65,2.57,;3.8,1.54,;3.68,3.72,;1.51,3.6,;.04,3.13,;-1.1,4.16,;-.78,5.66,;-1.93,6.69,;.68,6.14,;1.83,5.11,;1.52,-7.95,;2.91,-8.62,;.25,-8.81,)|
OC(=O)[C@@]1(F)CC[C@@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:15.18,3.2,wD:7.10,3.3,(2.91,-8.62,;1.52,-7.95,;.25,-8.81,;1.42,-6.41,;.2,-7.36,;.51,-5.16,;1.14,-3.76,;2.67,-3.6,;3.57,-4.84,;2.95,-6.25,;3.3,-2.19,;4.83,-2.03,;2.39,-.94,;.85,-.94,;.37,.52,;1.62,1.43,;2.87,.52,;.09,1.27,;-.54,-.14,;-2.07,-.3,;-2.97,.94,;-2.35,2.35,;-.82,2.51,;-4.51,.78,;-4.34,-.75,;-4.67,2.31,;-4.83,3.85,;-3.14,2.48,;-6.2,2.15,;-6.04,.62,;-7.57,.46,;-7.07,1.77,;-5.88,-.91,;2.65,2.57,;3.8,1.54,;3.68,3.72,;1.51,3.6,;.04,3.13,;-1.1,4.16,;-.78,5.66,;-1.93,6.69,;.68,6.14,;1.83,5.11,)|
CC[C@@]1(CC[C@@H](CC1)C(O)=O)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:2.1,5.8,wD:16.19,2.11,(-.36,-3.62,;-1.75,-2.95,;-3.02,-3.81,;-4.52,-4.18,;-4.94,-5.66,;-3.87,-6.77,;-2.38,-6.4,;-1.95,-4.92,;-4.3,-8.25,;-3.23,-9.36,;-5.79,-8.62,;-3.65,-2.4,;-5.18,-2.24,;-2.75,-1.16,;-1.21,-1.16,;-.73,.31,;-1.98,1.21,;-3.22,.31,;-.44,1.05,;.46,2.3,;1.99,2.14,;2.62,.73,;1.71,-.51,;.18,-.35,;4.15,.57,;4.31,2.1,;3.99,-.96,;3.83,-2.49,;2.46,-.8,;5.52,-1.12,;5.68,.41,;7.21,.25,;6.45,-.92,;5.84,1.94,;-3.01,2.36,;-4.15,1.33,;-4.04,3.5,;-1.86,3.39,;-2.18,4.9,;-1.04,5.93,;.43,5.45,;1.57,6.48,;.75,3.94,;-.4,2.91,)|
COC[C@@]1(CC[C@@H](CC1)C(O)=O)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:3.12,wD:17.20,6.9,(19.14,-49.19,;17.81,-48.42,;16.47,-49.19,;15.14,-48.42,;13.8,-47.66,;13.8,-46.11,;15.14,-45.33,;16.47,-46.1,;16.48,-47.64,;15.13,-43.79,;13.8,-43.03,;16.46,-43.02,;15.15,-49.96,;16.53,-50.66,;13.87,-50.81,;12.43,-50.26,;11.46,-51.46,;12.31,-52.75,;13.79,-52.35,;10.76,-52.75,;9.99,-54.08,;8.45,-54.08,;7.69,-52.76,;8.45,-51.43,;9.99,-51.42,;6.15,-52.76,;4.6,-52.75,;5.37,-51.43,;3.83,-51.43,;6.14,-50.09,;4.59,-50.08,;5.38,-54.1,;3.84,-54.1,;6.16,-55.43,;4.6,-55.42,;13.07,-54.08,;13.06,-55.62,;11.73,-54.85,;14.61,-54.09,;15.37,-55.42,;16.91,-55.42,;17.68,-54.09,;19.22,-54.09,;16.9,-52.75,;15.37,-52.76,)|
OC(=O)[C@H]1CC[C@@](F)(CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:3.2,6.6,wD:15.18,6.10,(-3.31,-8.88,;-4.38,-7.77,;-5.87,-8.15,;-3.95,-6.29,;-5.02,-5.18,;-4.6,-3.7,;-3.1,-3.33,;-1.83,-2.47,;-2.03,-4.44,;-2.46,-5.92,;-3.73,-1.92,;-5.26,-1.76,;-2.82,-.68,;-1.28,-.68,;-.81,.79,;-2.05,1.69,;-3.3,.79,;-.52,1.53,;.38,2.78,;1.91,2.61,;2.54,1.21,;1.63,-.04,;.1,.12,;4.07,1.05,;4.23,2.58,;3.91,-.48,;3.75,-2.02,;2.38,-.32,;5.44,-.65,;5.6,.89,;7.13,.73,;6.37,-.45,;5.76,2.42,;-3.09,2.84,;-4.23,1.8,;-4.12,3.98,;-1.94,3.87,;-2.26,5.37,;-1.12,6.4,;.35,5.93,;1.49,6.96,;.67,4.42,;-.48,3.39,)|
OC(=O)C1CCC(O)(CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@]1(CC[C@@H](CC1)C(O)=O)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:1.10,4.7,wD:15.18,(41.31,-8.68,;39.98,-7.91,;41.31,-7.13,;41.31,-5.59,;39.97,-4.82,;38.63,-5.6,;38.64,-7.15,;39.97,-3.28,;38.63,-2.52,;41.3,-2.51,;39.99,-9.45,;41.36,-10.15,;38.7,-10.3,;37.26,-9.75,;36.3,-10.95,;37.14,-12.24,;38.63,-11.84,;35.59,-12.24,;34.83,-13.57,;33.29,-13.57,;32.52,-12.25,;33.28,-10.92,;34.83,-10.91,;30.98,-12.25,;29.44,-12.23,;30.21,-10.92,;28.67,-10.92,;30.97,-9.58,;29.42,-9.57,;30.22,-13.59,;28.68,-13.59,;30.99,-14.92,;29.43,-14.91,;37.9,-13.57,;37.89,-15.11,;36.56,-14.34,;39.44,-13.58,;40.21,-14.91,;41.74,-14.91,;42.52,-13.58,;44.06,-13.58,;41.74,-12.24,;40.2,-12.25,)|
OC(=O)[C@H]1[C@H]2C[C@@H](C[C@@H]12)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C12CCC(CC1)(CC2)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C12CCC(CC1)(OC2)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:16.20,(-1.15,.45,;-2.05,2.08,;-3.48,1.02,;-1.75,4.01,;-.35,3.37,;-.63,4.79,;-2.01,5.41,;-3.51,4.75,;-3.31,3.34,;-1.94,7.08,;-1.49,5.95,;-2.48,3.55,;-3.94,2.45,;-.85,2.94,;.54,3.61,;1.61,2.5,;.88,1.14,;-.64,1.41,;.45,-.34,;1.52,-1.45,;1.09,-2.93,;-.41,-3.29,;-1.47,-2.18,;-1.04,-.7,;-.84,-4.77,;-1.27,-6.25,;.64,-5.2,;2.12,-5.63,;.21,-6.68,;1.07,-3.72,;-2.32,-4.34,;-3.79,-3.92,;-1.89,-2.87,;-2.74,-5.82,;2.61,1.03,;4.04,1.93,;2,-.46,;3.73,-.02,;5.21,.43,;6.33,-.63,;5.98,-2.13,;7.1,-3.18,;4.5,-2.57,;3.38,-1.52,)|
Fc1ccc(cc1)S(=O)(=O)[C@]1(CCN(C1)C(=O)C1CCC2(CC1)NC(=O)NC2=O)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wD:10.32,(5.5,-2.78,;3.96,-2.78,;3.19,-4.12,;1.65,-4.12,;.88,-2.78,;1.65,-1.45,;3.19,-1.45,;-.66,-2.78,;-.66,-4.32,;-1.99,-3.55,;-1.43,-1.45,;-2.33,-.2,;-1.43,1.04,;.04,.57,;.04,-.97,;.81,1.9,;.04,3.23,;2.35,1.9,;3.12,.57,;4.66,.57,;5.43,1.9,;4.66,3.23,;3.12,3.23,;6.33,.65,;7.8,1.13,;9.13,.36,;7.8,2.67,;6.33,3.14,;5.56,4.48,;-2.97,-1.45,;-3.74,-.12,;-5.28,-.12,;-6.05,-1.45,;-5.28,-2.78,;-3.74,-2.78,;-7.59,-1.45,;-9.13,-1.45,;-7.59,.09,;-8.92,.86,;-6.26,.86,;-7.99,1.58,;-7.59,-2.99,;-6.26,-3.76,;-8.92,-3.76,;-7.19,-4.48,)|
COC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:4.3,wD:15.18,7.10,(-10.36,-5.17,;-8.82,-5.33,;-7.92,-4.08,;-8.54,-2.67,;-6.39,-4.24,;-5.48,-3,;-3.95,-3.16,;-3.32,-4.56,;-4.23,-5.81,;-5.76,-5.65,;-1.79,-4.72,;-1.17,-6.13,;-.89,-3.48,;.65,-3.48,;1.13,-2.01,;-.12,-1.11,;-1.36,-2.01,;.91,.04,;.44,1.5,;1.47,2.64,;2.97,2.32,;3.45,.86,;2.42,-.28,;4,3.47,;5.04,4.61,;2.86,4.5,;1.72,5.53,;3.89,5.64,;1.83,3.36,;5.15,2.44,;6.29,1.41,;4.12,1.29,;6.18,3.58,;-1.15,.04,;-0,1.07,;-2.29,-.99,;-2.18,1.18,;-3.68,.86,;-4.71,2,;-4.24,3.47,;-5.27,4.61,;-2.73,3.79,;-1.7,2.64,)|
CS(=O)(=O)C1CCC(CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wD:15.18,(8.43,1.01,;7.66,2.34,;8.43,3.68,;7.66,3.88,;6.12,2.34,;5.35,1.01,;3.81,1.01,;3.04,2.34,;3.81,3.68,;5.35,3.68,;1.5,2.34,;.73,3.68,;.73,1.01,;-.73,1.48,;-1.64,.24,;-.73,-1.01,;.73,-.53,;-2.27,-1.01,;-3.04,.33,;-4.58,.33,;-5.35,-1.01,;-4.58,-2.34,;-3.04,-2.34,;-6.89,-1.01,;-8.43,-1.01,;-6.89,.53,;-8.23,1.3,;-5.56,1.3,;-7.66,1.87,;-6.89,-2.55,;-8.23,-3.32,;-5.56,-3.32,;-6.12,-3.88,;.04,-2.34,;.04,-3.88,;-.73,-3.68,;1.58,-2.34,;2.35,-3.68,;3.89,-3.68,;4.66,-2.34,;6.2,-2.34,;3.89,-1.01,;2.35,-1.01,)|
OC[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:13.16,2.1,wD:5.8,(-.06,-11.15,;-.96,-9.91,;-.33,-8.5,;-1.24,-7.26,;-.61,-5.85,;.92,-5.69,;1.82,-6.93,;1.2,-8.34,;1.54,-4.28,;3.08,-4.12,;.64,-3.03,;-.9,-3.03,;-1.38,-1.57,;-.13,-.67,;1.12,-1.57,;-1.16,.48,;-.69,1.94,;-1.72,3.09,;-3.22,2.77,;-3.7,1.3,;-2.67,.16,;-4.25,3.91,;-5.28,5.06,;-5.4,2.88,;-6.54,1.85,;-6.43,4.03,;-4.37,1.74,;-3.11,4.94,;-1.96,5.97,;-2.08,3.8,;-4.14,6.09,;.9,.48,;2.04,-.55,;-.24,1.51,;1.93,1.62,;1.45,3.09,;2.48,4.23,;3.99,3.91,;5.02,5.06,;4.47,2.45,;3.44,1.3,)|
CC1(CCS(=O)(=O)CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CCC1(CCS(=O)(=O)CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@]1(CCN(C1)C(=O)C1(F)CCS(=O)(=O)CC1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
OCC1(CCS(=O)(=O)CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
COC1(CCS(=O)(=O)CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CCC[C@@]1(CC[C@@H](CC1)C(O)=O)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:17.20,3.2,6.9,wD:3.12,(6.16,-6.82,;4.67,-6.45,;4.24,-4.97,;2.75,-4.6,;1.47,-3.74,;.09,-4.41,;-.02,-5.95,;1.26,-6.81,;2.64,-6.14,;-1.4,-6.62,;-1.51,-8.16,;-2.68,-5.76,;3.37,-3.19,;4.91,-3.03,;2.47,-1.95,;.93,-1.95,;.45,-.48,;1.7,.42,;2.95,-.48,;.17,.26,;-.46,-1.14,;-1.99,-1.31,;-2.9,-.06,;-2.27,1.35,;-.74,1.51,;-4.43,-.22,;-5.96,-.38,;-4.27,-1.75,;-4.1,-3.28,;-5.8,-1.91,;-2.73,-1.59,;-4.59,1.31,;-4.75,2.84,;-3.06,1.47,;-6.12,1.15,;2.73,1.57,;3.87,.54,;3.76,2.71,;1.59,2.6,;.12,2.12,;-1.02,3.15,;-.7,4.66,;-1.85,5.69,;.76,5.14,;1.91,4.1,)|
Fc1ccc(cc1)S(=O)(=O)[C@]1(CCN(C1)C(=O)C1CCS(=O)(=O)C1)c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
OC(=O)[C@H]1C[C@H]2[C@@H](C1)[C@@H]2C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C12CCC(CC1)(C2)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
NC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:14.17,3.2,wD:6.9,(.2,-10.82,;-.7,-9.58,;-2.23,-9.74,;-.07,-8.17,;-.98,-6.92,;-.35,-5.52,;1.18,-5.36,;2.08,-6.6,;1.46,-8.01,;1.8,-3.95,;3.34,-3.79,;.9,-2.7,;-.64,-2.7,;-1.12,-1.24,;.13,-.33,;1.38,-1.24,;-.9,.81,;-.43,2.28,;-1.46,3.42,;-2.96,3.1,;-3.44,1.64,;-2.41,.49,;-3.99,4.24,;-5.02,5.39,;-5.14,3.21,;-6.28,2.18,;-6.17,4.36,;-4.11,2.07,;-2.85,5.28,;-1.7,6.31,;-1.82,4.13,;-3.88,6.42,;1.16,.81,;2.3,-.22,;.02,1.84,;2.19,1.96,;1.71,3.42,;2.74,4.56,;4.25,4.24,;5.28,5.39,;4.73,2.78,;3.7,1.64,)|
CC[C@@]1(CC[C@@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1)C(O)=O |r,wU:13.16,2.44,wD:5.8,2.1,(3.05,-8.77,;1.67,-8.09,;1.56,-6.56,;.66,-5.31,;1.28,-3.9,;2.82,-3.74,;3.72,-4.99,;3.09,-6.4,;3.44,-2.34,;4.97,-2.17,;2.54,-1.09,;1,-1.09,;.52,.37,;1.77,1.28,;3.01,.37,;.24,1.12,;-.39,-.29,;-1.92,-.45,;-2.83,.8,;-2.2,2.2,;-.67,2.36,;-4.36,.64,;-5.89,.48,;-4.2,-.9,;-4.04,-2.43,;-5.73,-1.06,;-2.67,-.73,;-4.52,2.17,;-4.68,3.7,;-2.99,2.33,;-6.05,2.01,;2.8,2.42,;3.94,1.39,;3.83,3.57,;1.65,3.45,;.19,2.98,;-.96,4.01,;-.64,5.52,;-1.78,6.55,;.83,5.99,;1.97,4.96,;.35,-7.5,;.56,-9.03,;-1.08,-6.93,)|
CO[C@@]1(CC[C@@H](CC1)C(O)=O)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:2.11,wD:16.19,5.8,(85.51,-27.18,;84.17,-27.95,;82.84,-27.18,;81.5,-26.42,;81.5,-24.88,;82.83,-24.1,;84.17,-24.87,;84.18,-26.41,;82.83,-22.56,;81.49,-21.79,;84.16,-21.78,;82.85,-28.73,;84.23,-29.42,;81.56,-29.57,;80.12,-29.03,;79.16,-30.23,;80,-31.51,;81.49,-31.11,;78.46,-31.52,;77.69,-32.84,;76.15,-32.84,;75.39,-31.52,;76.15,-30.19,;77.69,-30.18,;73.85,-31.52,;72.3,-31.51,;73.07,-30.19,;71.53,-30.2,;73.84,-28.86,;72.29,-28.85,;73.08,-32.86,;71.54,-32.86,;73.85,-34.19,;72.29,-34.18,;80.76,-32.85,;80.76,-34.39,;79.43,-33.61,;82.31,-32.85,;83.07,-34.18,;84.61,-34.19,;85.38,-32.85,;86.92,-32.85,;84.6,-31.51,;83.07,-31.52,)|
OC(=O)[C@@H]1[C@H]2C[C@@H](C[C@@H]12)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)C12CCC(CC1)(CO2)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:16.20,(-1.15,.45,;-2.05,2.08,;-3.48,1.02,;-1.75,4.01,;-1.49,5.95,;-1.94,7.08,;-2.01,5.41,;-.63,4.79,;-.35,3.37,;-3.51,4.75,;-3.31,3.34,;-2.48,3.55,;-3.94,2.45,;-.85,2.94,;.54,3.61,;1.61,2.5,;.88,1.14,;-.64,1.41,;.45,-.34,;1.52,-1.45,;1.09,-2.93,;-.41,-3.29,;-1.47,-2.18,;-1.04,-.7,;-.84,-4.77,;-1.27,-6.25,;.64,-5.2,;2.12,-5.63,;.21,-6.68,;1.07,-3.72,;-2.32,-4.34,;-3.79,-3.92,;-1.89,-2.87,;-2.74,-5.82,;2.61,1.03,;4.04,1.93,;2,-.46,;3.73,-.02,;5.21,.43,;6.33,-.63,;5.98,-2.13,;7.1,-3.18,;4.5,-2.57,;3.38,-1.52,)|
O[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:12.15,1.0,wD:4.7,(-1.21,-4.9,;-.58,-3.49,;-1.49,-2.25,;-.86,-.84,;.67,-.68,;1.58,-1.92,;.95,-3.33,;1.3,.73,;2.83,.89,;.39,1.97,;-1.15,1.97,;-1.62,3.44,;-.38,4.34,;.87,3.44,;-1.13,5.69,;-2.67,5.7,;-3.43,7.04,;-2.65,8.37,;-1.11,8.35,;-.35,7.01,;-3.4,9.71,;-4.16,11.05,;-4.74,8.96,;-6.09,8.2,;-5.5,10.3,;-3.99,7.61,;-2.06,10.47,;-.72,11.22,;-1.3,9.13,;-2.82,11.81,;.38,5.69,;.2,7.22,;1.13,7.03,;1.72,4.93,;3.05,5.71,;4.39,4.96,;4.4,3.42,;5.74,2.66,;3.08,2.63,;1.74,3.39,)|
OC1(CCS(=O)(=O)CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
COC(=O)c1ccc(CS(=O)(=O)Nc2ccc(cc2)-c2ccc(cc2F)C(O)(C(F)(F)F)C(F)(F)F)cc1
OC(c1ccc(c(F)c1)-c1ccc(NC(=O)CCCC2CCCCC2)cc1)(C(F)(F)F)C(F)(F)F
CCCCCCC(=O)Nc1ccc(cc1)-c1ccc(cc1F)C(O)(C(F)(F)F)C(F)(F)F
CS(=O)(=O)c1ccc(CS(=O)(=O)Nc2ccc(cc2)-c2ccc(cc2F)C(O)(C(F)(F)F)C(F)(F)F)cc1
OC(c1ccc(c(F)c1)-c1ccc(NS(=O)(=O)Cc2ccc(cc2)C#N)cc1)(C(F)(F)F)C(F)(F)F
NC(=O)c1ccc(CS(=O)(=O)Nc2ccc(cc2)-c2ccc(cc2F)C(O)(C(F)(F)F)C(F)(F)F)cc1
OC(c1ccc(c(F)c1)-c1ccc(NS(=O)(=O)Cc2ccccc2[N+]([O-])=O)cc1)(C(F)(F)F)C(F)(F)F
COC(=O)c1cccc(CS(=O)(=O)Nc2ccc(cc2)-c2ccc(cc2F)C(O)(C(F)(F)F)C(F)(F)F)c1
Nc1ccccc1CC(=O)Nc1ccc(cc1)-c1ccc(cc1F)C(O)(C(F)(F)F)C(F)(F)F
CCCCCC(=O)Nc1ccc(cc1)-c1ccc(cc1F)C(O)(C(F)(F)F)C(F)(F)F
OC(c1ccc(c(F)c1)-c1ccc(NC(=O)CCC(F)(F)F)cc1)(C(F)(F)F)C(F)(F)F
CC(=O)CCCC(=O)Nc1ccc(cc1)-c1ccc(cc1F)C(O)(C(F)(F)F)C(F)(F)F
OC(c1ccc(c(F)c1)-c1ccc(NC(=O)CCc2ccccc2)cc1)(C(F)(F)F)C(F)(F)F
OC(c1ccc(c(F)c1)-c1ccc(NS(=O)(=O)Cc2cccc(c2)[N+]([O-])=O)cc1)(C(F)(F)F)C(F)(F)F
COC(=O)CCC(=O)Nc1ccc(cc1)-c1ccc(cc1F)C(O)(C(F)(F)F)C(F)(F)F
CNC(=O)c1ccc(CS(=O)(=O)Nc2ccc(cc2)-c2ccc(cc2F)C(O)(C(F)(F)F)C(F)(F)F)cc1
COC(=O)c1ccccc1CS(=O)(=O)Nc1ccc(cc1)-c1ccc(cc1F)C(O)(C(F)(F)F)C(F)(F)F
COC(=O)CCCC(=O)Nc1ccc(cc1)-c1ccc(cc1F)C(O)(C(F)(F)F)C(F)(F)F
OC(c1ccc(c(F)c1)-c1ccc(NS(=O)(=O)Cc2ccc(cc2)[N+]([O-])=O)cc1)(C(F)(F)F)C(F)(F)F
c1ccc(c(c1)Nc2cccc3c2CN(CCO3)S(=O)(=O)c4ccc(cc4)F)F
C[C@H]1CC[C@H](c2cccc(c2)C#N)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)C(C)=O |r|
C[C@H]1CC[C@H](c2ccccn2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)C(C)=O |r|
C[C@H]1CC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)C(C)=O |r|
C[C@H]1COC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)C(C)=O |r|
C[C@H]1CN(Cc2ccc(cc2F)N2CCN(CC2)C(C)=O)S(=O)(=O)[C@H](CO1)c1ccccc1 |r|
C[C@@H]1COC[C@H](c2ccccc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)C(C)=O |r|
CC(=O)N1CCN(CC1)c1ccc(CN2CCCC[C@H](c3ccccc3)S2(=O)=O)c(F)c1 |r|
C[C@H]1CC[C@H](c2cccs2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)C(C)=O |r|
C[C@H]1CC[C@H](c2ccsc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)C(C)=O |r|
C[C@H]1CC[C@H](c2ccncc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)C(C)=O |r|
C[C@H]1CC[C@H](c2cccc(Cl)c2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)C(C)=O |r|
COc1ccc(cc1)[C@H]1CC[C@H](C)N(Cc2ccc(cc2F)N2CCN(CC2)C(C)=O)S1(=O)=O |r|
COc1ccccc1[C@H]1CC[C@H](C)N(Cc2ccc(cc2F)N2CCN(CC2)C(C)=O)S1(=O)=O |r|
C[C@H]1CC[C@H](c2ccc(cc2)C#N)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)C(C)=O |r|
C[C@@H]1CN(Cc2ccc(cc2F)N2CCN(CC2)C(C)=O)S(=O)(=O)[C@H](CO1)c1ccccc1 |r|
C[C@H]1CC[C@H](c2ncccn2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)C(C)=O |r|
C[C@H]1CC[C@H](c2ccc(Cl)cc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)C(C)=O |r|
CC(=O)N1CCN(CC1)c1ccc(CN2CCOC[C@H](c3ccccc3)S2(=O)=O)c(F)c1 |r|
C[C@H]1CC[C@H](c2cccnc2)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)C(C)=O |r|
C[C@H]1CC[C@H](c2ccccc2Cl)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)C(C)=O |r|
C[C@H]1CC[C@H](c2ccccc2C#N)S(=O)(=O)N1Cc1ccc(cc1F)N1CCN(CC1)C(C)=O |r|
COc1cccc(c1)[C@H]1CC[C@H](C)N(Cc2ccc(cc2F)N2CCN(CC2)C(C)=O)S1(=O)=O |r|
CC(C)CCCc1nnc(C(CCO)CC(=O)Nc2ccc(C)cc2C)n1C1CC1
CC(C)Cc1cc(on1)-c1onc([C@@H](CCC([O-])=O)CC(=O)Nc2ccc(C)cc2Cl)c1C1CC1 |r|
Cc1ccc(NC(=O)C[C@H](CCC([O-])=O)c2noc(-c3cc(CC(C)(C)C)on3)c2C2CC2)c(Cl)c1 |r|
CC(C)CCCc1nnc(C(CCC(O)=O)CC(=O)Nc2ccc(C)cc2C)n1C1CC1
CNC(=O)CCC(CC(=O)Nc1ccc(C)cc1C)c1nnc(CCCC(C)C)n1C1CC1
CC(C)Cc1ccc(cc1)-c1onc([C@@H](CCC(O)=O)CC(=O)Nc2ccc(C)cc2Cl)c1C1CC1 |r|
CC(C)Cc1cnc(o1)-c1onc([C@@H](CCC([O-])=O)CC(=O)Nc2ccc(C)cc2Cl)c1C1CC1 |r|
CC(C)Cc1nc(cs1)-c1onc([C@@H](CCC([O-])=O)CC(=O)Nc2ccc(C)cc2Cl)c1C1CC1 |r|
CC(C)Cc1ncc(s1)-c1onc([C@@H](CCC([O-])=O)CC(=O)Nc2ccc(C)cc2Cl)c1C1CC1 |r|
CC(C)Cc1nnc(s1)-c1onc([C@@H](CCC([O-])=O)CC(=O)Nc2ccc(C)cc2Cl)c1C1CC1 |r|
CC(C)CC(F)(F)c1cc(no1)-c1onc([C@@H](CCC([O-])=O)CC(=O)Nc2ccc(C)cc2Cl)c1C1CC1 |r|
CC(C)(C)Cc1cc(no1)-c1onc([C@@H](CCC([O-])=O)CC(=O)Nc2ccc(Cl)cc2Cl)c1C1CC1 |r|
Cc1ccc(NC(=O)C[C@H](CCC([O-])=O)c2noc(-c3cc(on3)C(F)(F)C(C)(C)C)c2C2CC2)c(Cl)c1 |r|
CC(C)(C)C(F)(F)c1cc(no1)-c1onc([C@@H](CCC([O-])=O)CC(=O)Nc2ccc(Cl)cc2F)c1C1CC1 |r|
CC(C)CCCc1nnc(C(CCN)CC(=O)Nc2ccc(C)cc2C)n1C1CC1
CC(C)Cc1nc(no1)-c1onc([C@@H](CCC([O-])=O)CC(=O)Nc2ccc(C)cc2Cl)c1C1CC1 |r|
CC(C)CCCc1nnc(C(CCC(N)=O)CC(=O)Nc2ccc(C)cc2C)n1C1CC1
Cc4ccc(NC(=O)C[C@H](CCC(=O)[O-])c2noc(c1cc(CC(C)C)on1)c2C3CC3)c(Cl)c4
CC(C)C(F)(F)c1cc(no1)-c1onc([C@@H](CCC([O-])=O)CC(=O)Nc2ccc(C)cc2Cl)c1C1CC1 |r|
CCN(c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(cc1)[N+]([O-])=O
CC(C)CCCc1nnc(C(CCNC(C)=O)CC(=O)Nc2ccc(C)cc2C)n1C1CC1
CC(C)CCCc1nnc(C(CCC(=O)N(C)C)CC(=O)Nc2ccc(C)cc2C)n1C1CC1
CC(C)Cc1cnc(s1)-c1onc([C@@H](CCC([O-])=O)CC(=O)Nc2ccc(C)cc2Cl)c1C1CC1 |r|
CC(C)CCc1cc(no1)-c1onc([C@@H](CCC([O-])=O)CC(=O)Nc2ccc(C)cc2Cl)c1C1CC1 |r|
CC(C)(C)C(F)(F)c1cc(no1)-c1onc([C@@H](CCC([O-])=O)CC(=O)Nc2ccc(F)cc2Cl)c1C1CC1 |r|
CC(C)CCCc1nnc(C(CCN(C)C)CC(=O)Nc2ccc(C)cc2C)n1C1CC1
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@H]1CCS(=O)(=O)[C@@H](C)C1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
C[C@H]1C[C@@H](CC[C@H]1C(=O)N2CC[C@@]3([C@H]2CCc4c3ccc(c4)C(C(F)(F)F)(C(F)(F)F)F)S(=O)(=O)c5ccc(cc5)F)C(=O)O
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@@H]1CC[C@H](C[C@@H]1C)C(O)=O)S(=O)(=O)c1cccc(F)c1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@@H]1CC[C@H](C[C@H]1C)C(O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@@H]1CC[C@H]([C@@H](C)C1)C(O)=O)S(=O)(=O)c1cccc(F)c1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@H]1CC[C@H]([C@@H](C)C1)C(O)=O)S(=O)(=O)c1cccc(F)c1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@@H]1CC[C@H]([C@H](C)C1)C(O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@H]1CC[C@H]([C@H](C)C1)C(O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCCC[C@@H]2C)C(=O)NCC(C)(C)O)c(C(F)F)c1F)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCCC[C@@H]2C)C(=O)NCC(C)(C)O)c(C(F)F)c1F)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CC(F)(F)C[C@@H]2C)C(=O)NCC(C)(C)O)c(C(F)F)c1F)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CC(F)(F)C[C@@H]2C)C(=O)NCC(C)(C)O)c(C(F)F)c1F)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)(F)CC2)C(=O)NCC(C)(C)O)c(c1F)C(F)(F)F)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(=O)NCC(C)(C)O)c(Cl)c1C)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N(CC)CC)C(=O)NCC(C)(C)O)c(C(F)F)c1F)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N(CC)CC)C(=O)NCC(C)(C)O)c(C(F)F)c1Cl)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N(CC)CC)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(NCCC(C)(C)O)nc2C(=O)N2CCC(F)CC2)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(NC(=O)CC(C)(C)O)nc2C(=O)N2CCC(F)CC2)c(Cl)c1Cl)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(=O)NCCN2CCOCC2)c(Cl)c1Cl)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(=O)N2CC3(C2)CS(=O)(=O)C3)c(Cl)c1Cl)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(=O)NC2CC22CCOCC2)c(Cl)c1Cl)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(=O)NC2CCS(=O)(=O)CC2)c(Cl)c1Cl)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(=O)NCCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(=O)NCCC(C)(C)C(N)=O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(=O)NCC(C)(C)C#N)c(Cl)c1Cl)C(F)(F)F |r|
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)(F)CC2)c(s1)-c1ccc(c(Cl)c1Cl)S(=O)(=O)NC(C)(C)CF
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)(F)CC2)c(s1)-c1ccc(c(Cl)c1Cl)S(=O)(=O)NC1(CC1)C(F)(F)F
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
CCN(C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)N[C@@H](C)C(F)(F)F)C(=O)NCC(C)(C)O)C12CC(C1)C2 |r|
CCN(C1CC1)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)N[C@@H](C)C(F)(F)F)C(=O)NCC(C)(C)O |r|
CCN(CCC(F)(F)F)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)N[C@@H](C)C(F)(F)F)C(=O)NCC(C)(C)O |r|
CCN(CC(F)F)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)N[C@@H](C)C(F)(F)F)C(=O)NCC(C)(C)O |r|
CCN(CCCF)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)N[C@@H](C)C(F)(F)F)C(=O)NCC(C)(C)O |r|
CCN(CC(F)(F)F)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)N[C@@H](C)C(F)(F)F)C(=O)NCC(C)(C)O |r|
CCN(C(C)C)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)N[C@@H](C)C(F)(F)F)C(=O)NCC(C)(C)O |r|
CCCN(CC)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)N[C@@H](C)C(F)(F)F)C(=O)NCC(C)(C)O |r|
CCN(CC)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)N[C@@H](C)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CC(F)(F)C[C@@H]2C)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)(F)C2)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CC3CC3C2)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2C3CCC2CC3)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)(C)C2)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
CC[C@H]1CCCN1C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)N[C@@H](C)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC[C@@H]2CF)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC[C@@H]2C)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CC[C@@H](F)C[C@@H]2C)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CC[C@H](F)C[C@@H]2C)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)(F)CC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)(F)CC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCCC[C@@H]2C)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC3(CC3)CC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCCCC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCCCC2)C(=O)NCC(C)(C)O)c2ccccc12
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)(F)CC2)C(=O)NCC(C)(C)O)c(Cl)c1F)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(=O)NCC(C)(C)c2nn[nH]n2)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(=O)NCC(C)(C)c2noc(=O)[nH]2)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(=O)NCCC(C)(C)C#N)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(=O)N2CC(C)(C2)C#N)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(=O)N2CC3(C2)CC(O)(C3)C(F)(F)F)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(N)=O)c(Cl)c1Cl)C(F)(F)F |r|
COCC(C)(C)NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)(F)CC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)(F)CC2)c(s1)-c1ccc(c(Cl)c1Cl)S(=O)(=O)NC1(C)CC1
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)(F)CC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)CC2)c(s1)-c1ccc(c(Cl)c1Cl)S(=O)(=O)NC1(C)CC1
CC(C)(O)CNC(=O)c1nc(C(=O)N2CCC(F)CC2)c(s1)-c1ccc(c(Cl)c1Cl)S(=O)(=O)N[C@@H](C(C)(C)C)C(F)(F)F |r|
CC(C)[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
CCN(C1CCC1)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)N[C@@H](C)C(F)(F)F)C(=O)NCC(C)(C)O |r|
CC(C)CNC(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)N[C@@H](C)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(C)CC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCCC[C@H]2C)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCCC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
CCN(CC(C)C)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)N[C@@H](C)C(F)(F)F)C(=O)NCC(C)(C)O |r|
CC(C)N(C(C)C)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)N[C@@H](C)C(F)(F)F)C(=O)NCC(C)(C)O |r|
CCCN(C)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)N[C@@H](C)C(F)(F)F)C(=O)NCC(C)(C)O |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(CC(C)(C)C(O)=O)nc2CC2CCC2)c(Cl)c1Cl)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(CC(C)(C)C(O)=O)nc2CC2CCC2)c(Cl)c1Cl)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(CC(C)(C)C(O)=O)nc2CC2CCC2)c(Cl)c1)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(CC(C)(C)C(O)=O)nc2CC2CCC2)c(c1)C(F)(F)F)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(CC(C)(C)C(O)=O)nc2CC2CCC2)c(C(F)F)c1F)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2noc(CC(C)(C)C(O)=O)n2)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2nnc(CC(C)(C)C(O)=O)s2)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2cc(CC(C)(C)C(O)=O)on2)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2cc(CC(C)(C)C(O)=O)ncn2)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)-c2nnc(o2)[C@H]2C[C@@H](C2)C(O)=O)c(Cl)c1Cl)C(F)(F)F |r,wU:25.27,wD:27.32,1.0,(60.84,-8,;59.51,-7.23,;58.18,-8,;56.84,-7.23,;57.61,-5.9,;56.07,-5.9,;55.51,-8,;55.51,-9.54,;54.19,-10.31,;52.84,-9.55,;51.51,-10.32,;50.11,-9.69,;49.08,-10.84,;49.84,-12.17,;51.35,-11.85,;52.44,-12.94,;52.04,-14.42,;52.83,-15.78,;51.5,-16.55,;50.71,-15.2,;47.54,-10.84,;46.63,-9.59,;45.17,-10.07,;45.17,-11.61,;46.63,-12.08,;43.84,-12.38,;43.43,-13.89,;41.94,-13.49,;42.35,-11.97,;40.61,-14.26,;40.61,-15.8,;39.28,-13.49,;52.84,-8,;51.51,-7.23,;54.18,-7.24,;54.18,-5.7,;59.51,-5.69,;58.18,-4.93,;60.84,-4.93,;59.51,-4.17,)|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2Cc2ccc(F)cc2)-c2nnc(CC(C)(C)C(O)=O)o2)c(C(F)F)c1F)C(F)(F)F |r|
CC(C)Cc1nc(sc1-c1ccc(c(F)c1C(F)F)S(=O)(=O)N[C@@H](C)C(F)(F)F)-c1nnc(CC(C)(C)C(O)=O)o1 |r|
COC(C)(C)Cc1nc(sc1-c1ccc(c(F)c1C(F)F)S(=O)(=O)N[C@@H](C)C(F)(F)F)-c1nnc(CC(C)(C)C(O)=O)o1 |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CN2CCCC(F)(F)C2)-c2nnc(CC(C)(C)C(O)=O)o2)c(C(F)F)c1F)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCCC[C@@H]2C)-c2nnc(CC(C)(C)C(O)=O)o2)c(C(F)F)c1F)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2CC2CCC2)C(=O)NCC(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
CCN(CC)C(=O)c1nc(sc1-c1ccc(c(Cl)c1Cl)S(=O)(=O)N[C@@H](C)C(F)(F)F)-c1nnc(o1)C(C)(C)O |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)(F)CC2)-c2nnc(o2)C(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)-c2nnc(o2)C(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
CC[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)-c2nnc(CC(C)(C)O)o2)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)CC2)-c2noc(n2)C(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
C[C@H](NS(=O)(=O)c1ccc(-c2sc(nc2C(=O)N2CCC(F)(F)CC2)-c2nnc(n2C)C(C)(C)O)c(Cl)c1Cl)C(F)(F)F |r|
[H][C@]12CCc3c(nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2CCC)-c1ccnc(c1)C(F)(F)F)-c1ccccc1F |r,t:14|
[H][C@]12CCc3c(nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2CCC)-c1ccnc(CF)c1)-c1ccccc1F |r,t:14|
[H][C@]12CCc3c(nc(nc3[C@]1(C)C=C(C(N)=O)C(=O)[C@@H]2CCC)-c1ccnc(c1)C1CC1)-c1ccccc1F |r,t:14|
CC1=C2CCc3c(nc(nc3[C@]2(C)C=C(C#N)C1=O)-c1ccncc1)-c1ccccc1 |r,c:1,t:15|
[H][C@]12CCc3c(nc(nc3[C@]1(C)CC(C#N)C(=O)[C@@H]2C)-c1ccncc1)-c1ccccc1 |r|
[H][C@]12CCc3c(nc(nc3[C@]1(C)CC(C(N)=O)C(=O)[C@@H]2C)-c1ccncc1)-c1ccccc1 |r|
c1ccc(cc1)COc2ccc(cc2)C3(CCCC3)S(=O)(=O)c4ccc(cc4)F
Fc1ccc(cc1)S(=O)(=O)C1(CCN(C1)C(=O)CC1CCOCC1)c1ccc(OCc2ccccc2)cc1
Fc1ccc(cc1)S(=O)(=O)C1(CCN(C1)C(=O)C1CCOCC1)c1ccc(OCc2ccccc2)cc1
Fc1ccc(cc1)S(=O)(=O)C1(CCN(C1)C(=O)Cc1ccncc1)c1ccc(OCc2ccccc2)cc1
Fc1ccc(cc1)S(=O)(=O)C1(CCN(C1)C(=O)C1CCS(=O)(=O)CC1)c1ccc(OCc2ccccc2)cc1
Fc1ccc(cc1)S(=O)(=O)[C@]1(CCN(C1)C(=O)C1CCS(=O)(=O)CC1)c1ccc(OCc2ccccc2C(F)(F)F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@]1(CCN(C1)C(=O)C1CCS(=O)(=O)CC1)c1ccc(OCc2c(Cl)cccc2C(F)(F)F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@]1(CCN(C1)C(=O)C1CCS(=O)(=O)CC1)c1ccc(OCc2c(F)cccc2C(F)(F)F)cc1 |r|
[H][C@@]12CCc3cc(OCc4c(F)cccc4C(F)(F)F)ccc3[C@@]1(CCN2C(=O)C1CCS(=O)(=O)CC1)S(=O)(=O)c1ccc(F)cc1 |r|
[H][C@@]12CCc3cc(OCc4c(F)cccc4C(F)(F)F)ccc3[C@@]1(CCN2C(=O)C1(O)CCS(=O)(=O)CC1)S(=O)(=O)c1ccc(F)cc1 |r|
[H][C@@]12CCc3cc(OCc4c(F)cccc4C(F)(F)F)ccc3[C@@]1(CCN2C(=O)CN1CCS(=O)(=O)CC1)S(=O)(=O)c1ccc(F)cc1 |r|
[H][C@@]12CCc3cc(OCc4c(F)cccc4C(F)(F)F)ccc3[C@@]1(CCN2C(=O)[C@H]1CC[C@@H](CC1)NS(C)(=O)=O)S(=O)(=O)c1ccc(F)cc1 |r,wU:23.44,29.32,1.0,wD:32.39,(34.56,-11.06,;33.23,-10.3,;33.23,-11.85,;31.88,-12.62,;30.54,-11.85,;29.17,-12.77,;27.83,-12,;26.5,-12.77,;25.16,-12,;23.83,-12.76,;23.83,-14.3,;25.17,-15.06,;22.5,-15.07,;21.16,-14.3,;21.16,-12.76,;22.5,-11.99,;22.5,-10.45,;23.84,-9.68,;21.17,-9.68,;22.49,-8.91,;27.83,-10.45,;29.16,-9.68,;30.55,-10.29,;31.89,-9.51,;31.98,-8.14,;33.48,-7.82,;34.26,-9.15,;35.79,-9.3,;36.69,-8.05,;36.42,-10.71,;37.96,-10.85,;38.58,-12.27,;37.68,-13.51,;36.15,-13.35,;35.52,-11.95,;38.3,-14.92,;37.39,-16.16,;38.03,-17.57,;36.06,-16.92,;36.07,-15.38,;30.73,-8.57,;29.39,-9.33,;29.4,-7.79,;31.13,-7.08,;32.61,-6.69,;33.01,-5.21,;31.93,-4.12,;32.32,-2.63,;30.43,-4.52,;30.04,-6.01,)|
[H][C@@]12CCc3cc(OCc4c(F)cccc4C(F)(F)F)ccc3[C@@]1(CCN2C(=O)[C@H]1CC[C@@H](CC1)C(N)=O)S(=O)(=O)c1ccc(F)cc1 |r,wU:23.42,29.32,1.0,wD:32.39,(35.32,-11.24,;34,-10.47,;33.99,-12.03,;32.64,-12.8,;31.31,-12.03,;29.93,-12.95,;28.59,-12.18,;27.26,-12.95,;25.93,-12.17,;24.59,-12.94,;24.6,-14.48,;25.93,-15.24,;23.27,-15.25,;21.92,-14.48,;21.93,-12.94,;23.26,-12.17,;23.26,-10.63,;24.6,-9.86,;21.93,-9.85,;23.25,-9.08,;28.6,-10.63,;29.92,-9.86,;31.31,-10.47,;32.65,-9.69,;32.74,-8.32,;34.25,-8,;35.02,-9.33,;36.55,-9.48,;37.45,-8.23,;37.19,-10.89,;38.72,-11.03,;39.35,-12.44,;38.44,-13.69,;36.91,-13.53,;36.28,-12.13,;39.07,-15.1,;38.16,-16.35,;40.6,-15.26,;31.49,-8.75,;30.15,-9.51,;30.16,-7.97,;31.89,-7.26,;33.38,-6.87,;33.78,-5.39,;32.69,-4.3,;33.09,-2.81,;31.19,-4.7,;30.8,-6.19,)|
[H][C@@]12CCc3cc(OCc4c(F)cccc4C(F)(F)F)ccc3[C@@]1(CCN2C(=O)C1CCN(CC1)C(N)=O)S(=O)(=O)c1ccc(F)cc1 |r|
[H][C@@]12CCc3cc(OCc4c(F)cccc4C(F)(F)F)ccc3[C@@]1(CCN2C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1ccc(F)cc1 |r,wU:23.42,29.32,1.0,wD:32.39,(35.43,-10.87,;34.11,-10.1,;34.11,-11.66,;32.76,-12.43,;31.42,-11.65,;30.04,-12.57,;28.71,-11.8,;27.38,-12.57,;26.04,-11.8,;24.71,-12.57,;24.71,-14.1,;26.05,-14.87,;23.38,-14.87,;22.04,-14.1,;22.04,-12.56,;23.38,-11.79,;23.38,-10.25,;24.72,-9.49,;22.05,-9.48,;23.37,-8.71,;28.71,-10.26,;30.04,-9.49,;31.42,-10.1,;32.77,-9.32,;32.86,-7.95,;34.36,-7.62,;35.14,-8.95,;36.67,-9.11,;37.57,-7.86,;37.3,-10.51,;38.83,-10.66,;39.46,-12.07,;38.56,-13.32,;37.03,-13.16,;36.4,-11.76,;39.18,-14.73,;38.28,-15.97,;40.72,-14.89,;31.61,-8.38,;30.27,-9.14,;30.28,-7.6,;32.01,-6.89,;33.49,-6.5,;33.89,-5.01,;32.8,-3.92,;33.2,-2.44,;31.31,-4.33,;30.92,-5.81,)|
[H][C@@]12CCc3cc(OCc4c(F)cccc4C(F)(F)F)ccc3[C@@]1(CCN2C(=O)[C@H]1CC[C@@H](CC1)c1nn[nH]n1)S(=O)(=O)c1ccc(F)cc1 |r,wU:23.45,29.32,1.0,wD:32.39,(33.51,-12.97,;32.19,-12.21,;32.19,-13.76,;30.84,-14.53,;29.5,-13.76,;28.12,-14.68,;26.79,-13.91,;25.45,-14.68,;24.12,-13.91,;22.79,-14.68,;22.79,-16.21,;24.13,-16.98,;21.46,-16.98,;20.12,-16.21,;20.12,-14.67,;21.46,-13.9,;21.46,-12.36,;22.79,-11.6,;20.13,-11.59,;21.45,-10.82,;26.79,-12.37,;28.12,-11.6,;29.5,-12.2,;30.84,-11.42,;30.94,-10.06,;32.44,-9.73,;33.22,-11.06,;34.75,-11.22,;35.65,-9.97,;35.38,-12.62,;36.91,-12.77,;37.54,-14.18,;36.63,-15.43,;35.1,-15.26,;34.48,-13.86,;37.26,-16.83,;38.77,-17.15,;38.93,-18.69,;37.52,-19.31,;36.49,-18.17,;29.69,-10.48,;28.35,-11.25,;28.36,-9.71,;30.09,-9,;31.57,-8.61,;31.97,-7.12,;30.88,-6.03,;31.28,-4.54,;29.39,-6.44,;29,-7.92,)|
[H][C@@]12CCc3cc(OCc4c(F)cccc4C(F)(F)F)ccc3[C@@]1(CCN2C(=O)[C@@]1(C)CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1ccc(F)cc1 |r,wU:33.40,1.0,23.43,wD:29.32,(25.68,-18.35,;24.36,-17.58,;24.36,-19.14,;23.01,-19.91,;21.68,-19.13,;20.3,-20.06,;18.97,-19.29,;17.63,-20.06,;16.29,-19.28,;14.96,-20.06,;14.96,-21.59,;16.3,-22.35,;13.64,-22.36,;12.3,-21.59,;12.3,-20.05,;13.63,-19.28,;13.64,-17.74,;12.3,-16.97,;14.97,-16.98,;13.63,-16.2,;18.97,-17.74,;20.29,-16.98,;21.68,-17.58,;23.02,-16.8,;23.11,-15.44,;24.61,-15.11,;25.39,-16.44,;26.92,-16.59,;27.82,-15.35,;27.55,-18,;28.3,-16.66,;26.65,-19.24,;27.27,-20.64,;28.8,-20.8,;29.71,-19.56,;29.08,-18.14,;29.43,-22.21,;28.52,-23.46,;30.96,-22.37,;21.86,-15.87,;20.53,-15.09,;20.53,-16.63,;22.26,-14.38,;23.75,-13.99,;24.14,-12.51,;23.06,-11.41,;23.46,-9.92,;21.56,-11.82,;21.17,-13.3,)|
CNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)c(COc2cccc3c(cc(C)nc23)-n2ccnc2)c1Cl |r|
CNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)c(COc2cccc3c(cc(nc23)C(F)(F)F)-n2ccnc2)c1Cl |r|
CNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)c(COc2cccc3c(cc(C)nc23)C(F)(F)F)c1Cl |r|
CCc1cc(c2cccc(OCc3c(Cl)ccc(c3Cl)S(=O)(=O)N3CCC[C@H]3C(=O)NC)c2n1)C(F)(F)F |r|
CNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)c(COc2cccc3c(cc(nc23)C(C)C)C(F)(F)F)c1Cl |r|
Cc1cc(c2cccc(OCc3c(Cl)ccc(c3Cl)S(=O)(=O)N3CCC[C@H]3C(N)=O)c2n1)C(F)(F)F |r|
Cc1cc(c2cccc(OCc3c(Cl)ccc(c3Cl)S(=O)(=O)N3CCC[C@H]3CO)c2n1)C(F)(F)F |r|
COC[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)c(COc2cccc3c(cc(C)nc23)C(F)(F)F)c1Cl |r|
Cc1cc(c2cccc(OCc3c(Cl)ccc(c3Cl)S(=O)(=O)N3CCCC3)c2n1)C(F)(F)F
CNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)c(COc2cccc3c(cc(C)nc23)-c2cncn2C)c1Cl |r|
CNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)c(COc2cccc3c(cc(C)nc23)-c2ccccc2)c1Cl |r|
CNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)c(COc2cccc3c(cc(C)nc23)-c2ccccn2)c1Cl |r|
CNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)c(COc2cccc3c(cc(C)nc23)-c2cccnc2)c1Cl |r|
CNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)c(COc2cccc3c(cc(nc23)C(C)C)-c2ccncc2)c1Cl |r|
CNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)c(COc2cccc3c(OCc4ccccc4)cc(nc23)C(C)C)c1Cl |r|
CNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)c(COc2cccc3c(cc(nc23)C(C)C)-c2cncn2C)c1Cl |r|
CNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)c(COc2cccc3c(cc(nc23)C(C)C)-n2ccnc2)c1Cl |r|
CNC(=O)[C@@H]1CCCN1S(=O)(=O)c1cccc(COc2cccc3c(cc(C)nc23)C(F)(F)F)c1 |r|
Cc1cc(c2cccc(OCc3c(Cl)ccc(c3Cl)S(=O)(=O)N3CCC[C@H]3C(O)=O)c2n1)C(F)(F)F |r|
CN(C)[C@@H]1CCN(C1)S(=O)(=O)c1ccc(Cl)c(COc2cccc3c(cc(C)nc23)C(F)(F)F)c1Cl |r|
Cc1cc(c2cccc(OCc3c(Cl)ccc(c3Cl)S(=O)(=O)N3CCCCC3)c2n1)C(F)(F)F
Cc1cc(c2cccc(OCc3c(Cl)ccc(c3Cl)S(=O)(=O)N3CCC(CCO)CC3)c2n1)C(F)(F)F
C[C@H]1CN(C[C@@H](C)O1)S(=O)(=O)c1ccc(Cl)c(COc2cccc3c(cc(C)nc23)C(F)(F)F)c1Cl |r|
Cc1cc(c2cccc(OCc3c(Cl)ccc(c3Cl)S(=O)(=O)N3CCC(CC3)C#N)c2n1)C(F)(F)F
CNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)c(COc2cccc3c(cc(C)nc23)-c2nccn2C)c1Cl |r|
CNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)c(COc2cccc3c(OCc4ccccc4)cc(C)nc23)c1Cl |r|
CNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)c(COc2cccc3c(cc(C)nc23)-c2ccncc2)c1Cl |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@@H]1C[C@@H](F)C(=O)N1Cc1ccc(F)cc1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@@H]1C[C@@H](F)C(=O)N1Cc1ccc(cc1)C#N)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@@H]1C[C@@H](F)C(=O)N1CCC#N)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@@H]1C[C@@H](F)C(=O)N1CC(O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@@H]1C[C@@H](F)C(=O)N1C(C)C)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@@H]1C[C@@H](F)C(=O)N1CCO)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
CC(C)(CN1[C@@H](C[C@H](C1=O)F)C(=O)N2CC[C@@]3([C@H]2CCc4c3ccc(c4)C(C(F)(F)F)(C(F)(F)F)F)S(=O)(=O)c5ccc(cc5)F)O
[H][C@]12CCc3cc(ccc3[C@]1(CC[C@H]2C(=O)OCC)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@]12CCc3cc(ccc3[C@]1(CC[C@@H]2C(=O)OCC)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CC[C@H]2C(=O)OCC)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CC[C@@H]2C(=O)OCC)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CC[C@H]2C(O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CC[C@H]2C(=O)NC1CC1(F)F)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
CCC(C)n1c2cc(ncc2nc(N2CCN(C)CC2)c1=O)N(C)C1CCCCC1
CNS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)N2CC(C)(C)c3nc(ccc23)-c2c(OC)ncnc2C2CC2)cc1
CNS(=O)(=O)c1ccc(CNC(=O)N2CC3(CCCC3)c3nc(ccc23)-c2ccc(O)cc2C)cc1
CNS(=O)(=O)c1ccc(CNC(=O)c2cnc(OC)c3n(ncc23)-c2ccc(F)cc2)cc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(-c3ccccc3)c2=O)-c2c(OC)ncnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(c2=O)C(C)(C)O)-c2c(OC)ncnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(c2=O)C(C)(C)C)-c2c(OC)ncnc2C2CC2)nc1
CCCn1c2nc(ncc2nc(NCc2ccc(cn2)S(=O)(=O)CC)c1=O)-c1c(OC)ncnc1C1CC1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C(C)C)c2=O)-c2ccc(F)cc2C)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C(C)C)c2=O)-c2nccnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C(C)C)c2=O)-c2c(OC)ccc3ncccc23)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C(C)C)c2=O)-c2c(O)ncnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(nc3n(C(C)C)c2=O)-c2cncnc2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3nnc(cc3n([C@@H](C)C3CC3)c2=O)-c2c(OC)ncnc2C2CC2)nc1 |r|
CCS(=O)(=O)c1ccc(CNc2nc3ncc(nc3n(C(C)C)c2=O)-c2c(OC)ncnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3ncc(cc3n(C(C)C)c2=O)-c2c(OC)ncnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3cnc(cc3n(C(C)C)c2=O)-c2c(OC)ncnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3ccc(nc3n(C(C)C)c2=O)-c2c(OC)ncnc2C2CC2)nc1
CCS(=O)(=O)c1ccc(CNc2nc3ccc(cc3n(C(C)C)c2=O)-c2c(OC)ncnc2C2CC2)nc1
C[C@@H](C1CC1)n1c2nc(ncc2nc(NCc2ccc(cn2)[S@@](C)(=N)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
CCS(=O)(=O)C1CC2(CC(CNc3nc4cnc(nc4n([C@@H](C)C4CC4)c3=O)-c3c(C)ncnc3C3CC3)C2)C1 |r,wU:21.22,(68.95,-37.02,;67.62,-36.25,;66.28,-37.01,;67.37,-38.1,;65.88,-38.5,;64.95,-36.25,;63.47,-36.65,;63.07,-35.16,;61.58,-35.56,;61.18,-34.08,;59.85,-33.31,;58.52,-34.09,;57.18,-33.32,;55.84,-34.1,;54.5,-33.33,;53.16,-34.11,;51.82,-33.34,;51.82,-31.79,;53.16,-31.01,;54.5,-31.78,;55.83,-31,;55.83,-29.46,;54.49,-28.69,;57.16,-28.69,;58.7,-28.68,;57.92,-27.35,;57.17,-31.77,;58.51,-30.98,;50.49,-31.02,;50.49,-29.48,;51.82,-28.71,;49.16,-28.71,;47.82,-29.48,;47.83,-31.03,;49.16,-31.79,;49.17,-33.33,;48.41,-34.66,;49.95,-34.66,;62.66,-33.67,;64.56,-34.76,)|
C[C@@H](C1CC1)n1c2nc(ncc2nc(NCc2cnc(cn2)S(C)(=O)=O)c1=O)-c1c(C)ncnc1C1CC1 |r|
COc1ccc(Oc2c(Cl)cc(NC(=O)CN3CCN(CC3)S(C)(=O)=O)cc2Cl)cc1C(C)C
CC(C)c1cc(cnc1OC)Oc2c(cc(cc2Cl)NC(=O)CC3CCN(CC3)S(=O)(=O)C)Cl
COc1ncc(Oc2c(Cl)cc(NC(=O)Cc3cccnc3)cc2Cl)cc1C(C)C
COc1cc(Oc2c(Cl)cc(NC(=O)Cc3cccnc3)cc2Cl)cc(c1)C(C)C
CC(C)c1cc(Oc2c(Cl)cc(NC(=O)Cc3cccnc3)cc2Cl)cc(c1)C#N
CC(C)c1cc(F)cc(Oc2c(Cl)cc(NC(=O)Cc3cccnc3)cc2Cl)c1
CC(C)c1cc(Oc2c(Cl)cc(NC(=O)Cc3cccnc3)cc2Cl)ccc1F
CC(C)c1ccc(C)c(Oc2ccc(NC(=O)Cc3cccnc3)cc2Cl)c1
CC(C)c1cccc(Oc2c(Cl)cc(NC(=O)Cc3cccnc3)cc2Cl)c1
COc1ccc(Oc2c(Cl)cc(NC(=O)Cc3cccnc3)cc2Cl)cc1C
COc1ccc(Oc2c(Cl)ccc(CNC(=O)C3CN(C3)S(N)(=O)=O)c2Cl)cc1C(C)C
COc1ccc(Oc2c(Cl)ccc(CNC(=O)c3ccc(cc3)S(C)(=O)=O)c2Cl)cc1C(C)C
COc1ccc(Oc2c(Cl)ccc(C(=O)NCCC(N)=O)c2Cl)cc1C(C)C
COc1ccc(Oc2c(Cl)ccc(C(=O)NCc3ccc(cc3)S(N)(=O)=O)c2Cl)cc1C(C)C
COc1ccc(Oc2c(Cl)ccc(NC(=O)CC3CCN(CC3)S(C)(=O)=O)c2Cl)cc1C(C)C
COc1ccc(Oc2c(Cl)ccc(NC(=O)Cc3ccc(cc3)S(C)(=O)=O)c2Cl)cc1C(C)C
COc1ccc(Oc2c(Cl)cc(NC(=O)Cc3cnn(c3)S(C)(=O)=O)cc2Cl)cc1C(C)C
CC(C)c1cc(ccc1OC)Oc2c(cc(cc2Cl)NC(=O)Cc3cccnc3)Cl
COc1ccc(Oc2c(Cl)cc(NC(=O)Cc3ccncc3)cc2Cl)cc1C(C)C
COc1ccc(Oc2c(Cl)cc(NC(=O)Cc3ccccc3)cc2Cl)cc1C(C)C
CC(C)c1cc(ccc1OC)Oc2c(cc(cc2Cl)CO)Cl
Fc1ccc(cc1)S(=O)(=O)C1(CCCC1)c1ccc(cc1)C(OCc1cccc(c1)-c1ccccc1)(C(F)(F)F)C(F)(F)F
CC(=O)N1CCC(CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CC(C1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CC[C@@H](C1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CC[C@H](C1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCC(C)(CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCC(O)(CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
Fc1ccc(cc1)S(=O)(=O)[C@]1(CCN(C1)C(=O)C1CCOCC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r|
Fc1ccc(cc1)S(=O)(=O)[C@]1(CCN(C1)C(=O)N1CCOCC1)c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F |r|
CC(=O)N1CCN(CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CC(=O)N1CCN(CC1)C(=O)N2CC[C@](C2)(c3ccc(cc3)C(C(F)(F)F)(C(F)(F)F)OCc4c(cccc4F)C#N)S(=O)(=O)c5ccc(cc5)F
OC(=O)C1CCN(CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:14.17,3.2,wD:6.9,(2.12,-12.14,;1.22,-10.89,;-.31,-11.05,;1.85,-9.48,;.94,-8.24,;1.57,-6.83,;3.1,-6.67,;4,-7.92,;3.38,-9.32,;3.72,-5.26,;5.26,-5.1,;2.82,-4.02,;1.28,-4.02,;.8,-2.55,;2.05,-1.65,;3.3,-2.55,;1.02,-.5,;1.49,.96,;.46,2.11,;-1.04,1.79,;-1.52,.32,;-.49,-.82,;-2.07,2.93,;-3.1,4.07,;-4.61,3.75,;-5.64,4.9,;-5.16,6.36,;-3.66,6.68,;-6.19,7.51,;-7.7,7.19,;-8.18,5.72,;-7.15,4.58,;-7.62,3.11,;-3.22,1.9,;-4.36,.87,;-2.19,.76,;-4.25,3.04,;-.93,3.96,;.22,4.99,;.1,2.82,;-1.96,5.11,;3.08,-.5,;4.22,-1.53,;1.94,.53,;4.11,.64,;3.63,2.11,;4.66,3.25,;6.17,2.93,;7.2,4.07,;6.65,1.47,;5.62,.32,)|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(OCc1ccccc1OC(F)(F)F)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:14.17,3.2,wD:6.9,(-.76,-11.6,;.77,-11.44,;1.67,-12.68,;1.39,-10.03,;.49,-8.78,;1.11,-7.38,;2.65,-7.21,;3.55,-8.46,;2.92,-9.87,;3.27,-5.81,;4.8,-5.65,;2.37,-4.56,;.83,-4.56,;.35,-3.1,;1.6,-2.19,;2.84,-3.1,;.57,-1.05,;1.04,.42,;.01,1.56,;-1.49,1.24,;-1.97,-.22,;-.94,-1.37,;-2.52,2.39,;-3.56,3.53,;-3.08,4.99,;-4.11,6.14,;-5.62,5.82,;-6.65,6.96,;-6.17,8.43,;-4.66,8.75,;-3.63,7.6,;-2.13,7.92,;-1.65,9.39,;-2.05,10.88,;-.88,10.72,;-.11,9.39,;-1.38,3.42,;-.24,4.45,;-.35,2.27,;-2.41,4.56,;-3.67,1.36,;-4.81,.32,;-2.64,.21,;-4.7,2.5,;2.63,-1.05,;3.77,-2.08,;1.48,-.02,;3.66,.1,;3.18,1.56,;4.21,2.71,;5.72,2.39,;6.75,3.53,;6.19,.92,;5.16,-.22,)|
Cc1cccc(C)c1COC(c1ccc(cc1)[C@@]1(CCN(C1)C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F |r,wU:17.18,27.33,wD:24.26,(-5.99,4.58,;-5.51,6.05,;-6.54,7.19,;-6.07,8.66,;-4.56,8.98,;-3.53,7.83,;-2.03,8.15,;-4.01,6.37,;-2.98,5.22,;-3.45,3.76,;-2.42,2.62,;-1.39,1.47,;.11,1.79,;1.14,.65,;.67,-.82,;-.84,-1.14,;-1.87,.01,;1.7,-1.96,;.45,-2.87,;.93,-4.33,;2.47,-4.33,;2.95,-2.87,;3.37,-5.58,;4.91,-5.42,;2.75,-6.99,;1.22,-7.15,;.59,-8.55,;1.5,-9.8,;3.03,-9.64,;3.65,-8.23,;.87,-11.21,;-.66,-11.37,;1.77,-12.45,;2.73,-.82,;3.87,-1.85,;1.59,.21,;3.76,.33,;3.28,1.79,;4.31,2.94,;5.82,2.62,;6.85,3.76,;6.3,1.15,;5.27,.01,;-1.28,3.65,;-.13,4.68,;-.25,2.5,;-2.31,4.79,;-3.57,1.58,;-4.71,.55,;-2.54,.44,;-4.6,2.73,)|
Cc1cccc(F)c1COC(c1ccc(cc1)[C@@]1(CCN(C1)C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F |r,wU:17.18,27.33,wD:24.26,(-2.03,8.15,;-3.53,7.83,;-4.56,8.98,;-6.07,8.66,;-6.54,7.19,;-5.51,6.05,;-5.99,4.58,;-4.01,6.37,;-2.98,5.22,;-3.45,3.76,;-2.42,2.62,;-1.39,1.47,;.11,1.79,;1.14,.65,;.67,-.82,;-.84,-1.14,;-1.87,.01,;1.7,-1.96,;.45,-2.87,;.93,-4.33,;2.47,-4.33,;2.95,-2.87,;3.37,-5.58,;4.91,-5.42,;2.75,-6.99,;1.22,-7.15,;.59,-8.55,;1.5,-9.8,;3.03,-9.64,;3.65,-8.23,;.87,-11.21,;-.66,-11.37,;1.77,-12.45,;2.73,-.82,;3.87,-1.85,;1.59,.21,;3.76,.33,;3.28,1.79,;4.31,2.94,;5.82,2.62,;6.85,3.76,;6.3,1.15,;5.27,.01,;-1.28,3.65,;-.13,4.68,;-.25,2.5,;-2.31,4.79,;-3.57,1.58,;-4.71,.55,;-2.54,.44,;-4.6,2.73,)|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(OCc1c(F)cccc1Cl)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:14.17,3.2,wD:6.9,(-.66,-11.37,;.87,-11.21,;1.77,-12.45,;1.5,-9.8,;.59,-8.55,;1.22,-7.15,;2.75,-6.99,;3.65,-8.23,;3.03,-9.64,;3.37,-5.58,;4.91,-5.42,;2.47,-4.33,;.93,-4.33,;.45,-2.87,;1.7,-1.96,;2.95,-2.87,;.67,-.82,;1.14,.65,;.11,1.79,;-1.39,1.47,;-1.87,.01,;-.84,-1.14,;-2.42,2.62,;-3.45,3.76,;-2.98,5.22,;-4.01,6.37,;-5.51,6.05,;-5.99,4.58,;-6.54,7.19,;-6.07,8.66,;-4.56,8.98,;-3.53,7.83,;-2.03,8.15,;-1.28,3.65,;-.13,4.68,;-.25,2.5,;-2.31,4.79,;-3.57,1.58,;-4.71,.55,;-2.54,.44,;-4.6,2.73,;2.73,-.82,;3.87,-1.85,;1.59,.21,;3.76,.33,;3.28,1.79,;4.31,2.94,;5.82,2.62,;6.85,3.76,;6.3,1.15,;5.27,.01,)|
COc1cccc(F)c1COC(c1ccc(cc1)[C@@]1(CCN(C1)C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1ccc(F)cc1)(C(F)(F)F)C(F)(F)F |r,wU:18.19,28.34,wD:25.27,(-1.69,9.37,;-2.17,7.9,;-3.68,7.58,;-4.71,8.73,;-6.21,8.41,;-6.69,6.94,;-5.66,5.8,;-6.13,4.33,;-4.15,6.12,;-3.12,4.97,;-3.6,3.51,;-2.57,2.36,;-1.54,1.22,;-.03,1.54,;1,.4,;.52,-1.07,;-.98,-1.39,;-2.01,-.24,;1.56,-2.21,;.31,-3.12,;.79,-4.58,;2.33,-4.58,;2.8,-3.12,;3.23,-5.83,;4.76,-5.67,;2.6,-7.24,;1.07,-7.4,;.45,-8.8,;1.35,-10.05,;2.88,-9.89,;3.51,-8.48,;.73,-11.46,;-.81,-11.62,;1.63,-12.7,;2.59,-1.07,;3.73,-2.1,;1.44,-.04,;3.62,.08,;3.14,1.54,;4.17,2.68,;5.68,2.36,;6.71,3.51,;6.15,.9,;5.12,-.24,;-1.42,3.39,;-.28,4.43,;-.39,2.25,;-2.45,4.54,;-3.71,1.33,;-4.86,.3,;-2.68,.19,;-4.74,2.48,)|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(OCC1CC1)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:14.17,3.2,wD:6.9,(8,6.51,;6.75,7.41,;6.91,8.94,;5.34,6.78,;5.18,5.25,;3.77,4.63,;2.53,5.53,;2.69,7.06,;4.1,7.69,;1.12,4.9,;-.12,5.81,;.96,3.37,;2.11,2.34,;1.48,.94,;-.05,1.1,;-.37,2.6,;-.05,-.44,;-1.39,-1.21,;-1.39,-2.75,;-.05,-3.52,;1.28,-2.75,;1.28,-1.21,;-.05,-5.06,;-.05,-6.6,;1.28,-7.37,;1.28,-8.91,;2.05,-10.25,;.51,-10.25,;-1.59,-5.06,;-3.13,-5.06,;-1.59,-3.52,;-1.59,-6.6,;1.49,-5.06,;3.03,-5.06,;1.49,-3.52,;1.49,-6.6,;-1.58,.94,;-1.74,2.47,;-1.42,-.6,;-3.12,.78,;-3.74,-.63,;-5.27,-.79,;-6.18,.45,;-7.71,.29,;-5.55,1.86,;-4.02,2.02,)|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(OCC1CCC1)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:14.17,3.2,wD:6.9,(8.16,6.74,;6.91,7.65,;7.08,9.18,;5.51,7.02,;5.35,5.49,;3.94,4.86,;2.69,5.77,;2.85,7.3,;4.26,7.93,;1.29,5.14,;.04,6.05,;1.13,3.61,;2.27,2.58,;1.64,1.17,;.11,1.33,;-.21,2.84,;.11,-.21,;-1.22,-.98,;-1.22,-2.52,;.11,-3.29,;1.45,-2.52,;1.45,-.98,;.11,-4.83,;.11,-6.37,;1.45,-7.14,;1.45,-8.68,;2.54,-9.76,;1.45,-10.85,;.36,-9.76,;-1.43,-4.83,;-2.97,-4.83,;-1.43,-3.29,;-1.43,-6.37,;1.65,-4.83,;3.19,-4.83,;1.65,-3.29,;1.65,-6.37,;-1.42,1.17,;-1.58,2.71,;-1.26,-.36,;-2.95,1.01,;-3.58,-.39,;-5.11,-.55,;-6.01,.69,;-7.55,.53,;-5.39,2.1,;-3.86,2.26,)|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(OCC1CCCC1)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:14.17,3.2,wD:6.9,(-.49,-10.74,;1.05,-10.58,;1.95,-11.82,;1.67,-9.17,;.77,-7.93,;1.39,-6.52,;2.93,-6.36,;3.83,-7.6,;3.2,-9.01,;3.55,-4.95,;5.08,-4.79,;2.65,-3.71,;1.11,-3.71,;.63,-2.24,;1.88,-1.34,;3.12,-2.24,;.85,-.19,;1.32,1.27,;.29,2.42,;-1.22,2.1,;-1.69,.63,;-.66,-.51,;-2.25,3.24,;-3.28,4.39,;-4.78,4.07,;-5.81,5.21,;-7.34,5.05,;-7.97,6.46,;-6.83,7.49,;-5.49,6.72,;-1.1,4.27,;.04,5.3,;-.07,3.13,;-2.13,5.42,;-3.39,2.21,;-4.53,1.18,;-2.36,1.07,;-4.42,3.36,;2.91,-.19,;4.05,-1.22,;1.76,.84,;3.94,.95,;3.46,2.42,;4.49,3.56,;6,3.24,;7.03,4.39,;6.47,1.78,;5.44,.63,)|
OC(=O)[C@H]1CC[C@@H](CC1)C(=O)N1CC[C@](C1)(c1ccc(cc1)C(OCC1CCCCC1)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r,wU:3.2,wD:14.17,6.9,(-1,-12.22,;-.1,-10.97,;1.43,-11.13,;-.72,-9.56,;-2.26,-9.4,;-2.88,-7.99,;-1.98,-6.75,;-.45,-6.91,;.18,-8.32,;-2.6,-5.34,;-4.13,-5.18,;-1.7,-4.1,;-.16,-4.1,;.32,-2.63,;-.93,-1.73,;-2.17,-2.63,;.1,-.58,;1.61,-.9,;2.64,.24,;2.16,1.71,;.66,2.03,;-.37,.88,;3.19,2.85,;4.22,4,;3.75,5.46,;4.78,6.61,;4.3,8.07,;5.33,9.21,;6.84,8.89,;7.32,7.43,;6.29,6.29,;4.34,1.82,;5.48,.79,;3.31,.68,;5.37,2.97,;2.05,3.88,;.9,4.91,;1.02,2.74,;3.08,5.03,;-1.96,-.58,;-.81,.45,;-3.1,-1.61,;-2.99,.56,;-4.5,.24,;-5.53,1.39,;-5.05,2.85,;-6.08,4,;-3.54,3.17,;-2.51,2.03,)|
[H][C@@]12CCc3c(Br)c(ccc3[C@@]1(CCN2C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:17.19,wD:20.26,11.29,1.0,(37.63,-6.58,;36.31,-7.36,;36.31,-5.81,;34.96,-5.02,;33.62,-5.8,;32.29,-5.04,;32.28,-3.5,;30.96,-5.81,;30.96,-7.35,;32.29,-8.12,;33.62,-7.36,;34.97,-8.13,;35.29,-9.65,;36.83,-9.81,;37.45,-8.4,;38.96,-8.08,;39.44,-6.61,;39.99,-9.22,;41.49,-8.89,;42.52,-10.05,;42.04,-11.51,;40.53,-11.82,;39.51,-10.68,;43.07,-12.66,;44.58,-12.34,;42.59,-14.12,;33.87,-9.22,;32.77,-10.3,;32.38,-8.81,;34.26,-10.71,;33.16,-11.78,;33.54,-13.27,;35.03,-13.68,;35.42,-15.17,;36.13,-12.59,;35.74,-11.11,;29.62,-5.04,;28.28,-4.27,;29.62,-3.5,;28.29,-2.73,;30.96,-2.73,;29.61,-1.96,;28.29,-5.81,;26.96,-5.04,;28.29,-7.35,;26.95,-6.57,)|
[H][C@@]12CCc3c(C)c(ccc3[C@@]1(CCN2C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:17.19,wD:20.26,11.29,1.0,(59.6,-6.52,;58.27,-7.3,;58.27,-5.74,;56.93,-4.96,;55.59,-5.74,;54.25,-4.98,;54.25,-3.44,;52.92,-5.75,;52.92,-7.29,;54.25,-8.06,;55.58,-7.3,;56.93,-8.07,;57.25,-9.58,;58.79,-9.75,;59.42,-8.33,;60.93,-8.01,;61.4,-6.55,;61.96,-9.16,;63.46,-8.83,;64.49,-9.98,;64.01,-11.45,;62.5,-11.76,;61.48,-10.62,;65.03,-12.6,;66.54,-12.28,;64.55,-14.06,;55.83,-9.15,;54.74,-10.24,;54.34,-8.75,;56.22,-10.64,;55.12,-11.72,;55.51,-13.21,;57,-13.62,;57.38,-15.11,;58.09,-12.53,;57.7,-11.05,;51.59,-4.98,;50.25,-4.21,;51.59,-3.44,;50.25,-2.67,;52.92,-2.67,;51.58,-1.9,;50.26,-5.75,;48.92,-4.98,;50.26,-7.29,;48.91,-6.51,)|
[H][C@@]12CCc3cc(c(Br)cc3[C@@]1(CCN2C(=O)[C@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:17.19,wD:20.26,11.29,1.0,(81.03,-6.64,;79.7,-7.42,;79.71,-5.87,;78.36,-5.09,;77.02,-5.86,;75.68,-5.1,;74.36,-5.87,;74.35,-7.42,;73.02,-8.19,;75.69,-8.19,;77.02,-7.42,;78.37,-8.2,;78.69,-9.71,;80.22,-9.87,;80.85,-8.46,;82.36,-8.14,;82.84,-6.67,;83.39,-9.28,;84.89,-8.95,;85.92,-10.11,;85.44,-11.57,;83.93,-11.88,;82.91,-10.74,;86.47,-12.72,;87.97,-12.41,;85.99,-14.18,;77.27,-9.28,;76.17,-10.37,;75.78,-8.87,;77.65,-10.77,;76.56,-11.84,;76.94,-13.33,;78.43,-13.75,;78.82,-15.24,;79.53,-12.66,;79.14,-11.17,;73.02,-5.1,;71.68,-4.33,;73.02,-3.56,;71.69,-2.79,;74.36,-2.79,;73.01,-2.02,;71.69,-5.87,;70.36,-5.1,;71.69,-7.41,;70.35,-6.63,)|
c1cc(ccc1F)S(=O)(=O)[C@@]23CCN([C@@H]2CCc4c3cc(c(c4)C(C(F)(F)F)(C(F)(F)F)F)C#N)C(=O)C5CCC(CC5)C(=O)O
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2C(=O)[C@@H]1CC[C@H](C[C@@H]1C)C(O)=O)S(=O)(=O)c1ccccc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(c(F)cc3[C@@]1(CCN2C(=O)[C@@H]1CC[C@H](C[C@@H]1C)C(O)=O)S(=O)(=O)c1ccccc1)C(F)(C(F)(F)F)C(F)(F)F |r|
CC(=O)N1CCN(CC1)c1ccc2CN(Cc2c1)S(=O)(=O)Cc1ccccc1
CC(=O)N1CCN(CC1)c1ccc2N(CCc2c1)S(=O)(=O)Cc1ccccc1
CC(=O)N1CCN(CC1)c1ccc2CCCN(c2c1)S(=O)(=O)Cc1ccccc1
CC(=O)N1CCN(CC1)c1ccc2N(CCCc2c1)S(=O)(=O)Cc1ccccc1
CC(=O)N1CCN(CC1)c1ccc2CN(CCCc2c1)S(=O)(=O)Cc1ccccc1
CN(Cc1ccc(cc1)C(C)(C)C)S(=O)(=O)N1CCCc2cc(ccc12)N1CCN(CC1)C(C)=O
CN(Cc1ccc(cc1)-c1ccccc1)S(=O)(=O)N1CCCc2cc(ccc12)N1CCN(CC1)C(C)=O
CN(Cc1ccc(OC(F)(F)F)cc1)S(=O)(=O)N1CCCc2cc(ccc12)N1CCN(CC1)C(C)=O
CN(Cc1ccc(cc1)C#N)S(=O)(=O)N1CCCc2cc(ccc12)N1CCN(CC1)C(C)=O
CN(Cc1ccc(cc1)C(C)(C)C)S(=O)(=O)N1CCCc2cc(ccc12)N1CCN(CC1)S(C)(=O)=O
CCS(=O)(=O)N1CCN(CC1)c1ccc2N(CCCc2c1)S(=O)(=O)N(C)Cc1ccc(cc1)C(C)(C)C
CN(Cc1ccc(cc1)C(C)(C)C)S(=O)(=O)N1CCCc2cc(ccc12)N1CCOCC1
COC(=O)c1ccc(Nc2ccc3N(CCCc3c2)S(=O)(=O)N(C)Cc2ccc(cc2)C(C)(C)C)cc1
CN(Cc1ccc(cc1)C(C)(C)C)S(=O)(=O)N1CCCc2cc(Nc3ccc(cc3)C(O)=O)ccc12
CC(=O)N1CCN(CC1)c1ccc2N(CCCc2c1)S(=O)(=O)c1ccccc1
CN(Cc1ccccc1)S(=O)(=O)N1CCCc2cc(ccc12)N1CCN(CC1)C(C)=O
c1ccc(cc1)NC(=O)c2cc(ccc2Cl)[N+](=O)[O-]
Cc1ccccc1NC(=O)c1cc(ccc1Cl)[N+]([O-])=O
[O-][N+](=O)c1ccc(Cl)c(c1)C(=O)Nc1ccsc1
CCc1ccccc1NC(=O)c1cc(ccc1Cl)[N+]([O-])=O
[O-][N+](=O)c1ccc(Cl)c(c1)C(=O)Nc1ccccc1F
COc1ccccc1NC(=O)c1cc(ccc1Cl)[N+]([O-])=O
Cc1cccc(C)c1NC(=O)c1cc(ccc1Cl)[N+]([O-])=O
[O-][N+](=O)c1ccc(Cl)c(c1)C(=O)Nc1ccccc1C(F)(F)F
[O-][N+](=O)c1ccc(Cl)c(c1)C(=O)Nc1cccc2ccccc12
Nc1ccccc1NC(=O)c1cc(ccc1Cl)[N+]([O-])=O
Oc1ccccc1NC(=O)c1cc(ccc1Cl)[N+]([O-])=O
CC(C)CCC[C@@](C)([C@H]1CC[C@@H]2[C@@]1(CC[C@H]3[C@H]2CC=C4[C@@]3(CC[C@@H](C4)O)C)C)O
[H][C@@]12CCc3nc(ccc3[C@@]1(CCN2C(=O)C1CCS(=O)(=O)CC1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3nc(ccc3[C@@]1(CCN2C(=O)[C@@H]1CCC(=O)N1CCC#N)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ncc3[C@@]1(CCN2C(=O)C1CCS(=O)(=O)CC1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ncc3[C@@]1(CCN2C(=O)[C@@H]1CCC(=O)N1CCC#N)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(cnc3[C@@]1(CCN2C(=O)C1CCS(=O)(=O)CC1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(cnc3[C@@]1(CCN2C(=O)[C@@H]1CCC(=O)N1CCC#N)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3nc(ccc3[C@@]1(CC[C@H]2NC(=O)C(C)(C)O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3nc(ccc3[C@@]1(CC[C@H]2NC(=O)CC(C)(C)O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3nc(ccc3[C@@]1(CC[C@H]2NC(=O)C1CCS(=O)(=O)CC1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3nc(ccc3[C@@]1(CC[C@H]2NC(=O)[C@@](C)(O)CS(C)(=O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
C[C@@](CS(=O)(=O)C)(C(=O)N[C@@H]1CC[C@@]2([C@H]1CCc3c2ccc(n3)C(C(F)(F)F)(C(F)(F)F)F)S(=O)(=O)c4ccc(cc4)F)O
[H][C@@]12CCc3cc(ccc3[C@@]1(CC[C@H]2NC(=O)[C@@](C)(O)CS(C)(=O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CC[C@H]2NC(=O)[C@](C)(O)CS(C)(=O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
CC(=O)N1CCC(CC1)C(=O)N2C[C@H]([C@@](C2)(C)c3ccccc3)c4ccc(cc4)C(C(F)(F)F)(C(F)(F)F)O
C[C@@]1(CN(C[C@H]1c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)C(=O)c1ccccc1)c1ccccc1 |r|
C[C@@]1(CN(Cc2ccccc2)C[C@H]1c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)c1ccccc1 |r|
CC(=O)N1C[C@@H](c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)[C@](C)(C1)c1ccccc1 |r|
C[C@@]1(CNC[C@H]1c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)c1ccccc1 |r|
C[C@@]1(CN(CC(N)=O)C[C@H]1c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)c1ccccc1 |r|
C[C@@]1(CN(C[C@H]1c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O)c1ccccc1 |r|
CCOC(=O)N1C[C@@H](c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)[C@](C)(C1)c1ccccc1 |r|
CCNC(=O)N1C[C@@H](c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)[C@](C)(C1)c1ccccc1 |r|
C[C@@]1(CN(C[C@H]1c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCc1ccccc1)c1ccccc1 |r|
C[C@]1(CN(C[C@@H]1c1ccccc1)C(=O)NCc1ccccc1)c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F |r|
CC[C@@]1(CN(C[C@H]1c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCc1ccccc1)c1ccccc1 |r|
C[C@@]1(CN(C[C@H]1c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCc1ccccc1)c1ccc(F)cc1 |r|
OC[C@@]1(CN(C[C@H]1c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCc1ccccc1)c1ccc(F)cc1 |r|
C[C@]1(CN(C[C@@H]1c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCc1ccccc1)c1ccc(F)cc1 |r|
COc1ccc(CNC(=O)N2C[C@@H](c3ccc(cc3)C(O)(C(F)(F)F)C(F)(F)F)[C@](C)(C2)c2ccc(F)cc2)cc1 |r|
C[C@@]1(CN(C[C@H]1c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCc1ccc2OCOc2c1)c1ccc(F)cc1 |r|
C[C@@]1(CN(C[C@H]1c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCc1ccncc1)c1ccc(F)cc1 |r|
C[C@@]1(CN(C[C@H]1c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)C(=O)NCc1ccc(cc1)C#N)c1ccc(F)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)N2C[C@@H](c3ccc(cc3)C(O)(C(F)(F)F)C(F)(F)F)[C@](C)(C2)c2ccc(F)cc2)cc1 |r|
CC(=O)N1CCC(CC1)C(=O)N1C[C@H](c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)[C@@](C)(C1)c1ccccc1 |r|
CC(=O)N1CCC(CC1)C(=O)N1C[C@@H](c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)[C@](C)(C1)c1ccc(F)cc1 |r|
CC(=O)N1CCC(CC1)C(=O)N1C[C@@H](c2ccc(cc2)C(F)(C(F)(F)F)C(F)(F)F)[C@](C)(C1)c1ccc(F)cc1 |r|
C[C@@]1(CN(C[C@H]1c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)C(=O)C1CCN(CC1)S(C)(=O)=O)c1ccc(F)cc1 |r|
C[C@@]1(CN(C[C@H]1c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)C(=O)C1CCN(CC1)C(N)=O)c1ccc(F)cc1 |r|
C[C@@]1(CN(C[C@H]1c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)C(=O)C1CCN(CC1)C(=O)C(N)=O)c1ccc(F)cc1 |r|
C[C@@]1(CN(C[C@H]1c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)C(=O)C1CCN(CC1)C(=O)CO)c1ccc(F)cc1 |r|
COCC(=O)N1CCC(CC1)C(=O)N1C[C@@H](c2ccc(cc2)C(O)(C(F)(F)F)C(F)(F)F)[C@](C)(C1)c1ccc(F)cc1 |r|
C[C@@]1(CN(C[C@H]1c1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)C(=O)C1CCN(CC1)C(=O)CC#N)c1ccc(F)cc1 |r|
C[C@H]1CN(Cc2cc(F)cc(NC(=O)CC(CCC(O)=O)c3nccs3)c2C)CCN1C(=O)C1CCCC1 |r|
C[C@H]1CN(Cc2cc(F)cc(NC(=O)CC(CCC(O)=O)c3ccccc3)c2C)CCN1C(=O)C1CCCC1 |r|
C[C@H]1CN(Cc2cc(F)cc(NC(=O)CC(CC(O)=O)c3ccccc3)c2C)CCN1C(=O)C1CCCC1 |r|
C[C@H]1CN(Cc2cc(F)cc(NC(=O)CCCCC(O)=O)c2C)CCN1C(=O)C1CCCC1 |r|
C[C@H]1CN(Cc2cc(F)cc(NC(=O)CCc3ccccc3)c2C)CCN1C(=O)C1CCCC1 |r|
C[C@H]1C[C@H](CCN1C(=O)C1CCCC1)Oc1cc(Cl)cc(NC(=O)CC(CCC(O)=O)c2ccccc2)c1C |r|
C[C@H]1C[C@H](CCN1C(=O)C1CCCC1)Oc1cc(Cl)cc(NC(=O)CC(CCC(O)=O)c2ccccc2)c1Cl |r|
C[C@H]1CN(Cc2cc(Cl)cc(NC(=O)CC(CCC(O)=O)c3ccccc3)c2Cl)CCN1C(=O)C1CCCC1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(44.58,-1.86,;43.76,-3.16,;42.22,-3.1,;40.88,-2.33,;42.21,-1.55,;41.39,-4.4,;42.11,-5.76,;41.28,-7.06,;39.75,-6.99,;38.92,-8.29,;37.38,-8.22,;36.56,-9.52,;37.27,-10.89,;35.02,-9.46,;34.3,-8.09,;32.76,-8.03,;32.05,-6.66,;31.94,-9.32,;32.65,-10.69,;31.83,-11.99,;34.19,-10.76,;30.41,-9.26,;29.58,-10.57,;28.04,-10.49,;27.33,-9.12,;28.17,-7.82,;29.7,-7.89,;30.53,-6.6,;29.82,-5.23,;28.45,-5.93,;28.53,-4.39,;30.65,-3.93,;39.03,-5.64,;39.85,-4.34,)|
CCS(=O)(=O)c1ccc(OCC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(22.97,-19.33,;21.43,-19.26,;20.71,-17.9,;20.7,-16.36,;22.04,-17.12,;19.18,-17.84,;18.35,-19.14,;16.81,-19.07,;16.11,-17.71,;14.57,-17.64,;13.75,-18.94,;12.21,-18.88,;11.49,-17.51,;11.38,-20.18,;9.84,-20.11,;9.12,-18.74,;7.59,-18.68,;6.87,-17.32,;6.77,-19.98,;7.48,-21.35,;6.65,-22.65,;9.02,-21.41,;5.24,-19.91,;4.4,-21.22,;2.86,-21.15,;2.15,-19.78,;2.99,-18.48,;4.52,-18.55,;5.35,-17.25,;4.64,-15.88,;3.27,-16.58,;3.35,-15.04,;5.47,-14.59,;16.92,-16.41,;18.46,-16.47,)|
CCS(=O)(=O)c1ccc(CCNc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(44.93,-13.7,;44.1,-15,;42.56,-14.94,;41.22,-14.17,;42.56,-13.4,;41.74,-16.24,;42.45,-17.61,;41.63,-18.91,;40.09,-18.83,;39.27,-20.14,;37.73,-20.07,;36.9,-21.37,;35.36,-21.31,;34.64,-19.94,;33.11,-19.88,;32.39,-18.51,;32.29,-21.17,;33,-22.54,;32.17,-23.84,;34.54,-22.61,;30.76,-21.1,;29.92,-22.41,;28.38,-22.34,;27.67,-20.97,;28.51,-19.67,;30.04,-19.74,;30.87,-18.44,;30.16,-17.07,;28.79,-17.77,;28.87,-16.23,;30.99,-15.78,;39.37,-17.48,;40.19,-16.18,)|
CCS(=O)(=O)c1ccc(CCOc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(67.84,-12.25,;67.01,-13.55,;65.47,-13.49,;64.13,-12.72,;65.47,-11.94,;64.65,-14.79,;65.36,-16.15,;64.54,-17.45,;63,-17.38,;62.18,-18.68,;60.64,-18.61,;59.81,-19.92,;58.27,-19.85,;57.55,-18.48,;56.02,-18.42,;55.3,-17.06,;55.2,-19.71,;55.91,-21.08,;55.08,-22.38,;57.45,-21.15,;53.67,-19.65,;52.83,-20.96,;51.29,-20.88,;50.58,-19.51,;51.42,-18.22,;52.96,-18.28,;53.78,-16.99,;53.07,-15.62,;51.7,-16.32,;51.78,-14.78,;53.9,-14.32,;62.28,-16.03,;63.1,-14.73,)|
CCS(=O)(=O)c1ccc(COCc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(19.56,-25.41,;18.74,-26.71,;17.2,-26.65,;15.86,-25.88,;17.2,-25.1,;16.38,-27.95,;17.09,-29.32,;16.26,-30.61,;14.73,-30.54,;13.9,-31.84,;12.36,-31.78,;11.54,-33.08,;10,-33.01,;9.28,-31.64,;7.75,-31.58,;7.03,-30.22,;6.92,-32.88,;7.63,-34.24,;6.81,-35.54,;9.17,-34.31,;5.39,-32.81,;4.56,-34.12,;3.02,-34.05,;2.31,-32.68,;3.15,-31.38,;4.68,-31.45,;5.51,-30.15,;4.8,-28.78,;3.43,-29.48,;3.51,-27.94,;5.63,-27.48,;14.01,-29.19,;14.83,-27.89,)|
OCC(O)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(73.27,-4.31,;71.73,-4.25,;70.91,-5.55,;71.62,-6.91,;69.37,-5.49,;68.54,-6.79,;67.01,-6.72,;66.3,-5.36,;64.76,-5.29,;63.94,-6.59,;62.4,-6.53,;61.69,-5.16,;61.57,-7.83,;60.04,-7.76,;59.32,-6.39,;57.78,-6.33,;57.07,-4.97,;56.96,-7.63,;57.67,-9,;56.84,-10.3,;59.21,-9.06,;55.43,-7.56,;54.59,-8.87,;53.05,-8.8,;52.34,-7.43,;53.18,-6.13,;54.72,-6.2,;55.54,-4.9,;54.83,-3.53,;53.46,-4.23,;53.54,-2.69,;55.66,-2.24,;67.11,-4.06,;68.65,-4.12,)|
CC(C(O)=O)c1ccc(CNC(=O)Nc2ccc(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1
CC(C(O)=O)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccccc2OC(F)F)cc1 |(70.2,-5.84,;69.48,-4.48,;70.31,-3.17,;71.84,-3.24,;69.59,-1.81,;67.94,-4.41,;67.12,-5.71,;65.58,-5.65,;64.88,-4.28,;63.34,-4.22,;62.51,-5.52,;60.97,-5.46,;60.26,-4.09,;60.15,-6.76,;58.61,-6.69,;57.89,-5.32,;56.35,-5.26,;55.64,-3.9,;55.53,-6.55,;56.24,-7.92,;55.42,-9.22,;57.78,-7.99,;54,-6.49,;53.17,-7.8,;51.63,-7.72,;50.92,-6.35,;51.76,-5.06,;53.29,-5.13,;54.12,-3.83,;53.41,-2.46,;54.24,-1.16,;51.87,-2.39,;65.69,-2.98,;67.22,-3.04,)|
CC(C(O)=O)c1ccc(CNC(=O)Nc2cc(C)c(c(Cl)c2)-c2ccccc2OC(F)(F)F)cc1 |(20.66,-16.3,;19.94,-14.94,;20.76,-13.64,;22.3,-13.7,;20.05,-12.27,;18.4,-14.87,;17.57,-16.18,;16.04,-16.11,;15.33,-14.75,;13.79,-14.68,;12.97,-15.98,;11.43,-15.92,;10.72,-14.55,;10.61,-17.22,;9.07,-17.15,;8.24,-18.45,;6.7,-18.39,;5.87,-19.68,;5.99,-17.02,;6.81,-15.72,;6.1,-14.36,;8.35,-15.78,;4.46,-16.95,;3.63,-18.26,;2.08,-18.19,;1.38,-16.82,;2.21,-15.52,;3.75,-15.59,;4.57,-14.29,;3.86,-12.92,;2.49,-13.62,;2.57,-12.08,;4.69,-11.62,;16.14,-13.45,;17.68,-13.5,)|
CC(C(O)=O)c1ccc(CNC(=O)Nc2cc(Cl)c(c(c2)C#N)-c2ccccc2OC(F)(F)F)cc1 |(45.36,-15.77,;44.65,-14.41,;45.47,-13.11,;47.01,-13.17,;44.76,-11.74,;43.11,-14.34,;42.28,-15.65,;40.75,-15.58,;40.04,-14.22,;38.5,-14.15,;37.68,-15.45,;36.14,-15.39,;35.43,-14.02,;35.31,-16.69,;33.78,-16.62,;33.06,-15.25,;31.52,-15.19,;30.81,-13.83,;30.7,-16.49,;31.41,-17.86,;32.95,-17.92,;30.58,-19.15,;29.76,-20.46,;29.17,-16.42,;28.33,-17.73,;26.79,-17.66,;26.09,-16.29,;26.92,-14.99,;28.46,-15.06,;29.28,-13.76,;28.57,-12.39,;27.2,-13.09,;27.28,-11.55,;29.4,-11.09,;40.85,-12.92,;42.39,-12.98,)|
Cc1cc(NC(=O)NCc2ccc(CC(O)=O)cc2)cc(C)c1-c1ccccc1OC(F)(F)F |(55.97,-13.73,;56.68,-15.09,;58.22,-15.15,;58.94,-16.52,;60.48,-16.59,;61.3,-15.29,;60.59,-13.92,;62.84,-15.35,;63.67,-14.05,;65.21,-14.12,;65.91,-15.48,;67.45,-15.55,;68.27,-14.24,;69.81,-14.31,;70.64,-13.01,;72.18,-13.07,;69.92,-11.64,;67.55,-12.87,;66.02,-12.82,;58.11,-17.82,;56.57,-17.76,;55.75,-19.05,;55.86,-16.39,;54.33,-16.32,;53.5,-17.63,;51.96,-17.56,;51.25,-16.19,;52.08,-14.89,;53.62,-14.96,;54.45,-13.66,;53.74,-12.29,;52.36,-12.99,;52.45,-11.45,;54.56,-10.99,)|
Cc1cc(NC(=O)NCc2ccc(CC(O)=O)cn2)cc(C)c1-c1ccccc1OC(F)F |(5.75,-25.97,;6.47,-27.33,;8,-27.39,;8.72,-28.76,;10.26,-28.83,;11.09,-27.53,;10.37,-26.16,;12.63,-27.59,;13.45,-26.29,;14.99,-26.36,;15.8,-25.06,;17.34,-25.12,;18.06,-26.49,;19.6,-26.55,;20.42,-25.25,;21.96,-25.31,;19.71,-23.88,;17.23,-27.79,;15.69,-27.72,;7.9,-30.06,;6.36,-30,;5.53,-31.3,;5.65,-28.63,;4.12,-28.56,;3.28,-29.87,;1.74,-29.8,;1.03,-28.43,;1.87,-27.13,;3.4,-27.2,;4.23,-25.9,;3.52,-24.53,;4.35,-23.23,;1.98,-24.46,)|
OC(=O)Cc1ccc(CNC(=O)Nc2cc(F)c(c(F)c2)-c2ccccc2OC(F)(F)F)nc1 |(46.5,-23.85,;44.96,-23.79,;44.25,-22.42,;44.14,-25.09,;42.6,-25.02,;41.88,-23.65,;40.34,-23.6,;39.53,-24.9,;37.99,-24.83,;37.17,-26.13,;35.63,-26.07,;34.91,-24.7,;34.8,-27.37,;33.26,-27.3,;32.54,-25.93,;31.01,-25.87,;30.29,-24.51,;30.19,-27.17,;30.9,-28.54,;30.07,-29.83,;32.44,-28.6,;28.66,-27.1,;27.82,-28.41,;26.28,-28.34,;25.57,-26.97,;26.41,-25.67,;27.94,-25.74,;28.77,-24.44,;28.06,-23.07,;26.69,-23.77,;26.77,-22.23,;28.89,-21.77,;40.23,-26.26,;41.77,-26.33,)|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCCc4ccc(CC(C)C)cc34)cc2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc(CCN3CCCc4ccc(CC(C)C)cc34)cc2)nc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc(CCN3CCOc4ccc(OC(C)C)cc34)cc2)nc1
CC(C)Oc1ccc2OCCN(CCc3ccc(cc3)C(=O)NCc3ccc(cn3)S(C)(=O)=O)c2c1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCCc4ccccc34)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCCc4ccc(C)cc34)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCCc4c(C)cccc34)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCCc4ccc(F)cc34)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCCc4ccc(Cl)cc34)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCCc4ccc(OC)cc34)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCCc4ccc(cc34)C3CC3)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCCc4ccc(cc34)C(C)C)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCCc4ccc(cc34)C(C)(C)C)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCCc4ccc(CC(C)(C)C)cc34)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCCc4ccc(CC5CC5)cc34)cc2)cc1
[#6]-[#6]S(=O)(=O)c1ccc(-[#6]-[#6](=O)-[#7]-c2ccc(-[#6]-[#6]-[#7]-3-[#6]-[#6]-[#6]-c4ccc(\[#6]=[#6](/[#6])-[#6])cc-34)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCCc4ccc(CN(C)C)cc34)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCCc4ccc(OC(C)C)cc34)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCCc4ccc(OC(C)(C)C)cc34)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCCc4ccc(OC5CCC5)cc34)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCCc4ccc(OC5COC5)cc34)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCCc4ccc(CC(C)C)cc34)c(F)c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)Nc2ccc(CCN3CCCc4ccc(CC(C)C)cc34)cc2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc(CCN3CCCc4ccc(CC(C)C)cc34)cc2)cc1
CCS(=O)(=O)c1ccc(cc1)C(CO)NC(=O)c1ccc(CCN2CCCc3ccc(CC(C)C)cc23)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCCc4ccc(CC(C)C)cc34)cc2)nc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc(CCN3CCCc4ccc(OC(C)C)cc34)cc2)nc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc(CCN3CCCc4ccc(OC5CCC5)cc34)cc2)nc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc(CCN3CCCc4ccc(OC5COC5)cc34)cc2)nc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCOc4ccc(CC(C)C)cc34)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCOc4ccc(OC(C)C)cc34)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCOc4ccc(OC(C)C)cc34)c(F)c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc(CCN3CCOc4ccc(OC(C)C)cc34)c(Cl)c2)nc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc(CCN3CCOc4ccc(CC(C)C)cc34)cc2)nc1
CC(C)Oc1ccc2OCCN(CCc3ccc(NC(=O)Cc4ccc(cc4)S(C)(=O)=O)cc3)c2c1
CC(Oc1ccc2OCCN(CCc3ccc(NC(=O)Cc4ccc(cc4)S(C)(=O)=O)cc3)c2c1)C(F)(F)F
CS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCOc4ccc(cc34)C(F)(C(F)(F)F)C(F)(F)F)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CC(=O)N3CCCc4ccc(CC(C)C)cc34)cc2)cc1
CS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCN3CCOc4ccc(cc34)C(O)(C(F)(F)F)C(F)(F)F)cc2)cc1
[H][C@@]12CCc3cc(ccc3[C@@]1(CC[C@H]2NC(=O)C(C)(C)N1CCOCC1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CC[C@H]2NC(=O)[C@H]1C[C@H](F)C(=O)N1C([2H])([2H])[2H])S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CC[C@H]2NC1CCN(CC1)S(C)(=O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CC[C@H]2NC1CCS(=O)(=O)CC1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CC[C@H]2NC1(O)CCS(=O)(=O)CC1)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2N[C@@H]1CC[C@H](C[C@@H]1C)C(O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CC[C@H]2NC(=O)[C@H]1C[C@H](O)C(=O)N1CCC#N)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CC[C@H]2NC(=O)[C@H]1C[C@H](O)C(=O)N1C([2H])([2H])[2H])S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
[H][C@@]12CCc3cc(ccc3[C@@]1(CCN2N[C@H]1CC[C@@H](CC1)C(O)=O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r,wU:15.17,wD:1.0,10.27,18.24,(68.13,-45.44,;66.81,-46.22,;66.81,-44.67,;65.47,-43.9,;64.14,-44.67,;62.81,-43.91,;61.48,-44.68,;61.48,-46.22,;62.81,-46.99,;64.14,-46.22,;65.47,-46.99,;65.78,-48.5,;67.32,-48.67,;67.95,-47.26,;69.46,-46.94,;70.48,-48.09,;71.99,-47.77,;73.01,-48.93,;72.52,-50.39,;71.02,-50.7,;70,-49.55,;73.55,-51.54,;75.05,-51.23,;73.06,-53,;64.69,-48.31,;66.02,-49.08,;64.69,-49.85,;63.15,-48.31,;62.4,-46.97,;60.86,-46.96,;60.08,-48.29,;58.54,-48.28,;60.85,-49.63,;62.39,-49.63,;60.14,-43.91,;60.91,-42.57,;59.37,-42.57,;58.96,-41.08,;60.46,-41.47,;57.83,-42.58,;58.81,-44.68,;59.57,-46.01,;58.04,-46,;57.48,-43.91,)|
[H][C@@]12CCc3cc(ccc3[C@@]1(CC[C@H]2N(C)C(=O)C(C)(C)O)S(=O)(=O)c1ccc(F)cc1)C(F)(C(F)(F)F)C(F)(F)F |r|
OC(=O)c1cc(c2cc(ccc2n1)N1CCC2(CC(=C2)c2c(onc2-c2c(Cl)cncc2Cl)C2CC2)CC1)C(F)(F)F |c:20,(46.96,-23.25,;46.47,-24.71,;47.49,-25.87,;44.96,-25.01,;44.46,-26.48,;42.95,-26.78,;41.94,-25.62,;40.43,-25.91,;39.43,-24.74,;39.93,-23.29,;41.43,-22.99,;42.44,-24.16,;43.95,-23.86,;37.92,-25.03,;37.41,-26.48,;35.91,-26.76,;34.9,-25.6,;33.89,-24.44,;32.72,-25.45,;33.74,-26.62,;31.19,-25.35,;30.71,-23.88,;29.16,-23.89,;28.69,-25.36,;29.95,-26.26,;29.96,-27.8,;28.63,-28.57,;27.29,-27.8,;28.63,-30.11,;29.96,-30.88,;31.3,-30.11,;31.29,-28.56,;32.62,-27.79,;31.6,-22.64,;33.01,-22.01,;31.76,-21.1,;35.4,-24.15,;36.91,-23.86,;42.45,-28.23,;43.47,-29.39,;40.97,-27.83,;41.68,-29.57,)|
CN(Cc1ccccc1C(F)(F)F)S(=O)(=O)N1CCc2cc(ccc2C1)N1CCN(CC1)C(C)=O
CN(Cc1ccccc1Cl)S(=O)(=O)N1CCc2cc(ccc2C1)N1CCN(CC1)C(C)=O
CN(Cc1c(F)cccc1Cl)S(=O)(=O)N1CCc2cc(ccc2C1)N1CCN(CC1)C(C)=O
CN(c1nccc(n1)C(F)(F)F)S(=O)(=O)N1CCc2cc(ccc2C1)N1CCN(CC1)C(C)=O
CN(Cc1ccccn1)S(=O)(=O)N1CCc2cc(ccc2C1)N1CCN(CC1)C(C)=O
CN(Cc1ccccc1)S(=O)(=O)N1CCc2cc(ccc2C1)N1CCN(CC1)C(C)=O
CN(CCc1ccccc1)S(=O)(=O)N1CCc2cc(ccc2C1)N1CCN(CC1)C(C)=O
CN(CCCc1ccccc1)S(=O)(=O)N1CCc2cc(ccc2C1)N1CCN(CC1)C(C)=O
CN(Cc1ccc(C)cc1)S(=O)(=O)N1CCc2cc(ccc2C1)N1CCN(CC1)C(C)=O
CN(Cc1ccc(F)cc1)S(=O)(=O)N1CCc2cc(ccc2C1)N1CCN(CC1)C(C)=O
CN(Cc1cccc(c1)C(F)(F)F)S(=O)(=O)N1CCc2cc(ccc2C1)N1CCN(CC1)C(C)=O
CN(Cc1cccc(Cl)c1)S(=O)(=O)N1CCc2cc(ccc2C1)N1CCN(CC1)C(C)=O
CN(Cc1ccccc1C)S(=O)(=O)N1CCc2cc(ccc2C1)N1CCN(CC1)C(C)=O
CN(Cc1cccc(C)c1)S(=O)(=O)N1CCc2cc(ccc2C1)N1CCN(CC1)C(C)=O
CN(Cc1ccccc1F)S(=O)(=O)N1CCc2cc(ccc2C1)N1CCN(CC1)C(C)=O
CN(Cc1cccc(F)c1)S(=O)(=O)N1CCc2cc(ccc2C1)N1CCN(CC1)C(C)=O
CN(Cc1cc(F)ccc1F)S(=O)(=O)N1CCc2cc(ccc2C1)N1CCN(CC1)C(C)=O
C[C@@H]1CN(CCN1c1ccc2CN(CCc2c1)S(=O)(=O)N(C)Cc1c(F)cccc1Cl)C(C)=O |r|
C[C@H]1CN(CCN1C(C)=O)c1ccc2CN(CCc2c1)S(=O)(=O)N(C)Cc1c(F)cccc1Cl |r|
C[C@@H]1CN(CCN1C(C)=O)c1ccc2CN(CCc2c1)S(=O)(=O)N(C)Cc1c(F)cccc1Cl |r|
C[C@H]1CN(C[C@@H](C)N1C(C)=O)c1ccc2CN(CCc2c1)S(=O)(=O)N(C)Cc1c(F)cccc1Cl |r|
CN(Cc1c(F)cccc1Cl)S(=O)(=O)N1CCc2cc(ccc2C1)N1C2CC1CN(C2)C(C)=O
Fc1cccc(Cl)c1OCc1ccc2CCN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
CCN1c2ccc(cc2OCC1=O)N(CC(F)(F)F)S(=O)(=O)c3ccc(c(c3)C)C
CN(Cc1ccccc1Cl)S(=O)(=O)N1CCCc2cc(ccc12)N1CCN(CC1)C(C)=O
CN(Cc1ccc(cc1)C(F)(F)F)S(=O)(=O)N1CCc2cc(ccc2C1)N1CCN(CC1)C(C)=O
CCS(=O)(=O)c1ccc(nc1)C(NC(C)=O)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(nc1)C(NC(=O)OC)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(nc1)C(NC(=O)CC1CC1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(nc1)C(NC(=O)Cc1ccccc1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(nc1)C(NC(=O)Cc1ccccn1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(nc1)C(NC(=O)Cc1nccs1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)C(CC(=O)NC)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)[C@H](CC(=O)NC)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(cc1)[C@@H](CC(=O)NC)C(=O)Nc2ccc(cc2)C(C(F)(F)F)(C(F)(F)F)O
CCS(=O)(=O)c1ccc(cc1)C(CC(=O)N(C)C)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)C(Cc1nnco1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1)C(Cn1cccn1)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
CC(=O)NC(C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)c1ccc(cc1)S(C)(=O)=O
CC(=O)N1CCc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O
CC(=O)N1Cc2cc(ccc2[C@@H]1C(=O)Nc3ccc(cc3)C(C(F)(F)F)(C(F)(F)F)O)S(=O)(=O)C
CC(=O)N1Cc2cc(ccc2[C@H]1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(C)(=O)=O |r|
CCS(=O)(=O)c1ccc2[C@@H](N(Cc2c1)C(C)=O)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F |r|
CCS(=O)(=O)c1ccc2[C@H](N(Cc2c1)C(C)=O)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F |r|
CS(=O)(=O)c1ccc2C(N(Cc2c1)C(=O)CO)C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F
NCCC(=O)N1Cc2cc(ccc2C1C(=O)Nc1ccc(cc1)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)CC1CC1
COc1cc(ccc1F)S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(\C=C(/C)c3c(F)cccc3Cl)cc12 |r|
C\C(=C/c1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(OC(F)F)c1)c1c(F)cccc1Cl |r|
C\C(=C/c1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C(F)(F)F)c1c(F)cccc1Cl |r|
C\C(=C/c1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1ccc(F)c(c1)C1CC1)c1c(F)cccc1Cl |r|
C\C(=C/c1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1c(OCCO)nn2CCCCc12)c1c(F)cccc1Cl |r|
C\C(=C/c1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)c1ccccc1 |r|
C\C(=C/c1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)c1ccccc1C |r|
C\C(=C/c1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)c1ccccc1C(F)(F)F |r|
C\C(=C/c1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)c1ccccc1Cl |r|
C\C(=C/c1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F)c1c(Cl)cccc1Cl |r|
OC(=O)CC[C@H]1CN(c2cc(\C=C\c3c(F)cccc3Cl)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
OC(=O)CC[C@H]1CN(c2cc(\C=C\c3ccc(Cl)cc3F)ccc2O1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
Cc1ccc(\C=C\c2ccc3O[C@@H](CCC(O)=O)CN(c3c2)S(=O)(=O)c2cccc(c2)C(F)(F)F)cc1 |r|
OC(=O)CC[C@H]1CN(c2cc(ccc2O1)-c1ccccc1Cl)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
OC(=O)CC[C@H]1CN(c2cc(ccc2O1)-c1cccc(Cl)c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
OC(=O)CC[C@H]1CN(c2cc(ccc2O1)-c1ccc(Cl)cc1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
OC(=O)CC[C@H]1CN(c2cc(ccc2O1)-c1cccc(F)c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
COc1cccc(c1)-c1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
OC(=O)CC[C@H]1CN(c2cc(ccc2O1)-c1cccc(OC(F)F)c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CC(C)c1ccc(cc1)-c1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
OCCOc1cccc(c1)-c1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
OC(=O)CC[C@H]1CN(c2cc(ccc2O1)-c1cccc(F)c1Cl)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
OC(=O)CC[C@H]1CN(c2cc(ccc2O1)-c1cc(F)ccc1Cl)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
OC(=O)CC[C@H]1CN(c2cc(ccc2O1)-c1cc(F)cc(F)c1Cl)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
OC(=O)CC[C@H]1CN(c2cc(ccc2O1)-c1cc(F)ccc1F)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
OC(=O)CC[C@H]1CN(c2cc(ccc2O1)-c1cc(F)cc(F)c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
COc1cc(F)cc(c1)-c1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
OC(=O)CC[C@H]1CN(c2cc(ccc2O1)-c1cc(F)cc(OC(F)F)c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
C[C@@H](C[C@H]1CN(c2cc(ccc2O1)-c1cc(F)ccc1F)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(O)=O |r|
C[C@H](C[C@H]1CN(c2cc(ccc2O1)-c1cc(F)ccc1F)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(O)=O |r|
CC(C)(C[C@H]1CN(c2cc(ccc2O1)-c1cc(F)ccc1F)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(O)=O |r|
CC(C)(C[C@H]1CN(c2cc(ccc2O1)-c1cccc(Cl)c1F)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(O)=O |r|
OCC1(C[C@H]2CN(c3cc(Br)ccc3O2)S(=O)(=O)c2cccc(c2)C(F)(F)F)COC1 |r|
OC(=O)C1(C[C@H]2CN(c3cc(ccc3O2)-c2cc(F)cc(OC(F)F)c2)S(=O)(=O)c2cccc(c2)C(F)(F)F)COC1 |r|
OC(=O)C1(C[C@H]2CN(c3cc(ccc3O2)-c2cc(F)ccc2F)S(=O)(=O)c2cccc(c2)C(F)(F)F)COC1 |r|
OC(=O)C1(C[C@H]2CN(c3cc(ccc3O2)-c2cc(F)ccc2F)S(=O)(=O)c2cccc(c2)C(F)(F)F)CCOCC1 |r|
OC(=O)C1(C[C@H]2CN(c3cc(ccc3O2)-c2cc(F)cc(OC(F)F)c2)S(=O)(=O)c2cccc(c2)C(F)(F)F)CCOCC1 |r|
OC(=O)C1(C[C@H]2CN(c3cc(ccc3O2)-c2cccc(Cl)c2F)S(=O)(=O)c2cccc(c2)C(F)(F)F)CCOCC1 |r|
O[C@H](CC[C@H]1CN(c2cc(ccc2O1)-c1cc(F)ccc1F)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(O)=O |r|
O[C@@H](CC[C@H]1CN(c2cc(ccc2O1)-c1cc(F)ccc1F)S(=O)(=O)c1cccc(c1)C(F)(F)F)C(O)=O |r|
CCOc1nn2CCCCc2c1S(=O)(=O)N1C[C@H](CCC(O)=O)Oc2ccc(\C=C(/C)c3c(F)cccc3Cl)cc12 |r|
COc1ccccc1\C(C)=C\c1ccc2O[C@@H](CCC(O)=O)CN(c2c1)S(=O)(=O)c1cccc(c1)C(F)(F)F |r|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CCc2c1)C1CCOCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(C)(O)c2c1)C1CCOCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCOCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(C)c2c1)C1CCOCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(C=Cc2c1)C1CCOCC1 |c:23|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2nc(cc(O)c2c1)C1CCOCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c(CN)c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c2C(O)CCCc12
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c2C(O)CCc12
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2C(CCc2c1)OC1CCOCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(N)c2c1)C1CCOCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(OC)c2c1)C1CCOCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(OC3CCCCC3)c2c1)C1CCOCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC3CCOCC3)CC(O)c2c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCN(C)CC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCNCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCN(CC1)S(C)(=O)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCN(CC1)C(=O)C1CCCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C(C)C1CCOCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2O[C@@H](CC(O)c2c1)C1CCOCC1 |r|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2O[C@H](CC(O)c2c1)C1CCOCC1 |r|
CC(C)CN(c1ccc(C)cc1C)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCOCC1
CC(C)CN(c1ccccc1F)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCOCC1
CC(C)CN(c1cccc(F)c1)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCOCC1
CC(C)CN(c1ccc(F)cc1)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCOCC1
CC(C)CN(c1ccc(F)cc1F)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCOCC1
CC(C)CN(c1ccccc1C(F)(F)F)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCOCC1
CC(C)CN(Cc1ccccc1C(F)(F)F)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCOCC1
CC(C)CN(c1ccc(cc1)C#N)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCOCC1
CC(C)CN(c1ccc(cc1)N(C)C)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCOCC1
CCS(=O)(=O)c1ccc(CN(CC(C)C)S(=O)(=O)c2ccc3OC(CC(O)c3c2)C2CCOCC2)nc1
CC(C)CN(c1ccc(cc1C)C(O)(C(F)(F)F)C(F)(F)F)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCOCC1
CC(C)CN(C1CCc2ccc(F)cc12)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCOCC1
CC(C)CN(c1cc2ccccc2s1)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCOCC1
CCc1ccc2N(CC(C)Cc2c1)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCOCC1
OC1CC(Oc2ccc(cc12)S(=O)(=O)Nc1ccccc1C(F)(F)F)C1CCOCC1
CCc1ccc(cc1)N(C1CCC1)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCOCC1
CCc1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCOCC1
CCc1ccc(NS(=O)(=O)c2ccc3OC(CC(O)c3c2)C2CCOCC2)cc1
OC1CC(Oc2ccc(cc12)S(=O)(=O)N1CCCC1c1ccccc1C(F)(F)F)C1CCOCC1
CCc1ccc(cc1)N(CC1CCC1)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCOCC1
CCc1ccc(cc1)N(C1COC1)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCOCC1
Cc1ccc(N(C2CCC2)S(=O)(=O)c2ccc3OC(CC(O)c3c2)C2CCOCC2)c(C)c1
CCc1ccc(cc1)N(Cc1ccccc1)S(=O)(=O)c1ccc2OC(CC(O)c2c1)C1CCOCC1
OC1CC(Oc2ccc(cc12)S(=O)(=O)N1CCC(CC1)c1ccccc1)C1CCOCC1
Cc1c(CN2CCN(CC2)C(=O)C2CCCC2)cccc1Nc1nc2ccccc2s1
Cc1c(CN2CCN(CC2)C(=O)C2CCCC2)cccc1Nc1nc2ccccc2o1
Cc1c(CN2CCN(CC2)C(=O)C2CCCC2)cccc1NC(=O)Nc1ccccc1
Cc1c(CN2CCN(CC2)C(=O)C2CCCC2)cccc1NC(=S)Nc1ccccc1
Cc1c(CN2CCN(CC2)C(=O)C2CCCC2)cccc1Nc1nc2cccnc2s1
Cc1c(CN2CCN(CC2)C(=O)C2CCCC2)cccc1Nc1nc2ncccc2s1
Cc1c(CN2CCN(CC2)C(=O)C2CCCC2)cccc1Nc1nc2nccnc2s1
Cc1c(CN2CCN(CC2)C(=O)C2CCCC2)cccc1Nc1nc2CCCc2s1
Cc1c(CN2CCN(CC2)C(=O)C2CCCC2)cccc1Nc1nc2CCCCc2s1
Cc1c(CN2CCN(CC2)C(=O)C2CCCC2)cccc1Nc1nc2CCCCCc2s1
Cc1c(CN2CCN(CC2)C(=O)C2CCCC2)cccc1Nc1nc2CCOCc2s1
Cc1c(CN2CCN(CC2)C(=O)C2CCCC2)cccc1Nc1nc2CCCC(=O)c2s1
Cc1c(CN2CCN(CC2)C(=O)C2CCCC2)cccc1Nc1nc2c(CCCC2=O)s1
Cc1c(CN2CCN(CC2)C(=O)C2CCCC2)cccc1Nc1nc2c(CCC\C2=N/O)s1
CO\N=C1/CCCc2sc(Nc3cccc(CN4CCN(CC4)C(=O)C4CCCC4)c3C)nc12
Cc1c(CN2CCN(CC2)C(=O)C2CCCC2)cccc1Nc1nc2CCCC(O)c2s1
Cc1c(CN2CCN(CC2)C(=O)C2CCCC2)cccc1Nc1nc2C(O)CCCc2s1
COC1CCCc2sc(Nc3cccc(CN4CCN(CC4)C(=O)C4CCCC4)c3C)nc12
Cc1ccc(Nc2nc3ccccc3s2)c(C)c1CN1CCN(CC1)C(=O)C1CCCC1
Cc1c(Nc2nc3ccccc3s2)ccc(Cl)c1CN1CCN(CC1)C(=O)C1CCCC1
Cc1c(CN2CCN(CC2)C(=O)C2CCCC2)cc(F)cc1Nc1nc2ccccc2s1
Cc1c(CN2CCN(CC2)C(=O)C2CCCC2)cc(Cl)cc1Nc1nc2ccccc2s1
Cc1c(Nc2nc3ccccc3s2)cc(Cl)cc1OC1CCN(CC1)C(=O)CC(C(F)(F)F)C(F)(F)F
Cc1c(Nc2nc3CCCCc3s2)cc(Cl)cc1OC1CCN(CC1)C(=O)CC(C(F)(F)F)C(F)(F)F
Cc1c(Nc2nc3c(CCCC3=O)s2)cc(Cl)cc1OC1CCN(CC1)C(=O)CC(C(F)(F)F)C(F)(F)F
Cc1c(Nc2nc3C(O)CCCc3s2)cc(Cl)cc1OC1CCN(CC1)C(=O)CC(C(F)(F)F)C(F)(F)F
Cc1c(Nc2nc3[C@H](O)CCCc3s2)cc(Cl)cc1OC1CCN(CC1)C(=O)CC(C(F)(F)F)C(F)(F)F |r|
Cc1c(Nc2nc3[C@@H](O)CCCc3s2)cc(Cl)cc1OC1CCN(CC1)C(=O)CC(C(F)(F)F)C(F)(F)F |r|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c2C(=O)CCCc12
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2cc(OCC3CCOCC3)c(CO)cc2c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2cc(OCC3CCOCC3)c(cc2c1)C(=O)OC
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2cc(OCC3CCOCC3)c(cc2c1)C(=O)OCC1CCOCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2cc(OCC3CCOCC3)c(cc2c1)C(O)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2CN(C3CCOCC3)C(=O)c2c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2oc(cc(=O)c2c1)C1CCOCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc(OCC2CCOCC2)c2C(=O)CCc12
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(F)c2c1)C1CCOCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2O[C@@H](CC(=O)c2c1)C1CCOCC1 |r|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2O[C@H](CC(=O)c2c1)C1CCOCC1 |r|
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC3CCOCC3)CC(=O)c2c1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCN(CC1)C(=O)OC(C)(C)C
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCNCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCN(CC1)S(C)(=O)=O
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)c1c(C)noc1C
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCN(CC1)C(=O)C1CCCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCN(CC1)S(=O)(=O)C1CCCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C(C)C1CCOCC1
CCc1ccc(cc1)N(CC(C)C)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1(C)CCOCC1
CC(C)CN(c1ccc(C)cc1C)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CC(C)CN(c1ccccc1F)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CC(C)CN(c1cccc(F)c1)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CC(C)CN(c1ccc(F)cc1)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CC(C)CN(c1ccc(cc1)C#N)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CC(C)CN(Cc1ccccc1C(F)(F)F)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CC(C)CN(C1CCc2ccc(F)cc12)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CC(C)CN(c1cc2ccccc2s1)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CC(C)CN(c1ccc(nc1C)N1CCOCC1)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CC(C)CN(c1ccc(F)cc1F)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CC(C)CN(c1ccc(cc1)N(C)C)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CC(C)CN(c1ccc(cc1)C(C)(C)C)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CCc1ccc2N(CC(C)Cc2c1)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CCc1ccc(cc1)N(C1CCC1)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CCc1ccc(cc1)N(CC(F)(F)F)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CCc1ccc(NS(=O)(=O)c2ccc3OC(CC(=O)c3c2)C2CCOCC2)cc1
CCS(=O)(=O)c1ccc(CNS(=O)(=O)c2ccc3OC(CC(=O)c3c2)C2CCOCC2)nc1
FC(F)(F)c1ccccc1C1CCCN1S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CCc1ccc(cc1)N(CC1CCC1)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CCc1ccc(cc1)N(C1COC1)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
Cc1ccc(NS(=O)(=O)c2ccc3OC(CC(=O)c3c2)C2CCOCC2)c(C)c1
Cc1ccc(N(C2CCC2)S(=O)(=O)c2ccc3OC(CC(=O)c3c2)C2CCOCC2)c(C)c1
CCc1ccc(cc1)N(Cc1ccccc1)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CCc1ccc(cc1)N(CC1CC1)S(=O)(=O)c1ccc2OC(CC(=O)c2c1)C1CCOCC1
CS(=O)(=O)c1ccc(cc1)CNC(=O)c2cc3c(s2)C4(CCN(CC4)Cc5ccccc5Cl)OCC3
CS(=O)(=O)c1ccc(CNC(=O)c2cc3CCOC4(CCN(Cc5ccc(Cl)cc5Cl)CC4)c3s2)cc1
CS(=O)(=O)c1ccc(CNC(=O)c2cc3CCOC4(CCN(Cc5ccc(Cl)cc5)CC4)c3s2)cc1
CS(=O)(=O)c1ccc(CNC(=O)c2cc3CCOC4(CCN(Cc5ccc(cc5)C(F)(F)F)CC4)c3s2)cc1
CS(=O)(=O)c1ccc(CNC(=O)c2cc3CCOC4(CCN(Cc5ccc(cc5)C#N)CC4)c3s2)cc1
C[C@@H](N1CCC2(CC1)OCCc1cc(sc21)C(=O)NCc1ccc(cc1)S(C)(=O)=O)c1ccc(cc1)C#N |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cc3CCOC4(CCN(CC4)[C@H](C)c4ccc(cc4)C#N)c3s2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cc3CCOC4(CCN(CC4)[C@H](C)c4ccc(cc4)C(F)(F)F)c3s2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cc3CCOC4(CCN(CC4)[C@H](C)c4cnc(nc4)C(F)(F)F)c3s2)cc1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2cc3CCOC4(CCN(CC4)[C@H](C)c4ccc(cc4)C#N)c3s2)nc1 |r|
Clc1ccc(CN2CCC3(CC2)OCCc2ccsc32)c(Cl)c1
CCCN(Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1)Cc1ccccc1F
CCCN(Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1)Cc1ccccc1C
CCCN(Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1)Cc1ccccc1Cl
CCCN(Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1)Cc1cccc(Cl)c1
CCCN(Cc1ccc(Cl)cc1)Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CCCN(Cc1cccs1)Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CCCN(Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1)Cc1cccnc1
CCCN(Cc1nccs1)Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CCCN(CC1CC1)Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CCCN(CC1CCC1)Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CCCN(CC1CCCC1)Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CCCN(CC1CCCCC1)Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CCCN(CC1CCC(F)(F)CC1)Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CCCN(CC1CCOCC1)Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CCCN(CC1CCCO1)Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CNCc3ccccc3)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CN(C)Cc3ccccc3)cc2)cc1
CCN(Cc1ccccc1)Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CCCCN(Cc1ccccc1)Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CN(CC(C)C)Cc3ccccc3)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CN(CC3CC3)Cc3ccccc3)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CN(CC3CCC3)Cc3ccccc3)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(NCCc3ccccc3)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CCNc3ccccc3)cc2)cc1
CCCN(CCc1ccccc1)c1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CCCN(CCc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1)c1ccccc1
CCCN(Cc1ccccc1)Cc1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1Cl
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(CN(CC3CC3)Cc3ccccc3)c(Cl)c2)cc1
CCCN(Cc1ccccc1)Cc1c(Cl)cc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1Cl
CCCN(Cc1ccccc1)Cc1ccc(NC(=O)NCc2ccc(cc2)S(=O)(=O)CC)cc1
CCCN(Cc1ccccc1)Cc1ccc(cc1)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCCN(Cc1ccccc1)Cc1ccc(NCCc2ccc(cc2)S(=O)(=O)CC)cc1
CCCN(Cc1ccccc1)Cc1ccc(NC(=O)Cc2ccc(cc2)S(C)(=O)=O)cc1
CCCN(Cc1ccccc1)Cc1ccc(NC(=O)Cc2ccc(cc2)C(O)=O)cc1
CCCN(Cc1ccccc1)Cc1ccc(NC(=O)Cc2ccc(cc2)C#N)cc1
CCCN(Cc1ccccc1)Cc1ccc(NC(=O)Cc2ccccc2)cc1
CCCN(Cc1ccccc1)Cc1ccc(NC(=O)Cc2ccc(cn2)S(=O)(=O)CC)cc1
CCCN(CC1CCCCC1)Cc1ccc(NC(=O)Cc2ccc(cc2)S(C)(=O)=O)cc1Cl
CCCN(CC1CCCCC1)Cc1ccc(NC(=O)Cc2ccc(cc2)S(C)(=O)=O)cc1
CCCN(CC1CCCCC1)Cc1c(Cl)cc(NC(=O)Cc2ccc(cc2)S(C)(=O)=O)cc1Cl
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C(C)C)c(Cc4ccccc4C(F)(F)F)cc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C(C)C)c(Cc4ccc(F)cc4C(F)(F)F)cc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C(C)C)c(Cc4ccc(Cl)cc4C(F)(F)F)cc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C4CC4)c(Cc4ccc(Cl)cc4C(F)(F)F)cc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CCF)c(Cc4ccc(Cl)cc4C(F)(F)F)cc3c2)cc1
CCS(=O)(=O)c1ccc(cc1)[C@@H](CO)NC(=O)c1ccc2n(CCF)c(Cc3ccc(Cl)cc3C(F)(F)F)cc2c1 |r|
CCS(=O)(=O)c1ccc(cc1)[C@H](CO)NC(=O)c1ccc2n(CCF)c(Cc3ccc(Cl)cc3C(F)(F)F)cc2c1 |r|
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C(C)C)c(Cc4ccccc4OC(F)(F)F)cc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C(C)C)c(Cc4ccccc4OC)cc3c2)cc1
CCc1ccccc1Cc1cc2cc(ccc2n1C(C)C)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C(C)C)c(Cc4ccccc4Br)cc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C(C)C)c(Cc4ccccc4Cl)cc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C(C)C)c(Cc4ccccc4C)cc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C(C)C)c(Cc4ccccc4)cc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C(C)C)c(Cc4cccc(c4)C(F)(F)F)cc3c2)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(C(C)C)c(Cc4ccc(cc4)C(F)(F)F)cc3c2)cc1
CCOC(=O)C1C(NC(=O)N=C1C)c1ccc(OCc2ccccc2)c(OC)c1 |c:10|
CCCOc1cc(Oc2ccccc2)ccc1COc1c(Cl)cc(cc1OC)C1NC(=O)NC(C)=C1C(=O)OCC |c:37|
CC(C)n1c2ccc(NC(=O)N3CCOC(C3)C(=O)Nc3ccc(C#N)c(Cl)c3)cc2c(=O)n(CC2CC2)c1=O
FC(F)(F)Oc1ccccc1S(=O)(=O)N1Cc2ccccc2COC[C@H]1Cc1ccccc1 |r|
c1cc(cc(c1)S(=O)(=O)N2CCOc3ccc(cc3C2)NC(=O)c4c(cccc4Cl)F)C(F)(F)F
C[C@H]1CN(Cc2c(C)c(NC(=O)c3cnc(C)nc3)cn3ccnc23)CCN1c1noc(n1)C(C)(C)C |r|
OC(=O)c1ccc(OCc2c(noc2-c2cc[nH]c2)-c2c(Cl)cccc2C(F)(F)F)cc1 |(43.77,-15.96,;42.3,-15.49,;41.16,-16.52,;41.98,-13.98,;40.51,-13.51,;40.18,-12.01,;41.33,-10.98,;41,-9.47,;39.54,-9,;39.21,-7.5,;37.8,-6.88,;37.96,-5.34,;39.46,-5.02,;40.24,-6.35,;41.76,-6.5,;42.53,-7.83,;44.04,-7.51,;44.19,-5.97,;42.78,-5.35,;36.47,-7.65,;36.48,-9.2,;37.81,-9.97,;35.14,-9.97,;33.81,-9.2,;33.81,-7.65,;35.14,-6.88,;35.13,-5.34,;36.47,-4.57,;33.8,-4.58,;35.12,-3.8,;42.79,-11.44,;43.12,-12.94,)|
OC(=O)c1ccc(SCc2c(noc2-c2cc[nH]c2)-c2c(Cl)cccc2C(F)(F)F)cc1 |(61.1,-16.42,;59.63,-15.95,;58.49,-16.99,;59.3,-14.45,;57.83,-13.98,;57.51,-12.47,;58.65,-11.44,;58.33,-9.94,;56.86,-9.47,;56.54,-7.96,;55.13,-7.34,;55.28,-5.81,;56.79,-5.48,;57.56,-6.81,;59.08,-6.97,;59.86,-8.3,;61.36,-7.97,;61.52,-6.44,;60.11,-5.82,;53.8,-8.11,;53.81,-9.66,;55.14,-10.43,;52.47,-10.43,;51.13,-9.66,;51.14,-8.12,;52.47,-7.35,;52.46,-5.81,;53.79,-5.04,;51.13,-5.04,;52.45,-4.26,;60.11,-11.9,;60.44,-13.4,)|
CN(Cc1c(noc1-c1cc[nH]c1)-c1c(Cl)cccc1C(F)(F)F)c1ccc(cc1)C(O)=O |(75.8,-9.43,;74.66,-10.47,;73.19,-10,;72.86,-8.49,;71.45,-7.87,;71.61,-6.34,;73.11,-6.01,;73.89,-7.35,;75.41,-7.5,;76.19,-8.83,;77.69,-8.5,;77.85,-6.97,;76.44,-6.35,;70.13,-8.64,;70.13,-10.2,;71.47,-10.96,;68.8,-10.97,;67.46,-10.2,;67.46,-8.65,;68.79,-7.88,;68.79,-6.34,;70.12,-5.57,;67.45,-5.58,;68.77,-4.79,;74.98,-11.97,;73.84,-13,;74.16,-14.51,;75.63,-14.98,;76.77,-13.94,;76.44,-12.44,;75.96,-16.48,;77.42,-16.95,;74.82,-17.52,)|
OC(=O)c1ccc(\C=C\c2c(noc2-c2cc[nH]c2)-c2c(Cl)cccc2C(F)(F)F)cc1 |(14.41,-34.54,;12.94,-34.07,;11.81,-35.11,;12.62,-32.56,;11.15,-32.09,;10.82,-30.59,;11.97,-29.56,;11.64,-28.05,;10.18,-27.58,;9.85,-26.08,;8.44,-25.46,;8.6,-23.93,;10.1,-23.6,;10.88,-24.93,;12.4,-25.08,;13.17,-26.41,;14.68,-26.09,;14.83,-24.56,;13.42,-23.93,;7.12,-26.23,;7.12,-27.78,;8.46,-28.55,;5.78,-28.55,;4.45,-27.78,;4.45,-26.24,;5.78,-25.47,;5.78,-23.93,;7.11,-23.15,;4.44,-23.16,;5.76,-22.38,;13.43,-30.02,;13.76,-31.52,)|
OC(=O)c1ccc(\C=C/c2c(noc2-c2cc[nH]c2)-c2c(Cl)cccc2C(F)(F)F)cc1 |(-2.23,-6.05,;-3.56,-5.28,;-4.9,-6.05,;-3.56,-3.74,;-2.22,-2.97,;-2.23,-1.42,;-3.56,-.65,;-3.57,.89,;-2.24,1.66,;-.9,.9,;.51,1.54,;1.54,.39,;.78,-.94,;-.73,-.62,;-.76,-2.16,;-2.02,-3.05,;-1.57,-4.52,;-.03,-4.55,;.47,-3.09,;.82,3.03,;-.33,4.05,;-1.79,3.57,;-.02,5.56,;1.45,6.05,;2.6,5.02,;2.28,3.51,;3.43,2.49,;3.12,.98,;4.9,2.97,;4.52,1.4,;-4.89,-1.42,;-4.9,-2.97,)|
OC(=O)c1ccc(NCc2c(noc2-c2cc[nH]c2)-c2c(Cl)cccc2C(F)(F)F)cc1F |(45.61,-34.71,;44.15,-34.24,;43.01,-35.27,;43.82,-32.73,;42.35,-32.26,;42.03,-30.76,;43.17,-29.73,;42.85,-28.22,;41.38,-27.75,;41.05,-26.25,;39.64,-25.63,;39.8,-24.09,;41.3,-23.77,;42.08,-25.1,;43.6,-25.25,;44.38,-26.58,;45.88,-26.26,;46.04,-24.72,;44.63,-24.1,;38.32,-26.4,;38.32,-27.95,;39.66,-28.72,;36.99,-28.72,;35.65,-27.95,;35.65,-26.4,;36.98,-25.63,;36.98,-24.09,;38.31,-23.32,;35.64,-23.33,;36.96,-22.55,;44.63,-30.19,;44.96,-31.69,;46.43,-32.15,)|
OC(=O)c1ccc(OCc2c(noc2-c2cc[nH]c2)-c2c(Cl)cccc2C(F)(F)F)cc1F |(63.42,-34.59,;61.95,-34.12,;60.81,-35.16,;61.62,-32.62,;60.15,-32.15,;59.83,-30.64,;60.97,-29.61,;60.65,-28.11,;59.18,-27.64,;58.86,-26.13,;57.45,-25.51,;57.6,-23.98,;59.11,-23.65,;59.88,-24.98,;61.4,-25.14,;62.18,-26.47,;63.68,-26.14,;63.84,-24.61,;62.43,-23.99,;56.12,-26.28,;56.13,-27.83,;57.46,-28.6,;54.79,-28.61,;53.45,-27.83,;53.46,-26.29,;54.78,-25.52,;54.78,-23.98,;56.11,-23.21,;53.44,-23.21,;54.77,-22.43,;62.43,-30.07,;62.76,-31.57,;64.23,-32.04,)|
OC(=O)c1ccc(OCc2c(noc2-c2ccc[nH]2)-c2c(Cl)cccc2C(F)(F)F)cc1 |(80.73,-36.17,;79.26,-35.7,;78.12,-36.74,;78.94,-34.2,;77.47,-33.73,;77.14,-32.22,;78.29,-31.19,;77.96,-29.69,;76.5,-29.22,;76.17,-27.71,;74.76,-27.09,;74.92,-25.56,;76.42,-25.23,;77.2,-26.56,;78.72,-26.72,;79.49,-28.05,;81,-27.72,;81.15,-26.19,;79.74,-25.57,;73.43,-27.86,;73.44,-29.41,;74.77,-30.18,;72.1,-30.18,;70.77,-29.41,;70.77,-27.87,;72.1,-27.1,;72.09,-25.56,;73.43,-24.78,;70.76,-24.79,;72.08,-24.01,;79.75,-31.65,;80.08,-33.15,)|
OC(=O)c1ccc(OCc2c(noc2-c2cn[nH]c2)-c2c(Cl)cccc2C(F)(F)F)cc1 |(13.95,-52.84,;12.48,-52.37,;11.34,-53.41,;12.15,-50.87,;10.69,-50.4,;10.36,-48.89,;11.51,-47.86,;11.18,-46.36,;9.71,-45.89,;9.39,-44.38,;7.98,-43.76,;8.13,-42.23,;9.64,-41.9,;10.41,-43.23,;11.94,-43.39,;12.71,-44.72,;14.22,-44.39,;14.37,-42.86,;12.96,-42.24,;6.65,-44.53,;6.66,-46.08,;7.99,-46.85,;5.32,-46.85,;3.99,-46.08,;3.99,-44.54,;5.32,-43.77,;5.31,-42.23,;6.64,-41.45,;3.98,-41.46,;5.3,-40.68,;12.97,-48.32,;13.3,-49.82,)|
Cn1ccc(c1)-c1onc(c1COc1ccc(cc1)C(O)=O)-c1c(Cl)cccc1C(F)(F)F |(33.85,-41.98,;32.52,-42.75,;32.37,-44.28,;30.86,-44.61,;30.09,-43.28,;31.11,-42.13,;28.57,-43.13,;27.79,-41.79,;26.29,-42.12,;26.13,-43.65,;27.54,-44.27,;27.87,-45.78,;29.33,-46.25,;29.66,-47.75,;28.51,-48.78,;28.84,-50.29,;30.31,-50.76,;31.45,-49.72,;31.12,-48.22,;30.63,-52.26,;32.1,-52.73,;29.49,-53.3,;24.8,-44.42,;24.81,-45.98,;26.14,-46.74,;23.47,-46.75,;22.14,-45.98,;22.14,-44.43,;23.47,-43.66,;23.46,-42.12,;24.8,-41.35,;22.13,-41.36,;23.45,-40.57,)|
Cc1cc(c[nH]1)-c1onc(c1COc1ccc(cc1)C(O)=O)-c1c(Cl)cccc1C(F)(F)F |(52.23,-44.54,;51.09,-43.52,;49.58,-43.84,;48.81,-42.51,;49.83,-41.36,;51.24,-41.98,;47.29,-42.36,;46.51,-41.03,;45.01,-41.35,;44.85,-42.89,;46.26,-43.51,;46.58,-45.01,;48.05,-45.48,;48.38,-46.99,;47.23,-48.02,;47.56,-49.52,;49.02,-49.99,;50.17,-48.95,;49.84,-47.45,;49.35,-51.5,;50.82,-51.97,;48.21,-52.53,;43.52,-43.66,;43.53,-45.21,;44.86,-45.98,;42.19,-45.98,;40.86,-45.21,;40.86,-43.66,;42.19,-42.89,;42.18,-41.35,;43.51,-40.58,;40.85,-40.59,;42.17,-39.81,)|
Cc1ccc(cc1)S(=O)(=O)Nc1ccc(cc1)-c1nc2ccc(C)cc2s1
Cc1ccc2nc(sc2c1)-c1ccc(NS(=O)(=O)c2ccc(cc2)C(C)(C)C)cc1
Cc1ccc2nc(sc2c1)-c1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1
Cc1ccc2nc(sc2c1)-c1ccc(NS(=O)(=O)c2ccc(OC(F)(F)F)cc2)cc1
Cc1ccc2nc(sc2c1)-c1ccc(NS(=O)(=O)c2cccc(c2)[N+]([O-])=O)cc1
Cc1ccc2nc(sc2c1)-c1ccc(NS(=O)(=O)c2ccccc2[N+]([O-])=O)cc1
Cc1ccc2nc(sc2c1)-c1ccc(NS(=O)(=O)c2cccc(c2)S(C)(=O)=O)cc1
Cc1ccc2nc(sc2c1)-c1ccc(NS(=O)(=O)c2ccc(F)cc2F)cc1
Cc1ccc2nc(sc2c1)-c1ccc(NS(=O)(=O)Cc2ccc(F)cc2)cc1
Cc1ccc2nc(sc2c1)-c1ccc(NS(=O)(=O)Cc2ccc(cc2)C(F)(F)F)cc1
Cc1ccc2nc(sc2c1)-c1ccc(NS(=O)(=O)Cc2ccc(cc2)[N+]([O-])=O)cc1
Cc1ccc2nc(sc2c1)-c1ccc(NS(=O)(=O)Cc2ccc(cc2)S(C)(=O)=O)cc1
COC(=O)c1ccc(CS(=O)(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3s2)cc1
Cc1ccc2nc(sc2c1)-c1ccc(NS(=O)(=O)Cc2ccc(cc2)C(O)=O)cc1
CCC(=O)Oc1ccc(CS(=O)(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3s2)cc1
Cc1ccc2nc(sc2c1)-c1ccc(NS(=O)(=O)Cc2cccc(c2)[N+]([O-])=O)cc1
Cc1ccc2nc(sc2c1)-c1ccc(NS(=O)(=O)Cc2ccccc2[N+]([O-])=O)cc1
COC(=O)c1cccc(CS(=O)(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3s2)c1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3s2)cc1
Cc1ccc2nc(sc2c1)-c1ccc(NC(=O)Cc2ccccc2[N+]([O-])=O)cc1
CCCn1c(nc2ccc(C)cc12)-c1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CCCCn1c(nc2ccc(C)cc12)-c1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CCCCCn1c(nc2ccc(C)cc12)-c1ccc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2C(C)C)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2CC(C)C)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2CCC(C)C)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2C2CCC2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2CC2CCC2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2CC2CCCCC2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2Cc2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2Cc2ccc(C)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2CCc2ccccc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2CCc2ccc(C)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2C(C)c2ccc(C)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2[C@H](C)c2ccc(C)cc2)cc1 |r|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2[C@@H](C)c2ccc(C)cc2)cc1 |r|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2Cc2ccc(F)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2Cc2cccc(F)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2Cc2ccccc2F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2CCc2ccc(F)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2Cc2c(F)cccc2F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2Cc2ccc(cc2)C(F)(F)F)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2Cc2ccc(cc2)S(C)(=O)=O)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2Cc2ccc(cc2)C(=O)OC)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2Cc2ccc(cc2)C(O)=O)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2Cc2ccncc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2Cc2cccnc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(C)cc3n2Cc2ccccn2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(cc3n2[C@H](C)c2ccc(C)cc2)C(F)(F)F)cc1 |r|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(OC)cc3n2[C@H](C)c2ccc(C)cc2)cc1 |r|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(cc3n2[C@H](C)c2ccc(C)cc2)C(=O)NC(C)C)cc1 |r|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3cc(C)ccc3n2[C@H](C)c2ccc(C)cc2)cc1 |r|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3cc(OC)ccc3n2[C@H](C)c2ccc(C)cc2)cc1 |r|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3cc(ccc3n2[C@H](C)c2ccc(C)cc2)C(=O)NC(C)C)cc1 |r|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(cc3n2[C@H](C)c2ccc(F)cc2)C(F)(F)F)cc1 |r|
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(cc2)-c2nc3ccc(cc3n2[C@@H](C)c2ccc(F)cc2)C(F)(F)F)cc1 |r|
[H][C@]12CCc3c(nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2C)-c1ccncc1C)-c1ccccc1 |r,t:14|
[H][C@@]12CC[C@]3(C)C(=CC(=O)C4C5CC(C)(C)CC[C@@]5(CC[C@@]34C)C(=O)OC)[C@@]1(C)C=C(C#N)C(=O)[C@@]2(C)O |r,c:6,t:33|
CCS(=O)(=O)c1ccc(CNc2nc3c(C)nc(nc3n([C@@H](C)C3CC3)c2=O)-c2c(C)ncnc2C2CC2)nc1 |r|
[H][C@@]12CC[C@@](c3nnc(cc13)-c1c(F)cccc1F)(c1ccnc(n1)N1CCCCC1)C2(C)C |r|
[H][C@@]12CC[C@@](c3nnc(cc13)-c1c(F)cccc1F)(c1ccncn1)C2(C)C |r|
CC(C)CN(c1ccc(C)cc1C)S(=O)(=O)c1ccc2n(CC3CCOCC3)c(=O)[nH]c2c1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(Cl)c(c(Cl)c2)C2(CC2)c2noc(n2)-c2ccc(F)cc2)cc1
C[C@H]1CN(Cc2cc(F)cc(NC(=O)c3cnc(C)nc3)c2C)CCN1C(=O)C1CCCC1 |r|
[H][C@]12CCCc3c(nc(nc3[C@]1(C)C=C(C#N)C(=O)[C@@H]2C)-c1ccncc1C)-c1ccccc1 |r,t:15|
CCn1c(nc2cc(NC(=O)Cc3ccc(cc3)S(=O)(=O)CC)ccc12)C(C)(C)Oc1ccc(F)cc1F
C[C@H]1CN(Cc2cncc(NS(=O)(=O)c3c(Cl)cc(Cl)cc3Cl)c2)CCN1C(=O)C1CCCC1 |r|
COc1c(NC(=O)c2cccc(c2)C#N)cnc2n(C)cc(C3CCN(CC3)C(=O)C3CCCC3)c12
COc1ccc2[C@@H](N(CCc2n1)C(=O)[C@@H]1C[C@H](CC(O)=O)C1)C(=O)Nc1cc2CCC(C)(C)c2c(F)c1 |r,wU:6.24,14.15,16.18,(64.98,-30.47,;63.66,-31.25,;63.67,-32.79,;62.34,-33.58,;62.36,-35.12,;63.7,-35.87,;63.7,-37.41,;65.03,-38.17,;66.35,-37.41,;66.35,-35.87,;65.03,-35.09,;65.01,-33.55,;65.03,-39.71,;63.69,-40.48,;66.36,-40.48,;66.75,-41.97,;68.24,-41.57,;69.58,-42.34,;70.91,-41.57,;72.24,-42.34,;70.91,-40.03,;67.84,-40.08,;62.36,-38.18,;62.36,-39.72,;61.03,-37.41,;59.7,-38.18,;59.7,-39.72,;58.38,-40.49,;58.07,-42,;56.53,-42.18,;55.89,-40.77,;54.55,-41.53,;54.56,-39.99,;57.03,-39.73,;57.03,-38.18,;55.7,-37.41,;58.36,-37.41,)|
c1cc(c(c(c1)Cl)C(=O)n2c3cccnc3c(n2)c4cc(c(cc4F)C(=O)O)O)C(F)(F)F
OC(=O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C3(CC3)C(F)(F)F)c3cccnc23)c(F)c1
Cc1noc(C)c1[C@H](O)c1cc2cc(CC(=O)N[C@H](c3ccccc3)c3ccc(C)cc3C)ccc2o1 |r|
COc1cc2C(=O)C(Cc3cccc(c3)C(F)(F)F)Cc2cc1N1CCOCC1
COc1nc2ccc(cc2c(Cl)c1Cc1ccc(cc1)C(F)(F)F)[C@@](O)(c1cnnn1C)c1ccc(C)nc1C |r|
OC(c1ccc(NC(=O)c2ccccc2Cl)cc1)(C(F)(F)F)C(F)(F)F
COc1ccccc1COc1ccc(NC(=O)[C@@H]2N(CCc3nc(ON)ccc23)C(C)=O)cc1 |r|
Fc1ccccc1C(=O)Nc1sc2CCCCc2c1C(=O)N1CCN(Cc2ccccc2)CC1
CSc1ncc(Cl)c(n1)C(=O)Nc1sc2CCCCc2c1C(=O)NCc1ccccc1
CSc1ncc(Cl)c(n1)C(=O)Nc1sc2CC(C)CCc2c1C(=O)NC1CCS(=O)(=O)C1
CCC1CCc2c(C1)sc(NC(=O)c1ccnn1C)c2C(=O)Nc1ccccc1C
CN1CCN(CC1)C(=O)c1c(NC(=O)c2ccccc2F)sc2CC(CCc12)C(C)(C)C
CC1CCc2c(C1)sc(NC(=O)c1ccccc1F)c2C(=O)N1CCN(C)CC1
FC(F)(F)C(=O)Nc1sc2CCCCc2c1C(=O)NCc1ccccc1
Cc1ccnc(SCC(=O)Nc2sc3CCCCc3c2C(=O)NCc2ccccc2)n1
O=C(CN1CCCCC1)Nc1sc2CCCCc2c1C(=O)NCc1ccccc1
CN1CCN(CC(=O)Nc2sc3CCCCc3c2C(=O)NCc2ccccc2)CC1
CC1CCN(CC(=O)Nc2sc3CCCCc3c2C(=O)NCc2ccccc2)CC1
CC1CCCN1C(=O)c1c(NC(=O)c2cccnc2)sc2CCCCc12
C[C@@H]1CCN([C@H](C)C1)C(=O)c1c(NC(=O)c2cccnc2)sc2CCCCc12 |r|
O[C@H]1CC[C@@H](CC1)NC(=O)c1c(NC(=O)c2cccnc2)sc2CCCCc12 |r,wU:1.0,wD:4.7,(-1.98,-5.78,;-1.51,-4.31,;-2.55,-3.18,;-2.08,-1.71,;-.58,-1.38,;.46,-2.52,;-.01,-3.99,;-.11,.09,;1.39,.42,;2.43,-.72,;1.86,1.88,;.95,3.12,;-.59,3.12,;-1.37,4.44,;-.61,5.78,;-2.91,4.44,;-3.69,5.76,;-5.23,5.76,;-5.99,4.42,;-5.21,3.09,;-3.67,3.09,;1.85,4.37,;3.31,3.91,;4.64,4.69,;5.99,3.92,;5.99,2.38,;4.66,1.61,;3.31,2.37,)|
CCC1CCN(C1)C(=O)c1c(NC(=O)c2cccnc2)sc2CCCCc12
Cn1ccnc1SCC(=O)Nc1sc2CCCCc2c1C(=O)NCc1ccccc1
OCC1CCN(C1)C(=O)c1c(NC(=O)c2cccnc2)sc2CCCCc12
CC1(C)CCc2c(C1)sc(NC(=O)c1cnccn1)c2C(=O)N1CCOCC1
Cn1cnc(CNC(=O)c2c(NC(=O)c3cccnc3)sc3CCCCc23)n1
C[C@H](NC(=O)c1c(NC(=O)c2cccnc2)sc2CCCCc12)C#N |r|
O=C(NCC1CCNCC1)c1c(NC(=O)c2cccnc2)sc2CCCCc12
O=C(Nc1sc2CCCCc2c1C(=O)c1ccccc1)c1cnccn1
Cc1cnc(nc1C(=O)Nc1sc2CCCCc2c1C(=O)c1ccccc1)S(C)(=O)=O
CCn1c2ccc(cc2c2cccc(OC(C)C)c12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCn1c2ccc(OC3COC3)cc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCn1c2ccc(CC3COC3)cc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCn1c2ccc(cc2c3c1ccc(c3)OC(C)C)C(=O)NCc4ccc(cc4)S(=O)(=O)CC
CCn1c2ccc(cc2c2c(OC(C)C)cccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCn1c2ccc(cc2c2ccc(OC(C)C)cc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCn1c2ccc(cc2c3c1ccc(c3)OC4CCC4)C(=O)NCc5ccc(cc5)S(=O)(=O)CC
CCn1c2ccc(OCC(C)C)cc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCn1c2ccc(OC(C)C(F)(F)F)cc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCn1c2ccc(CC(C)C)cc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCn1c2ccc(CC(C)(C)F)cc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCn1c2ccc(CN(C)C)cc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCn1c2ccc(CC3CCC3)cc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCn1c2ccc(OC3CC3)cc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCn1c2ccc(CC3CC3)cc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
CCn1c2ccc(OC(C)C)cc2c2cc(ccc12)C(=O)NC(CO)c1ccc(cc1)S(=O)(=O)CC
CCn1c2ccc(OC(C)C)cc2c2cc(ccc12)C(=O)NCc1ccc(cn1)S(=O)(=O)CC
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CCF)c4ccc(OC(C)C)cc4c3c2)cc1
CCn1c2ccc(OC(C)C)cc2c2cc(ccc12)C(=O)NCc1ccc(cn1)S(C)(=O)=O
CCn1c2ccc(OC(C)C)cc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(C)(=O)=O
CCn1c2ccc(CC3CC3)cc2c2cc(ccc12)C(=O)NC(COC)c1ccc(cc1)S(=O)(=O)CC
CCS(=O)(=O)c1ccc(CNC(=O)c2ccc3n(CCF)c4ccc(CC5CC5)cc4c3c2)cc1
CCn1c2ccc(CC3CC3)cc2c2cc(ccc12)C(=O)NC(CO)c1ccc(cc1)S(=O)(=O)CC
CCn1c2ccc(CC3CC3)cc2c2cc(ccc12)C(=O)NCc1ccc(cn1)S(=O)(=O)CC
CCn1c2ccc(CC3CC3)cc2c2cc(ccc12)C(=O)NCc1ccc(cn1)S(C)(=O)=O
CCn1c2ccc(CC3CC3)cc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(C)(=O)=O
CCS(=O)(=O)c1ccc(cc1)C(COC)NC(=O)c1ccc2n(CCF)c3ccc(CC4CC4)cc3c2c1
CCn1c2ccc(CC3CC3)cc2c2cc(ccc12)C(=O)N[C@H](COC)c1ccc(cc1)S(=O)(=O)CC |r|
CCn1c2ccc(CC3CC3)cc2c2cc(ccc12)C(=O)N[C@@H](COC)c1ccc(cc1)S(=O)(=O)CC |r|
CCn1c2ccc(CC(C)C(F)(F)F)cc2c2cc(ccc12)C(=O)NCc1ccc(cc1)S(=O)(=O)CC
OC(=O)c1ccc(Nc2nc(Oc3ccccc3C(F)(F)F)nc(n2)-c2ccccc2)cc1
OC(=O)c1ccc(Nc2nc(Cc3c(Cl)cccc3C(F)(F)F)nc(n2)-c2ccccc2)cc1
OC(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3Cl)nc(n2)-c2ccccc2)cc1
OC(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3Cl)nc(n2)C2CCCCC2)cc1
OC(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3Cl)nc(n2)N2CCCCC2)cc1
OC(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3Cl)nc(n2)C2CCOCC2)cc1
OC(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3Cl)nc(n2)C2CCCC2)cc1
Cc1ccccc1-c1nc(Nc2ccc(cc2)C(O)=O)nc(Oc2c(Cl)cccc2Cl)n1
Cc1cccc(c1)-c1nc(Nc2ccc(cc2)C(O)=O)nc(Oc2c(Cl)cccc2Cl)n1
Cc1ccc(cc1)-c1nc(Nc2ccc(cc2)C(O)=O)nc(Oc2c(Cl)cccc2Cl)n1
COc1ccc(cc1)-c1nc(Nc2ccc(cc2)C(O)=O)nc(Oc2c(Cl)cccc2Cl)n1
CCc1ccc(cc1)-c1nc(Nc2ccc(cc2)C(O)=O)nc(Oc2c(Cl)cccc2Cl)n1
CC(C)c1ccc(cc1)-c1nc(Nc2ccc(cc2)C(O)=O)nc(Oc2c(Cl)cccc2Cl)n1
OC(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3Cl)nc(n2)-c2ccc(cc2)C2CC2)cc1
CC(C)(C)c1ccc(cc1)-c1nc(Nc2ccc(cc2)C(O)=O)nc(Oc2c(Cl)cccc2Cl)n1
CC(C)Cc1ccc(cc1)-c1nc(Nc2ccc(cc2)C(O)=O)nc(Oc2c(Cl)cccc2Cl)n1
OC(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3Cl)nc(n2)-c2ccc(F)cc2)cc1
OC(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3Cl)nc(n2)-c2ccc(Cl)cc2)cc1
OC(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3Cl)nc(n2)-c2ccc(cc2)C(F)(F)F)cc1
COc1ccc(cc1)-c1nc(Nc2cccc(c2)C(O)=O)nc(Oc2c(Cl)cccc2Cl)n1
COc1ccc(cc1)-c1nc(Nc2ccc(cc2OC)C(O)=O)nc(Oc2c(Cl)cccc2Cl)n1
COc1ccc(cc1)-c1nc(Nc2ccc(C(O)=O)c(OC)c2)nc(Oc2c(Cl)cccc2Cl)n1
COc1ccc(cc1)-c1nc(Nc2ccc(C(O)=O)c(O)c2)nc(Oc2c(Cl)cccc2Cl)n1
COc1ccc(cc1)-c1nc(Nc2ccc(C(O)=O)c(F)c2)nc(Oc2c(Cl)cccc2Cl)n1
COc1ccc(cc1)-c1nc(Nc2ccc(C(O)=O)c(Cl)c2)nc(Oc2c(Cl)cccc2Cl)n1
COc1ccc(cc1)-c1nc(Nc2ccc(C(O)=O)c(c2)C(O)=O)nc(Oc2c(Cl)cccc2Cl)n1
COc1ccc(cc1)-c1nc(Nc2ccc(nc2)C(O)=O)nc(Oc2c(Cl)cccc2Cl)n1
COc1ccc(cc1)-c1nc(N[C@H]2CC[C@H](CC2)C(O)=O)nc(Oc2c(Cl)cccc2Cl)n1 |r,wU:12.12,15.19,(-8.66,4.24,;-7.33,5.01,;-6,4.24,;-4.67,5.01,;-3.33,4.24,;-3.33,2.7,;-4.67,1.93,;-6,2.7,;-2,1.93,;-.66,2.7,;.66,1.93,;2,2.7,;3.33,1.93,;4.67,2.7,;6,1.93,;6,.39,;4.67,-.38,;3.33,.38,;7.33,-.38,;7.33,-1.92,;8.66,.39,;.66,.39,;-.66,-.38,;-.66,-1.92,;.67,-2.69,;.67,-4.24,;-.66,-5.01,;2.01,-5,;3.34,-4.23,;3.34,-2.69,;2.01,-1.92,;2.01,-.38,;-2,.38,)|
COc1ccc(cc1)-c1nc(N[C@H]2CC[C@@H](CC2)C(O)=O)nc(Oc2c(Cl)cccc2Cl)n1 |r,wU:15.19,wD:12.12,(-8.66,4.24,;-7.33,5.01,;-6,4.24,;-4.67,5.01,;-3.33,4.24,;-3.33,2.7,;-4.67,1.93,;-6,2.7,;-2,1.93,;-.66,2.7,;.66,1.93,;2,2.7,;3.33,1.93,;3.33,.38,;4.67,-.38,;6,.39,;6,1.93,;4.67,2.7,;7.33,-.38,;7.33,-1.92,;8.66,.39,;.66,.39,;-.66,-.38,;-.66,-1.92,;.67,-2.69,;.67,-4.24,;-.66,-5.01,;2.01,-5,;3.34,-4.23,;3.34,-2.69,;2.01,-1.92,;2.01,-.38,;-2,.38,)|
COc1ccc(cc1)-c1nc(NC2CCC(C2)C(O)=O)nc(Oc2c(Cl)cccc2Cl)n1
COC(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3Cl)nc(n2)-c2ccc(OC)cc2)cc1
COc1ccc(cc1)-c1nc(Nc2ccc(CC(O)=O)cc2)nc(Oc2c(Cl)cccc2Cl)n1
COc1ccc(cc1)-c1nc(Nc2ccc(cc2)C(C)C(O)=O)nc(Oc2c(Cl)cccc2Cl)n1
COc1ccc(cc1)-c1nc(Nc2ccc(cc2)C(N)=O)nc(Oc2c(Cl)cccc2Cl)n1
CNC(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3Cl)nc(n2)-c2ccc(OC)cc2)cc1
COc1ccc(cc1)-c1nc(Nc2ccc(cc2)C(=O)NC(C)C)nc(Oc2c(Cl)cccc2Cl)n1
COc1ccc(cc1)-c1nc(Nc2ccc(CC(N)=O)cc2)nc(Oc2c(Cl)cccc2Cl)n1
COc1ccc(cc1)-c1nc(Nc2ccc(NC(C)=O)cc2)nc(Oc2c(Cl)cccc2Cl)n1
COc1ccc(cc1)-c1nc(Nc2ccc(cc2)S(N)(=O)=O)nc(Oc2c(Cl)cccc2Cl)n1
CNS(=O)(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3Cl)nc(n2)-c2ccc(OC)cc2)cc1
COc1ccc(cc1)-c1nc(Nc2ccc(NS(C)(=O)=O)cc2)nc(Oc2c(Cl)cccc2Cl)n1
COc1ccc(cc1)-c1nc(Nc2ccc(cc2)S(C)(=O)=O)nc(Oc2c(Cl)cccc2Cl)n1
CC(=O)Nc1ccc(Nc2nc(Oc3c(Cl)cccc3Cl)nc(n2)-c2ccc(cc2)C(F)(F)F)cc1
COc1ccc(cc1)-c1nc(Nc2ccc(NC(C)=O)cc2)nc(Oc2c(Cl)cccc2C(F)(F)F)n1
CC(=O)Nc1ccc(Nc2nc(Oc3c(Cl)cccc3C(F)(F)F)nc(n2)-c2ccc(cc2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3Cl)nc(n2)-c2ccc(cc2)C(F)(F)F)cc1
CNC(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3C(F)(F)F)nc(n2)-c2ccc(OC)cc2)cc1
CNC(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3C(F)(F)F)nc(n2)-c2ccc(cc2)C(F)(F)F)cc1
CS(=O)(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3Cl)nc(n2)-c2ccc(cc2)C(F)(F)F)cc1
COc1ccc(cc1)-c1nc(Nc2ccc(cc2)S(C)(=O)=O)nc(Oc2c(Cl)cccc2C(F)(F)F)n1
CS(=O)(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3C(F)(F)F)nc(n2)-c2ccc(cc2)C(F)(F)F)cc1
NC(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3Cl)nc(n2)-c2ccc(cc2)C(F)(F)F)cc1
COc1ccc(cc1)-c1nc(Nc2ccc(cc2)C(N)=O)nc(Oc2c(Cl)cccc2C(F)(F)F)n1
NC(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3C(F)(F)F)nc(n2)-c2ccc(cc2)C(F)(F)F)cc1
COc1ccc(cc1)-c1nc(Nc2ccc(cc2)C(O)=O)nc(Oc2c(Cl)cccc2C(F)(F)F)n1
OC(=O)c1ccc(Nc2nc(Oc3c(Cl)cccc3C(F)(F)F)nc(n2)-c2ccc(cc2)C(F)(F)F)cc1
CCc1ccc(cc1C#N)-c1c(Cl)cc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1Cl
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccc(CC(C)C)c(c2)C#N)cc1
CCS(=O)(=O)c1ccc(CNC(=O)c2cc(Cl)c(c(Cl)c2)-c2ccc(CC(C)C)c(c2)C#N)cc1
CCS(=O)(=O)c1ccc(CNC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccc(CC(C)C)c(c2)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccc(CC(C)C)cc2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccc(CC(C)C)c(F)c2)cc1
[#6]-[#6]S(=O)(=O)c1ccc(-[#6]-[#6](=O)-[#7]-c2cc(Cl)c(c(Cl)c2)-c2ccc(\[#6]=[#6](\[#6])-[#6])c(c2)C#N)cc1
CCC(C)Cc1ccc(cc1C#N)-c1c(Cl)cc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1Cl
CC\C(C)=C\c1ccc(cc1C#N)-c1c(Cl)cc(NC(=O)Cc2ccc(cc2)S(=O)(=O)CC)cc1Cl
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccc(CC3CCC3)c(c2)C#N)cc1
[#6]-[#6]S(=O)(=O)c1ccc(-[#6]-[#6](=O)-[#7]-c2cc(Cl)c(c(Cl)c2)-c2ccc(\[#6]=[#6]-3/[#6]-[#6]-[#6]-3)c(c2)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccc(CC3CCCC3)c(c2)C#N)cc1
[#6]-[#6]S(=O)(=O)c1ccc(-[#6]-[#6](=O)-[#7]-c2cc(Cl)c(c(Cl)c2)-c2ccc(\[#6]=[#6]-3/[#6]-[#6]-[#6]-[#6]-3)c(c2)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccc(OC(C)C)c(c2)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccc(CN(C)C)c(c2)C#N)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2cc(Cl)c(c(Cl)c2)-c2ccc(CC(C)C)c(c2)C#N)nc1
CCS(=O)(=O)c1ccc(CNC(=O)c2cnc3c(c2)CN(C[C@H]2CC[C@H](C(F)(F)F)CC2)[C@H]3C(C)C)nc1
O=C(O)c1ccc(-c2nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c3cc(C(=O)NCCOCCOCCNC(=S)Nc4ccc5c(c4)C(=O)OC54c5ccc(O)cc5Oc5cc(O)ccc54)ccc23)cc1
O=C(O)c1ccc(-c2nn(C(=O)c3ccccc3C(F)(F)F)c3ccccc23)cc1
O=C(O)c1ccc(-c2nn(C(=O)c3ccccc3)c3ccccc23)cc1
Cc1ccc(NCc2cn(-c3ccc(C(=O)O)s3)c3ccccc23)cc1C
COc1cccc(-c2cc(C(F)(F)F)c3c(C)nn(-c4ccc(C(=O)O)cc4)c3n2)c1
Cc1cccc(c1)-c1nc(Nc2ccc(cc2)C(O)=O)c2ccccc2n1
O=C(O)c1ccc(-n2cc(CNc3ccccc3)c3ccccc32)s1
O=C(O)c1ccc(-n2cc(CNc3ccccc3)c3ccccc32)o1
O=C(O)c1ccc(-n2cc(CNc3ccccc3)c3ccccc32)cc1
O=C(O)c1cccc(-n2cc(CNc3ccccc3)c3ccccc32)c1
CC(Nc1ccccc1)c1cn(-c2ccc(C(=O)O)s2)c2ccccc12
O=C(O)c1ccc(-n2cc(CNc3ccccc3Cl)c3ccccc32)s1
O=C(O)c1ccc(-n2cc(C(=O)c3ccccc3)c3ccccc32)s1
Cc1ccccc1C(=O)c1cn(-c2ccc(C(=O)O)s2)c2ccccc12
Cc1cccc(C(=O)c2cn(-c3ccc(C(=O)O)s3)c3ccccc23)c1
Cc1ccc(C(=O)c2cn(-c3ccc(C(=O)O)s3)c3ccccc23)cc1
O=C(O)c1ccc(-n2cc(C(=O)c3c(Cl)cccc3C(F)(F)F)c3ccccc32)s1
O=C(O)c1ccc(-n2cc(C(=O)c3ccccc3Cl)c3ccccc32)s1
O=C(O)c1ccc(-n2cc(C(=O)c3cccc(Cl)c3)c3ccccc32)s1
O=C(O)c1ccc(-n2cc(C(=O)c3ccc(Cl)cc3)c3ccccc32)s1
O=C(O)c1ccc(-n2cc(C(=O)c3c(Cl)cccc3Cl)c3ccccc32)s1
Cc1cccc(Cl)c1C(=O)c1cn(-c2ccc(C(=O)O)s2)c2ccccc12
Cc1cc(-n2cc(C(=O)c3c(Cl)cccc3Cl)c3ccccc32)sc1C(=O)O
Cc1csc(-n2cc(C(=O)c3c(Cl)cccc3Cl)c3ccccc32)c1
Cc1ccc(NC(=O)CC(c2nnc([C@H]3C[C@@H](CC(C)C)C3)n2C2CC2)C2CNC2)c(C)c1
Cc1ccc(NC(=O)CC(c2nnc([C@H]3C[C@@H](CC(C)C)C3)n2C2CC2)C2CN(C)C2)c(C)c1
Cc1ccc(NC(=O)C[C@H](c2nnc([C@H]3C[C@@H](CC(C)C)C3)n2C2CC2)[C@H]2C[C@@H](O)C2)c(C)c1
Cc1ccc(NC(=O)C[C@H](CC(C)(C)O)c2nnc([C@H]3C[C@@H](CC(C)C)C3)n2C2CC2)c(C)c1
Cc1ccc(NC(=O)CC(CC(=O)O)c2nnc([C@H]3C[C@@H](CC(C)C)C3)n2C2CC2)c(C)c1
Cc1ccc(NC(=O)CC(CC(=O)N(C)C)c2nnc([C@H]3C[C@@H](CC(C)C)C3)n2C2CC2)c(C)c1
Cc1ccc(NC(=O)CC(Cc2nnn[nH]2)c2nnc([C@H]3C[C@@H](CC(C)C)C3)n2C2CC2)c(C)c1
Cc1ccc(NC(=O)CC(Cc2ncco2)c2nnc([C@H]3C[C@@H](CC(C)C)C3)n2C2CC2)c(C)c1
Cc1ccc(NC(=O)C[C@H](Cc2nccs2)c2nnc([C@H]3C[C@@H](CC(C)C)C3)n2C2CC2)c(C)c1
Cc1ccc(NC(=O)C[C@H](CC(=O)O)c2noc([C@H]3C[C@@H](CC(C)C)C3)c2C2CC2)c(C)c1
Cc1ccc(NC(=O)C[C@H](CC(=O)O)c2noc([C@H]3C[C@@H](CC(C)(C)C)C3)c2C2CC2)c(C)c1
Cc1ccc(NC(=O)C[C@H](CC(=O)O)c2noc([C@H]3C[C@@H](CCC(C)C)C3)c2C2CC2)c(C)c1
CCC(C)(C)C[C@H]1C[C@@H](c2onc([C@@H](CC(=O)O)CC(=O)Nc3ccc(C)cc3C)c2C2CC2)C1
Cc1ccc(NC(=O)C[C@H](CC(=O)O)c2noc([C@H]3C[C@@H](CCC(C)(C)C)C3)c2C2CC2)c(C)c1
Cc1ccc(NC(=O)C[C@H](CC(=O)O)c2noc([C@H]3C[C@@H](C(C)(C)C(C)C)C3)c2C2CC2)c(C)c1
CCC(CC)C[C@H]1C[C@@H](c2onc([C@@H](CC(=O)O)CC(=O)Nc3ccc(C)cc3C)c2C2CC2)C1
CCc1c([C@@H](CC(=O)O)CC(=O)Nc2ccc(C)cc2C)noc1[C@H]1C[C@@H](CC(C)C)C1
Cc1ccc(NC(=O)C[C@H](CC(=O)O)c2noc([C@H]3C[C@@H](CC(C)C)C3)c2C(C)C)c(C)c1
C=C(C)c1c([C@@H](CC(=O)O)CC(=O)Nc2ccc(C)cc2C)noc1[C@H]1C[C@@H](CC(C)C)C1
Cc1ccc(NC(=O)C[C@H](CCC(=O)O)c2noc([C@H]3C[C@@H](CC(C)C)C3)c2C2CC2)c(C)c1
Cc1ccc(NC(=O)C[C@@H](c2noc([C@H]3C[C@@H](CC(C)C)C3)c2C2CC2)C(C)(C)C(=O)O)c(C)c1
Cc1ccc(NC(=O)C[C@@H](c2noc([C@H]3C[C@@H](CC(C)C)C3)c2C2CC2)C(C)(C)CC(=O)O)c(C)c1
Cc1ccc(NC(=O)C[C@H](OCC(=O)O)c2noc([C@H]3C[C@@H](CC(C)C)C3)c2C2CC2)c(C)c1
Cc1ccc(NC(=O)C[C@H](Cc2ccc(C(=O)O)cc2)c2noc([C@H]3C[C@@H](CC(C)C)C3)c2C2CC2)c(C)c1
Cc1ccc(NC(=O)C[C@H](Cc2nc(C(=O)O)cs2)c2noc([C@H]3C[C@@H](CC(C)C)C3)c2C2CC2)c(C)c1
Cc1ccc(NC(=O)C[C@H](C[C@H]2C[C@@H](C(=O)O)C2)c2noc([C@H]3C[C@@H](CC(C)C)C3)c2C2CC2)c(C)c1
Cc1ccc(NC(=O)C[C@H](Cc2nnn[nH]2)c2noc([C@H]3C[C@@H](CC(C)C)C3)c2C2CC2)c(C)c1
Cc1cccc(NC(=O)C[C@H](CC(=O)O)c2noc([C@H]3C[C@@H](CC(C)C)C3)c2C2CC2)c1C
Cc1ccc(C)c(NC(=O)C[C@H](CC(=O)O)c2noc([C@H]3C[C@@H](CC(C)C)C3)c2C2CC2)c1
Cc1cccc(C)c1NC(=O)C[C@H](CC(=O)O)c1noc([C@H]2C[C@@H](CC(C)C)C2)c1C1CC1
Cc1cc(C)cc(NC(=O)C[C@H](CC(=O)O)c2noc([C@H]3C[C@@H](CC(C)C)C3)c2C2CC2)c1
Cc1ccc(NC(=O)C[C@H](CC(=O)O)c2noc([C@H]3C[C@@H](CC(C)C)C3)c2C2CC2)cc1C
Cc1cc(C)c(NC(=O)C[C@H](CC(=O)O)c2noc([C@H]3C[C@@H](CC(C)C)C3)c2C2CC2)cc1C
Cc1ccc(NC(=O)C[C@H](CC(=O)O)c2noc([C@H]3C[C@@H](CC(C)C)C3)c2C2CC2)c(C)c1C
Cc1cc(C)c(C)c(NC(=O)C[C@H](CC(=O)O)c2noc([C@H]3C[C@@H](CC(C)C)C3)c2C2CC2)c1
Cc1ccc(NC(=O)C[C@H](CC(=O)O)c2noc([C@H]3C[C@@H](CC(C)C)C3)c2C2CC2)c(F)c1
Cc1cc(F)ccc1NC(=O)C[C@H](CC(=O)O)c1noc([C@H]2C[C@@H](CC(C)C)C2)c1C1CC1
CC(C)C[C@H]1C[C@@H](c2onc([C@@H](CC(=O)O)CC(=O)Nc3ccc(Cl)cc3F)c2C2CC2)C1
CC(C)C[C@H]1C[C@@H](c2onc([C@@H](CC(=O)O)CC(=O)Nc3ccc(F)cc3Cl)c2C2CC2)C1
Cc1ccc(NC(=O)C[C@H](CCC(=O)O)c2nnn([C@H]3C[C@@H](CC(C)(C)C)C3)c2C2CC2)c(Cl)c1
Cc1ccc(NC(=O)C[C@H](CCC(=O)O)n2nnc([C@H]3C[C@@H](CC(C)(C)C)C3)c2C2CC2)c(Cl)c1
Cc1ccc(NC(=O)C[C@H](CCC(=O)O)n2ncc([C@H]3C[C@@H](CC(C)(C)C)C3)c2C2CC2)c(Cl)c1
Cc1ccc(NC(=O)CC(CCC(=O)O)c2ncnc([C@H]3C[C@@H](CC(C)(C)C)C3)c2C2CC2)c(Cl)c1
Cc1ccc(NC(=O)C[C@H](CCC(=O)O)C(=O)N(C[C@H]2C[C@@H](CC(C)(C)C)C2)C2CC2)c(Cl)c1
CCC(=O)Nc1ccccc1-c1ccc(NC(=O)Cc2ccc(S(=O)(=O)CC)cc2)cc1C
C=CC(=O)Nc1ccccc1-c1ccc(NC(=O)Cc2ccc(S(=O)(=O)CC)cc2)cc1C
C=C(C)C(=O)Nc1ccccc1-c1ccc(NC(=O)Cc2ccc(S(=O)(=O)CC)cc2)cc1C
C/C=C/C(=O)Nc1ccccc1-c1ccc(NC(=O)Cc2ccc(S(=O)(=O)CC)cc2)cc1C
C=C(F)C(=O)Nc1ccccc1-c1ccc(NC(=O)Cc2ccc(S(=O)(=O)CC)cc2)cc1C
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(-c3ccccc3NC(=O)/C=C/COC)c(C)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(-c3ccccc3NC(=O)CCl)c(C)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(-c3ccccc3NC(=O)CC#N)c(C)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(-c3ccccc3NC(=O)C(C)(C)C#N)c(C)c2)cc1
CCS(=O)(=O)c1ccc(CC(=O)Nc2ccc(-c3ccccc3NC(=O)C3(C#N)CC3)c(C)c2)cc1
C=CC(=O)Nc1ccccc1-c1ccc(NC(=O)Cc2ccc(S(C)(=O)=O)cc2)cc1C
C=CC(=O)Nc1ccccc1-c1ccc(NC(=O)Cc2ccc(C#N)cc2)cc1C
C=CC(=O)Nc1ccccc1-c1ccc(NC(=O)Cc2cccc(C#N)c2)cc1C
C=CC(=O)Nc1ccccc1-c1ccc(NC(=O)Cc2ccccc2[N+](=O)[O-])cc1C
C=CC(=O)Nc1ccccc1-c1ccc(NC(=O)c2ccc(S(C)(=O)=O)cc2)cc1C
C=CC(=O)Nc1ccccc1-c1ccc(NC(=O)c2ccc(S(C)(=O)=O)cn2)cc1C
C=CC(=O)Nc1ccccc1-c1ccc(NC(=O)c2ccc(OC)nc2)cc1C
C=CC(=O)Nc1ccccc1-c1ccc(NC(=O)c2cnc(C)nc2)cc1C
C=CC(=O)Nc1ccccc1-c1ccc(NC(=O)c2cccc(C#N)c2)cc1C
C=CC(=O)Nc1ccccc1-c1ccc(NS(=O)(=O)Cc2ccc([N+](=O)[O-])cc2)cc1C
C=CC(=O)Nc1ccccc1-c1ccc(NC(=O)Cc2ccc(S(=O)(=O)CC)cc2)cc1C(F)(F)F
C=CC(=O)Nc1ccccc1-c1ccc(NC(=O)Cc2ccc(S(=O)(=O)CC)cc2)cc1F
C=CC(=O)Nc1ccccc1-c1ccc(NC(=O)Cc2ccc(S(=O)(=O)CC)cc2)cc1Cl
C=CC(=O)Nc1ccccc1-c1c(Cl)cc(NC(=O)Cc2ccc(S(=O)(=O)CC)cc2)cc1Cl
C=CC(=O)Nc1ccccc1-c1ccc(NC(=O)Cc2ccc(S(=O)(=O)CC)cc2)cc1
C=CC(=O)Nc1ccccc1-c1ccc(NC(=O)Cc2ccc(S(=O)(=O)CC)cc2)cn1
CC(=C)[C@@H]1CC[C@]2([C@H]1[C@H]3CC[C@@H]4[C@]5(CC[C@@H](C([C@@H]5CC[C@]4([C@@]3(CC2)C)C)(C)C)O)C)C(=O)O
C=C(C)[C@@H]1CC[C@]2(C(=O)Nc3nccs3)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)N[C@@H]3CCN(C)C3)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)N[C@H]3CCN(C)C3)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)NC3CCNCC3)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)N[C@@H]3CCCN(C)C3)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)N[C@H]3CCCN(C)C3)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)NC3CCCN(C)CC3)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)N[C@@H]3CN4CCC3CC4)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)NCc3cncs3)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)NCc3cc[nH]n3)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)NC[C@@H]3CCN(C)C3)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)NC[C@H]3CCN(C)C3)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)NC[C@@H]3CCCN3C)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)NC[C@H]3CCCN3C)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)NCCN3CCCC3)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)NCCN3CCC(O)C3)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)NCCNc3ccncc3)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)NCCN(CC)CC)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)NCCCN(C)C)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)NCCN(C)CCN(C)C)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)NCC(C)(C)CN(C)C)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)NCCN(CC)CCO)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C(C)[C@@H]1CC[C@]2(C(=O)NCCOCCN(C)C)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
CN(C)CCCNC(=O)[C@]12CC[C@@H](C3(C)CC3)[C@@H]1[C@H]1CC[C@@H]3[C@@]4(C)CC[C@H](O)C(C)(C)[C@@H]4CC[C@@]3(C)[C@]1(C)CC2
C=C(C)[C@@H]1CC[C@]2(C(=O)NCCCN(C)C)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)C[C@H](O)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
C=C1C[C@]2(C)[C@H]3CC[C@@H]4[C@H]5[C@H](C(=C)C)CC[C@]5(C(=O)NCCCN(C)C)CC[C@@]4(C)[C@]3(C)CC[C@H]2C(C)(C)C1=O
C=C(C)[C@@H]1CC[C@]2(C(=O)NCCCN(C)C)CC[C@]3(C)[C@H](CC[C@@H]4[C@@]5(C)CC[C@H](N)C(C)(C)[C@@H]5CC[C@]43C)[C@@H]12
Cc1cc2c(s1)c(-c1ccc(C(=O)O)cc1)nn2C(=O)c1c(Cl)cccc1C(F)(F)F
Cc1cc2c(s1)c(-c1ccc(C(=O)O)cc1)nn2C(=O)c1c(C)cccc1Cl
Cc1cc2c(s1)c(-c1ccc(C(=O)O)cc1)nn2C(=O)c1c(Cl)cccc1Br
Cc1cc2c(s1)c(-c1ccc(C(=O)O)cc1F)nn2C(=O)c1c(Cl)cccc1C(F)(F)F
Cc1cc2c(s1)c(-c1ccc(C(=O)O)cc1F)nn2C(=O)c1c(Cl)cccc1Cl
Cc1cc2c(s1)c(-c1ccc(C(=O)O)cc1F)nn2C(=O)c1c(F)cccc1C(F)(F)F
Cc1cc2c(s1)c(-c1ccc(C(=O)O)c(F)c1)nn2C(=O)c1c(F)cccc1C(F)(F)F
CN(C)C(=O)c1cc2c(s1)c(-c1ccc(C(=O)O)cc1F)nn2C(=O)c1c(F)cccc1C(F)(F)F
C[C@H](CCC(=O)NCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)c1ccc2c(-c3ccc(C(=O)O)cc3)nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)[C@H]1CC[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C