1324 SMILES Strings for Protein cereblon

Compound Name
SMILES String
Nc1cccc2C(=O)N(Cc12)C1CCC(=O)NC1=O
Nc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12
c1ccc2c(c1)C(=O)N(C2=O)[C@H]3CCC(=O)NC3=O
c1ccc2c(c1)C(=O)N(C2=O)[C@@H]3CCC(=O)NC3=O
CN1C(=O)CCC(N2C(=O)c3cccc(NCCOCCOCCOc4ccc(COc5ccc6oc(nc6c5)-c5ccc(=O)n(C)n5)nc4)c3C2=O)C1=O
Cn1nc(ccc1=O)-c1nc2cc(OCc3ccc(OCCOCCOCCNc4cccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c45)cn3)ccc2o1
Cn1nc(ccc1=O)-c1nc2cc(NC(=O)c3ccc(OCCOCCOCCOCCOCCOCCNc4cccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c45)cn3)ccc2o1
Cn1nc(ccc1=O)-c1nc2cc(NC(=O)c3ccc(OCCOCCOCCNc4cccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c45)cn3)ccc2o1
Cn1nc(ccc1=O)-c1nc2cc(NC(=O)c3ccc(OCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNc4cccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c45)cn3)ccc2o1
Cn1nc(ccc1=O)-c1nc2cc(NC(=O)c3ccc(OCCOCCOCCOCCNc4cccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c45)cn3)ccc2o1
Cn1nc(ccc1=O)-c1nc2cc(NC(=O)c3ccc(OCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNc4cccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c45)cn3)ccc2o1
Cn1nc(ccc1=O)-c1nc2cc(NC(=O)c3ccc(OCCOCCOCCOCCOCCOCCOCCOCCOCCNc4cccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c45)cn3)ccc2o1
CN1C(=O)CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCCOCCOc4ccc(nc4)C(=O)Nc4ccc5oc(nc5c4)-c4ccc(=O)n(C)n4)c3C2=O)C1=O
CN1C(=O)CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOc4ccc(nc4)C(=O)Nc4ccc5oc(nc5c4)-c4ccc(=O)n(C)n4)c3C2=O)C1=O
CN1C(=O)CCC(N2C(=O)c3cccc(NCCOCCOCCOc4ccc(nc4)C(=O)Nc4ccc5oc(nc5c4)-c4ccc(=O)n(C)n4)c3C2=O)C1=O
O=C1CCc2cc(ccc2N1)-n1ccnc1
CNC(=O)c1ccc2n(c(nc2c1)-c1cc(nc2ccccc12)-c1cncn1C)-c1ccc2NC(=O)CCc2c1
CCc1nc2cc(ccc2n1-c1ccc2NC(=O)CCc2c1)C(=O)NC
CNC(=O)c1ccc2n(c(nc2c1)-c1ccnc2ccccc12)-c1ccc2NC(=O)CCc2c1
Cn1cncc1-c1cc(C(=O)Nc2ccc3NC(=O)CCc3c2)c2ccccc2n1
CNC(=O)c1ccc2n(c(Cc3ccccc3)nc2c1)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)C1CC1)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(COCc3ccccc3)nc2c1)-c1ccc2NC(=O)CCc2c1
O=C1CCc2cc(cnc2N1)-n1ccnc1
CNC(=O)c1ccc2n(c(Cc3ccccc3OC)nc2c1)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)C1(CC1)c1ccccc1)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1cn[nH]c1)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1ccnc(OC)c1)-c1ccc2NC(=O)CCc2c1
O=C1CCc2cc(ccc2N1)-n1cncc1-c1ccccc1
CNC(=O)c1ccc2n(c(CO)nc2c1)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(CCNC(=O)C3CC3)nc2c1)-c1ccc2NC(=O)CCc2c1
CCOC(=O)c1nc2cc(ccc2n1-c1ccc2NC(=O)CCc2c1)C(=O)NC
CNC(=O)c1ccc2n(c(CCN)nc2c1)-c1ccc2NC(=O)CCc2c1
COC(=O)c1ccc(Nc2ccc3NC(=O)CCc3c2)cc1
CNC(=O)c1ccc2n(c(nc2c1)C(=O)N1CCOCC1)-c1ccc2NC(=O)CCc2c1
O=C(Nc1cnc2NC(=O)CCc2c1)C1CCCc2ccccc12
COC(=O)c1ccc2n(c(nc2c1)-c1ccnc(OC)c1)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1cccc(OC)n1)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1ccc(OC)nc1)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1cc(OC)ccn1)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1cccnc1OC)-c1ccc2NC(=O)CCc2c1
COc1ccc(cc1)-c1cncn1-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)C(C)C)-c1cnc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1ccnc(OC)c1)-c1cnc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1ccccc1C(C)=O)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1ccccc1C(=O)NC)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1cccc(OC)c1)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1ccc(CNC(C)=O)cc1)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1cc(OC)ccc1F)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1ccccc1CO)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1ccccc1NC(C)=O)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1ccccc1N)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1cc(OC)cc(C)n1)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1ncccc1C(=O)OC)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(Cc3ccccc3C(=O)OC)nc2c1)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1ncccc1NC(C)=O)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1ncccc1N)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1cc(OC)ncc1F)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1ccncc1C(F)(F)F)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1ccnc(CO)c1)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(Cc3ccc(cc3OC)C(F)(F)F)nc2c1)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1cccnc1C(C)=O)-c1ccc2NC(=O)CCc2c1
CNC(=O)c1ccc2n(c(nc2c1)-c1ncccc1C(=O)NC)-c1ccc2NC(=O)CCc2c1
COC(=O)c1ccc2n(c(nc2c1)C(C)C)-c1ccc2NC(=O)CCc2n1
CNC(=O)c1ccc2n(c(nc2c1)C(C)C)-c1ccc2NC(=O)CCc2n1
CC(C)c1nc2cc(ccc2n1-c1ccc2NC(=O)CCc2n1)C(=O)N(C)C
O=C1CCc2ccc(cc2N1)-n1ccnc1
O=C(N1CCc2ccccc12)c1ccc2NC(=O)CCc2c1
O=C(N1CCc2cccnc12)c1ccc2NC(=O)CCc2c1
O=C(N1CCCc2ccccc12)c1ccc2NC(=O)CCc2c1
CC(=O)N1CCC(CC1)NC(=O)c1ccc2NC(=O)CCc2c1
O=C(N1CCc2ccccc12)c1cnc2NC(=O)CCc2c1
O=C(N1CCc2cccnc12)c1cnc2NC(=O)CCc2c1
O=C(N1CCCc2ccccc12)c1cnc2NC(=O)CCc2c1
CC(C)c1nc2ccccc2n1-c1ccc2NC(=O)NCc2c1
CNC(=O)c1ccc2n(c(nc2c1)C(C)C)-c1ccc2NC(=O)NCc2c1
Cc1nnc2[C@H](CC(=O)NCCCCCCCCCCNC(=O)c3ccc4n(c(nc4c3)-c3cc(nc4ccccc34)-c3cncn3C)-c3ccc4NC(=O)CCc4c3)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1 |r,c:66|
Cc1nnc2[C@H](CC(=O)NCCCCCNC(=O)c3ccc4n(c(nc4c3)-c3cc(nc4ccccc34)-c3cncn3C)-c3ccc4NC(=O)CCc4c3)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1 |r,c:61|
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)NCCOCCOCCNC(=O)c1ccc3n(c(nc3c1)-c1cc(nc3ccccc13)-c1cncn1C)-c1ccc3NC(=O)CCc3c1)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
O=C(NCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1)Nc1ccccc1
Clc1ccc(NC(=O)NCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1
Clc1cccc(NC(=O)NCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
Clc1ccccc1NC(=O)NCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
COc1ccc(NC(=O)NCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1
COc1cccc(NC(=O)NCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
COc1ccccc1NC(=O)NCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Cc1ccc(NC(=O)NCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1Cl
Brc1ccc(NC(=O)NCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1
CC(C)(C)NC(=O)NCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
CC(C)(C)c1ccccc1NC(=O)NCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
CC(C)NC(=O)NCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
CCCCCCNC(=O)NCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
CCCNC(=O)NCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
CCNC(=O)NCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
CCOc1ccc(NC(=O)NCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1
COc1ccc(C)cc1NC(=O)NCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
CCc1ccc(NC(=O)NCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1
Cc1c(Cl)cccc1NC(=O)NCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Cc1cc(C)cc(NC(=O)NCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
Cc1ccc(NC(=O)NCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1
CCOc1ccccc1NC(=O)NCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
COc1ccc(NC(=O)NCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c(C)c1
O=C(NCc1ccccc1)NCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C1CCC(Sc2ccccc2)C(=O)N1
O=C1CCC(Sc2ccccn2)C(=O)N1
Fc1ccc(SC2CCC(=O)NC2=O)cc1
Clc1ccc2nc(SC3CCC(=O)NC3=O)[nH]c2c1
COc1ccc(SC2CCC(=O)NC2=O)cc1
OC(=O)c1ccc(SC2CCC(=O)NC2=O)cc1
CCn1c(SC2CCC(=O)NC2=O)nc2ccccc12
Cn1c(SC2CCC(=O)NC2=O)nc2ccccc12
CC(=O)Nc1ccc(SC2CCC(=O)NC2=O)cc1
Nc1ccc(SC2CCC(=O)NC2=O)cc1
Clc1ccc(SC2CCC(=O)NC2=O)cc1
FC(F)(F)c1ccc(SC2CCC(=O)NC2=O)cc1
CCc1ccc(SC2CCC(=O)NC2=O)cc1
c1ccc(cc1)N2CCC(=O)NC2=O
O=C1CCN(C(=O)N1)c1ccccn1
O=C1CCN(Cc2ccccc2)C(=O)N1
O=C1CCN(Cc2ccccn2)C(=O)N1
O=c1ccn(-c2ccccc2)c(=O)[nH]1
O=c1ccn(-c2ccccn2)c(=O)[nH]1
O=C1NC(=O)C(S1)N1CC(OC1=O)c1ccccc1
Cn1c2ccccc2n(C2SC(=O)NC2=O)c1=O
O=C1CCC(Sc2ccncc2)C(=O)N1
CC(C)(C)n1c(SC2CCC(=O)NC2=O)nc2ccccc12
CCc1ccc(cc1)S(=O)C1CCC(=O)NC1=O
CCc1ccc(cc1)S(=O)(=O)C1CCC(=O)NC1=O
Cc1ccc(SC2CCC(=O)NC2=O)cc1
O=C1CCC(Sc2ccc(cc2)C#N)C(=O)N1
CC(C)c1ccc(SC2CCC(=O)NC2=O)cc1
Cc1cccc(SC2CCC(=O)NC2=O)c1
O=C1CCC(Sc2nc3ccccc3n2C2CC2)C(=O)N1
Cn1cc(C2SC(=O)NC2=O)c2ccccc12
O=C1CCC(Sc2cccs2)C(=O)N1
Cn1ccnc1SC1CCC(=O)NC1=O
Oc1ccccc1SC1CCC(=O)NC1=O
COc1ccccc1SC1CCC(=O)NC1=O
Cn1ccc(n1)N1CCC(=O)NC1=O
O=C1NC(=O)C(S1)N1CCNC(=O)C1
CCc1ccc(OC2CCC(=O)NC2=O)cc1
Cc1ccc(SC2CCC(=O)NC2=O)c(C)c1
Cc1occc1SC1CCC(=O)NC1=O
Cn1nc(C2SC(=N)NC2=O)c2ccccc12
O=C1NC(=O)C(S1)N1CCN(CC1=O)c1ccccc1
O=C1CCC(Sc2ncccn2)C(=O)N1
CCCCc1ccc(SC2CCC(=O)NC2=O)cc1
CN(C)c1ccc(SC2CCC(=O)NC2=O)cc1
CCOc1cccc(SC2CCC(=O)NC2=O)c1
COc1cccc(SC2CCC(=O)NC2=O)c1
Cn1nc(cc1-c1ccccc1)N1CCC(=O)NC1=O
Cc1cc(C)nc(SC2CCC(=O)NC2=O)n1
Clc1ccc(SC2CCC(=O)NC2=O)nc1
FC(F)(F)c1cc(SC2CCC(=O)NC2=O)cc(c1)C(F)(F)F
O=C1CCC(Sc2nc(=O)cc([nH]2)-c2ccccc2)C(=O)N1
Cc1cc(O)nc(SC2CCC(=O)NC2=O)n1
O=C1CCC(Sc2nc3ccccc3[nH]2)C(=O)N1
O=C1CCC(Sc2cccc3cccnc23)C(=O)N1
FC(F)(F)c1ccc(SC2CCC(=O)NC2=O)nc1
FC(F)(F)Oc1ccccc1SC1CCC(=O)NC1=O
Clc1ccc(Cl)c(SC2CCC(=O)NC2=O)c1
Clc1cc(Cl)c(SC2CCC(=O)NC2=O)cc1Cl
O=C1CCC(Oc2ccccc2)C(=O)N1
Brc1ccc(SC2CCC(=O)NC2=O)nc1
Cn1ccc(CN2CCC(=O)NC2=O)n1
O=C1CCC(SCc2ccccc2)C(=O)N1
Brc1cccc(SC2CCC(=O)NC2=O)c1
FC(F)(F)c1ccccc1SC1CCC(=O)NC1=O
[O-][n+]1ccccc1SC1CCC(=O)NC1=O
OC(=O)c1ccnc(SC2CCC(=O)NC2=O)c1
OCc1ccc(SC2CCC(=O)NC2=O)cc1
Nc1cc(=O)nc(SC2CCC(=O)NC2=O)[nH]1
Fc1ccc(SC2CCC(=O)NC2=O)cc1F
CC(C)(C)c1ccc(OC2CCC(=O)NC2=O)cc1
O=C1CCC(SC2CCCCC2)C(=O)N1
O=C1CCC(Sc2ccccc2C#N)C(=O)N1
Cn1c2ccccc2cc(C2SC(=O)NC2=O)c1=O
O=C1CCC(Oc2ccc3ccccc3c2)C(=O)N1
Nc1cc(ccc1SC1CCC(=O)NC1=O)C(F)(F)F
CCc1cccc(SC2CCC(=O)NC2=O)c1
Clc1cccc(SC2CCC(=O)NC2=O)c1
OC(=O)c1cccc(SC2CCC(=O)NC2=O)c1
CCCCc1ccc(OC2CCC(=O)NC2=O)cc1
CN(C)c1ccc(OC2CCC(=O)NC2=O)cc1
OC(=O)c1cccnc1SC1CCC(=O)NC1=O
OCc1cccc(SC2CCC(=O)NC2=O)c1
CN1CCN(CC1)c1ccc(OC2CCC(=O)NC2=O)cc1
O=C1CCC(Oc2cccc3cccnc23)C(=O)N1
NC(=O)c1ccnc(SC2CCC(=O)NC2=O)c1
CNC(=O)c1ccnc(SC2CCC(=O)NC2=O)c1
CN(C)C(=O)c1ccnc(SC2CCC(=O)NC2=O)c1
OC(=O)c1ccc(SC2CCC(=O)NC2=O)nc1
O=C1CCC(Sc2cccc(c2)C#N)C(=O)N1
CCN(CC)c1ccc(SC2CCC(=O)NC2=O)cc1
OC(=O)c1cccc(SC2CCC(=O)NC2=O)n1
Cc1c(SC2CCC(=O)NC2=O)cccc1C(O)=O
Cc1coc(n1)-c1ccnc(SC2CCC(=O)NC2=O)c1
O=C1CCC(Sc2cc(ccn2)-c2nn[nH]n2)C(=O)N1
NC(=O)c1cccnc1SC1CCC(=O)NC1=O
CN(C)C(=O)c1cccnc1SC1CCC(=O)NC1=O
COCCOCCNC(=O)c1cccnc1SC1CCC(=O)NC1=O
Cn1cccc(N2CCC(=O)NC2=O)c1=O
Cn1c2ccccc2cc(N2CCC(=O)NC2=O)c1=O
CN1Cc2ccccc2C(N2CCC(=O)NC2=O)C1=O
Cn1cc2ccccc2c(N2CCC(=O)NC2=O)c1=O
Fc1ccccc1Nc1nccc(NCC(=O)Nc2cccc3C(=O)N(Cc23)C2CCC(=O)NC2=O)n1
O=C(CNc1ccnc(Nc2ccc3CCCc3c2)n1)Nc1cccc2C(=O)N(Cc12)C1CCC(=O)NC1=O
O=C(CNc1ccnc(NCc2ccc3OCOc3c2)n1)Nc1cccc2C(=O)N(Cc12)C1CCC(=O)NC1=O
OC[C@@H]1CCCN1c1nccc(NCC(=O)Nc2cccc3C(=O)N(Cc23)C2CCC(=O)NC2=O)n1 |r|
O=C(CNc1ccnc(Nc2ccc3OCOc3c2)n1)Nc1cccc2C(=O)N(Cc12)C1CCC(=O)NC1=O
O=C(CNc1ccnc(NCCCN2CCCC2=O)n1)Nc1cccc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1ccc(Nc2nccc(NCC(=O)Nc3cccc4C(=O)N(Cc34)C3CCC(=O)NC3=O)n2)cc1
COc1cccc(c1)-c1nccc(NCC(=O)Nc2cccc3C(=O)N(Cc23)C2CCC(=O)NC2=O)n1
COc1ccc(OC)c(c1)-c1nccc(NCC(=O)Nc2cccc3C(=O)N(Cc23)C2CCC(=O)NC2=O)n1
Fc1ccc(cc1)-c1nccc(NCC(=O)Nc2cccc3C(=O)N(Cc23)C2CCC(=O)NC2=O)n1
CC(=O)c1ccc(cc1)-c1nccc(NCC(=O)Nc2cccc3C(=O)N(Cc23)C2CCC(=O)NC2=O)n1
O=C(CNc1ccnc(n1)-c1cc2ccccc2o1)Nc1cccc2C(=O)N(Cc12)C1CCC(=O)NC1=O
OC[C@H]1CCCN1c1nccc(NCC(=O)Nc2cccc3C(=O)N(Cc23)C2CCC(=O)NC2=O)n1 |r|
COc1ccccc1Nc1nccc(NCC(=O)Nc2cccc3C(=O)N(Cc23)C2CCC(=O)NC2=O)n1
FC(F)(F)c1cccc(c1)N1CCN(CC1)c1nccc(NCC(=O)Nc2cccc3C(=O)N(Cc23)C2CCC(=O)NC2=O)n1
CN(c1ccccc1)c1nccc(NCC(=O)Nc2cccc3C(=O)N(Cc23)C2CCC(=O)NC2=O)n1
O=C1Cc2ccc(cc2N1)-c1ccccc1
O=C1Cc2ccc(cc2N1)-c1ccncc1
O=C1Cc2ccc(cc2N1)-c1cccnc1
O=C1Cc2ccc(cc2N1)-c1ccccn1
Cc1cc(ccn1)-c1ccc2CC(=O)Nc2c1
Cc1cnccc1-c1ccc2CC(=O)Nc2c1
CC1C(=O)Nc2cc(ccc12)-c1ccncc1
CN1C(=O)Cc2ccc(cc12)-c1ccncc1
Clc1cc(ccn1)-c1ccc2CC(=O)Nc2c1
COc1cc(ccn1)-c1ccc2CC(=O)Nc2c1
Nc1cc(ccn1)-c1ccc2CC(=O)Nc2c1
Nc1cnccc1-c1ccc2CC(=O)Nc2c1
Nc1ccc(cn1)-c1ccc2CC(=O)Nc2c1
CCOC(=O)c1cc(ccn1)-c1ccc2CC(=O)Nc2c1
Cn1cc(cn1)-c1ccc2CC(=O)Nc2c1
O=C1Cc2ccc(cc2N1)-c1ccc2[nH]ccc2c1
O=C1Cc2ccc(cc2N1)-c1cnc2[nH]ccc2c1
O=C1Cc2ccc(cc2N1)-c1ccc(CN2CCNCC2)cc1
O=C1Cc2ccc(cc2N1)-c1cccc(CN2CCNCC2)c1
O=C(N1CCNCC1)c1ccc(cc1)-c1ccc2CC(=O)Nc2c1
O=C(N1CCNCC1)c1cccc(c1)-c1ccc2CC(=O)Nc2c1
CNC(=O)c1ccc(cc1)-c1ccc2CC(=O)Nc2c1
CNC(=O)c1cccc(c1)-c1ccc2CC(=O)Nc2c1
O=C(Nc1ccccc1)c1ccc2CC(=O)Nc2c1
O=C(NC1CCCCC1)c1ccc2CC(=O)Nc2c1
CC(=O)N1CCC(CC1)C(=O)Nc1ccc2CC(=O)Nc2c1
CN1CCC(CC1)NC(=O)c1ccc2CC(=O)Nc2c1
CN1CCN(CCNC(=O)c2ccc3CC(=O)Nc3c2)CC1
O=C(N1CCCCC1)c1ccc2CC(=O)Nc2c1
Clc1cc2CC(=O)Nc2cc1C(=O)N1CCCCC1
O=C(Nc1ccncc1)c1ccc2CC(=O)Nc2c1
O=C(Nc1ccc2CC(=O)Nc2c1)c1ccncc1
O=C(NCc1cccnc1)c1ccc2CC(=O)Nc2c1
O=C1Cc2ccc(OC3CCNCC3)cc2N1
Clc1nccc(Oc2ccc3CC(=O)Nc3c2)n1
COC(=O)COc1ccc2CC(=O)Nc2c1
O=C1Cc2cccc(c2N1)-c1ccncc1
O=C1Cc2c(N1)cccc2-c1ccncc1
O=C1Cc2cc(ccc2N1)-c1ccncc1
Nc1cc(ccn1)-c1ccc2NC(=O)Cc2c1
COc1cc(ccn1)-c1ccc2NC(=O)Cc2c1
Nc1ccc(cn1)-c1ccc2NC(=O)Cc2c1
Cc1cc(N)ncc1-c1ccc2NC(=O)Cc2c1
Cc1nc(N)ccc1-c1ccc2NC(=O)Cc2c1
Nc1ncccc1-c1ccc2NC(=O)Cc2c1
CNc1ccc(cn1)-c1ccc2NC(=O)Cc2c1
CNc1cc(ccn1)-c1ccc2NC(=O)Cc2c1
CC(=O)Nc1ncc(cc1C)-c1ccc2NC(=O)Cc2c1
CC(=O)Nc1ccc(c(C)n1)-c1ccc2NC(=O)Cc2c1
CC(=O)Nc1cc(C)c(cn1)-c1ccc2NC(=O)Cc2c1
O=C1Cc2cc(ccc2N1)-c1ccccc1
CC(C)(C)OC(=O)N1CCN(CC1)C(=O)c1ccc(cc1)-c1ccc2NC(=O)Cc2c1
CC(C)(C)OC(=O)N1CCN(CC1)C(=O)c1cccc(c1)-c1ccc2NC(=O)Cc2c1
O=C(N1CCNCC1)c1ccc(cc1)-c1ccc2NC(=O)Cc2c1
O=C(N1CCNCC1)c1cccc(c1)-c1ccc2NC(=O)Cc2c1
O=C1Cc2cc(ccc2N1)-c1cccnc1
O=C1Cc2cc(ccc2N1)-c1ccc(nc1)N1CCCCC1
O=C(N1CCCCC1)c1ccc2NC(=O)Cc2c1
O=C(Nc1ccc2NC(=O)Cc2c1)c1ccncc1
CC(=O)N1CCC(CC1)C(=O)Nc1ccc2NC(=O)Cc2c1
FC1(F)C(=O)Nc2cc(ccc12)-c1ccncc1
CC1(C)C(=O)Nc2cc(ccc12)-c1ccncc1
O=C(OCc1ccccc1)N1CCC(=CC1)c1ccc2CC(=O)Nc2c1 |c:14|
O=C1Cc2ccc(cc2N1)-c1ccc(nc1)N1CCCCC1
O=C1Cc2ccc(cc2N1)-c1ccc(nc1)N1CCNCC1
CN1CCN(CC1)C(=O)c1ccc2NC(=O)Cc2c1
O=C(N1CCC(CC1)c1ccccc1)c1ccc2NC(=O)Cc2c1
O=C(N1CCC(Cc2ccccc2)CC1)c1ccc2NC(=O)Cc2c1
Fc1ccc(cn1)-c1ccc2CC(=O)Nc2c1
O=C(Nc1ccc2CC(=O)Nc2c1)c1cccnc1
O=C(Nc1ccc2NC(=O)Cc2c1)c1cccnc1
O=C1Cc2cc(ncc2N1)-c1ccncc1
O=C1Cc2cnc(cc2N1)-c1ccncc1
O=C1Cc2ncc(cc2N1)-c1ccncc1
Fc1cc(ccn1)C(=O)Nc1ccc2NC(=O)Cc2c1
NC1CCN(CC1)C(=O)c1ccc2CC(=O)Nc2c1
NC1CCN(CC1)C(=O)c1ccc2NC(=O)Cc2c1
COC(=O)c1ccccc1-c1ccc2CC(=O)Nc2c1
NC1CCCN(C1)C(=O)c1ccc2CC(=O)Nc2c1
NC1CCCN(C1)C(=O)c1ccc2NC(=O)Cc2c1
CC(C)C1C(=O)Nc2ccc(cc12)-c1ccncc1
CN1C(=O)Cc2cc(ccc12)C(=O)N1CCCCC1
[N-]=[N+]=NCCOCCOCCOCCNC(=O)c1cc(ccn1)-c1ccc2CC(=O)Nc2c1
[N-]=[N+]=NCCOCCOCCOCCNc1cc(ccn1)-c1ccc2CC(=O)Nc2c1
[N-]=[N+]=NCCOCCOCCOCCNc1ccc(cn1)C(=O)Nc1ccc2NC(=O)Cc2c1
NCCCCCNc1cc(ccn1)-c1ccc2CC(=O)Nc2c1
[N-]=[N+]=NCCOCCOCCOCCNc1cc(ccn1)-c1ccc2NC(=O)Cc2c1
[N-]=[N+]=NCCOCCOCCOCCNc1ccc(cn1)-c1ccc2CC(=O)Nc2c1
Nc1ccc(OCCOCCOCCOCCNC(=O)c2cccc(c2)-c2ccc3CC(=O)Nc3c2)cc1
Nc1ccc(OCCOCCOCCOCCNC(=O)c2cccc(c2)-c2ccc3NC(=O)Cc3c2)cc1
[N-]=[N+]=NCCOCCOCCOCCNc1ccc(cn1)-c1ccc2NC(=O)Cc2c1
Nc1ccc(OCCOCCOCCOCCNc2ccc(cn2)-c2ccc3NC(=O)Cc3c2)cc1
[N-]=[N+]=NCCOCCOCCOCCNc1ncccc1-c1ccc2NC(=O)Cc2c1
[N-]=[N+]=NCCOCCOCCOCCNc1ncccc1-c1ccc2CC(=O)Nc2c1
O=C1CCC2(CCNC2)C(=O)N1
CN1CC2(CC1=O)CCC(=O)NC2=O
O=C(Cc1ccccc1)N1CCC2(C1)CCC(=O)NC2=O
O=C(C1CCc2ccccc12)N1CCC2(C1)CCC(=O)NC2=O
[O-][N+](=O)c1cccc(c1)C(=O)N1CCC2(C1)CCC(=O)NC2=O
COC(=O)c1ccc(nc1)N1CCC2(C1)CCC(=O)NC2=O
O=C1CCC2(CCN(C2)c2nc3ncccc3s2)C(=O)N1
[O-][N+](=O)c1ccc(cc1)N1CCC2(C1)CCC(=O)NC2=O
[O-][N+](=O)c1ccc2[nH]c(nc2c1)N1CCC2(C1)CCC(=O)NC2=O
[O-][N+](=O)c1ccc2[nH]c(nc2c1)N1CCC2(C1)CCC(=O)NC2=O
[O-][N+](=O)c1ccc2[nH]c(nc2c1)N1CCC2(C1)CCC(=O)NC2=O
O=C1CCC2(CCN(C2)c2nc3ccccc3s2)C(=O)N1
COC(=O)c1cccc2nc([nH]c12)N1CCC2(C1)CCC(=O)NC2=O
COC(=O)c1ccnc(n1)N1CCC2(C1)CCC(=O)NC2=O
O=C1CCC2(CCN(C2)c2ccc3ccccc3n2)C(=O)N1
Nc1ccc2nc(sc2c1)N1CCC2(C1)CCC(=O)NC2=O
O=C1CCC2(CCN(C2)c2nc3ncccc3o2)C(=O)N1
O=C1CCC2(CCN(C2)c2nc3ccccc3o2)C(=O)N1
Cn1c(nc2ccccc12)N1CCC2(C1)CCC(=O)NC2=O
O=C1CCC2(CCN(C2)c2nc3cnccc3s2)C(=O)N1
COC(=O)c1ccc2nc(sc2c1)N1CCC2(C1)CCC(=O)NC2=O
COC(=O)c1csc(n1)N1CCC2(C1)CCC(=O)NC2=O
COC(=O)c1cnc(s1)N1CCC2(C1)CCC(=O)NC2=O
CC(C)(C)OC(=O)c1ccc(nc1)N1CCC2(C1)CCC(=O)NC2=O
O=C(N1CCC2(C1)CCC(=O)NC2=O)c1ccc2ncsc2c1
[O-][N+](=O)c1ccnc(c1)C(=O)N1CCC2(C1)CCC(=O)NC2=O
O=C(N1CCC2(C1)CCC(=O)NC2=O)c1cccc2NC(=O)Cc12
COC(=O)c1ccc(cc1)C(=O)N1CCC2(C1)CCC(=O)NC2=O
O=C(N1CCC2(C1)CCC(=O)NC2=O)c1ccc2scnc2c1
[O-][N+](=O)c1ccc(nc1)N1CCC2(C1)CCC(=O)NC2=O
CC(C(=O)N1CCC2(C1)CCC(=O)NC2=O)c1cccnc1
COC(=O)c1cccc(n1)N1CCC2(C1)CCC(=O)NC2=O
[O-][N+](=O)c1ccc2[nH]c(nc2c1)N1CCC2(C1)CCC(=O)NC2=O
[O-][N+](=O)c1ccc2[nH]c(nc2c1)N1CCC2(C1)CCC(=O)NC2=O
CC(=O)N1CCc2c1cccc2C(=O)N1CCC2(C1)CCC(=O)NC2=O
O=C(N1CCC2(C1)CCC(=O)NC2=O)c1ccccc1
CC(=O)Nc1cccc(c1)C(=O)N1CCC2(C1)CCC(=O)NC2=O
O=C(N1CCC2(C1)CCC(=O)NC2=O)c1cccc2[nH]ncc12
Nc1ccc(nc1)N1CCC2(C1)CCC(=O)NC2=O
O=C(N1CCC2(C1)CCC(=O)NC2=O)c1cccc2NCCc12
O=C(N1CCC2(C1)CCC(=O)NC2=O)c1ccc2CCNc2c1
CC(=O)N1CCc2ccc(cc12)C(=O)N1CCC2(C1)CCC(=O)NC2=O
CC(=O)Nc1ccc(nc1)N1CCC2(C1)CCC(=O)NC2=O
O=C(N1CCC2(C1)CCC(=O)NC2=O)c1coc2ccccc12
O=C(N1CCC2(C1)CCC(=O)NC2=O)c1cnn2ccccc12
O=C(N1CCC2(C1)CCC(=O)NC2=O)c1ccc2ncoc2c1
O=C(N1CCC2(C1)CCC(=O)NC2=O)c1ccc2NCCc2c1
O=C([C@@H]1CCCc2ccccc12)N1CCC2(C1)CCC(=O)NC2=O |r|
O=C([C@H]1CCCc2ccccc12)N1CCC2(C1)CCC(=O)NC2=O |r|
CC(=O)Nc1nc2cc(ccc2s1)C(=O)N1CCC2(C1)CCC(=O)NC2=O
CC(=O)Nc1nc2ccc(cc2s1)C(=O)N1CCC2(C1)CCC(=O)NC2=O
CC(=O)N1CCc2cc(ccc12)C(=O)N1CCC2(C1)CCC(=O)NC2=O
CC(C)(C)OC(=O)Nc1nc2cc(ccc2s1)C(=O)N1CCC2(C1)CCC(=O)NC2=O
CC(C)(C)OC(=O)Nc1nc2ccc(cc2s1)C(=O)N1CCC2(C1)CCC(=O)NC2=O
Nc1nc2ccc(cc2s1)C(=O)N1CCC2(C1)CCC(=O)NC2=O
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)NCCCCCCCC(=O)Nc1cccc(c1)C(=O)N1CCC3(C1)CCC(=O)NC3=O)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
O=C([C@H]1CCCc2ccccc12)N1CCC2(CC1)NC(=O)NC2=O |r|
O=C([C@@H]1CCCc2ccccc12)N1CCC2(CC1)NC(=O)NC2=O |r|
O=C(N1CCC2(CC1)NC(=O)NC2=O)c1ccccc1
O=C1NC(=O)C2(CCN(CC2)c2nc3ccccc3s2)N1
O=C1NC(=O)C2(CCN(CC2)c2nc3ncccc3s2)N1
COC(=O)c1ccc(nc1)N1CCC2(CC1)NC(=O)NC2=O
CC(=O)Nc1ccc(cc1)C(=O)N1CCC2(CC1)NC(=O)NC2=O
CC(=O)Nc1cccc(c1)C(=O)N1CCC2(CC1)NC(=O)NC2=O
O=C(N1CCC2(CC1)NC(=O)NC2=O)c1coc2ccccc12
O=C(N1CCC2(CC1)NC(=O)NC2=O)c1cnn2ccccc12
O=C1CC2(CCN(CC2)c2nc3ncccc3s2)C(=O)N1
[O-][N+](=O)c1ccc(nc1)N1CCC2(CC1)NC(=O)NC2=O
[O-][N+](=O)c1ccc(nc1)N1CCC2(CC(=O)NC2=O)CC1
O=C1CC2(CCN(CC2)c2nc3ccccc3s2)C(=O)N1
[O-][N+](=O)c1ccc(cc1)N1CCC2(CC1)NC(=O)NC2=O
[O-][N+](=O)c1ccc(cc1)N1CCC2(CC(=O)NC2=O)CC1
COC(=O)c1ccc(nc1)N1CCC2(CC(=O)NC2=O)CC1
O=C(N1CCC2(CC(=O)NC2=O)CC1)c1ccccc1
O=C(N1CCC2(CC(=O)NC2=O)CC1)c1ccc2scnc2c1
O=C([C@H]1CCCc2ccccc12)N1CCC2(CC(=O)NC2=O)CC1 |r|
O=C([C@@H]1CCCc2ccccc12)N1CCC2(CC(=O)NC2=O)CC1 |r|
O=C(N1CCC2(CC(=O)NC2=O)CC1)c1cnn2ccccc12
O=C(N1CCC2(CC(=O)NC2=O)CC1)c1coc2ccccc12
O=C(N1CCC2(CC1)NC(=O)NC2=O)c1ccc2scnc2c1
O=C1CCC(C(=O)N1)n1c2ccccc2oc1=O
Cn1c2ccccc2n(C2CCC(=O)NC2=O)c1=O
O=C1Cc2ccccc2N1C1CCC(=O)NC1=O
O=C1CC(CN1C1CCC(=O)NC1=O)c1ccccc1
C[C@]1(CCC(=O)NC1=O)N2C(=O)c3ccc(cc3C2=O)C(=O)O
Oc1c2C(=O)N(C3CCC(=O)NC3=O)C(=O)c2ccc1-c1cn[nH]c1
C[C@]1(CCC(=O)NC1=O)N1C(=O)c2ccc(-c3cn[nH]c3)c(O)c2C1=O |r|
C[C@]1(CCC(=O)NC1=O)N1C(=O)c2ccc(cc2C1=O)-c1n[nH]c(=S)o1 |r|
Cc1ccc(NC(=O)OCc2cc3C(=O)N(Cc3c(Br)c2)C2CCC(=O)NC2=O)cc1Cl
Cc1ccc(NC(=O)OCc2cc3C(=O)N(Cc3c(c2)C#N)C2CCC(=O)NC2=O)cc1Cl
Cc1ccc(NC(=O)OCc2cc3C(=O)N(Cc3c(F)c2)C2CCC(=O)NC2=O)cc1Cl
Cc1ccc(NC(=O)OCc2cc3C(=O)N(Cc3c(Cl)c2)C2CCC(=O)NC2=O)cc1Cl
COc1cc(COC(=O)Nc2ccc(C)c(Cl)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
FC(F)Oc1cc(F)cc(NC(=O)OCc2cc3C(=O)N(Cc3c(F)c2)C2CCC(=O)NC2=O)c1
FC(F)Oc1cc(NC(=O)OCc2cc3C(=O)N(Cc3c(F)c2)C2CCC(=O)NC2=O)ccc1F
Fc1cc(COC(=O)Nc2ccc(nc2)-c2ccccc2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
CC(C)(C)c1ccc(NC(=O)OCc2cc3C(=O)N(Cc3c(F)c2)C2CCC(=O)NC2=O)cn1
CC(C)(C)c1ccc(NC(=O)OCc2cc3C(=O)N(Cc3c(F)c2)C2CCC(=O)NC2=O)cc1
Fc1cc(COC(=O)Nc2ccc(cc2)-c2ccccn2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
Fc1cc(NC(=O)OCc2cc3C(=O)N(Cc3c(F)c2)C2CCC(=O)NC2=O)cc(OC(F)(F)F)c1
CC1(CC1)c1ccc(NC(=O)OCc2cc3C(=O)N(Cc3c(F)c2)C2CCC(=O)NC2=O)cc1
Fc1cc(COC(=O)Nc2ccc(F)c(OC(F)(F)F)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
Fc1cc(COC(=O)Nc2cccc(OC(F)(F)F)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
CC1CCCCN1c1ccc(NC(=O)OCc2cc3C(=O)N(Cc3c(F)c2)C2CCC(=O)NC2=O)cn1
CC1(C)COc2cc(NC(=O)OCc3cc4C(=O)N(Cc4c(F)c3)C3CCC(=O)NC3=O)ccc12
Fc1cc(COC(=O)Nc2ccc(nc2)-c2ccccc2F)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
Cc1ccccc1-c1ccc(NC(=O)OCc2cc3C(=O)N(Cc3c(F)c2)C2CCC(=O)NC2=O)cn1
Cc1cc(NC(=O)OCc2cc3C(=O)N(Cc3c(F)c2)C2CCC(=O)NC2=O)cnc1-c1ccccc1
Fc1cc(COC(=O)Nc2cccc(OC3CC3)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
Fc1cc(COC(=O)Nc2ccc(cc2)C2CCC2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
C[C@@H]1CCCN1c1ccc(NC(=O)OCc2cc3C(=O)N(Cc3c(F)c2)C2CCC(=O)NC2=O)cn1 |r|
Fc1cc(COC(=O)Nc2cc(ccn2)-c2ccccc2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
CC(C)(C)c1cccc(NC(=O)OCc2cc3C(=O)N(Cc3c(F)c2)C2CCC(=O)NC2=O)c1
FC(F)Oc1cccc(NC(=O)OCc2cc3C(=O)N(Cc3c(F)c2)C2CCC(=O)NC2=O)c1
Cc1cc(Cl)cc(NC(=O)OCc2cc3C(=O)N(Cc3c(F)c2)C2CCC(=O)NC2=O)c1
Fc1cc(COC(=O)Nc2cc(Cl)cc(Cl)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
Fc1cc(COC(=O)Nc2ccc(c(F)c2)-c2ccccc2F)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
Fc1cc(COC(=O)Nc2cc(F)c(c(F)c2)-c2ccccc2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
Cc1cc(C)cc(NC(=O)OCc2cc3C(=O)N(Cc3c(F)c2)C2CCC(=O)NC2=O)c1
Fc1cc(COC(=O)Nc2ccc(F)c(Cl)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
Fc1cc(Cl)cc(NC(=O)OCc2cc3C(=O)N(Cc3c(F)c2)C2CCC(=O)NC2=O)c1
FC(F)Oc1cc(Cl)cc(NC(=O)OCc2cc3C(=O)N(Cc3c(F)c2)C2CCC(=O)NC2=O)c1
Cc1ccc(NC(=O)OCc2cc3C(=O)N(Cc3c(F)c2)C2CCC(=O)NC2=O)cc1OC(F)F
COc1cc(COC(=O)Nc2ccc(nc2)-c2ccccc2F)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2ccc3c(OCC3(C)C)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2ccc(nc2)N2CCCCC2C)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2ccc(F)c(OC(F)(F)F)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2ccc(cc2)C2(C)CC2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2cc(F)cc(OC(F)(F)F)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2ccc(cc2)-c2ccccn2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2ccc(cc2)C(C)(C)C)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2ccc(nc2)C(C)(C)C)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2ccc(nc2)-c2ccccc2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2ccc(F)c(OC(F)F)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2cc(F)cc(OC(F)F)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2ccc(C)c(OC(F)F)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2cc(Cl)cc(OC(F)F)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2cc(F)cc(Cl)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2ccc(F)c(Cl)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2cc(C)cc(C)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2cccc(OC(F)F)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2cccc(c2)C(C)(C)C)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2cccc(OC(F)(F)F)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2cc(ccn2)-c2ccccc2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2ccc(cc2)C2CCC2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2cccc(OC3CC3)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2cnc(c(C)c2)-c2ccccc2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2ccc(nc2)-c2ccccc2C)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
Fc1cc(COC(=O)Nc2cc(F)c(F)c(Cl)c2)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O
COc1cc(COC(=O)Nc2ccc(nc2)N2CCC[C@@H]2C)cc2C(=O)N(Cc12)C1CCC(=O)NC1=O |r|
COc1c2C(=O)N(Cc2ccc1COC(=O)Nc1ccc(C)c(Cl)c1)C1CCC(=O)NC1=O
Cc1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2F)cc1Cl
Cc1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2Cl)cc1Cl
Cc1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2C)cc1Cl
O=C1N(Cc2c1ccc1OC3(CCNCC3)COc21)[C@H]1CCC(=O)NC1=O
O=C1N(Cc2c1ccc1OC3(CNC3)COc21)C1CCC(=O)NC1=O
Fc1c2C(=O)N(Cc2cc2OC3(CCNCC3)COc12)[C@H]1CCC(=O)NC1=O
O=C1N(Cc2cc3OC4(CNC4)COc3cc12)[C@H]1CCC(=O)NC1=O
O=C1N(C2CCC(=O)NC2=O)C(=O)c2cc3OC4(CNC4)COc3cc12
O=C1N(Cc2c1ccc1O[C@H](COCc3ccccc3)COc21)[C@H]1CCC(=O)NC1=O |r|
OC[C@@H]1COc2c3CN([C@H]4CCC(=O)NC4=O)C(=O)c3ccc2O1 |r|
O=C1N(Cc2c1ccc1O[C@@H](COCc3ccccc3)COc21)[C@H]1CCC(=O)NC1=O |r|
OC[C@H]1COc2c3CN([C@H]4CCC(=O)NC4=O)C(=O)c3ccc2O1 |r|
O=C1N(Cc2c1ccc1N[C@@H](COCc3ccccc3)COc21)C1CCC(=O)NC1=O |r|
OC[C@H]1COc2ccc3C(=O)N(Cc3c2O1)[C@H]1CCC(=O)NC1=O |r|
OC[C@@H]1COc2ccc3C(=O)N(Cc3c2O1)[C@H]1CCC(=O)NC1=O |r|
OC[C@@H]1COc2ccc3C(=O)N(Cc3c2O1)C1CCC(=O)NC1=O |r|
O=C1N(Cc2c1ccc1OC[C@H](COCc3ccccc3)Oc21)C1CCC(=O)NC1=O |r|
O=C1N(Cc2c1ccc1OC[C@@H](COCc3ccccc3)Oc21)C1CCC(=O)NC1=O |r|
OC[C@H]1COc2cc3C(=O)N(Cc3cc2O1)[C@H]1CCC(=O)NC1=O |r|
O=C1N(Cc2cc3O[C@@H](COCc4ccccc4)COc3cc12)[C@H]1CCC(=O)NC1=O |r|
O=C1N(C2CCC(=O)NC2=O)C(=O)c2cc3O[C@@H](COCc4ccccc4)COc3cc12 |r|
Fc1c2C(=O)N(C3CCC(=O)NC3=O)C(=O)c2cc2O[C@@H](COCc3ccccc3)COc12 |r|
OCC1COc2cc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c3cc2O1
COc1cc(C)c(Cl)cc1NC(=O)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Cc1c(Cl)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1CN1CCOCC1
FC(F)(F)Oc1cccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
FC(F)(F)Oc1cc(CN2CCOCC2)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
FC(F)Oc1cccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
Cc1ncc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1Cl
Cc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc(C)n1
Cc1cc(C)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
Fc1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1Cl
Cc1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1Cl
FC(F)(F)Oc1cc(Cl)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
Fc1cc(Cl)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
Cc1c(Cl)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1CN1CC2CC1CO2 |THB:31:32:37.38:35|
COc1ccc(Cl)cc1NC(=O)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C(Nc1ccc(nc1)N1CCCCC1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Clc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc(OCC2CCNC2)c1
CC(OC(=O)Nc1ccc(C)c(Cl)c1)c1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C(Nc1ccc2CCOc2c1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
FC(F)Oc1cc(Cl)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
Clc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc(OC2CCNC2)c1
Cc1c(Cl)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1CN1CC2CCC(C1)O2 |TLB:31:32:39:35.36|
O=C(NCC1CC1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C(OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1)N1CCCCC1
Cc1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1OC(F)F
Cc1c(CN2CCOCC2)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1OC(F)F
O=C(OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1)N1CCCC1
CC(C)CCNC(=O)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C(NC1CCCCC1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C(NC1CCCC1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C(OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1)N1CCC(C1)Oc1ccccc1
FC(F)Oc1cc(F)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
FC(F)Oc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)ccc1F
CCOc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)ccc1C
Cc1c(CN2CCOCC2)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1OC(F)(F)F
O=C(NC1CCN(CC1)c1ccccn1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C(OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1)N1CCN(CC1)c1ccccc1
COc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)ccc1C
COc1cc(Cl)ccc1NC(=O)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C(Nc1ccc(cc1)C1CC1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
CN1CCC(COc2cc(Cl)cc(NC(=O)OCc3ccc4CN(C5CCC(=O)NC5=O)C(=O)c4c3)c2)C1
Cc1c(F)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1CN1CCOCC1
O=C(Nc1ccc(nc1)-c1ccccc1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
CC(C)(C)c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cn1
Cc1c(Cl)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1OC1CCNC1
CCc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc(Cl)c1C
CN1CCC(C1)Oc1cc(Cl)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
CC(C)(C)c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1
Cc1c(Cl)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1OCCN1CCOCC1
CCc1ncc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1C
O=C(Nc1ccc(cc1)-c1ccccn1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
COc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cnc1C
Cc1c(Cl)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1OCC1CCNC1
O=C(Nc1cnc2CCCc2c1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C(Nc1cnc2CCOCc2c1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
CCc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cnc1C
O=C(Nc1ccc2CCCc2c1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Fc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc(OC(F)(F)F)c1
CC1(CC1)c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1
FC(F)(F)Oc1ccnc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
O=C(Nc1ccc(nc1)N1CCCC1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Fc1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1OC(F)(F)F
CC1(COC1)c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1
CCc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)ccn1
O=C(Nc1cnc(nc1)N1CCCCC1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C(Nc1ccc(nc1)N1CC2CCC(C1)O2)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1 |TLB:6:9:16:12.13|
O=C(Nc1ccc2OCCc2c1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C(Nc1ccc2OCCCc2c1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
CN1CCC(C1)Oc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc(Cl)c1C
CC1CCN(C1)c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cn1
CN1CCC(COc2cc(NC(=O)OCc3ccc4CN(C5CCC(=O)NC5=O)C(=O)c4c3)cc(Cl)c2C)C1
CCc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc(C)n1
Fc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cnc1N1CCCCC1
FC1(F)CCCN(C1)c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cn1
CC1CCCN1c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cn1
O=C(Nc1ccc(nn1)N1CCCCC1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C(Nc1ccc(nc1)N1CCOCC1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
CC1CCCCN1c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cn1
FC1(F)CCN(CC1)c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cn1
FC1(F)Oc2ccc(NC(=O)OCc3ccc4CN(C5CCC(=O)NC5=O)C(=O)c4c3)cc2O1
O=C(Nc1ccc(nc1)C1CC1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C(Nc1ccc(cc1)C1COC1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
CN1CCN(CC1)c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cn1
CC1(C)COc2cc(NC(=O)OCc3ccc4CN(C5CCC(=O)NC5=O)C(=O)c4c3)ccc12
Fc1ccccc1-c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cn1
Fc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cnc1-c1ccccc1
Cc1ccccc1-c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cn1
COc1ccccc1-c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cn1
Cc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cnc1-c1ccccc1
CN(C)C1CN(C1)c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cn1
COc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cnc1-c1ccccc1
Cc1ncc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1OC(F)(F)F
O=C(Nc1ccc2CCCOc2c1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C(Nc1cccc(OC2CC2)c1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C(Nc1cnc(cn1)N1CCCCC1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
FC(F)Oc1cc(CN2CCOCC2)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
FC(F)Oc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc(OCCN2CCOCC2)c1
COc1ccccc1CNC(=O)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C(NCc1ccccc1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
CC(F)(F)c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1
FC(F)Oc1cc(CN2CC3CC2CO3)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1 |THB:7:8:13.14:11|
FC1(F)CC1c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1
CC(NC(=O)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1)c1ccccc1
CC1COc2cc(NC(=O)OCc3ccc4CN(C5CCC(=O)NC5=O)C(=O)c4c3)ccc12
O=C(Nc1ccc(cc1)C1CCC1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C(Nc1ccc(nc1)C1CCC1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
FC(F)(F)Oc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc(OCCN2CCOCC2)c1
O=C(Nc1ccc(nc1)N1CCC1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Cc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc(C)c1C#N
Cc1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1C#N
Clc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc(c1)C#N
Cc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc(c1)C#N
FC1(F)Cc2cc(NC(=O)OCc3ccc4CN(C5CCC(=O)NC5=O)C(=O)c4c3)ccc2O1
CC(C)(C)c1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)ccn1
FC1(CC1)c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1
Cc1c(F)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1Cl
Cc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc(F)c1C
Cc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc(n1)C(C)(C)C
Cc1cc(Cl)c(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1Cl
CC(C)(C)C12CC(C1)(C2)NC(=O)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
CC(OC(=O)Nc1cccc(OC(F)(F)F)c1)c1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Cc1cc(C)c(F)c(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
Cc1cc(C)c(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1Cl
Cc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc(C)c1F
FC(F)(F)Oc1ccc(Cl)c(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
O=C(NC12CC(C1)(C2)c1ccccc1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Cc1c(F)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1F
Cc1ccc(OC(F)(F)F)cc1NC(=O)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Cc1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1C
O=C(NC1COC(OC1)c1ccccc1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1 |(-2.93,1.33,;-2.93,-.21,;-4.26,-.98,;-5.6,-.21,;-6.93,-.98,;-8.27,-.21,;-8.27,1.33,;-6.93,2.1,;-5.6,1.33,;-9.6,2.1,;-9.6,3.64,;-10.93,4.41,;-12.27,3.64,;-12.27,2.1,;-10.93,1.33,;-1.6,-.98,;-.26,-.21,;1.07,-.98,;1.07,-2.52,;2.4,-3.29,;3.74,-2.52,;5.2,-2.99,;6.11,-1.75,;7.65,-1.75,;8.42,-.41,;9.96,-.41,;10.73,-1.75,;12.27,-1.75,;9.96,-3.08,;8.42,-3.08,;7.65,-4.41,;5.2,-.5,;5.68,.96,;3.74,-.98,;2.4,-.21,)|
CC(C)(C)c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)nc1
Fc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc(Cl)c1F
Cc1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1F
Fc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc(F)c1-c1ccccc1
Fc1cc(ccc1NC(=O)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1)-c1ccccn1
Fc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)ccc1-c1ccccc1
Cc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)ccc1-c1ccccc1
FC(F)(F)c1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)sn1
FC1(F)CC1Oc1cccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
Cc1cc(F)c(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1Cl
CC(C)(C)c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c(F)c1
O=C(Nc1ccc(cn1)-c1ccccc1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Cc1cc(Cl)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
Fc1ccc(OC(F)(F)F)cc1NC(=O)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Cc1cc(F)cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
CCc1nscc1NC(=O)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Fc1cc(OC(F)(F)F)ccc1NC(=O)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C(Nc1ccnc(c1)-c1ccccc1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
CN1CCOCC1Cc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc(Cl)c1C
CCc1cc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)sn1
CC1(CC1)c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cn1
CC(C)(C)c1cccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)c1
FC(F)(F)Oc1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cc1
O=C(Nc1cc(ccn1)-c1ccccc1)OCc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
C[C@H]1CCCN1c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cn1 |r|
C[C@@H]1CCCN1c1ccc(NC(=O)OCc2ccc3CN(C4CCC(=O)NC4=O)C(=O)c3c2)cn1 |r|
C[C@@H](NC(=O)c1nc(no1)C(C)(C)C)c1ccc(cc1C)-c1cc(Nc2ccc(cn2)N2CCN(CCc3ccc(cc3)N3CCC(=O)NC3=O)C[C@@H]2C)ncn1 |r|
C[C@@H](NC(=O)c1nc(no1)C(C)(C)C)c1ccc(cc1C)-c1cc(Nc2ccc(cn2)N2CCN(CCc3ccc(cc3)N3CCC(=O)NC3=O)C[C@H]2C)ncn1 |r|
C[C@@H](NC(=O)c1nc(no1)C(C)(C)C)c1ccc(cc1C)-c1cc(Nc2ccc(cn2)N2CCN(CCc3ccc(cc3)N3CCC(=O)NC3=O)CC2)ncn1 |r|
C[C@@H](NC(=O)c1nc(no1)C(C)(C)C)c1ccc(cc1C)-c1cc(Nc2ccc(cn2)N2CCN(CCc3ccc(N4CCC(=O)NC4=O)c(F)c3)C[C@@H]2C)ncn1 |r|
C[C@@H](NC(=O)c1nc(no1)C(C)(C)C)c1ccc(cc1C)-c1cc(Nc2ccc(cn2)N2CCN(CCc3ccc(N4CCC(=O)NC4=O)c(F)c3)C[C@H]2C)ncn1 |r|
CC[C@H]1CN(CCc2ccc(cc2)N2CCC(=O)NC2=O)CCN1c1ccc(Nc2cc(ncn2)-c2ccc([C@@H](C)NC(=O)c3nc(no3)C(C)(C)C)c(C)c2)nc1 |r|
CC[C@H]1CN(CCc2ccc(N3CCC(=O)NC3=O)c(F)c2)CCN1c1ccc(Nc2cc(ncn2)-c2ccc([C@@H](C)NC(=O)c3nc(no3)C(C)(C)C)c(C)c2)nc1 |r|
CC[C@@H]1CN(CCc2ccc(cc2)N2CCC(=O)NC2=O)CCN1c1ccc(Nc2cc(ncn2)-c2ccc([C@@H](C)NC(=O)c3nc(no3)C(C)(C)C)c(C)c2)nc1 |r|
C[C@@H](NC(=O)c1nc(no1)C(C)(C)C)c1ccc(cc1C)-c1cc(Nc2ccc(cn2)N2CCN(CCc3ccc(cc3)N3CCC(=O)NC3=O)CC2(C)C)ncn1 |r|
C[C@@H](NC(=O)c1nc(no1)C(C)(C)C)c1ccc(c(F)c1C)-c1cc(Nc2ccc(cn2)N2CCN(CCc3ccc(cc3)N3CCC(=O)NC3=O)C[C@@H]2C)ncn1 |r|
C[C@@H](NC(=O)c1nc(no1)C(C)(C)C)c1ccc(c(F)c1C)-c1cc(Nc2ccc(cn2)N2CCN(CCc3ccc(cc3)N3CCC(=O)NC3=O)CC2)ncn1 |r|
C[C@@H](NC(=O)c1nc(no1)C(C)(C)C)c1cc(F)c(cc1C)-c1cc(Nc2ccc(cn2)N2CCN(CCc3ccc(cc3)N3CCC(=O)NC3=O)CC2)ncn1 |r|
CC(C)[C@H]1CN(CCc2ccc(cc2)N2CCC(=O)NC2=O)CCN1c1ccc(Nc2cc(ncn2)-c2ccc([C@@H](C)NC(=O)c3nc(no3)C(C)(C)C)c(C)c2)nc1 |r|
C[C@@H](NC(=O)c1nc(no1)C(C)(C)C)c1ccc(cc1Cl)-c1cc(Nc2ccc(cn2)N2CCN(CCc3ccc(cc3)N3CCC(=O)NC3=O)C[C@@H]2C)ncn1 |r|
COC[C@H]1CN(CCc2ccc(cc2)N2CCC(=O)NC2=O)CCN1c1ccc(Nc2cc(ncn2)-c2ccc([C@@H](C)NC(=O)c3nc(no3)C(C)(C)C)c(C)c2)nc1 |r|
C[C@@H](NC(=O)c1nc(no1)C(C)(C)C)c1ccc(cc1C(F)(F)F)-c1cc(Nc2ccc(cn2)N2CCN(CCc3ccc(cc3)N3CCC(=O)NC3=O)C[C@@H]2C)ncn1 |r|
C[C@@H](NC(=O)c1nc(no1)C(C)(C)C)c1ccc(cc1F)-c1cc(Nc2ccc(cn2)N2CCN(CCc3ccc(cc3)N3CCC(=O)NC3=O)C[C@@H]2C)ncn1 |r|
C[C@@H](NC(=O)c1nc(no1)C(C)(C)C)c1ccc(cc1C)-c1cc(Nc2ccc(cc2)N2CCN(CCc3ccc(cc3)N3CCC(=O)NC3=O)C[C@@H]2C)ncn1 |r|
C[C@@H](NC(=O)c1nc(no1)C(C)(C)C)c1ccc(cc1C)-c1cc(Nc2ccc(CCN3CCN(CC3)c3ccc(cc3)N3CCC(=O)NC3=O)cn2)ncn1 |r|
FC(F)(F)Oc1ccccc1S(=O)(=O)Nc1ccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c2c1
FC(F)(F)Oc1cccc(c1)S(=O)(=O)Nc1ccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c2c1
Cc1c(Cl)cccc1S(=O)(=O)Nc1ccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c2c1
Cc1ccc(cc1Cl)S(=O)(=O)Nc1ccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c2c1
O=C1N(C2CCC(=O)NC2=O)C(=O)c2cc(NS(=O)(=O)c3ccccc3)ccc12
O=C1CCC(N2C(=O)c3cccc4cccc(C2=O)c34)C(=O)N1
Oc1cc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c3cccc(c1)c23
Nc1cc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c3cccc(c1)c23
FC(F)(F)Oc1cccc(c1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
FC(F)(F)Oc1ccccc1C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
Clc1ccc(C2CN(C2)[C@@H]2CCCC[C@@H]2Oc2ccc3C(=O)N(Cc3c2)C2CCC(=O)NC2=O)c(c1)C#N |r|
Clc1ccc(C2CN(C2)[C@H]2CCCC[C@@H]2Oc2ccc3C(=O)N(Cc3c2)C2CCC(=O)NC2=O)c(c1)C#N |r|
Clc1ccc(C2CN(C2)[C@H]2CCCC[C@H]2Oc2ccc3C(=O)N(Cc3c2)C2CCC(=O)NC2=O)c(c1)C#N |r|
Clc1c2CN(C3CCC(=O)NC3=O)C(=O)c2ccc1O[C@H]1CCCC[C@@H]1N1CC(C1)c1ccccc1 |r|
Fc1ccc(C2CN(C2)[C@@H]2CCCC[C@H]2Oc2ccc3C(=O)N(Cc3c2)C2CCC(=O)NC2=O)c(c1)C#N |r|
Fc1ccc(C2CN(C2)[C@H]2CCCC[C@@H]2Oc2ccc3C(=O)N(Cc3c2)C2CCC(=O)NC2=O)c(c1)C#N |r|
Fc1ccc(C2CN(C2)[C@H]2CCCC[C@H]2Oc2ccc3C(=O)N(Cc3c2)C2CCC(=O)NC2=O)c(c1)C#N |r|
Clc1cc(ccc1C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O)C#N |r|
Clc1cc(ccc1C1CN(C1)[C@H]1CCCC[C@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O)C#N |r|
Fc1ccc(cc1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
Fc1cc2C(=O)N(Cc2cc1O[C@H]1CCCC[C@@H]1N1CC(C1)c1ccccc1)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@@H]3CCCC[C@H]3N3CCC3c3ccccc3)ccc12)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@H]3CCCC[C@@H]3N3CCC3c3ccccc3)ccc12)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@H]3CCCC[C@H]3N3CCC3c3ccccc3)ccc12)C1CCC(=O)NC1=O |r|
Fc1ccc(C2CN(C2)[C@H]2CCCC[C@@H]2Oc2ccc3C(=O)N(Cc3c2)C2CCC(=O)NC2=O)c(F)c1 |r|
FC(F)(F)c1ccc(cc1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
FC(F)(F)c1ccc(cc1)C1CN(C1)[C@H]1CCCC[C@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
FC(F)(F)Oc1ccc(cc1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
FC(F)(F)Oc1ccc(cc1)C1CN(C1)[C@H]1CCCC[C@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
FC(F)(F)Oc1ccc(cc1)C1CN(C1)[C@@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
Fc1cccc(C2CN(C2)[C@H]2CCCC[C@@H]2Oc2ccc3C(=O)N(Cc3c2)C2CCC(=O)NC2=O)c1F |r|
Fc1c2CN(C3CCC(=O)NC3=O)C(=O)c2ccc1O[C@H]1CCCC[C@@H]1N1CC(C1)c1ccccc1 |r|
FC(F)(F)Oc1cccc(c1)C1CN(C1)C1CCCCC1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O
FC(F)(F)Oc1ccccc1C1CN(C1)C1CCCCC1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O
FC(F)(F)c1ccccc1C1CN(C1)C1CCCCC1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O
Fc1ccc(C2CN(C2)[C@@H]2CCC[C@@H]2Oc2ccc3C(=O)N(Cc3c2)C23CC(C2)C(=O)NC3=O)c(c1)C#N |r,wD:13.15,9.9,(-7.27,-6.88,;-6.95,-5.38,;-5.48,-4.9,;-5.16,-3.4,;-6.31,-2.37,;-5.99,-.86,;-6.82,.43,;-5.53,1.27,;-4.69,-.02,;-5.21,2.78,;-6.24,3.92,;-5.47,5.26,;-3.97,4.94,;-3.81,3.4,;-2.47,2.63,;-1.14,3.4,;-1.14,4.94,;.2,5.71,;1.53,4.94,;2.99,5.42,;3.47,6.88,;3.9,4.17,;2.99,2.93,;1.53,3.4,;.2,2.63,;5.44,4.17,;6.21,5.51,;7.75,5.51,;6.93,4.57,;8.52,4.17,;10.06,4.17,;7.75,2.84,;6.21,2.84,;5.44,1.51,;-7.77,-2.84,;-8.09,-4.35,;-8.91,-1.81,;-10.06,-.78,)|
Fc1ccc(C2CN(C2)[C@@H]2CCC[C@H]2Oc2ccc3C(=O)N(Cc3c2)C23CC(C2)C(=O)NC3=O)c(c1)C#N |r,wU:13.15,wD:9.9,(-7.27,-6.88,;-6.95,-5.38,;-5.48,-4.9,;-5.16,-3.4,;-6.31,-2.37,;-5.99,-.86,;-6.82,.43,;-5.53,1.27,;-4.69,-.02,;-5.21,2.78,;-6.24,3.92,;-5.47,5.26,;-3.97,4.94,;-3.81,3.4,;-2.47,2.63,;-1.14,3.4,;-1.14,4.94,;.2,5.71,;1.53,4.94,;2.99,5.42,;3.47,6.88,;3.9,4.17,;2.99,2.93,;1.53,3.4,;.2,2.63,;5.44,4.17,;6.21,5.51,;7.75,5.51,;6.93,4.57,;8.52,4.17,;10.06,4.17,;7.75,2.84,;6.21,2.84,;5.44,1.51,;-7.77,-2.84,;-8.09,-4.35,;-8.91,-1.81,;-10.06,-.78,)|
O=C1N(Cc2cc(O[C@H]3CCC[C@@H]3N3CCC(CC3)c3ccccc3)ccc12)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@H]3CCC[C@@H]3N3CC(C3)c3ccc(cc3)-n3cccn3)ccc12)C1CCC(=O)NC1=O |r|
Clc1cc(ccc1C1CN(C1)[C@@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O)C#N |r|
O=C1N(Cc2cc(O[C@@H]3CCCC[C@@H]3N3CC(C3)c3cccc(c3)C#N)ccc12)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@@H]3CCCC[C@@H]3N3CC(C3)c3cccc(c3)C#N)ccc12)C12CC(C1)C(=O)NC2=O |r,wU:8.7,13.14,(1.68,6.68,;1.2,5.21,;2.11,3.97,;1.2,2.72,;-.26,3.2,;-1.6,2.43,;-2.93,3.2,;-4.26,2.43,;-5.6,3.2,;-5.6,4.74,;-6.93,5.51,;-8.27,4.74,;-8.27,3.2,;-6.93,2.43,;-6.93,.89,;-8.02,-.2,;-6.93,-1.29,;-5.84,-.2,;-6.93,-2.83,;-8.27,-3.6,;-8.27,-5.14,;-6.93,-5.91,;-5.6,-5.14,;-5.6,-3.6,;-4.26,-5.91,;-2.93,-6.68,;-2.93,4.74,;-1.6,5.51,;-.26,4.74,;3.65,3.97,;4.42,5.3,;5.96,5.3,;5.13,4.37,;6.73,3.97,;8.27,3.97,;5.96,2.63,;4.42,2.63,;3.65,1.3,)|
O=C1N(Cc2cc(O[C@H]3CCCC[C@@H]3N3CC(C3)c3cccc(c3)C#N)ccc12)C12CC(C1)C(=O)NC2=O |r,wU:13.14,wD:8.7,(1.68,6.68,;1.2,5.21,;2.11,3.97,;1.2,2.72,;-.26,3.2,;-1.6,2.43,;-2.93,3.2,;-4.26,2.43,;-5.6,3.2,;-5.6,4.74,;-6.93,5.51,;-8.27,4.74,;-8.27,3.2,;-6.93,2.43,;-6.93,.89,;-8.02,-.2,;-6.93,-1.29,;-5.84,-.2,;-6.93,-2.83,;-8.27,-3.6,;-8.27,-5.14,;-6.93,-5.91,;-5.6,-5.14,;-5.6,-3.6,;-4.26,-5.91,;-2.93,-6.68,;-2.93,4.74,;-1.6,5.51,;-.26,4.74,;3.65,3.97,;4.42,5.3,;5.96,5.3,;5.13,4.37,;6.73,3.97,;8.27,3.97,;5.96,2.63,;4.42,2.63,;3.65,1.3,)|
O=C1N(Cc2cc(O[C@H]3CCCC[C@@H]3N3CCC(CC3)c3ccccc3)ccc12)C1CCC(=O)NC1=O |r|
FC(F)Oc1cccc(c1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1F)C1CCC(=O)NC1=O |r|
FC(F)Oc1ccc(cc1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1F)C1CCC(=O)NC1=O |r|
Clc1ccccc1C1CN(C1)[C@H]1CCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C12CC(C1)C(=O)NC2=O |r,wU:11.12,wD:15.18,(-9.49,-2.56,;-8.34,-3.59,;-8.66,-5.1,;-7.52,-6.13,;-6.05,-5.66,;-5.73,-4.15,;-6.88,-3.12,;-6.56,-1.61,;-7.4,-.32,;-6.1,.52,;-5.27,-.77,;-5.78,2.02,;-6.82,3.17,;-6.05,4.5,;-4.54,4.18,;-4.38,2.65,;-3.04,1.88,;-1.71,2.65,;-1.71,4.19,;-.38,4.96,;.96,4.19,;2.42,4.67,;2.9,6.13,;3.33,3.42,;2.42,2.17,;.96,2.65,;-.38,1.88,;4.87,3.42,;5.64,4.75,;7.18,4.75,;6.41,3.42,;7.95,3.42,;9.49,3.42,;7.18,2.09,;5.64,2.09,;4.87,.75,)|
Clc1ccc(C2CN(C2)[C@H]2CCC[C@@H]2Oc2ccc3C(=O)N(Cc3c2)C2CCC(=O)NC2=O)c(c1)C#N |r|
Clc1ccc(C2CN(C2)[C@H]2CCC[C@H]2Oc2ccc3C(=O)N(Cc3c2)C2CCC(=O)NC2=O)c(c1)C#N |r|
Fc1ccc(C2CN(C2)[C@H]2CCCC[C@@H]2Oc2ccc3C(=O)N(Cc3c2)C23CC(C2)C(=O)NC3=O)c(Cl)c1 |r,wU:9.9,wD:14.16,(-6.27,-7.06,;-6.27,-5.52,;-4.93,-4.75,;-4.93,-3.21,;-6.27,-2.44,;-6.27,-.9,;-7.35,.18,;-6.27,1.27,;-5.18,.18,;-6.27,2.81,;-7.6,3.58,;-7.6,5.12,;-6.27,5.89,;-4.93,5.12,;-4.93,3.58,;-3.6,2.81,;-2.26,3.58,;-2.26,5.12,;-.93,5.89,;.4,5.12,;1.87,5.6,;2.34,7.06,;2.77,4.35,;1.87,3.11,;.4,3.58,;-.93,2.81,;4.31,4.35,;5.08,5.69,;6.62,5.69,;5.8,4.75,;7.39,4.35,;8.93,4.35,;6.62,3.02,;5.08,3.02,;4.31,1.69,;-7.6,-3.21,;-8.93,-2.44,;-7.6,-4.75,)|
Fc1ccc(C2CN(C2)[C@H]2CCC[C@@H]2Oc2ccc3C(=O)N(Cc3c2)C23CC(C2)C(=O)NC3=O)c(Cl)c1 |r,wU:9.9,wD:13.15,(-7.84,-6.88,;-7.52,-5.38,;-6.05,-4.9,;-5.73,-3.4,;-6.88,-2.37,;-6.56,-.86,;-7.4,.43,;-6.1,1.27,;-5.27,-.02,;-5.78,2.78,;-6.82,3.92,;-6.05,5.26,;-4.54,4.94,;-4.38,3.4,;-3.04,2.63,;-1.71,3.4,;-1.71,4.94,;-.38,5.71,;.96,4.94,;2.42,5.42,;2.9,6.88,;3.33,4.17,;2.42,2.93,;.96,3.4,;-.38,2.63,;4.87,4.17,;5.64,5.51,;7.18,5.51,;6.41,4.17,;7.95,4.17,;9.49,4.17,;7.18,2.84,;5.64,2.84,;4.87,1.51,;-8.34,-2.84,;-9.49,-1.81,;-8.66,-4.35,)|
Fc1cccc(c1)C1CN(C1)[C@H]1CCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C12CC(C1)C(=O)NC2=O |r,wU:11.12,wD:15.18,(-9.81,-5.58,;-8.34,-5.1,;-7.2,-6.13,;-5.73,-5.66,;-5.41,-4.15,;-6.56,-3.12,;-8.02,-3.59,;-6.24,-1.61,;-7.08,-.32,;-5.78,.52,;-4.95,-.77,;-5.46,2.02,;-6.49,3.17,;-5.72,4.5,;-4.22,4.18,;-4.06,2.65,;-2.72,1.88,;-1.39,2.65,;-1.39,4.19,;-.06,4.96,;1.28,4.19,;2.74,4.67,;3.22,6.13,;3.65,3.42,;2.74,2.17,;1.28,2.65,;-.06,1.88,;5.19,3.42,;5.96,4.75,;7.5,4.75,;6.73,3.42,;8.27,3.42,;9.81,3.42,;7.5,2.09,;5.96,2.09,;5.19,.75,)|
Fc1cccc(c1)C1CN(C1)[C@H]1CCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
Fc1cccc(c1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C12CC(C1)C(=O)NC2=O |r,wU:11.12,wD:16.19,(-4.26,-6.29,;-5.6,-5.52,;-6.93,-6.29,;-8.27,-5.52,;-8.27,-3.98,;-6.93,-3.21,;-5.6,-3.98,;-6.93,-1.67,;-8.02,-.59,;-6.93,.5,;-5.84,-.59,;-6.93,2.04,;-8.27,2.81,;-8.27,4.35,;-6.93,5.12,;-5.6,4.35,;-5.6,2.81,;-4.26,2.04,;-2.93,2.81,;-2.93,4.35,;-1.6,5.12,;-.26,4.35,;1.2,4.83,;1.68,6.29,;2.11,3.58,;1.2,2.34,;-.26,2.81,;-1.6,2.04,;3.65,3.58,;4.42,4.92,;5.96,4.92,;5.13,3.98,;6.73,3.58,;8.27,3.58,;5.96,2.25,;4.42,2.25,;3.65,.92,)|
Fc1cc(ccc1C1CN(C1)[C@H]1CCCC[C@H]1Oc1ccc2C(=O)N(Cc2c1)C12CC(C1)C(=O)NC2=O)C#N |r,wU:11.12,16.19,(-8.93,-1.67,;-7.6,-2.44,;-7.6,-3.98,;-6.27,-4.75,;-4.93,-3.98,;-4.93,-2.44,;-6.27,-1.67,;-6.27,-.13,;-7.35,.95,;-6.27,2.04,;-5.18,.95,;-6.27,3.58,;-7.6,4.35,;-7.6,5.89,;-6.27,6.66,;-4.93,5.89,;-4.93,4.35,;-3.6,3.58,;-2.26,4.35,;-2.26,5.89,;-.93,6.66,;.4,5.89,;1.87,6.37,;2.34,7.83,;2.77,5.12,;1.87,3.88,;.4,4.35,;-.93,3.58,;4.31,5.12,;5.08,6.46,;6.62,6.46,;5.8,5.52,;7.39,5.12,;8.93,5.12,;6.62,3.79,;5.08,3.79,;4.31,2.46,;-6.27,-6.29,;-6.27,-7.83,)|
Fc1cc(ccc1C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C12CC(C1)C(=O)NC2=O)C#N |r,wU:11.12,wD:16.19,(-8.93,-1.67,;-7.6,-2.44,;-7.6,-3.98,;-6.27,-4.75,;-4.93,-3.98,;-4.93,-2.44,;-6.27,-1.67,;-6.27,-.13,;-7.35,.95,;-6.27,2.04,;-5.18,.95,;-6.27,3.58,;-7.6,4.35,;-7.6,5.89,;-6.27,6.66,;-4.93,5.89,;-4.93,4.35,;-3.6,3.58,;-2.26,4.35,;-2.26,5.89,;-.93,6.66,;.4,5.89,;1.87,6.37,;2.34,7.83,;2.77,5.12,;1.87,3.88,;.4,4.35,;-.93,3.58,;4.31,5.12,;5.08,6.46,;6.62,6.46,;5.8,5.52,;7.39,5.12,;8.93,5.12,;6.62,3.79,;5.08,3.79,;4.31,2.46,;-6.27,-6.29,;-6.27,-7.83,)|
O=C1N(Cc2cc(O[C@@H]3CCCC[C@@H]3N3CC(C3)c3ccc(cc3)C#N)ccc12)C12CC(C1)C(=O)NC2=O |r,wU:13.14,8.7,(1.68,7.83,;1.2,6.37,;2.11,5.12,;1.2,3.88,;-.26,4.35,;-1.6,3.58,;-2.93,4.35,;-4.26,3.58,;-5.6,4.35,;-5.6,5.89,;-6.93,6.66,;-8.27,5.89,;-8.27,4.35,;-6.93,3.58,;-6.93,2.04,;-8.02,.95,;-6.93,-.13,;-5.84,.95,;-6.93,-1.67,;-8.27,-2.44,;-8.27,-3.98,;-6.93,-4.75,;-5.6,-3.98,;-5.6,-2.44,;-6.93,-6.29,;-6.93,-7.83,;-2.93,5.89,;-1.6,6.66,;-.26,5.89,;3.65,5.12,;4.42,6.46,;5.96,6.46,;5.13,5.52,;6.73,5.12,;8.27,5.12,;5.96,3.79,;4.42,3.79,;3.65,2.46,)|
O=C1N(Cc2cc(O[C@H]3CCCC[C@@H]3N3CC(C3)c3ccc(cc3)C#N)ccc12)C12CC(C1)C(=O)NC2=O |r,wU:13.14,wD:8.7,(1.68,7.83,;1.2,6.37,;2.11,5.12,;1.2,3.88,;-.26,4.35,;-1.6,3.58,;-2.93,4.35,;-4.26,3.58,;-5.6,4.35,;-5.6,5.89,;-6.93,6.66,;-8.27,5.89,;-8.27,4.35,;-6.93,3.58,;-6.93,2.04,;-8.02,.95,;-6.93,-.13,;-5.84,.95,;-6.93,-1.67,;-8.27,-2.44,;-8.27,-3.98,;-6.93,-4.75,;-5.6,-3.98,;-5.6,-2.44,;-6.93,-6.29,;-6.93,-7.83,;-2.93,5.89,;-1.6,6.66,;-.26,5.89,;3.65,5.12,;4.42,6.46,;5.96,6.46,;5.13,5.52,;6.73,5.12,;8.27,5.12,;5.96,3.79,;4.42,3.79,;3.65,2.46,)|
O=C1N(Cc2cc(O[C@@H]3CCCC[C@@H]3N3CC(C3)c3ccccc3C#N)ccc12)C12CC(C1)C(=O)NC2=O |r,wU:13.14,8.7,(3.01,6.29,;2.53,4.83,;3.44,3.58,;2.53,2.34,;1.07,2.81,;-.26,2.04,;-1.6,2.81,;-2.93,2.04,;-4.26,2.81,;-4.26,4.35,;-5.6,5.12,;-6.93,4.35,;-6.93,2.81,;-5.6,2.04,;-5.6,.5,;-6.69,-.59,;-5.6,-1.67,;-4.51,-.59,;-5.6,-3.21,;-4.26,-3.98,;-4.26,-5.52,;-5.6,-6.29,;-6.93,-5.52,;-6.93,-3.98,;-8.27,-3.21,;-9.6,-2.44,;-1.6,4.35,;-.26,5.12,;1.07,4.35,;4.98,3.58,;5.75,4.92,;7.29,4.92,;6.47,3.98,;8.06,3.58,;9.6,3.58,;7.29,2.25,;5.75,2.25,;4.98,.92,)|
O=C1N(Cc2cc(O[C@H]3CCCC[C@@H]3N3CC(C3)c3ccccc3C#N)ccc12)C12CC(C1)C(=O)NC2=O |r,wU:13.14,wD:8.7,(3.01,6.29,;2.53,4.83,;3.44,3.58,;2.53,2.34,;1.07,2.81,;-.26,2.04,;-1.6,2.81,;-2.93,2.04,;-4.26,2.81,;-4.26,4.35,;-5.6,5.12,;-6.93,4.35,;-6.93,2.81,;-5.6,2.04,;-5.6,.5,;-6.69,-.59,;-5.6,-1.67,;-4.51,-.59,;-5.6,-3.21,;-4.26,-3.98,;-4.26,-5.52,;-5.6,-6.29,;-6.93,-5.52,;-6.93,-3.98,;-8.27,-3.21,;-9.6,-2.44,;-1.6,4.35,;-.26,5.12,;1.07,4.35,;4.98,3.58,;5.75,4.92,;7.29,4.92,;6.47,3.98,;8.06,3.58,;9.6,3.58,;7.29,2.25,;5.75,2.25,;4.98,.92,)|
CC1(CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O)c1ccccc1 |r|
CC1(CN(C1)[C@@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O)c1ccccc1 |r|
O=C1N(Cc2cc(OC3CCCC3N3CC(C3)c3ccc(cc3)C#N)ccc12)C1CCC(=O)NC1=O
Fc1ccc(C2CN(C2)[C@H]2CCCC[C@@H]2Oc2ccc3C(=O)N(Cc3c2)C2CCC(=O)NC2=O)c(Cl)c1 |r|
Fc1ccc(C2CN(C2)[C@H]2CCC[C@@H]2Oc2ccc3C(=O)N(Cc3c2)C2CCC(=O)NC2=O)c(Cl)c1 |r|
O=C1N(Cc2cc(O[C@H]3CCC[C@@H]3N3CC(C3)c3ccccc3)ccc12)C12CC(C1)C(=O)NC2=O |r,wU:12.13,wD:8.7,(2.49,6.13,;2.01,4.67,;2.91,3.42,;2.01,2.17,;.54,2.65,;-.79,1.88,;-2.12,2.65,;-3.46,1.88,;-4.79,2.65,;-4.95,4.18,;-6.46,4.5,;-7.23,3.17,;-6.2,2.02,;-6.52,.52,;-7.81,-.32,;-6.97,-1.61,;-5.68,-.77,;-7.29,-3.12,;-8.75,-3.59,;-9.07,-5.1,;-7.93,-6.13,;-6.47,-5.66,;-6.15,-4.15,;-2.12,4.19,;-.79,4.96,;.54,4.19,;4.45,3.42,;5.22,4.75,;6.76,4.75,;5.99,3.42,;7.53,3.42,;9.07,3.42,;6.76,2.09,;5.22,2.09,;4.45,.75,)|
O=C1N(Cc2cc(O[C@H]3CCCC[C@@H]3N3CCC(C3)c3ccccc3)ccc12)C12CC(C1)C(=O)NC2=O |r,wU:13.14,wD:8.7,(1.68,6.03,;1.2,4.56,;2.11,3.32,;1.2,2.07,;-.26,2.55,;-1.6,1.78,;-2.93,2.55,;-4.26,1.78,;-5.6,2.55,;-5.6,4.09,;-6.93,4.86,;-8.27,4.09,;-8.27,2.55,;-6.93,1.78,;-6.93,.24,;-8.18,-.67,;-7.7,-2.13,;-6.16,-2.13,;-5.69,-.67,;-5.26,-3.38,;-5.88,-4.78,;-4.98,-6.03,;-3.45,-5.87,;-2.82,-4.46,;-3.73,-3.22,;-2.93,4.09,;-1.6,4.86,;-.26,4.09,;3.65,3.32,;4.42,4.65,;5.96,4.65,;5.13,3.72,;6.73,3.32,;8.27,3.32,;5.96,1.99,;4.42,1.99,;3.65,.65,)|
O=C1N(Cc2cc(O[C@H]3CCC[C@@H]3N3CCC(C3)c3ccccc3)ccc12)C12CC(C1)C(=O)NC2=O |r,wU:12.13,wD:8.7,(1.91,6.16,;1.43,4.69,;2.34,3.45,;1.43,2.2,;-.03,2.68,;-1.36,1.91,;-2.7,2.68,;-4.03,1.91,;-5.37,2.68,;-5.53,4.21,;-7.03,4.53,;-7.8,3.19,;-6.77,2.05,;-7.09,.54,;-8.5,-.08,;-8.34,-1.62,;-6.83,-1.94,;-6.06,-.6,;-6.21,-3.34,;-7.11,-4.59,;-6.48,-5.99,;-4.95,-6.16,;-4.05,-4.91,;-4.67,-3.5,;-2.7,4.22,;-1.36,4.99,;-.03,4.22,;3.88,3.45,;4.65,4.78,;6.19,4.78,;5.37,3.84,;6.96,3.45,;8.5,3.45,;6.19,2.11,;4.65,2.11,;3.88,.78,)|
O=C1N(Cc2cc(O[C@H]3CCCC[C@@H]3N3CC(C3)c3ccccc3C#N)ccc12)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@@H]3CCCC[C@@H]3N3CC(C3)c3ccccc3C#N)ccc12)C1CCC(=O)NC1=O |r|
Fc1cc(ccc1C#N)C1CN(C1)C1CCCC1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O
Fc1cccc(c1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@H]3CCCC[C@@H]3N3CC(C3)c3cccc(c3)N3CCOCC3)ccc12)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@H]3CCCC[C@@H]3N3CC(C3)c3cccc(c3)C#N)ccc12)C1CCC(=O)NC1=O |r|
Fc1cc(ccc1C1CN(C1)[C@@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O)C#N |r|
Fc1cc(ccc1C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O)C#N |r|
O=C1N(Cc2cc(OC3CCCCC3N3CC(C3)c3ccc(cc3)C#N)ccc12)C1CCC(=O)NC1=O
O=C1N(Cc2cc(OC3CCCCC3N3CC(C3)c3ccccc3)ccc12)C1CCC(=O)NC1=O
Fc1cc(ccc1C#N)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@H]3CCC[C@@H]3N3CC(C3)c3ccccc3)ccc12)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@H]3CCC[C@@H]3N3CCC(C3)c3ccccc3)ccc12)C1CCC(=O)NC1=O |r|
Fc1cc(ccc1C#N)C1CN(C1)[C@@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@H]3CCCC[C@@H]3N3CC(C3)c3ccc(cc3)N3CCOCC3)ccc12)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@H]3CCCC[C@@H]3N3CC(C3)c3ccccc3)ccc12)[C@@H]1CCC(=O)NC1=O |r|
COc1cccc(c1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@H]3CCCC[C@@H]3N3CC(C3)c3ccccc3)ccc12)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@H]3CCCC[C@H]3N3CC(C3)c3ccccc3)ccc12)C1CCC(=O)NC1=O |r|
FC(F)(F)c1ccccc1C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@H]3CCCCC[C@@H]3N3CC(C3)c3ccccc3)ccc12)C1CCC(=O)NC1=O |r|
Oc1ccc(cc1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
Oc1ccccc1C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
Oc1cccc(c1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@H]3CCCC[C@@H]3N3CC(C3)C3CCCCC3)ccc12)C1CCC(=O)NC1=O |r|
FC1(F)CCC(CC1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@H]3CCCC[C@@H]3N3CC(C3)C3CC3)ccc12)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@H]3CCCC[C@@H]3N3CC(C3)C3CCC3)ccc12)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@H]3CCCC[C@@H]3N3CC(C3)C3CCCC3)ccc12)C1CCC(=O)NC1=O |r|
CO[C@H]1CCC(CC1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r,wU:12.13,2.1,wD:17.20,(-8.27,-7.45,;-6.93,-6.68,;-6.93,-5.14,;-8.27,-4.37,;-8.27,-2.83,;-6.93,-2.06,;-5.6,-2.83,;-5.6,-4.37,;-6.93,-.52,;-8.02,.57,;-6.93,1.66,;-5.84,.57,;-6.93,3.2,;-8.27,3.97,;-8.27,5.51,;-6.93,6.28,;-5.6,5.51,;-5.6,3.97,;-4.26,3.2,;-2.93,3.97,;-2.93,5.51,;-1.6,6.28,;-.26,5.51,;1.2,5.98,;1.68,7.45,;2.11,4.74,;1.2,3.49,;-.26,3.97,;-1.6,3.2,;3.65,4.74,;4.42,6.07,;5.96,6.07,;6.73,4.74,;8.27,4.74,;5.96,3.4,;4.42,3.4,;3.65,2.07,)|
CO[C@H]1CCC(CC1)C1CN(C1)[C@H]1CCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r,wU:12.13,2.1,wD:16.19,(-7.11,-7.4,;-8.25,-6.37,;-7.93,-4.86,;-9.07,-3.83,;-8.75,-2.33,;-7.29,-1.85,;-6.15,-2.88,;-6.47,-4.39,;-6.97,-.34,;-7.81,.95,;-6.52,1.79,;-5.68,.49,;-6.2,3.29,;-7.23,4.44,;-6.46,5.77,;-4.95,5.45,;-4.79,3.92,;-3.46,3.15,;-2.12,3.92,;-2.12,5.46,;-.79,6.23,;.54,5.46,;2.01,5.94,;2.49,7.4,;2.91,4.69,;2.01,3.44,;.54,3.92,;-.79,3.15,;4.45,4.69,;5.22,6.02,;6.76,6.02,;7.53,4.69,;9.07,4.69,;6.76,3.36,;5.22,3.36,;4.45,2.02,)|
CO[C@H]1CCC(CC1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C12CC(C1)C(=O)NC2=O |r,wU:12.13,2.1,wD:17.20,(-8.27,-7.45,;-6.93,-6.68,;-6.93,-5.14,;-8.27,-4.37,;-8.27,-2.83,;-6.93,-2.06,;-5.6,-2.83,;-5.6,-4.37,;-6.93,-.52,;-8.02,.57,;-6.93,1.66,;-5.84,.57,;-6.93,3.2,;-8.27,3.97,;-8.27,5.51,;-6.93,6.28,;-5.6,5.51,;-5.6,3.97,;-4.26,3.2,;-2.93,3.97,;-2.93,5.51,;-1.6,6.28,;-.26,5.51,;1.2,5.98,;1.68,7.45,;2.11,4.74,;1.2,3.49,;-.26,3.97,;-1.6,3.2,;3.65,4.74,;4.42,6.07,;5.96,6.07,;5.19,4.74,;6.73,4.74,;8.27,4.74,;5.96,3.4,;4.42,3.4,;3.65,2.07,)|
CO[C@H]1CCC(CC1)C1CN(C1)[C@H]1CCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C12CC(C1)C(=O)NC2=O |r,wU:12.13,2.1,wD:16.19,(-7.11,-7.4,;-8.25,-6.37,;-7.93,-4.86,;-9.07,-3.83,;-8.75,-2.33,;-7.29,-1.85,;-6.15,-2.88,;-6.47,-4.39,;-6.97,-.34,;-7.81,.95,;-6.52,1.79,;-5.68,.49,;-6.2,3.29,;-7.23,4.44,;-6.46,5.77,;-4.95,5.45,;-4.79,3.92,;-3.46,3.15,;-2.12,3.92,;-2.12,5.46,;-.79,6.23,;.54,5.46,;2.01,5.94,;2.49,7.4,;2.91,4.69,;2.01,3.44,;.54,3.92,;-.79,3.15,;4.45,4.69,;5.22,6.02,;6.76,6.02,;5.99,4.69,;7.53,4.69,;9.07,4.69,;6.76,3.36,;5.22,3.36,;4.45,2.02,)|
FC1(F)CCC(CC1)C1CN(C1)[C@H]1CCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
FC1(F)CCC(CC1)C1CN(C1)[C@H]1CCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C12CC(C1)C(=O)NC2=O |r,wU:12.13,wD:16.19,(1.81,-4.16,;.32,-3.76,;.72,-5.25,;-1.14,-4.24,;-2.29,-3.21,;-1.97,-1.7,;-.5,-1.22,;.64,-2.25,;-3.11,-.67,;-4.65,-.75,;-4.73,.79,;-3.19,.87,;-5.87,1.82,;-7.38,1.5,;-8.15,2.83,;-7.12,3.98,;-5.71,3.35,;-4.38,4.12,;-3.05,3.35,;-3.05,1.81,;-1.71,1.04,;-.38,1.81,;1.09,1.33,;1.56,-.13,;1.99,2.58,;1.09,3.83,;-.38,3.35,;-1.71,4.12,;3.53,2.58,;4.3,1.25,;5.84,1.25,;5.02,2.18,;6.61,2.58,;8.15,2.58,;5.84,3.91,;4.3,3.91,;3.53,5.25,)|
FC1(F)CCC(CC1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C12CC(C1)C(=O)NC2=O |r,wU:12.13,wD:17.20,(-7.7,-6.96,;-6.93,-5.63,;-6.16,-6.96,;-8.27,-4.86,;-8.27,-3.32,;-6.93,-2.55,;-5.6,-3.32,;-5.6,-4.86,;-6.93,-1.01,;-8.02,.08,;-6.93,1.17,;-5.84,.08,;-6.93,2.71,;-8.27,3.48,;-8.27,5.02,;-6.93,5.79,;-5.6,5.02,;-5.6,3.48,;-4.26,2.71,;-2.93,3.48,;-2.93,5.02,;-1.6,5.79,;-.26,5.02,;1.2,5.5,;1.68,6.96,;2.11,4.25,;1.2,3,;-.26,3.48,;-1.6,2.71,;3.65,4.25,;4.42,5.58,;5.96,5.58,;5.13,4.65,;6.73,4.25,;8.27,4.25,;5.96,2.92,;4.42,2.92,;3.65,1.58,)|
CC(C)O[C@H]1CCC(CC1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r,wU:14.15,wD:19.22,4.3,(-5.6,-8.22,;-5.6,-6.68,;-4.26,-5.91,;-6.93,-5.91,;-6.93,-4.37,;-5.6,-3.6,;-5.6,-2.06,;-6.93,-1.29,;-8.27,-2.06,;-8.27,-3.6,;-6.93,.25,;-8.02,1.34,;-6.93,2.43,;-5.84,1.34,;-6.93,3.97,;-8.27,4.74,;-8.27,6.28,;-6.93,7.05,;-5.6,6.28,;-5.6,4.74,;-4.26,3.97,;-2.93,4.74,;-2.93,6.28,;-1.6,7.05,;-.26,6.28,;1.2,6.75,;1.68,8.22,;2.11,5.51,;1.2,4.26,;-.26,4.74,;-1.6,3.97,;3.65,5.51,;4.42,6.84,;5.96,6.84,;6.73,5.51,;8.27,5.51,;5.96,4.17,;4.42,4.17,;3.65,2.84,)|
FC1(F)CC(C1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
CCOC1CCC(CC1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r,wU:13.14,wD:18.21,(-5.6,-8.22,;-5.6,-6.68,;-6.93,-5.91,;-6.93,-4.37,;-8.27,-3.6,;-8.27,-2.06,;-6.93,-1.29,;-5.6,-2.06,;-5.6,-3.6,;-6.93,.25,;-8.02,1.34,;-6.93,2.43,;-5.84,1.34,;-6.93,3.97,;-8.27,4.74,;-8.27,6.28,;-6.93,7.05,;-5.6,6.28,;-5.6,4.74,;-4.26,3.97,;-2.93,4.74,;-2.93,6.28,;-1.6,7.05,;-.26,6.28,;1.2,6.75,;1.68,8.22,;2.11,5.51,;1.2,4.26,;-.26,4.74,;-1.6,3.97,;3.65,5.51,;4.42,6.84,;5.96,6.84,;6.73,5.51,;8.27,5.51,;5.96,4.17,;4.42,4.17,;3.65,2.84,)|
FC1(F)CCCC(C1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r|
FC(F)OC1CCC(CC1)C1CN(C1)[C@H]1CCCC[C@@H]1Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O |r,wU:14.15,wD:19.22,(-5.6,-8.22,;-5.6,-6.68,;-4.26,-5.91,;-6.93,-5.91,;-6.93,-4.37,;-8.27,-3.6,;-8.27,-2.06,;-6.93,-1.29,;-5.6,-2.06,;-5.6,-3.6,;-6.93,.25,;-8.02,1.34,;-6.93,2.43,;-5.84,1.34,;-6.93,3.97,;-8.27,4.74,;-8.27,6.28,;-6.93,7.05,;-5.6,6.28,;-5.6,4.74,;-4.26,3.97,;-2.93,4.74,;-2.93,6.28,;-1.6,7.05,;-.26,6.28,;1.2,6.75,;1.68,8.22,;2.11,5.51,;1.2,4.26,;-.26,4.74,;-1.6,3.97,;3.65,5.51,;4.42,6.84,;5.96,6.84,;6.73,5.51,;8.27,5.51,;5.96,4.17,;4.42,4.17,;3.65,2.84,)|
O=C1N(Cc2cc(O[C@H]3CCC[C@@H]3N3CC(C3)C3CC3)ccc12)C1CCC(=O)NC1=O |r|
O=C1N(Cc2cc(O[C@H]3CCCC[C@@H]3N3CC(C3)C3(CCC3)C#N)ccc12)C1CCC(=O)NC1=O |r|
Fc1c2CN(C3CCC(=O)NC3=O)C(=O)c2ccc1O[C@H]1CCCC[C@@H]1N1CC(C1)C1CC1 |r|
Fc1c2CN(C3CCC(=O)NC3=O)C(=O)c2ccc1O[C@H]1CCCC[C@@H]1N1CC(C1)C1CCC1 |r|
Fc1cc2C(=O)N(Cc2cc1O[C@H]1CCCC[C@@H]1N1CC(C1)C1CC1)C1CCC(=O)NC1=O |r|
Fc1cc2C(=O)N(Cc2cc1O[C@H]1CCCC[C@@H]1N1CC(C1)C1CCC1)C1CCC(=O)NC1=O |r|
COCCOCC1COCCN1Cc1ccc(COc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)cc1
COCCCCC1COCCN1Cc1ccc(COc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)cc1
COCCNC(=O)C1CCCN(Cc2ccc(COc3cccc4c3CN(C3CCC(=O)NC3=O)C4=O)cc2)C1
COCCCC(=O)C1CCN(Cc2ccc(COc3cccc4c3CN(C3CCC(=O)NC3=O)C4=O)cc2)CC1
COCCNC(=O)C1CCN(Cc2ccc(COc3cccc4c3CN(C3CCC(=O)CC3=O)C4=O)cc2)C1
COCCOCC1CCN(Cc2ccc(COc3cccc4c3CN(C3CCC(=O)NC3=O)C4=O)cc2)CC1
COCCOc1cc(OCc2ccc(CN3CCOCC3)cc2)c2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2
COCCCc1cc(COc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)ccc1CN1CCOCC1
COCCNc1cc(CN2CCOCC2)ccc1COc1cccc2c1CN(C1CCC(=O)NC1=O)C2=O
COCCCC(=O)c1cc(COc2cccc3c2CN([C@H]2CCC(=O)NC2=O)C3=O)ccc1CN1CCOCC1
O=C1N(C2CCC(=O)NC2=O)C(=O)c2ccccc12
Cc6cc(c5cc(Nc4ccc(N3CCN(CCc2ccc(N1CCC(=O)NC1=O)cc2)C[C@@H]3C)cn4)ncn5)ccc6[C@@H](C)NC(=O)c7nc(C(C)(C)C)no7
Cc6cc(c5cc(Nc4ccc(N3CCN(CCc2ccc(N1CCC(=O)NC1=O)cc2)C[C@H]3C)cn4)ncn5)ccc6[C@@H](C)NC(=O)c7nc(C(C)(C)C)no7
Cc6cc(c5cc(Nc4ccc(N3CCN(CCc2ccc(N1CCC(=O)NC1=O)cc2)CC3)cn4)ncn5)ccc6[C@@H](C)NC(=O)c7nc(C(C)(C)C)no7
Cc6cc(c5cc(Nc4ccc(N3CCN(CCc2ccc(N1CCC(=O)NC1=O)c(F)c2)C[C@@H]3C)cn4)ncn5)ccc6[C@@H](C)NC(=O)c7nc(C(C)(C)C)no7
Cc6cc(c5cc(Nc4ccc(N3CCN(CCc2ccc(N1CCC(=O)NC1=O)c(F)c2)C[C@H]3C)cn4)ncn5)ccc6[C@@H](C)NC(=O)c7nc(C(C)(C)C)no7
CC[C@H]3CN(CCc2ccc(N1CCC(=O)NC1=O)cc2)CCN3c7ccc(Nc6cc(c5ccc([C@@H](C)NC(=O)c4nc(C(C)(C)C)no4)c(C)c5)ncn6)nc7
CC[C@H]3CN(CCc2ccc(N1CCC(=O)NC1=O)c(F)c2)CCN3c7ccc(Nc6cc(c5ccc([C@@H](C)NC(=O)c4nc(C(C)(C)C)no4)c(C)c5)ncn6)nc7
CC[C@@H]3CN(CCc2ccc(N1CCC(=O)NC1=O)cc2)CCN3c7ccc(Nc6cc(c5ccc([C@@H](C)NC(=O)c4nc(C(C)(C)C)no4)c(C)c5)ncn6)nc7
Cc6cc(c5cc(Nc4ccc(N3CCN(CCc2ccc(N1CCC(=O)NC1=O)cc2)CC3(C)C)cn4)ncn5)ccc6[C@@H](C)NC(=O)c7nc(C(C)(C)C)no7
Cc6c(F)c(c5cc(Nc4ccc(N3CCN(CCc2ccc(N1CCC(=O)NC1=O)cc2)C[C@@H]3C)cn4)ncn5)ccc6[C@@H](C)NC(=O)c7nc(C(C)(C)C)no7
Cc6c(F)c(c5cc(Nc4ccc(N3CCN(CCc2ccc(N1CCC(=O)NC1=O)cc2)CC3)cn4)ncn5)ccc6[C@@H](C)NC(=O)c7nc(C(C)(C)C)no7
Cc6cc(c5cc(Nc4ccc(N3CCN(CCc2ccc(N1CCC(=O)NC1=O)cc2)CC3)cn4)ncn5)c(F)cc6[C@@H](C)NC(=O)c7nc(C(C)(C)C)no7
Cc6cc(c5cc(Nc4ccc(N3CCN(CCc2ccc(N1CCC(=O)NC1=O)cc2)C[C@@H]3C(C)C)cn4)ncn5)ccc6[C@@H](C)NC(=O)c7nc(C(C)(C)C)no7
C[C@H]3CN(CCc2ccc(N1CCC(=O)NC1=O)cc2)CCN3c7ccc(Nc6cc(c5ccc([C@@H](C)NC(=O)c4nc(C(C)(C)C)no4)c(Cl)c5)ncn6)nc7
COC[C@H]3CN(CCc2ccc(N1CCC(=O)NC1=O)cc2)CCN3c7ccc(Nc6cc(c5ccc([C@@H](C)NC(=O)c4nc(C(C)(C)C)no4)c(C)c5)ncn6)nc7
C[C@H]3CN(CCc2ccc(N1CCC(=O)NC1=O)cc2)CCN3c7ccc(Nc6cc(c5ccc([C@@H](C)NC(=O)c4nc(C(C)(C)C)no4)c(C(F)(F)F)c5)ncn6)nc7
C[C@H]3CN(CCc2ccc(N1CCC(=O)NC1=O)cc2)CCN3c7ccc(Nc6cc(c5ccc([C@@H](C)NC(=O)c4nc(C(C)(C)C)no4)c(F)c5)ncn6)nc7
Cc6cc(c5cc(Nc4ccc(N3CCN(CCc2ccc(N1CCC(=O)NC1=O)cc2)C[C@@H]3C)cc4)ncn5)ccc6[C@@H](C)NC(=O)c7nc(C(C)(C)C)no7
Cc6cc(c5cc(Nc4ccc(CCN3CCN(c2ccc(N1CCC(=O)NC1=O)cc2)CC3)cn4)ncn5)ccc6[C@@H](C)NC(=O)c7nc(C(C)(C)C)no7
Cc1nc2cccc(N)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(C#CCCCCCCN3CCN(C)CC3)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCCCCCCNC34CC5CC(CC(C5)C3)C4)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(SCCCN3CCN(CCC45CC6CC(CC(C6)C4)C5)CC3)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCCNC3C4CC5CC(C4)CC3C5)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(CCCCCNC34CC5CC(CC(C5)C3)C4)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCCCCCNC34CC5CC(CC3C5)C4)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(CCCCCCCCNC34CC5CC(CC(C5)C3)C4)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCCCCCCNC34CC5CC(CC3C5)C4)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(CCCCCCCCN3CCC(N4CCN(C)CC4)CC3)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCCCCCCN3CCCN(C)CC3)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(CCCCCCCCN3CC4CC(C3)O4)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCCCCCCO)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCOCCNC34CC5CC(CC(C5)C3)C4)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NC34CC5CC(CC(C5)C3)C4)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCOCCNC34CC5CC(CC3C5)C4)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCCCCCCN3CC4CC(C3)O4)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCN3CCN(CCC45CC6CC(CC(C6)C4)C5)CC3)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCCCCCCN3CCC(N4CCOCC4)CC3)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCCCCNC34CC5CC(CC3C5)C4)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCCCCCCN3CCN(C4COC4)CC3)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCCCNC3C4CC5CC(C4)CC3C5)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCCCCCCN[C@@]34CC5CC(C)(C[C@@](C)(C5)C3)C4)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCCCCNC3C4CC5CC(C4)CC3C5)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCCCCCCNC(C)C34CC5CC(CC(C5)C3)C4)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCCCCCCNC34CCC5(F)CCC53C4)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCCCCCCN3CCC4(CC3)CC(F)(F)C4)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(NCCCCCCCNC34CC5CC(CC3C5)C4)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(N3C4CC3CN(CCC35CC6CC(CC(C6)C3)C5)C4)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(SCCN3CCN(CCC45CC6CC(CC(C6)C4)C5)CC3)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(SCCN3CCN(Cc4ccc(C56CC7CC(CC(C7)C5)C6)cc4)CC3)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(CN3CCN(CCC45CC6CC(CC(C6)C4)C5)CC3)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(CN3CCN(C(=O)C45CC6CC(CC(C6)C4)C5)CC3)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(C#CCN3CCN(CCC45CC6CC(CC(C6)C4)C5)CC3)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(CCCN3CCN(CCCNC45CC6CC(CC(C6)C4)C5)CC3)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(CN3CCNCC3)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(SCCN3CCN(CC45CC6CC(CC(C6)C4)C5)CC3)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(SCCCN3CCN(CC45CC6CC(CC(C6)C4)C5)CC3)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(CN3CCN(Cc4ccc(C56CC7CC(CC(C7)C5)C6)cc4)CC3)c2c(=O)n1C1CCC(=O)NC1=O
Cc1nc2cccc(C#CCN3CCN(Cc4ccc(C56CC7CC(CC(C7)C5)C6)cc4)CC3)c2c(=O)n1C1CCC(=O)NC1=O
COc1cccc(C(=O)NCc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)c1
O=C1CCC(N2Cc3c(CNC(=O)c4cccc(Cl)c4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4ccccc4C(F)(F)F)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4ccc(Cl)cc4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4ccc(F)cc4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4cccc(F)c4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4cccc(C(F)(F)F)c4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4ccc(C(F)(F)F)cc4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4ccc(F)c(Cl)c4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4ccc(C(F)(F)F)c(F)c4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4ccc(F)cc4Cl)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4ccc(Br)cc4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4ccc(Cl)c(F)c4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4cccc(OC(F)(F)F)c4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4ccc(Cl)c(C(F)(F)F)c4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4ccc(F)c(C(F)(F)F)c4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4cccc(C(F)F)c4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4ccc(C(F)F)cc4)cccc3C2=O)C(=O)N1
COc1ccc(C(=O)NCc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)cc1
N#Cc1cccc(C(=O)NCc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)c1
O=C1CCC(N2Cc3c(CNC(=O)c4cccs4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4ccc(Cl)cc4Cl)cccc3C2=O)C(=O)N1
COc1ccccc1C(=O)NCc1cccc2c1CN(C1CCC(=O)NC1=O)C2=O
CCCc1ccc(C(=O)NCc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)cc1
O=C1CCC(N2Cc3c(CNC(=O)c4ccccc4F)cccc3C2=O)C(=O)N1
Cc1ccc(F)cc1C(=O)NCc1cccc2c1CN(C1CCC(=O)NC1=O)C2=O
O=C1CCC(N2Cc3c(CNC(=O)c4c(F)ccc(F)c4Cl)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4ccc(OC(F)(F)F)cc4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4cc(C(F)(F)F)cc(Cl)c4F)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4ccc(Cl)cc4F)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4cc(F)ccc4F)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4cccc5cc[nH]c45)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4cccc5[nH]ccc45)cccc3C2=O)C(=O)N1
O=C(Cc1ccc(O)cc1)NCc1cccc2c1CN(C1CCC(=O)NC1=O)C2=O
O=C(Cc1ccccc1Br)NCc1cccc2c1CN(C1CCC(=O)NC1=O)C2=O
O=C1CCC(N2Cc3c(CNC(=O)c4ccc5nc[nH]c5c4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4ccccc4Nc4cccc(C(F)(F)F)c4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4ccc(-c5ccc(Cl)cc5)o4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4ccccc4Nc4ccccc4)cccc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CNC(=O)c4ccccc4Cl)cccc3C2=O)C(=O)N1
CCC[C@H](C)Nc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O
COc1ccc([C@@H](C)Nc2cccc3c2CN(C2CCC(=O)NC2=O)C3)cc1
C[C@H](CO)Nc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O
O=C1CCC(N2C(=O)c3cc4c(cc3C2=O)OC2(CCNCC2)C(F)(F)C4)C(=O)N1
O=C1CCC(N2Cc3ccc4c(c3C2=O)CC2(CCNCC2)CO4)C(=O)N1
O=C1CCC(N2C(=O)c3cc4c(cc3C2=O)OC2(CC4)CNC2)C(=O)N1
O=C1CCC(N2C(=O)c3cc4c(cc3C2=O)OCC2(CCNCC2)C4)C(=O)N1
O=C1CCC(N2C(=O)c3cc4c(cc3C2=O)OC2(CCNCC2)CO4)C(=O)N1
O=C1CCC(N2C(=O)c3cc4c(cc3C2=O)OC2(CCNCC2)C4)C(=O)N1
O=C1CCC(N2C(=O)c3cc4c(cc3C2=O)CC2CNCC2C4)C(=O)N1
O=C1CCC2(CC1)CCc1cc3c(cc1O2)C(=O)N(C1CCC(=O)NC1=O)C3=O
O=C1CCC(N2C(=O)c3cc4c(cc3C2=O)C(F)(F)CC2(CCNCC2)O4)C(=O)N1
O=C1CCC(N2C(=O)c3cc4c(cc3C2=O)C(F)(F)CC2(CNC2)O4)C(=O)N1
O=C1CCC(N2C(=O)c3cc4c(cc3C2=O)OC2(CCNCC2)C(F)(F)C4)C(=O)N1
O=C1CCC(N2C(=O)c3cc4c(cc3C2=O)OC2(CCNCC2)CC4)C(=O)N1
O=C1CCC(N2C(=O)c3cc4c(cc3C2=O)OC2(CC4)CNC2)C(=O)N1
O=C1CCC(N2Cc3cc4c(cc3C2=O)OC2(CCNCC2)CC4)C(=O)N1
O=C1CCC(N2Cc3cc4c(cc3C2=O)OC2(CC4)CNC2)C(=O)N1
O=C1CCC(N2C(=O)c3cc4c(cc3C2=O)OC2(CCNCC2)CO4)C(=O)N1
O=C1CCC(N2C(=O)c3cc4c(cc3C2=O)C2(CCNCC2)CO4)C(=O)N1
O=C5CCC(N4Cc3cc2OCC1(CCNCC1)c2cc3C4=O)C(=O)N5
O=C5CCC(N4Cc3ccc2CCC1(CCNCC1)Oc2c3C4=O)C(=O)N5
O=C5NCC(N4Cc3ccc2CCC1(CCC1)Oc2c3C4=O)C(=O)N5
O=C5CCC(N4Cc3c(ccc2CCC1(CCNCC1)Oc23)C4=O)C(=O)N5
O=C1CCC(N2Cc3c(ccc4c3OCC43CCNCC3)C2=O)C(=O)N1
O=C5CCC(n4c(=O)c3ccc2CCC1(CCNCC1)Oc2c3c4=O)C(=O)N5
O=C5CCC(n4c(=O)c3ccc2CCC1(CNC1)Oc2c3c4=O)C(=O)N5
O=C1CCC(N2C(=O)c3ccc4c(c3C2=O)OCC42CCNCC2)C(=O)N1
O=C1CCC(N2Cc3ccc4c(c3C2=O)OCC2(CCNCC2)C4)C(=O)N1
O=C1CCC(N2C(=O)c3ccc4c(c3C2=O)C2(CCNCC2)CO4)C(=O)N1
O=C5CCC(N4Cc3ccc2OCC1(CCNCC1)Cc2c3C4=O)C(=O)N5
O=C1CCC(N2C(=O)c3ccc(N4C5CNCC4C5)cc3C2=O)C(=O)N1
O=C1CCC(N2C(=O)c3cc(F)c(N4C5CNCC4C5)cc3C2=O)C(=O)N1
O=C1CCC(N2C(=O)c3ccc(N4CC5CC(C4)N5)cc3C2=O)C(=O)N1
O=C1CCC(N2C(=O)c3cc(F)c(N4CC5CC(C4)N5)cc3C2=O)C(=O)N1
O=C1CCC(N2C(=O)c3ccc(N4C5CCC4CNC5)cc3C2=O)C(=O)N1
O=C1CCC(N2C(=O)c3ccc(N4CC5CCC(C4)N5)cc3C2=O)C(=O)N1
O=C1CCC(N2C(=O)c3cc(F)c(N4C5CCC4CNC5)cc3C2=O)C(=O)N1
[2H]C1([2H])NC([2H])([2H])C([2H])([2H])N(c2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1([2H])[2H]
O=C1CCC(N2C(=O)c3ccc(N4CC5CCC4CN5)cc3C2=O)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OCC4CC5(CCC5)C4)C3)cc2F)C(=O)N1
COc1c(N2CC(C)(NC(=O)OCC3CC4(CCC4)C3)C2)ccc(C2CCC(=O)NC2=O)c1F
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC[C@@H]4C[C@H]5CC[C@@H]4C5)C3)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC45CC(C(=O)c6ccccc6)(C4)C5)C3)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC4CN(C(=O)N5Cc6ccccc6C5)C4)C3)cc2F)C(=O)N1
Cc1ccnc(N2CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)C2)c1
Cn1nccc1N1CC(OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1
CN(C(=O)N1CC(OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1)c1cccc(Cl)c1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC4CN(C(=O)N5CCc6ccccc65)C4)C3)cc2F)C(=O)N1
Cc1cccc(N(C)C(=O)N2CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)C2)c1
CN(C(=O)N1CC(OC(=O)NC2(C(F)(F)F)CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1)C1CC1
CN(C(=O)N1CC(OC(=O)NC2(C)CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1)C1CC1
COc1ccc(N(C)C(=O)N2CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)C2)cc1
CN(C)C(=O)N1CC(OC(=O)NC2(C)CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1
Cc1cc(N2CC(NC(=O)OC3CN(C(=O)N(C)C4CC4)C3)C2)cc(F)c1C1CCC(=O)NC1=O
CN(C(=O)N1CC[C@H](OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1)C1CC1
CN(C(=O)N1CC(OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1)c1ccccc1
CN(C)C(=O)N1CC[C@@H](OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1
CN(C)C(=O)N1CCC(OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)CC1
N#Cc1ccc(C(=O)N2CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)C2)cc1
COc1ccc(C(=O)N2CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)C2)cc1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC4CN(C(=O)c5ccc(F)cc5)C4)C3)cc2F)C(=O)N1
Cc1ccc(C(=O)N2CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)C2)cc1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC4CN(C(=O)c5ccccc5)C4)C3)cc2F)C(=O)N1
CN(C(=O)N1CC[C@@H](OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1)C1CC1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC4CN(C(=O)c5ccc(Cl)cc5)C4)C3)cc2F)C(=O)N1
CN(C)C(=O)N1CC[C@H](OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1
O=C1CCC(c2c(Cl)cc(N3CC(NC(=O)OCC4CC5(CCC5)C4)C3)cc2Cl)C(=O)N1
Cc1cccnc1N1CC(OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC4CN(C(=O)N5CCC5)C4)C3)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC4CN(C(=O)N5CC6(CCC6)C5)C4)C3)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC4CN(C(=O)N5CCCC5)C4)C3)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC4CN(C(=O)N5CCC56CCC6)C4)C3)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OCCc4ccccc4)C3)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OCc4ccc(OC(F)(F)F)cc4)C3)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC4CN(C(=O)N5CCCCC5)C4)C3)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OCc4ccccc4)C3)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc([C@@H]3C[C@H]3NC(=O)OCC3CC4(CCC4)C3)cc2F)C(=O)N1
CC(C)O[C@H]1C[C@@H](OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1
CN(C(=O)N1CC(OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1)C1CC1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC4CN(C(=O)C5CC5)C4)C3)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC4CN(S(=O)(=O)C5CC5)C4)C3)cc2F)C(=O)N1
CN(CC1CC1)C(=O)N1CC(OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1
COc1c(N2CC(NC(=O)OCC3CC4(CCC4)C3)C2)ccc(C2CCC(=O)NC2=O)c1F
CN(C)C(=O)N1CC(OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1
CC(C)(C)O[C@H]1C[C@@H](OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1
CC(C)(C)[Si](C)(C)O[C@H]1C[C@H](OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1
CC(C)(C)[Si](C)(C)O[C@H]1C[C@@H](OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1
CC(C)(C)[Si](C)(C)O[C@H]1C[C@@H](COC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1
CC(C)(C)[Si](C)(C)O[C@H]1C[C@H](COC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OCC4CCCCC4)C3)cc2F)C(=O)N1
C[C@H]1CC[C@H](COC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)CC1
CC1(C)CCC(COC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)CC1
O=C1CC[C@H](c2c(F)cc(N3CC[C@@H](NC(=O)OCC4CC5(CCC5)C4)C3=O)cc2F)C(=O)N1
O=C1CC[C@@H](c2c(F)cc(N3CC[C@@H](NC(=O)OCC4CC5(CCC5)C4)C3=O)cc2F)C(=O)N1
CC1(NC(=O)OCC2CC3(CCC3)C2)CN(c2cc(F)c(C3CCC(=O)NC3=O)c(F)c2)C1
O=C1CCC(c2c(F)cc(N3C[C@@H](NC(=O)OCC4CC5(CCC5)C4)CC3=O)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc(N3C[C@H](NC(=O)OCC4CC5(CCC5)C4)CC3=O)cc2F)C(=O)N1
O=C1CCC(c2ccc(N3CC(NC(=O)OCC4CC5(CCC5)C4)C3)cc2F)C(=O)N1
O=C1CCC(c2ccc(N3CC(NC(=O)OCC4CC5(CCC5)C4)C3)cc2Cl)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC[C@H](NC(=O)OCC4CC5(CCC5)C4)C3)cc2F)C(=O)N1
O=C1CCC(c2ccc(N3CC(NC(=O)OCC4CC5(CCC5)C4)C3)cc2)C(=O)N1
COc1c(N2CC(NC(=O)OCC3CC4(CCC4)C3)C2)ccc(C2CCC(=O)NC2=O)c1Cl
O=C1CCC(c2c(F)cc(N3CC[C@@H](NC(=O)OCC4CC5(CCC5)C4)C3)cc2F)C(=O)N1
CC(C)(CCOC(=O)NC1CN(c2cc(F)c(C3CCC(=O)NC3=O)c(F)c2)C1)C1CC1
CC1(CCCOC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)CC1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC4CC5(CCCCC5)C4)C3)cc2F)C(=O)N1
CC(C)C1CC(COC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC4CN(c5nc6ccccc6o5)C4)C3)cc2F)C(=O)N1
Cc1ccccc1N(C)C(=O)N1CC(OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1
CN(C(=O)N1CC(OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1)c1ccccc1Cl
CN(C(=O)N1CC(OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1)c1ccc(F)cc1
CN(C(=O)N1CC(OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1)c1ccc(C#N)cc1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC4CN(C(=O)Cc5ccccc5)C4)C3)cc2F)C(=O)N1
Cn1c(N2CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)C2)nc2ccccc21
CN(C)C(=O)C12CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)(C1)C2
Cn1ccnc1N1CC(OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1
CN(C(=O)C12CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)(C1)C2)C1CC1
Cc1ccc(N2CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)C2)nc1
Cc1cccc(N2CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)C2)n1
CN(C(=O)C12CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)(C1)C2)c1ccccc1
CN(CC1CC1)C(=O)C12CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)(C1)C2
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC4CN(c5ccccn5)C4)C3)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OCC#CC4CC4)C3)cc2F)C(=O)N1
Cc1cc(N2CC(NC(=O)OC3CN(C(=O)N(C)C4CC4)C3)C2)cc(C)c1C1CCC(=O)NC1=O
Cc1cc(N2CC(NC(=O)OC3CN(C(=O)N(C)C4CC4)C3)C2)cc(Cl)c1C1CCC(=O)NC1=O
CN(C(=O)N1CCC(OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)CC1)C1CC1
N#Cc1cc(C2CCC(=O)NC2=O)ccc1N1CC(Nc2nnc(C3CC4(CCC4)C3)o2)C1
COc1c(N2CC(Nc3nnc(-c4ccc(OC(F)(F)F)cc4)o3)C2)ccc(C2CCC(=O)NC2=O)c1F
COc1c(N2CC(Nc3nnc(C4CC5(CCC5)C4)o3)C2)ccc(C2CCC(=O)NC2=O)c1Cl
O=C1CCC(c2c(F)cc(N3C[C@H](Nc4nnc(C5CC6(CCC6)C5)o4)CC3=O)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(Nc4nnc(-c5ccc(Cl)cc5)o4)C3)cc2F)C(=O)N1
COc1c(N2CC(Nc3nnc(C4CC5(CCC5)C4)o3)C2)ccc(C2CCC(=O)NC2=O)c1F
N#Cc1ccc(-c2nnc(NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)o2)cc1
Cc1ccccc1-c1nnc(NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)o1
Cc1cccc(-c2nnc(NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)o2)c1
COc1ccc(-c2nnc(NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)o2)cc1
Cc1ccc(-c2nnc(NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)o2)cc1
O=C1CCC(c2c(F)cc(N3CC(Nc4nnc(Cc5ccccc5)o4)C3)cc2F)C(=O)N1
CC1(Nc2nnc(C3CC4(CCC4)C3)o2)CN(c2cc(F)c(C3CCC(=O)NC3=O)c(F)c2)C1
O=C1CCC(c2c(Cl)cc(N3CC(Nc4nnc(C5CC6(CCC6)C5)o4)C3)cc2Cl)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(Nc4nnc(-c5ccc(OC(F)(F)F)cc5)o4)C3)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(Nc4nnc(-c5ccccc5)o4)C3)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(Nc4ncn(C5CC6(CCC6)C5)n4)C3)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(Nc4cc(C5CC6(CCC6)C5)ccn4)C3)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(Nc4nnc(C5CC6(CCC6)C5)o4)C3)cc2F)C(=O)N1
CN(C(=O)N1CC(OC(=S)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1)C1CC1
Cc1ccc(N(C)C(=O)N2CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)C2)cn1
Cc1ccc(N(C)C(=O)N2CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)C2)nc1
Cc1ccc(C)c(N(C)C(=O)C23CC(OC(=O)NC4CN(c5cc(F)c(C6CCC(=O)NC6=O)c(F)c5)C4)(C2)C3)c1
Cc1cc(Cl)ccc1N(C)C(=O)C12CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)(C1)C2
Cc1cc(Cl)ccc1N(C)C(=O)N1CC(OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1
Cc1cccc(N(C)C(=O)C23CC(OC(=O)NC4CN(c5cc(F)c(C6CCC(=O)NC6=O)c(F)c5)C4)(C2)C3)c1C
Cc1c(Cl)cccc1N(C)C(=O)C12CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)(C1)C2
Cc1ccc(N(C)C(=O)N2CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)C2)c(C)c1
Cc1ccc(N(C)C(=O)C23CC(OC(=O)NC4CN(c5cc(F)c(C6CCC(=O)NC6=O)c(F)c5)C4)(C2)C3)c(C)c1
[2H]C([2H])([2H])N(C(=O)N1CC(OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1)c1ccc(C)cc1
[2H]C([2H])([2H])N(C(=O)N1CC(OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1)c1ccc(Cl)cc1
CN(C(=O)C12CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)(C1)C2)c1ccc(C#N)cc1
COc1c(N2CC(C)(Nc3nnc(C4CC5(CCC5)C4)o3)C2)ccc(C2CCC(=O)NC2=O)c1F
CC1(CCc2nnc(NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)o2)CC1
CN(C(=O)C12CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)(C1)C2)c1cccc(C#N)c1
O=C1CCC(c2c(F)cc(N3CC(Nc4nnc(-c5ccccn5)o4)C3)cc2F)C(=O)N1
CN(C(=O)C12CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)(C1)C2)c1ccc(OC(F)(F)F)cc1
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC45CC(C(=O)N6CCC6)(C4)C5)C3)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(Nc4nnc(CCC5CC5)o4)C3)cc2F)C(=O)N1
O=C1CCC(c2c(F)cc(N3CC(Nc4nnc(-c5cccnc5)o4)C3)cc2F)C(=O)N1
CN(C(=O)C12CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)(C1)C2)c1ccc(Cl)cc1
COc1cccc(N(C)C(=O)C23CC(OC(=O)NC4CN(c5cc(F)c(C6CCC(=O)NC6=O)c(F)c5)C4)(C2)C3)c1
CN(C(=O)C12CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)(C1)C2)c1cccc(Cl)c1
CN(C(=O)C12CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)(C1)C2)c1ccc(F)cc1
Cc1ccc(N(C)C(=O)C23CC(OC(=O)NC4CN(c5cc(F)c(C6CCC(=O)NC6=O)c(F)c5)C4)(C2)C3)cc1
Cc1cccc(N(C)C(=O)C23CC(OC(=O)NC4CN(c5cc(F)c(C6CCC(=O)NC6=O)c(F)c5)C4)(C2)C3)c1
Cc1ccccc1N(C)C(=O)C12CC(OC(=O)NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)(C1)C2
COc1c(N2CC(C)(Nc3nnc(-c4ccc(OC(F)(F)F)cc4)o3)C2)ccc(C2CCC(=O)NC2=O)c1F
O=C1CCC(c2c(F)cc(N3CC(NC(=O)OC45CC(C(=O)c6ccccc6)(C4)C5)C3)cc2F)C(=O)N1
CN(C(=O)N1CC(OC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)C1)c1ccc(Cl)cc1
COC12CC(c3nnc(N[C@H]4CN(c5cc(F)c(C6CCC(=O)NC6=O)c(F)c5)[C@@H]4C)o3)(C1)C2
C[C@@H]1[C@@H](Nc2nnc(C34CC(C(F)(F)F)(C3)C4)o2)CN1c1cc(F)c(C2CCC(=O)NC2=O)c(F)c1
C[C@@H]1[C@@H](Nc2nnc(-c3ccc(C(F)(F)F)cc3)o2)CN1c1cc(F)c(C2CCC(=O)NC2=O)c(F)c1
C[C@@H]1[C@@H](Nc2nnc(C3CC4(CCC4)C3)o2)CN1c1cc(F)c(C2CCC(=O)NC2=O)c(F)c1
Cc1ccc(-c2nnc(N[C@H]3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)[C@@H]3C)o2)cc1
C[C@@H]1[C@@H](Nc2nnc(-c3ccc(OC(F)(F)F)cc3)o2)CN1c1cc(F)c(C2CCC(=O)NC2=O)c(F)c1
CC1(C)[C@@H]2CC[C@@]1(C)[C@@H](NCCCCCCCSc1cc(F)cc3c1CN(C1CCC(=O)NC1=O)C3=O)C2
O=C1CCC(N2Cc3c(SCc4ccc(CN5CCCCC5)cc4)cc(F)cc3C2=O)C(=O)N1
CC1(C)[C@@H]2CC[C@@]1(C)[C@@H](NCc1ccc(CSc3cc(F)cc4c3CN(C3CCC(=O)NC3=O)C4=O)cc1)C2
O=C1CCC(N2Cc3c(SCc4ccc(CN5CCC(F)(F)CC5)cc4)cc(F)cc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(SCc4ccc(CNC56CC7CC(CC(C7)C5)C6)cc4)cc(F)cc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(SCCCCNC45CC6CC(CC(C6)C4)C5)cc(F)cc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(SCCCCCCCNC4CC5(CCC5)C4)cc(F)cc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(SCCCCCCCCN4CCOCC4)cc(F)cc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(CCCCCCCCNC45CC6CC(CC(C6)C4)C5)cc(F)cc3C2=O)C(=O)N1
CCN(CC)CCCCCCCCSc1cc(F)cc2c1CN(C1CCC(=O)NC1=O)C2=O
O=C1CCC(N2Cc3c(SCc4ccc(CN5CCC(F)(F)CC5)c(F)c4)cc(F)cc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(SCCCCCCCN4CCCCC4)cc(F)cc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(SCc4ccc(CCNC56CC7CC(CC(C7)C5)C6)cc4)cc(F)cc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(SCCCCCCCN4CCC(F)(F)CC4)cc(F)cc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(SCc4ccc(CN5CCCCC5)c(F)c4)cc(F)cc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(SCCCCCCC(=O)N4CCCCC4)cc(F)cc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(SCCCCCCCNC4CCCCC4)cc(F)cc3C2=O)C(=O)N1
O=C1CCC(N2Cc3c(SCCCCCCC(=O)N4CCC(F)(F)CC4)cc(F)cc3C2=O)C(=O)N1
CN(CCCCCCCSc1cc(F)cc2c1CN(C1CCC(=O)NC1=O)C2=O)C12CC3CC(CC(C3)C1)C2
O=C1CCC(N2Cc3c(SCc4ccc(CNC56CC7CC(CC(C7)C5)C6)cc4)cc(F)cc3C2=O)C(=O)N1
Fc1c(Cl)cccc1[C@H]1[C@@H](NC2(CCCCC2)[C@@]11C(=O)Nc2cc(Cl)ccc12)C(=O)NCCCCCc1cccc2C(=O)N(Cc12)C1CCC(=O)NC1=O |r|
Fc1c(Cl)cccc1[C@H]1[C@@H](NC2(CCCCC2)[C@@]11C(=O)Nc2cc(Cl)ccc12)C(=O)Nc1ccc(cc1)C(=O)NCCCCCc1cccc2C(=O)N(Cc12)C1CCC(=O)NC1=O |r|
CNC(=O)[C@@H]1NC2(CCCCC2)[C@]2([C@H]1c1cccc(Cl)c1F)C(=O)Nc1cc(Cl)ccc21 |r|
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)Nc1ccc(OCCOCCOCCOCCNc3cccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c34)cc1)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
O=C1CCC(Nc2ccccc2N2CCOCC2)C(=O)N1
Nc1ccc(C(=O)NC2CCC(=O)NC2=O)c2ncccc12
Nc1ccnc2c(cccc12)C(=O)NC1CCC(=O)NC1=O
OC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1ccc(=O)[nH]c1=O |r|
COc1c(cc(cc1C(C)(C)C)-n1ccc(=O)[nH]c1=O)-c1ccc2cc(NS(C)(=O)=O)ccc2c1
CC(C)OC(=O)[C@@H](C)NP(=O)(OC[C@H]1O[C@@H](n2ccc(=O)[nH]c2=O)[C@](C)(F)[C@@H]1O)Oc1ccccc1 |r|
O=C1CCC(=O)N1
C1=CN(C(=O)NC1=O)[C@H]2[C@@H]([C@@H]([C@H](O2)COP(=O)(O)O)O)O
C1C(=O)NC(=O)N1
O=C1CNCN1
CN1CC(=O)NC1=O
O=C1CNC(=S)N1
NN1CC(=O)NC1=O
[O-][N+](=O)c1ccc(\C=C\C=N\N2CC(=O)NC2=O)o1
c1cc2c(c(c1)OCc3ccc(cc3)CN4CCOCC4)CN(C2=O)[C@H]5CCC(=O)NC5=O
COc1ccc(cc1OC2CCCC2)[C@H]3CC(=O)NC3
C1=CNC(=O)NC1=O
Cn1ccc(=O)[nH]c1=O
Nn1ccc(=O)[nH]c1=O
CC(C)c1ccn2ncnc(N[C@H]3CC[C@H](CC3)N3CCN(CC3)C(=O)CCC(=O)N3CCC(CN4CCN(CC4)c4ccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c5c4)CC3)c12 |r,wU:12.11,15.18,(9.52,-11.75,;9.89,-12.93,;11.08,-13.21,;8.83,-14.06,;7.31,-13.87,;6.65,-15.27,;7.78,-16.32,;7.76,-17.86,;9.08,-18.65,;10.42,-17.9,;10.45,-16.36,;11.8,-15.61,;13.12,-16.41,;14.47,-15.67,;15.79,-16.46,;15.76,-18.01,;14.41,-18.76,;13.09,-17.96,;17.08,-18.81,;17.05,-20.34,;18.37,-21.15,;19.71,-20.4,;19.75,-18.86,;18.42,-18.06,;21.04,-21.19,;21.01,-22.43,;22.39,-20.44,;23.71,-21.24,;25.06,-20.49,;25.08,-19.26,;26.38,-21.29,;27.72,-20.54,;29.05,-21.34,;29.02,-22.88,;30.34,-23.67,;30.31,-25.22,;31.62,-26.01,;31.58,-27.55,;30.24,-28.3,;28.92,-27.5,;28.96,-25.97,;30.2,-29.84,;28.85,-30.59,;28.81,-32.12,;30.14,-32.93,;30.41,-34.43,;29.56,-35.34,;31.94,-34.63,;32.69,-35.98,;34.22,-35.9,;35.06,-37.19,;34.35,-38.57,;35.03,-39.6,;32.82,-38.65,;31.98,-37.35,;30.75,-37.42,;32.6,-33.24,;33.81,-33.01,;31.48,-32.18,;31.52,-30.64,;27.67,-23.63,;26.35,-22.83,;9.13,-15.57,)|
CC(C)c1ccn2ncnc(N[C@H]3CC[C@H](CC3)N3CCN(CC3)C(=O)CCC(=O)N3CCC(CCN4CCN(CC4)c4ccc5C(=O)N(C6CCC(=O)NC6=O)C(=O)c5c4)CC3)c12 |r,wU:12.11,15.18,(12.72,-9.27,;13.1,-10.45,;14.3,-10.7,;12.07,-11.59,;10.53,-11.42,;9.91,-12.83,;11.05,-13.86,;11.04,-15.41,;12.38,-16.18,;13.71,-15.41,;13.72,-13.87,;15.05,-13.1,;16.39,-13.88,;17.72,-13.12,;19.05,-13.89,;19.05,-15.43,;17.71,-16.2,;16.38,-15.42,;20.38,-16.21,;20.37,-17.75,;21.71,-18.53,;23.04,-17.77,;23.04,-16.23,;21.71,-15.44,;24.38,-18.54,;24.37,-19.77,;25.71,-17.77,;27.04,-18.55,;28.39,-17.78,;28.39,-16.55,;29.72,-18.55,;31.05,-17.79,;32.38,-18.56,;32.38,-20.11,;33.71,-20.88,;33.7,-22.42,;35.03,-23.2,;35.02,-24.74,;36.36,-25.52,;37.69,-24.75,;37.7,-23.22,;36.37,-22.43,;39.03,-25.53,;40.36,-24.76,;41.7,-25.54,;41.69,-27.08,;42.84,-28.11,;44.05,-27.86,;42.21,-29.51,;43.05,-30.8,;42.26,-32.12,;43,-33.47,;44.54,-33.5,;45.14,-34.58,;45.33,-32.18,;44.59,-30.83,;45.22,-29.77,;40.67,-29.35,;39.84,-30.27,;40.36,-27.85,;39.02,-27.07,;31.04,-20.87,;29.71,-20.09,;12.38,-13.1,)|
CC(C)c1ccn2ncnc(N[C@H]3CC[C@H](CC3)N3CCN(CC3)C(=O)CCC(=O)N3CCC(CCN4CCN(CC4)c4ccc5C(=O)N(C6CCC(=O)N(C)C6=O)C(=O)c5c4)CC3)c12 |r,wU:12.11,15.18,(12.72,-9.27,;13.1,-10.45,;14.3,-10.7,;12.07,-11.59,;10.53,-11.42,;9.91,-12.83,;11.05,-13.86,;11.04,-15.41,;12.38,-16.18,;13.71,-15.41,;13.72,-13.87,;15.05,-13.1,;16.39,-13.88,;17.72,-13.12,;19.05,-13.89,;19.05,-15.43,;17.71,-16.2,;16.38,-15.42,;20.38,-16.21,;20.37,-17.75,;21.71,-18.53,;23.04,-17.77,;23.04,-16.23,;21.71,-15.44,;24.38,-18.54,;24.37,-19.77,;25.71,-17.77,;27.04,-18.55,;28.39,-17.78,;28.39,-16.55,;29.72,-18.55,;31.05,-17.79,;32.38,-18.56,;32.38,-20.11,;33.71,-20.88,;33.7,-22.42,;35.03,-23.2,;35.02,-24.74,;36.36,-25.52,;37.69,-24.75,;37.7,-23.22,;36.37,-22.43,;39.03,-25.53,;40.36,-24.76,;41.7,-25.54,;41.69,-27.08,;42.84,-28.11,;44.05,-27.86,;42.21,-29.51,;43.05,-30.8,;42.26,-32.12,;43,-33.47,;44.54,-33.5,;45.14,-34.58,;45.33,-32.18,;46.84,-32.21,;44.59,-30.83,;45.22,-29.77,;40.67,-29.35,;39.84,-30.27,;40.36,-27.85,;39.02,-27.07,;31.04,-20.87,;29.71,-20.09,;12.38,-13.1,)|
C\C(=N/Nc1nc(cs1)-c1ccc(cc1)-c1ccccc1)C(=O)NCCCCNc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12
[O-][N+](=O)c1ccccc1\C(=N\Nc1nc(cs1)-c1ccc(cc1)-c1ccccc1)C(=O)NCCCCNc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12
C\C(=N/Nc1nc(c(CC(=O)NCCNc2cccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c23)s1)-c1ccc(Cl)c(Cl)c1)C(=O)OCOC(=O)C(C)(C)C
CCS(=O)(=O)N1CC(CC#N)(C1)n1cc(cn1)-c1nc(Nc2ccc(cc2)C(=O)NCCCCNc2cccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c23)nc2[nH]ccc12
CCS(=O)(=O)N1CC(CC#N)(C1)n1cc(cn1)-c1nc(Nc2ccc(cc2)C(=O)NCCCCOc2cccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c23)nc2[nH]ccc12
CCS(=O)(=O)N1CC(CC#N)(C1)n1cc(cn1)-c1nc(Nc2ccc(cc2)C(=O)NC2CCN(CC2)c2ccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c3c2)nc2[nH]ccc12
CCS(=O)(=O)N1CC(CC#N)(C1)n1cc(cn1)-c1nc(Nc2ccc(cc2)C(=O)NCCN2CCN(CC2)c2ccc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c3c2)nc2[nH]ccc12
CCS(=O)(=O)N1CC(CC#N)(C1)n1cc(cn1)-c1nc(Nc2ccc(cc2)C(=O)NCCCCNc2cccc(c2)C2CCC(=O)NC2=O)nc2[nH]ccc12
CCS(=O)(=O)N1CC(CC#N)(C1)n1cc(cn1)-c1nc(Nc2ccc(cc2)C(=O)NCCCCOc2ccc(cc2)C2CCC(=O)NC2=O)nc2[nH]ccc12
CCS(=O)(=O)N1CC(CC#N)(C1)n1cc(cn1)-c1nc(Nc2ccc(cc2)C(=O)NCCCCOc2cccc(c2)C2CCC(=O)NC2=O)nc2[nH]ccc12
CCS(=O)(=O)N1CC(CC#N)(C1)n1cc(cn1)-c1nc(Nc2ccc(cc2)C(=O)NC2CCN(CC2)c2ccc(cc2)C2CCC(=O)NC2=O)nc2[nH]ccc12
CCS(=O)(=O)N1CC(CC#N)(C1)n1cc(cn1)-c1nc(Nc2ccc(cc2)C(=O)NCCN2CCN(CC2)c2ccc(cc2)C2CCC(=O)NC2=O)nc2[nH]ccc12
CCS(=O)(=O)N1CC(CC#N)(C1)n1cc(cn1)-c1nc(Nc2ccc(cc2)C(=O)NCCCN2CCN(CC2)c2ccc(cc2)C2CCC(=O)NC2=O)nc2[nH]ccc12
CCS(=O)(=O)N1CC(CC#N)(C1)n1cc(cn1)-c1nc(Nc2ccc(cc2)C(=O)NCCCN2CC3CC2CN3c2ccc(cc2)C2CCC(=O)NC2=O)nc2[nH]ccc12
CCS(=O)(=O)N1CC(CC#N)(C1)n1cc(cn1)-c1nc(Nc2ccc(cc2)C(=O)NCCCN2CCC3(CC2)CCN(CC3)c2ccc(cc2)C2CCC(=O)NC2=O)nc2[nH]ccc12
Oc1cc(-c2c(Cl)cc3c(nc(NCCCN4CCN(CCCNc5cccc6C(=O)N(C7CCC(=O)NC7=O)C(=O)c56)CC4)nc3c2F)N2CCN(CC2)C(=O)C=C)c2ccccc2c1 |(-16.45,-1.93,;-15.12,-2.7,;-13.8,-1.93,;-12.46,-2.69,;-11.12,-1.92,;-11.12,-.38,;-12.46,.39,;-9.79,.39,;-8.46,-.38,;-7.14,.38,;-5.81,-.38,;-5.8,-1.91,;-4.47,-2.68,;-3.13,-1.91,;-1.8,-2.68,;-.47,-1.91,;.87,-2.68,;2.2,-1.91,;3.53,-2.68,;3.53,-4.22,;4.87,-4.99,;6.2,-4.22,;7.53,-4.99,;8.87,-4.22,;10.2,-4.99,;10.2,-6.53,;11.54,-7.29,;12.87,-6.53,;12.87,-4.98,;13.99,-3.95,;15.48,-4.35,;13.37,-2.54,;14.14,-1.2,;15.68,-1.2,;16.45,.13,;15.68,1.46,;16.45,2.8,;14.14,1.46,;13.37,.13,;11.83,.13,;11.88,-2.69,;10.79,-1.6,;11.54,-4.22,;2.2,-4.99,;.87,-4.22,;-7.12,-2.68,;-8.46,-1.92,;-9.79,-2.69,;-9.79,-4.23,;-7.14,1.92,;-8.47,2.69,;-8.47,4.23,;-7.14,5,;-5.8,4.23,;-5.8,2.69,;-7.14,6.54,;-8.47,7.31,;-5.8,7.31,;-4.47,6.54,;-12.46,-4.24,;-11.13,-5,;-11.13,-6.54,;-12.46,-7.31,;-13.79,-6.55,;-13.79,-5,;-15.12,-4.24,)|
[H][C@@]12CCC[C@]1([H])[C@H](N(C2)C(=O)[C@@H](NC(=O)[C@@H](NC(=O)c1cnc(cn1)C(=O)NCCOCCOCCOc1cc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c3cccc(c1)c23)C1CCCCC1)C(C)(C)C)C(=O)N[C@@H](CCC)C(=O)C(=O)NC1CC1 |r|
CC(C)Nc1cc(ccc1C(=O)N[C@H]1CC[C@@H](CC1)C(=O)NCCOCCNC(=O)COc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12)-n1ccc2cc(cnc12)C#N |r,wU:13.13,wD:16.20,(-14.01,4.43,;-12.49,4.7,;-11.97,6.15,;-11.5,3.52,;-12.03,2.08,;-13.54,1.81,;-14.07,.36,;-13.08,-.82,;-11.56,-.55,;-11.04,.9,;-9.52,1.17,;-9,2.61,;-8.53,-.01,;-7.01,.26,;-6.49,1.7,;-4.97,1.97,;-3.98,.79,;-4.51,-.65,;-6.02,-.92,;-2.49,1.19,;-2.09,2.68,;-1.4,.1,;.08,.5,;1.17,-.59,;2.66,-.19,;3.75,-1.28,;5.24,-.88,;6.33,-1.97,;7.82,-1.57,;8.91,-2.66,;8.21,-.08,;9.7,.32,;10.1,1.81,;9.01,2.89,;9.41,4.38,;10.9,4.78,;11.99,3.69,;13.56,3.77,;14.33,5.1,;14.1,2.36,;15.58,1.97,;16.67,3.05,;18.16,2.66,;18.56,1.17,;20.05,.77,;17.47,.08,;15.98,.48,;14.89,-.61,;12.89,1.39,;12.89,-.15,;11.6,2.21,;-15.59,.09,;-16.69,1.16,;-18.05,.44,;-17.79,-1.08,;-18.73,-2.29,;-18.15,-3.72,;-16.63,-3.93,;-15.68,-2.72,;-16.26,-1.29,;-19.1,-4.94,;-20.05,-6.15,)|
Oc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12
Oc1ccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c2c1
Nc1ccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c2c1
O=C1N(Cc2ccccc12)C1CCC(=O)NC1=O
Oc1cccc2C(=O)N(Cc12)C1CCC(=O)NC1=O
Oc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O
Oc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Oc1cccc2CN(C3CCC(=O)NC3=O)C(=O)c12
Nc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O
Nc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Nc1cccc2CN(C3CCC(=O)NC3=O)C(=O)c12
O=C1N(C2CCC(=O)NC2=O)C(=O)c2cc3CNCc3cc12
C1CC(=O)NC(=O)C1
C1CCNC(=O)C1
C1CNC(=O)NC1=O
O=C1CCN1
CC(=O)NC(N)=O
C[C@H]1CN(CCN1c1ccc(Nc2cc(cn(C)c2=O)-c2ccnc(N3CCn4c5CC(C)(C)Cc5cc4C3=O)c2CO)nc1)C(=O)CNc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12 |r|
C[C@H]1CN(CCN1c1ccc(Nc2cc(cn(C)c2=O)-c2ccnc(N3CCn4c5CC(C)(C)Cc5cc4C3=O)c2CO)nc1)C(=O)c1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12 |r|
C[C@H]1CN(CCN1c1ccc(Nc2cc(cn(C)c2=O)-c2ccnc(N3CCn4c5CC(C)(C)Cc5cc4C3=O)c2CO)nc1)C(=O)CCCCCCCCCCCNc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12 |r|
CC(C)Nc1cc(ncc1C(=O)N[C@H]1CC[C@@H](CC1)C(=O)NCCOCCNC(=O)COc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12)-n1ccc2cc(cnc12)C#N |r,wU:16.20,wD:13.13,(-16.22,-3.7,;-14.89,-2.92,;-14.89,-1.38,;-13.55,-3.7,;-12.22,-2.92,;-12.22,-1.38,;-10.89,-.61,;-9.55,-1.38,;-9.55,-2.92,;-10.89,-3.69,;-10.89,-5.23,;-12.22,-6,;-9.55,-6,;-8.22,-5.23,;-6.89,-6.01,;-5.55,-5.23,;-5.55,-3.69,;-6.89,-2.92,;-8.22,-3.69,;-4.22,-2.92,;-4.22,-1.38,;-2.88,-3.69,;-1.55,-2.92,;-.22,-3.69,;1.12,-2.92,;2.45,-3.69,;3.78,-2.92,;5.12,-3.69,;6.45,-2.92,;6.45,-1.38,;7.79,-3.69,;9.12,-2.92,;10.45,-3.69,;10.45,-5.23,;11.79,-6,;13.12,-5.23,;13.12,-3.69,;14.25,-2.66,;15.74,-3.06,;13.63,-1.24,;14.4,.09,;13.63,1.43,;14.4,2.76,;15.94,2.76,;16.71,4.09,;16.71,1.43,;15.94,.09,;16.71,-1.24,;12.13,-1.39,;11.04,-.3,;11.79,-2.92,;-10.89,.92,;-9.76,1.96,;-10.38,3.38,;-11.87,3.23,;-13.03,4.29,;-14.53,3.83,;-14.88,2.29,;-13.72,1.23,;-12.22,1.69,;-15.62,4.92,;-16.71,6.01,)|
O=C1CCC(CSc2ccccc2)C(=O)N1
Clc1ccc(SCC2CCC(=O)NC2=O)cc1
Cc1ccc(SCC2CCC(=O)NC2=O)cc1
Fc1ccc(SCC2CCC(=O)NC2=O)cc1
Brc1ccc(SCC2CCC(=O)NC2=O)cc1
Cc1cc(C)c(SCC2CCC(=O)NC2=O)c(C)c1
Cn1cnnc1SCC1CCC(=O)NC1=O
COC(=O)c1ccccc1SCC1CCC(=O)NC1=O
[O-][N+](=O)c1ccccc1SCC1CCC(=O)NC1=O
[O-][N+](=O)c1cccc(SCC2CCC(=O)NC2=O)c1
[O-][N+](=O)c1ccc(SCC2CCC(=O)NC2=O)cc1
O=C1CCC(CSCc2ccccc2)C(=O)N1
COc1ccc(CSCC2CCC(=O)NC2=O)cc1
O=C1CCC(CSc2ccccn2)C(=O)N1
O=C1CCC(CSc2ncccn2)C(=O)N1
Cc1ccnc(SCC2CCC(=O)NC2=O)n1
Nc1ccccc1SCC1CCC(=O)NC1=O
Nc1cccc(SCC2CCC(=O)NC2=O)c1
Nc1ccc(SCC2CCC(=O)NC2=O)cc1
CC(=O)Nc1ccccc1SCC1CCC(=O)NC1=O
CC(=O)Nc1cccc(SCC2CCC(=O)NC2=O)c1
CC(=O)Nc1ccc(SCC2CCC(=O)NC2=O)cc1
O=C1CCC(CS(=O)(=O)c2ccccc2)C(=O)N1
Clc1ccc(cc1)S(=O)(=O)CC1CCC(=O)NC1=O
Cc1ccc(cc1)S(=O)(=O)CC1CCC(=O)NC1=O
Fc1ccc(cc1)S(=O)(=O)CC1CCC(=O)NC1=O
O=C1CCC(CS(=O)(=O)Cc2ccccc2)C(=O)N1
COc1ccc(CS(=O)(=O)CC2CCC(=O)NC2=O)cc1
O=C1N(C2CCC(=O)NC2=O)C(=O)c2cc(ccc12)N1CCC1
CN1CCN(CC1)c1cc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c2cc1F
CN1Cc2cc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c3cc2C1
CN1CCc2cc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c3cc2C1
CN1CCc2cc3C(=O)N(C4CCC(=O)NC4=O)C(=O)c3cc2CC1
O=C(NC1CCC(=O)NC1=O)c1ccccc1
Fc1cc(C(=O)NC2CCC(=O)NC2=O)c(F)c(F)c1F
Nc1cccc(c1)C(=O)NC1CCC(=O)NC1=O
Nc1cccc(C(=O)NC2CCC(=O)NC2=O)c1F
Nc1ccc(cc1)C(=O)NC1CCC(=O)NC1=O
Nc1ccc(C(=O)NC2CCC(=O)NC2=O)c(F)c1
Nc1ccccc1C(=O)NC1CCC(=O)NC1=O
Nc1cccc(F)c1C(=O)NC1CCC(=O)NC1=O
Nc1ccc(C(=O)NC2CCC(=O)NC2=O)c(Cl)c1
Nc1ccc(C(=O)NC2CCC(=O)NC2=O)c(c1)C(F)(F)F
Cc1cc(N)ccc1C(=O)NC1CCC(=O)NC1=O
COc1cc(N)ccc1C(=O)NC1CCC(=O)NC1=O
Nc1ccc(C(=O)NC2CCC(=O)NC2=O)c(O)c1
COc1c(N)c(F)cc(C(=O)NC2CCC(=O)NC2=O)c1F
CCCCNc1ccc(C(=O)NC2CCC(=O)NC2=O)c(F)c1
CCCCNC(=O)CNc1ccc(C(=O)NC2CCC(=O)NC2=O)c(F)c1
CCCCOc1ccc(C(=O)NC2CCC(=O)NC2=O)c(F)c1
CCCCNc1c(F)cc(C(=O)NC2CCC(=O)NC2=O)c(F)c1OC
CCCCNc1ccc2c(c1)nnn(C1CCC(=O)NC1=O)c2=O
CCCCOc1ccc(cc1)C1CCC(=O)NC1=O
CCCCNc1ccc2C(=O)N(Cc2c1)C1CCC(=O)NC1=O
O=C(NC1CCC(=O)NC1=O)c1ccccn1
CC(=O)Nc1sccc1C(=O)NC1CCC(=O)NC1=O
Cc1cc2cccc(C(=O)NC3CCC(=O)NC3=O)c2o1
FS(=O)(=O)c1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
FS(=O)(=O)Oc1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C1N(Cc2ccc(cc12)S(=O)(=O)n1nccn1)C1CCC(=O)NC1=O
O=C1N(Cc2ccc(cc12)S(=O)(=O)n1cncn1)C1CCC(=O)NC1=O
O=C1N(Cc2ccc(cc12)S(=O)(=O)n1ccnc1)C1CCC(=O)NC1=O
Cc1cn(cn1)S(=O)(=O)c1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Fc1cn(cn1)S(=O)(=O)c1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
FC(F)(F)c1cn(cn1)S(=O)(=O)c1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Cc1cnn(c1)S(=O)(=O)c1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Fc1ccn(n1)S(=O)(=O)c1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Fc1cnn(c1)S(=O)(=O)c1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
FC(F)(F)c1ccn(n1)S(=O)(=O)c1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
FC(F)(F)c1cnn(c1)S(=O)(=O)c1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Cc1cn(c(=O)[nH]c1=O)S(=O)(=O)c1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
O=C1N(Cc2ccc(cc12)S(=O)(=O)n1ccc(=O)[nH]c1=O)C1CCC(=O)NC1=O
Nc1ccn(c(=O)n1)S(=O)(=O)c1ccc2CN(C3CCC(=O)NC3=O)C(=O)c2c1
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)N1CCC(CC1)c1ccc3C(=O)N(Cc3c1)C1CCC(=O)NC1=O)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)NCCN1CCC(CC1)c1ccc3C(=O)N(Cc3c1)C1CCC(=O)NC1=O)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)NCCCN1CCC(CC1)c1ccc3C(=O)N(Cc3c1)C1CCC(=O)NC1=O)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)NCCCCN1CCC(CC1)c1ccc3C(=O)N(Cc3c1)C1CCC(=O)NC1=O)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)NCCCCCN1CCC(CC1)c1ccc3C(=O)N(Cc3c1)C1CCC(=O)NC1=O)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)NCCCCCCN1CCC(CC1)c1ccc3C(=O)N(Cc3c1)C1CCC(=O)NC1=O)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)Nc1ccc(Cc3ccc4C(=O)N(Cc4c3)C3CCC(=O)NC3=O)cc1)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)NCCNc1ccc(Cc3ccc4C(=O)N(Cc4c3)C3CCC(=O)NC3=O)cc1)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)NCCCNc1ccc(Cc3ccc4C(=O)N(Cc4c3)C3CCC(=O)NC3=O)cc1)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)NCCCCNc1ccc(Cc3ccc4C(=O)N(Cc4c3)C3CCC(=O)NC3=O)cc1)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)NCCCCCNc1ccc(Cc3ccc4C(=O)N(Cc4c3)C3CCC(=O)NC3=O)cc1)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)NCCCCCCNc1ccc(Cc3ccc4CN(C5CCC(=O)NC5=O)C(=O)c4c3)cc1)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)NCCN1CCC3(CCC(CC3)c3ccc4C(=O)N(Cc4c3)C3CCC(=O)NC3=O)CC1)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)NCCN1CC3(C1)CCC(CC3)c1ccc3C(=O)N(Cc3c1)C1CCC(=O)NC1=O)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
Cc1sc-2c(c1C)C(=N[C@@H](CC(=O)NCCN1CC(C1)N1CCC(CC1)c1ccc3C(=O)N(Cc3c1)C1CCC(=O)NC1=O)c1nnc(C)n-21)c1ccc(Cl)cc1 |r,c:8|
O=C(Cc1ccccc1)NC1CCC(=O)NC1=O
O=C(NCc1ccccc1)[C@@H]1CCC(=O)N1 |r|
O=C(NCc1ccccc1)[C@H]1CCC(=O)N1 |r|
CN1C(=O)CCC(N2Cc3ccc(cc3C2=O)S(F)(=O)=O)C1=O
O=C1CCC(N2Cc3ccccc3C2)C(=O)N1
FS(=O)(=O)c1cccc(CC(=O)NC2CCC(=O)NC2=O)c1
FS(=O)(=O)c1cccc(CNC(=O)[C@@H]2CCC(=O)N2)c1 |r|
FS(=O)(=O)c1cccc(CNC(=O)[C@H]2CCC(=O)N2)c1 |r|
FS(=O)(=O)c1ccc2CN(C3CCC(=O)NC3)C(=O)c2c1
FS(=O)(=O)c1ccc2CN(Cc2c1)C1CCC(=O)NC1=O
FS(=O)(=O)c1ccc(CC(=O)NC2CCC(=O)NC2=O)cc1
FS(=O)(=O)c1ccc(CNC(=O)[C@@H]2CCC(=O)N2)cc1 |r|
FS(=O)(=O)c1ccc(CNC(=O)[C@H]2CCC(=O)N2)cc1 |r|
O=C1CCC(N2Cc3cccc(OCc4ccc(CN5CCOCC5)cc4)c3C2)C(=O)N1
CN(CCCC#Cc1cccc2C(=O)N(Cc12)C1CCC(=O)NC1=O)C(=O)CCN(C(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)c1cc2cc(ccc2s1)C(F)(F)P(O)(O)=O)C(C)(C)C)c1ccc(cc1)-c1nccs1 |r|
CN(CCCC#Cc1cccc2C(=O)N(Cc12)C1CCC(=O)N(C)C1=O)C(=O)CCN(C(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)c1cc2cc(ccc2s1)C(F)(F)P(O)(O)=O)C(C)(C)C)c1ccc(cc1)-c1nccs1 |r|
O=C1CCC(C(=O)N1)c1ccccc1
COc1nc(OCc2cccc(-c3ccccc3)c2C)ccc1CNCCNC(=O)CCCCCCCCNC(=O)COc1ccc(C2CCC(=O)NC2=O)cc1
c1cc2c(c[nH]c2c(c1)NS(=O)(=O)c3ccc(cc3)S(=O)(=O)N)Cl
Cc1ccc(c2c1c(c[nH]2)C#N)NS(=O)(=O)c3cccc(c3)C#N
CO[C@H]1CC[C@@H](CC1)n1c(nc2cc(ccc12)-c1c(C)noc1C)[C@@H]1CCCC(=O)N1c1ccc(F)c(F)c1 |r,wU:24.27,5.8,wD:2.1,(-5.83,-7.85,;-6.97,-6.82,;-6.65,-5.31,;-5.19,-4.84,;-4.87,-3.33,;-6.01,-2.3,;-7.48,-2.77,;-7.8,-4.28,;-5.69,-.79,;-4.29,-.17,;-4.45,1.37,;-5.95,1.69,;-6.72,3.02,;-8.26,3.02,;-9.03,1.69,;-8.26,.35,;-6.72,.35,;-9.03,4.35,;-8.41,5.76,;-6.9,6.08,;-9.55,6.79,;-10.89,6.02,;-10.57,4.51,;-11.6,3.37,;-2.95,-.94,;-2.95,-2.48,;-1.62,-3.25,;-.29,-2.48,;-.29,-.94,;1.05,-.17,;-1.62,-.17,;-1.62,1.37,;-.29,2.14,;-.29,3.68,;-1.62,4.45,;-1.62,5.99,;-2.95,3.68,;-4.29,4.45,;-2.95,2.14,)|
CC(=O)c1cc(C(=O)Nc2cc(CO)cc(-c3cnn(C)c3)c2F)c2cc(O)ccn12
CC(=O)c1cc(C(=O)Nc2cc(CO)cc(-c3cnn(C)c3)c2F)c2cc(OCCCCC(=O)NCCCc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)ccn12
CC(=O)c1cc(C(=O)Nc2cc(CO)cc(-c3cnn(C)c3)c2F)c2cc(OCCCCCC(=O)NCCCc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)ccn12
CC(=O)c1cc(C(=O)Nc2cc(CO)cc(-c3cnn(C)c3)c2F)c2cc(OCCCCCCC(=O)NCCCc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)ccn12
CC(=O)c1cc(C(=O)Nc2cc(CO)cc(-c3cnn(C)c3)c2F)c2cc(OCC(=O)NCCCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)ccn12
CC(=O)c1cc(C(=O)Nc2cc(CO)cc(-c3cnn(C)c3)c2F)c2cc(OCCCC(=O)NCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)ccn12
O=C1CCC2(CC(c3ccccc3Cl)=NO2)C(=O)N1
O=C1CCC2(CC(c3ccc(Cl)cc3Cl)=NO2)C(=O)N1
O=C1CCC2(CC(c3c(Cl)cccc3Cl)=NO2)C(=O)N1
O=C1CCC2(CC(c3ccccc3Br)=NO2)C(=O)N1
O=C1CCC2(CC(c3ccccc3I)=NO2)C(=O)N1
O=C1CCC2(CC(c3ccccc3F)=NO2)C(=O)N1
O=C1CCC2(CC(c3ccccc3[N+](=O)[O-])=NO2)C(=O)N1
COc1ccccc1C1=NOC2(CCC(=O)NC2=O)C1
COc1ccc(C2=NOC3(CCC(=O)NC3=O)C2)c(OC)c1OC
O=C1CCC2(CC(c3ccc(C(=O)O)cc3)=NO2)C(=O)N1
O=C1CCC2(CC(c3cccnc3)=NO2)C(=O)N1
O=C1CCC2(CC(C3CCCCC3)=NO2)C(=O)N1
O=C1CCC2(CC(C3CCCC3)=NO2)C(=O)N1
CCCC1=NOC2(CCC(=O)NC2=O)C1
CC(C)(C)C1=NOC2(CCC(=O)NC2=O)C1
CCC(CC)C1=NOC2(CCC(=O)NC2=O)C1
CC1CC(=O)NC(=O)C1
CC1(C)CC(=O)NC(=O)C1
CC(C)(O)c1cc2nn(CCCCCCCCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)cc2cc1NC(=O)c1cccc(C(F)(F)F)n1
CC(C)(O)c1cc2c(cnn2CCCCCCCCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1NC(=O)c1cccc(C(F)(F)F)n1
CC(C)(O)c1cc2nn(CCCCCNCCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)cc2cc1NC(=O)c1cccc(C(F)(F)F)n1
CN(CCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C[C@H]1CC[C@H](n2cc3cc(NC(=O)c4cccc(C(F)(F)F)n4)c(C(C)(C)O)cc3n2)CC1
CN(CCCN(C)c1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C[C@H]1CC[C@H](n2cc3cc(NC(=O)c4cccc(C(F)(F)F)n4)c(C(C)(C)O)cc3n2)CC1
CN(CCCCc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C[C@H]1CC[C@H](n2cc3cc(NC(=O)c4cccc(C(F)(F)F)n4)c(C(C)(C)O)cc3n2)CC1
CN(CCCOCCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C[C@H]1CC[C@H](n2cc3cc(NC(=O)c4cccc(C(F)(F)F)n4)c(C(C)(C)O)cc3n2)CC1
CN(CCCO[C@H]1C[C@@H](Nc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C1)C[C@H]1CC[C@H](n2cc3cc(NC(=O)c4cccc(C(F)(F)F)n4)c(C(C)(C)O)cc3n2)CC1
CN(CCCO[C@H]1C[C@H](Nc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C1)C[C@H]1CC[C@H](n2cc3cc(NC(=O)c4cccc(C(F)(F)F)n4)c(C(C)(C)O)cc3n2)CC1
COc1cc2nn([C@H]3CC[C@H](CN(C)CCCO[C@H]4C[C@H](Nc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)cc2cc1NC(=O)c1cccc(C(F)(F)F)n1
CN(CCCO[C@H]1C[C@H](Nc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C1)C[C@H]1CC[C@H](n2cc3cc(NC(=O)c4cccc(C(F)(F)F)n4)ccc3n2)CC1
CN(CCCO[C@H]1C[C@H](Nc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C1)C[C@H]1CC[C@H](n2cc3cc(NC(=O)c4cccc(C(F)(F)F)n4)c(C(F)F)cc3n2)CC1
CC(C)(O)c1cc2nn([C@H]3CC[C@H](CN4CCC(O[C@H]5C[C@H](Nc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)CC3)cc2cc1NC(=O)c1cccc(C(F)(F)F)n1
CN(C[C@H]1CC[C@H](n2cc3cc(NC(=O)c4cccc(C(F)(F)F)n4)c(C(C)(C)O)cc3n2)CC1)[C@H]1CCC2(CC1)C[C@H](Nc1cccc3c1C(=O)N(C1CCC(=O)NC1=O)C3=O)C2
CC(C)(O)c1cc2nn([C@H]3CC[C@H](CN4CCC5(CC4)CC(Nc4cccc6c4C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)cc2cc1NC(=O)c1cccc(C(F)(F)F)n1
CC(C)(O)c1cc2nn([C@H]3CC[C@H](CN4CCC5(CC4)CC(CNc4cccc6c4C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)cc2cc1NC(=O)c1cccc(C(F)(F)F)n1
COc1cc2nn([C@H]3CC[C@H](CN4CCC5(CC4)CC(CNc4cccc6c4C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)cc2cc1NC(=O)c1cccc(C(F)(F)F)n1
O=C1CCC(N2C(=O)c3cccc(NCC4CC5(CCN(C[C@H]6CC[C@H](n7cc8cc(NC(=O)c9cccc(C(F)(F)F)n9)c(C(F)F)cc8n7)CC6)CC5)C4)c3C2=O)C(=O)N1
COc1cc2nn([C@H]3CC[C@H](CN4CC5(CC(CCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)CC3)cc2cc1NC(=O)c1cccc(C(F)(F)F)n1
CC(C)(O)c1cc2nc([C@H]3CC[C@H](CN4CC5(CC(CCNc6cccc7c6C(=O)N([C@H]6CCC(=O)NC6=O)C7=O)C5)C4)CC3)sc2cc1NC(=O)c1cccc(C(F)(F)F)n1
CC(C)(O)c1cc2nc([C@H]3CC[C@H](CN4CC5(CC(CCNc6cccc7c6C(=O)N([C@@H]6CCC(=O)NC6=O)C7=O)C5)C4)CC3)sc2cc1NC(=O)c1cccc(C(F)(F)F)n1
Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCN(C(=O)CN2CCN(CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)CC1
Cc1cc(-c2nc(Nc3cnn(C4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)c3)ncc2F)ccc1CNC(=O)c1cn(C(C)(C)C)nn1
CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(C(=O)CN3Cc4cc5c(cc4C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)C1
CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCC(CCN3Cc4cc5c(cc4C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)C1
CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2[C@H]2CC[C@H](CN3Cc4cc5c(cc4C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)C1
CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2[C@H]2CC[C@@H](CN3Cc4cc5c(cc4C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)C1
CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C[C@H]2CC[C@H](CN3Cc4cc5c(cc4C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)C1
CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2CC2CCC(N3Cc4cc5c(cc4C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)C1
CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCC(N3Cc4cc5c(cc4C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)C1
Fc1c2C(=O)N(C3CCC(=O)NC3=O)C(=O)c2c(F)c(F)c1F
CN1Cc2cc3c(cc2C1)C(=O)N(C1CCC(=O)NC1=O)C3
CS(=O)(=O)C
CNc1ccccc1C(=O)NCCn1ccc(=O)[nH]c1=O