3527 SMILES Strings for Prostaglandin D2 receptor 2

Compound Name
SMILES String
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3ccccc3)C2=O)c2cc(Cl)ccc12
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3ccccc3)C2=O)c2cc(F)ccc12
COc1ccc2N(CC(O)=O)C(=O)C3(CC(=O)N(Cc4ccccc4)C3=O)c2c1
CN(C)C(=O)CN1C(=O)CC2(C1=O)C(=O)N(CC(O)=O)c1ccc(F)cc21
CN(C)C(=O)CN1C(=O)CC2(C1=O)C(=O)N(CC(O)=O)c1ccc(Cl)cc21
COCCOCN1C(=O)CC2(C1=O)C(=O)N(CC(O)=O)c1ccc(F)cc21
OC(=O)CCCN1C(=O)C2(CC(=O)N(CC=C)C2=O)c2cc(Cl)ccc12
CN1C(=O)C2(CC(=O)N(Cc3ccccc3)C2=O)c2cc(Cl)ccc12
CN1C(=O)CC2(C1=O)C(=O)N(CC(O)=O)c1ccc(Cl)cc21
COCCN1C(=O)CC2(C1=O)C(=O)N(CC(O)=O)c1ccc(Cl)cc21
OC(=O)CCCN1C(=O)C2(CC(=O)N(Cc3ccccc3)C2=O)c2cc(Cl)ccc12
CN1C(=O)CC2(C1=O)C(=O)N(CCCC(O)=O)c1ccc(F)cc21
OC(=O)CCCN1C(=O)C2(CC(=O)N(CC=C)C2=O)c2cc(F)ccc12
OC(=O)CCCN1C(=O)C2(CC(=O)N(Cc3ccccc3)C2=O)c2cc(F)ccc12
CCOC(=O)CN1C(=O)C2(CC(=O)N(Cc3ccccc3)C2=O)c2cc(Cl)ccc12
OC(=O)CCCN1C(=O)C2(CC(=O)N(Cc3ccccc3F)C2=O)c2cc(Cl)ccc12
COc1ccc(CN2C(=O)CC3(C(=O)N(CCCC(O)=O)c4ccc(Cl)cc34)C2=O)cc1
OC(=O)CCCN1C(=O)C2(CC(=O)N(Cc3ccc(Cl)cc3)C2=O)c2cc(Cl)ccc12
Clc1ccc2N(Cc3nnn[nH]3)C(=O)C3(CC(=O)N(Cc4ccccc4)C3=O)c2c1
OC(=O)CN1C(=O)C2(CC(=O)N(CCc3ccccc3)C2=O)c2cc(Cl)ccc12
OC(=O)CN1C(=O)C2(CC(=O)N(C\C=C\c3ccccc3)C2=O)c2cc(Cl)ccc12
CC(N1C(=O)CC2(C(=O)N(CC(O)=O)c3ccc(Cl)cc23)C1=O)c1ccccc1
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3ccccc3F)C2=O)c2cc(Cl)ccc12
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3ccc(F)cc3)C2=O)c2cc(Cl)ccc12
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3cccc(Cl)c3)C2=O)c2cc(Cl)ccc12
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3ccc(Cl)cc3)C2=O)c2cc(Cl)ccc12
COc1ccccc1CN1C(=O)CC2(C(=O)N(CC(O)=O)c3ccc(Cl)cc23)C1=O
COc1cccc(CN2C(=O)CC3(C(=O)N(CC(O)=O)c4ccc(Cl)cc34)C2=O)c1
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3ccc(Oc4ccccc4)cc3)C2=O)c2cc(Cl)ccc12
CS(=O)(=O)c1ccc(CN2C(=O)CC3(C2=O)C(=O)N(CC(O)=O)c2ccc(Cl)cc32)cc1
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3cccc(F)c3F)C2=O)c2cc(Cl)ccc12
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3cc(F)ccc3F)C2=O)c2cc(Cl)ccc12
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3cc(F)cc(F)c3)C2=O)c2cc(Cl)ccc12
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3ccc(F)c(F)c3)C2=O)c2cc(Cl)ccc12
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3cc(F)ccc3Cl)C2=O)c2cc(Cl)ccc12
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3cc(Cl)ccc3F)C2=O)c2cc(Cl)ccc12
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3cc(Cl)cc(Cl)c3)C2=O)c2cc(Cl)ccc12
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3cc(F)cc(Cl)c3)C2=O)c2cc(Cl)ccc12
COc1ccc(CN2C(=O)CC3(C2=O)C(=O)N(CC(O)=O)c2ccc(Cl)cc32)cc1F
Cn1nnc2cc(CN3C(=O)CC4(C3=O)C(=O)N(CC(O)=O)c3ccc(Cl)cc43)ccc12
Cc1nc(CN2C(=O)CC3(C2=O)C(=O)N(CC(O)=O)c2ccc(Cl)cc32)cs1
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3csc(n3)-c3cccc(Cl)c3)C2=O)c2cc(Cl)ccc12
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3csc(n3)-c3ccc(Cl)cc3)C2=O)c2cc(Cl)ccc12
COc1ccc(cc1)-c1nc(CN2C(=O)CC3(C2=O)C(=O)N(CC(O)=O)c2ccc(Cl)cc32)no1
CC(C)(C)c1nc(CN2C(=O)CC3(C2=O)C(=O)N(CC(O)=O)c2ccc(Cl)cc32)no1
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3ncco3)C2=O)c2cc(Cl)ccc12
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3nnc(s3)C3CC3)C2=O)c2cc(Cl)ccc12
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3ccoc3)C2=O)c2cc(Cl)ccc12
OC(=O)CN1C(=O)C2(CC(=O)N(Cc3c[nH]c4ccccc34)C2=O)c2cc(Cl)ccc12
Cc1noc(C)c1CN1C(=O)CC2(C1=O)C(=O)N(CC(O)=O)c1ccc(Cl)cc21
Cc1onc(c1CN1C(=O)CC2(C1=O)C(=O)N(CC(O)=O)c1ccc(Cl)cc21)-c1ccccc1
Cc1noc(c1CN1C(=O)CC2(C1=O)C(=O)N(CC(O)=O)c1ccc(Cl)cc21)-c1ccccc1
COc1c(C)cnc(CN2C(=O)CC3(C2=O)C(=O)N(CC(O)=O)c2ccc(Cl)cc32)c1C
OC(=O)CN1C(=O)C2(CN(Cc3ccccc3)C(=O)C2)c2cc(Cl)ccc12
OC(=O)CN1C(=O)C2(CN(Cc3cc(Cl)ccc3F)C(=O)C2)c2cc(Cl)ccc12
Cc1noc(c1CN1CC2(CC1=O)C(=O)N(CC(O)=O)c1ccc(Cl)cc21)-c1ccccc1
Cc1onc(c1CN1CCC2(C1=O)C(=O)N(CC(O)=O)c1ccc(Cl)cc21)-c1ccccc1
OC(=O)CN1C(=O)[C@@]2(CC(=O)N(Cc3ccccc3)C2=O)c2cc(Cl)ccc12 |r|
OC(=O)CN1C(=O)[C@]2(CC(=O)N(Cc3ccccc3)C2=O)c2cc(Cl)ccc12 |r|
OC(=O)CN1C(=O)[C@@]2(CC(=O)N(Cc3ccccc3F)C2=O)c2cc(Cl)ccc12 |r|
OC(=O)CN1C(=O)[C@]2(CC(=O)N(Cc3ccccc3F)C2=O)c2cc(Cl)ccc12 |r|
OC(=O)CN1C(=O)[C@@]2(CC(=O)N(Cc3cccc(Cl)c3)C2=O)c2cc(Cl)ccc12 |r|
OC(=O)CN1C(=O)[C@]2(CC(=O)N(Cc3cccc(Cl)c3)C2=O)c2cc(Cl)ccc12 |r|
COc1cccc(CN2C(=O)C[C@@]3(C(=O)N(CC(O)=O)c4ccc(Cl)cc34)C2=O)c1 |r|
COc1cccc(CN2C(=O)C[C@]3(C(=O)N(CC(O)=O)c4ccc(Cl)cc34)C2=O)c1 |r|
OC(=O)CN1C(=O)[C@]2(CC(=O)N(Cc3cc(Cl)ccc3F)C2=O)c2cc(Cl)ccc12 |r|
OC(=O)CN1C(=O)[C@@]2(CC(=O)N(Cc3cc(Cl)ccc3F)C2=O)c2cc(Cl)ccc12 |r|
OC(=O)CN1C(=O)[C@]2(CN(Cc3cc(Cl)ccc3F)C(=O)C2)c2cc(Cl)ccc12 |r|
OC(=O)CN1C(=O)[C@@]2(CN(Cc3cc(Cl)ccc3F)C(=O)C2)c2cc(Cl)ccc12 |r|
Cc1c(Cc2cccnc2S(=O)(=O)c2ccccc2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2cccnc2S(=O)(=O)c2ccc(F)cc2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2cccnc2S(=O)(=O)c2ccc(Cl)cc2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(cc2)S(C)(=O)=O)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccncc2S(=O)(=O)c2ccccc2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ncccc2S(=O)(=O)c2ccccc2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2cccn2S(=O)(=O)c2ccccc2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2cccnc2)c2cc(F)ccc2n1CC(O)=O
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CCC(CC1)n1cc(C)c2ccccc12
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CCC(CC1)n1cc(C)c2cc(Cl)ccc12
CCOc1ccc(cc1)S(=O)(=O)N1CCC(CC1)n1cc(C)c2cc(Cl)ccc12
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CCC(C1)n1cc(C)c2cc(Cl)ccc12
CCOc1ccc(cc1)S(=O)(=O)N1CCC(C1)n1cc(C)c2cc(Cl)ccc12
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CCC(CC1)n1cc(C)c2ccc(Cl)cc12
CCOc1ccc(cc1)S(=O)(=O)N1CCC(CC1)n1cc(C)c2ccc(Cl)cc12
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CCC(C1)n1cc(C)c2ccc(Cl)cc12
CCOc1ccc(cc1)S(=O)(=O)N1CCC(C1)n1cc(C)c2ccc(Cl)cc12
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CCC(CC1)n1cc(C)c2cc(F)ccc12
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CCC(CC1)n1cc(CC(O)=O)c2ccc(F)cc12
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CC[C@H](C1)n1cc(CC(O)=O)c2ccccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CC[C@@H](C1)n1nc(CC(O)=O)c2cc(Cl)ccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CCC(CC1)n1cc(OC=O)c2ccccc12
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CC[C@H](C1)n1cc(CC(O)=O)c2ccc(Cl)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CC[C@H](C1)n1cc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CC[C@H](C1)n1cc(C(O)=O)c2ccc(Cl)cc12 |r|
OC(=O)Cc1cc(C2CCN(CC2)S(=O)(=O)c2ccccc2)c2cc(F)ccc2c1
Cc1ccc(cc1)S(=O)(=O)N1CCC(CC1)c1cc(CC(O)=O)cc2ccc(F)cc12
OC(=O)Cc1cc(C2CCN(CC2)S(=O)(=O)c2ccccn2)c2cc(F)ccc2c1
OC(=O)Cc1cc(C2CCN(CC2)S(=O)(=O)c2cccnc2)c2cc(F)ccc2c1
OC(=O)Cc1cc(C2CCN(CC2)S(=O)(=O)c2ccncc2)c2cc(F)ccc2c1
OC(=O)Cc1cc(C2CCN(CC2)S(=O)(=O)c2ccccc2Cl)c2cc(F)ccc2c1
OC(=O)Cc1cc(C2CCN(CC2)S(=O)(=O)c2cccc(Cl)c2)c2cc(F)ccc2c1
OC(=O)Cc1cc(C2CCN(CC2)S(=O)(=O)c2ccc(Cl)cc2)c2cc(F)ccc2c1
CS(=O)(=O)c1cccc(c1)S(=O)(=O)N1CCC(CC1)c1cc(CC(O)=O)cc2ccc(F)cc12
OC(=O)Cc1cc(C2CCN(CC2)S(=O)(=O)c2cc(Cl)ccc2Cl)c2cc(F)ccc2c1
OC(=O)Cc1cc(C2CCN(CC2)S(=O)(=O)c2ccc(Cl)cc2Cl)c2cc(F)ccc2c1
OC(=O)Cc1cc(C2CCN(CC2)S(=O)(=O)c2cc(Cl)cc(Cl)c2)c2cc(F)ccc2c1
OC(=O)Cc1cc(C2CCN(CC2)S(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2cc(F)ccc2c1
OC(=O)Cn1c2CC[C@@H](Cc2c2cc(F)ccc12)Nc1ncc(F)cn1
OC(=O)Cn1c2CC[C@H](Cc2c2cc(F)ccc12)Nc1ncc(F)cn1
OC(=O)Cn1c2CC[C@@H](Cc2c2cc(F)ccc12)Nc1ncc(Cl)cn1
OC(=O)Cn1c2CC[C@H](Cc2c2cc(F)ccc12)Nc1ncc(Cl)cn1
OC(=O)Cn1c2CC[C@H](Cc2c2cc(F)ccc12)Nc1ncc(cn1)C(F)(F)F
OC(=O)Cn1c2CC[C@H](Cc2c2cc(F)ccc12)Nc1nccc(n1)C(F)(F)F
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1ncc(F)cn1
CN([C@@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1ncc(F)cn1
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1ncc(Cl)cn1
CN([C@@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1ncc(Cl)cn1
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1ncc(cn1)C(F)(F)F
CN([C@@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1ncc(cn1)C(F)(F)F
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1nccc(n1)C(F)(F)F
CN([C@@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1nccc(n1)C(F)(F)F
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1ncccn1
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1nc(C)cc(C)n1
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1nccc(C)n1
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1nc2cc(Cl)ccc2o1
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1nc2ccccc2o1
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1nc2ccccc2s1
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1ncnc2ccccc12
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1nc(nc2ccccc12)C(F)(F)F
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1nc(C)nc2ccccc12
CCN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1ncc(Cl)cn1
CCCN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1ncc(Cl)cn1
CC(C)N([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1ncc(Cl)cn1
OC(=O)Cn1c2CC[C@@H](Cc2c2cc(F)ccc12)N(CC1CC1)c1ncc(Cl)cn1
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1ncc2ccccc2n1
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1nc2cc(F)ccc2o1
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1ncc(cn1)-c1ccccc1
COc1cnc(nc1)N(C)[C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1nc2ccc(Cl)cc2s1
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1nc2cc(Cl)ccc2s1
COCCN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1ncc(Cl)cn1
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1ccc(cn1)C(F)(F)F
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1ccc(F)cn1
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1ccc(Cl)cn1
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1nc2ccc(F)cc2s1
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1nc2cc(F)ccc2s1
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1nc2ccc(Cl)cc2o1
OC(=O)Cn1c2CC[C@@H](Cc2c2cc(F)ccc12)N(CC(F)F)c1ncc(Cl)cn1
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1nc2ccc(F)cc2o1
CN([C@H]1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1cnc2ccccc2n1
CN(C1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1nc(C)cs1
CN(C1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1nc(cs1)C(C)(C)C
CN(C1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1cc(on1)C(C)(C)C
CN(C1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1ccn(C)n1
CN(C1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1nnc(C)s1
CN(C1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1ccon1
CN(C1CCc2c(C1)c1cc(F)ccc1n2CC(O)=O)c1cc(C)on1
CN(C1CCc2c(C1)c1ccccc1n2CC(O)=O)c1ncc(Cl)cn1
CN(C1CCc2c(C1)c1cc(Cl)ccc1n2CC(O)=O)c1ncc(Cl)cn1
CN(C1CCc2c(C1)c1cc(C)ccc1n2CC(O)=O)c1ncc(Cl)cn1
CN(C1CCc2c(C1)c1cc(OC(F)(F)F)ccc1n2CC(O)=O)c1ncc(Cl)cn1
COc1ccc2n(CC(O)=O)c3CCC(Cc3c2c1)N(C)c1ncc(Cl)cn1
CN(C1CCc2c(C1)c1cc(ccc1n2CC(O)=O)C(F)(F)F)c1ncc(Cl)cn1
Cc1nn(Cc2ccc(NC(=O)c3cc4ccccc4[nH]3)cc2F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3cc4ccccc4[nH]3)cc2Cl)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3cc4ccccc4n3Cc3ccccc3)cc2F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3oc4ccc(F)cc4c3C)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3cc4ccccc4o3)cc2Cl)c(C)c1CC(O)=O
COc1ccc2oc(cc2c1)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)cc1
Cc1nn(Cc2ccc(NC(=O)c3oc4c(F)cccc4c3C)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3cc4cc(Cl)ccc4o3)cc2)c(C)c1CC(O)=O
COc1cccc2cc(oc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)cc1
Cc1nn(Cc2ccc(NC(=O)c3cc4ccccc4[nH]3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3cc4ccc(F)cc4[nH]3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3cc4cc(F)ccc4[nH]3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3c(C)c4ccccc4n3C)cc2)c(C)c1CC(O)=O
COc1ccc2[nH]c(C(=O)Nc3ccc(Cn4nc(C)c(CC(O)=O)c4C)cc3)c(C)c2c1
Cc1nn(Cc2ccc(NC(=O)c3cc4ccccc4s3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3cc4ccccc4n3C)cc2)c(C)c1CC(O)=O
CCn1c(cc2ccccc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)cc1
Cc1nn(Cc2ccc(NC(=O)c3cc4ccccc4n3Cc3ccccc3)cc2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3cc4cc(Cl)ccc4o3)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3cc4ccccc4[nH]3)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3cc4ccccc4n3C)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3cc4ccccc4n3CC)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3cc4cc(F)ccc4[nH]3)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3c(C)c4ccccc4n3C)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3cc4ccc(F)cc4[nH]3)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3cc4ccccc4o3)cc2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3oc4ccc(F)cc4c3C)cc2F)c(C)c1CC(O)=O
CCCn1c(cc2ccc(F)cc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)cc1
CCn1c(cc2ccc(F)cc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)cc1
Cc1nn(Cc2ccc(NC(=O)c3cc4ccccc4n3C)cc2F)c(C)c1CC(O)=O
CCn1c(cc2ccccc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)c(F)c1
CCn1c(cc2cc(F)ccc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)c(F)c1
Cc1nn(Cc2ccc(NC(=O)c3oc4c(Cl)cccc4c3C)cc2)c(C)c1CC(O)=O
CCc1c(oc2c(F)cccc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)cc1
CCc1c(oc2c(F)cc(F)cc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)cc1
Cc1nn(Cc2ccc(NC(=O)c3cc4ccc(Cl)cc4o3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3oc4c(Cl)cccc4c3C)cc2F)c(C)c1CC(O)=O
CCc1c(oc2c(Cl)cccc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)c(F)c1
Cc1nn(Cc2ccc(NC(=O)c3cc4ccc(Cl)cc4o3)cc2F)c(C)c1CC(O)=O
CCn1c(cc2c(F)cccc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)c(F)c1
CCn1c(cc2ccc(F)cc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)c(F)c1
CCCn1c(cc2ccc(F)cc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)c(F)c1
COCc1c(oc2ccccc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)c(F)c1
Cc1nn(Cc2ccc(NC(=O)c3oc4ccc(Cl)cc4c3C)cc2F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3oc4cc(Br)ccc4c3C)cc2F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3sc4ccc(F)cc4c3C)cc2F)c(C)c1CC(O)=O
CCc1c(oc2ccc(F)cc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)c(F)c1
CCc1c(oc2ccc(F)cc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)cc1
COc1ccc2oc(C(=O)Nc3ccc(Cn4nc(C)c(CC(O)=O)c4C)c(F)c3)c(C)c2c1
Cc1nn(Cc2ccc(NC(=O)c3oc4c(F)cccc4c3C)cc2F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3cc4cc(F)ccc4n3C)cc2F)c(C)c1CC(O)=O
CCCc1c(oc2ccc(F)cc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)c(F)c1
CCCCn1c(cc2ccccc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)c(F)c1
CCCn1c(cc2cc(F)ccc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)c(F)c1
CCCCn1c(cc2cc(F)ccc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)c(F)c1
CCCn1c(cc2ccccc12)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)c(F)c1
Cc1nn(Cc2ccc(NC(=O)c3coc4ccccc34)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3c[nH]c4ccccc34)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3csc4ccccc34)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(Cl)cc3C)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccccc3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(C)cc3)cc2)c(C)c1CC(O)=O
COc1ccc(cc1)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)cc1
Cc1nn(Cc2ccc(NC(=O)c3ccc(Cl)cc3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc4ccccc4c3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(Cl)c(Cl)c3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc4ccccc4n3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)CCc3ccccc3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(cc3C)C(F)(F)F)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(C)cc3C)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)\C=C\c3ccccc3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)\C=C\c3ccc(Cl)cc3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(cc3)C(C)(C)C)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(Br)cc3C)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3cc(C)c(Br)cc3C)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(Cl)cc3Cl)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(Cl)cc3F)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(C)cc3F)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(C)cc3C(F)(F)F)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(cc3F)C(F)(F)F)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3cc4ccccc4cc3Cl)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3c(C)cc(C)cc3C)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3cc4ccccc4cc3C)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc4ccccc4c3C)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(Br)cc3Cl)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(Cl)cc3Br)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3cccc4CCCCc34)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc4ccccc4c3Br)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3cc(C)ccc3Br)cc2)c(C)c1CC(O)=O
CC(C)C(=O)Nc1ccc(Cn2nc(C)c(CC(O)=O)c2C)cc1
Cc1nn(Cc2ccc(NC(=O)C3CCCCC3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)C3[C@H]4C[C@@H]5C[C@@H](C[C@H]3C5)C4)cc2)c(C)c1CC(O)=O |r,wU:13.13,17.16,wD:15.15,19.18,THB:21:17:13.14.12:20,(2.62,6.84,;3.39,5.51,;2.92,4.04,;4.16,3.14,;4.56,1.65,;3.47,.56,;1.99,.96,;.9,-.13,;1.29,-1.62,;.21,-2.7,;-1.28,-2.31,;-1.68,-.82,;-2.37,-3.39,;-2.68,-5.45,;-2.29,-6.93,;-3.37,-8.02,;-4.86,-7.62,;-5.26,-6.14,;-4.89,-4.04,;-3.55,-4.38,;-2.95,-6.7,;-4.17,-5.05,;2.78,-2.01,;3.87,-.93,;5.41,4.04,;6.74,3.27,;4.93,5.51,;5.7,6.84,;4.93,8.18,;5.7,9.51,;3.39,8.18,)|
Cc1nn(Cc2ccc(NC(=O)C3CCC3)cc2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3ccc(Cl)cc3C)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3ccccc3)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3ccc(C)cc3)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3ccc(Cl)cc3)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3ccc(Cl)c(Cl)c3)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3ccc4ccccc4c3)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3ccc(C)cc3C)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)C3CCC(CC3)C(F)(F)F)cc2)c(CC)c1CC(O)=O |(-9.77,.07,;-8.43,.84,;-7.1,.07,;-7.1,-1.47,;-5.63,-1.95,;-4.86,-3.28,;-3.32,-3.28,;-2.55,-4.62,;-1.01,-4.62,;-.24,-3.28,;1.3,-3.28,;2.07,-1.95,;1.3,-.61,;3.61,-1.95,;4.38,-3.28,;5.92,-3.28,;6.69,-1.95,;5.92,-.61,;4.38,-.61,;8.23,-1.95,;9.77,-1.95,;8.23,-3.49,;8.23,-.41,;-1.01,-1.95,;-2.55,-1.95,;-4.73,-.7,;-3.19,-.7,;-2.42,.63,;-5.63,.54,;-5.08,1.98,;-6.05,3.18,;-5.5,4.62,;-7.57,2.94,)|
CCc1nn(Cc2ccc(NC(=O)c3ccc(Br)cc3C)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)C3CCCCC3)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3cc(C)ccc3Br)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3cccc(Cl)c3Cl)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3cccc4CCCCc34)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3ccc(Br)cc3Cl)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3ccccc3CC)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3ccc(Cl)cc3Br)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3cccc(C)c3Br)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3ccc4ccccc4c3Br)cc2)c(CC)c1CC(O)=O
CCCc1c(C)cccc1C(=O)Nc1ccc(Cn2nc(CC)c(CC(O)=O)c2CC)cc1
CCc1nn(Cc2ccc(NC(=O)c3cccc(C)c3CC(C)C)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3ccccc3C3CCCCC3)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)C(C)(C)C)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)C3CCC3)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)C3CCCC3)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)C3[C@H]4C[C@@H]5C[C@@H](C[C@H]3C5)C4)cc2)c(CC)c1CC(O)=O |r,wU:16.22,14.24,wD:18.17,20.21,(1.28,4.24,;2.77,4.64,;3.86,3.55,;3.38,2.09,;4.63,1.18,;4.63,-.36,;3.3,-1.13,;1.96,-.36,;.63,-1.13,;.63,-2.67,;-.71,-3.44,;-2.04,-2.67,;-2.04,-1.13,;-3.37,-3.44,;-4.7,-3.06,;-6.38,-4.77,;-6.67,-6.13,;-7.07,-4.64,;-5.98,-3.55,;-4.49,-3.95,;-4.1,-5.43,;-5.19,-6.52,;-5.23,-1.62,;1.96,-3.44,;3.3,-2.67,;5.87,2.09,;7.36,1.69,;7.76,.2,;5.4,3.55,;6.49,4.64,;6.09,6.13,;7.18,7.22,;4.6,6.53,)|
CCc1nn(Cc2ccc(NC(=O)C(C)C)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3ccccc3C3CC3)cc2)c(CC)c1CC(O)=O
Cc1c(CC(O)=O)c(nn1Cc1ccc(NC(=O)c2ccc(cc2)C(F)(F)F)cc1)C1CCCCC1
Cc1nn(Cc2ccc(NC(=O)c3ccc4ccccc4c3)cc2)c(c1CC(O)=O)-c1ccccc1
Cc1nn(Cc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2)c(c1CC(O)=O)-c1ccccc1
Cc1nn(Cc2ccc(NC(=O)c3ccc(Cl)c(Cl)c3)cc2)c(c1CC(O)=O)-c1ccccc1
Cc1c(CC(O)=O)c(nn1Cc1ccc(NC(=O)c2ccc(cc2)C(F)(F)F)cc1)-c1ccccc1
Cc1c(CC(O)=O)c(nn1Cc1ccc(NC(=O)c2ccc3ccccc3c2)cc1)-c1ccccc1
Cc1c(CC(O)=O)c(nn1Cc1ccc(NC(=O)c2ccc(Cl)c(Cl)c2)cc1)-c1ccccc1
CCCc1nn(Cc2ccc(NC(=O)c3ccc(cc3C)C(F)(F)F)cc2)c(C(C)C)c1CC(O)=O
CCCc1nn(Cc2ccc(NC(=O)c3ccc(Cl)cc3)cc2)c(C(C)C)c1CC(O)=O
CCCc1nn(Cc2ccc(NC(=O)c3ccc(Cl)cc3C)cc2)c(C(C)C)c1CC(O)=O
CCCc1nn(Cc2ccc(NC(=O)c3ccccc3)cc2)c(C(C)C)c1CC(O)=O
CCCc1nn(Cc2ccc(NC(=O)c3ccc(Cl)c(Cl)c3)cc2)c(C(C)C)c1CC(O)=O
CCCc1nn(Cc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2)c(C(C)C)c1CC(O)=O
CCCc1nn(Cc2ccc(NC(=O)c3ccc4ccccc4c3)cc2)c(C(C)C)c1CC(O)=O
OC(=O)Cc1c(nn(Cc2ccc(NC(=O)c3ccc(Cl)cc3)cc2)c1-c1ccccc1)-c1ccccc1
OC(=O)Cc1c(nn(Cc2ccc(NC(=O)c3ccc4ccccc4c3)cc2)c1-c1ccccc1)-c1ccccc1
OC(=O)Cc1c(nn(Cc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2)c1-c1ccccc1)-c1ccccc1
CCc1c(CC(O)=O)c(nn1Cc1ccc(NC(=O)c2ccc(Cl)cc2C)cc1)C1CC1
CCc1c(CC(O)=O)c(nn1Cc1ccc(NC(=O)c2ccc(cc2)C(F)(F)F)cc1)C1CC1
CCc1nn(Cc2ccc(NC(=O)c3cccc4ccccc34)cc2)c(C2CC2)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3ccc(Cl)cc3C)cc2)c(C2CC2)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2)c(C2CC2)c1CC(O)=O
CCc1c(CC(O)=O)c(nn1Cc1ccc(NC(=O)c2cccc3ccccc23)cc1)C1CC1
CCc1c(CC(O)=O)c(C)nn1Cc1ccc(NC(=O)c2ccc(cc2)C(F)(F)F)cc1
CCc1nn(Cc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2)c(C)c1CC(O)=O
Cc1c(CC(O)=O)cnn1Cc1ccc(NC(=O)c2ccc3ccccc3c2)cc1
Cc1c(CC(O)=O)cnn1Cc1ccc(NC(=O)c2ccc(Cl)c(Cl)c2)cc1
Cc1nn(Cc2ccc(NC(=O)c3ccc4ccccc4c3)cc2)cc1CC(O)=O
CCc1c(CC(O)=O)cnn1Cc1ccc(NC(=O)c2ccc3ccccc3c2)cc1
COc1c(CC(O)=O)c(C)nn1Cc1ccc(NC(=O)c2ccc3ccccc3c2)cc1
Cc1nn(Cc2ccc(NC(=O)OCc3ccccc3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)OCc3ccccc3)cc2)c(C)c1CCC(O)=O
CCc1nn(Cc2ccc(NC(=O)OCc3ccccc3)cc2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)OCc3ccc(Cl)c(Cl)c3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)OCc3ccccc3Cl)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)OCc3ccccc3Br)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)OCc3ccc4ccccc4c3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)OC(C)(C)C)cc2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)OCc3ccc(Cl)c(Cl)c3)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)OCc3ccccc3Cl)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)OCc3ccccc3Br)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(NC(=O)OCc3ccc4ccccc4c3)cc2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)OCc3ccccc3)cc2Cl)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)OCc3ccccc3)cc2F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)NCc3ccccc3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NS(=O)(=O)c3ccccc3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NS(=O)(=O)c3ccc(Cl)cc3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NS(=O)(=O)c3ccc(Cl)c(Cl)c3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NS(=O)(=O)c3ccc(cc3)C(F)(F)F)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NCc3ccc(Cl)cc3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NCc3ccccc3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NCc3ccc(cc3)C(F)(F)F)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccccc3)c(C)c2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(Cl)cc3)c(C)c2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)c(C)c2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(Cl)c(Cl)c3)c(C)c2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc4ccccc4c3)cc2C)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(Cl)cc3)cc2Cl)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(Cl)cc3C)cc2Cl)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2Cl)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)CCc3ccccc3)cc2Cl)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccccc3)cc2Cl)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)\C=C\c3ccccc3)cc2Cl)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(C)cc3C)cc2Cl)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc4ccccc4c3)cc2Cl)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(cc3C)C(F)(F)F)cc2Cl)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(Cl)c(Cl)c3)cc2Cl)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(cc3C)C(F)(F)F)cc2F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(Cl)c(Cl)c3)cc2F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(Cl)cc3C)cc2F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc4ccccc4c3)cc2F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)\C=C\c3ccccc3)cc2F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(Cl)cc3C)cc2)c(C)c1CCC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2)c(C)c1CCC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccccc3)cc2)c(C)c1CCC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(cc3)C(C)(C)C)cc2)c(C)c1CCC(O)=O
Cc1nn(Cc2ccc(NC(=O)CCc3ccccc3)cc2)c(C)c1CCC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(Cl)c(Cl)c3)cc2)c(C)c1CCC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(cc3C)C(F)(F)F)cc2)c(C)c1CCC(O)=O
Cc1nn(Cc2ccc(cc2)C(=O)Nc2cccc(F)c2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)C(=O)Nc2ccc(Cl)c(F)c2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)C(=O)Nc2ccc(Cl)c(Cl)c2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)C(=O)Nc2ccc(F)c(Cl)c2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)C(=O)Nc2cccc(c2)C(F)(F)F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)C(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Cl)c2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)C(=O)Nc2cc(Cl)cc(Cl)c2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)C(=O)Nc2ccc(Br)c(F)c2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)C(=O)Nc2cccc(F)c2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)C(=O)Nc2ccc(Cl)c(F)c2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)C(=O)Nc2ccc(F)c(Cl)c2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)C(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)C(=O)Nc2ccc(F)c(Br)c2)c(CC)c1CC(O)=O
CC(C)(C)c1nn(Cc2ccc(cc2)C(=O)Nc2ccc(F)c(Cl)c2)c(c1CC(O)=O)C(C)(C)C
CCc1nn(Cc2ccc(cc2)C(=O)Nc2ccc(Br)c(F)c2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)C(=O)NCc2ccc3ccccc3c2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)C(=O)NCc2ccc(Cl)c(Cl)c2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)C(=O)NCc2ccc(Cl)c(c2)C(F)(F)F)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)C(=O)NCc2ccc(cc2)C(F)(F)F)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)C(=O)N[C@H]2CC[C@@H](CC2)c2ccccc2)c(CC)c1CC(O)=O |r,wU:15.15,wD:18.22,(-5.21,4.34,;-6.55,3.57,;-6.55,2.03,;-5.3,1.13,;-5.78,-.34,;-5.01,-1.67,;-3.47,-1.67,;-2.7,-3.01,;-1.16,-3.01,;-.39,-1.67,;-1.16,-.34,;-2.7,-.34,;1.15,-1.67,;1.92,-.34,;1.92,-3.01,;3.46,-3.01,;4.23,-1.67,;5.77,-1.67,;6.54,-3.01,;5.77,-4.34,;4.23,-4.34,;8.08,-3.01,;8.85,-4.34,;10.39,-4.34,;11.16,-3.01,;10.39,-1.67,;8.85,-1.67,;-7.32,-.34,;-8.09,-1.67,;-9.63,-1.67,;-7.79,1.13,;-9.28,1.52,;-9.68,3.01,;-8.59,4.1,;-11.16,3.41,)|
CCc1nn(Cc2ccc(cc2)C(=O)N[C@@H]2CCC[C@@H](C2)c2ccccc2)c(CC)c1CC(O)=O |r|
CCc1nn(Cc2ccc(cc2)C(=O)Nc2ccc3ccccc3n2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)C(=O)NC2CCC(C)(C)CC2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)C(=O)NC2CCC3CCCCC3C2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)C(=O)NC2CCC(CC2)C(C)(C)C)c(CC)c1CC(O)=O |(-4.06,4.34,;-5.39,3.57,;-5.39,2.03,;-4.14,1.13,;-4.62,-.34,;-3.85,-1.67,;-2.31,-1.67,;-1.54,-3.01,;-0,-3.01,;.77,-1.67,;-0,-.34,;-1.54,-.34,;2.31,-1.67,;3.08,-.34,;3.08,-3.01,;4.62,-3.01,;5.39,-4.34,;6.93,-4.34,;7.7,-3.01,;6.93,-1.67,;5.39,-1.67,;9.24,-3.01,;10.01,-4.34,;10.01,-1.67,;8.47,-4.34,;-6.16,-.34,;-6.93,-1.67,;-8.47,-1.67,;-6.64,1.13,;-8.12,1.52,;-8.52,3.01,;-7.43,4.1,;-10.01,3.41,)|
CCc1nn(Cc2ccc(cc2F)C(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)C(=O)NCc2cc3ccccc3o2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)S(=O)(=O)Nc2ccc(F)cc2)c(C)c1CC(O)=O
COc1ccc(CCNS(=O)(=O)c2ccc(Cn3nc(C)c(CC(O)=O)c3C)cc2)cc1OC
CCc1nn(Cc2ccc(cc2)S(=O)(=O)Nc2ccc(C)c(Cl)c2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)S(=O)(=O)Nc2ccc(Cl)c(Cl)c2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)S(=O)(=O)Nc2ccc(Cl)c(F)c2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2)c(C)c1CC(=O)NS(=O)(=O)C(C)(C)C
Cc1nn(Cc2ccc(cc2)C#Cc2ccc(cc2)C(F)(F)F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(\C=C\c3ccc(cc3)C(F)(F)F)cc2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(\C=C\c3ccc(Cl)cc3)cc2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(OCc3ccc(Cl)c(Cl)c3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(OCc3ccc(cc3)C(F)(F)F)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(OCc3ccc(Cl)cc3C)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(OCc3ccccc3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(OCc3ccc(Cl)c(c3)C(F)(F)F)cc2)c(C)c1CC(O)=O
COc1ccc(COc2ccc(Cn3nc(C)c(CC(O)=O)c3C)cc2)cc1C(F)(F)F
CCc1nn(Cc2ccc(OCc3ccc(Cl)c(c3)C(F)(F)F)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(OCc3cc(Cl)cc(Cl)c3)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(OCc3cccc(Cl)c3)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(OCc3cccc(c3)C(F)(F)F)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(OCc3ccc(OC(F)(F)F)c(Cl)c3)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(OCc3ccc(OC)c(c3)C(F)(F)F)cc2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(OCc3cccc(C)c3)cc2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(COc3ccc(cc3)C(F)(F)F)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(COc3ccc(Cl)c(Cl)c3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(COc3ccccc3)cc2)c(C)c1CC(O)=O
CC(Oc1ccc(Cl)c(Cl)c1)c1ccc(Cn2nc(C)c(CC(O)=O)c2C)cc1
CC(Oc1ccc(cc1)C(F)(F)F)c1ccc(Cn2nc(C)c(CC(O)=O)c2C)cc1
CC(Oc1ccccc1)c1ccc(Cn2nc(C)c(CC(O)=O)c2C)cc1
Cc1nn(Cc2ccc(cc2)C(O)Cc2ccccc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)C(=O)Cc2ccccc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(CSc3ccc(cc3)C(F)(F)F)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(CS(=O)c3ccc(cc3)C(F)(F)F)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(CS(=O)(=O)c3ccc(cc3)C(F)(F)F)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(CSc3ccc(Cl)c(Cl)c3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(CS(=O)c3ccc(Cl)c(Cl)c3)cc2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(CS(=O)(=O)c3ccc(Cl)c(Cl)c3)cc2)c(C)c1CC(O)=O
CCc1nn(C(C)c2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2)c(CC)c1CC(O)=O
CCc1nn(C(C)c2ccc(cc2)C(=O)Nc2ccc(cc2)C(F)(F)F)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(NC(=O)c3ccc(Cl)c(Cl)c3)cn2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)S(=O)Cc2ccc3ccccc3c2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)S(=O)Cc2ccc(Cl)c(Cl)c2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)S(=O)Cc2ccc(Cl)c(Cl)c2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)S(=O)Cc2ccccc2)c(CC)c1CC(O)=O
FC(F)(F)c1ccccc1S(=O)(=O)Nc1nccnc1-c1ccc(Cn2ccc3ccccc23)cc1
CN(Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccccc1Cl)c1ccc(OC(F)(F)F)cc1
CCc1nc2ccccc2n1Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccccc1C(F)(F)F
CN(Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccccc1Cl)c1ccccc1
Clc1ccccc1S(=O)(=O)Nc1nccnc1-c1ccc(COc2ccc3ccccc3c2)cc1
Clc1ccccc1S(=O)(=O)Nc1nccnc1-c1ccc(Cn2ccc3ccccc23)cc1
Clc1ccccc1S(=O)(=O)Nc1nccnc1-c1ccc(COc2ccc3CCCCc3c2)cc1
CCc1nc2ccccc2n1Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccccc1Cl
FC(F)(F)c1ccccc1S(=O)(=O)Nc1nccnc1-c1ccc(CNc2ccc3OCOc3c2)cc1
COc1cccc(COCc2ccc(cc2)-c2nccnc2NS(=O)(=O)c2ccccc2C(F)(F)F)c1
CN(Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1cccc(Cl)c1)c1ccc(OC(F)(F)F)cc1
CN(Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1cccs1)c1ccc(Cl)cc1
O=S(=O)(Nc1nccnc1N1CCN(Cc2ccc3ccccc3n2)CC1)c1ccc(Oc2ccccc2)cc1
CN(Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccc(C)cc1)c1ccc(OC(F)(F)F)cc1
CN(Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccc(Cl)cc1)c1ccccc1
CN(Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccc(cc1)C#N)c1ccc(OC(F)(F)F)cc1
CN(Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccccc1C(F)(F)F)c1ccc(F)cc1
CN(Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccccc1C(F)(F)F)c1ccccc1
CN(Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccccc1C(F)(F)F)c1ccc(cc1)C#N
Fc1ccc(OCc2ccc(cc2)-c2nccnc2NS(=O)(=O)c2ccccc2C(F)(F)F)cc1
CCN(Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccccc1C(F)(F)F)c1ccccc1
FC(F)(F)c1ccccc1S(=O)(=O)Nc1nccnc1-c1ccc(CN2CCOc3ccccc23)cc1
CN(Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccccc1C(F)(F)F)c1cccc(F)c1
FC(F)(F)c1ccccc1S(=O)(=O)Nc1nccnc1-c1ccc(COc2ccc(Cl)nc2)cc1
FC(F)(F)c1ccccc1S(=O)(=O)Nc1nccnc1-c1ccc(Cn2c(cc3ccccc23)-c2ccccn2)cc1
Fc1ccc2n(Cc3ccc(cc3)-c3nccnc3NS(=O)(=O)c3ccccc3C(F)(F)F)ccc2c1
FC(F)(F)c1ccccc1S(=O)(=O)Nc1nccnc1-c1ccc(COc2ccccc2)cc1
CN(Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccccc1C(F)(F)F)c1ccc(Cl)cc1
CN(Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccccc1Cl)c1ccc(cc1)C#N
CN(Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccccc1C(F)(F)F)c1ccc(Cl)c(Cl)c1
FC(F)(F)c1ccccc1S(=O)(=O)Nc1nccnc1-c1ccc(COc2ccc(cc2)C#N)cc1
Fc1ccc2ccn(Cc3ccc(cc3)-c3nccnc3NS(=O)(=O)c3ccccc3C(F)(F)F)c2c1
COc1ccc2n(Cc3ccc(cc3)-c3nccnc3NS(=O)(=O)c3ccccc3Cl)c(C)cc2c1
COc1ccc(OCc2ccc(cc2)-c2nccnc2NS(=O)(=O)c2ccccc2C(F)(F)F)cc1
Clc1ccccc1S(=O)(=O)Nc1nccnc1-c1ccc(CN(Cc2ccccc2)c2ccccn2)cc1
FC(F)(F)c1ccccc1S(=O)(=O)Nc1nccnc1-c1ccc(CN2CCc3ccccc23)cc1
CN(Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccccc1C(F)(F)F)c1ccc(Cl)cc1Cl
FC(F)(F)c1ccccc1S(=O)(=O)Nc1nccnc1-c1ccc(COc2cccc(Cl)c2)cc1
CN(Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccccc1Cl)c1ccc(F)cc1F
Cc1cc2ccccc2n1Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccccc1C(F)(F)F
Fc1ccc2n(Cc3ccc(cc3)-c3nccnc3NS(=O)(=O)c3ccccc3Cl)ccc2c1
CN(Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccccc1Cl)c1ccccc1F
Cc1cc2ccccc2n1Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccccc1Cl
FC(F)(F)c1ccccc1S(=O)(=O)Nc1nccnc1-c1ccc(CN(Cc2ccccc2)c2ccccn2)cc1
CCN(Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccccc1Cl)c1ccccn1
Cc1cc2cc(Cl)ccc2n1Cc1ccc(cc1)-c1nccnc1NS(=O)(=O)c1ccccc1C(F)(F)F
Cc1ccccc1S(=O)(=O)c1ccc(cc1)-c1c(C)c(CC(O)=O)cc2ccc(F)cc12
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(C)(=O)=O
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)N1CCOCC1
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cn1)S(C)(=O)=O
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(NS(=O)(=O)c2ccccc2)cc1
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)cc1
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(NS(=O)(=O)c2ccccc2C(F)(F)F)cc1
Cc1ccccc1S(=O)(=O)Nc1ccc(cc1)-c1c(C)c(CC(O)=O)cc2ccc(Cl)cc12
CC(=O)Nc1ccc(cc1)-c1c(C)c(CC(O)=O)cc2ccc(Cl)cc12
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(NC(=O)c2ccccc2)cc1
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(NC(=O)Nc2ccccc2)cc1
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(=O)(=O)c1ccccc1Cl
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(=O)(=O)c1cccc(Cl)c1
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(=O)(=O)c1ccc(Cl)cc1
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(=O)(=O)c1ccccc1C(F)(F)F
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(=O)(=O)c1ccccc1OC(F)(F)F
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(=O)(=O)c1ccc(OC(F)(F)F)cc1
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(=O)(=O)c1ccc(Cl)cc1Cl
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(=O)(=O)c1cc(Cl)ccc1Cl
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(=O)(=O)c1ccc(F)cc1F
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(=O)(=O)c1c(F)cccc1F
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(=O)(=O)c1cc(Cl)cc(Cl)c1
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(=O)(=O)c1cc(F)cc(F)c1
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)c1cccc(Cl)c1
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)c1ccc(Cl)cc1
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)c1ccccc1C(F)(F)F
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)c1ccccc1OC(F)(F)F
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)c1ccc(OC(F)(F)F)cc1
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)c1cc(Cl)ccc1Cl
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)c1ccc(F)cc1F
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)c1c(F)cccc1F
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)c1cc(Cl)cc(Cl)c1
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)c1cc(F)cc(F)c1
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)Nc1ccc(F)cc1
Cc1ccc(NS(=O)(=O)c2ccc(cc2)-c2c(C)c(CC(O)=O)cc3ccc(Cl)cc23)cc1
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)Nc1ccc(OC(F)(F)F)cc1
Cc1c(Cl)cccc1NS(=O)(=O)c1ccc(cc1)-c1c(C)c(CC(O)=O)cc2ccc(Cl)cc12
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)Nc1cccc(Cl)c1
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)N1CCCC1
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)N1CCCCC1
CCN(CC)S(=O)(=O)c1ccc(cc1)-c1c(C)c(CC(O)=O)cc2ccc(Cl)cc12
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)NC1CCCCC1
CC(C)NS(=O)(=O)c1ccc(cc1)-c1c(C)c(CC(O)=O)cc2ccc(Cl)cc12
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)NCc1ccccc1
COc1ccc(CNS(=O)(=O)c2ccc(cc2)-c2c(C)c(CC(O)=O)cc3ccc(Cl)cc23)cc1
COc1ccc(CN(C(C)C)S(=O)(=O)c2ccc(cc2)-c2c(C)c(CC(O)=O)cc3ccc(Cl)cc23)cc1
Cc1ccc(NS(=O)(=O)c2ccc(cc2)-c2c(C)c(CC(O)=O)cc3ccc(F)cc23)cc1
Cc1c(Cl)cccc1NS(=O)(=O)c1ccc(cc1)-c1c(C)c(CC(O)=O)cc2ccc(F)cc12
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(=O)(=O)Nc1cccc(Cl)c1
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(=O)(=O)N1CCCC1
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(=O)(=O)N1CCCCC1
CCN(CC)S(=O)(=O)c1ccc(cc1)-c1c(C)c(CC(O)=O)cc2ccc(F)cc12
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(=O)(=O)NC1CCCCC1
CC(C)NS(=O)(=O)c1ccc(cc1)-c1c(C)c(CC(O)=O)cc2ccc(F)cc12
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(=O)(=O)NCc1ccccc1
COc1ccc(CNS(=O)(=O)c2ccc(cc2)-c2c(C)c(CC(O)=O)cc3ccc(F)cc23)cc1
COc1ccc(CN(C(C)C)S(=O)(=O)c2ccc(cc2)-c2c(C)c(CC(O)=O)cc3ccc(F)cc23)cc1
Cc1c(CC(O)=O)cc2ccc(Cl)cc2c1-c1ccc(cc1)S(=O)(=O)NCCO
Cc1c(CC(O)=O)cc2ccc(F)cc2c1-c1ccc(cc1)S(=O)(=O)NCCO
CN(C1CCc2c(CC(O)=O)c3ccccc3n2C1)c1ncc(Cl)cn1
CN(C1CCc2c(CC(O)=O)c3ccccc3n2C1)c1ncc(F)cn1
CN(C1CCc2c(CC(O)=O)c3ccccc3n2C1)c1ncc(cn1)C(F)(F)F
CN(C1CCc2c(CC(O)=O)c3ccccc3n2C1)c1nc2ccc(F)cc2s1
CN(C1CCc2c(CC(O)=O)c3ccccc3n2C1)c1nc2cc(F)ccc2o1
CN(C1CCc2c(CC(O)=O)c3ccccc3n2C1)c1nc2cc(F)ccc2s1
CN(C1CCc2c(CC(O)=O)c3cc(F)ccc3n2C1)c1ncc(F)cn1
CN(C1CCc2c(CC(O)=O)c3cc(F)ccc3n2C1)c1nc2cc(F)ccc2o1
CN(C1CCc2c(CC(O)=O)c3ccc(F)cc3n2C1)c1ncc(F)cn1
CN(C1CCc2c(CC(O)=O)c3ccc(F)cc3n2C1)c1nc2cc(F)ccc2o1
COc1ccc2n3CC(CCc3c(CC(O)=O)c2c1)N(C)c1ncc(F)cn1
COc1ccc2n3CC(CCc3c(CC(O)=O)c2c1)N(C)c1nc2cc(F)ccc2o1
CN(C1CCc2c(CC(O)=O)c3cc(C)ccc3n2C1)c1ncc(F)cn1
CN(C1CCc2c(CC(O)=O)c3cc(C)ccc3n2C1)c1nc2cc(F)ccc2o1
CN(C1CCc2c(CC(O)=O)c3cc(Cl)ccc3n2C1)c1ncc(F)cn1
CN(C1CCc2c(CC(O)=O)c3cc(Cl)ccc3n2C1)c1nc2cc(F)ccc2o1
CN(C1CCc2c(CC(O)=O)c3ccc(F)cc3n2C1)c1ncc(Cl)cn1
CN(C1CCc2c(CC(O)=O)c3ccc(F)cc3n2C1)c1ncc(cn1)C(F)(F)F
CN(C1CCc2c(CC(O)=O)c3ccc(F)cc3n2C1)c1nc2cc(F)ccc2s1
CN(C1CCc2c(CC(O)=O)c3ccc(F)cc3n2C1)c1nc2ccc(F)cc2o1
CN(C1CCc2c(CC(O)=O)c3ccc(Cl)cc3n2C1)c1ncc(Cl)cn1
CN(C1CCc2c(CC(O)=O)c3ccc(cc3n2C1)C(F)(F)F)c1ncc(Cl)cn1
CN(C1CCc2c(CC(O)=O)c3cc(OC(F)(F)F)ccc3n2C1)c1ncc(Cl)cn1
CN(C1CCc2c(CC(O)=O)c3ccc(cc3n2C1)C(F)(F)F)c1ncc(F)cn1
CN(C1CCc2c(CC(O)=O)c3cc(OC(F)(F)F)ccc3n2C1)c1ncc(F)cn1
CN(C1CCc2c(CC(O)=O)c3ccc(cc3n2C1)C(F)(F)F)c1nc2ccc(F)cc2s1
CN(C1CCc2c(CC(O)=O)c3cc(OC(F)(F)F)ccc3n2C1)c1nc2ccc(F)cc2s1
CN(C1CCc2c(CC(O)=O)c3ccc(cc3n2C1)C(F)(F)F)c1nc2cc(F)ccc2o1
CN(C1CCc2c(CC(O)=O)c3cc(OC(F)(F)F)ccc3n2C1)c1nc2cc(F)ccc2o1
CN(C1CCc2c(CC(O)=O)c3ccc(Cl)cc3n2C1)c1ncc(F)cn1
CN(C1CCc2c(CC(O)=O)c3ccc(Cl)cc3n2C1)c1nc2cc(F)ccc2o1
CN([C@H]1CCc2c(CC(O)=O)c3ccc(Cl)cc3n2C1)c1ncc(F)cn1
CN([C@@H]1CCc2c(CC(O)=O)c3ccc(Cl)cc3n2C1)c1ncc(F)cn1
OC(=O)Cc1c2CCC(Cn2c2cc(F)ccc12)Nc1ncc(F)cn1
OC(=O)Cc1c2CCC(Cn2c2cc(F)ccc12)Nc1nc2cc(F)ccc2o1
OC(=O)Cc1c2CCC(Cn2c2cc(Cl)ccc12)Nc1ncc(F)cn1
OC(=O)Cc1c2CCC(Cn2c2cc(Cl)ccc12)Nc1ncc(Cl)cn1
CN(C1CCc2c(CC(O)=O)c3ccc(Cl)cc3n2C1)c1ncc(C)cn1
CN(C1CCc2c(CC(O)=O)c3ccc(Cl)cc3n2C1)c1ncc2ccccc2n1
CN(C1CCc2c(CC(O)=O)c3ccc(Cl)cc3n2C1)c1ncc2cc(F)ccc2n1
CN(C1CCc2c(CC(O)=O)c3ccc(Cl)cc3n2C1)c1ncc2ccc(F)cc2n1
CN(C1CCc2c(CC(O)=O)c3ccc(Cl)cc3n2C1)c1nc(C)nc2ccccc12
CN(C1CCc2c(CC(O)=O)c3ccc(Cl)cc3n2C1)c1cnc2cc(F)ccc2n1
OC(=O)Cc1c2CCC(Cn2c2cc(Cl)ccc12)N(CC(F)F)c1nc2cc(F)ccc2o1
CCN(C1CCc2c(CC(O)=O)c3ccc(Cl)cc3n2C1)c1ncc(F)cn1
CC(C)N(C1CCc2c(CC(O)=O)c3ccc(Cl)cc3n2C1)c1nc2cc(F)ccc2o1
COCCN(C1CCc2c(CC(O)=O)c3ccc(Cl)cc3n2C1)c1ncc(F)cn1
CC(C)CN(C1CCc2c(CC(O)=O)c3ccc(Cl)cc3n2C1)c1nc2cc(F)ccc2o1
CCCN(C1CCc2c(CC(O)=O)c3ccc(Cl)cc3n2C1)c1ncc(F)cn1
CCN(C1CCc2c(CC(O)=O)c3ccc(Cl)cc3n2C1)c1nc2cc(F)ccc2o1
OC(=O)Cc1c2CCC(Cn2c2cc(Cl)ccc12)N(CC1CC1)c1ncc(F)cn1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)NCc1ccccc1F
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)NCc1cccc(F)c1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)NCc1ccc(F)cc1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)NCc1ccccc1
OC(=O)COc1ccc(Cl)cc1[C@H]1N(CCc2ncsc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
OC(=O)COc1ccc(Cl)cc1[C@H]1N(CCc2ncsc12)C(=O)[C@H]1C[C@@H]1c1ccccc1
OC(=O)COc1ccc(Cl)cc1[C@H]1N(CCc2ncsc12)C(=O)[C@@H]1C[C@H]1c1cccc(F)c1
OC(=O)COc1ccc(Cl)cc1[C@H]1N(CCc2ncsc12)C(=O)[C@@H]1C[C@H]1c1ccc(F)cc1
OC(=O)COc1ccc(Cl)cc1[C@H]1N(CCc2ncsc12)C(=O)[C@H]1C[C@@H]1c1ccc(F)cc1
Cc1nc2CCN([C@@H](c2s1)c1cc(Cl)ccc1OCC(O)=O)C(=O)[C@@H]1C[C@H]1c1ccccc1
Cc1nc2CCN([C@H](c2s1)c1cc(Cl)ccc1OCC(O)=O)C(=O)[C@@H]1C[C@H]1c1ccccc1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2nc(sc12)C(F)(F)F)C(=O)OCc1ccccc1
CC(C)c1nc2CCN(C(c2s1)c1cc(Cl)ccc1OCC(O)=O)C(=O)OCc1ccccc1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2nc(sc12)C1CC1)C(=O)OCc1ccccc1
Cc1nc2CCN(C(c2s1)c1cc(Cl)ccc1OCC(O)=O)C(=O)OCc1ccccc1
CCc1nc2CCN(C(c2s1)c1cc(Cl)ccc1OCC(O)=O)C(=O)OCc1ccccc1
Nc1nc2CCN(C(c2s1)c1cc(Cl)ccc1OCC(O)=O)C(=O)OCc1ccccc1
Cc1nc2CCN([C@H](c2s1)c1cc(Cl)ccc1OCC(O)=O)C(=O)OCc1ccccc1
Cc1nc2CCN([C@@H](c2s1)c1cc(Cl)ccc1OCC(O)=O)C(=O)OCc1ccccc1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2nc(Br)sc12)C(=O)OCc1ccccc1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)CCOc1ccc(F)cc1
OC(=O)COc1ccc(Cl)cc1[C@@H]1N(CCc2ncsc12)C(=O)C1CC1c1ccccc1
OC(=O)COc1ccc(Cl)cc1[C@@H]1N(CCc2ncsc12)C(=O)C1CC1c1ccccc1C(F)(F)F
OC(=O)COc1ccc(Cl)cc1[C@@H]1N(CCc2ncsc12)C(=O)C1CC1c1ccccc1Cl
Cc1ccccc1C1CC1C(=O)N1CCc2ncsc2[C@@H]1c1cc(Cl)ccc1OCC(O)=O
COc1ccc2[nH]cc(CCC(=O)N3CCc4ncsc4C3c3cc(Cl)ccc3OCC(O)=O)c2c1
Cc1[nH]c2ccccc2c1CCC(=O)N1CCc2ncsc2C1c1cc(Cl)ccc1OCC(O)=O
Cn1cc(CCC(=O)N2CCc3ncsc3C2c2cc(Cl)ccc2OCC(O)=O)c2ccccc12
Cc1ccccc1CCC(=O)N1CCc2ncsc2C1c1cc(Cl)ccc1OCC(O)=O
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)CCCc1ccccc1F
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)COCc1ccccc1Cl
Cc1ccc(OCC(=O)N2CCc3ncsc3C2c2cc(Cl)ccc2OCC(O)=O)c(C)n1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)CCn1ncc2ccccc12
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)COc1ccccc1
C[C@@H](CC(=O)N1CCc2ncsc2C1c1cc(Cl)ccc1OCC(O)=O)c1ccccc1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)C1Cc2ccccc2C1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)CC1(CC1)c1ccccc1
C[C@H](CC(=O)N1CCc2ncsc2C1c1cc(Cl)ccc1OCC(O)=O)c1ccccc1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)CC1OCCc2ccccc12
CC(C)(C)CC(=O)N1CCc2ncsc2C1c1cc(Cl)ccc1OCC(O)=O
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)CC1CC1
Cc1noc(C)c1CCC(=O)N1CCc2ncsc2C1c1cc(Cl)ccc1OCC(O)=O
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)C1CC1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)Cc1n[nH]c2ccccc12
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)\C=C\c1ccccc1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)CC1Cc2ccccc2C1
CC1(C)CC1C(=O)N1CCc2ncsc2C1c1cc(Cl)ccc1OCC(O)=O
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)CC1CCCCC1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)Cc1ccc2ccccc2c1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)Cc1cccc2ccccc12
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)CCCc1ccc(F)cc1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)CCN1CCc2ccccc12
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)CCN1CCCc2ccccc12
COc1ccc(\C=C\C(=O)N2CCc3ncsc3C2c2cc(Cl)ccc2OCC(O)=O)cc1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)\C=C\c1ccc(F)cc1
Cc1ccc(\C=C\C(=O)N2CCc3ncsc3C2c2cc(Cl)ccc2OCC(O)=O)cc1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)\C=C\c1ccc(F)cc1F
OC(=O)COc1ccc(Cl)cc1[C@H]1N(CCc2ncsc12)C(=O)OCc1cc(F)ccc1F
OC(=O)COc1ccc(Cl)cc1[C@H]1N(CCc2ncsc12)C(=O)OCc1ccc(F)cc1F
CCC(C)(C)COC(=O)N1CCc2ncsc2[C@H]1c1cc(Cl)ccc1OCC(O)=O
OC(=O)COc1ccc(Cl)cc1[C@H]1N(CCc2ncsc12)C(=O)OCc1ccc(F)cc1
COC(C)(C)CCOC(=O)N1CCc2ncsc2[C@H]1c1cc(Cl)ccc1OCC(O)=O
Cc1ccc(COC(=O)N2CCc3ncsc3[C@H]2c2cc(Cl)ccc2OCC(O)=O)c(C)c1
OC(=O)COc1ccc(Cl)cc1[C@H]1N(CCc2ncsc12)C(=O)OCc1cc(F)ccc1Cl
CC(C)(C)CCOC(=O)N1CCc2ncsc2[C@H]1c1cc(Cl)ccc1OCC(O)=O
OC(=O)COc1ccc(Cl)cc1[C@H]1N(CCc2ncsc12)C(=O)OCC1CCCCC1
CC(C)CCOC(=O)N1CCc2ncsc2[C@H]1c1cc(Cl)ccc1OCC(O)=O
OC(=O)COc1ccc(Cl)cc1[C@H]1N(CCc2ncsc12)C(=O)OCc1cc(Cl)ccc1F
OC(=O)COc1ccc(Cl)cc1[C@H]1N(CCc2ncsc12)C(=O)OCC1CCC1
CCC(C)COC(=O)N1CCc2ncsc2[C@H]1c1cc(Cl)ccc1OCC(O)=O
OC(=O)COc1ccc(Cl)cc1[C@H]1N(CCc2ncsc12)C(=O)OCc1cccc(F)c1F
Cc1cccc(COC(=O)N2CCc3ncsc3[C@H]2c2cc(Cl)ccc2OCC(O)=O)c1C
OC(=O)COc1ccc(Cl)cc1[C@H]1N(CCc2ncsc12)C(=O)OCc1c(F)cccc1F
OC(=O)COc1ccc(Cl)cc1[C@H]1N(CCc2ncsc12)C(=O)OCCCF
OC(=O)COc1ccc(Cl)cc1[C@H]1N(CCc2ncsc12)C(=O)OCc1ccccc1F
OC(=O)COc1ccc(Cl)cc1[C@H]1N(CCc2ncsc12)C(=O)OCc1cccc(F)c1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCCc1cccc(F)c1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1cccc(F)c1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1ccccc1F
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1ccc(F)cc1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1cccc(Cl)c1Cl
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1cccc(F)c1F
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1ccc(F)cc1F
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1ccccc1Cl
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1cccc(Cl)c1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1ccc(Cl)cc1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1c(Cl)cccc1Cl
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCCc1ccccc1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1c(F)cccc1F
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCn1ncc2ccccc12
CCn1nc(C)cc1CCOC(=O)N1CCc2ncsc2C1c1cc(Cl)ccc1OCC(O)=O
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1cc(F)ccc1Cl
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1cc(F)ccc1F
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1ccc(Cl)cc1Cl
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1cnccn1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCC1CCCCC1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1nc2ccccc2o1
CC(C)COC(=O)N1CCc2ncsc2C1c1cc(Cl)ccc1OCC(O)=O
CCCCOC(=O)N1CCc2ncsc2C1c1cc(Cl)ccc1OCC(O)=O
Cc1ccc(COC(=O)N2CCc3ncsc3C2c2cc(Cl)ccc2OCC(O)=O)c(C)c1
Cc1cccc(COC(=O)N2CCc3ncsc3C2c2cc(Cl)ccc2OCC(O)=O)c1C
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1cc(Cl)ccc1F
OC(=O)COc1ccc(Cl)cc1[C@H]1N(CCc2ncsc12)C(=O)OCc1ccccc1
OC(=O)COc1ccc(Cl)cc1[C@@H]1N(CCc2ncsc12)C(=O)OCc1ccccc1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1ccccc1
OC(=O)COc1ccc(cc1C1N(CCc2ncsc12)C(=O)OCc1ccccc1)C#N
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)NCCc1ccccc1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)NCc1ccccc1Cl
COc1ccccc1CNC(=O)N1CCc2ncsc2C1c1cc(Cl)ccc1OCC(O)=O
COc1ccccc1CNC(=S)N1CCc2ncsc2C1c1cc(Cl)ccc1OCC(O)=O
CCCc1nc2CCN(C(c2s1)c1cc(Cl)ccc1OCC(O)=O)C(=O)OCc1ccccc1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2nc(sc12)-c1ccccc1)C(=O)OCc1ccccc1
CS(=O)(=O)Nc1nc2CCN(C(c2s1)c1cc(Cl)ccc1OCC(O)=O)C(=O)OCc1ccccc1
OC(=O)COc1ccc(Cl)cc1N(C1N(CCc2ncsc12)C(=O)OCc1ccccc1)S(=O)(=O)C1CC1
OC(=O)COc1ccc(Cl)cc1C1N(CCc2nc(NC(=O)C3CC3)sc12)C(=O)OCc1ccccc1
CC(=O)Nc1nc2CCN(C(c2s1)c1cc(Cl)ccc1OCC(O)=O)C(=O)OCc1ccccc1
CN(C)c1nc2CCN(C(c2s1)c1cc(Cl)ccc1OCC(O)=O)C(=O)OCc1ccccc1
OC(=O)COc1ccc(F)cc1C1N(CCc2ncsc12)C(=O)OCc1ccccc1
C[C@@H](Oc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1ccccc1)C(O)=O
C[C@H](Oc1ccc(Cl)cc1C1N(CCc2ncsc12)C(=O)OCc1ccccc1)C(O)=O
Cc1nn(Cc2ccc(cc2)-c2cc3ccc(Cl)cc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2cc3cc(ccc3[nH]2)C(F)(F)F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2cc3cc(Cl)ccc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2cc3ccc(cc3[nH]2)C(F)(F)F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2F)-c2cc3ccc(cc3[nH]2)C(F)(F)F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2F)-c2cc3ccc(Cl)cc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2cccc(c2)-c2cc3ccc(Cl)cc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccccc2-c2cc3ccc(Cl)cc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2cccc(c2)-c2cc3ccc(cc3[nH]2)C(F)(F)F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2cc3ncccc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2C(F)(F)F)-c2cc3ccc(cc3[nH]2)C(F)(F)F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2F)-c2cc3cccnc3[nH]2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)-c2nc3cccnc3[nH]2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3ccccc3[nH]2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3ccccc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3cc(Cl)c(Cl)cc3[nH]2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3cc(Cl)c(Cl)cc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3cc4ccccc4cc3[nH]2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3cc4ccccc4cc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3ccc(cc3[nH]2)C(F)(F)F)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3ccc(cc3[nH]2)C(F)(F)F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(-c3nc4ccccc4[nH]3)c(C)c2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3cc(Cl)c(Cl)cc3[nH]2)c(C2CC2)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3cc(Cl)ccc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3cc(Cl)ccc3n2C)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3cncc(C)c3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3cc(F)c(Cl)cc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3cc(Br)c(Cl)cc3[nH]2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3c(C)cncc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3ccccc3n2C)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3cccnc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3cc(Br)ccc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3cc(ccc3[nH]2)C(C)(C)C)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3cc(ccc3[nH]2)C#N)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3cc(Cl)c(Cl)cc3n2C)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3c(F)cc(F)cc3[nH]2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3cncnc3[nH]2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3cc(Br)cnc3[nH]2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3cc(OC)ccc3[nH]2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3cc(Cl)cnc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3cc(C)ccc3[nH]2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3cc(Cl)cnc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3c(F)c(F)ccc3[nH]2)c(CC)c1CC(O)=O
COc1ccc2[nH]c(nc2n1)-c1ccc(Cn2nc(C)c(CC(O)=O)c2C)cc1
CCc1nn(Cc2ccc(cc2)-c2nc3cc(Cl)ccc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3ccccc3n2C)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3c(F)c(F)ccc3[nH]2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3cccnc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3c(F)cc(F)cc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3c(C)cccc3[nH]2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3c(F)cccc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3cc(F)c(Cl)cc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3cc(C)c(Cl)cc3[nH]2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3cc(C)c(Cl)cc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3cc(F)ccc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3cc(Br)cnc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3cc(C)ccc3[nH]2)c(CC)c1CC(O)=O
COc1ccc2[nH]c(nc2c1)-c1ccc(Cn2nc(C)c(CC(O)=O)c2C)cc1
Cc1nn(Cc2ccc(cc2)-c2nc3ccncc3[nH]2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3ccncc3[nH]2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3cc(ccc3[nH]2)C#N)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3c(C)cccc3[nH]2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3nc(OC)ccc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3c(Cl)cc(Cl)cc3[nH]2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3c(Cl)cc(Cl)cc3[nH]2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3c(F)cccc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3cc(ccc3[nH]2)C(C)(C)C)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2)-c2nc3cc(Cl)ccc3n2C)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3cncnc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2)-c2nc3cc(F)ccc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2F)-c2nc3ccncc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2F)-c2nc3c(Cl)cc(Cl)cc3[nH]2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)-c2nc3c(F)cccc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)-c2nc3cc(OC)ccc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)-c2nc3cc(F)c(Cl)cc3[nH]2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(cc2F)-c2nc3c(F)cc(F)cc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2F)-c2nc3cc(ccc3[nH]2)C#N)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)-c2nc3nc(OC)ccc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)-c2nc3cc(Cl)ccc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)-c2nc3cc(ccc3[nH]2)C#N)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)-c2nc3cc(F)ccc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)-c2nc3c(C)cccc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)-c2nc3c(F)c(F)ccc3[nH]2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(cc2F)-c2nc3cncc(C)c3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2F)-c2nc3cc(F)ccc3[nH]2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)-c2nc3cc(Br)ccc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)-c2nc3cc(ccc3[nH]2)C(C)(C)C)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)-c2nc3cc(Br)cnc3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)-c2nc3ccncc3[nH]2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(cc2F)-c2nc3cc(C)ccc3[nH]2)c(C)c1CC(O)=O
COc1ccc2[nH]c(nc2n1)-c1ccc(Cn2nc(C)c(CC(O)=O)c2C)c(F)c1
Cc1nn(Cc2ccc(cc2F)-c2nc3c(C)cccc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2F)-c2nc3cc(Br)ccc3[nH]2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)-c2nc3cc(Cl)cnc3[nH]2)c(CC)c1CC(O)=O
COc1ccc2[nH]c(nc2c1)-c1ccc(Cn2nc(C)c(CC(O)=O)c2C)c(F)c1
Cc1nn(Cc2ccc(cc2F)-c2nc3cc(ccc3[nH]2)C(C)(C)C)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2F)-c2nc3c(F)cccc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2F)-c2nc3cc(Cl)cnc3[nH]2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)-c2nc3c(F)cc(F)cc3[nH]2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(cc2F)-c2nc3cc(F)c(Cl)cc3[nH]2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)-c2nc3cncc(C)c3[nH]2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)-c2nc3c(Cl)cc(Cl)cc3[nH]2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(cc2F)-c2nc3c(F)c(F)ccc3[nH]2)c(C)c1CC(O)=O
CCc1nn(Cc2ccc(cc2F)-c2nc3cc(C)c(Cl)cc3[nH]2)c(CC)c1CC(O)=O
Cc1nn(Cc2ccc(cc2F)-c2nc3cccnc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2F)-c2nc3cc(Cl)ccc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2F)-c2nc3cc(C)c(Cl)cc3[nH]2)c(C)c1CC(O)=O
Cc1nn(Cc2cccc(c2)-c2nc3cc(ccc3[nH]2)C(F)(F)F)c(C)c1CC(O)=O
Cc1nn(Cc2ccc(cc2F)-c2nc3cc(ccc3[nH]2)C(F)(F)F)c(C)c1CC(O)=O
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccc(F)cc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccc(Cl)cc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1Cl
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1F
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1CC1c1ccccc1C
Cc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1ccc(c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1)C(F)(F)F
OC(=O)Cc1ccc(Cl)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1ccc(F)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1cc(ccc1Cl)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1cc(ccc1F)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1ccc(cc1CC(O)=O)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1cc(F)cc(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1cc(CC(O)=O)cc(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1cccc(c1F)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(CCc12)C(=O)OCc1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1cc(Cl)cc(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
CS(=O)(=O)c1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1ccc(OC(F)(F)F)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
CC(C)Oc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1ccc(F)c(c1)-c1cccc2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1cccc(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(c2CCN(Cc12)C(=O)OCc1ccccc1)S(C)(=O)=O
OC(=O)Cc1ccc(OC(F)(F)F)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
CC(C)Oc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
OC(=O)Cc1ccc(Cl)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
CS(=O)(=O)c1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
OC(=O)Cc1ccccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1ccc(CC(O)=O)cc1-c1cc(F)c(F)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1ccc(CC(O)=O)cc1-c1cc(F)cc2CCN(Cc12)C(=O)OCc1ccccc1
COc1ccc(CC(O)=O)cc1-c1c(F)ccc2CCN(Cc12)C(=O)OCc1ccccc1 |(4,-5.39,;2.67,-4.62,;1.33,-5.39,;1.33,-6.93,;,-7.7,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-1.33,-10.01,;-1.33,-5.39,;,-4.62,;,-3.08,;-1.33,-2.31,;-2.67,-3.08,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;2.67,-3.08,;1.33,-2.31,;5.33,-3.08,;6.67,-2.31,;5.33,-4.62,;6.67,-5.39,;8,-4.62,;8,-3.08,;9.34,-2.31,;10.67,-3.08,;10.67,-4.62,;9.34,-5.39,)|
COc1ccc(CC(O)=O)cc1-c1cc(F)cc2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
COc1ccc(CC(O)=O)cc1-c1c(F)ccc2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1 |wU:25.27,wD:27.31,(4,-5.39,;2.67,-4.62,;1.33,-5.39,;1.33,-6.93,;,-7.7,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-1.33,-10.01,;-1.33,-5.39,;,-4.62,;,-3.08,;-1.33,-2.31,;-2.67,-3.08,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;2.67,-3.08,;1.33,-2.31,;5.33,-3.08,;6.67,-2.31,;5.33,-4.62,;4.56,-5.95,;6.1,-5.95,;7.44,-6.72,;8.77,-5.95,;10.11,-6.72,;10.11,-8.26,;8.77,-9.03,;7.44,-8.26,)|
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(CCc12)C(=O)C1CC1c1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CN(Cc12)C(=O)C1CC1c1ccccc1
COc1ccc(CC(O)=O)cc1-c1c(F)cc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1 |wU:26.28,wD:28.32,(4,-5.39,;2.67,-4.62,;1.33,-5.39,;1.33,-6.93,;,-7.7,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-1.33,-10.01,;-1.33,-5.39,;,-4.62,;,-3.08,;-1.33,-2.31,;-2.67,-3.08,;-1.33,-.77,;;,1.54,;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;2.67,-3.08,;1.33,-2.31,;5.33,-3.08,;6.67,-2.31,;5.33,-4.62,;4.56,-5.95,;6.1,-5.95,;7.44,-6.72,;8.77,-5.95,;10.11,-6.72,;10.11,-8.26,;8.77,-9.03,;7.44,-8.26,)|
COc1ccc(CC(O)=O)cc1-c1c(F)cc(F)c2CCN(Cc12)C(=O)OCc1ccccc1 |(4,-5.39,;2.67,-4.62,;1.33,-5.39,;1.33,-6.93,;,-7.7,;-1.33,-6.93,;-2.67,-7.7,;-2.67,-9.24,;-4,-10.01,;-1.33,-10.01,;-1.33,-5.39,;,-4.62,;,-3.08,;-1.33,-2.31,;-2.67,-3.08,;-1.33,-.77,;;,1.54,;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;2.67,-3.08,;1.33,-2.31,;5.33,-3.08,;6.67,-2.31,;5.33,-4.62,;6.67,-5.39,;8,-4.62,;8,-3.08,;9.34,-2.31,;10.67,-3.08,;10.67,-4.62,;9.34,-5.39,)|
OC(=O)Cc1ccc(cc1Cl)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1ccc(cc1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCOc1ccc(F)cc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)COc1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)COc1ccc(F)cc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCCc1ccccc1F
CCOCC(=O)N1CCc2c(F)ccc(c2C1)-c1cc(CC(O)=O)ccc1OC
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)COC(C)(C)C
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1CC1c1cccc(F)c1
COc1ccc2onc(CC(=O)N3CCc4c(F)ccc(c4C3)-c3cc(CC(O)=O)ccc3OC)c2c1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1C(C)(C)C1(C)C
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1cccnc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1CC1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCN1CCCc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1CC1(C)C
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1ccccc1C
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCn1cc(C)c2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)COCc1ccccc1Cl
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCN1CCc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1CC1c1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1c(C)[nH]c2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1cn(C)c2ccccc12
COc1ccc2[nH]cc(CCC(=O)N3CCc4c(F)ccc(c4C3)-c3cc(CC(O)=O)ccc3OC)c2c1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1cccc(F)c1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCn1ncc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(Cl)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccc(Cl)cc1
COc1ccc(CC(O)=O)cc1-c1ccc(Cl)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1cccc(F)c1
COc1ccc(CC(O)=O)cc1-c1ccc(Cl)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1F
COc1ccc(CC(O)=O)cc1-c1ccc(Cl)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(Cl)c2CCN(Cc12)C(=O)CCn1ncc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(Cl)c2CCN(Cc12)C(=O)COCc1ccccc1Cl
COc1ccc(CC(O)=O)cc1-c1ccc(Cl)c2CCN(Cc12)C(=O)CCCc1ccccc1F
COc1ccc(CC(O)=O)cc1-c1ccc(Cl)c2CCN(Cc12)C(=O)CCc1cn(C)c2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(Cl)c2CCN(Cc12)C(=O)CCc1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(Cl)c2CCN(Cc12)C(=O)CCN1CCCc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(Cl)c2CCN(Cc12)C(=O)CCN1CCc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(Cl)c2CCN(Cc12)C(=O)CCc1c(C)[nH]c2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@H]1C[C@@H]1c1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(c2CCN(Cc12)C(=O)C1CC1)C(F)(F)F
COc1ccc(CC(O)=O)cc1-c1ccc(c2CCN(Cc12)C(=O)C1CC1c1ccccc1)C(F)(F)F
COc1ccc(CC(O)=O)cc1-c1cc(F)c(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)\C=C\c1ccccc1
COc1ccc(\C=C\C(=O)N2CCc3c(F)ccc(c3C2)-c2cc(CC(O)=O)ccc2OC)cn1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)\C=C\c1sc(C)nc1C
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)\C=C\c1nc2ccccc2s1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)\C=C\c1cccnc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)\C=C\c1cc(C)nn1C
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1ccccn1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1cccc(C)n1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1ncccn1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)COc1cccnc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1CC1c1ccccc1C(F)(F)F
COc1ccc(cc1)C1CC1C(=O)N1CCc2c(F)ccc(c2C1)-c1cc(CC(O)=O)ccc1OC
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(c1ccccc1)c1ccc(Cl)cc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1CC1c1ccc(Cl)cc1Cl
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CN(CCc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CN(CCc12)C(=O)CCCc1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CN(CCc12)C(=O)CCc1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CN(CCc12)C(=O)CCOc1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CN(CCc12)C(=O)COCc1ccccc1Cl
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CN(CCc12)C(=O)CCN1CCCc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CN(CCc12)C(=O)CCc1cn(C)c2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C[C@@H](C)c1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C[C@H](C)c1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)(C)c1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C(C)Cc1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1Cc2ccccc2C1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1Cc2ccccc2C1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1CCc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1COc2ccccc2C1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1CC(=O)c2ccccc2C1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1CCc2ccccc2O1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1Cc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCCc1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCC(=O)c1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)Cc1cn(C)c2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)NCc1ccccc1F
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)Cc1noc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1CC(=O)c2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1CCc2ccccc2C1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)Cc1n[nH]c2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCn1nc(C)c2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCn1ncc2cc(F)ccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCCCC1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1(O)CCCCC1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)(C)C
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)NCc1cccc(F)c1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)NCc1ccc(F)cc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)NCCc1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)NCc1ccccc1Cl
COc1ccccc1CNC(=O)N1CCc2c(F)ccc(c2C1)-c1cc(CC(O)=O)ccc1OC
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)NCc1ccccc1
CCCNC(=O)N1CCc2c(F)ccc(c2C1)-c1cc(CC(O)=O)ccc1OC
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1cccc(F)c1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccc(F)cc1
COc1ccc(cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1F)C(C)C(O)=O
CCOC(=O)N1CCc2c(F)ccc(c2C1)-c1cc(CC(O)=O)ccc1OC
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCC(C)C
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OC(C)C
OC(=O)COc1cc(Cl)cc(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)COc1ccc(Cl)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1F
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1cccc(F)c1F
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccnn1C
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1cc(C)nn1C
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1csc(C)n1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1cnc(C)s1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1cncnc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCCc1scnc1C
COc1ccc(CC(O)=O)cc1-c1ccc(Cl)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(C)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1ccc(c2CN(CCc12)C(=O)OCc1ccccc1)-c1cc(CC(O)=O)ccc1OC
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(c2CCN(Cc12)C(=O)OCc1ccccc1)C(F)(F)F
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CN(CCc12)C(=O)OCc1ccccc1
OC(=O)COc1ccc(OC(F)(F)F)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
CC(C)Oc1ccc(OCC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
OC(=O)COc1ccc(OC(F)(F)F)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
CC(C)Oc1ccc(OCC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1ccc(c(F)c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1ccc(c(Cl)c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1cc2OCOc2c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1cc2OCCOc2c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(C#N)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1ccc(CC(O)=O)cc1-c1cccc2CCN(Cc12)C(=O)OCc1ccccc1
COc1ccc(cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1)C(C)C(O)=O
OC(=O)COc1ccc(cc1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)COc1ccc(F)cc1-c1cccc2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)CCCOc1ccc(F)cc1-c1cccc2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)COc1cccc(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)COc1ccc(Cl)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1ccc(OCC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)COc1ccc(Cl)c(c1)-c1ccc(Cl)c2CCN(Cc12)C(=O)OCc1ccccc1
Cc1ccc(c2CN(CCc12)C(=O)OCc1ccccc1)-c1cc(OCC(O)=O)ccc1Cl
OC(=O)COc1ccc(Cl)c(c1)-c1ccc(c2CCN(Cc12)C(=O)OCc1ccccc1)C(F)(F)F
OC(=O)COc1ccc(Cl)c(c1)-c1cccc2CCN(Cc12)C(=O)OCc1ccccc1
COc1ccc(OCC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
COc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1cn(C)c2ccccc12
COc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
COc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CCCc1ccccc1F
COc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1c(C)[nH]c2ccccc12
COc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CCCc1ccccc1
COc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)(C)c1ccccc1
COc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)C[C@@H](C)c1ccccc1
COc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CCn1ncc2cc(F)ccc12
COc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CCN1CCc2ccccc12
COc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CCOc1ccc(F)cc1
COc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)COCc1ccccc1Cl
COc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1ccccc1C
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1ccc(OCC2CC2)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
CCCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
CC(C)COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
COCCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCOc2ccccc12
COc1cc(OC(C)C(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)c1ccccn1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1OCCc2ccccc12
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1COc2ccccc12
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1COCc2ccccc12
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)c1ccc(F)cc1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C(C)Cc1ccccc1
CCCc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
CC(C)c1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
CC(C)Oc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1cc(CC(O)=O)cc(OC)c1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1 |(4,-5.39,;2.67,-4.62,;1.33,-5.39,;1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-10.01,;-1.33,-11.55,;-2.67,-9.24,;-1.33,-6.93,;-1.33,-5.39,;-2.67,-4.62,;-2.67,-3.08,;,-4.62,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;,1.54,;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;2.67,-3.08,;1.33,-2.31,;5.33,-3.08,;6.67,-2.31,;5.33,-4.62,;6.67,-5.39,;8,-4.62,;8,-3.08,;9.34,-2.31,;10.67,-3.08,;10.67,-4.62,;9.34,-5.39,)|
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCc2ccccc12
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C[C@@H](C)c1ccccc1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1(CC1)c1ccccc1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)(C)c1ccc(F)cc1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1OCCc2ccccc12
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)(C)c1ccccc1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCOc2ccccc12
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1(CC1)c1ccccc1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1COCc2ccccc12
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCc2ccccc12
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)C[C@@H](C)c1ccccc1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1COc2ccccc12
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCOc2ccccc12
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)(C)c1ccc(F)cc1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)(C)c1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1(C)CCCc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CC(C)(C)Oc2ccccc12
COc1cccc2CCC(Cc12)C(=O)N1CCc2c(F)ccc(c2C1)-c1cc(CC(O)=O)ccc1OC
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1COc2ccccc2C1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCOc2cc(F)ccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCOc2ccc(F)cc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)C1CC1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCOc2c(F)cccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCCc2ccncc12
COc1cccc(n1)C(C)CC(=O)N1CCc2c(F)ccc(c2C1)-c1cc(CC(O)=O)ccc1OC
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)c1cccc(C)n1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1(CCC1)c1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1(CCC1)c1ccc(F)cc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)(C)c1cccc(F)c1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CN(C)C(c1ccccc1)c1ccc(Cl)cc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CC1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@H](C)c1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)(O)c1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1OCCc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1(CC1)c1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1N(C)CCc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCc2ccccc2C1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCOc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCCc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C(C)C)c1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)c1ccccn1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)c1cccnc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)c1ccncc1
CCC(CC(=O)N1CCc2c(F)ccc(c2C1)-c1cc(CC(O)=O)ccc1OC)c1ccccc1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1CCCc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1COc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1COCc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1CCOc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1OCCc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1Cc2ccccc2CO1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1(CC1)c1cccc(F)c1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1(CC1)c1ccccc1F
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1(CC1)c1ccc(F)cc1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)c1cccc(F)c1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)c1ccccc1F
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)c1cnccn1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)c1ccccc1OC
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)c1nccs1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CC(C)(C)Oc2ncccc12
OC(=O)Cc1ccc(c(OCC(F)(F)F)c1)-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCOc2ccccc12
CC(C)(CC(=O)N1CCc2c(F)ccc(c2C1)-c1ccc(CC(O)=O)cc1OCC(F)(F)F)c1ccccc1
C[C@@H](CC(=O)N1CCc2c(F)ccc(c2C1)-c1ccc(CC(O)=O)cc1OCC(F)(F)F)c1ccccc1
CC(CC(=O)N1CCc2c(F)ccc(c2C1)-c1ccc(CC(O)=O)cc1OCC(F)(F)F)c1ccccn1
OC(=O)Cc1ccc(c(OCC(F)(F)F)c1)-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
CC(C)Oc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCOc2ccccc12
CC(C)Oc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)(C)c1ccccc1
CC(C)Oc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C[C@@H](C)c1ccccc1
CC(C)Oc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)c1ccccn1
CC(C)Oc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)c1cccc(C)n1
CC(C)Oc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1cccc(C)n1
CC(C)Oc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1COCc2ccccc12
CC(C)Oc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1OCCc2ccccc12
CC(C)Oc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1COc2ccccc12
OC(=O)Cc1ccc(OCC(F)(F)F)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCOc2ccccc12
CC(C)(CC(=O)N1CCc2c(F)ccc(c2C1)-c1cc(CC(O)=O)ccc1OCC(F)(F)F)c1ccccc1
C[C@H](CC(=O)N1CCc2c(F)ccc(c2C1)-c1cc(CC(O)=O)ccc1OCC(F)(F)F)c1ccccc1
CC(CC(=O)N1CCc2c(F)ccc(c2C1)-c1cc(CC(O)=O)ccc1OCC(F)(F)F)c1ccccn1
CC(CC(=O)N1CCc2c(F)ccc(c2C1)-c1cc(CC(O)=O)ccc1OCC(F)(F)F)c1cccc(C)n1
Cc1cccc(CCC(=O)N2CCc3c(F)ccc(c3C2)-c2cc(CC(O)=O)ccc2OCC(F)(F)F)n1
OC(=O)Cc1ccc(OCC(F)(F)F)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)CC1COCc2ccccc12
OC(=O)Cc1ccc(OCC(F)(F)F)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)CC1OCCc2ccccc12
OC(=O)Cc1ccc(OCC(F)(F)F)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)CC1COc2ccccc12
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(CC)c1ccccn1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1ncccc1OC
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1ccc(F)cc1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1cccc(F)c1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1ccccc1F
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(CC)c1ccccn1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1ncccc1OC
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1ccc(F)cc1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1cccc(F)c1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1ccccc1F
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C1CC1)c1ccccn1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C1CC1)c1ccccn1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)c1cccc(C)n1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1cccc(C)n1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)C1CC1c1ccccn1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CC(C)(C)Oc2ccccc12
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1COc2ccccc2C1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)C1CCc2cccc(OC)c2C1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1(C)CCCc2ccccc12
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCOc2cc(F)ccc12
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)c1cccc(C)n1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1cccc(C)n1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1CC1c1ccccn1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CC(C)(C)Oc2ccccc12
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1COc2ccccc2C1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1CCc2cccc(OC)c2C1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1(C)CCCc2ccccc12
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCOc2cc(F)ccc12
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)\C=C\c1ccccn1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)\C=C\c1ccn(C)n1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)\C=C\c1ccccn1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)\C=C\c1cnn(C)c1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)Cc1ccccn1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)\C=C\c1cnn(C)c1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)Cc1ccccn1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C(C)Cc1cccnc1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)c1ccccn1
CC(C)Oc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)c1ccccn1
C[C@H](CC(=O)N1CCc2c(F)ccc(c2C1)-c1ccc(CC(O)=O)cc1OCC(F)(F)F)c1ccccc1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1ccccn1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CCc1ccccn1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCCc2cccnc12
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C(C)Cc1ccccn1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)C(C)Cc1ccccn1
CC(C)Oc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCOc2ccccc12
CC(C)Oc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)(C)c1ccccc1
CC(C)Oc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)C[C@H](C)c1ccccc1
CC(C)Oc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)C[C@@H](C)c1ccccc1
CC(C)Oc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
COc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)(C)c1ccc(F)cc1
COc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1CCc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)C1CC1c1ccccn1
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC1OCc2ccccc12
COc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)CC(C)(C)c1ccc(F)cc1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)O[C@H](C)c1ccccc1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1cnccn1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ncc(C)cc1F
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)O[C@@H](C)c1ccccc1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCC1CCCC1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCCC(C)C
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1cccc(C)n1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCC1CC1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCCc1ccccc1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OC[C@H](C)c1ccccc1
[#6]-[#6]-[#8]-c1ccc(-[#6]-[#6](-[#8])=O)cc1-c1ccc(F)c2-[#6]-[#6]-[#7](-[#6]-c12)-[#6](=O)-[#8]-[#6]\[#6]=[#6](\[#6])-[#6]
CCCCOC(=O)N1CCc2c(F)ccc(c2C1)-c1cc(CC(O)=O)ccc1OCC
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCC(C)C
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCCOC
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCCC(C)=C
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCC(C)CC
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCCC#C
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCCC(C)(C)O
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCCC(C)(C)OC
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCC1CCCO1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)O[C@H](C)c1ccccc1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1cnccn1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ncc(C)cc1F
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccnn1C
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)O[C@@H](C)c1ccccc1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1cccc(C)n1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCC1CC1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCC1CCCC1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCCC(C)C
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccn1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccn1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCC1CCCCC1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCC1CCCCC1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccc(F)cc1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1cccc(F)c1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1F
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1cc(F)ccc1F
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1cc(Cl)ccc1F
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccc(F)cc1F
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccc(F)cc1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1cccc(F)c1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1F
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1cc(F)ccc1F
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1cc(Cl)ccc1F
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccc(F)cc1F
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1ccc(c(OCC(F)(F)F)c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1ccc(OC(F)F)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1ccc(OCC(F)F)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1ccc(OC(C)C(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
CCC(Oc1ccc(OC)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1)C(O)=O
OC(=O)Cc1ccc(Cl)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1cccc(OCC(O)=O)c1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1 |(-2.67,-3.08,;-2.67,-4.62,;-1.33,-5.39,;-1.33,-6.93,;,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;5.33,-7.7,;,-4.62,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;,1.54,;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;2.67,-3.08,;1.33,-2.31,;5.33,-3.08,;6.67,-2.31,;5.33,-4.62,;6.67,-5.39,;8,-4.62,;8,-3.08,;9.34,-2.31,;10.67,-3.08,;10.67,-4.62,;9.34,-5.39,)|
COc1cccc(CC(O)=O)c1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1 |(4,-5.39,;2.67,-4.62,;1.33,-5.39,;1.33,-6.93,;,-7.7,;-1.33,-6.93,;-1.33,-5.39,;-2.67,-4.62,;-4,-5.39,;-5.33,-4.62,;-4,-6.93,;,-4.62,;,-3.08,;-1.33,-2.31,;-1.33,-.77,;;,1.54,;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;2.67,-3.08,;1.33,-2.31,;5.33,-3.08,;6.67,-2.31,;5.33,-4.62,;6.67,-5.39,;8,-4.62,;8,-3.08,;9.34,-2.31,;10.67,-3.08,;10.67,-4.62,;9.34,-5.39,)|
CC(C)(C)Oc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
CN(C)c1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1ccc(OCC(F)(F)F)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
OC(=O)Cc1ccc(OCCF)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1c(CC(O)=O)cccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
COc1cc(OCC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
CCOc1cc(ccc1-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1)C(C)C(O)=O
OC(=O)Cc1ccc(OCC(F)(F)F)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
OC(=O)Cc1ccc(OCCF)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
CC(C)(C)Oc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1
COc1ccc(cc1-c1ccc(F)c2CCN(Cc12)C(=O)[C@@H]1C[C@H]1c1ccccc1)C1(CC1)C(O)=O
OC(=O)Cc1ccc(OC2CC2)c(c1)-c1ccc(F)c2CCN(Cc12)C(=O)OCc1ccccc1
CC(C)Oc1ccc(CC(O)=O)cc1-c1ccc(C#N)c2CCN(Cc12)C(=O)OCc1ccccc1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)NCc1ccccc1F
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)NCc1cccc(F)c1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)NCc1ccc(F)cc1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)NCCc1ccccc1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)NCc1ccccc1Cl
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)NCc1ccccc1OC
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)NCc1ccccc1
CCCNC(=O)N1CCc2c(F)ccc(c2C1)-c1cc(CC(O)=O)ccc1OCC
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)NCc1ccccc1F
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)NCc1cccc(F)c1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)NCc1ccc(F)cc1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)NCCc1ccccc1
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)NCc1ccccc1Cl
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)NCc1ccccc1OC
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)NCc1ccccc1
CCCNC(=O)N1CCc2c(F)ccc(c2C1)-c1ccc(CC(O)=O)cc1OCC
CCOc1cc(CC(O)=O)ccc1-c1ccc(F)c2CCN(Cc12)C(=O)NCc1ccccn1
CCOc1ccc(CC(O)=O)cc1-c1ccc(F)c2CCN(Cc12)C(=O)NCc1ccccn1
C[C@@H](NC(=O)c1ccc2c(c1)cc(CCCCC(O)=O)n(Cc1ccccc1)c2=O)c1ccc(F)cc1
C[C@@H](NC(=O)c1ccc2c(c1)cc(CCCCC(O)=O)n(Cc1ccc(F)cc1)c2=O)c1ccc(F)cc1
C[C@@H](NC(=O)c1ccc2c(c1)cc(CC(O)=O)n(-c1ccc(F)cc1)c2=O)c1ccc(F)cc1
OC(=O)CCCCc1cc2cc(ccc2c(=O)n1-c1ccc(F)cc1)C(=O)N[C@@H]1CCCc2ccccc12
OC(=O)CCCCc1cc2cc(ccc2c(=O)n1-c1ccc(F)cc1)C(=O)N[C@@H]1CCCc2cc(F)ccc12
COc1ccc(cc1)-n1c(CCCCC(O)=O)cc2cc(ccc2c1=O)C(=O)N[C@H](C)c1ccc(F)cc1
C[C@@H](NC(=O)c1ccc2c(cc(CCCCC(O)=O)n(-c3ccc(cc3)C#N)c2=O)c1)c1ccc(F)cc1
COc1cccc(c1)-n1c(CCCCC(O)=O)cc2cc(ccc2c1=O)C(=O)N[C@H](C)c1ccc(F)cc1
COc1ccccc1-n1c(CCCCC(O)=O)cc2cc(ccc2c1=O)C(=O)N[C@H](C)c1ccc(F)cc1 |wD:29.32,(2.67,6.16,;2.67,4.62,;4,3.85,;5.33,4.62,;6.67,3.85,;6.67,2.31,;5.33,1.54,;4,2.31,;2.67,1.54,;1.33,2.31,;1.33,3.85,;,4.62,;-1.33,3.85,;-2.67,4.62,;-4,3.85,;-4,2.31,;-5.33,4.62,;,1.54,;;-1.33,-.77,;-1.33,-2.31,;,-3.08,;1.33,-2.31,;1.33,-.77,;2.67,,;4,-.77,;-2.67,-3.08,;-4,-2.31,;-2.67,-4.62,;-1.33,-5.39,;,-4.62,;-1.33,-6.93,;,-7.7,;,-9.24,;-1.33,-10.01,;-1.33,-11.55,;-2.67,-9.24,;-2.67,-7.7,)|
C[C@@H]1CN(CCN1C(=O)c1ccc2c(cc(CCCCC(O)=O)n(-c3ccc(F)cc3)c2=O)c1)c1ccc(F)cc1
C[C@@H]1CN(CCN1C(=O)c1ccc2c(cc(CCCCC(O)=O)n(-c3ccc(F)cc3)c2=O)c1)c1ccccc1
OC(=O)CCCCc1cc2cc(ccc2c(=O)n1-c1ccc(F)cc1)C(=O)NC1CC(=O)Nc2ccccc12
C[C@@H](NC(=O)c1ccc2c(c1)cc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1ccc(F)cc1
OC(=O)CCCCc1cc2cc(ccc2c(=O)n1-c1ccc(F)cc1)-c1cc(Cc2ccc(F)cc2)on1
CC1(CC(=NO1)c1ccc2c(c1)c(Cl)c(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1nc2ccc(F)cc2o1 |c:3|
CC1(CC(=NO1)c1ccc2c(cc(CCCCC(O)=O)n(-c3ccc(F)cc3)c2=O)c1)c1nc2ccc(F)cc2o1 |c:3|
OC(=O)CCCCc1cc2cc(ccc2c(=O)n1-c1ccc(F)cc1)-c1noc(n1)C1Cc2ccccc2C1
OC(=O)CCCCc1cc2cc(ccc2c(=O)n1-c1ccc(F)cc1)-c1noc(Cc2ccc(F)cc2)n1
CC(c1nc(no1)-c1ccc2c(c1)cc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1ccc(F)cc1
OC(=O)CCCCc1cc2cc(ccc2c(=O)n1-c1ccc(F)cc1)-c1noc(n1)-c1ccc(cc1)C(F)(F)F
Fc1ccc(cc1)-n1c(CCCCC(=O)NS(=O)(=O)C2CC2)cc2cc(ccc2c1=O)C(=O)N[C@@H]1CCCc2cc(F)ccc12
C[C@@H](NC(=O)c1ccc2c(cc(CCCCC(=O)NS(=O)(=O)C3CC3)n(-c3ccc(F)cc3)c2=O)c1)c1ccc(F)cc1
C[C@@H]1CN(CCN1C(=O)c1ccc2c(cc(CCCCC(=O)NS(=O)(=O)C3CC3)n(-c3ccc(F)cc3)c2=O)c1)c1ccc(F)cc1
C[C@@H]1CN(CCN1C(=O)c1ccc2c(cc(CCCCC(=O)NS(=O)(=O)C3CC3)n(-c3ccc(F)cc3)c2=O)c1)c1ccccc1
Fc1ccc(Cc2cc(no2)-c2ccc3c(cc(CCCCC(=O)NS(=O)(=O)C4CC4)n(-c4ccc(F)cc4)c3=O)c2)cc1
Fc1ccc(Cc2nc(no2)-c2ccc3c(cc(CCCCC(=O)NS(=O)(=O)C4CC4)n(-c4ccc(F)cc4)c3=O)c2)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3)c(cc12)C#N
CC1(CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3)c(cc12)C#N)C(O)=O
CC1(C)CC(C(O)=O)c2cc(C#N)c(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3)cc2O1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3Cl)c(cc12)C#N
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccccc3)c(cc12)C#N
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3Cc4ccccc4C3)c(cc12)C#N
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NOCc3ccc(Cl)cc3)c(cc12)C#N
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)Nc3ccc(Cl)c(Cl)c3)c(cc12)C#N
OC(=O)C1CCOc2cc(Oc3ccc(cc3[N+]([O-])=O)C(=O)NCCc3ccc(Cl)cc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3)c(Cl)cc12
OC(=O)[C@@H]1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccccc3)c(Cl)cc12 |r|
OC(=O)[C@H]1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccccc3)c(Cl)cc12 |r|
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCCCc3ccccc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCCCc3cccc(Cl)c3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCCCc3ccc(Cl)cc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCC\C=C/c3ccccc3Cl)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCCCc3ccccc3Cl)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCC\C=C/c3ccc(Cl)cc3Cl)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCCCc3ccc(Cl)cc3Cl)c(Cl)cc12
Cc1ccccc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
Cc1ccc(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3Cl)cc2)c(C)c1
Cc1ccc(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3Cl)cc2)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Br)cc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(cc3)C3CC3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCC3CC3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(cc3)-c3ccccc3Cl)c(Cl)cc12
Cc1cc(Cl)ccc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Br)cc3Cl)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(cc3Cl)-c3ccccc3Cl)c(Cl)cc12
[Na]OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(cc3Cl)C3CC3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(cc3Cl)-c3ccccc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3Br)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3-c3ccccc3Cl)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3C3CC3)c(Cl)cc12
COc1cc(Br)ccc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(=O)O[Na])c3cc2Cl)cc1
COc1cc(ccc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1)C1CC1
COc1cc(Cl)cc(Cl)c1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
OC(=O)C1CCOc2c(Br)c(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3)c(Cl)cc12
OC(=O)C1CCOc2c1cc(C1CC1)c(Oc1ccc(cc1)C(=O)NCCc1ccc(Cl)cc1)c2C1CC1
OC(=O)C1CCOc2c1cc(C1CC1)c(Oc1ccc(cc1)C(=O)NCCc1ccc(Cl)cc1Cl)c2C1CC1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3)c(cc12)C1CC1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3Cl)c(cc12)C1CC1
OC(=O)C1CCOc2c1cc(Cl)c(Oc1ccc(cc1)C(=O)NCCc1ccc(Cl)cc1Cl)c2C1CC1
CN(C)Cc1ccc(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3C#N)cc2)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)Nc3ccc4CCNCc4c3)c(cc12)C#N
OC(=O)C1CCOc2c(Cl)c(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CC3c3ccccc3)c(cc12)C#N
COc1cccc(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3C#N)cc2)c1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(F)cc3)c(cc12)C#N
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(cc3)C(F)(F)F)c(cc12)C#N
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CC3c3ccc(Cl)cc3)c(cc12)C#N
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3COc4ccccc4C3)c(cc12)C#N
COc1ccc2CC(CCc2c1)NC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2C#N)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCc3cccc4ccccc34)c(cc12)C#N
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3cccc4ccccc34)c(cc12)C#N
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc4ccccc4c3)c(cc12)C#N
CC(C)(C)c1ccc(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3C#N)cc2)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(cc3)-c3ccccc3)c(cc12)C#N
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(cc3)-c3ccccc3)c(Cl)cc12
C[C@@H](CNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1)c1ccccc1 |r|
C[C@H](CNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1)c1ccccc1 |r|
CC(CNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1)c1ccc(Cl)cc1
COc1ccccc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccccc3OC(F)(F)F)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccccc3Oc3ccccc3)c(Cl)cc12
Cc1ccc(cc1C)-c1cccc(NC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3C#N)cc2)c1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)Nc3cccc(c3)-c3ccccc3)c(cc12)C#N
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)Nc3ccc(cc3)-c3ccccc3)c(cc12)C#N
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)Nc3ccc(cc3)-c3ccc(Cl)cc3)c(cc12)C#N
Cc1nccc(n1)-c1cccc(NC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3C#N)cc2)c1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)Nc3ccc(F)c(c3)-c3ccc(Cl)cc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CCc4ccccc4C3)c(cc12)C#N
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3Cc4ccc(Cl)cc4C3)c(cc12)C#N
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)Nc3ccc(Cl)cc3)c(cc12)C#N
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)Nc3ccc(cc3)C(F)(F)F)c(cc12)C#N
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)Nc3ccc4ccccc4c3)c(cc12)C#N
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCCc3ccc(Cl)cc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCCc3ccccc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccccc3Cl)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3c(Cl)cccc3Cl)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(F)cc3F)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3c(F)cccc3Cl)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3cccc(O)c3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(O)cc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(F)cc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3cccc4ccccc34)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc4ccccc4c3)c(Cl)cc12
COc1ccc(OC)c(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3Cl)cc2)c1
COc1cccc(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3Cl)cc2)c1OC
COc1ccc(Br)cc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccccc3Br)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccccc3-c3ccccc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccccc3C3CC3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccccc3-c3ccc(Cl)cc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccccc3-c3cccc(Cl)c3)c(Cl)cc12
[Na]OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccccc3-c3ccccc3Cl)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(F)cc3Cl)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(cc3Cl)C(F)(F)F)c(Cl)cc12
COc1cc(Cl)ccc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
COc1ccc(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3Cl)cc2)c(Cl)c1
COc1cc(F)ccc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
COc1cc(ccc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1)C(F)(F)F
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3cc(Cl)ccc3Cl)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3cc(Cl)ccc3F)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3Cl)c(Cl)cc12
OC(=O)[C@H]1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3Cl)c(Cl)cc12 |r|
OC(=O)[C@@H]1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3Cl)c(Cl)cc12 |r|
Cc1ccc(cc1)-c1cccc(NC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3C#N)cc2)c1
Cc1cccc(c1)-c1cccc(NC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3C#N)cc2)c1
Cc1cccc(c1C)-c1cccc(NC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3C#N)cc2)c1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc4OCOc4c3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCC3Cc4ccccc4C3)c(Cl)cc12
Cc1ccc(SCCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3Cl)cc2)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCSc3ccc(Cl)cc3)c(Cl)cc12
CCOc1ccccc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCOc3ccccc3Cl)c(Cl)cc12
CC(C)(C)Oc1ccccc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
CSc1ccccc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
CSc1ccc(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3Cl)cc2)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CCN(C3)c3cccc(Cl)c3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CCN(CC3)c3cccc(Cl)c3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CN(C3)c3cccc(c3)C(F)(F)F)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CCN(C3)c3cccc(c3)C(F)(F)F)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CCN(CC3)c3cccc(c3)C(F)(F)F)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CCN(CC3)c3ccc(Cl)cc3Cl)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)N[C@H]3CCCN(C3)c3cccc(Cl)c3)c(Cl)cc12 |r|
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCC3Cc4ccccc4C3)c(cc12)C#N
CC(C)(C)C1CCC(CC1)NC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2C#N)cc1 |(8,-5.39,;6.67,-6.16,;6.67,-7.7,;6.67,-4.62,;5.33,-5.39,;4,-6.16,;2.67,-5.39,;2.67,-3.85,;4,-3.08,;5.33,-3.85,;1.33,-3.08,;,-3.85,;,-5.39,;-1.33,-3.08,;-2.67,-3.85,;-4,-3.08,;-4,-1.54,;-5.33,-.77,;-5.33,.77,;-6.67,1.54,;-6.67,3.08,;-8,3.85,;-8,5.39,;-6.67,6.16,;-5.33,5.39,;-4,6.16,;-2.67,5.39,;-4,7.7,;-5.33,3.85,;-4,3.08,;-3.95,1.51,;-2.62,.74,;-1.29,-.03,;-2.67,-.77,;-1.33,-1.54,)|
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3)ccc12
Cc1cc(ccc1Oc1cc2OCCC(C(O)=O)c2cc1C#N)C(=O)NCCc1ccc(Cl)cc1
C[C@@H](CNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2C#N)cc1)c1ccccc1 |r|
C[C@H](CNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2C#N)cc1)c1ccccc1 |r|
CC(Cc1ccc(Cl)cc1)NC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2C#N)cc1
COc1cc(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3C#N)cc2)ccc1Cl
CC(C)(C)c1cccc(NC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3C#N)cc2)c1
CC(C)Oc1cccc(NC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3C#N)cc2)c1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCc3ccc(Cl)c(Cl)c3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(cc3)C(F)(F)F)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)c(Cl)c3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3cccc(Cl)c3Cl)c(Cl)cc12
COc1ccc(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3Cl)cc2)cc1
COc1ccc(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3Cl)cc2)cc1OC
CC(C)(C)c1ccc(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3Cl)cc2)cc1
COc1cccc(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3Cl)cc2)c1
COc1ccc(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3Cl)cc2)c(OC)c1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3cccc(F)c3)c(Cl)cc12
Cc1cccc(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3Cl)cc2)c1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(SC(F)(F)F)cc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3cc(Cl)cc(Cl)c3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3cccc(Oc4ccccc4)c3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3cccc(Cl)c3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3cccc(c3)C(F)(F)F)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccccc3C(F)(F)F)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccccc3F)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)Nc3cccc(c3)C(F)(F)F)c(cc12)C#N
OC(=O)[C@@H]1CCOc2cc(Oc3ccc(cc3)C(=O)NCCC3CCC(CC3)c3ccccc3)c(Cl)cc12 |r,wU:3.2,(-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-6.67,5.39,;-8,4.62,;-8,3.08,;-6.67,2.31,;-6.67,.77,;-5.33,,;-5.33,-1.54,;-4,-2.31,;-4,-3.85,;-2.67,-4.62,;-1.33,-3.85,;-1.33,-2.31,;-2.67,-1.54,;,-4.62,;,-6.16,;1.33,-3.85,;2.67,-4.62,;4,-3.85,;5.33,-4.62,;5.33,-6.16,;6.67,-6.93,;8,-6.16,;8,-4.62,;6.67,-3.85,;9.34,-6.93,;9.34,-8.47,;10.67,-9.24,;12,-8.47,;12,-6.93,;10.67,-6.16,;-4,.77,;-2.67,,;-4,2.31,;-5.33,3.08,)|
OC(=O)[C@H]1CCOc2cc(Oc3ccc(cc3)C(=O)NCCC3CCC(CC3)c3ccccc3)c(Cl)cc12 |r,wD:3.2,(-2.67,4.62,;-4,5.39,;-4,6.93,;-5.33,4.62,;-6.67,5.39,;-8,4.62,;-8,3.08,;-6.67,2.31,;-6.67,.77,;-5.33,,;-5.33,-1.54,;-4,-2.31,;-4,-3.85,;-2.67,-4.62,;-1.33,-3.85,;-1.33,-2.31,;-2.67,-1.54,;,-4.62,;,-6.16,;1.33,-3.85,;2.67,-4.62,;4,-3.85,;5.33,-4.62,;5.33,-6.16,;6.67,-6.93,;8,-6.16,;8,-4.62,;6.67,-3.85,;9.34,-6.93,;9.34,-8.47,;10.67,-9.24,;12,-8.47,;12,-6.93,;10.67,-6.16,;-4,.77,;-2.67,,;-4,2.31,;-5.33,3.08,)|
CC(C)(C)C1CCC(CC1)NC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1 |(8,-5.39,;6.67,-6.16,;6.67,-7.7,;6.67,-4.62,;5.33,-5.39,;4,-6.16,;2.67,-5.39,;2.67,-3.85,;4,-3.08,;5.33,-3.85,;1.33,-3.08,;,-3.85,;,-5.39,;-1.33,-3.08,;-2.67,-3.85,;-4,-3.08,;-4,-1.54,;-5.33,-.77,;-5.33,.77,;-6.67,1.54,;-6.67,3.08,;-8,3.85,;-8,5.39,;-6.67,6.16,;-5.33,5.39,;-4,6.16,;-2.67,5.39,;-4,7.7,;-5.33,3.85,;-4,3.08,;-4,1.54,;-2.67,.77,;-2.67,-.77,;-1.33,-1.54,)|
CC1(C)CCC(CC1)NC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CCCC(C3)c3ccccc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CCCC(C3)c3cccc(Cl)c3)c(Cl)cc12
Cc1ccc(cc1)C1CCCC(C1)NC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
COc1ccc(cc1)C1CCCC(C1)NC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
CSc1ccc(cc1)C1CCCC(C1)NC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
COc1cccc(c1)C1CCCC(C1)NC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CCCC(C3)c3ccc(Cl)cc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CCC(C3)c3ccccc3)c(Cl)cc12
Cc1ccc(cc1)C1CCC(C1)NC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CCC(C3)c3cccc(Cl)c3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CCC(C3)c3ccc(Cl)cc3)c(Cl)cc12
Cc1cccc(c1)C1CCC(C1)NC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CCC(C3)c3cccc(c3)C(F)(F)F)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CCC(C3)c3cccc(F)c3)c(Cl)cc12
CSc1cccc(c1)C1CCC(C1)NC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CCC(C3)c3ccc(Cl)c(Cl)c3)c(Cl)cc12
COc1ccc(cc1)C1CCC(C1)NC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
CSc1ccc(cc1)C1CCC(C1)NC(=O)c1ccc(Oc2cc3OCCC(C(=O)O[Na])c3cc2Cl)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CCC(CC3)c3ccc(Cl)cc3)c(Cl)cc12 |(.28,-10.52,;1.61,-9.75,;2.95,-10.52,;1.61,-8.21,;2.95,-7.44,;2.95,-5.9,;1.61,-5.13,;.28,-5.9,;-1.05,-5.13,;-2.39,-5.9,;-3.72,-5.13,;-3.72,-3.59,;-5.05,-2.82,;-5.05,-1.28,;-3.72,-.51,;-2.39,-1.28,;-2.39,-2.82,;-3.72,1.03,;-5.05,1.8,;-2.39,1.8,;-2.39,3.34,;-3.72,4.11,;-3.72,5.65,;-2.39,6.42,;-1.05,5.65,;-1.05,4.11,;-2.39,7.96,;-3.72,8.73,;-3.72,10.27,;-2.39,11.04,;-2.39,12.58,;-1.05,10.27,;-1.05,8.73,;-2.39,-7.44,;-3.72,-8.21,;-1.05,-8.21,;.28,-7.44,)|
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3CC(C3)c3ccccc3)c(Cl)cc12 |(.54,-9.32,;1.87,-8.55,;3.2,-9.32,;1.87,-7.01,;3.2,-6.24,;3.2,-4.7,;1.87,-3.93,;.54,-4.7,;-.8,-3.93,;-2.13,-4.7,;-3.47,-3.93,;-3.47,-2.39,;-4.8,-1.62,;-4.8,-.08,;-3.47,.69,;-2.13,-.08,;-2.13,-1.62,;-3.47,2.23,;-4.8,3,;-2.13,3,;-2.13,4.54,;-3.22,5.63,;-2.13,6.72,;-1.04,5.63,;-2.13,8.26,;-3.47,9.03,;-3.47,10.57,;-2.13,11.34,;-.8,10.57,;-.8,9.03,;-2.13,-6.24,;-3.47,-7.01,;-.8,-7.01,;.54,-6.24,)|
OCC(Cc1ccc(Cl)cc1)NC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
CC(C)(C)CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCC3CCCCC3)c(Cl)cc12
Cc1cc(ccc1Oc1cc2OCCC(C(O)=O)c2cc1Cl)C(=O)NCCc1ccc(Cl)cc1
Cc1cc(ccc1Oc1cc2OCCC(C(O)=O)c2cc1Cl)C(=O)NCCc1ccc(Cl)cc1Cl
Cc1cc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)ccc1C(=O)NCCc1ccc(Cl)cc1Cl
OC(CNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1)c1ccc(Cl)cc1
OC(CNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1)c1ccccc1Cl
[Na]OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCC3CCCC3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NC3COC4(CCCC4)C3)c(Cl)cc12
COC(CNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1)c1ccc(Cl)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCC(F)c3ccc(Cl)cc3)c(Cl)cc12
COc1cc(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3Cl)cc2)cc(OC)c1
COc1c(Cl)cccc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3C(F)(F)F)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3cccc4OCOc34)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3cccn3-c3ccc(cc3)C(F)(F)F)c(Cl)cc12
FC(F)(CNC(=O)c1ccc(Oc2cc3OCCC(C(=O)O[Na])c3cc2Cl)cc1)c1ccc(Cl)cc1
CCc1ccccc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(=O)O[Na])c3cc2Cl)cc1
OC(CNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1)c1ccc(Cl)cc1Cl
CCOc1cc(Cl)ccc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(=O)O[Na])c3cc2Cl)cc1
[Na]OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3OCC3CC3)c(Cl)cc12
COCCOc1cc(Cl)ccc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
CCOc1cc(Cl)c(Cl)cc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
CC(C)Oc1cc(Cl)ccc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3OC(F)(F)F)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCC3CCCc4ccccc34)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccccc3Oc3ccc(Cl)cc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3Oc3ccccc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3Oc3ccc(Cl)cc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccccc3Oc3cccc(Cl)c3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccccc3Oc3ccccc3Cl)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3Oc3cccc(Cl)c3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3cc(F)ccc3Oc3ccc(Cl)c(Cl)c3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3cc(F)ccc3Oc3ccc(Cl)cc3Cl)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3OCCF)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3OCCCF)c(Cl)cc12
COc1cccc(Cl)c1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
COc1cccc(OC)c1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3)cc(Cl)c12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCC3(CC3)c3ccc(Cl)cc3)c(cc12)C#N
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCOc3ccccc3)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(cc3C(F)(F)F)C(F)(F)F)c(Cl)cc12
COc1cc(OC)c(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3Cl)cc2)c(OC)c1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(OC(F)F)cc3)c(Cl)cc12
COc1cc(Cl)c(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3Cl)cc2)c(Cl)c1
CCOc1ccc(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3Cl)cc2)c(OCC)c1
COc1cc(Cl)c(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3Cl)cc2)c(OC)c1
CCOc1ccc(CCNC(=O)c2ccc(Oc3cc4OCCC(C(O)=O)c4cc3Cl)cc2)c(OC)c1
CCOc1cc(OC)ccc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
CSc1cc(Cl)ccc1CCNC(=O)c1ccc(Oc2cc3OCCC(C(O)=O)c3cc2Cl)cc1
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3F)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCC3CCc4cc(Cl)ccc34)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(cc3C3CC3)C(F)(F)F)c(Cl)cc12
OC(=O)C1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3O)c(Cl)cc12
OC(=O)[C@@H]1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3C3CC3)c(Cl)cc12 |r|
OC(=O)[C@H]1CCOc2cc(Oc3ccc(cc3)C(=O)NCCc3ccc(Cl)cc3C3CC3)c(Cl)cc12 |r|
COc1cc(ccc1CCNC(=O)c1ccc(Oc2cc3OCC[C@@H](C(O)=O)c3cc2Cl)cc1)C1CC1 |r|
COc1cc(ccc1CCNC(=O)c1ccc(Oc2cc3OCC[C@H](C(O)=O)c3cc2Cl)cc1)C1CC1 |r|
COc1cc(Cl)cc(Cl)c1CCNC(=O)c1ccc(Oc2cc3OCC[C@@H](C(O)=O)c3cc2Cl)cc1 |r|
COc1cc(Cl)cc(Cl)c1CCNC(=O)c1ccc(Oc2cc3OCC[C@H](C(O)=O)c3cc2Cl)cc1 |r|
COc1cc(Cl)ccc1CCNC(=O)c1ccc(Oc2cc3OCC[C@@H](C(O)=O)c3cc2Cl)cc1 |r|
COc1cc(Cl)ccc1CCNC(=O)c1ccc(Oc2cc3OCC[C@H](C(O)=O)c3cc2Cl)cc1 |r|
COc1cc(ccc1CCNC(=O)c1ccc(Oc2cc3OCC[C@@H](C(O)=O)c3cc2Cl)cc1)C(F)(F)F |r|
COc1ccc(CCNC(=O)c2ccc(Oc3cc4OCC[C@@H](C(O)=O)c4cc3Cl)cc2)c(OC)c1 |r|
COc1ccc(CCNC(=O)c2ccc(Oc3cc4OCC[C@H](C(O)=O)c4cc3Cl)cc2)c(OC)c1 |r|
CNC(=O)[C@@H]1C[C@H](CN1S(=O)(=O)c1ccc(OC(C)C)cc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@H]1CO)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@H]1C)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@H]1C)n1nc(CC(O)=O)c2cc(Cl)ccc12 |r|
CO\N=C\[C@H]1C[C@H](CN1S(=O)(=O)c1ccc(OC(C)C)cc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1Cn1cccn1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CO[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(F)cc12)S(=O)(=O)c1ccc(OC(C)C)cc1 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(Cl)cc12 |r|
CCC[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(F)cc12)S(=O)(=O)c1ccc(OC(C)C)cc1 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@H]([C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12)N1CCCC1 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(F)cc12)S(=O)(=O)c1ccc(Cl)cc1 |r|
CC(C)Oc1ccc(c(F)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cccc(F)c12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(C)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CC[C@@H]([C@@H](C)C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
C[C@H]1C[C@H](CCN1S(=O)(=O)c1ccc(F)cc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@H](n2nc(CC(O)=O)c3ccc(F)cc23)[C@@](C)(F)C1 |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@]1(C)C#N)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(F)cc12)S(=O)(=O)c1ccc(cc1)C1CC1 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(F)cc12)S(=O)(=O)c1ccc(C)cc1 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(F)cc12)S(=O)(=O)c1cccc(Cl)c1 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(cc12)C(F)(F)F |r|
CC(C)Oc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(cc12)C(F)(F)F |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(=O)NS(C)(=O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(=O)NC#N)c2ccc(F)cc12 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(Cl)cc12)S(=O)(=O)c1ccc(OC(F)(F)F)cc1 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1cc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cccnc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1cc(CC(O)=O)c2cccnc12 |r|
CC(C)Oc1ccc(nc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2c(F)cccc12 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccccc12)S(=O)(=O)c1cc2ccccc2s1 |r|
CC1Cc2cc(ccc2O1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(Cc2nnn[nH]2)c2ccc(F)cc12 |r|
CCOc1ncc(s1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(cc12)C#N |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cc3OCOc3cc12 |r|
CCOc1ccc(s1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CC[C@H]([C@@H]1C)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccccc12)S(=O)(=O)c1ccc2occc2c1 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(cc12)N1CCOCC1 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(cc12)C1=CCCCC1 |r,t:35|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(cc12)N1CCCC1 |r|
CC(C)C1CC1S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCOc1ccc(nc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(c(CCCNC(C)=O)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(c(CCCO)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1cc(CC(O)=O)c2ccc(cc12)-c1ncco1 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(C(C)C(O)=O)c2ccccc12 |r|
C[C@@H]1CN(C[C@@H]1n1c(C)c(CC(O)=O)c2ccccc12)S(=O)(=O)c1ccc(C)cc1 |r|
C[C@H]1C[C@H](CN1S(=O)(=O)c1ccc(OC(F)F)cc1)n1c(C)c(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1[N+]#[C-])n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(c(N)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(c2ccccc12)C1(CC1)C(O)=O |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](CC11COC1)n1nc(CC(O)=O)c2ccccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1c1ccccc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1c1ncc[nH]1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@H]([C@@H]2COC[C@H]12)n1nc(CC(O)=O)c2ccccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CC[C@H]([C@H]1C)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@H]1C(N)=O)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1C(N)=O)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@H]1C(=O)N(C)C)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)NC(=O)[C@@H]1C[C@H](CN1S(=O)(=O)c1ccc(OC(C)C)cc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@H]1C#N)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@H](C[C@H]1C)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1CO)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@H]1CF)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1CF)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@H]1CC#N)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
COC[C@@H]1C[C@H](CN1S(=O)(=O)c1ccc(OC(C)C)cc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
COC[C@H]1C[C@H](CN1S(=O)(=O)c1ccc(OC(C)C)cc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1CC#N)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1Cn1ccnc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1C(F)F)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1Cn1cccc(C)c1=O)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](CC1(C)C)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@H](O)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CC(F)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CC(C(=O)C1)n1nc(CC(O)=O)c2ccc(F)cc12
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CC=C(C1)n1nc(CC(O)=O)c2ccc(F)cc12 |c:16|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](CC=C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@H](C)[C@@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C=C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(F)cc12)S(=O)(=O)c1ccc(OC(C)C)cc1 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](CCO)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C2CC2)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](CF)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CC(C(=C)C1)n1nc(CC(O)=O)c2ccc(F)cc12
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](CC(F)F)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](CCF)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1C)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(F)cc12)S(=O)(=O)c1ccc(F)cc1 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(F)cc12)S(=O)(=O)c1ccc(OC(F)F)cc1 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(F)cc12)S(=O)(=O)c1ccc(cc1Cl)C1CC1 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](CC11CC1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1c1nc[nH]n1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(c(c1)C#N)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1C)n1nc(CC(O)=O)c2cccc(F)c12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cccc(Cl)c12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](CO)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CON=C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(F)cc12)S(=O)(=O)c1ccc(OC(C)C)cc1 |r,w:2.1|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cc(F)c(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cc(F)ccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@H](C)[C@H](C1)n1nc(CC(O)=O)c2cccc(F)c12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CC[C@@H](C[C@H]1CO)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1[C@@H](C)C[C@H](C[C@H]1C)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CC[C@@H]([C@H](C)C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CC[C@@H](C[C@@H]1C)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1CC[C@@H](C[C@H]1C)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
C[C@@H]1C[C@H](CCN1S(=O)(=O)c1ccc(F)cc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
OC(=O)Cc1nn([C@H]2C[C@@H]3CC[C@H](C2)N3S(=O)(=O)c2ccc(F)cc2)c2cc(F)ccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1[C@H]2CC[C@@H]1C[C@H](C2)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
OC(=O)Cc1nn([C@@H]2C[C@@H]3CC[C@H](C2)N3S(=O)(=O)c2ccc(F)cc2)c2cc(F)ccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1[C@H]2CC[C@@H]1C[C@@H](C2)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@H](n2nc(CC(O)=O)c3ccc(F)cc23)[C@@](C)(O)C1 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@H](n2nc(CC(O)=O)c3ccccc23)[C@@](C)(O)C1 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@H](n2nc(CC(O)=O)c3ccc(C)cc23)[C@@](C)(O)C1 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@H](n2nc(CC(O)=O)c3ccccc23)[C@](C)(F)C1 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@H](n2nc(CC(O)=O)c3ccc(C)cc23)[C@](C)(F)C1 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1C(F)F)n1nc(CC(O)=O)c2ccccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1C)n1nc(CC(O)=O)c2ccccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1C(F)F)n1nc(CC(O)=O)c2ccc(C)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1C(F)F)n1nc(CC(O)=O)c2ccc(Cl)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1C)n1nc(CC(O)=O)c2ccc(C)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1C)n1nc(CC(O)=O)c2ccc(Cl)cc12 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccccc12)S(=O)(=O)c1ccc(OC(F)F)cc1 |r|
CC(C)Oc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(\C=C\C(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CCC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1C=C)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC[C@H]1C[C@H](CN1S(=O)(=O)c1ccc(OC(C)C)cc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@]1(C)C#N)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(C)cc12 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(C)cc12)S(=O)(=O)c1ccc(OC(F)F)cc1 |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(C)cc12 |r|
COc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(C)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
COc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(F)cc12)S(=O)(=O)c1ccc(cc1)C(F)(F)F |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(F)cc12)S(=O)(=O)c1ccc(OC(F)(F)F)cc1 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(F)cc12)S(=O)(=O)c1ccccc1Cl |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(F)cc12)S(=O)(=O)c1ccccc1C#N |r|
CCOc1cc(F)c(c(F)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(cc12)C(F)(F)F |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(cc12)C(F)(F)F)S(=O)(=O)c1ccc(OC(F)F)cc1 |r|
COc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(cc12)C(F)(F)F |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(cc12)C(F)(F)F |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(cc12)C(F)(F)F |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1C(F)F)n1nc(CC(O)=O)c2cccc(F)c12 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(Cl)cc12)S(=O)(=O)c1ccc(OC(F)F)cc1 |r|
C[C@H]1CN(C[C@H]1n1nc(CC(O)=O)c2ccc(F)cc12)S(=O)(=O)c1ccc(OC(F)F)cc1 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(Cl)cc12 |r|
COc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(Cl)cc12 |r|
CCc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(Cl)cc12 |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(Cl)cc12 |r|
CC(C)Oc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(Cl)cc12 |r|
CCOc1ccc(c(F)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCCCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@H]([C@@H](C)[C@@H]1C#N)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@@H](C1)n1nc(CC(O)=O)c2cc(Br)c(F)cc12 |r|
C[C@]1(O)CN(C[C@@H]1n1nc(CC(O)=O)c2ccccc12)S(=O)(=O)c1ccc(F)cc1 |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cc(ccc12)C#N |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cc(ccc12)C#N |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cc(Cl)ccc12 |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cc(Cl)ccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cc(Cl)ccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cc(C#N)c(F)cc12 |r|
CCOc1ncc(s1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(s1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCOc1ncc(s1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(C)cc12 |r|
CCOc1ccc(s1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(C)cc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(cc12)C#N |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cc3OCOc3cc12 |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cc3OCOc3cc12 |r|
COc1ccc(s1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
COc1ccc(s1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
COc1ccc(s1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(C)cc12 |r|
CCOc1ccc(c(C=NOC)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r,w:9.9|
CCOc1ccc(c(\C=C\COC)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(c(CCCOC)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(c(COC)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(c(\C=C\c2ccccc2)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(c(CCc2ccccc2)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(c(c1)-c1ccccc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1[N+]([O-])=O)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
COCCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CC(C)OCCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOCCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccccc12)S(=O)(=O)c1ccc(OCCOc2ccccc2)cc1 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccccc12)S(=O)(=O)c1ccc(OCCOC(C)(C)C)cc1 |r|
C[C@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccccc12)S(=O)(=O)c1ccc(OC(F)F)cc1 |r|
C[C@@H]1CN(C[C@H]1n1nc(CC(O)=O)c2ccccc12)S(=O)(=O)c1ccc(OC(F)F)cc1 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1C)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(c(c1)C#N)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cc(C)ccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cc(C)ccc12 |r|
COc1ccc2c(CC(O)=O)nn([C@H]3CN(C[C@H]3C)S(=O)(=O)c3ccc(OC(C)C)cc3)c2c1 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2c(C)cccc12 |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2c(C)cccc12 |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@H](n2nc(CC(O)=O)c3ccccc23)[C@@](C)(F)C1 |r|
COc1ccc(cn1)S(=O)(=O)N1C[C@H](n2nc(CC(O)=O)c3ccccc23)[C@@](C)(F)C1 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1CF)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(=O)NS(C)(=O)=O)c2ccccc12 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccccc12)S(=O)(=O)c1ccc(Oc2ccccc2)nc1 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccccc12)S(=O)(=O)c1ccc2nc(C)sc2c1 |r|
CCOc1ccc(c(Br)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H]([C@H](C)[C@H]1C#N)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
COc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cc(Cl)ccc12 |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(cc12)C1=CCCCC1 |r,t:35|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(cc12)C1CCCCC1 |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(cc12)C1CCCCC1 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(OC)cc12 |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(OC)cc12 |r|
C[C@]1(F)CN(C[C@@H]1n1nc(CC(O)=O)c2ccccc12)S(=O)(=O)c1ccc(F)cc1 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@H](n2nc(CC(O)=O)c3ccccc23)[C@@](C)(F)C1 |r|
CC(C)Oc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(C)cc12 |r|
COc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(C)cc12 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(C)cc12)S(=O)(=O)c1ccc(OC(F)(F)F)cc1 |r|
CCc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(C)cc12 |r|
COc1ccc(c(F)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
COc1ccc(nc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCOc1ccc(nc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
COc1ccc(c(F)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(C)cc12 |r|
CCOc1ccc(c(F)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(C)cc12 |r|
CC(C)C1CC1S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
COc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
COc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccccc12)S(=O)(=O)c1ccc(OC(F)(F)F)cc1 |r|
CCc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
COc1ccc(c(F)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(c(F)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
COc1ccc(nc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CC(C)Oc1ccc(nc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CC(C)C1CC1S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccc(C)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2c(C)cccc12 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2cc(F)ccc12)S(=O)(=O)c1ccc(OC(F)F)cc1 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cc(F)ccc12 |r|
COCCOCCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1cc(CC(O)=O)c2ccc(cc12)C#N |r|
CCOc1ccc(c(CF)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(c(CNC(C)=O)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(c(OC)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cc(ccc12)C#N |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2c(F)cccc12 |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2cc(C)ccc12 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccccc12)S(=O)(=O)C1CCCCC1 |r|
COc1ccc2n(nc(CC(O)=O)c2c1)[C@H]1CN(C[C@H]1C)S(=O)(=O)c1ccc(OC(C)C)cc1 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2cc(C)ccc12)S(=O)(=O)c1ccc(OCF)cc1 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccc(F)cc12)S(=O)(=O)c1ccc(OCF)cc1 |r|
C[C@@H]1CN(C[C@@H]1n1nc(CC(O)=O)c2ccccc12)S(=O)(=O)c1ccc(OCF)cc1 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1cc(CC(O)=O)c2ccc(C)cc12 |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1cc(CC(O)=O)c2ccc(C)cc12 |r|
CCOCCCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
COCCCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@@H](C[C@@H]1CF)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(c(C=C)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(c(CO)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(c(c1)C#C)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(c(\C=C\CO)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(c2ccccc12)C(C)(O)C(O)=O |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(c2ccccc12)C(C)(OC)C(O)=O |r|
C[C@@H]1CN(C[C@@H]1n1c(C)c(CC(O)=O)c2ccccc12)S(=O)(=O)c1ccc(F)cc1 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1COCCCOc1ccccc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(c2ccccc12)C(F)(F)C(O)=O |r|
COCCOCCOC[C@H]1C[C@H](CN1S(=O)(=O)c1ccc(OC(C)C)cc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1COc1ccccc1O)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@@H]([C@H](C)[C@H]1C#N)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@H]([C@H](C)[C@H]1[N+]#[C-])n1nc(CC(O)=O)c2ccccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1COc1cccc(I)c1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(Cc2noc(=O)[nH]2)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC2=NNC(=O)C2)c2ccccc12 |r,t:24|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H]([C@@H](C)[C@@H]1C(N)=O)n1nc(CC(O)=O)c2ccccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1Cn1ncnn1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@H]1COc1nc2ccccc2s1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@H](C[C@@H]1c1ccccc1F)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1c1ccccc1F)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1COc1cccc(F)c1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H]([C@@H](C)[C@@H]1[N+]#[C-])n1nc(CC(O)=O)c2ccccc12 |r|
CCS(=O)(=O)CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(C(O)C(O)=O)c2ccccc12 |r|
CCSCCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](n2nc(CC(O)=O)c3ccccc23)[C@](C)(F)C1 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(=O)NO)c2ccccc12 |r|
CCOc1ccc(c(c1)C(C)O)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@H](F)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(c(CCO)c1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1C)n1c(C)c(CC(O)=O)c2ccccc12 |r|
C[C@H]1C[C@H](CN1S(=O)(=O)c1ccc(F)cc1)n1c(C)c(CC(O)=O)c2ccccc12 |r|
C[C@H]1C[C@H](CN1S(=O)(=O)c1ccc(C)cc1)n1c(C)c(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1C(N)=O)n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@H]1[N+]#[C-])n1nc(CC(O)=O)c2ccccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1COCC=C)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCOc1ccc(c(c1)[N+]([O-])=O)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(CC(O)=O)c2ccccc12 |r|
CC#CCOC[C@H]1C[C@H](CN1S(=O)(=O)c1ccc(OC(C)C)cc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCCOC[C@H]1C[C@H](CN1S(=O)(=O)c1ccc(OC(C)C)cc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1cc(CC(O)=O)c2ccc(cc12)-c1cnn(C)c1 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1c(C)c(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cn1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1c(C)c(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@H](n2nc(CC(O)=O)c3ccc(F)cc23)C(C)(C)C1 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H]([C@H](C)[C@H]1[N+]#[C-])n1nc(CC(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H]([C@H](C)[C@@H]1[N+]#[C-])n1nc(CC(O)=O)c2ccccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1COc1nc2ccccc2s1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(C(F)C(O)=O)c2ccccc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C)[C@H](C1)n1nc(Cc2cc(O)no2)c2ccccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1COCCCO)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1CCc1ccccc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
COc1ccccc1OC[C@H]1C[C@H](CN1S(=O)(=O)c1ccc(OC(C)C)cc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](CC1c1cccnc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1COc1cccc(O)c1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1COc1ccc(O)cc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1Cc1ccccc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1Cc1ccccc1)n1nc(CC(O)=O)c2ccccc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@H]1c1ccccn1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1c1ccccn1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1CC1COC1)n1nc(CC(O)=O)c2ccccc12 |r|
CSC[C@H]1C[C@H](CN1S(=O)(=O)c1ccc(OC(C)C)cc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1CS(C)(=O)=O)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CCOc1ccc(cc1)S(=O)(=O)N1C[C@H](n2nc(CC(O)=O)c3ccccc23)C(C)(C)C1 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@H]1c1ccccc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1c1ccncc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@H]1c1ccncc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1c1nc(C)no1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1COc1ccccc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
CC(C)Oc1ccc(cc1)S(=O)(=O)N1C[C@@H](C[C@@H]1COc1ccc(F)cc1)n1nc(CC(O)=O)c2ccc(F)cc12 |r|
Cc1c(C2=CS(=O)(=O)c3ccccc23)c2cc(F)ccc2n1CC(O)=O |t:3|
Cc1c(C2CS(=O)(=O)c3ccccc23)c2cc(F)ccc2n1CC(O)=O
Cc1c(C2=CS(=O)(=O)c3ccccc23)c2ccc(F)cc2n1CC(O)=O |t:3|
Cc1c(C2=CS(=O)(=O)c3ccccc23)c2ccc(Cl)cc2n1CC(O)=O |t:3|
Cc1c(C2=CS(=O)(=O)c3ccccc23)c2cc(Cl)ccc2n1CC(O)=O |t:3|
Cc1c(C2=CCS(=O)(=O)c3ccccc23)c2cc(F)ccc2n1CC(O)=O |t:3|
Cc1c(C2=CCCS(=O)(=O)c3ccccc23)c2cc(F)ccc2n1CC(O)=O |t:3|
Cc1c(C2=CS(=O)(=O)c3ccncc23)c2cc(F)ccc2n1CC(O)=O |t:3|
Cc1c(C2=CS(=O)(=O)c3ncccc23)c2cc(F)ccc2n1CC(O)=O |t:3|
Cc1c(C2=CS(=O)(=O)c3ccc(cc23)C(F)(F)F)c2cc(F)ccc2n1CC(O)=O |t:3|
Cc1c(C2=CS(=O)(=O)c3cc(ccc23)C(F)(F)F)c2cc(F)ccc2n1CC(O)=O |t:3|
Cc1c(C2=CS(=O)(=O)c3ccc(cc23)C(F)(F)F)c2cc(C)ccc2n1CC(O)=O |t:3|
Cc1c(C2=CS(=O)(=O)c3ccc(cc23)C(F)(F)F)c2ccc(F)cc2n1CC(O)=O |t:3|
Cc1c(C2=CS(=O)(=O)c3cc(ccc23)C(F)(F)F)c2cc(Cl)ccc2n1CC(O)=O |t:3|
Cc1c(C2=CS(=O)(=O)c3cc(ccc23)C(F)(F)F)c2ccc(Cl)cc2n1CC(O)=O |t:3|
Cc1c(C2=CS(=O)(=O)c3cc(ccc23)C(F)(F)F)c2cc(C)ccc2n1CC(O)=O |t:3|
Cc1c(C2=CS(=O)(=O)c3cc(ccc23)C(F)(F)F)c2ccc(F)cc2n1CC(O)=O |t:3|
Cc1c(C2=CS(=O)(=O)c3cc(Br)ccc23)c2cc(F)ccc2n1CC(O)=O |t:3|
Cc1c(C2=CS(=O)(=O)c3cc(ccc23)-c2cc(F)cc(Cl)c2)c2cc(F)ccc2n1CC(O)=O |t:3|
Cc1c(C2=CS(=O)(=O)c3ccc(F)cc23)c2cc(F)ccc2n1CC(O)=O |t:3|
Cc1c(C2=CS(=O)(=O)c3cc(ccc23)S(C)(=O)=O)c2cc(F)ccc2n1CC(O)=O |t:3|
Cc1c(C2=CS(=O)(=O)c3ccc(Cl)cc23)c2cc(F)ccc2n1CC(O)=O |t:3|
Cc1c(C2=CS(=O)(=O)c3ccc(Cl)cc23)c2cc(Cl)ccc2n1CC(O)=O |t:3|
Cc1c(C2=CS(=O)(=O)c3ccc(Cl)cc23)c2ccc(cc2n1CC(O)=O)C(F)(F)F |t:3|
Cc1c(C2=CS(=O)(=O)c3cc(Cl)ccc23)c2cc(F)ccc2n1CC(O)=O |t:3|
Cc1c(Cc2ccc3c(CCS3(=O)=O)c2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc3c(C=CS3(=O)=O)c2)c2cc(F)ccc2n1CC(O)=O |c:9|
CC(C1=CS(=O)(=O)c2ccccc12)c1c(C)n(CC(O)=O)c2ccc(F)cc12 |t:2|
Cc1c(Cc2ccc3C(F)C(F)(F)S(=O)(=O)c3c2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc3c(CNS3(=O)=O)c2)c2cc(F)ccc2n1CC(O)=O
CN1c2cc(Cc3c(C)n(CC(O)=O)c4ccc(F)cc34)ccc2C=CS1(=O)=O |c:27|
Cc1c(Cc2cccc3c2CCS3(=O)=O)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc3c(CCS3(=O)=O)c2)c2ccccc2n1CC(O)=O
Cc1c(Cc2ccc3c(CCS3(=O)=O)c2)c2cc(Cl)ccc2n1CC(O)=O
Cc1c(Cc2ccc3c(CCS3(=O)=O)c2)c2cc(C)ccc2n1CC(O)=O
OC(=O)Cn1c(c(Cc2ccc3c(CCS3(=O)=O)c2)c2ccccc12)-c1ccccc1
Cc1c(Cc2ccc3c(CCS3(=O)=O)c2)c2ccc(Cl)cc2n1CC(O)=O
Cc1c(Cc2ccc3c(CCS3(=O)=O)c2)c2cc(Br)ccc2n1CC(O)=O
Cc1c(Cc2ccc3c(CCS3(=O)=O)c2)c2ccc(cc2n1CC(O)=O)C(F)(F)F
Cc1c(Cc2ccc3c(CCS3(=O)=O)c2)c2cc(ccc2n1CC(O)=O)[N+]([O-])=O
Cc1c(Cc2ccc3c(CCS3(=O)=O)c2)c2cc(NC(=O)C3CC3)ccc2n1CC(O)=O
CC(=O)Nc1ccc2n(CC(O)=O)c(C)c(Cc3ccc4c(CCS4(=O)=O)c3)c2c1
OC(=O)Cn1cc(Cc2ccc3c(CCS3(=O)=O)c2)c2cc(F)ccc12
Cc1c(Cc2ccc3c(c2)C(C)(C)CS3(=O)=O)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2cc3c(cc2C(F)(F)F)S(=O)(=O)CCC3(F)F)c2cc(F)ccc2n1CC(O)=O
CN1CC(F)(F)c2cc(Cc3c(C)n(CC(O)=O)c4ccc(F)cc34)c(cc2S1(=O)=O)C(F)(F)F
Cc1c(Cc2ccc3c(n2)C(F)(F)CCS3(=O)=O)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc3c(N=CNS3(=O)=O)n2)c2cc(F)ccc2n1CC(O)=O |c:9|
CN1C=Nc2cc(Cc3c(C)n(CC(O)=O)c4ccc(F)cc34)ccc2S1(=O)=O |c:2|
CN1CN(C)S(=O)(=O)c2ccc(Cc3c(C)n(CC(O)=O)c4ccc(F)cc34)cc12
Cc1c(Cc2ccc3c(c2)N=C(C)NS3(=O)=O)c2cc(F)ccc2n1CC(O)=O |t:11|
CN1CN(C2CC2)S(=O)(=O)c2ccc(Cc3c(C)n(CC(O)=O)c4ccc(F)cc34)cc12
CN1CN(C)S(=O)(=O)c2cc(c(Cc3c(C)n(CC(O)=O)c4ccc(F)cc34)cc12)C(F)(F)F
Cc1c(Cc2ccc3c(c2)C(F)(F)CCS3(=O)=O)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc3CCS(=O)(=O)c3c2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2cccc3CCS(=O)(=O)c23)c2cc(F)ccc2n1CC(O)=O
CN1CC(F)(F)c2cc(Cc3c(C)n(CC(O)=O)c4ccc(F)cc34)ccc2S1(=O)=O
CN1CC(F)(F)c2cc(Cc3c(C)n(CC(O)=O)c4ccc(F)cc34)c(F)cc2S1(=O)=O
Cc1c(Cc2ccc3c(c2)C(F)(F)CCS3(=O)=O)c2cccnc2n1CC(O)=O
Cc1c(Cc2ccc3c(c2)C(F)(F)CCS3(=O)=O)c2ncccc2n1CC(O)=O
Cc1c(Cc2ccc3c(c2)C(F)(F)CCS3(=O)=O)c2cnccc2n1CC(O)=O
Cc1c(Cc2ccc3c(c2)C(F)(F)CCS3(=O)=O)c2cc(F)ccc2n1Cc1nn[nH]n1
OC(=O)CN1C2CCCCCC2c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12
OC(=O)CCn1c2CCCCc2c2cc(NC(=O)c3ccccc3)ccc12
OC(=O)CCn1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(O)cc3)ccc12
CC(C)(C)C1CCc2c(C1)c1cc(NS(=O)(=O)c3ccc(F)cc3)ccc1n2CC(O)=O
OC(=O)CCn1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12
OC(=O)CCn1c2CCCCc2c2cc(NS(=O)(=O)c3cccc(F)c3)ccc12
Nc1ccc2n(CCC(O)=O)c3CCCCc3c2c1
CC1CCc2c(C1)c1cc(NS(=O)(=O)c3ccc(F)cc3)ccc1n2CC(O)=O
c1ccc2c(c1)c3c(n2CCC(=O)O)CC[C@H](C3)NS(=O)(=O)c4ccc(cc4)F
OC(=O)CCn1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(Cl)cc3)ccc12
OC(=O)c1ccccc1-n1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12 |(.19,-1.35,;.24,-2.9,;-1.07,-3.71,;1.62,-3.64,;1.69,-5.19,;3.04,-5.93,;4.35,-5.09,;4.28,-3.55,;2.93,-2.83,;2.86,-1.28,;4.12,-.38,;5.61,-.71,;6.66,.44,;6.17,1.89,;4.68,2.22,;3.65,1.07,;2.11,1.07,;1.11,2.24,;-.41,1.94,;-1.42,3.11,;-2.93,2.8,;-3.24,4.32,;-2.63,1.3,;-4.45,2.5,;-5.46,3.67,;-6.97,3.36,;-7.46,1.91,;-9.01,1.61,;-6.46,.75,;-4.94,1.05,;-.9,.49,;.1,-.68,;1.62,-.37,)|
OC(=O)Cn1c2CCCc2c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12
OC(=O)CCn1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(F)c(F)c3)ccc12
OC(=O)CCn1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(F)c(Cl)c3)ccc12
OP(O)(=O)CCn1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12
OC(=O)Cn1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12
OC(=O)CCn1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(F)cc3F)ccc12
Cc1ccc(cc1)S(=O)(=O)Nc1ccc2n(CCC(O)=O)c3CCCCc3c2c1
OC(=O)c1cccc(c1)-n1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12
OC(=O)Cn1c2CCC(Cc2c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12)c1ccccc1
CCC(C(O)=O)n1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12
OC(=O)CCCn1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12
OS(=O)(=O)CCn1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12
OC(=O)CCCCn1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12
OC(=O)CCn1c2CCCCc2c2cc(NCc3ccccc3)ccc12
COc1ccc(cc1)S(=O)(=O)Nc1ccc2n(CCC(O)=O)c3CCCCc3c2c1
Cc1ccccc1S(=O)(=O)Nc1ccc2n(CCC(O)=O)c3CCCCc3c2c1
OC(=O)CCn1c2CCCCc2c2cc(NS(=O)(=O)c3cccs3)ccc12
OC(=O)CCn1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(cc3)-c3ccccc3)ccc12
Cc1cccc(c1)S(=O)(=O)Nc1ccc2n(CCC(O)=O)c3CCCCc3c2c1
OC(=O)CCn1c2CCCCc2c2cc(NS(=O)(=O)c3ccc4ccccc4c3)ccc12
CC(C(O)=O)n1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12
OC(=O)CCn1c2CCCCc2c2cc(NS(=O)(=O)c3ccccc3)ccc12
CC(CC(O)=O)n1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12
OC(=O)CCn1c2CCCCc2c2cc(NS(=O)(=O)c3ccccc3F)ccc12
OC(=O)CCn1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(Oc4ccccc4)cc3)ccc12
OC(=O)c1ccc(cc1)-n1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12
OC(=O)\C=C/n1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12
OC(=O)CCn1c2CCCCc2c2cc(NC(=O)Nc3ccccc3)ccc12
CC(Cn1c2CCCCc2c2cc(NS(=O)(=O)c3ccc(F)cc3)ccc12)C(O)=O
CCCS(=O)(=O)Nc1ccc2n(CCC(O)=O)c3CCCCc3c2c1
OC(=O)Cc1sc(Cc2cccc3ccccc23)nc1-c1ccc(Cl)cc1
OC(=O)Cc1sc(nc1-c1ccc(Cl)cc1)C1COc2ccccc2O1
OC(=O)Cc1sc(Nc2cccc3ccccc23)nc1-c1ccc(Cl)cc1
OC(=O)Cc1sc(CS(=O)(=O)c2ccc(Cl)cc2)nc1-c1ccc(Cl)cc1
OC(=O)Cc1sc(COc2ccc(Cl)cc2)nc1-c1ccc(Cl)cc1
OC(=O)Cc1sc(nc1-c1ccc(cc1)C#N)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)Cc1sc(nc1-c1cc(F)cc(F)c1)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)Cc1sc(nc1-c1ccc(Cl)cc1)C(c1ccccc1)c1cccc(Cl)n1
OC(=O)Cc1sc(nc1-c1ccccc1)C(c1ccccc1)c1ccccc1
COc1ccc(Cl)cc1-c1nc(sc1CC(O)=O)C(c1ccccc1)c1ccccc1
OC(=O)Cc1sc(nc1-c1ccccc1)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)Cc1sc(nc1-c1ccc(cc1)C(F)(F)F)C(c1ccccc1)c1ccccc1
OC(=O)Cc1sc(nc1-c1ccc(F)c(F)c1)C(c1ccccc1)c1ccccc1
OC(=O)Cc1sc(nc1-c1ccc(F)cc1)C(c1ccccc1)c1ccccc1
OC(=O)Cc1sc(nc1-c1ccnc(Cl)c1)C(c1ccc(F)cc1)c1ccc(F)cc1
COc1ccc(cc1)-c1nc(sc1CC(O)=O)C(c1ccccc1)c1ccccc1
OC(=O)Cc1sc(nc1-c1cccc(F)c1)C(c1ccccc1)c1ccccc1
OC(=O)Cc1sc(nc1-c1cc(F)nc(F)c1)C(c1ccc(F)cc1)c1ccc(F)cc1
Cc1cc(ccn1)-c1nc(sc1CC(O)=O)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)Cc1sc(nc1-c1ccc(Cl)cc1)-c1ccccc1
OC(=O)Cc1sc(nc1-c1ccc(F)cc1)C(c1ccc(F)cc1)c1ccc(F)cc1
COc1ccc(cc1)C(c1nc(c(CC(O)=O)s1)-c1ccc(F)cc1)c1ccccc1
COc1ccc(cc1)C(c1nc(c(CC(O)=O)s1)-c1ccc(F)cc1)c1ccc(OC)cc1
OC(=O)Cc1sc(nc1-c1ccc(F)cc1)C(c1ccccc1)c1ccc(F)c(F)c1
OC(=O)Cc1sc(nc1-c1cccc(F)c1)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)Cc1sc(nc1-c1ccc(F)cc1)C(c1ccccc1)c1ccc(Cl)cc1
COc1ccc(OC)c(c1)-c1nc(sc1CC(O)=O)C(c1ccccc1)c1ccccc1
COc1ccc(cc1)C(c1nc(c(CC(O)=O)s1)-c1ccc(Cl)cc1)c1ccccn1
OC(=O)Cc1sc(nc1-c1ccc(Cl)cc1)C(c1ccccc1)c1ccccn1
COc1ccc(cc1)C(c1nc(c(CC(O)=O)s1)-c1ccc(Cl)cc1)c1ccccc1
OC(=O)Cc1sc(nc1-c1ccc(Cl)cc1)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)Cc1sc(nc1-c1ccc(F)c(F)c1)C(c1ccc(F)cc1)c1ccc(F)cc1
CN(C)c1cc(ccn1)-c1nc(sc1CC(O)=O)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)Cc1sc(nc1-c1ccnc(c1)N1CCC1)C(c1ccc(F)cc1)c1ccc(F)cc1
CC(=O)N1CCC(CC1)(c1nc(c(CC(O)=O)s1)-c1ccc(Cl)cc1)c1ccccc1
CNc1cc(ccn1)-c1nc(sc1CC(O)=O)C(c1ccc(F)cc1)c1ccc(F)cc1
CCC(c1nc(c(CC(O)=O)s1)-c1ccc(Cl)cc1)c1ccccc1
OC(=O)Cc1sc(nc1-c1ccc(Cl)cc1)C1(CCNCC1)c1ccccc1
OC(=O)Cc1sc(nc1-c1ccc(F)c(c1)C#N)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)Cc1sc(Cc2ccccc2)nc1-c1ccc(Cl)cc1
OC(=O)Cc1sc(nc1-c1ccnc(c1)N1CCCC1)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)Cc1sc(Cc2ccccc2-c2ccccc2)nc1-c1ccc(Cl)cc1
OC(=O)Cc1sc(nc1-c1ccco1)C(c1ccc(F)cc1)c1ccc(F)cc1
COc1cc(ccn1)-c1nc(sc1CC(O)=O)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)Cc1sc(nc1-c1ccoc1)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)Cc1sc(nc1-c1cc[nH]c(=O)c1)C(c1ccc(F)cc1)c1ccc(F)cc1
CS(=O)(=O)Nc1cccc(c1)-c1nc(sc1CC(O)=O)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)Cc1sc(nc1-c1cccc(c1)C#N)C(c1ccc(F)cc1)c1ccc(F)cc1
Nc1nc(c(CC(O)=O)s1)-c1ccc(Cl)cc1
CS(=O)(=O)c1cccc(c1)-c1nc(sc1CC(O)=O)C(c1ccc(F)cc1)c1ccc(F)cc1
NS(=O)(=O)c1cccc(c1)-c1nc(sc1CC(O)=O)C(c1ccc(F)cc1)c1ccc(F)cc1
Nc1cc(ccn1)-c1nc(sc1CC(O)=O)C(c1ccc(F)cc1)c1ccc(F)cc1
NS(=O)(=O)c1ccc(cc1)-c1nc(sc1CC(O)=O)C(c1ccc(F)cc1)c1ccc(F)cc1
Nc1cc(cc(F)n1)-c1nc(sc1CC(O)=O)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)Cc1sc(nc1-c1cccnc1)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)Cc1sc(nc1-c1ccn[nH]1)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)Cc1sc(nc1-c1ccncc1)C(c1ccc(F)cc1)c1ccc(F)cc1
Cn1cc(cn1)-c1nc(sc1CC(O)=O)C(c1ccc(F)cc1)c1ccc(F)cc1
Cc1nc(c(CC(O)=O)s1)-c1ccc(Cl)cc1
OC(=O)Cc1sc(nc1-c1ccc(Cl)cc1)-c1ccco1
OC(=O)Cc1sc(Nc2ccccc2)nc1-c1ccc(Cl)cc1
OC(=O)Cc1sc(CSc2ccccc2)nc1-c1ccc(Cl)cc1
OC(=O)Cc1sc(NC(=O)c2ccccc2)nc1-c1ccc(Cl)cc1
OC(=O)Cc1sc(NCCc2ccccc2)nc1-c1ccc(Cl)cc1
OC(=O)Cc1sc(NCc2ccccc2)nc1-c1ccc(Cl)cc1
OC(=O)Cc1sc(nc1-c1cncc(F)c1)C(c1ccc(F)cc1)c1ccc(F)cc1
Cc1cc(cnc1N)-c1nc(sc1CC(O)=O)C(c1ccc(F)cc1)c1ccc(F)cc1
Nc1ccc(cn1)-c1nc(sc1CC(O)=O)C(c1ccc(F)cc1)c1ccc(F)cc1
CC(=O)N1CCN(CC1)c1cc(ccn1)-c1nc(sc1CC(O)=O)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)Cc1sc(nc1-c1ccc(Cl)cc1)C(Cc1ccccc1)c1ccccc1
OC(=O)Cc1sc(nc1-c1ccc(F)cc1)C(c1ccccc1)c1ccc(O)cc1
OC(=O)Cc1sc(nc1-c1ccc(Cl)cc1)-c1ccc(Oc2ccccc2)cc1
OC(=O)Cc1sc(CC(c2ccccc2)c2ccccc2)nc1-c1ccc(Cl)cc1
OC(=O)Cc1sc(nc1-c1ccc(Cl)cc1)C(c1ccccc1)c1ccc(F)cc1
OC(=O)Cc1sc(nc1-c1ccc(Cl)cc1)C(C1CCCCC1)c1ccccc1
OC(=O)Cc1sc(nc1-c1ccc(Cl)cc1)C(c1ccccc1)c1ccc(Cl)cc1
OC(=O)Cc1sc(nc1-c1ccc(Cl)cc1)C(c1ccccc1)c1ccccc1
OC(=O)Cc1sc(nc1-c1ccnc(F)c1)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)Cc1sc(nc1-c1cn[nH]c1)C(c1ccc(F)cc1)c1ccc(F)cc1
C[C@H]1CN(Cc2cc(Cl)ccc2OCC(O)=O)CCN1C(=O)Cc1ccccc1Cl |r|
C[C@H]1CN(Cc2cc(Cl)ccc2OCC(O)=O)CCN1C(=O)Cc1ccc(Cl)cc1 |r|
C[C@H]1CN(Cc2cc(ccc2OCC(O)=O)C(F)(F)F)CCN1C(=O)Cc1ccc(F)cc1 |r|
C[C@H]1CN(Cc2cc(Cl)ccc2OCC(O)=O)CCN1C(=O)Cc1cccc(Cl)c1 |r|
C[C@H](Oc1ccc(Cl)cc1CN1CCN([C@@H](C)C1)C(=O)Cc1ccc(Cl)cc1)C(O)=O |r|
C[C@H]1CN(Cc2cc(Cl)ccc2OCC(O)=O)CCN1C(=O)C(C)(C)c1ccc(Cl)cc1 |r|
CC[C@H]1CN(Cc2cc(Cl)ccc2OCC(O)=O)CCN1S(=O)(=O)c1ccccc1 |r|
CCC[C@H]1CN(Cc2cc(Cl)ccc2OCC(O)=O)CCN1S(=O)(=O)c1ccccc1 |r|
C[C@H]1CN(Cc2cc(Cl)ccc2OCC(O)=O)C[C@@H](C)N1C(=O)Cc1ccccc1 |r|
OC(=O)COc1ccc(Cl)cc1CN1CCCN(CC1)S(=O)(=O)c1ccccc1
C[C@H]1CN(Cc2cc(Cl)ccc2OCC(O)=O)CCN1C(=O)Cc1ccccc1 |r|
OC(=O)COc1ccc(Cl)cc1CN1CCCN(CC1)S(=O)(=O)Cc1ccccc1
C[C@H]1CN(Cc2cc(Cl)ccc2OCC(O)=O)CCN1C(=O)Cc1ccc(F)cc1 |r|
OC(=O)COc1ccc(Cl)cc1CN1CCN(CC1)C(=O)Cc1ccccc1
OC(=O)COc1ccc(cc1CN1CCN(CC1)S(=O)(=O)c1ccccc1)C(F)(F)F
OC(=O)COc1ccc(Cl)cc1CN1CCN(CC1)S(=O)(=O)Cc1ccccc1
OC(=O)COc1ccc(Cl)cc1CN1CCN(CC1)S(=O)(=O)c1ccccc1
C[C@H]1CN(Cc2cc(Cl)ccc2CC(=O)NS(C)(=O)=O)CCN1S(=O)(=O)Cc1ccccc1 |r|
C[C@H]1CN(Cc2cc(Cl)ccc2CCC(O)=O)CCN1C(=O)Cc1ccccc1 |r|
C[C@H]1CN(Cc2cc(Cl)ccc2CC(O)=O)CCN1S(=O)(=O)Cc1ccccc1 |r|
C[C@H]1CN(Cc2cc(Cl)ccc2OC(C)(C)C(O)=O)CCN1S(=O)(=O)c1ccccc1 |r|
C[C@H]1CN(Cc2cc(Cl)ccc2CC(O)=O)CCN1C(=O)Cc1ccc(Cl)cc1 |r|
CC1CN(Cc2cc(Cl)ccc2OCC(O)=O)CCN1C(=O)c1ccccc1
CC1CN(CCN1Cc1cc(Cl)ccc1OCC(O)=O)S(=O)(=O)c1ccccc1
C[C@H]1CN(Cc2cc(Cl)ccc2OCC(O)=O)CCN1S(=O)(=O)c1ccccc1 |r|
C[C@@H]1CN(Cc2cc(Cl)ccc2OCC(O)=O)CCN1S(=O)(=O)c1ccccc1 |r|
OC(=O)COc1ccc(Cl)cc1CN1CCN(CC1)S(=O)(=O)c1ccc(F)cc1
OC(=O)COc1ccc(cc1CN1CCN(CC1)C(=O)c1ccccc1)C(F)(F)F
Cc1c(CC(O)=O)c2cccnc2n1Cc1ccc(cc1)S(C)=O
Cc1c(CC(O)=O)c2cccnc2n1Cc1ccc(cc1)S(C)(=O)=O
Cc1c(CC(O)=O)c2cccnc2n1Cc1ccc(cc1)[N+]([O-])=O
Cc1c(CC(O)=O)c2cccnc2n1S(=O)(=O)c1ccc(Cl)cc1
Cc1c(CC(O)=O)c2cccnc2n1Cc1ccc(Cl)cc1
Cc1c(CC(O)=O)c2cccnc2n1S(=O)(=O)c1ccc(F)c(F)c1
Cc1c(CC(O)=O)c2cccnc2n1Cc1ccc(cc1)C#N
Cc1c(CC(O)=O)c2cccnc2n1Cc1ccc(cc1)S(=O)(=O)C(F)(F)F
Cc1c(-c2cn(Cc3ccccc3)c(=O)c3CCCCc23)c2cc(F)ccc2n1CC(O)=O |(10.49,-20.94,;9.02,-21.42,;7.78,-20.51,;7.78,-18.97,;9.12,-18.2,;9.12,-16.66,;10.46,-15.89,;11.79,-16.66,;11.79,-18.2,;13.12,-18.98,;14.46,-18.21,;14.46,-16.65,;13.12,-15.89,;7.78,-15.89,;7.78,-14.34,;6.44,-16.67,;5.12,-15.9,;3.79,-16.67,;3.79,-18.21,;5.12,-18.97,;6.44,-18.2,;6.53,-21.42,;5.03,-21.1,;4,-22.24,;2.49,-21.92,;4.48,-23.71,;5.98,-24.02,;7,-22.88,;8.54,-22.88,;9.45,-24.13,;10.98,-23.97,;11.61,-22.56,;11.89,-25.22,)|
Cc1c(-c2cn(CCCC(F)(F)F)c(=O)c3CCCCc23)c2cc(F)ccc2n1CC(O)=O |(35.97,-7.05,;34.5,-7.52,;33.26,-6.62,;33.26,-5.08,;34.6,-4.31,;34.6,-2.77,;35.93,-2,;37.27,-2.78,;38.6,-2.01,;39.94,-2.78,;41.27,-2.01,;39.94,-4.32,;41.42,-3.18,;33.26,-2,;33.26,-.46,;31.93,-2.78,;30.6,-2.02,;29.27,-2.78,;29.28,-4.32,;30.61,-5.08,;31.93,-4.32,;32.01,-7.53,;30.51,-7.21,;29.48,-8.35,;27.98,-8.03,;29.96,-9.81,;31.46,-10.12,;32.48,-8.99,;34.02,-8.99,;34.93,-10.24,;36.46,-10.08,;37.09,-8.67,;37.37,-11.32,)|
Cc1c(-c2cn(CC(F)(F)F)c(=O)c3CCCCc23)c2cc(F)ccc2n1CC(O)=O |(25.15,-8.13,;23.68,-8.61,;22.44,-7.7,;22.44,-6.15,;23.78,-5.39,;23.78,-3.84,;25.12,-3.07,;26.46,-3.84,;27.55,-4.93,;26.46,-5.39,;27.8,-3.07,;22.44,-3.07,;22.44,-1.52,;21.1,-3.85,;19.77,-3.08,;18.44,-3.85,;18.45,-5.4,;19.78,-6.16,;21.1,-5.39,;21.19,-8.61,;19.68,-8.29,;18.65,-9.43,;17.14,-9.11,;19.13,-10.9,;20.63,-11.21,;21.66,-10.08,;23.2,-10.08,;24.11,-11.33,;25.65,-11.17,;26.28,-9.76,;26.56,-12.42,)|
CC(C)n1cc(-c2c(C)n(CC(O)=O)c3ccc(F)cc23)c2CCCCc2c1=O |(11.06,-2.57,;9.73,-1.79,;9.73,-.27,;8.39,-2.56,;8.38,-4.11,;7.04,-4.87,;7.04,-6.42,;8.29,-7.33,;9.76,-6.85,;7.81,-8.8,;8.72,-10.05,;10.25,-9.89,;10.88,-8.48,;11.16,-11.14,;6.26,-8.8,;5.24,-9.93,;3.74,-9.62,;3.26,-8.15,;1.75,-7.83,;4.29,-7.01,;5.79,-7.33,;5.71,-4.11,;4.38,-4.88,;3.05,-4.12,;3.05,-2.57,;4.38,-1.8,;5.71,-2.57,;7.05,-1.79,;7.05,-.24,)|
Cc1c(-c2cn(Cc3ccccc3)c(=O)c3ccccc23)c2cc(F)ccc2n1CC(O)=O |(48.93,-55.96,;47.46,-56.43,;46.22,-55.53,;46.22,-53.98,;47.56,-53.22,;47.56,-51.67,;48.9,-50.9,;50.24,-51.68,;50.23,-53.22,;51.56,-53.99,;52.9,-53.22,;52.9,-51.67,;51.57,-50.9,;46.22,-50.9,;46.22,-49.36,;44.89,-51.68,;43.56,-50.91,;42.23,-51.68,;42.24,-53.23,;43.57,-53.99,;44.89,-53.22,;44.97,-56.43,;43.47,-56.11,;42.44,-57.25,;40.93,-56.93,;42.92,-58.72,;44.42,-59.03,;45.44,-57.9,;46.99,-57.9,;47.89,-59.15,;49.43,-58.99,;50.06,-57.58,;50.33,-60.24,)|
Cc1c(-c2cn(CC(C)(C)C)c(=O)c3ccccc23)c2cc(F)ccc2n1CC(O)=O |(34.69,-56,;33.23,-56.48,;31.99,-55.57,;31.99,-54.03,;33.32,-53.27,;33.33,-51.73,;34.66,-50.96,;36,-51.73,;35.99,-53.27,;37.33,-50.96,;37.32,-52.49,;31.99,-50.95,;31.99,-49.41,;30.66,-51.73,;29.33,-50.97,;28,-51.74,;28.01,-53.28,;29.33,-54.04,;30.66,-53.27,;30.74,-56.48,;29.24,-56.16,;28.21,-57.3,;26.7,-56.98,;28.69,-58.76,;30.19,-59.08,;31.21,-57.94,;32.75,-57.94,;33.66,-59.19,;35.19,-59.03,;35.82,-57.62,;36.09,-60.28,)|
Cc1c(-c2cn(CCCC(F)(F)F)c(=O)c3ccccc23)c2cc(F)ccc2n1CC(O)=O |(20.58,-56.23,;19.11,-56.7,;17.87,-55.8,;17.87,-54.26,;19.21,-53.49,;19.21,-51.95,;20.54,-51.18,;21.88,-51.96,;23.21,-51.19,;24.55,-51.96,;25.88,-51.19,;24.55,-53.5,;26.03,-52.36,;17.87,-51.18,;17.87,-49.64,;16.54,-51.96,;15.21,-51.19,;13.88,-51.96,;13.89,-53.5,;15.22,-54.26,;16.54,-53.49,;16.62,-56.71,;15.12,-56.39,;14.1,-57.53,;12.59,-57.21,;14.57,-58.99,;16.07,-59.3,;17.09,-58.17,;18.63,-58.17,;19.54,-59.42,;21.07,-59.26,;21.7,-57.85,;21.98,-60.5,)|
Cc1c(-c2cn(CC(F)(F)F)c(=O)c3ccccc23)c2cc(F)ccc2n1CC(O)=O |(7.05,-54.88,;5.58,-55.35,;4.34,-54.45,;4.34,-52.9,;5.68,-52.13,;5.68,-50.59,;7.02,-49.82,;8.36,-50.59,;8.36,-52.14,;9.7,-49.82,;9.45,-51.68,;4.34,-49.81,;4.34,-48.27,;3,-50.6,;1.67,-49.83,;.34,-50.6,;.35,-52.15,;1.68,-52.91,;3,-52.14,;3.09,-55.36,;1.58,-55.04,;.55,-56.18,;-.96,-55.86,;1.03,-57.65,;2.53,-57.96,;3.56,-56.82,;5.1,-56.82,;6.01,-58.08,;7.55,-57.92,;8.18,-56.5,;8.46,-59.17,)|
CC(C)n1cc(-c2c(C)n(CC(O)=O)c3ccc(F)cc23)c2ccccc2c1=O |(57.2,-40.02,;55.86,-39.25,;55.86,-37.71,;54.53,-40.02,;54.52,-41.56,;53.19,-42.33,;53.19,-43.87,;54.43,-44.77,;55.89,-44.3,;53.95,-46.24,;54.86,-47.48,;56.39,-47.32,;57.02,-45.92,;57.29,-48.57,;52.41,-46.24,;51.39,-47.37,;49.89,-47.06,;49.41,-45.59,;47.9,-45.27,;50.44,-44.45,;51.94,-44.77,;51.86,-41.56,;50.54,-42.33,;49.21,-41.57,;49.2,-40.03,;50.53,-39.26,;51.86,-40.03,;53.19,-39.25,;53.19,-37.71,)|
Cc1c(-c2ccc(=O)n(CC(F)(F)F)c2)c2cc(F)ccc2n1CC(O)=O
CC(C)n1cc(ccc1=O)-c1c(C)n(CC(O)=O)c2ccc(F)cc12
CC(C)n1cc(Cc2c(C)n(CC(O)=O)c3ccc(F)cc23)ccc1=O
Cc1c(-c2ccc(=O)n(Cc3c(F)cccc3F)c2)c2cc(F)ccc2n1CC(O)=O
Cc1c(-c2ccc(=O)n(Cc3ccc(F)cc3)c2)c2cc(F)ccc2n1CC(O)=O
Cc1c(-c2ccc(=O)n(Cc3ccc(F)cc3F)c2)c2cc(F)ccc2n1CC(O)=O
Cc1c(-c2ccc(=O)n(Cc3ccccc3)c2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(CCCC(F)(F)F)c2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(CCCC(F)(F)F)n2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(CC(F)(F)F)c2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(CC(F)(F)F)n2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3ccc(F)cc3F)c2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3cc(F)ccc3F)c2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3cc(F)ccc3F)n2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3c(F)cccc3F)c2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3c(F)cccc3F)n2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3ccc(F)cc3)c2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3ccc(F)cc3)n2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3cccc(F)c3)c2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3cccc(F)c3)n2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3ccccc3F)c2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3ccccc3F)n2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3ccccc3)c2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3ccccc3)n2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3cccc(F)c3F)c2)c2cc(F)ccc2n1CC(=O)ONS(C)(=O)=O
Cc1c(Cc2ccc(=O)n(Cc3cccc(F)c3F)c2)c2cc(F)ccc2n1CC(=O)N1CCCC1
CN(C)C(=O)Cn1c(C)c(Cc2ccc(=O)n(Cc3cccc(F)c3F)c2)c2cc(F)ccc12
Cc1c(Cc2ccc(=O)n(Cc3cccc(F)c3F)c2)c2cc(F)ccc2n1CC(N)=O
Cc1c(Cc2ccc(=O)n(Cc3cccc(F)c3F)c2)c2cc(F)ccc2n1CC(O)=O
Cc1c(-c2ccc(=O)n(CCCC(F)(F)F)c2)c2cc(F)ccc2n1CC(O)=O
Cc1c(-c2ccc(=O)n(Cc3c(F)cccc3F)c2)c2ccccc2n1CC(O)=O
Cc1c(-c2ccc(=O)n(Cc3c(F)cccc3F)c2)c2cc(Cl)ccc2n1CC(O)=O
Cc1c(-c2ccc(=O)n(Cc3ccccc3)c2)c2ccccc2n1CC(O)=O
Cc1c(-c2ccc(=O)n(Cc3ccccc3)c2)c2cc(Cl)ccc2n1CC(O)=O
COc1ccc2n(CC(O)=O)c(C)c(-c3ccc(=O)n(CC(F)(F)F)c3)c2c1
Cc1c(-c2ccc(=O)n(CC(F)(F)F)c2)c2cc(C)ccc2n1CC(O)=O
Cc1c(-c2ccc(=O)n(CC(F)(F)F)c2)c2ccccc2n1CC(O)=O
Cc1c(-c2ccc(=O)n(CC(F)(F)F)c2)c2cc(Cl)ccc2n1CC(O)=O
CC(C)n1cc(ccc1=O)-c1c(C)n(CC(O)=O)c2ccccc12
CC(C)n1cc(ccc1=O)-c1c(C)n(CC(O)=O)c2ccc(Cl)cc12
Cc1c(-c2ccc(OCCCC(F)(F)F)nc2)c2cc(F)ccc2n1CC(O)=O
C[C@@H](C(O)=O)n1c(C)c(Cc2ccc(=O)n(Cc3cccc(F)c3F)c2)c2cc(F)ccc12 |r|
C[C@H](C(O)=O)n1c(C)c(Cc2ccc(=O)n(Cc3cccc(F)c3F)c2)c2cc(F)ccc12 |r|
Cc1c(Cc2ccc(=O)n(Cc3ccc(F)cc3F)n2)c2cc(F)ccc2n1CC(O)=O
COc1cc(CC(O)=O)ccc1Oc1ccc2n(C)ccc2c1NS(=O)(=O)c1ccc(Cl)cc1Cl
COc1cc(CC(O)=O)ccc1Oc1ccc2[nH]c(cc2c1NS(=O)(=O)c1ccc(Cl)cc1Cl)C1CC1
COc1cc(CC(O)=O)ccc1Oc1ccc2[nH]c(CC(C)C)cc2c1NS(=O)(=O)c1ccc(Cl)cc1Cl
COc1cc(CC(O)=O)ccc1Oc1ccc2[nH]c(cc2c1NS(=O)(=O)c1ccc(Cl)cc1Cl)C(C)(C)C
CCCc1cc2c(NS(=O)(=O)c3ccc(Cl)cc3Cl)c(Oc3ccc(CC(O)=O)cc3OC)ccc2[nH]1
COc1cc(CC(O)=O)ccc1Oc1ccc2n(C)c(C)cc2c1NS(=O)(=O)c1ccc(Cl)cc1Cl
COc1cc(CC(O)=O)ccc1Oc1ccc2[nH]c(C)c(Cl)c2c1NS(=O)(=O)c1ccc(Cl)cc1Cl
COc1cc(CC(O)=O)ccc1Oc1ccc2[nH]c(cc2c1NS(=O)(=O)c1ccc(Cl)cc1Cl)C#N
COc1cc(CC(O)=O)ccc1Oc1ccc2NC(=O)Cc2c1NS(=O)(=O)c1ccc(Cl)cc1Cl
CCCCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
OC(=O)Cn1c2CC[C@H](Cc2c2ccccc12)NS(=O)(=O)c1ccc(F)cc1
CN([C@@H]1CCc2c(c3ccccc3n2CC(=O)O)C1)S(=O)(=O)c4ccc(cc4)F
CN([C@@H]1CCc2c(C1)c1ccccc1n2CCC(O)=O)S(=O)(=O)c1ccc(F)cc1
CCCCC[C@H](O)\C=C\[C@@H]1[C@@H](C\C=C\CCCC(O)=O)[C@@H](O)CC1=O
CCCCC[C@@](C)(O)\C=C\[C@@H]1[C@@H](C\C=C\CCCC(O)=O)[C@@H](O)CC1=O
CCCCC[C@](C)(O)\C=C\[C@@H]1[C@@H](C\C=C\CCCC(O)=O)[C@@H](O)CC1=O
Cc1c(CC(O)=O)c2cc(F)ccc2n1S(=O)(=O)c1ccccc1
Cc1c(CC(O)=O)c2cc(F)ccc2n1S(=O)(=O)c1ccc(F)cc1
Cc1c(CC(O)=O)c2cc(F)ccc2n1S(=O)(=O)c1ccc(Cl)cc1
Cc1c(CC(O)=O)c2cc(F)ccc2n1S(=O)(=O)c1ccc(C)cc1
Cc1c(c2cc(ccc2n1C(=O)c3ccc(cc3)Cl)OC)CC(=O)O
CCCCS(=O)(=O)n1c(C)c(CC(O)=O)c2cc(F)ccc12
Cc1c(CC(O)=O)c2cc(F)ccc2n1S(=O)(=O)c1cccc(F)c1
Cc1c(CC(O)=O)c2cc(F)ccc2n1S(=O)(=O)c1cc(Cl)ccc1Cl
COc1ccc(cc1)S(=O)(=O)n1c(C)c(CC(O)=O)c2cc(F)ccc12
Cc1c(CC(O)=O)c2cc(F)ccc2n1S(=O)(=O)c1ccc(cc1)S(C)(=O)=O
Cc1nc(cn1C)S(=O)(=O)n1c(C)c(CC(O)=O)c2cc(F)ccc12
CC\1=C(c2cc(ccc2/C1=C\c3ccc(cc3)SC)F)CC(=O)O
OC(=O)C[C@@H]1CCn2c1c(Sc1ccc(Cl)cc1)c1ccc(F)cc21
COc1ccc2n(CC(O)=O)c(C)c(-c3ccnc4cc(Cl)ccc34)c2c1 |(5.11,-4.86,;5.12,-3.32,;6.45,-2.56,;6.45,-1.01,;7.78,-.24,;9.11,-1,;10.59,-.52,;11.06,.95,;12.57,1.27,;13.61,.13,;13.05,2.74,;11.51,-1.77,;13.05,-1.76,;10.6,-3.03,;11.09,-4.5,;12.59,-4.8,;13.08,-6.25,;12.05,-7.41,;10.54,-7.1,;9.53,-8.24,;8.03,-7.94,;7.02,-9.09,;7.55,-6.48,;8.56,-5.34,;10.06,-5.64,;9.12,-2.56,;7.78,-3.33,)|
Cc1c(-c2ccnc3c(F)cccc23)c2cc(C)ccc2n1CC(O)=O |(24.76,-.53,;23.22,-.54,;22.31,-1.8,;22.79,-3.27,;24.3,-3.56,;24.78,-5.02,;23.76,-6.18,;22.25,-5.87,;21.24,-7.01,;21.73,-8.47,;19.74,-6.71,;19.25,-5.25,;20.27,-4.1,;21.77,-4.41,;20.83,-1.33,;19.49,-2.1,;18.16,-1.33,;16.82,-2.1,;18.16,.22,;19.49,.99,;20.82,.22,;22.3,.71,;22.77,2.17,;24.28,2.5,;25.32,1.36,;24.75,3.97,)|
Cc1c(-c2ccnc3ccccc23)c2cc(C)ccc2n1CC(O)=O |(12.8,-17.54,;11.26,-17.55,;10.36,-18.82,;10.84,-20.28,;12.34,-20.58,;12.83,-22.03,;11.81,-23.19,;10.3,-22.88,;9.29,-24.02,;7.79,-23.72,;7.3,-22.26,;8.32,-21.12,;9.82,-21.43,;8.87,-18.34,;7.54,-19.11,;6.2,-18.34,;4.87,-19.11,;6.21,-16.8,;7.53,-16.02,;8.87,-16.79,;10.35,-16.31,;10.82,-14.84,;12.32,-14.51,;13.36,-15.65,;12.8,-13.04,)|
Cc1c(-c2ccnc3c(C)cccc23)c2cc(C)ccc2n1CC(O)=O |(-2.12,-2.68,;-3.66,-2.69,;-4.56,-3.95,;-4.08,-5.41,;-2.58,-5.71,;-2.09,-7.17,;-3.11,-8.33,;-4.62,-8.02,;-5.63,-9.15,;-5.14,-10.61,;-7.13,-8.85,;-7.62,-7.39,;-6.6,-6.25,;-5.1,-6.56,;-6.04,-3.48,;-7.38,-4.24,;-8.72,-3.47,;-10.05,-4.24,;-8.71,-1.93,;-7.38,-1.16,;-6.05,-1.92,;-4.57,-1.44,;-4.1,.03,;-2.6,.35,;-1.56,-.78,;-2.12,1.82,)|
Cc1c(-c2ccnc3c(cccc23)C#N)c2cc(C)ccc2n1CC(O)=O |(27.67,-17.48,;26.13,-17.49,;25.23,-18.76,;25.71,-20.22,;27.21,-20.52,;27.7,-21.97,;26.68,-23.13,;25.17,-22.82,;24.15,-23.96,;22.66,-23.66,;22.17,-22.2,;23.19,-21.06,;24.68,-21.37,;24.65,-25.42,;25.14,-26.88,;23.74,-18.28,;22.41,-19.05,;21.07,-18.28,;19.73,-19.05,;21.07,-16.73,;22.4,-15.96,;23.74,-16.73,;25.22,-16.24,;25.69,-14.78,;27.19,-14.45,;28.23,-15.59,;27.67,-12.98,)|
COc1ccc2n(c(C)c(CC(O)=O)c2c1)-c1ccnc2cc(Cl)ccc12 |(-9.26,-.49,;-7.93,.28,;-6.59,-.48,;-6.59,-2.03,;-5.26,-2.8,;-3.92,-2.03,;-2.44,-2.5,;-1.53,-1.24,;.01,-1.23,;-2.45,.01,;-1.98,1.47,;-.47,1.8,;.57,.66,;0,3.27,;-3.93,-.48,;-5.26,.29,;-1.96,-3.97,;-.45,-4.26,;.04,-5.72,;-.99,-6.88,;-2.5,-6.57,;-3.51,-7.71,;-5.01,-7.41,;-6.02,-8.56,;-5.5,-5.95,;-4.48,-4.8,;-2.98,-5.11,)|
Cc1c(CC(O)=O)c2ccccc2n1-c1ccncn1
Cc1c(-c2ccnc3cc(Cl)ccc23)c2ccc(C)cc2n1CC(O)=O |(27.14,-1.36,;25.6,-1.36,;24.69,-2.63,;25.18,-4.09,;26.68,-4.39,;27.17,-5.85,;26.14,-7.01,;24.63,-6.69,;23.62,-7.83,;22.13,-7.53,;21.11,-8.69,;21.64,-6.07,;22.66,-4.93,;24.15,-5.24,;23.21,-2.16,;21.88,-2.92,;20.54,-2.15,;20.54,-.61,;19.21,.16,;21.87,.16,;23.21,-.6,;24.68,-.12,;25.16,1.35,;26.66,1.67,;27.7,.54,;27.14,3.15,)|
Cc1c(-c2ccnc3cc(Cl)ccc23)c2cc(C)ccc2n1CC(O)=O |(-.89,-17.71,;-2.43,-17.72,;-3.33,-18.98,;-2.85,-20.44,;-1.35,-20.74,;-.86,-22.2,;-1.89,-23.36,;-3.4,-23.04,;-4.41,-24.19,;-5.9,-23.88,;-6.92,-25.04,;-6.39,-22.43,;-5.37,-21.28,;-3.88,-21.59,;-4.82,-18.51,;-6.15,-19.27,;-7.49,-18.5,;-8.82,-19.27,;-7.49,-16.96,;-6.16,-16.19,;-4.82,-16.95,;-3.34,-16.47,;-2.87,-15,;-1.37,-14.68,;-.33,-15.81,;-.89,-13.21,)|
COc1cccc2c(ccnc12)-c1c(C)n(CC(O)=O)c2ccc(C)cc12 |(-5.5,-28.92,;-4.48,-27.76,;-4.97,-26.3,;-6.47,-26,;-6.96,-24.54,;-5.94,-23.4,;-4.44,-23.71,;-3.42,-22.56,;-1.92,-22.86,;-1.43,-24.32,;-2.45,-25.48,;-3.96,-25.16,;-3.9,-21.1,;-3,-19.84,;-1.46,-19.83,;-3.91,-18.59,;-3.44,-17.12,;-1.93,-16.8,;-.89,-17.93,;-1.46,-15.33,;-5.39,-19.07,;-6.72,-18.31,;-8.05,-19.08,;-8.05,-20.62,;-9.39,-21.39,;-6.72,-21.39,;-5.38,-20.63,)|
Cc1c(-c2cc(C)nc3ccccc23)c2cc(C)ccc2n1CC(O)=O |(28.12,-18.42,;26.58,-18.43,;25.68,-19.69,;26.16,-21.15,;27.66,-21.45,;28.15,-22.91,;29.66,-23.22,;27.13,-24.07,;25.62,-23.76,;24.61,-24.9,;23.11,-24.59,;22.62,-23.14,;23.64,-21.99,;25.14,-22.3,;24.2,-19.22,;22.86,-19.99,;21.52,-19.22,;20.19,-19.98,;21.53,-17.67,;22.86,-16.9,;24.19,-17.66,;25.67,-17.18,;26.14,-15.72,;27.64,-15.39,;28.68,-16.53,;28.12,-13.92,)|
Cc1c(-c2ccnc3c(cccc23)C(F)(F)F)c2cc(C)ccc2n1CC(O)=O |(26.72,-33.91,;25.18,-33.91,;24.27,-35.18,;24.75,-36.64,;26.26,-36.94,;26.74,-38.39,;25.72,-39.55,;24.21,-39.24,;23.2,-40.38,;21.7,-40.08,;21.21,-38.62,;22.23,-37.48,;23.73,-37.79,;23.69,-41.84,;24.08,-43.32,;25.16,-41.4,;22.22,-42.29,;22.79,-34.71,;21.45,-35.47,;20.12,-34.7,;18.78,-35.47,;20.12,-33.16,;21.45,-32.39,;22.78,-33.15,;24.26,-32.67,;24.73,-31.2,;26.24,-30.88,;27.28,-32.01,;26.71,-29.41,)|
Cc1c(-c2ccnc3ccc(cc23)C(F)(F)F)c2cc(C)ccc2n1CC(O)=O |(-.91,-35.57,;-2.45,-35.58,;-3.36,-36.84,;-2.87,-38.3,;-1.37,-38.6,;-.88,-40.06,;-1.91,-41.22,;-3.42,-40.91,;-4.43,-42.05,;-5.92,-41.74,;-6.41,-40.29,;-5.39,-39.14,;-3.9,-39.45,;-7.92,-39.98,;-9.42,-39.57,;-8.28,-41.48,;-7.55,-38.48,;-4.84,-36.37,;-6.18,-37.14,;-7.51,-36.37,;-8.84,-37.13,;-7.51,-34.82,;-6.18,-34.05,;-4.84,-34.81,;-3.37,-34.33,;-2.9,-32.87,;-1.39,-32.54,;-.35,-33.68,;-.91,-31.07,)|
Cc1c(-c2ccnc3c(Cl)cccc23)c2cc(C)ccc2n1CC(O)=O |(10.93,-.53,;9.39,-.54,;8.49,-1.8,;8.97,-3.27,;10.47,-3.56,;10.96,-5.02,;9.94,-6.18,;8.43,-5.87,;7.42,-7.01,;7.91,-8.47,;5.92,-6.71,;5.43,-5.25,;6.45,-4.1,;7.95,-4.41,;7.01,-1.33,;5.67,-2.1,;4.34,-1.33,;3,-2.1,;4.34,.22,;5.67,.99,;7,.22,;8.48,.71,;8.95,2.17,;10.46,2.5,;11.5,1.36,;10.93,3.97,)|
Cc1c(-c2ccnc3cc(ccc23)C(F)(F)F)c2cc(C)ccc2n1CC(O)=O |(11.76,-35.94,;10.22,-35.95,;9.31,-37.22,;9.8,-38.68,;11.3,-38.98,;11.79,-40.43,;10.76,-41.59,;9.25,-41.28,;8.24,-42.42,;6.75,-42.12,;6.26,-40.66,;7.28,-39.52,;8.77,-39.82,;5.73,-43.27,;4.63,-44.36,;6.85,-44.33,;4.61,-42.21,;7.83,-36.74,;6.49,-37.51,;5.16,-36.74,;3.83,-37.51,;5.16,-35.19,;6.49,-34.42,;7.83,-35.19,;9.3,-34.7,;9.77,-33.24,;11.28,-32.91,;12.32,-34.05,;11.76,-31.44,)|
Cc1c(-c2ccnc3c(cccc23)S(C)(=O)=O)c2cc(C)ccc2n1CC(O)=O |(13.57,-17.56,;12.03,-17.57,;11.12,-18.83,;11.61,-20.29,;13.11,-20.59,;13.6,-22.05,;12.57,-23.21,;11.06,-22.89,;10.05,-24.03,;8.56,-23.73,;8.07,-22.27,;9.09,-21.13,;10.58,-21.44,;10.54,-25.49,;11.04,-26.95,;11.87,-24.71,;9.2,-26.25,;9.64,-18.36,;8.31,-19.12,;6.97,-18.35,;5.64,-19.12,;6.97,-16.81,;8.3,-16.04,;9.64,-16.8,;11.12,-16.32,;11.59,-14.85,;13.09,-14.53,;14.13,-15.66,;13.57,-13.06,)|
COc1ccc(OCC(O)=O)c(c1)C(=O)c1cnn(c1)-c1ccccc1
Cc1ccc(OCC(O)=O)c(c1)C(=O)c1cnn(c1)-c1ccccc1
CCOC(=O)COc1ccc(Br)cc1C(=O)c1cnn(c1)-c1ccccc1
COc1ccc(cc1)-n1cc(cn1)C(=O)c1cc(Br)ccc1OCC(O)=O
CC(C)(C)c1cc(Br)ccc1OCC(O)=O
OCc1cc(Br)ccc1OCC(O)=O
OC(=O)COc1ccc(Br)cc1C(=O)c1cnn(c1)-c1ccccc1Br
OC(=O)COc1ccc(Br)cc1C(=O)c1ccno1
OC(=O)COc1ccc(Br)cc1C(=O)c1cnn(c1)-c1ccccc1
OC(=O)COc1ccccc1C=O
OC(=O)COc1ccc(Br)cc1C=O
OC(=O)COc1ccc(cc1C(=O)c1cnn(c1)-c1ccccc1)-c1ccccc1
OC(=O)COc1ccccc1C=NNC(=O)COc1ccc(Cl)cc1Cl |w:12.13|
OC(=O)COc1ccc(Br)cc1C(=O)c1cnn(c1)-c1ccc(Br)cc1
OC(=O)COc1ccc(Cl)cc1C(=O)c1cnn(c1)-c1ccccc1
OC(=O)COc1ccccc1C=NNC(=O)Cn1cnc2ccccc12 |w:12.13|
Cc1ccc(NCC(=O)NN=Cc2ccccc2OCC(O)=O)cc1 |w:10.9|
OC(=O)COc1ccc(F)cc1C(=O)c1cnn(c1)-c1ccccc1
OC(=O)COc1ccc(Br)cc1CN=Nc1ccccn1 |w:13.13|
CC(=O)c1cc(Br)ccc1OCC(O)=O
OC(=O)COc1ccc(Br)cc1CN=Nc1cccc2cccnc12 |w:13.13|
OC(=O)COc1ccc(Br)cc1C(=O)c1cnn(c1)-c1cccc(Br)c1
OC(=O)COc1ccc(Br)cc1C(=O)c1ccccc1
OC(=O)COc1ccc(cc1C(=O)c1cnn(c1)-c1ccccc1)-c1cc(F)cc(F)c1
COc1ccc(cc1)-c1cnnc(N=NCc2ccccc2OCC(O)=O)n1 |w:14.15|
OC(=O)COc1ccc(cc1C(=O)c1cnn(c1)-c1ccccc1)[N+]([O-])=O
OC(=O)COc1ccccc1C(=O)c1cnn(c1)-c1ccccc1
Cc1cc([nH]n1)C(=O)NN=Cc1ccccc1OCC(O)=O |w:9.9|
OC(=O)COc1ccc(Br)cc1C(=O)c1cnn(c1)-c1ccc(Cl)cc1
OC(=O)COc1ccc(Br)cc1CN=Nc1nncc(n1)-c1ccccc1 |w:13.13|
OC(=O)COc1ccc(cc1C(=O)c1cnn(c1)-c1ccccc1)-c1ccc(Cl)cc1
CS(=O)(=O)c1cc(F)cc2c3CC[C@H](CC(O)=O)c3n(Cc3ccc(Cl)cc3)c12
CC1(CCCCC1)c1cc(Cl)ccc1OCC(O)=O
OC(=O)COc1ccc(Cl)cc1C1CCCC1
OC(=O)COc1ccc(Cl)cc1C1CCCCCC1
C[C@H](Oc1ccc(Cl)cc1C1CCCCC1)C(O)=O
C[C@@H](Oc1ccc(Cl)cc1C1CCCCC1)C(O)=O
COC(=O)COc1ccc(Cl)cc1C1CCCCC1
OC(=O)COc1ccccc1C1CCCCC1
OC(=O)CCOc1ccc(Cl)cc1C1CCCCC1
OC(=O)CCCOc1ccc(Cl)cc1C1CCCCC1
OC(=O)COc1ccc(cc1C1CCCCC1)C#N
OC(=O)COc1ccc(Cl)cc1C1CCCCC1
Cc1ccc(OCC(O)=O)c(c1)C1CCCCC1
COc1ccc(OCC(O)=O)c(c1)C1CCCCC1
OC(=O)COc1ccc(cc1C1CCCCC1)-c1ccc(F)cc1
OC(=O)COc1ccc(Br)cc1C1CCCCC1
OCCOc1ccc(Cl)cc1C1CCCCC1
OC(=O)COc1ccc(F)cc1C1CCCCC1
CS(=O)(=O)NC(=O)COc1ccc(Cl)cc1C1CCCCC1
OC(=O)COc1ccc(Cl)cc1CC=C
OC(=O)COc1ccc(cc1C1CCCCC1)C(F)(F)F
Cc1cc(Cl)ccc1OCC(O)=O
Clc1ccc(OCc2nnn[nH]2)c(c1)C1CCCCC1
CC(C)c1nccc2n3CC[C@@H](CC(O)=O)c3c(Sc3ccc(Cl)c(Cl)c3)c12 |r|
CC(C)c1nccc2n3CC[C@H](CC(O)=O)c3c(Sc3ccc(Cl)c(Cl)c3)c12 |r|
Cc1c(CC(O)=O)c2cccnc2n1S(=O)(=O)c1ccccc1Cl
COc1ccc(cc1)S(=O)(=O)n1c(C)c(CC(O)=O)c2cccnc12
Cc1c(CC(O)=O)c2cccnc2n1S(=O)(=O)c1ccc(Cl)c(Cl)c1
Cc1c(CC(O)=O)c2cccnc2n1S(=O)(=O)c1ccc(Cl)c(c1)C#N
Cc1c(CC(O)=O)c2cccnc2n1S(=O)(=O)c1ccc(F)c(c1)C#N
Cc1c(CC(O)=O)c2cccnc2n1S(=O)(=O)c1ccccc1
CCOc1cc(ccc1C#N)S(=O)(=O)n1c(C)c(CC(O)=O)c2cccnc12
Cc1c(CC(O)=O)c2cccnc2n1S(=O)(=O)c1cccc(Cl)c1
Cc1c(CC(O)=O)c2cccnc2n1S(=O)(=O)c1ccc(C)cc1
COc1cc(ccc1F)S(=O)(=O)n1c(C)c(CC(O)=O)c2cccnc12
Cc1c(CC(O)=O)c2cccnc2n1S(=O)(=O)c1ccc(cc1)[N+]([O-])=O
Cc1c(CC(O)=O)c2cccnc2n1S(=O)(=O)c1ccc(F)c(Cl)c1
Cc1c(CC(O)=O)c2cccnc2n1S(=O)(=O)c1ccc(Cl)c(c1)C(F)(F)F
CN([C@@H]1CCc2c(CC(O)=O)c3ccccn3c2C1)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(C1)c1nccnc1n2CC(O)=O)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(C1)c1cccnc1n2CC(O)=O)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(C1)c1ccncc1n2CC(O)=O)S(=O)(=O)c1ccc(F)cc1 |r|
CN(C)c1nc(Cc2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2)nc(N(C)C)c1CC(O)=O
CN([C@@H]1CCc2c(CC(O)=O)c3ncccc3n2C1)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(C1)c1ncccc1n2CC(O)=O)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)S(=O)(=O)c1ccc(F)cc1 |r|
Cc1c(Cc2ccc3ccccc3n2)c2cc(F)ccc2n1CC(O)=O
CN([C@@H]1CCc2c(CC(O)=O)n3ccccc3c2C1)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCC2=C(C1)C1C=CC=CC1N2CC(O)=O)S(=O)(=O)c1ccc(F)cc1 |r,c:5,10,12|
OC(=O)c1ccc(CNC(=O)c2c(Cl)sc(Cl)c2Cc2cccc(Cl)c2)cc1
C[C@H](NC(=O)c1c(C)sc(C)c1Cc1ccc(Cl)cc1)c1ccc(cc1)C(O)=O |r|
C[C@H](NC(=O)c1c(C)sc(C)c1Cc1ccc(cc1)C(F)(F)F)c1ccc(cc1)C(O)=O |r|
C[C@H](NC(=O)c1cscc1Cc1cccc(Cl)c1)c1ccc(cc1)C(O)=O |r|
C[C@H](NC(=O)c1c(C)sc(C)c1Cc1cccc(Cl)c1)c1ccc(cc1)C(O)=O |r|
C[C@H](NC(=O)c1c(Cl)sc(Cl)c1Cc1cccc(Cl)c1)c1ccc(cc1)C(O)=O |r|
C[C@H](NC(=O)c1c(C)sc(C)c1Cc1cccc(c1)C(F)(F)F)c1ccc(cc1)C(O)=O |r|
Cc1sc(C)c(C(=O)NC2(CC2)c2ccc(cc2)C(O)=O)c1Cc1cccc(c1)C(F)(F)F
Cc1sc(C)c(C(=O)NC2(CC2)c2ccc(cc2)C(O)=O)c1Cc1ccc(cc1)C(F)(F)F
Cc1sc(C)c(C(=O)NC2(CC2)c2ccc(cc2)-c2nnn[nH]2)c1Cc1ccc(cc1)C(F)(F)F
C[C@@H](NC(=O)c1c(Cl)sc(Cl)c1Cc1cccc(Cl)c1)c1ccc(cc1)C(O)=O |r|
OC(=O)Cc1sc(nc1-c1ccccc1)-c1ccccc1
COc1ccccc1Nc1nc(c(CC(O)=O)s1)-c1ccc(Cl)cc1
COc1ccccc1Nc1nc(c(CC(O)=O)s1)-c1ccc(cc1)-c1ccccc1
OC(=O)Cc1sc(nc1-c1ccc(F)cc1)-c1ccccc1
COc1ccc(cc1)-c1nc(sc1CC(O)=O)-c1ccc(Cl)cc1
Cc1ccc(-c2nc(sc2CC(O)=O)-c2ccc(Cl)cc2)c(C)c1
CN(C)c1ccc(cc1)-c1nc(c(CC(O)=O)s1)-c1ccc(Br)cc1
COc1ccc(cc1)-c1nc(c(CC(O)=O)s1)-c1ccc(Br)cc1
COc1ccc(cc1)-c1nc(Cc2ccc(Cl)cc2)sc1CC(O)=O
OC(=O)Cc1sc(Nc2ccccc2)nc1-c1ccccc1
COc1ccc(cc1)-c1nc(c(CC(O)=O)s1)-c1ccccc1
COc1ccc(cc1)-c1nc(sc1CC(O)=O)-c1ccc(Oc2ccccc2)cc1
OC(=O)Cc1sc(nc1-c1ccccc1)-c1ccc(Oc2ccccc2)cc1
COc1ccc(Cc2nc(c(CC(O)=O)s2)-c2ccccc2)cc1OC
OC(=O)Cc1sc(Cc2ccc(Cl)cc2)nc1-c1ccccc1
Cc1ccc(Cc2nc(c(CC(O)=O)s2)-c2ccccc2)cc1
OC(=O)Cc1sc(Nc2ccc3ccccc3c2)nc1-c1ccc(Oc2ccccc2)cc1
OC(=O)Cc1sc(Cc2ccc(Cl)cc2)nc1-c1ccc(Cl)cc1
COc1ccccc1Nc1nc(c(CC(O)=O)s1)-c1ccc(Oc2ccccc2)cc1
OC(=O)Cc1sc(Cc2ccccc2-c2ccc3OCOc3c2)nc1-c1ccc(F)cc1
OC(=O)Cc1sc(Nc2ccc(Cl)cc2)nc1-c1ccc(cc1)-c1ccccc1
OC(=O)Cc1sc(Nc2ccc(Cl)cc2)nc1-c1ccc(F)cc1
OC(=O)Cc1sc(Nc2ccc3ccccc3c2)nc1-c1ccc(Br)cc1
COc1ccccc1-c1ccccc1Cc1nc(c(CC(O)=O)s1)-c1ccc(F)cc1
OC(=O)Cc1sc(Cc2ccccc2-c2cccc(OC(F)(F)F)c2)nc1-c1ccc(F)cc1
COc1cccc(c1)-c1ccccc1Cc1nc(c(CC(O)=O)s1)-c1ccc(F)cc1
OC(=O)Cc1sc(Nc2ccccc2F)nc1-c1ccc(Oc2ccccc2)cc1
OC(=O)Cc1sc(Cc2ccccc2Br)nc1-c1ccc(F)cc1
OC(=O)Cc1sc(Nc2ccc(F)cc2)nc1-c1ccc(Oc2ccccc2)cc1
OC(=O)Cc1sc(Cc2ccccc2-c2ccccc2)nc1-c1ccc(F)cc1
OC(=O)Cc1sc(Nc2ccccc2Cl)nc1-c1ccc(Oc2ccccc2)cc1
OC(=O)Cc1sc(Cc2ccccc2)nc1-c1ccc(F)cc1
OC(=O)Cc1sc(Nc2ccccc2)nc1-c1ccc(cc1)-c1ccccc1
COc1ccccc1Nc1nc(c(CC(O)=O)s1)-c1ccc(F)cc1
OC(=O)Cc1sc(Nc2ccccc2)nc1-c1ccc(F)cc1
COc1ccc(cc1)-c1nc(Nc2ccccc2)sc1CC(O)=O
COc1ccccc1-c1nc(c(CC(O)=O)s1)-c1ccc(Br)cc1
COc1ccc(cc1)-c1nc(c(CC(O)=O)s1)-c1ccc(OC)cc1
CCc1ccc(cc1)-c1nc(sc1CC(O)=O)-c1ccccc1OC
Cc1ccc(Nc2nc(c(CC(O)=O)s2)-c2ccc(Cl)cc2)cc1
CC(C)c1ccc(Nc2nc(c(CC(O)=O)s2)-c2ccc(Cl)cc2)cc1
OC(=O)Cc1sc(Nc2ccc(cc2)C(F)(F)F)nc1-c1ccc(Cl)cc1
OC(=O)Cc1sc(nc1-c1ccccc1)-c1ccc(F)cc1
OC(=O)Cc1sc(nc1-c1ccc(cc1)-c1ccccc1)-c1ccccc1
OC(=O)Cc1sc(nc1-c1ccccc1)-c1ccc(Cl)cc1
OC(=O)Cc1sc(Cc2ccc3ccccc3c2)nc1-c1ccc(Cl)cc1
CCc1ccc(cc1)-c1nc(sc1CC(O)=O)-c1ccccc1
OC(=O)Cc1sc(Cc2ccccc2Oc2ccccc2)nc1-c1ccc(Cl)cc1
COc1ccc(cc1)-c1nc(sc1CC(O)=O)-c1ccccc1
OC(=O)Cc1sc(Cc2ccc(Cl)cc2)nc1-c1ccc(Oc2ccccc2)cc1
OC(=O)Cc1sc(Cc2ccccc2-c2ccc(cc2)C#N)nc1-c1ccc(F)cc1
COc1ccc(cc1)-c1ccccc1Cc1nc(c(CC(O)=O)s1)-c1ccc(F)cc1
OC(=O)Cc1sc(Nc2ccccc2)nc1-c1ccc(Oc2ccccc2)cc1
OC(=O)Cc1sc(Cc2ccccc2-c2cccc(c2)C#N)nc1-c1ccc(F)cc1
COc1ccc(Nc2nc(c(CC(O)=O)s2)-c2ccccc2)cc1
CC1CC(N(C(C)=O)c2ccccc2)c2ccccc2N1Cc1ccccc1
COc1cccc(c1)C(=O)N1[C@@H](C)C[C@@H](N(C(C)=O)c2ccccc2)c2ccccc12 |r|
CC1CC(N(C(C)=O)c2ccccc2)c2ccccc2N1C(=O)c1cccc(C)c1
CC1CC(N(C(C)=O)c2ccccc2)c2ccccc2N1S(=O)(=O)c1ccccc1
C[C@H]1C[C@@H](N(C(=O)CCC(O)=O)c2ccccc2)c2ccccc2N1C(=O)c1ccccc1 |r|
C[C@@H]1C[C@H](N(C(=O)CCC(O)=O)c2ccccc2)c2ccccc2N1C(=O)c1ccccc1 |r|
CC1CC(N(C(C)=O)c2ccccc2)c2ccccc2N1C(=O)\C=C\c1ccccc1
CC1CC(N(C(C)=O)c2ccccc2)c2ccccc2N1C(=O)OCc1ccccc1
CC1CC(N(C(C)=O)c2ccccc2)c2ccccc2N1C(=O)Cc1ccccc1
CC1CC(N(C(C)=O)c2ccccc2)c2ccccc2N1C(=O)c1ccc(C)c(C)c1
CC1CC(N(C(C)=O)c2ccccc2)c2ccccc2N1C(=O)c1ccc(Oc2ccccc2)cc1
CC1CC(N(C(C)=O)c2ccccc2)c2ccccc2N1C(=O)c1ccccc1C
CC1CC(N(C(C)=O)c2ccccc2)c2ccccc2N1C(=O)c1ccc(C)cc1
CCN(C1CC(C)N(C(=O)c2ccccc2)c2ccccc12)C(C)=O
CC1CC(NC(C)=O)c2ccccc2N1C(=O)c1ccccc1
C[C@@H]1C[C@H](N(C(C)=O)c2ccccc2)c2ccccc2N1C(=O)c1cccc(OC(F)(F)F)c1 |r|
CC1CC(N(C(=O)c2cccc(c2)C(O)=O)c2ccccc2)c2ccccc2N1C(=O)c1ccccc1
C[C@H]1C[C@@H](N(C(C)=O)c2ccccc2)c2ccccc2N1C(=O)c1cccc(OC(F)(F)F)c1 |r|
CC1CC(N(C(=O)\C=C\C(O)=O)c2ccccc2)c2ccccc2N1C(=O)c1ccccc1
COc1cccc(c1)C(=O)N1[C@H](C)C[C@H](N(C(C)=O)c2ccccc2)c2ccccc12 |r|
CC1CC(N(C(=O)CCCC(O)=O)c2ccccc2)c2ccccc2N1C(=O)c1ccccc1
CC1CC(N(C(C)=O)c2ccccc2)c2ccccc2N1
CC1CC(N(C(=O)CCC(O)=O)c2ccccc2)c2ccccc2N1C(=O)c1ccccc1
C[C@H]1C[C@@H](N(C(C)=O)c2ccccc2)c2ccccc2N1C(=O)c1ccccc1 |r|
CC1CC(N(Cc2ccccc2)C(C)=O)c2ccccc2N1C(=O)c1ccccc1
CC1CC(N(C(=O)CC(O)=O)c2ccccc2)c2ccccc2N1C(=O)c1ccccc1
C[C@@H]1C[C@H](N(C(C)=O)c2ccccc2)c2ccccc2N1C(=O)c1ccccc1 |r|
COc1ccc(cc1)C(=O)N1C(C)CC(N(C(C)=O)c2ccccc2)c2ccccc12
CC1CC(N(C(C)=O)c2ccccc2)c2ccccc2N1C(=O)c1ccc(OC(F)(F)F)cc1
CC1CC(N(C(C)=O)c2ccccc2)c2ccccc2N1C(=O)c1ccc(cc1)C(C)(C)C
CC1CC(N(C(C)=O)c2ccccc2)c2ccccc2N1C(=O)c1ccc(Cl)cc1
CC1CC(N(c2ccccc2)S(=O)(=O)c2ccccc2)c2ccccc2N1C(=O)c1ccccc1
CCN(C1CC(C)N(C(=O)c2ccccc2)c2ccccc12)c1ccccc1
C[C@@H]1C[C@H](Nc2ccccc2)c2ccccc2N1C(=O)c1ccccc1
CC1CC(N(C(=O)CCC(=O)ON)c2ccccc2)c2ccccc2N1C(=O)c1ccccc1
C[C@H]1C[C@H](N(C(C)=O)c2ccccc2)c2ccccc2N1C(=O)c1ccccc1 |r|
CCCCC(=O)N1C(C)CC(N(C(C)=O)c2ccccc2)c2ccccc12
CCCCC(=O)N(C1CC(C)N(C(=O)c2ccccc2)c2ccccc12)c1ccccc1
CC1CC(N(C(=O)c2ccccc2)c2ccccc2)c2ccccc2N1C(=O)c1ccccc1
OC(=O)CCc1sc(nc1-c1cccc(F)c1)C(c1ccc(F)cc1)c1ccc(F)cc1
COc1ccc(cc1)N(c1ccc(OC)cc1)c1ncc(CC(O)=O)c(n1)-c1cccc(F)c1
OC(=O)Cc1cnc(nc1-c1cccc(F)c1)N(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)Cc1sc(nc1-c1ccc(F)cc1)N(c1ccccc1)c1cccnc1
OC(=O)Cc1sc(nc1-c1ccc(F)cc1)N(c1ccccc1)c1ccc(cc1)C#N
CC(c1nc(c(CC(O)=O)s1)-c1ccc(F)cc1)(c1ccccc1)c1ccccc1
OC(=O)Cc1sc(nc1-c1ccc(Cl)cc1)N(c1ccccc1)c1ccccc1
OC(=O)Cc1sc(nc1-c1ccc(F)cc1)N(c1ccccc1)c1ccccc1
OC(=O)Cc1sc(nc1-c1ccc(F)cc1)N(c1ccc(F)cc1)c1ccc(F)cc1
CS(=O)(=O)c1ccc(cc1)N(c1nc(c(CC(O)=O)s1)-c1ccc(F)cc1)c1ccccc1
OC(=O)Cc1cnc(nc1-c1cccc(F)c1)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)COc1sc(nc1-c1cccc(F)c1)C(c1ccc(F)cc1)c1ccc(F)cc1
COc1ccc(cc1)N(c1nc(c(CC(O)=O)s1)-c1cccc(F)c1)c1ccc(OC)cc1
OC(=O)Cc1[nH]c(nc1-c1ccc(F)cc1)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)CCc1cnc(nc1-c1cccc(F)c1)C(c1ccc(F)cc1)c1ccc(F)cc1
OC(=O)Cc1sc(nc1-c1cccc(F)c1)N(c1ccccc1)c1ccccc1
Cc1c(C2NS(=O)(=O)c3ccccc23)c2cc(Cl)ccc2n1CC(O)=O
Cc1c(C2NS(=O)(=O)c3ccccc23)c2cc(C)ccc2n1CC(O)=O
CC(C)CCN1C(c2ccccc2S1(=O)=O)c1cn(CC(O)=O)c2ccccc12
CN1C(c2ccccc2S1(=O)=O)c1cn(CC(O)=O)c2ccccc12
Cc1noc(C)c1CN1C(C)(c2ccccc2S1(=O)=O)c1c(C)n(CC(O)=O)c2ccccc12
Cc1c(C2NS(=O)(=O)c3ccccc23)c2cc(F)ccc2n1CC(O)=O
Cc1c(C2N(CCOc3ccc(Cl)cc3)S(=O)(=O)c3ccccc23)c2ccccc2n1CC(O)=O
Cc1c(C2N(CCOc3ccccc3)S(=O)(=O)c3ccccc23)c2ccccc2n1CC(O)=O
OC(=O)Cn1cc(C2NS(=O)(=O)c3ccccc23)c2cc(ccc12)C#N
Cc1noc(C)c1CN1C(c2ccccc2S1(=O)=O)c1c(C)n(CC(O)=O)c2ccccc12
Cc1c(C2N(CCO)S(=O)(=O)c3ccccc23)c2ccccc2n1CC(O)=O
Cc1c(C2NS(=O)(=O)c3ccccc23)c2ccccc2n1CC(O)=O
Cc1c(C2N(c3ccccc3)S(=O)(=O)c3ccccc23)c2ccccc2n1CC(O)=O
CC(C)N1C(c2ccccc2S1(=O)=O)c1c(C)n(CC(O)=O)c2ccccc12
CC(C)CCN1C(c2ccccc2S1(=O)=O)c1c(C)n(CC(O)=O)c2ccccc12
Cc1noc(C)c1CN1C(c2ccccc2S1(=O)=O)c1c(C)n(CC(O)=O)c2ccc(Cl)cc12
OC(=O)Cn1cc(C2NS(=O)(=O)c3ccccc23)c2ccccc12
Cc1ccc2n(CC(O)=O)cc(C3NS(=O)(=O)c4ccccc34)c2c1
OC(=O)Cn1cc(C2NS(=O)(=O)c3ccccc23)c2cc(Cl)ccc12
Cc1noc(c1CN1C(c2ccccc2S1(=O)=O)c1c(C)n(CC(O)=O)c2ccccc12)-c1ccccc1
Cc1c(C2N(CCCOc3ccccc3)S(=O)(=O)c3ccccc23)c2ccccc2n1CC(O)=O
Cc1c(C2N(CCc3ccccc3)S(=O)(=O)c3ccccc23)c2ccccc2n1CC(O)=O
Cc1noc(C)c1CN1C(c2ccccc2S1(=O)=O)c1cn(CC(O)=O)c2ccccc12
OC(=O)Cn1cc(C2N(CCc3ccccc3)S(=O)(=O)c3ccccc23)c2ccccc12
OC(=O)Cn1cc(C2N(Cc3ccccc3)S(=O)(=O)c3ccccc23)c2ccccc12
Cc1noc(C)c1CN1C(CCS1(=O)=O)c1c(C)n(CC(O)=O)c2ccccc12
OC(=O)c1ccc(cc1)C1(CC1)NC(=O)c1cccc2ccn(Cc3ccc(cc3)C(F)(F)F)c12
CN([C@@H]1CCc2c(CC(O)=O)c3cccnc3n2C1)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccc(nc3n2C1)-c1ccc(F)cc1)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccc(Cl)nc3n2C1)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccncc3n2C1)S(=O)(=O)c1ccc(F)cc1 |r|
C[C@@H](C(=O)N(C)[C@@H]1CCc2c(CC(O)=O)c3cccnc3n2C1)c1ccc(F)cc1 |r|
C[C@H](C(=O)N(C)[C@@H]1CCc2c(CC(O)=O)c3cccnc3n2C1)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3cnccc3n2C1)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3cccnc3n2C1)C(=O)C1(CC1(C)C)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3cccnc3n2C1)C(=O)C(C)(C)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3cccnc3n2C1)C(=O)C1(CCC1)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3cccnc3n2C1)C(=O)C1(CC1)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3cccnc3n2C1)C(=O)C1(CCCC1)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3cccnc3n2C1)C(=O)C1(CCOCC1)c1ccc(F)cc1 |r|
CN(C)C(=O)c1sc2c(C)cc(C)cc2c1-c1ccc(CCNC(=O)NS(=O)(=O)c2ccc(C)cc2)cc1
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)S(=O)(=O)Cc1ccc(F)cc1 |r|
CCc1ccc(cc1)S(=O)(=O)N(C)[C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccc(F)c(F)c3n2C1)S(=O)(=O)c1ccc(F)cc1 |r|
COc1ccc(cc1)S(=O)(=O)N(C)[C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)S(=O)(=O)c1ccc(cc1)C(F)(F)F |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccc(cc3n2C1)-c1ccccc1)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccc(cc3n2C1)S(C)(=O)=O)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccc(cc3n2C1)C(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)S(=O)(=O)c1ccccc1C |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccc(Cl)cc3n2C1)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)S(=O)(=O)c1ccccc1F |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)S(=O)(=O)c1cccc(C)c1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)S(=O)(=O)c1cccc(F)c1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)S(=O)(=O)c1ccc(Cl)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)S(=O)(=O)c1ccccc1 |r|
OC(=O)Cc1c2CC[C@H](Cn2c2ccccc12)N(CC(F)(F)F)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)S(=O)(=O)c1c(C)noc1C |r|
CN([C@@H]1CCc2c(CC(O)=O)c3cc(F)cc(F)c3n2C1)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)S(=O)(=O)c1cnn(C)c1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3cccc(F)c3n2C1)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)S(=O)(=O)c1ccc(Cl)s1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)S(=O)(=O)c1ccccn1 |r|
OC(=O)Cc1c2CC[C@H](Cn2c2ccccc12)N(Cc1ccc(F)cc1)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)Cc1c2CC[C@H](Cn2c2ccccc12)N(CC1CC1)S(=O)(=O)c1ccc(F)cc1 |r|
CCCCCN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)S(=O)(=O)c1ccc(F)cc1 |r|
CCN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccc(F)cc3n2C1)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3cc(F)ccc3n2C1)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccc(cc3n2C1)C#N)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3cc(F)c(F)cc3n2C1)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3cc(ccc3n2C1)S(C)(=O)=O)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3c(F)cccc3n2C1)S(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3c(Cl)cc(Cl)cc3n2C1)S(=O)(=O)c1ccc(F)cc1 |r|
OC(=O)Cc1c2CC[C@H](Cn2c2ccccc12)NS(=O)(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3cc(F)c(Cl)cc3n2C1)S(=O)(=O)c1ccc(F)cc1 |r|
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)-c1cnc2ccccc2c1)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)-c1ccc(F)cn1)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)C(O)=O)C(=O)OCc1ccccc1
CCOc1ccc(cn1)-c1ccc(c(CN(CC)C(=O)C2CC2)c1)-c1cc(CC([O-])=O)ccc1OC
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)-c1cnn(C)c1)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)C(C)(C)O)C(=O)OCc1ccccc1
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)-c1ncc(OC)cn1)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)S(C)(=O)=O)C(=O)OCc1ccccc1
CCN(Cc1cc(NC(C)=O)ccc1-c1cc(CC(O)=O)ccc1OC)C(=O)OCc1ccccc1
CCN(Cc1cc(F)ccc1-c1cc(CC(O)=O)ccc1OC)C(=O)OCc1ccccc1
CCN(Cc1cc(NS(=O)(=O)c2ccc(Cl)cc2)ccc1-c1cc(CC(O)=O)ccc1OC)C(=O)OCc1ccccc1
Cc1c(CC(O)=O)c2ccsc2n1Cc1ccc(cc1Cl)S(C)(=O)=O
Cc1c(CC(O)=O)c2ccsc2n1Cc1ccc(cc1)S(C)(=O)=O
CN(C1CCCCC1)S(=O)(=O)c1ccc(Cn2c(C)c(CC(O)=O)c3ccsc23)cc1
Cc1csc2n(c(C)c(CC(O)=O)c12)S(=O)(=O)c1ccc(cc1)S(C)(=O)=O
Cc1c(CC(O)=O)c2ccsc2n1S(=O)(=O)c1ccc(F)cc1
Cc1c(CC(O)=O)c2ccsc2n1S(=O)(=O)c1ccccc1
Cc1cc2c(CC(O)=O)c(C)n(Cc3ccc(cc3)S(C)(=O)=O)c2s1
Cc1c(CC(O)=O)c2ccsc2n1S(=O)(=O)c1ccc(cc1)C#N
Cc1csc2n(Cc3ccc(cc3)S(C)(=O)=O)c(C)c(CC(O)=O)c12
Cc1c(CC(O)=O)c2ccsc2n1S(=O)(=O)c1ccc(cc1)C(F)(F)F
Cc1c(CC(O)=O)c2ccsc2n1S(=O)(=O)c1ccc(cc1)S(C)(=O)=O
Cc1cc2c(CC(O)=O)c(C)n(Cc3ccc(cc3Cl)S(C)(=O)=O)c2s1
Cc1c(CC(O)=O)c2ccsc2n1S(=O)(=O)c1ccc(cc1)S(=O)(=O)N1CCCC1
CS(=O)(=O)c1ccc(cc1)S(=O)(=O)n1cc(CC(O)=O)c2sccc12
Cc1c(CC(O)=O)c2ccsc2n1S(=O)(=O)c1ccc(cc1)S(=O)(=O)N1CCOCC1
CS(=O)(=O)c1ccc(cc1)S(=O)(=O)n1cc(CC(O)=O)c2ccsc12
Cc1c(CC(O)=O)c2ccsc2n1Cc1ccc(cc1)S(=O)(=O)N1CCOCC1
CN(C)S(=O)(=O)c1ccc(Cn2c(C)c(CC(O)=O)c3ccsc23)cc1
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)Cc1ccccc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)Cc1ccc(F)cc1 |r|
C[C@@H](C(=O)N(C)[C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)c1ccc(F)cc1 |r|
CN(C)c1ccc(CC(=O)N(C)[C@@H]2CCc3c(CC(O)=O)c4ccccc4n3C2)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)C1(CC1)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)Cc1ccc(cc1)C(F)(F)F |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)C1(CCC1)c1ccc(F)cc1 |r|
COc1ccc(CC(=O)N(C)[C@@H]2CCc3c(CC(O)=O)c4ccccc4n3C2)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)C1(CCOCC1)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)Cc1ccc(Cl)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)c1ccc2ccccc2c1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)C(C)(C)c1ccc(F)cc1 |r|
C[C@H](C(=O)N(C)[C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)C1Cc2ccccc12 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)C1(CCCC1)c1ccc(F)cc1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)C1CCCc2ccccc12 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)C1CCc2ccccc12 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)Cc1ccc(F)cc1F |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)Cc1ccc(F)cc1C(F)(F)F |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)Cc1ccc(F)cc1Cl |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)c1cccc2ccccc12 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)C1CCCC1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)Cc1ccc(F)c(F)c1 |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)Cc1ccc(F)c(c1)C(F)(F)F |r|
CN([C@@H]1CCc2c(CC(O)=O)c3ccccc3n2C1)C(=O)Cc1ccc(F)c(Cl)c1 |r|
OC(=O)COc1ccc(cc1-c1ccccc1)C#N
OC(=O)COc1ccc(Br)cc1-c1ccccc1
OC(=O)COc1ccc(cc1-c1ccccc1)-c1nccs1
OC(=O)COc1ccc(cc1-c1cc(ccc1F)C#N)C(F)(F)F
CN(c1ccc(c(Cl)c1)-c1cc(F)ccc1OCC(O)=O)S(C)(=O)=O
Cc1ccc(OCC(O)=O)c(c1)-c1ccccc1
CCS(=O)(=O)c1ccc(c(C)c1)-c1cc(ccc1OCC(O)=O)C(F)(F)F
OC(=O)COc1ccc(cc1-c1ccccc1)[N+]([O-])=O
OC(=O)COc1ccc(Cl)cc1-c1cccc(c1)C#N
CN(c1ccc(cc1)-c1cc(ccc1OCC(O)=O)C(F)(F)F)S(C)(=O)=O
OC(=O)COc1ccc(cc1-c1ccc(cc1)C#N)C(F)(F)F
CCS(=O)(=O)c1cccc(c1)-c1cc(ccc1OCC(O)=O)C(F)(F)F
OC(=O)COc1ccc(cc1-c1cccc(c1)C#N)C(F)(F)F
CCCCOc1ccccc1-c1cc(ccc1OCC(O)=O)C(F)(F)F
OC(=O)COc1ccc(cc1-c1ccccc1-c1ccccc1)C(F)(F)F
CN(c1ccc(c(C)c1)-c1cc(ccc1OCC(O)=O)C(F)(F)F)S(C)(=O)=O
CN(c1ccc(c(Cl)c1)-c1cc(ccc1OCC(O)=O)C(F)(F)F)S(C)(=O)=O
C[C@@H](Oc1ccc(cc1-c1cccc(c1)C#N)C(F)(F)F)C(O)=O |r|
OC(=O)COc1ccc(cc1-c1ccc(Cl)cc1)C(F)(F)F
CCS(=O)(=O)c1ccc(c(Cl)c1)-c1cc(ccc1O[C@H](C)C(O)=O)C(F)(F)F |r|
CCN(CC)S(=O)(=O)c1ccc(cc1)-c1cc(ccc1OCC(O)=O)C(F)(F)F
COc1ccc(cc1)-c1cc(ccc1OCC(O)=O)C(F)(F)F
Nc1ccc(OCC(O)=O)c(c1)-c1ccccc1
CS(=O)(=O)c1ccc(OCC(O)=O)c(c1)-c1ccccc1
CCSc1ccc(cc1)-c1cc(ccc1OCC(O)=O)C(F)(F)F
CS(=O)(=O)c1ccc(cc1)-c1cc(ccc1OCC(O)=O)C(F)(F)F
CCS(=O)(=O)c1ccc(c(C)c1)-c1cc(Cl)ccc1OCC(O)=O
OC(=O)COc1ccc(Cl)cc1-c1ccccc1
CCS(=O)(=O)c1ccc(-c2cc(Cl)ccc2OCC(O)=O)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(c(Cl)c1)-c1cc(Cl)ccc1OCC(O)=O
OC(=O)COc1ccc(cc1-c1ccccc1)C(F)(F)F
CCS(=O)(=O)c1ccc(c(C)c1)-c1cc(ccc1O[C@@H](C)C(O)=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(c(C)c1)-c1cc(ccc1O[C@H](C)C(O)=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(c(C)c1)-c1cc(ccc1OC(C)(C)C(O)=O)C(F)(F)F
CCC(Oc1ccc(cc1-c1ccc(cc1C)S(=O)(=O)CC)C(F)(F)F)C(O)=O
CCS(=O)(=O)c1ccc(c(C)c1)-c1cc(ccc1OCC(N)=O)C(F)(F)F
CCS(=O)(=O)c1ccc(c(C)c1)-c1cc(ccc1CCC(O)=O)C(F)(F)F
CCS(=O)(=O)c1ccc(c(C)c1)-c1cc(ccc1OCc1nnn[nH]1)C(F)(F)F
Cc1ccc(cc1-c1cc(ccc1OCC(O)=O)C(F)(F)F)C#N
CCS(=O)(=O)c1ccc(c(Cl)c1)-c1cc(ccc1OCC(O)=O)C(F)(F)F
CS(=O)(=O)c1ccc(c(Cl)c1)-c1cc(ccc1OCC(O)=O)C(F)(F)F
OC(=O)COc1ccc(cc1-c1ccc2c(CCS2(=O)=O)c1)C(F)(F)F
CS(=O)(=O)c1ccc(c(Cl)c1)-c1cc(Cl)ccc1OCC(O)=O
CCS(=O)(=O)c1ccc(cc1)-c1cc(Cl)ccc1OCC(O)=O
CCS(=O)(=O)c1ccc(c(F)c1)-c1cc(Cl)ccc1OCC(O)=O
CCc1ccc(OCC(O)=O)c(c1)-c1ccc(cc1)S(C)(=O)=O
CCCS(=O)(=O)c1cccc(c1)C#Cc1c(OCC(O)=O)cccc1-c1ccccc1
CCNS(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CCCS(=O)(=O)c1cccc(c1)C#Cc1c(OCC(O)=O)cccc1-c1sc(C)nc1C
OC(=O)COc1ccc(Cl)cc1C#Cc1ccccc1Cl
OC(=O)COc1ccc(Cl)cc1C#Cc1ccccc1
OC(=O)COc1ccc(Cl)cc1C#Cc1cccc(Cl)c1
CC(C)N(C)S(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
OC(=O)COc1ccc(Cl)cc1C#Cc1ccc(Cl)cc1
COc1ccccc1C#Cc1cc(Cl)ccc1OCC(O)=O
CC(C)NS(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
OC(=O)COc1ccc(Cl)cc1C#Cc1ccccc1F
OC(=O)COc1ccc(Cl)cc1C#Cc1ccccc1C(F)(F)F
CCCS(=O)(=O)c1cccc(c1)C#Cc1c(OCC(O)=O)cccc1-c1ccsc1
CCCS(=O)(=O)c1cccc(c1)C#Cc1c(OCC(O)=O)cccc1-c1cccs1
CCCS(=O)(=O)c1ccc(F)c(c1)C#Cc1cc(Cl)ccc1OC(C)C(O)=O
CN(C)S(=O)(=O)c1ccc(F)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CCCS(=O)(=O)c1ccc(F)c(c1)C#Cc1cc(Cl)ccc1OC(C)(C)C(O)=O
CN(C)S(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CCCS(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OC(C)C(O)=O
CCCS(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OC(CC)C(O)=O
CCCC(Oc1ccc(Cl)cc1C#Cc1cc(ccc1C)S(=O)(=O)CCC)C(O)=O
CCCS(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OC(CC(C)C)C(O)=O
OC(=O)COc1ccc(Cl)cc1C#Cc1cccc(c1)C(F)(F)F
OC(=O)COc1ccc(Cl)cc1C#Cc1ccc(F)cc1F
OC(=O)COc1ccc(Cl)cc1C#Cc1ccc(Cl)s1
Cn1ccnc1C#Cc1cc(Cl)ccc1OCC(O)=O
OCc1ccc(F)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
OCc1ccc(C#Cc2cc(Cl)ccc2OCC(O)=O)c(F)c1
OCc1cccc(C#Cc2cc(Cl)ccc2OCC(O)=O)c1F
COCc1ccc(F)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
COCc1ccc(C#Cc2cc(Cl)ccc2OCC(O)=O)c(F)c1
OC(=O)COc1ccc(Cl)cc1C#Cc1ccccn1
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)-c1ccc(OC)cn1)C(=O)C1CC1
COCCNS(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
COCCN(C)S(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CC1CCCCN1S(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CCCS(=O)(=O)c1cccc(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
OCCCS(=O)(=O)c1cccc(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
OCCS(=O)(=O)c1cccc(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
OC(=O)COc1ccc(Cl)cc1C#Cc1cccnc1
Cc1ccc(cc1C#Cc1cc(Cl)ccc1OCC(O)=O)S(C)(=O)=O
OC(=O)COc1ccc(Cl)cc1C#Cc1ccncc1
CS(=O)(=O)c1ccc(F)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
Cc1ncccc1C#Cc1cc(Cl)ccc1OCC(O)=O
CS(=O)(=O)c1ccc(Cl)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
Cc1ccncc1C#Cc1cc(Cl)ccc1OCC(O)=O
CCCc1ccc(cc1C#Cc1cc(Cl)ccc1OCC(O)=O)S(C)(=O)=O
CCCc1ccncc1C#Cc1cc(Cl)ccc1OCC(O)=O
CN(C)S(=O)(=O)c1cncc(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CC(C)Cc1ccncc1C#Cc1cc(Cl)ccc1OCC(O)=O
CCCCCCc1ccncc1C#Cc1cc(Cl)ccc1OCC(O)=O
OC(=O)COc1ccc(Cl)cc1C#Cc1ccc2-c3ccccc3S(=O)(=O)c2c1
Cc1cc[n+]([O-])cc1C#Cc1cc(Cl)ccc1OCC(O)=O
CS(=O)(=O)c1cccc(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CCCS(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CC(C)c1ccc(cc1C#Cc1cc(Cl)ccc1OCC(O)=O)S(C)(=O)=O
CCS(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CC(C)S(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CC(C)CS(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
Cc1ccc(cc1C#Cc1cc(Cl)ccc1OCC(O)=O)S(=O)(=O)Cc1ccccc1
Cc1ccc(cc1C#Cc1cc(Cl)ccc1OCC(O)=O)S(=O)(=O)CCc1ccccc1
Cc1ccc(cc1C#Cc1cc(Cl)ccc1OCC(O)=O)S(=O)(=O)c1ccccc1
Cc1ccc(cc1C#Cc1cc(Cl)ccc1OCC(O)=O)S(=O)(=O)CCO
Cc1ccc(cc1C#Cc1cc(Cl)ccc1OCC(O)=O)S(=O)(=O)CCCO
CCCS(=O)(=O)c1ccc(F)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CC(C)S(=O)(=O)c1ccc(F)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CCCS(=O)(=O)c1ccc(Cl)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CC(C)S(=O)(=O)c1ccc(Cl)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CN(C)S(=O)(=O)c1cccc(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CCN(CC)S(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CC1(C)C(=O)c2ccc(cc2S1(=O)=O)C#Cc1cc(Cl)ccc1OCC(O)=O
Cc1ccc(cc1C#Cc1cc(Cl)ccc1OCC(O)=O)S(=O)(=O)NC(C)(C)C
CC1(C)C(O)c2ccc(cc2S1(=O)=O)C#Cc1cc(Cl)ccc1OCC(O)=O
CNS(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CC1(C)C(C)(O)c2ccc(cc2S1(=O)=O)C#Cc1cc(Cl)ccc1OCC(O)=O
COC1c2ccc(cc2S(=O)(=O)C1(C)C)C#Cc1cc(Cl)ccc1OCC(O)=O
COC1(C)c2ccc(cc2S(=O)(=O)C1(C)C)C#Cc1cc(Cl)ccc1OCC(O)=O
CS(=O)(=O)c1cc(ccc1-c1ccccc1)C#Cc1cc(Cl)ccc1OCC(O)=O
COc1ccc(cc1)-c1ccc(cc1S(C)(=O)=O)C#Cc1cc(Cl)ccc1OCC(O)=O
COc1cccc(c1)-c1ccc(cc1S(C)(=O)=O)C#Cc1cc(Cl)ccc1OCC(O)=O
CC(C)CN(C)S(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
Cc1ccc(cc1C#Cc1cc(Cl)ccc1OCC(O)=O)S(=O)(=O)N1CCCCC1
Cc1ccc(cc1C#Cc1cc(Cl)ccc1OCC(O)=O)S(=O)(=O)N1CCOCC1
CN1CCN(CC1)S(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CN(C)CCCN(C)S(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CN(C)CCN(C)S(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CS(=O)(=O)c1ccc(cc1)C#Cc1cc(Cl)ccc1OCC(O)=O
CN(C)C(=O)c1ccc(cc1)C#Cc1cc(Cl)ccc1OCC(O)=O
CN(C)C(=O)c1cccc(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CS(=O)(=O)Cc1cccc(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CS(=O)c1cccc(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CS(=O)(=O)Nc1cccc(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CN(c1cccc(c1)C#Cc1cc(Cl)ccc1OCC(O)=O)S(C)(=O)=O
CS(=O)(=O)c1cncc(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CS(=O)(=O)c1cc(ccc1-c1ccc(cc1)C(F)(F)F)C#Cc1cc(Cl)ccc1OCC(O)=O
CS(=O)(=O)c1cc(ccc1-c1ccc(Cl)cc1)C#Cc1cc(Cl)ccc1OCC(O)=O
CS(=O)(=O)Nc1cncc(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CN(c1cncc(c1)C#Cc1cc(Cl)ccc1OCC(O)=O)S(C)(=O)=O
OCCNS(=O)(=O)c1cncc(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
OC(=O)COc1ccc(Cl)cc1C#Cc1cncc(c1)S(=O)(=O)N1CCOCC1
CN(C)S(=O)(=O)c1cnc(C)c(c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CS(=O)(=O)c1cc(ccc1-c1cccc(Cl)c1)C#Cc1cc(Cl)ccc1OCC(O)=O
CS(=O)(=O)c1cc(ccc1-c1ccccc1Cl)C#Cc1cc(Cl)ccc1OCC(O)=O
OC(=O)COc1ccc(Cl)cc1C#Cc1ccc2C=CS(=O)(=O)c2c1 |c:19|
OC(=O)COc1ccc(Cl)cc1C#Cc1ccc2CCS(=O)(=O)c2c1
CCCS(=O)(=O)c1cc(C#Cc2cc(Cl)ccc2OCC(O)=O)c(C)cc1NC(C)=O
CC(C)(C)N1C(=O)c2ccc(cc2S1(=O)=O)C#Cc1cc(Cl)ccc1OCC(O)=O
CC(C)S(=O)(=O)c1cc(ccc1C(=O)N(C)C)C#Cc1cc(Cl)ccc1OCC(O)=O
CCN(CC)C(=O)c1ccc(cc1S(=O)(=O)C(C)C)C#Cc1cc(Cl)ccc1OCC(O)=O
CC(C)S(=O)(=O)c1cc(ccc1C(=O)N1CCOCC1)C#Cc1cc(Cl)ccc1OCC(O)=O
OC(=O)COc1ccccc1C#Cc1ccccc1Cl
Cc1ccc(OCC(O)=O)c(c1)C#Cc1ccccc1Cl
CCCS(=O)(=O)c1cccc(c1)C#Cc1cc(F)ccc1OCC(O)=O
OC(=O)COc1cc(F)ccc1C#Cc1ccccc1Cl
CCCS(=O)(=O)c1cccc(c1)C#Cc1c(Cl)cccc1OCC(O)=O
CCCS(=O)(=O)c1cccc(c1)C#Cc1c(OCC(O)=O)ccc2ccccc12
OC(=O)COc1ccc(cc1C#Cc1ccccc1Cl)C(F)(F)F
CCCS(=O)(=O)c1cccc(c1)C#Cc1cc(ccc1OCC(O)=O)C(F)(F)F
OC(=O)COc1ccc(cc1C#Cc1ccccc1Cl)C#N
CCCS(=O)(=O)c1cccc(c1)C#Cc1cc(ccc1OCC(O)=O)C#N
CCCS(=O)(=O)c1ccc(C)c(c1)C#Cc1cc(ccc1OCC(O)=O)C#N
CC(C)c1ccc(cc1C#Cc1cc(ccc1OCC(O)=O)C#N)S(C)(=O)=O
Cc1c(Sc2ccc(Cl)cc2)c2c(C)c(F)ccc2n1CC(O)=O
CC(=O)Nc1cccc2n(CC(O)=O)c(C)c(Sc3ccc(Cl)cc3)c12
Cc1c(Sc2ccc(Cl)cc2)c2c(C#N)c(Cl)ccc2n1CC(O)=O
Cc1c(Sc2ccc(Cl)cc2)c2c(Cl)cccc2n1CC(O)=O
Cc1c(Sc2ccc(Cl)cc2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Sc2ccc(Cl)cc2)c2ccc(Cl)cc2n1CC(O)=O
Cc1c(Sc2ccc(Cl)cc2)c2c(Cl)nccc2n1CC(O)=O
Cc1c(Oc2ccc(Cl)cc2)c2c(cccc2n1CC(O)=O)-c1ccccc1
Cc1c(Sc2ccc(Cl)cc2)c2nc(C)ccc2n1CC(O)=O
Cc1c(Sc2ccccc2)c2cc(C)ccc2n1CC(O)=O
CCS(=O)(=O)c1ccc(Oc2c(C)n(CC(O)=O)c3ccc(cc23)C(F)(F)F)cc1
Cc1c(Sc2ccc(Cl)cc2)c2cc(C)ccc2n1CC(O)=O
Cc1c(Sc2ccc(Cl)cc2)c2cc(Cl)ccc2n1CC(O)=O
CCS(=O)(=O)Nc1cccc2n(CC(O)=O)c(C)c(Oc3ccc(Cl)cc3)c12
Cc1c(Oc2ccc(Cl)cc2)c2c(NS(C)(=O)=O)cccc2n1CC(O)=O
CC(=O)Nc1cccc2n(CC(O)=O)c(C)c(Oc3ccc(Cl)cc3)c12
Cc1c(Sc2ccc(Cl)cc2)c2cc(Cl)ccc2n1Cc1nnn[nH]1
Cc1c(Oc2ccc(Cl)cc2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Sc2ccc(Cl)cc2)c2cccc(Cl)c2n1CC(O)=O
Cc1c(Oc2ccc(Cl)cc2)c2cc(ccc2n1CC(O)=O)C(F)(F)F
OC(=O)Cn1cc(Sc2ccc(Cl)cc2)c2cc(Cl)ccc12
CC(C(O)=O)n1c(C)c(Sc2ccc(Cl)cc2)c2cc(Cl)ccc12
Cc1c(c2cc(C)ccc2n1CC(O)=O)S(=O)(=O)c1c(Cl)cccc1Cl
Cc1c(c2cc(C)ccc2n1CC(O)=O)S(=O)(=O)c1ccccc1Cl
Cc1c(c2cc(C)ccc2n1CC(O)=O)S(=O)(=O)c1cccc(Cl)c1
CC(=O)Nc1cccc2n(CC(O)=O)c(C)c(c12)S(=O)(=O)c1ccc(Cl)cc1
Cc1c(c2c(NS(C)(=O)=O)cccc2n1CC(O)=O)S(=O)(=O)c1ccc(Cl)cc1
Cc1c(c2cc(F)ccc2n1CC(O)=O)S(=O)(=O)c1ccc(Cl)cc1
COc1cccc(c1)S(=O)(=O)c1c(C)n(CC(O)=O)c2ccc(C)cc12
Cc1c(S(=O)c2ccc(Cl)cc2)c2cc(C)ccc2n1CC(O)=O
Cc1c(c2cc(C)ccc2n1CC(O)=O)S(=O)(=O)c1ccc(Cl)cc1
Cc1c(Sc2ccc(cc2)S(C)(=O)=O)c2cc(C)ccc2n1CC(O)=O
COc1ccc(Sc2c(C)n(CC(O)=O)c3ccc(C)cc23)cc1
Cc1c(Sc2ccccc2Cl)c2cc(C)ccc2n1CC(O)=O
Cc1c(Sc2ccc(Cl)cc2)c2c(cccc2n1CC(O)=O)-c1cnccn1
Cc1c(Sc2cccc(Cl)c2)c2cc(C)ccc2n1CC(O)=O
Cc1c(Sc2ccc(Cl)cc2)c2c(cccc2n1CC(O)=O)-c1ccccc1
Cc1c(Sc2ccc(Cl)cc2)c2cc(ccc2n1CC(O)=O)-c1ccccc1
CC(=O)Nc1ccc2n(CC(O)=O)c(C)c(Sc3ccc(Cl)cc3)c2c1
Cc1c(Sc2ccc(Cl)cc2)c2c(cccc2n1CC(O)=O)-c1nccs1
CCN(C(C)=O)c1cccc2n(CC(O)=O)c(C)c(Sc3ccc(Cl)cc3)c12
CNC(=O)c1cccc2n(CC(O)=O)c(C)c(Sc3ccc(Cl)cc3)c12
Cc1c(Sc2ccc(Cl)cc2)c2c(NS(C)(=O)=O)cccc2n1CC(O)=O
Cn1c(CC(O)=O)c(Sc2ccccc2)c2ccccc12
Cc1c(Sc2ccc(Cl)cc2)c2cc(ccc2n1CC(O)=O)S(C)(=O)=O
Cc1c(Sc2ccc(Cl)cc2)c2c(cccc2n1CC(O)=O)S(C)(=O)=O
Cc1c(Sc2ccc(Cl)cc2)c2cc(Cl)c(cc2n1CC(O)=O)C#N
Cc1c(Sc2ccc(Cl)cc2)c2ccc(cc2n1CC(O)=O)S(C)(=O)=O
COc1ccc(CC(O)=O)cc1-c1ccc(cc1CN(C1CCC1)C(=O)OCc1ccccc1)C(F)(F)F
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)C(F)(F)F)C(=O)OCc1ccc(Cl)cc1
COc1ccc(CC(O)=O)cc1-c1ccc(cc1CN(C1CC1)C(=O)OCc1ccccc1)C(F)(F)F
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)C(F)(F)F)C(=O)OCc1cccc(Cl)c1
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)C(F)(F)F)C(=O)OCc1ccccc1Cl
COc1ccc(CC(O)=O)cc1-c1ccc(cc1CNCCc1ccccc1)C(F)(F)F
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)C(F)(F)F)C(=O)OC
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)C(F)(F)F)C(=O)OCc1ccc(F)cc1
COc1ccc(CC(O)=O)cc1-c1ccc(cc1CN(C1CCCC1)C(=O)OCc1ccccc1)C(F)(F)F
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)C(F)(F)F)C(=O)OCc1cc(Cl)cc(Cl)c1
C[C@H]1[C@H](OC(=O)N1Cc1cc(ccc1-c1ccccc1CC(O)=O)C(F)(F)F)c1ccccc1 |r|
C[C@H]1[C@H](OC(=O)N1Cc1cc(ccc1-c1cccc(CCC(O)=O)c1)C(F)(F)F)c1ccccc1 |r|
C[C@H]1[C@H](OC(=O)N1Cc1cc(ccc1-c1cccc(c1)C(O)=O)C(F)(F)F)c1ccccc1 |r|
C[C@H]1[C@H](OC(=O)N1Cc1cc(ccc1-c1cccc(CC(O)=O)c1)C(F)(F)F)c1ccccc1 |r|
COc1ccc(CC(O)=O)cc1-c1ccc(cc1CN1[C@@H](C)[C@H](OC1=O)c1ccccc1)C(F)(F)F |r|
C[C@H]1[C@H](OC(=O)N1Cc1cc(ccc1-c1ccccc1CCC(O)=O)C(F)(F)F)c1ccccc1 |r|
COC(=O)N(Cc1ccccc1)Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)C(F)(F)F
COC(=O)N(CCc1ccccc1)Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)C(F)(F)F
COc1ccc(c(CN2[C@@H](C)[C@H](OC2=O)c2ccccc2)c1)-c1cc(CC(O)=O)ccc1OC |r|
COc1ccc(CC(O)=O)cc1-c1ccccc1CN1[C@@H](C)[C@H](OC1=O)c1ccccc1 |r|
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)C(F)(F)F)C(=O)OCc1ccccc1
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)C(F)(F)F)C(=O)OCc1cc(F)cc(F)c1
COc1ccc(CC(O)=O)cc1-c1ccc(F)cc1CN1[C@@H](C)[C@H](OC1=O)c1ccccc1 |r|
COc1ccc(CC(O)=O)cc1-c1ccc(cc1CN(C)C(=O)OCc1ccccc1)C(F)(F)F
C[C@H]1[C@H](OC(=O)N1Cc1cc(F)ccc1-c1ccc(CC(O)=O)cc1)c1ccccc1 |r|
COc1ccc(CC(O)=O)cc1-c1ccc(cc1CNC(=O)OCc1ccccc1)C(F)(F)F
CCC(=O)Nc1ccc(Oc2cc(CC(O)=O)ccc2OC)c(c1)C(=O)N[C@H](C)c1ccc(Cl)cc1 |r|
CCC(=O)Nc1ccc(Oc2cc(CC(O)=O)ccc2OC)c(c1)C(=O)NCc1ccc(Cl)cc1
CCNC(=O)c1ccc(Oc2cccc(CC(O)=O)c2)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(c1)S(=O)(=O)Nc1ccc(Cl)cc1
COc1cc(CC(O)=O)ccc1Oc1ccc(cc1CS(=O)(=O)c1ccc(Cl)cc1Cl)C(=O)NC1CCC1
CCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(NC(=O)NCc2ccc(Cl)cc2)c1
CCCCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(NCCc2ccccc2)c1
CCC(=O)Nc1ccc(Oc2cc(CC(O)=O)ccc2OC)c(c1)C(=O)NC(C)(C)Cc1ccc(F)cc1
CCNC(=O)c1ccc(Oc2c(OC)cc(CC(O)=O)cc2OC)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCC(=O)Nc1ccc(Oc2cc(CC(O)=O)ccc2OC)c(c1)C(=O)N[C@@H](C)c1ccc(Cl)cc1 |r|
CCC(=O)Nc1ccc(Oc2cc(CC(O)=O)ccc2OC)c(c1)C(=O)NCCc1ccc(F)cc1
CCC(=O)Nc1ccc(Oc2cc(CC(O)=O)ccc2OC)c(c1)C(=O)N[C@@H](C)c1ccccc1 |r|
CCCCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(NS(=O)(=O)c2ccc(Cl)cc2)c1
CCCCNC(=O)c1ccc(Oc2ccc(CC(=O)NS(C)(=O)=O)cc2OC)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCCNC(=O)c1ccc(Oc2ccc(Cc3nnn[nH]3)cc2OC)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCCNC(=O)c1ccc(Oc2ccc(cc2OC)C(F)(F)C(O)=O)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCCNC(=O)c1ccc(Oc2ccc(cc2OC)C2(CCCC2)C(O)=O)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCCNC(=O)c1ccc(Oc2ccc(cc2OC)C2(CC2)C(O)=O)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(NCc2ccc(Cl)cc2)c1
Cc1ccc(cc1)C(c1ccc(C)cc1)c1ccc(=O)n(CCCc2cccc(OCC(O)=O)c2)c1
OC(=O)COc1cccc(CCCn2cc(ccc2=O)C(c2ccc(Cl)cc2)c2ccc(Cl)cc2)c1
OC(=O)COc1cccc(OCCn2cc(ccc2=O)C(c2ccccc2)c2ccccc2)c1
COc1ccc(cc1)C(c1ccc(OC)cc1)c1ccc(=O)n(CCCc2cccc(OCC(O)=O)c2)c1
COc1ccc(cc1)C(=O)N(CCCc1cccc(OCC(O)=O)c1)CCC(c1ccccc1)c1ccccc1
OC(=O)COc1cccc(CCCn2nc(ccc2=O)C(c2ccccc2)c2ccccc2)c1
OC(=O)COc1cccc(CCCN(CCC(c2ccccc2)c2ccccc2)C(=O)c2ccccc2)c1
OC(=O)COc1cccc(CCCn2cc(ccc2=O)C(c2ccccc2)c2ccccc2)c1
OC(=O)CCCOc1cccc(CCCn2nc(ccc2=O)C(c2ccccc2)c2ccccc2)c1
OC(=O)COc1cccc(CCCn2cc(ccc2=O)C(c2ccc(F)cc2)c2ccc(F)cc2)c1
CCC(Oc1cccc(CCCn2cc(ccc2=O)C(c2ccccc2)c2ccccc2)c1)C(O)=O
CC(Oc1cccc(CCCn2cc(ccc2=O)C(c2ccccc2)c2ccccc2)c1)C(O)=O
OC(=O)CCCOc1cccc(CCCn2cc(ccc2=O)C(c2ccccc2)c2ccccc2)c1
CCCCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(NS(=O)(=O)c2ccc(cc2Cl)C(F)(F)F)c1
COc1cc(CC(O)=O)ccc1Oc1ccc(cc1NS(=O)(=O)c1ccc(Cl)cc1Cl)C(=O)NC1CC1
OC(=O)Cc1cc(F)c(Oc2ccc(cc2NS(=O)(=O)c2ccc(OC(F)(F)F)cc2Cl)C(=O)NC2CCC2)cc1F
OC(=O)Cc1cc(Cl)c(Oc2ccc(cc2NS(=O)(=O)c2ccc(OC(F)(F)F)cc2Cl)C(=O)NC2CCC2)cc1F
CC(C)(C)NC(=O)c1ccc(Oc2cc(F)c(CC(O)=O)cc2Cl)c(NS(=O)(=O)c2ccc(OC(F)(F)F)cc2Cl)c1
CC(C)(C)NC(=O)c1ccc(Oc2cc(F)c(CC(O)=O)cc2Cl)c(NS(=O)(=O)c2ccc(cc2Cl)C2CC2)c1
CCCCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2C)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2Cl)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2F)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2C#N)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCCNC(=O)c1ccc(Oc2cc(F)c(CC(O)=O)cc2F)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
OC(=O)Cc1ccc(Oc2ccc(cc2NS(=O)(=O)c2ccc(Cl)cc2Cl)C(=O)NC2CC2)c(Cl)c1
OC(=O)Cc1ccc(Oc2ccc(cc2NS(=O)(=O)c2ccc(Cl)cc2Cl)C(=O)NC2CCC2)c(Cl)c1
CC(C)(C)NC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2Cl)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
COc1cc(CC(O)=O)ccc1Oc1ccc(cc1NS(=O)(=O)c1ccc(cc1Cl)C(F)(F)F)C(=O)NC1CCC1
OC(=O)Cc1cc(F)c(Oc2ccc(cc2NS(=O)(=O)c2ccc(cc2Cl)C(F)(F)F)C(=O)NC2CCC2)cc1F
CCCCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(NS(=O)(=O)c2cc(Cl)cc(Cl)c2)c1
CCCCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(NS(=O)(=O)c2cccc(Cl)c2Cl)c1
CCCCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(NS(=O)(=O)c2c(Cl)cccc2Cl)c1
OC(=O)Cc1ccc(Oc2ccc(cc2NS(=O)(=O)c2ccc(Cl)cc2)C(=O)NC2CCC2)c(Cl)c1
CC(C)(C)NC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2Cl)c(NS(=O)(=O)c2ccc(Cl)cc2)c1
CCCCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(NS(=O)(=O)c2ccc(Cl)c(Cl)c2)c1
CCCCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(NS(=O)(=O)c2cc(Cl)ccc2Cl)c1
CCCCNC(=O)c1ccc(Oc2ccc3C(CC(O)=O)COc3c2)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCc1cc(n[nH]1)-c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCCNC(=O)c1ccc(Oc2ccc3n(CC(O)=O)ccc3c2)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCCNC(=O)c1ccc(Oc2ccc3c(CC(O)=O)c[nH]c3c2)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCc1nc(c[nH]1)-c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCCNC(=O)c1ccc(c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1)S(=O)c1ccc(CC(O)=O)cc1
CCCCNC(=O)c1ccc(Sc2ccc(CC(O)=O)cc2)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCCNC(=O)c1ccc(Cc2ccc(CC(O)=O)cc2OC)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCCNC(=O)c1ccc(Oc2ccc3c(CC(O)=O)coc3c2)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCCNC(=O)c1ccc(Oc2ccc(CC(O)=O)nc2)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCc1nnc([nH]1)-c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cn2)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCc1noc(n1)-c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCc1nnc([nH]1)-c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCCNC(=O)c1ccc(c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1)S(=O)(=O)c1ccc(CC(O)=O)cc1
Cc1c(Cc2ccccc2S(=O)(=O)c2ccccc2)c2c(CCNC2=O)n1CC(O)=O
COc1ccc(c(Cc2c(C)n(CC(O)=O)c3CCNC(=O)c23)c1)S(=O)(=O)c1ccc(F)cc1
Cc1c(Cc2ccccc2S(=O)(=O)c2ccccc2)c2c(CC(C)(C)NC2=O)n1CC(O)=O
COc1cccc(Cc2c(C)n(CC(O)=O)c3CCNC(=O)c23)c1S(=O)(=O)c1ccccc1
Cc1c(Cc2ccc(cc2S(=O)(=O)c2ccccc2)C(F)(F)F)c2c(CCNC2=O)n1CC(O)=O
Cc1c(Cc2ccc(cc2S(=O)(=O)c2ccccc2)C(O)=O)c2c(CCNC2=O)n1CC(O)=O
COC(=O)c1ccc(Cc2c(C)n(CC(O)=O)c3CCNC(=O)c23)c(c1)S(=O)(=O)c1ccccc1
CNC(=O)c1ccc(Cc2c(C)n(CC(O)=O)c3CCNC(=O)c23)c(c1)S(=O)(=O)c1ccccc1
Cc1c(Cc2cc(F)ccc2S(=O)(=O)c2ccccc2)c2c(CCNC2=O)n1CC(O)=O
COc1ccc(c(Cc2c(C)n(CC(O)=O)c3CCNC(=O)c23)c1)S(=O)(=O)c1ccccc1
Cc1c(Cc2cc(Br)ccc2S(=O)(=O)c2ccccc2)c2c(CCNC2=O)n1CC(O)=O
Cc1c(Cc2cc(ccc2S(=O)(=O)c2ccccc2)C#N)c2c(CCNC2=O)n1CC(O)=O
COc1cccc(c1Cc1c(C)n(CC(O)=O)c2CCNC(=O)c12)S(=O)(=O)c1ccccc1
Cc1c(Cc2ccccc2S(=O)(=O)c2ccccc2F)c2c(CCNC2=O)n1CC(O)=O
Cc1c(Cc2ccccc2S(=O)(=O)c2cccc(F)c2)c2c(CCNC2=O)n1CC(O)=O
Cc1c(Cc2ccccc2S(=O)(=O)c2cccc(Cl)c2)c2c(CCNC2=O)n1CC(O)=O
COc1cccc(c1)S(=O)(=O)c1ccccc1Cc1c(C)n(CC(O)=O)c2CCNC(=O)c12
CNC(=O)c1cccc(c1)S(=O)(=O)c1ccccc1Cc1c(C)n(CC(O)=O)c2CCNC(=O)c12
Cc1c(Cc2ccccc2S(=O)(=O)c2ccc(F)cc2)c2c(CCNC2=O)n1CC(O)=O
Cc1c(Cc2ccccc2S(=O)(=O)c2ccc(Cl)cc2)c2c(CCNC2=O)n1CC(O)=O
COc1ccc(cc1)S(=O)(=O)c1ccccc1Cc1c(C)n(CC(O)=O)c2CCNC(=O)c12
Cc1c(Cc2ccccc2S(=O)(=O)c2ccc(OC(F)(F)F)cc2)c2c(CCNC2=O)n1CC(O)=O
C[C@@H](C(O)=O)n1c(C)c(Cc2ccccc2S(=O)(=O)c2ccccc2)c2c1CCNC2=O |r|
C[C@H](C(O)=O)n1c(C)c(Cc2ccccc2S(=O)(=O)c2ccccc2)c2c1CCNC2=O |r|
CCS(=O)(=O)c1ccccc1Cc1c(C)n(CC(O)=O)c2CCNC(=O)c12
Cc1c(Cc2ccccc2S(=O)(=O)C2CCCCC2)c2c(CCNC2=O)n1CC(O)=O
Cc1c(Cc2ccccc2S(=O)(=O)N2CCOCC2)c2c(CCNC2=O)n1CC(O)=O
CN(Cc1ccccc1)S(=O)(=O)c1ccccc1Cc1c(C)n(CC(O)=O)c2CCNC(=O)c12
Cc1c(Cc2ccc(cc2)S(C)(=O)=O)c2c(CCNC2=O)n1CC(O)=O
Cc1c(Cc2ccc(cc2)S(=O)(=O)c2ccccc2)c2c(CCNC2=O)n1CC(O)=O
Cc1c(Cc2ccc(cc2)S(=O)(=O)Cc2ccccc2)c2c(CCNC2=O)n1CC(O)=O
Cc1c(Cc2ccccc2Cn2ccnn2)c2c(CCNC2=O)n1CC(O)=O
CCN(Cc1ccccc1Cc1c(C)n(CC(O)=O)c2CCNC(=O)c12)C(=O)C1CC1
Cc1c(Cc2ccccc2C(=O)c2ccccc2)c2c(CCNC2=O)n1CC(O)=O
Cc1c(Cc2ccccc2C(O)c2ccccc2)c2c(CCNC2=O)n1CC(O)=O
Cc1c(Cc2ccccc2Cc2ccccc2)c2c(CCNC2=O)n1CC(O)=O
Cc1c(Cc2ccccc2-c2cccc3ccccc23)c2c(CCNC2=O)n1CC(O)=O
Cc1c(Cc2ccccc2Oc2ccccc2)c2c(CCNC2=O)n1CC(O)=O
CN1CCc2c(c(Cc3ccccc3S(=O)(=O)c3ccccc3)c(C)n2CC(O)=O)C1=O
Cc1c(Cc2ccccc2S(=O)(=O)c2ccccc2)c2c(CCN(Cc3ccccc3)C2=O)n1CC(O)=O
CC(C)N1CCc2c(c(Cc3ccccc3S(=O)(=O)c3ccccc3)c(C)n2CC(O)=O)C1=O
CC(N1CCc2c(c(Cc3ccccc3S(=O)(=O)c3ccccc3)c(C)n2CC(O)=O)C1=O)C(F)(F)F
Cc1c(Cc2ccccc2S(=O)(=O)c2ccc(F)cc2)c2c(CC(C)(C)NC2=O)n1CC(O)=O
COc1ccc(c(Cc2c(C)n(CC(O)=O)c3CC(C)(C)NC(=O)c23)c1)S(=O)(=O)c1ccc(F)cc1
Cc1c(Cc2ccccc2S(=O)(=O)c2ccccc2)c2c(Cl)nccc2n1CC(O)=O
Cc1c(Cc2ccccc2S(=O)(=O)c2ccccc2)c2c(cc[nH]c2=O)n1CC(O)=O
Cc1c(Cc2ccccc2S(=O)(=O)c2ccccc2)c2c(ccn(C)c2=O)n1CC(O)=O
Cc1c(Cc2ccccc2S(=O)(=O)c2ccccc2)c2c(ccn(C(F)F)c2=O)n1CC(O)=O
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)cc2cnn(C)c12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)cc2cn(C)nc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)cn2cnnc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)cn2ccnc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)cn2nccc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)c2ccnn2c1)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)c2cccn2c1)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1nn(CC(O)=O)c2ccccc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cn(CC(O)=O)c2ccccc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cn(CC(O)=O)c2cccnc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cn(CC(O)=O)c2ccncc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccccc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2cccnc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)n2cccnc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)c2ccncn12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1nc(CC(O)=O)c2ccccn12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1nn(CC(O)=O)c2cccc(Cl)c12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1nn(CC(O)=O)c2cccc(F)c12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1nn(CC(O)=O)c2cccc(OC)c12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1nn(CC(O)=O)c2cccc(C)c12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1nn(CC(O)=O)c2cccc(C#N)c12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1nn(CC(O)=O)c2ccc(Cl)cc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1nn(CC(O)=O)c2ccc(C)cc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1nn(CC(O)=O)c2ccc(F)cc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1nn(CC(O)=O)c2ccc(Cl)c(F)c12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1nn(CC(O)=O)c2ccc(F)c(Cl)c12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1nn(CC(O)=O)c2cc(F)ccc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(C)nc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(CC)nc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(nc12)C1CC1)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(nc12)C(F)F)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(nc12)C(F)(F)F)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(OC)nc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(F)ccc1-n1cc(CC(O)=O)c2cccnc12)C(=O)C1CC1
CCN(Cc1cc(F)ccc1-n1cc(CC(O)=O)c2ccc(C)nc12)C(=O)C1CC1
CCN(Cc1ccccc1-n1cc(CC(O)=O)c2ccc(C)nc12)C(=O)C1CC1
CCN(Cc1cc(Cl)ccc1-n1cc(CC(O)=O)c2ccc(C)nc12)C(=O)C1CC1
CCN(Cc1cc(C)ccc1-n1cc(CC(O)=O)c2ccc(C)nc12)C(=O)C1CC1
CCN(Cc1cc(OC(F)(F)F)ccc1-n1cc(CC(O)=O)c2ccc(C)nc12)C(=O)C1CC1
CCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(C)nc12)S(C)(=O)=O)C(=O)C1CC1
CCN(Cc1cc(F)ccc1-c1cn(CC(O)=O)c2ccccc12)C(=O)C1CC1
CCN(Cc1cc(F)ccc1-c1cn(CC(O)=O)c2ccc(cc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cn(CC(O)=O)c2ccc(C)nc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cn(CC(O)=O)c2ccc(nc12)C(F)(F)F)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(C)cc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1ccccc1-n1cc(CC(O)=O)c2ccc(cc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)n2ccc(C)nc12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)c2ccc(C)nn12)C(F)(F)F)C(=O)C1CC1
CCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(C)nc12)C(F)(F)F)C(C)=O
CCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(C)nc12)C(F)(F)F)C(=O)C1CCC1
CCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(C)nc12)C(F)(F)F)C(=O)CC1CC1
CCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(C)nc12)C(F)(F)F)C(=O)COC
CCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(C)nc12)C(F)(F)F)C(=O)Cc1ccccc1
CCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(C)nc12)C(F)(F)F)C(=O)c1ccccn1
CCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(C)nc12)C(F)(F)F)C(=O)NCc1ccccc1
CCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(C)nc12)C(F)(F)F)C(=O)CN(C)C
CC(C)N(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(C)nc12)C(F)(F)F)C(=O)C1CC1
Cc1ccc2c(CC(O)=O)cn(-c3ccc(cc3CN(CC3CC3)C(=O)C3CC3)C(F)(F)F)c2n1
Cc1ccc2c(CC(O)=O)cn(-c3ccc(cc3CN(CCOc3ccccc3)C(=O)C3CC3)C(F)(F)F)c2n1
COCCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(C)nc12)C(F)(F)F)C(=O)C1CC1
Cc1ccc2c(CC(O)=O)cn(-c3ccc(cc3CN(CCO)C(=O)C3CC3)C(F)(F)F)c2n1
CCN(Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(C)nc12)C(=O)NCCc1ccccc1)C(=O)C1CC1
Cc1ccc2c(CC(O)=O)cn(-c3ccc(cc3CSC(C)(C)C)C(=O)NCCc3ccccc3)c2n1
COc1ccc(CC(O)=O)cc1-c1ccc(cc1Cn1c(C)nnc1C1CC1)C(F)(F)F
CCCc1nc2ccccc2n1Cc1ccccc1-n1cc(CC(O)=O)c2ccc(C)nc12
Cc1cnn(C)c1Cc1cc(F)ccc1-n1cc(CC(O)=O)c2ccc(C)nc12
Cc1noc(C)c1Cc1cc(F)ccc1-n1cc(CC(O)=O)c2ccc(C)nc12
Cc1nnc(C)n1Cc1cc(C)ccc1-n1cc(CC(O)=O)c2ccc(C)nc12
Cc1ccc2c(CC(O)=O)cn(-c3ccccc3Cn3ccnn3)c2n1
Cc1cnnn1Cc1cc(C)ccc1-n1cc(CC(O)=O)c2ccc(C)nc12
OC(=O)Cn1cc(-c2ccc(cc2Cc2ocnc2C2CC2)C(F)(F)F)c2cc(F)ccc12
Cc1ccc2c(CC(O)=O)cn(-c3ccccc3Cn3ccnc3)c2n1
Cc1nccn1Cc1cc(C)ccc1-n1cc(CC(O)=O)c2ccc(C)nc12
Cc1ccc(c(Cn2ccnc2-c2ccccc2)c1)-n1cc(CC(O)=O)c2ccc(C)nc12
Cc1ccc2c(CC(O)=O)cn(-c3ccc(Cl)cc3Cc3cncnc3)c2n1
CC(C)c1ncncc1Cc1cc(Cl)ccc1-n1cc(CC(O)=O)c2ccc(C)nc12
Cc1ccc(c(Cc2ccnn2Cc2ccccc2)c1)-n1cc(CC(O)=O)c2ccc(C)nc12
Cc1cnn(C)c1Cc1cc(ccc1-c1cn(CC(O)=O)c2ccc(F)cc12)C(F)(F)F
Cc1cnn(CC2CC2)c1Cc1cc(C)ccc1-n1cc(CC(O)=O)c2ccc(C)nc12
Cc1nnc(C)n1Cc1cc(C)ccc1-n1cc(CC(O)=O)c2ccc(Cc3ccccc3)nc12
Cc1nnc(C2CC2)n1Cc1cc(Cl)ccc1-n1cc(CC(O)=O)c2ccc(C)nc12
Cc1nnc(C2CC2)n1Cc1cc(ccc1-c1cn(CC(O)=O)c2ccc(F)cc12)C(F)(F)F
Cc1nnc(C2CC2)n1Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(F)cc12)C(F)(F)F
Cc1nnc(Cc2ccccc2)n1Cc1cc(Cl)ccc1-n1cc(CC(O)=O)c2ccc(C)nc12
Cc1nnc(CCc2ccccc2)n1Cc1cc(Cl)ccc1-n1cc(CC(O)=O)c2ccc(C)nc12
Cc1noc(C)c1Cc1cc(ccc1-c1cn(CC(O)=O)c2ccc(C)nc12)C(F)(F)F
Cc1noc(C)c1Cc1cc(ccc1-c1cn(CC(O)=O)c2ccc(F)cc12)C(F)(F)F
Cc1noc(C2CC2)c1Cc1cc(ccc1-c1cn(CC(O)=O)c2ccc(F)cc12)C(F)(F)F
Cc1noc(C2CC2)c1Cc1cc(F)ccc1-c1cn(CC(O)=O)c2ccc(cc12)C(F)(F)F
Cc1noc(C2CC2)c1Cc1cc(ccc1-c1cc(CC(O)=O)n2ccc(C)nc12)C(F)(F)F
Cc1noc(C2CC2)c1Cc1cc(ccc1-c1cc(CC(O)=O)c2ccc(C)nn12)C(F)(F)F
Cc1noc(C2CC2)c1Cc1cc(ccc1-c1cn(CC(O)=O)c2ccc(nc12)C(F)(F)F)C(F)(F)F
Cc1noc(C2CC2)c1Cc1cc(F)ccc1-n1cc(CC(O)=O)c2ccc(C)nc12
Cc1noc(C2CC2)c1Cc1cc(ccc1-n1cc(CC(O)=O)c2ccc(C)nc12)C(F)(F)F
Cc1noc(C2CC2)c1Cc1cc(Cl)ccc1-n1cc(CC(O)=O)c2ccc(Cc3ccccc3)nc12
Cc1ccc2c(CC(O)=O)cn(-c3ccc(cc3Cc3c(noc3C3CC3)C3CC3)C(F)(F)F)c2n1
Cc1ccc2c(CC(O)=O)cn(-c3ccc(Cl)cc3Cc3c(noc3C3CC3)C3CC3)c2n1
Cc1noc(Cc2ccccc2)c1Cc1cc(Cl)ccc1-n1cc(CC(O)=O)c2ccc(C)nc12
Cc1c(-c2cccc3CN(CCc23)S(C)(=O)=O)c2cc(F)ccc2n1CC(O)=O |(5.67,-9.17,;5.99,-10.68,;7.4,-11.31,;8.74,-10.54,;10.07,-11.31,;11.42,-10.54,;11.41,-8.98,;10.07,-8.23,;10.07,-6.7,;8.74,-5.93,;7.42,-6.7,;7.41,-8.23,;8.74,-8.99,;8.74,-4.38,;10.09,-3.62,;7.2,-4.37,;7.98,-3.04,;7.24,-12.84,;8.26,-13.97,;7.79,-15.43,;8.83,-16.57,;6.29,-15.75,;5.26,-14.61,;5.74,-13.15,;4.96,-11.82,;3.42,-11.67,;2.52,-12.92,;.98,-12.77,;3.15,-14.33,)|
Cc1noc(C)c1-c1cccc(c1)-c1c(C)n(CC(O)=O)c2ccc(F)cc12
Fc1ccc2n(ccc2c1)-c1cc(Cl)c2OCCN(Cc3cc[nH]c(=O)c3)Cc2c1
Cc1c(CC(O)=O)c2ccncn2c1Cc1ccccc1S(=O)(=O)c1ccccc1
COc1ccc(c(Cc2c(C)c(CC(O)=O)c3ccncn23)c1)S(=O)(=O)c1ccc(F)cc1
COc1ccc(c(Cn2cc(CC(O)=O)c3ccc(C)nc23)c1)S(=O)(=O)c1ccc(F)cc1
COc1ccc(c(Cn2c(C)c(CC(O)=O)c3ccc(C)nc23)c1)S(=O)(=O)c1ccc(F)cc1
COc1ccc(c(Cc2c(C)n(CC(O)=O)c3CCCC(=O)c23)c1)S(=O)(=O)c1ccc(F)cc1
Cc1c(CC(O)=O)c2ccc(C)nc2n1Cc1ccccc1S(=O)(=O)c1ccccc1
OC(=O)Cc1cc(Cc2ccccc2S(=O)(=O)c2ccccc2)c2nc(ccn12)C(F)(F)F
OC(=O)Cc1nc(Cc2ccccc2S(=O)(=O)c2ccccc2)n2ccccc12
OC(=O)CN1c2cccnc2N(Cc2ccccc2S(=O)(=O)c2ccccc2)S1(=O)=O
OC(=O)Cc1nn(Cc2ccccc2S(=O)(=O)c2ccccc2)c(=O)c2ccccc12
Cc1c(Cc2ccccc2S(=O)(=O)c2ccc(F)cc2)c2c(CCCC2=O)n1CC(O)=O
Cc1c(Cc2ccccc2S(=O)(=O)c2ccc(F)cc2)c2CCCCc2n1CC(O)=O
OC(=O)Cc1cc(Cl)c(=O)n(Cc2ccccc2S(=O)(=O)c2ccccc2)c1
OC(=O)Cc1ccc(=O)n(Cc2ccccc2S(=O)(=O)c2ccccc2)c1
Cc1c(Cc2ccccc2S(=O)(=O)c2ccc(F)cc2)nc(-c2ccccc2)n1CC(O)=O
OC(=O)Cn1c(nn(Cc2ccccc2S(=O)(=O)c2ccccc2)c1=O)-c1ccccc1
Cc1c(-c2ccccc2)n(CC(O)=O)c(=O)n1Cc1ccccc1S(=O)(=O)c1ccc(F)cc1
Cc1c(Cc2ccccc2S(=O)(=O)c2ccccc2)c(=O)n(-c2ccccc2)n1CC(O)=O
Cc1c(Cc2ccccc2S(=O)(=O)c2ccccc2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccccc2S(=O)(=O)c2ccccc2)c(nn1CC(O)=O)-c1ccccc1
Cc1c(CC(O)=O)c(nn1Cc1ccccc1S(=O)(=O)c1ccccc1)-c1ccccc1
Cc1c(c2cccnc2n1Cc3ccc(cc3C(F)(F)F)S(=O)(=O)C)CC(=O)O
Cc1c(CC(O)=O)c2cccnc2n1Cc1ccc(cc1C)S(C)(=O)=O
CCS(=O)(=O)c1ccc(Cn2c(C)c(CC(O)=O)c3cccnc23)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cn2c(C)c(CC(O)=O)c3cccnc23)c(Cl)c1
Cc1c(CC(O)=O)c2ccccc2n1Cc1ccc(cc1)S(C)(=O)=O
Cc1c(CC(O)=O)c2cccnc2n1Cc1ccc(cc1Cl)S(C)(=O)=O
Cc1c(CC(O)=O)c2cccnc2n1Cc1ccc(c(c1)C(F)(F)F)S(C)(=O)=O
Cc1c(CC(O)=O)c2ccc(C)nc2n1Cc1ccc(cc1)S(C)(=O)=O
Cc1c(CC(O)=O)c2cccnc2n1Cc1ccc(cc1C(F)(F)F)C(F)(F)F
Cc1c(CC(O)=O)c2c(Cl)ccnc2n1Cc1ccc(cc1)S(C)(=O)=O
CCS(=O)(=O)c1ccc(Cn2c(C)c(CC(O)=O)c3cccnc23)cc1
Cc1c(CC(O)=O)c2cc(C)cnc2n1Cc1ccc(cc1)S(C)(=O)=O
CCc1ccc2c(CC(O)=O)c(C)n(Cc3ccc(cc3)S(C)(=O)=O)c2n1
CC(C)S(=O)(=O)c1ccc(Cn2c(C)c(CC(O)=O)c3cccnc23)cc1
Cc1c(CC(O)=O)c2cc(Br)cnc2n1Cc1ccc(cc1)S(C)(=O)=O
CC(C)(Oc1cccc(CCCn2cc(ccc2=O)C(c2ccccc2)c2ccccc2)c1)C(O)=O
CS(=O)(=O)c1cc(F)cc2n3CCC[C@H](CC(O)=O)c3c(C(=O)c3ccc(Cl)cc3)c12
CCNC(=O)c1ccc(Oc2cc(Cl)cc(CC(O)=O)c2)c(NS(=O)(=O)c2cc(C)c(Cl)cc2Cl)c1
CCNC(=O)c1ccc(Oc2cc(Cl)cc(CC(O)=O)c2)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCNC(=O)c1ccc(Oc2cc(Cl)cc(CC(O)=O)c2)c(NS(=O)(=O)c2ccccc2)c1
CCNC(=O)c1ccc(Oc2cc(Cl)cc(CC(O)=O)c2)c(NS(=O)(=O)c2ccc(C)cc2)c1
CCNC(=O)c1ccc(Oc2cc(Cl)cc(CC(O)=O)c2)c(NS(=O)(=O)c2ccc(Cl)cc2)c1
CCNC(=O)c1ccc(Oc2cc(Cl)cc(CC(O)=O)c2)c(NS(=O)(=O)c2ccccc2Cl)c1
CCNC(=O)c1ccc(Oc2cc(Cl)cc(CC(O)=O)c2)c(NS(=O)(=O)c2ccc(C)c(Cl)c2)c1
CCNC(=O)c1ccc(Oc2cc(Cl)cc(CC(O)=O)c2)c(NS(=O)(=O)c2ccc(cc2Cl)C(F)(F)F)c1
CCNC(=O)c1ccc(Oc2cccc(CC(O)=O)c2)c(NS(=O)(=O)c2ccccc2)c1
NC(=O)c1ccc(Oc2cccc(CC(O)=O)c2)c(NS(=O)(=O)c2ccccc2)c1
CCNC(=O)c1ccc(Oc2cccc(CC(O)=O)c2)c(NS(=O)(=O)c2ccc(C)cc2)c1
CCN(CC)C(=O)c1ccc(Oc2cccc(CC(O)=O)c2)c(NS(=O)(=O)c2ccc(C)cc2)c1
CC(=O)c1ccc(Oc2cccc(CC(O)=O)c2)c(NS(=O)(=O)c2ccccc2)c1
CCNCc1ccc(Oc2cccc(CC(O)=O)c2)c(NS(=O)(=O)c2ccccc2)c1
OC(=O)Cc1cccc(Oc2ccc(Cl)cc2NS(=O)(=O)c2ccccc2)c1
COc1ccc(Oc2cccc(CC(O)=O)c2)c(NS(=O)(=O)c2ccccc2)c1
Nc1ccc(Oc2cccc(CC(O)=O)c2)c(NS(=O)(=O)c2ccc(Cl)cc2)c1
CCC(=O)Nc1ccc(Oc2cccc(CC(O)=O)c2)c(NS(=O)(=O)c2ccc(Cl)cc2)c1
CCNC(=O)Nc1ccc(Oc2cccc(CC(O)=O)c2)c(NS(=O)(=O)c2ccc(Cl)cc2)c1
CCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCNC(=O)c1ccc(Oc2ccc(Cc3nnn[nH]3)cc2)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCNC(=O)c1ccc(Oc2ccc(cc2)C(C)C(O)=O)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2F)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2OCC)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCNC(=O)c1ccc(Oc2ccc(cc2OC)C(O)=O)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCNC(=O)c1ccc(Oc2ccc(CCC(O)=O)cc2OC)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
CCCCCNC(=O)c1ccc(Oc2ccc(CC(O)=O)cc2OC)c(NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
COc1cc(CC(O)=O)ccc1Oc1ccc(cc1NS(=O)(=O)c1ccc(Cl)cc1Cl)C(=O)NC(C)C
COc1cc(CC(O)=O)ccc1Oc1ccc(cc1NS(=O)(=O)c1ccc(Cl)cc1Cl)C(=O)NCC(C)C
COc1cc(CC(O)=O)ccc1Oc1ccc(cc1NS(=O)(=O)c1ccc(Cl)cc1Cl)C(=O)NC1CCC1
COc1cc(CC(O)=O)ccc1Oc1ccc(cc1NS(=O)(=O)c1ccc(Cl)cc1Cl)C(=O)NC1CCCC1
COc1ccc(CC(O)=O)cc1C1=NCC(=O)N(Cc2ccccc2)c2ccccc12 |t:13|
COc1ccc(CC(O)=O)cc1C1=NCC(=O)N(Cc2ccc(F)cc2)c2ccccc12 |t:13|
COc1ccc(CC(O)=O)cc1C1=NCC(=O)N(Cc2ccc(F)c(F)c2)c2ccccc12 |t:13|
COc1ccc(CC(O)=O)cc1C1=NCC(=O)N(Cc2ccc(Cl)cc2)c2ccccc12 |t:13|
COc1ccc(CC(O)=O)cc1C1=NCC(=O)N(Cc2cccc(Cl)c2)c2ccccc12 |t:13|
COc1ccc(CC(O)=O)cc1C1=NCC(=O)N(Cc2ccc(Cl)cc2Cl)c2ccccc12 |t:13|
COc1ccc(CC(O)=O)cc1C1=NCC(=O)N(Cc2ccc(C)cc2)c2ccccc12 |t:13|
COc1ccc(CC(O)=O)cc1C1=NCC(=O)N(Cc2ccc(cc2)C(F)(F)F)c2ccccc12 |t:13|
COc1ccc(CC(O)=O)cc1C1=NCC(=O)N(Cc2ccc(OC(F)(F)F)cc2)c2ccccc12 |t:13|
COc1ccc(CC(O)=O)cc1-c1nc(=O)n(Cc2ccccc2)c2ccccc12
OC(=O)Cc1cccc(Oc2ccccc2NS(=O)(=O)c2ccccc2)c1
COc1ccc(CC(O)=O)cc1C(=O)c1ccccc1NS(=O)(=O)c1ccc(C)cc1
OC(=O)Cc1cccc(Oc2ccccc2NS(=O)(=O)c2ccc(Cl)cc2Cl)c1
COc1ccc(CC(O)=O)cc1C(=O)c1ccccc1NS(=O)(=O)c1ccc(Cl)cc1Cl
CC(=O)Nc1ccc(cc1)C(=O)c1ncc(CC(O)=O)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3ccccc3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3ccc4ccccc4c3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3cc4ccccc4[nH]3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3ccncc3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3ncccn3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3cccc(Cl)c3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3ccc(Cl)cc3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3ccccc3Cl)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3ccc(cc3)C(F)(F)F)cc2)c2ccccc12
COc1ccc(cc1)C(=O)Nc1ccc(cc1)C(=O)c1ncc(CC(O)=O)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3ccc(Cl)c(Cl)c3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)CCc3ccc(Cl)c(Cl)c3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)\C=C\c3ccc(Cl)c(Cl)c3)cc2)c2ccccc12
CN(C(=O)c1ccc(Cl)c(Cl)c1)c1ccc(cc1)C(=O)c1ncc(CC(O)=O)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NCc3ccc(Cl)c(Cl)c3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NS(=O)(=O)c3ccc(Cl)c(Cl)c3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(OCc3ccc(Cl)c(Cl)c3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(cc2)C(=O)Nc2ccc(Cl)c(Cl)c2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(cc2)C(=O)NCCc2ccc(Cl)cc2)c2ccccc12
OC(=O)COc1cnc(C(=O)c2ccc(cc2)C(=O)NCCc2ccc(Cl)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)C3CCCCC3)cc2)c2ccccc12
CC(C)(C(O)=O)c1cnc(C(=O)c2ccc(cc2)C(=O)NCCc2ccc(Cl)cc2)c2ccccc12
CCc1nn(Cc2cccc(Br)c2)c(CC)c1CC(O)=O
CCc1nn(Cc2ccc3ccccc3c2)c(CC)c1CC(O)=O
CCc1nn(Cc2cc(Cl)ccc2Cl)c(CC)c1CC(O)=O
CCc1nn(CC(O)=O)c(CC)c1Cc1ccc2ccccc2c1
OC(=O)Cn1cnc2CN(CCc12)C(=O)c1csc(n1)-c1ccccc1
OC(=O)COc1ccccc1COc1ccc(Cl)cc1-c1ccno1
CCCNC(=O)c1ccccc1OCc1cccc(C)c1OCC(O)=O
Cc1ccc2cccc(OCc3ccccc3OCC(O)=O)c2n1
Cc1ccc(Cl)cc1OCc1ccccc1OCC(O)=O
OC(=O)COc1ccccc1COc1ccc(F)cc1C1CC1
CS(=O)(=O)c1ccc(CN(C(=O)C2CCOCC2)c2cc(F)cc(c2)-c2nnn[nH]2)cc1
CS(=O)(=O)c1ccc(CN(C(=O)c2cccnc2)c2cc(F)cc(c2)-c2nnn[nH]2)cc1
CS(=O)(=O)c1ccc(CN(C(=O)c2ccncc2)c2cc(F)cc(c2)-c2nnn[nH]2)cc1
CCCCC(=O)N(Cc1ccc2OCCOc2c1)c1cccc(CC(O)=O)c1
CCCCC(=O)N(Cc1cccc(OC)c1)c1cccc(c1)C(O)=O
CCCCC(=O)N(Cc1ccc2OCCOc2c1)c1cc(F)cc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1cccc(OC)c1)c1cc(F)cc(c1)-c1nnn[nH]1
CCCCC(=O)N(Cc1ccc(OC)cc1)c1cc(Cl)cc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1ccc(cc1)C(F)(F)F)c1cc(F)cc(c1)-c1nnn[nH]1
CCCCC(=O)N(Cc1ccc(OC(F)(F)F)cc1)c1cc(Cl)cc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1cccc(O)c1)c1cc(F)cc(c1)-c1nnn[nH]1
CC(C)CC(=O)N(Cc1ccc(cc1)S(C)(=O)=O)c1cc(F)cc(c1)-c1nnn[nH]1
CS(=O)(=O)c1ccc(CN(C(=O)C2CCCC2)c2cc(F)cc(c2)-c2nnn[nH]2)cc1
CS(=O)(=O)c1ccc(CN(C(=O)Cc2ccccc2)c2cc(F)cc(c2)-c2nnn[nH]2)cc1
CC(=O)N(Cc1cccc(c1)C#C)c1cc(ccc1F)-c1nnn[nH]1
CCCCC(=O)N(Cc1cccc(c1)C#C)c1cc(ccc1F)-c1nnn[nH]1
CCCCC(=O)N(Cc1ccc2OCCOc2c1)c1cc(ccc1F)-c1nnn[nH]1
CCCCC(=O)N(Cc1ccc2ccccc2c1)c1cccc(c1)-c1nnn[nH]1
CCCCC(=O)N(Cc1ccc2cnccc2c1)c1cccc(c1)-c1nnn[nH]1
CCCCC(=O)N(Cc1cccs1)c1cccc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1ccccc1)c1cccc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1cccc(OC)c1)c1cccc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1ccc(OC)cc1)c1cccc(c1)-c1nnn[nH]1
CCCCC(=O)N(Cc1cccc(OC)c1)c1cccc(c1)-c1nnn[nH]1
CCCCC(=O)N(Cc1cccc(OC)c1)c1cc(F)cc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1ccc(OC)cc1)c1cc(F)cc(c1)-c1nnn[nH]1
CCCCC(=O)N(Cc1ccc(OC)cc1)c1cc(F)cc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1cccc(OC(C)C)c1)c1cc(F)cc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1ccccc1F)c1cccc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1cccc(F)c1)c1cccc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1ccc(F)cc1)c1cccc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1cccc(C)c1)c1cccc(c1)-c1nnn[nH]1
CCCCC(=O)N(Cc1cc2ccccc2o1)c1cc(ccc1F)-c1nnn[nH]1
CCC(=O)N(Cc1ccc2ccccc2n1)c1cc(F)cc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1ccc2OCCOc2c1)c1cccc(c1)-c1nnn[nH]1
CCCC(=O)N(Cc1ccc2OCCOc2c1)c1cccc(c1)-c1nnn[nH]1
CCCCC(=O)N(Cc1ccc2OCCOc2c1)c1cccc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1ccc2OCCOc2c1)c1cc(ccc1F)-c1nnn[nH]1
CC(C)CC(=O)N(Cc1ccc2OCCOc2c1)c1cc(ccc1F)-c1nnn[nH]1
CCCC(=O)N(Cc1ccc2OCCOc2c1)c1cc(ccc1F)-c1nnn[nH]1
CCCCC(=O)N(Cc1ccc2OCCOc2c1)c1cc(-c2nnn[nH]2)c(F)cc1F
CCC(=O)N(Cc1ccc2OCOc2c1)c1cccc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1cccc(c1)C(F)(F)F)c1cccc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1ccc(cc1)C(F)(F)F)c1cccc(c1)-c1nnn[nH]1
CCCCC(=O)N(Cc1ccc(cc1)C(F)(F)F)c1cc(F)cc(c1)-c1nnn[nH]1
CCCCC(=O)N(Cc1cccc(OC(F)(F)F)c1)c1cc(F)cc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1ccc(OC(F)(F)F)cc1)c1cc(F)cc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1ccc(cc1)S(=O)(=O)C(F)(F)F)c1cc(F)cc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1ccc(O)cc1)c1cc(F)cc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1ccc(cc1)S(C)(=O)=O)c1cccc(c1)-c1nnn[nH]1
CCC(=O)N(Cc1ccc(cc1)S(C)(=O)=O)c1cc(F)cc(c1)-c1nnn[nH]1
CC(C)C(=O)N(Cc1ccc(cc1)S(C)(=O)=O)c1cc(F)cc(c1)-c1nnn[nH]1
CS(=O)(=O)c1ccc(CN(C(=O)c2ccccc2)c2cc(F)cc(c2)-c2nnn[nH]2)cc1
Cc1ccc(CCC(=O)N(Cc2ccc(cc2)S(C)(=O)=O)c2cc(F)cc(c2)-c2nnn[nH]2)cc1
CCCCC(=O)N(Cc1ccc(OC)cc1)c1cccc(c1)-c1nnn[nH]1
CCCCC(=O)N(Cc1ccc2ccccc2c1)c1cc(ccc1F)-c1nnn[nH]1
CCCCC(=O)N(Cc1ccc(OC(F)(F)F)cc1)c1cc(F)cc(c1)-c1nnn[nH]1
OC(=O)CN1C(=O)C2(NC(=O)N(Cc3ccccc3F)C2=O)c2cc(Cl)ccc12
OC(=O)CN1C(=O)C2(NC(=O)N(Cc3cc(Cl)ccc3F)C2=O)c2cc(Cl)ccc12
Cc1onc(c1CN1C(=O)NC2(C1=O)C(=O)N(CC(O)=O)c1ccc(Cl)cc21)-c1ccccc1
OC(=O)CN1C(=O)[C@@]2(NC(=O)N(Cc3cc(Cl)ccc3F)C2=O)c2cc(Cl)ccc12 |r|
CN1C(=O)N(Cc2cc(Cl)ccc2F)C(=O)[C@]11C(=O)N(CC(O)=O)c2ccc(Cl)cc12 |r|
CCN1C(=O)N(Cc2cc(Cl)ccc2F)C(=O)[C@]11C(=O)N(CC(O)=O)c2ccc(Cl)cc12 |r|
CCCN1C(=O)N(Cc2cc(Cl)ccc2F)C(=O)[C@]11C(=O)N(CC(O)=O)c2ccc(Cl)cc12 |r|
CC(C)c1nc(CN2C(=O)N(C)C3(C2=O)C(=O)N(CC(O)=O)c2ccc(Cl)cc32)cs1
CN1C(=O)N(Cc2cn(nc2-c2ccccc2)-c2ccccc2)C(=O)C11C(=O)N(CC(O)=O)c2ccc(Cl)cc12
CN1C(=O)N(Cc2c(C)onc2-c2ccccc2)C(=O)C11C(=O)N(CC(O)=O)c2ccc(Cl)cc12
CN1C(=O)N(Cc2csc(n2)-c2ccccc2)C(=O)C11C(=O)N(CC(O)=O)c2ccc(Cl)cc12
CN1C(=O)N(Cc2nc3ccccc3s2)C(=O)C11C(=O)N(CC(O)=O)c2ccc(Cl)cc12
COc1c(C)cnc(CN2C(=O)N(C)C3(C2=O)C(=O)N(CC(O)=O)c2ccc(Cl)cc32)c1C
CN1C(=O)N(Cc2cc(F)ccc2F)C(=O)C11C(=O)N(CC(O)=O)c2ccc(Cl)cc12
OC(=O)Cn1c(SCCOc2ccc3ccccc3c2)nc2ccccc12
COCCCn1c2nc3c(C)cccn3c(=O)c2cc(C#N)\c1=N/C(=O)c1ccncc1
OC(=O)Cn1c(SCCOc2ccc(Cl)cc2)nc2ccccc12
CCCOc1ccc(cc1CSc1nc2cc(F)ccc2n1CC(O)=O)C(C)=O
CCCCOc1ccc(cc1CSc1nc2cc(F)ccc2n1CC(O)=O)C(C)=O
COC(=O)c1ccc(OC)c(CSc2nc3ccccc3n2CC(O)=O)c1
OC(=O)Cn1c(SCc2cccc(Cl)c2)nc2ccccc12
COc1ccc(cc1CSc1nc2cc(F)ccc2n1CC(O)=O)C(=O)N1CCc2ccccc12
CCCCNC(=O)c1ccc(OC)c(CSc2nc3cc(F)ccc3n2CC(O)=O)c1
COc1ccc(cc1CSc1nc2cc(F)ccc2n1CC(O)=O)C(C)=O
COc1ccc(cc1CSc1nc2ccccc2n1CC(O)=O)C(C)=O
COc1ccc(cc1CSc1nc2cc(F)ccc2n1CC(O)=O)C(=O)N1CCOCC1
CCN(Cc1ccccc1)C(=O)c1ccc(OC)c(CSc2nc3cc(F)ccc3n2CC(O)=O)c1
CCN(CC)C(=O)c1ccc(OC)c(CSc2nc3cc(F)ccc3n2CC(O)=O)c1
COc1ccc(cc1CSc1nc2cc(F)ccc2n1CC(O)=O)C(=O)NCc1ccccc1
CCNC(=O)c1ccc(OC)c(CSc2nc3cc(F)ccc3n2CC(O)=O)c1
COc1ccc(cc1CSc1nc2cc(F)ccc2n1CC(O)=O)C(=O)c1ccccc1
CCOc1ccc(cc1CSc1nc2cc(F)ccc2n1CC(O)=O)C(C)=O
COc1ccc(cc1CSc1nc2cc(C=O)ccc2n1CC(O)=O)C(C)=O
COc1ccc(cc1CSc1nc2cc(ccc2n1CC(O)=O)C(C)=O)C(C)=O
COc1ccc(cc1CSc1nc2cc(ccc2n1CC(O)=O)S(C)(=O)=O)C(C)=O
COc1ccc(cc1CSc1nc2cc(ccc2n1CC(O)=O)C(F)(F)F)C(C)=O
COc1ccc(cc1CSc1nc2cc(ccc2n1CC(O)=O)[N+]([O-])=O)C(C)=O
COc1ccc(cc1CSc1nc2ccc(F)cc2n1CC(O)=O)C(C)=O
COc1ccc(cc1CSc1nc2c(F)cccc2n1CC(O)=O)C(C)=O
COc1ccc(cc1CSc1nc2ccccc2n1CC(O)=O)C(C)O
CC(=O)c1cccc(CSc2nc3ccccc3n2CC(O)=O)c1
COc1ccc(cc1CSc1nc2ccccc2n1CC(O)=O)C(=O)OC(C)C
COC(=O)c1ccc(Br)c(CSc2nc3ccccc3n2CC(O)=O)c1
COC(=O)c1cc(Br)cc(CSc2nc3ccccc3n2CC(O)=O)c1
COC(=O)c1cc(CSc2nc3ccccc3n2CC(O)=O)ccc1Br
COC(=O)c1cccc(CSc2nc3ccccc3n2CC(O)=O)c1Br
COc1ccc(OC)c(CSc2nc3ccccc3n2CC(O)=O)c1
COc1ccc(Cl)cc1CSc1nc2ccccc2n1CC(O)=O
COc1ccc(C)cc1CSc1nc2ccccc2n1CC(O)=O
OC(=O)Cn1c(SCc2cc(Cl)ccc2Cl)nc2ccccc12
OC(=O)Cn1c(SCc2ccc(Cl)c(Cl)c2)nc2ccccc12
COC(=O)c1ccccc1CSc1nc2ccccc2n1CC(O)=O
COC(=O)c1cccc(CSc2nc3ccccc3n2CC(O)=O)c1
COC(=O)c1ccc(CSc2nc3ccccc3n2CC(O)=O)cc1
OC(=O)Cn1c(SCc2ccccc2Br)nc2ccccc12
OC(=O)Cn1c(SCc2cccc(Br)c2)nc2ccccc12
OC(=O)Cn1c(SCc2ccc(Br)cc2)nc2ccccc12
Cc1ccccc1CSc1nc2ccccc2n1CC(O)=O
Cc1cccc(CSc2nc3ccccc3n2CC(O)=O)c1
Cc1ccc(CSc2nc3ccccc3n2CC(O)=O)cc1
COc1ccccc1CSc1nc2ccccc2n1CC(O)=O
COc1cccc(CSc2nc3ccccc3n2CC(O)=O)c1
COc1ccc(CSc2nc3ccccc3n2CC(O)=O)cc1
OC(=O)Cn1c(SCc2ccccc2Cl)nc2ccccc12
OC(=O)Cn1c(SCc2ccc(Cl)cc2)nc2ccccc12
CCNC(=O)CCCCSc1nc2ccccc2n1CC(O)=O
CCOC(=O)CCCCCSc1nc2ccccc2n1CC(O)=O
CCOC(=O)CCCCSc1nc2ccccc2n1CC(O)=O
CCOC(=O)CCCSc1nc2ccccc2n1CC(O)=O
CCOC(=O)CCSc1nc2ccccc2n1CC(O)=O
CCCCSc1nc2ccccc2n1CC(O)=O
CCCCCSc1nc2ccccc2n1CC(O)=O
CCCCCCSc1nc2ccccc2n1CC(O)=O
OC(=O)Cn1c(SCCNc2ccccc2)nc2ccccc12
OC(=O)Cn1c(SCCCNc2ccccc2)nc2ccccc12
OC(=O)Cn1c(SCc2ccccc2)nc2ccccc12
OC(=O)Cn1c(SCCc2ccccc2)nc2ccccc12
OC(=O)Cn1c(SCCCc2ccccc2)nc2ccccc12
OC(=O)Cn1c(SCCCCOc2ccccc2)nc2ccccc12
OC(=O)Cn1c(SCCCOc2ccccc2)nc2ccccc12
OC(=O)Cn1c(SCCOc2cccc3ccccc23)nc2ccccc12
Cc1c(CC(O)=O)cc2ccc(F)cc2c1Oc1ncc(cc1Br)S(C)(=O)=O
CCN(Cc1cc(ccc1-c1cc(CC(O)=O)ccc1OC)C(F)(F)F)C(=O)NCc1ccccc1
C[C@H](Oc1ccc(F)cc1-c1ccc(C(=O)N2CCCC2(C)C)c(Cl)c1)C(O)=O |r|
Cc1c(CC(O)=O)c2ccc(F)cn2c1Sc1ccc(cc1F)S(C)(=O)=O
Cc1c(Sc2ccc(Cl)cc2)c2cc(Cl)ncc2n1CC(O)=O
Cc1c(Sc2ccc(Cl)cc2)c2ncccc2n1CC(O)=O
Cc1c(Cc2ccc3ccccc3c2)c2cc(F)ccc2n1CC(O)=O
Cc1c(CC(O)=O)c2cc(F)ccc2n1Cc1ccc2ccccc2c1
Cc1c(Cc2nc3ccccc3s2)c2cc(F)ccc2n1CC(O)=O
Cc1c(CC(O)=O)c2cc(F)ccc2n1Cc1nc2ccccc2s1
CN(C(=O)C1(C)CCc2c(C1)c1ccccc1n2CC(O)=O)c1cccc(Cl)c1
OC(=O)Cn1c2CC[C@H](Cc2c2cc(F)ccc12)NC(=O)CC(c1ccccc1)c1ccccc1 |r|
OC(=O)Cn1c2CCN(Cc2c2cc(ccc12)C(F)(F)F)C(=O)c1ccccc1
CN(c1ccc2n(CC(O)=O)c3ccccc3c2c1)S(=O)(=O)c1ccc(F)cc1
CN(CCc1c(C)n(CC(O)=O)c2ccccc12)S(=O)(=O)c1ccc(F)cc1
OC(=O)[C@@H]1CCOc2cc(Oc3ccc(cc3)C(=O)Nc3cccc(n3)-c3ccc(Cl)cc3)c(Cl)cc12 |r|
CCc1nc2c(F)ccc(OCC(O)=O)c2c(OC(F)F)c1Cc1ccc(cc1)-n1cccn1
Cc1cc(CC(O)=O)c2c(C)c(Cc3ccccc3)c(=O)oc2c1
Cc1c(-c2nn(Cc3ccccc3)c(=O)c3ccccc23)c2ccccc2n1CCC(O)=O |(22.19,-53.06,;20.65,-53.06,;19.74,-51.8,;20.51,-50.48,;22.05,-50.48,;22.83,-49.16,;24.37,-49.16,;25.13,-50.5,;24.35,-51.82,;25.11,-53.16,;26.65,-53.16,;27.43,-51.82,;26.66,-50.49,;22.06,-47.82,;22.84,-46.49,;20.52,-47.81,;19.75,-46.48,;18.2,-46.48,;17.43,-47.83,;18.2,-49.16,;19.74,-49.15,;18.26,-52.28,;16.93,-51.52,;15.6,-52.29,;15.59,-53.83,;16.93,-54.6,;18.26,-53.83,;19.74,-54.31,;20.21,-55.78,;19.18,-56.92,;17.68,-56.6,;17.19,-55.14,;16.64,-57.75,)|
CC(C(O)=O)n1c(C)c(-c2nn(Cc3ccccc3)c(=O)c3ccccc23)c2ccccc12 |(8.1,-55.32,;6.59,-55,;5.56,-56.14,;4.05,-55.83,;6.04,-57.61,;6.11,-53.53,;7.02,-52.28,;8.56,-52.28,;6.11,-51.02,;6.89,-49.7,;8.43,-49.71,;9.2,-48.38,;10.74,-48.38,;11.51,-49.72,;10.73,-51.04,;11.49,-52.38,;13.03,-52.39,;13.81,-51.05,;13.04,-49.72,;8.44,-47.04,;9.21,-45.71,;6.9,-47.03,;6.12,-45.7,;4.57,-45.7,;3.8,-47.05,;4.58,-48.38,;6.12,-48.37,;4.64,-51.5,;3.3,-50.74,;1.97,-51.51,;1.97,-53.05,;3.3,-53.82,;4.64,-53.05,)|
Cc1c(-c2nn(Cc3ccccc3)c(=O)c3ccccc23)c2ccccc2n1CCO |(39.21,-35.7,;37.67,-35.7,;36.75,-34.45,;37.53,-33.12,;39.07,-33.13,;39.84,-31.8,;41.38,-31.81,;42.15,-33.15,;41.37,-34.47,;42.13,-35.8,;43.67,-35.81,;44.44,-34.47,;43.68,-33.14,;39.08,-30.47,;39.85,-29.14,;37.54,-30.46,;36.76,-29.13,;35.22,-29.13,;34.45,-30.48,;35.22,-31.81,;36.76,-31.8,;35.28,-34.93,;33.94,-34.17,;32.62,-34.94,;32.61,-36.48,;33.95,-37.25,;35.28,-36.48,;36.75,-36.96,;37.23,-38.42,;36.2,-39.57,;34.69,-39.25,)|
Cc1c(-c2nn(Cc3ccccc3)c(=O)c3ccccc23)c2ccccc2n1-c1nnn[nH]1 |(26.03,-37.21,;24.5,-37.21,;23.58,-35.96,;24.36,-34.63,;25.9,-34.64,;26.67,-33.31,;28.21,-33.32,;28.98,-34.65,;28.19,-35.97,;28.96,-37.31,;30.5,-37.32,;31.27,-35.98,;30.51,-34.65,;25.91,-31.97,;26.68,-30.64,;24.37,-31.97,;23.59,-30.63,;22.05,-30.63,;21.28,-31.98,;22.05,-33.31,;23.59,-33.31,;22.11,-36.44,;20.77,-35.67,;19.45,-36.44,;19.44,-37.99,;20.78,-38.76,;22.11,-37.99,;23.58,-38.46,;24.06,-39.93,;25.53,-40.4,;25.53,-41.94,;24.07,-42.42,;23.16,-41.17,)|
Cc1c(-c2nn(Cc3ccccc3)c(=O)c3ccccc23)c2ccccc2n1CC(=O)NS(C)(=O)=O |(10,-36.32,;8.46,-36.32,;7.55,-35.06,;8.32,-33.74,;9.87,-33.75,;10.64,-32.42,;12.18,-32.42,;12.94,-33.76,;12.16,-35.08,;12.93,-36.42,;14.47,-36.43,;15.24,-35.09,;14.48,-33.76,;9.88,-31.08,;10.65,-29.75,;8.33,-31.07,;7.56,-29.74,;6.01,-29.74,;5.24,-31.09,;6.02,-32.42,;7.56,-32.41,;6.08,-35.54,;4.74,-34.78,;3.41,-35.55,;3.41,-37.09,;4.74,-37.86,;6.08,-37.09,;7.55,-37.57,;8.03,-39.04,;7,-40.18,;7.47,-41.65,;5.49,-39.87,;4.46,-41.01,;2.95,-40.7,;5.79,-41.78,;4.45,-42.55,)|
Cc1c(-c2nn(Cc3ccccc3)c(=O)c3ccccc23)c2ccccc2n1CC(=O)N1CCCC1 |(37.67,-22.1,;36.13,-22.1,;35.22,-20.85,;35.99,-19.52,;37.53,-19.53,;38.31,-18.21,;39.85,-18.21,;40.61,-19.55,;39.83,-20.87,;40.59,-22.2,;42.13,-22.21,;42.91,-20.87,;42.14,-19.54,;37.54,-16.87,;38.32,-15.54,;36,-16.86,;35.23,-15.53,;33.68,-15.53,;32.91,-16.88,;33.69,-18.21,;35.23,-18.2,;33.75,-21.33,;32.41,-20.57,;31.09,-21.34,;31.08,-22.88,;32.42,-23.65,;33.75,-22.88,;35.22,-23.36,;35.7,-24.82,;34.67,-25.96,;35.14,-27.43,;33.16,-25.65,;32.53,-24.25,;31,-24.42,;30.69,-25.92,;32.02,-26.69,)|
CN(C)C(=O)Cn1c(C)c(-c2nn(Cc3ccccc3)c(=O)c3ccccc23)c2ccccc12 |(15.98,-25.02,;16.46,-26.48,;15.43,-27.63,;17.97,-26.8,;18.44,-28.27,;19,-25.65,;18.52,-24.19,;19.43,-22.93,;20.97,-22.93,;18.52,-21.68,;19.29,-20.35,;20.83,-20.36,;21.61,-19.03,;23.15,-19.04,;23.91,-20.38,;23.13,-21.7,;23.89,-23.03,;25.43,-23.04,;26.21,-21.7,;25.44,-20.37,;20.84,-17.7,;21.62,-16.37,;19.3,-17.69,;18.53,-16.35,;16.98,-16.36,;16.21,-17.71,;16.99,-19.04,;18.53,-19.03,;17.04,-22.16,;15.71,-21.4,;14.38,-22.17,;14.38,-23.71,;15.71,-24.48,;17.04,-23.71,)|
Cc1c(-c2nn(Cc3ccccc3)c(=O)c3ccccc23)c2ccccc2n1CC(N)=O |(7.37,-22.45,;5.83,-22.45,;4.92,-21.19,;5.69,-19.87,;7.23,-19.88,;8.01,-18.55,;9.55,-18.55,;10.31,-19.89,;9.53,-21.21,;10.29,-22.55,;11.83,-22.56,;12.61,-21.22,;11.84,-19.89,;7.24,-17.21,;8.02,-15.88,;5.7,-17.21,;4.93,-15.87,;3.38,-15.87,;2.61,-17.22,;3.39,-18.55,;4.93,-18.55,;3.45,-21.67,;2.11,-20.91,;.78,-21.68,;.78,-23.22,;2.11,-23.99,;3.45,-23.22,;4.92,-23.7,;5.4,-25.17,;4.37,-26.31,;2.86,-25.99,;4.84,-27.78,)|
Cc1c(-c2nn(Cc3ccccc3)c(=O)c3ccccc23)c2ccccc2n1CC(O)=O |(37.95,-7.39,;36.41,-7.39,;35.5,-6.14,;36.27,-4.81,;37.81,-4.82,;38.59,-3.49,;40.13,-3.5,;40.89,-4.83,;40.11,-6.16,;40.87,-7.49,;42.41,-7.5,;43.19,-6.16,;42.42,-4.83,;37.82,-2.15,;38.6,-.82,;36.28,-2.15,;35.51,-.81,;33.96,-.81,;33.19,-2.16,;33.97,-3.49,;35.51,-3.49,;34.03,-6.62,;32.69,-5.85,;31.36,-6.62,;31.36,-8.17,;32.69,-8.94,;34.03,-8.17,;35.5,-8.65,;35.98,-10.11,;34.95,-11.25,;33.44,-10.94,;35.42,-12.72,)|
Cc1c(-c2ccc(=O)n(Cc3ccc(F)cc3)n2)c2cc(F)ccc2n1CC(O)=O
Cc1c(-c2nn(CCOc3ccc(Cl)cc3)c(=O)c3ccccc23)c2cc(Cl)ccc2n1CC(O)=O |(7.71,-8.01,;6.17,-8.01,;5.26,-6.75,;6.03,-5.43,;7.57,-5.44,;8.35,-4.11,;9.89,-4.11,;10.65,-5.45,;12.19,-5.46,;12.96,-6.8,;12.18,-8.12,;12.94,-9.46,;14.48,-9.46,;15.25,-10.8,;15.26,-8.13,;14.49,-6.79,;7.58,-2.77,;8.36,-1.44,;6.04,-2.76,;5.27,-1.43,;3.73,-1.43,;2.96,-2.77,;3.73,-4.1,;5.27,-4.1,;3.78,-7.23,;2.45,-6.47,;1.12,-7.24,;-.22,-6.47,;1.12,-8.79,;2.45,-9.56,;3.78,-8.79,;5.26,-9.26,;5.73,-10.73,;4.7,-11.87,;3.19,-11.56,;5.18,-13.34,)|
Cc1c(Cc2ccc(=O)n(Cc3ccc(F)cc3F)n2)c2cc(F)cc(F)c2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3ccccc3)n2)c2ccccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3ccc(cc3)C(O)(C(F)(F)F)C(F)(F)F)n2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3ccc(cc3)C(F)(F)F)n2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3ccncc3)n2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3ccc(F)cc3F)n2)c2ccccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3ccccc3)n2)c2cc(Cl)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3cc(F)c(F)cc3F)n2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3ccncc3F)n2)c2cc(F)ccc2n1CC(O)=O
Cc1c(Cc2ccc(=O)n(Cc3ccc(cc3)C(C)(C)O)n2)c2cc(F)ccc2n1CC(O)=O
Cc1c(-c2ccc(=O)n(Cc3ccc(F)cc3F)n2)c2cc(F)ccc2n1CC(O)=O
Cc1c(CC2=NN(Cc3ccc(F)cc3F)C(=O)CC2)c2cc(F)ccc2n1CC(O)=O |t:4|
Cc1c(CC2=NN(Cc3ccccc3)C(=O)CC2)c2cc(F)ccc2n1CC(O)=O |t:4|
Cc1c(C2=NN(Cc3ccccc3)C(=O)C3CCCCC23)c2cc(F)ccc2n1CC(O)=O |t:3|
Cc1c(-c2nn(Cc3ccccc3)c(=O)c3ccccc23)c2cc(F)ccc2n1CC(O)=O |(8.23,-6.54,;6.69,-6.54,;5.77,-5.29,;6.5,-3.93,;8.04,-3.88,;8.76,-2.52,;10.3,-2.47,;11.12,-3.77,;10.39,-5.13,;11.2,-6.43,;12.75,-6.38,;13.47,-5.01,;12.65,-3.71,;7.94,-1.21,;8.66,.16,;6.4,-1.28,;5.59,.03,;4.05,-.04,;3.34,-1.4,;4.16,-2.69,;5.68,-2.63,;4.3,-5.77,;2.96,-5,;1.63,-5.78,;.3,-5,;1.63,-7.32,;2.96,-8.09,;4.3,-7.32,;5.77,-7.8,;6.49,-9.16,;5.67,-10.47,;4.13,-10.41,;6.39,-11.83,)|
Cc1c(Cc2nn(Cc3ccccc3)c(=O)c3ccccc23)c2cc(Cl)ccc2n1CC(O)=O
Cc1c(-c2nn(Cc3ccccc3)c(=O)c3ccccc23)c2cc(Cl)ccc2n1CC(O)=O |(23.87,-56.05,;22.33,-56.05,;21.42,-54.8,;22.14,-53.44,;23.68,-53.39,;24.41,-52.03,;25.95,-51.98,;26.76,-53.28,;26.03,-54.64,;26.85,-55.94,;28.39,-55.89,;29.11,-54.52,;28.29,-53.22,;23.59,-50.72,;24.31,-49.36,;22.04,-50.79,;21.23,-49.49,;19.7,-49.55,;18.98,-50.91,;19.8,-52.2,;21.32,-52.14,;19.94,-55.28,;18.61,-54.51,;17.28,-55.28,;15.94,-54.51,;17.27,-56.83,;18.61,-57.6,;19.94,-56.83,;21.42,-57.31,;22.14,-58.67,;21.31,-59.98,;19.77,-59.92,;22.03,-61.34,)|
Cc1c(-c2ccc(=O)n(Cc3ccccc3)n2)c2cc(cc(F)c2n1CC(O)=O)S(C)(=O)=O
Cc1c(-c2ccc(=O)n(Cc3ccccc3)n2)c2cc(F)cc(c2n1CC(O)=O)S(C)(=O)=O
Cc1c(-c2ccc(=O)n(Cc3ccccc3)n2)c2cc(F)cc(Cl)c2n1CC(O)=O
Cc1c(-c2ccc(=O)n(Cc3ccccc3)n2)c2cc(F)cc(F)c2n1CC(O)=O
Cc1c(-c2ccc(=O)n(Cc3ccccc3)n2)c2cc(Cl)cc(Cl)c2n1CC(O)=O
Cc1c(-c2ccc(=O)n(Cc3ccccc3)n2)c2cc(Cl)cc(F)c2n1CC(O)=O
Cc1c(-c2ccc(=O)n(Cc3ccccc3)n2)c2cccc(Br)c2n1CC(O)=O
COc1ccc2n(CC(O)=O)c(C)c(-c3ccc(=O)n(Cc4ccccc4)n3)c2c1
Cc1c(-c2ccc(=O)n(Cc3ccccc3)n2)c2cc(ccc2n1CC(O)=O)S(C)(=O)=O
Cc1c(-c2ccc(=O)n(Cc3ccccc3)n2)c2cc(C)ccc2n1CC(O)=O
Cc1c(-c2ccc(=O)n(Cc3ccccc3)n2)c2cc(F)ccc2n1CC(O)=O
Cc1c(-c2ccc(=O)n(Cc3ccccc3)n2)c2cc(Cl)ccc2n1CC(O)=O
Cc1c(-c2ccc(=O)n(Cc3ccccc3)n2)c2cc(Br)ccc2n1CC(O)=O
Cc1c(-c2ccc(=O)n(Cc3ccccc3)n2)c2ccccc2n1CC(O)=O
OC(=O)Cn1cc(CCN(Cc2ccccc2)S(=O)(=O)c2ccc(F)cc2)c2ccccc12
Cc1c(CC(O)=O)c(nn1Cc1ccccc1S(=O)(=O)c1ccccc1)-c1ccncc1
Cc1nn(Cc2ccccc2S(=O)(=O)c2ccccc2)c(C)c1CC(O)=O
Cc1c(CC(O)=O)c(=O)[nH]n1Cc1ccccc1S(=O)(=O)c1ccccc1
Cc1c(CC(O)=O)c(nn1Cc1ccccc1S(=O)(=O)c1ccccc1)-c1ccc(Cl)cc1
Cc1nn(c(C)c1CC(O)=O)-c1cccc(NC(=O)[C@H]2C[C@@H]2c2ccccc2)c1 |r|
Cc1nn(Cc2ccc(cc2)S(C)(=O)=O)c(C)c1CC(O)=O
Cc1c(CC(O)=O)c(nn1Cc1ccc2ccccc2n1)-c1ccccc1
Cc1nn(Cc2ccc3ccccc3n2)c(C)c1CC(O)=O
Cc1c(CC(O)=O)c(nn1-c1ccnc2ccccc12)-c1ccccc1
Cc1c(CC(O)=O)c(nn1S(=O)(=O)c1ccc(Cl)c(Cl)c1)-c1ccccc1
Cc1c(CC(O)=O)c(nn1C(c1ccc(F)cc1)c1ccc(cc1)S(C)(=O)=O)-c1ccccc1
Cc1c(CC(O)=O)c(nn1C(c1ccc(F)cc1)c1ccc(F)cc1)-c1ccccc1
Cc1c(CC(O)=O)c(nn1C(c1ccc(F)cc1)c1ccc(F)cc1)-c1ccncc1F
OC(=O)Cc1cn(nc1-c1ccncc1)C(c1ccc(F)cc1)c1ccc(F)cc1
Cc1c(CC(O)=O)c(nn1Cc1ccc(F)cc1)-c1ccncc1
Cc1c(CC(O)=O)c(nn1C(c1ccc(F)cc1)c1ccc(F)cc1)-c1ccncc1
CC(c1ccccc1S(=O)(=O)c1ccccc1)n1nc(c(CC(O)=O)c1C)-c1ccccc1
CN(C)S(=O)(=O)c1ccccc1Cn1nc(c(CC(O)=O)c1C)-c1ccccc1
Cc1c(CC(O)=O)c(nn1Cc1ccc(F)cc1S(=O)(=O)N1CCNCC1)-c1ccccc1
Cc1c(CC(O)=O)c(nn1Cc1ccccc1S(=O)(=O)N1CCCCC1)-c1ccccc1
Cc1c(CC(O)=O)c(nn1Cc1ccccc1S(=O)(=O)N1CCOCC1)-c1ccccc1
COc1ccc(c(Cn2nc(c(CC(O)=O)c2C)-c2ccccc2)c1)S(=O)(=O)c1ccc(F)cc1
Cc1c(CC(O)=O)c(nn1Cc1ccccc1Oc1ccccc1)-c1ccccc1
Cc1c(CC(O)=O)c(nn1Cc1ccccc1-c1ccccc1)-c1ccccc1
Cc1c(CC(O)=O)c(nn1Cc1ccccc1C(=O)c1ccccc1)-c1ccccc1
Cc1c(CC(O)=O)c(nn1Cc1ccccc1Cc1ccccc1)-c1ccccc1
Cc1c(CC(O)=O)c(nn1Cc1ccccc1CS(=O)(=O)c1ccccc1)-c1ccccc1
COc1c(CC(O)=O)c(C)nn1-c1cccc(NC(=O)[C@H]2C[C@@H]2c2ccccc2)c1 |r|
CCc1ccc(cc1)-c1ccc(cc1)C(=O)N1CCc2c(C1)c1cccc(Cl)c1n2CC(O)=O
OC(=O)Cn1c2CCN(Cc2c2cc(ccc12)C(F)(F)F)C(=O)c1cccc2ccccc12
OC(=O)Cn1c2CCN(Cc2c2ccccc12)C(=O)c1ccccc1
OC(=O)Cn1c2CCN(Cc2c2cc(F)ccc12)C(=O)Cc1c[nH]c2ccccc12
OC(=O)Cn1c2CCN(Cc2c2cc(F)ccc12)C(=O)c1cccs1
Cc1ccc2n(CC(O)=O)c3CCN(Cc3c2c1)C(=O)c1ccccc1
OC(=O)Cn1c2CCN(Cc2c2cc(F)ccc12)C(=O)CCc1cccc2ccccc12
OC(=O)Cn1c2CCN(Cc2c2ccccc12)C(=O)c1cccc(Cl)c1
OC(=O)Cn1c2CCN(Cc2c2ccccc12)C(=O)c1cccc2ccccc12
OC(=O)Cn1c2CCN(Cc2c2cc(F)ccc12)C(=O)c1cccc(Cl)c1
CCc1ccc(cc1)-c1ccc(cc1)C(=O)N1CCc2c(C1)c1ccccc1n2CC(O)=O
OC(=O)Cn1c2CCN(Cc2c2cc(F)ccc12)C(=O)c1ccccc1
OC(=O)Cn1c2CCN(Cc2c2cc(F)ccc12)C(=O)c1cccc2ccccc12
Cc1ccc2n(CC(O)=O)c3CCN(Cc3c2c1)C(=O)c1cccc2ccccc12
OC(=O)Cn1c2CCN(Cc2c2cc(Cl)ccc12)C(=O)c1ccccc1
OC(=O)Cn1c2CCN(Cc2c2cc(F)cc(Cl)c12)C(=O)c1cccc(Cl)c1
OC(=O)Cn1c2CCN(Cc2c2cccc(Cl)c12)C(=O)c1ccccc1
OC(=O)Cn1c2CCN(Cc2c2cc(F)cc(Cl)c12)C(=O)c1cccc2ccccc12
OC(=O)Cn1c2CCN(Cc2c2cc(F)ccc12)C(=O)Cc1cccc2ccccc12
OC(=O)Cn1c2CCN(Cc2c2ccccc12)C(=O)C1CCCCC1
OC(=O)Cn1c2CCN(Cc2c2cc(Cl)ccc12)C(=O)c1cccc2ccccc12
Cc1cccc2c3CN(CCc3n(CC(O)=O)c12)C(=O)c1ccccc1
COc1ccc2n(CC(O)=O)c3CCN(Cc3c2c1)C(=O)c1ccccc1
CC(C)c1ccc2n(CC(O)=O)c3CCN(Cc3c2c1)C(=O)c1ccccc1
OC(=O)Cn1c2CCN(Cc2c2cc(F)cc(F)c12)C(=O)c1ccccc1
Cc1ccc2c3CN(CCc3n(CC(O)=O)c2c1)C(=O)c1ccccc1
OC(=O)Cn1cc(\C=C(/C#N)C(=O)N2CCCc3ccccc23)c2ccccc12
OC(=O)Cn1c2CCN(Cc2c2ccccc12)C(=O)Nc1ccccc1
OC(=O)Cn1c2CCC(Cc2c2ccccc12)C(=O)Nc1ccccc1
OC(=O)Cn1c2ccccc2c2cc(ccc12)C(=O)Nc1ccccc1
CN(C(=O)C(=C\c1cn(CC(O)=O)c2c(C)cccc12)\C#N)c1ccccc1
CN(C(=O)C(=C\c1cn(CC(O)=O)c2cc(C)ccc12)\C#N)c1ccccc1
CN(C(=O)C(=C\c1cn(CC(O)=O)c2ccc(C)cc12)\C#N)c1ccccc1
CN(C(=O)C(=C\c1cn(CC(O)=O)c2cccc(C)c12)\C#N)c1ccccc1
CN(C(=O)C(=C\c1cn(CC(O)=O)c2c(Cl)cccc12)\C#N)c1ccccc1
CN(C(=O)C(=C\c1cn(CC(O)=O)c2cc(Cl)ccc12)\C#N)c1ccccc1
CN(C(=O)C(=C\c1cn(CC(O)=O)c2ccc(Cl)cc12)\C#N)c1ccccc1
CN(C(=O)C(=C\c1cn(CC(O)=O)c2cccc(Cl)c12)\C#N)c1ccccc1
CN(C(=O)C(=C\c1cn(CC(O)=O)c2c(F)cccc12)\C#N)c1ccccc1
CN(C(=O)C(=C\c1cn(CC(O)=O)c2cc(F)ccc12)\C#N)c1ccccc1
CN(C(=O)C(=C\c1cn(CC(O)=O)c2ccc(F)cc12)\C#N)c1ccccc1
CN(C(=O)C(=C\c1cn(CC(O)=O)c2cccc(F)c12)\C#N)c1ccccc1
OC(=O)Cn1cc(\C=C(/C#N)C(=O)N2Cc3ccccc3Cc3ccccc23)c2ccccc12
OC(=O)Cn1cc(\C=C(/C#N)C(=O)N2CCc3ccccc23)c2ccccc12
OC(=O)Cn1cc(\C=C(/C#N)C(=O)N(CCc2ccccc2)c2ccccc2)c2ccccc12
OC(=O)Cn1cc(\C=C(/C#N)C(=O)N(Cc2ccccc2)c2ccccc2)c2ccccc12
OC(=O)Cn1cc(\C=C(/C#N)C(=O)N(C2CCCCC2)c2ccccc2)c2ccccc12
CCCCN(C(=O)C(=C\c1cn(CC(O)=O)c2ccccc12)\C#N)c1ccccc1
CN(C(=O)C(=C\c1cn(CC(O)=O)c2ccccc12)\C#N)c1ccccc1
OC(=O)Cn1cc(\C=C\C(=O)Nc2ccccc2)c2ccccc12
OC(=O)Cn1cc(\C=C(/Cl)C(=O)Nc2ccccc2)c2ccccc12
C\C(=C(\C#N)C(=O)Nc1ccccc1)c1cn(CC(O)=O)c2ccccc12
OC(=O)CCCn1cc(\C=C(/C#N)C(=O)Nc2ccccc2)c2ccccc12
OC(=O)CCn1cc(\C=C(/C#N)C(=O)Nc2ccccc2)c2ccccc12
OC(=O)Cn1cc(\C=C(/C#N)C(=O)Nc2ccccc2)c2ccccc12
OC(=O)Cn1cc(\C=C(/C#N)C(=O)Nc2cccc(Br)c2)c2ccccc12
CC(=O)N1CCc2c(C1)c1ccccc1n2CC(O)=O
CCCCCC(=O)N1CCc2c(C1)c1ccccc1n2CC(O)=O
OC(=O)Cn1c2CCN(Cc2c2ccccc12)C(=O)Cc1ccccc1
Cc1c(CC(O)=O)c2cccnc2n1Cc1ccccn1
Cc1c(CC(O)=O)c2cccnc2n1Cc1ccncc1
Cc1c(CC(O)=O)c2cccnc2n1Cc1cccnc1
Cc1c(CC(O)=O)c2cccnc2n1Cc1ccc(F)c(F)c1
Cc1c(CC(O)=O)c2cccnc2n1Cc1ccc(Cl)c(Cl)c1
Cc1c(CC(O)=O)c2cccnc2n1Cc1ccc(cc1)C(F)(F)F
Cc1c(CC(O)=O)c2cccnc2n1Cc1ccc(C)cc1
COc1ccc(Cn2c(C)c(CC(O)=O)c3cccnc23)cc1
Cc1c(CC(O)=O)c2cccnc2n1Cc1ccccc1
Cc1c(CC(O)=O)c2cccnc2n1Cc1ccccc1Cl
Cc1c(CC(O)=O)c2cccnc2n1Cc1cccc(Cl)c1
[H][C@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1ccccc1[C@@H]2N(C(C)C)C(=O)CCC(O)=O |r|
[H][C@@]12CC[C@]1([H])N(C(=O)c1ccc(F)cc1)c1ccccc1[C@@H]2N(C1CC1)C(=O)OCC(O)=O |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1ccccc1[C@@H]2N(C1CC1)C(=O)CCc1nn[nH]n1 |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1ccc(cc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O)-c1cncnc1 |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)OCc1ccccc1)c1ccccc1[C@@H]2N(CC)c1nc(cs1)C(O)=O |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)c1ccccc1)c1ccccc1[C@@H]2N(CC)C(C)=O |r|
[H][C@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1ccccc1[C@@H]2N(CC)C(=O)CCC(O)=O |r|
[H][C@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1ccccc1[C@@H]2N(CCC(F)(F)F)C(=O)CCC(O)=O |r|
[H][C@@]12CC[C@]1([H])N(C(=O)c1cccc(F)c1)c1ccccc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O |r|
[H][C@@]12CCC[C@]1([H])N(CC(=O)Nc1ccc(F)cc1)c1ccccc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O |r|
[H][C@@]12CCC[C@]1([H])N(c1nnc(o1)-c1ccccc1)c1ccccc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)OCc1ccccc1)c1ccccc1[C@@H]2N(C1CC1)C(=O)C[C@@H](C)C(O)=O |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1ccc(F)cc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1ccc(cc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O)C(F)F |r|
OC(=O)CCC(=O)N(C1CC1)C1C2CCC2N(C(=O)OCc2ccccc2)c2ccccc12
OC(=O)CCC(=O)N(C1CC1)C1C2CCCC2N(C(=O)OCc2ccccc2)c2ccccc12
[H][C@@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1cc(F)ccc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O |r|
OC(=O)CCC(=O)N(C1CC1)C1C2CCCC2N(C(=O)c2ccccc2)c2ccccc12
[H][C@@]12CC[C@]1([H])N(C(=O)c1cccc(OC(F)(F)F)c1)c1ccccc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1cc(Cl)ccc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O |r|
[H][C@@]12CC[C@]1([H])N(C(=O)c1ccc(F)cc1)c1ccccc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1cc(Cl)c(F)cc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O |r|
[H][C@@]12CC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1ccccc1[C@@H]2N(C1CC1)C(=O)OCC(O)=O |r|
[H][C@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1ccccc1[C@@H]2N(CC1CCC1)C(=O)CCC(O)=O |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)OCc1ccc(F)cc1)c1ccccc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1ccccc1[C@@H]2N(C1CC1)C(=O)c1ccccc1C(O)=O |r|
[H][C@@]12CC[C@]1([H])N(C(=O)c1cccc(F)c1)c1ccccc1[C@@H]2N(C1CC1)C(=O)OCC(O)=O |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)OCc1ccccc1)c1ccccc1[C@@H]2N(C1CC1)C(=O)CC(C)(C)C(O)=O |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1ccc(CC)cc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O |r|
OC(=O)COC(=O)N(C1CC1)C1C2CCCC2N(C(=O)c2ccccc2)c2ccccc12
[H][C@@]12CC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1ccccc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O |r|
[H][C@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1ccccc1[C@@H]2N(C)C(=O)CCC(O)=O |r|
[H][C@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1ccccc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O |r|
[H][C@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1ccccc1[C@@H]2N(C1CCC1)C(=O)CCC(O)=O |r|
[H][C@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1ccccc1[C@@H]2N(C(=O)CCC(O)=O)C1(C)CC1 |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)Nc1ccccc1)c1ccccc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)O[C@H](C)c1ccc(F)cc1)c1ccccc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)O[C@@H](C)c1ccc(F)cc1)c1ccccc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)OCc1ccccc1)c1ccccc1[C@@H]2N(C1CC1)C(=O)CC(C)C(O)=O |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)c1ccc(SC(F)(F)F)cc1)c1ccc(F)cc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1ccc(CO)cc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1ccc(cc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O)C1CC1 |r|
[H][C@@]12CCC[C@]1([H])N(C(=O)c1ccc(OC(F)(F)F)cc1)c1ccc(cc1[C@@H]2N(C1CC1)C(=O)CCC(O)=O)-c1ccc(F)cc1 |r|
OC(=O)CCCC(=O)N(C1CC1)C1C2CCCC2N(C(=O)OCc2ccccc2)c2ccccc12
OC(=O)CCC(=O)N(C1CC1)C1C2CCCCC2N(C(=O)OCc2ccccc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3ccc(cc3)C#N)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3ccc(OC(F)(F)F)cc3)cc2)c2ccccc12
Cc1ccc(cc1)C(=O)Nc1ccc(cc1)C(=O)c1ncc(CC(O)=O)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3cscn3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3cccnn3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3ccccn3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3cc4ccccc4o3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3cccc4ccccc34)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)C3CCOCC3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)CC34CC5CC(CC(C5)C3)C4)cc2)c2ccccc12 |TLB:21:22:26:20.25.19,THB:23:22:25.24.26:19|
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)CC3CCCCC3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)C3CC3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(OCCCc3ccc(Cl)cc3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(OCCc3ccc(Cl)cc3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(cc2)C(=O)NCCc2ccc(Cl)c(Cl)c2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(cc2)C(=O)Nc2ccc(Cl)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)OCc3ccc(Cl)c(Cl)c3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)Nc3ccc(Cl)c(Cl)c3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)Cc3ccc(Cl)c(Cl)c3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3ccc(Oc4ccccc4)cc3)cc2)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3ccc(cc3)-c3ccccc3)cc2)c2ccccc12
CN(C)c1ccc(cc1)C(=O)Nc1ccc(cc1)C(=O)c1ncc(CC(O)=O)c2ccccc12
OC(=O)Cc1cnc(C(=O)c2ccc(NC(=O)c3ccc(cc3)[N+]([O-])=O)cc2)c2ccccc12
Cc1c(Cc2ccccc2S(=O)(=O)c2ccccc2)c(nn1CC(O)=O)-c1cccc(c1)C(F)(F)F
Cc1c(Cc2ccccc2S(=O)(=O)c2ccc(F)cc2)c(nn1CC(O)=O)-c1ccccc1
Cc1c(Cc2ccccc2S(=O)(=O)c2ccccc2)c(nn1CC(O)=O)C(=O)N1CCOCC1
Cc1c(Cc2ccccc2S(=O)(=O)c2ccccc2)c(nn1CC(O)=O)-c1cc(Cl)ccc1Cl
Cc1c(Cc2ccccc2S(=O)(=O)c2ccccc2)c(nn1CC(O)=O)-c1ccncc1
Cc1c(Cc2ccccc2S(=O)(=O)c2ccccc2)c(nn1CC(O)=O)-c1cncnc1
Cc1nn(CC(O)=O)c(C)c1Cc1ccccc1S(=O)(=O)c1ccccc1
Cc1c(Cc2ccccc2S(=O)(=O)c2cccc3cccnc23)c(nn1CC(O)=O)-c1ccccc1
Cc1c(Cc2ccccc2S(=O)(=O)Cc2ccccc2)c(nn1CC(O)=O)-c1ccccc1
Cc1c(Cc2ccccc2S(=O)(=O)c2ccc(cc2)S(C)(=O)=O)c(nn1CC(O)=O)-c1ccccc1
CN(C)c1ccc(cc1)S(=O)(=O)c1ccccc1Cc1c(C)n(CC(O)=O)nc1-c1ccccc1
Cc1c(Cc2ccccc2S(=O)(=O)c2ccc(OC(F)(F)F)cc2)c(nn1CC(O)=O)-c1ccccc1
COc1ccc(cc1)S(=O)(=O)c1ccccc1Cc1c(C)n(CC(O)=O)nc1-c1ccccc1
Cc1c(Cc2ccccc2S(=O)(=O)c2ccc(Cl)cc2)c(nn1CC(O)=O)-c1ccccc1
Cc1c(Cc2ccccc2S(=O)(=O)c2ccc(C)c(C)c2)c(nn1CC(O)=O)-c1ccccc1
Cc1c(Cc2ccccc2S(=O)c2ccc(C)c(C)c2)c(nn1CC(O)=O)-c1ccccc1
Cc1c(Cc2ccccc2Sc2ccc(C)c(C)c2)c(nn1CC(O)=O)-c1ccccc1
CN(C)C(=O)c1cccc(c1)S(=O)(=O)c1ccccc1Cc1c(C)n(CC(O)=O)nc1-c1ccccc1
COc1cccc(c1)S(=O)(=O)c1ccccc1Cc1c(C)n(CC(O)=O)nc1-c1ccccc1
COc1cccc(Sc2ccccc2Cc2c(C)n(CC(O)=O)nc2-c2ccccc2)c1
Cc1c(Cc2ccccc2S(=O)(=O)c2cccc(c2)C(F)(F)F)c(nn1CC(O)=O)-c1ccccc1
Cc1c(Cc2ccccc2S(=O)(=O)c2cccc(Cl)c2)c(nn1CC(O)=O)-c1ccccc1
Cc1c(Cc2ccccc2S(=O)(=O)c2cccc(F)c2)c(nn1CC(O)=O)-c1ccccc1
Cc1c(Cc2ccccc2S(=O)(=O)c2c(C)cccc2C)c(nn1CC(O)=O)-c1ccccc1
Cc1c(Cc2ccccc2S(=O)(=O)c2ccccc2C)c(nn1CC(O)=O)-c1ccccc1
COc1ccc(c(Cc2c(C)n(CC(O)=O)nc2-c2ccccc2)c1)S(=O)(=O)c1ccccc1
Cc1c(Cc2cc(F)ccc2S(=O)(=O)c2ccccc2)c(nn1CC(O)=O)-c1ccccc1
Cc1c(Cc2ccncc2S(=O)(=O)c2ccccc2)c(nn1CC(O)=O)-c1ccccc1
COC(=O)c1ccc(Cc2c(C)n(CC(O)=O)nc2-c2ccccc2)c(c1)S(=O)(=O)c1ccccc1
Cc1c(Cc2ccc(cc2S(=O)(=O)c2ccccc2)C(O)=O)c(nn1CC(O)=O)-c1ccccc1
COc1ccc(Cc2c(C)n(CC(O)=O)nc2-c2ccccc2)c(c1)S(=O)(=O)c1ccccc1
Cc1c(Cc2ccc(cc2S(=O)(=O)c2ccccc2)C(F)(F)F)c(nn1CC(O)=O)-c1ccccc1
Cc1c(Cc2ccccc2S(=O)(=O)c2ccccc2F)c(nn1CC(O)=O)-c1ccccc1
OC(=O)CCCCc1nc2cc(ccc2c(=O)n1-c1ccc(F)cc1)-c1cc(on1)-c1ccccc1
CC1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1ccccc1 |c:3|
CCC1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1ccccc1 |c:4|
CCCC1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1ccccc1 |c:5|
CCCCC1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1ccccc1 |c:6|
OCC1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1ccccc1 |c:4|
COCC1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1ccccc1 |c:5|
OC(=O)CCCCc1nc2cc(ccc2c(=O)n1-c1ccc(F)cc1)C1=NOC(C1)(c1ccccc1)c1ccccc1 |t:28|
OC(=O)CCCCc1nc2cc(ccc2c(=O)n1-c1ccc(F)cc1)C1=NOC2(C1)Cc1ccccc1C2 |t:28|
C[C@]1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1ccccc1 |r,c:3|
C[C@]1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1ccc(F)cc1 |r,c:3|
C[C@]1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1cc(F)cc(F)c1 |r,c:3|
C[C@]1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1ccc(Cl)cc1 |r,c:3|
C[C@]1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1cccc(c1)C#N |r,c:3|
C[C@@]1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1ccccc1 |r,c:3|
C[C@@]1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1ccc(F)cc1 |r,c:3|
C[C@@]1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1cc(F)cc(F)c1 |r,c:3|
C[C@@]1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1ccc(Cl)cc1 |r,c:3|
C[C@@]1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1cccc(c1)C#N |r,c:3|
C[C@@]1(Cc2ccccc2)CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O |r,c:11|
C[C@]1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)[C@@H](O)c1ccccc1 |r,c:3|
C[C@]1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)[C@H](O)c1ccccc1 |r,c:3|
C[C@]1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1nc2ccccc2o1 |r,c:3|
C[C@]1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1nc2ccccc2s1 |r,c:3|
C[C@]1(Cc2ccccc2)CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O |r,c:11|
C[C@@]1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)[C@@H](O)c1ccccc1 |r,c:3|
C[C@@]1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)[C@H](O)c1ccccc1 |r,c:3|
C[C@@]1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1nc2ccccc2o1 |r,c:3|
C[C@@]1(CC(=NO1)c1ccc2c(c1)nc(CCCCC(O)=O)n(-c1ccc(F)cc1)c2=O)c1nc2ccccc2s1 |r,c:3|
OC(=O)CCCCc1cc2cc(ccc2c(=O)n1-c1ccc(F)cc1)C(=O)Nc1noc(Cc2ccc(F)cc2)n1
C[C@@H](NC(=O)c1ccc2c(cc(CCCCC(O)=O)[nH]c2=O)c1)c1ccc(F)cc1 |r|
OC(=O)CCCCc1cc2cc(ccc2c(=O)n1-c1ccc(F)cc1)C(=O)Nc1cc(Cc2ccc(F)cc2)on1
OC(=O)CCCCc1cc2cc(ccc2c(=O)n1-c1ccc(F)cc1)C(=O)Nc1noc(n1)C1Cc2ccccc2C1
CC(c1nc(NC(=O)c2ccc3c(cc(CCCCC(O)=O)n(-c4ccc(F)cc4)c3=O)c2)no1)c1ccc(F)cc1
CC1(CC(NC(=O)c2ccc3c(cc(CCCCC(O)=O)n(-c4ccc(F)cc4)c3=O)c2)=NO1)c1nc2ccc(F)cc2o1 |c:34|
Cc1c(nc2ccc(Br)cc2c1C(=O)NC[C@H](CCC(O)=O)c1ccccc1Cl)N1CCCC1 |r|