3798 SMILES Strings for Serine/threonine-protein kinase B-raf

Compound Name
SMILES String
CNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(cc3F)C3CC3)c(F)c2F)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
NS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CCNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
Fc1cc(I)ccc1Nc1c(F)c(F)c(Cc2ccnc(NS(=O)(=O)NC3CC3)c2F)cc1C(=O)NC1CC1
FCCNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CNC(=O)c1cc(Cc2ccnc(NS(=O)(=O)NC)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NOC(C)(C)C)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
COCCNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NOC(C)(C)C)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NOC(C)C)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
COCCNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NOC(C)C)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CC(C)ONC(=O)c1cc(Cc2ccnc(NS(=O)(=O)NC3(C)CCC3)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NOC)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
COCCNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NOC)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CONC(=O)c1cc(Cc2ccnc(NS(=O)(=O)NC3(C)CCC3)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
COCC1(CC1)NS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CC(O)CNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(SC)cc3F)c(F)c2F)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(C=C)cc3F)c(F)c2F)c1F
CCCNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(cc3F)C#C)c(F)c2F)c1F
NC(=O)c1cc(Cc2ccnc(NS(=O)(=O)NCC3COC3)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
NC(=O)c1cc(Cc2ccnc(NS(=O)(=O)NC3C4COCC34)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
CC1(CC1)NS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
COCC(C)(C)NS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(cc3F)C#C)c(F)c2F)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(Br)cc3F)c(F)c2F)c1F
NC(=O)c1cc(Cc2ccnc(NS(=O)(=O)NC34CC(C3)C4)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
NC(=O)c1cc(Cc2ccnc(NS(=O)(=O)NC3CCOCC3)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
NC(=O)c1cc(Cc2ccnc(NS(=O)(=O)NC3CC3)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
CC(C)NS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
NC(=O)c1cc(Cc2ccnc(NS(=O)(=O)NC3CCC3)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
COCCNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CC(C)CNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CC1(CCC1)NS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
NC(=O)c1cc(Cc2ccnc(NS(=O)(=O)NCC3CC3)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
CC(C)(C)NS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CCS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CCS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CCNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CCCNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
NC(=O)c1cc(Cc2ccnc(NS(=O)(=O)NCCF)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
Nc1nccc(Cc2cc(C(O)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CCNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NOCCO)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CCCNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NOCCO)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CC1(CCC1)NS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(cc3F)C3CC3)c(F)c2F)c1F
CC1(CCC1)NS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NOCCO)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NOCCOC)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NC3CC3C)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)N[C@H]3C[C@H]3C)c(Nc3ccc(I)cc3F)c(F)c2F)c1F |r|
CNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)N[C@@H]3C[C@H]3C)c(Nc3ccc(I)cc3F)c(F)c2F)c1F |r|
CNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NC3CC3(F)F)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CCCS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
NC(=O)c1cc(Cc2ccnc(NS(=O)(=O)NCCO)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
NC(=O)c1cc(Cc2ccnc(NS(N)(=O)=O)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
NC(=O)c1cc(Cc2ccnc(NS(=O)(=O)NC3CC3)c2F)c(F)c(F)c1Nc1ccc(I)cc1Cl
Fc1c(F)c(Nc2ccc(I)cc2Cl)c(cc1Cc1ccnc(NS(=O)(=O)NC2CC2)c1F)C(=O)NC1CC1
CC(C)(C)ONC(=O)c1cc(Cc2ccnc(NS(=O)(=O)NC3CC3)c2F)c(F)c(F)c1Nc1ccc(I)cc1Cl
CS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CONC(=O)c1cc(Cc2ccnc(NS(C)(=O)=O)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
CCS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NOC)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
NC(=O)c1cc(Cc2ccnc(NS(N)(=O)=O)c2)c(F)c(F)c1Nc1ccc(I)cc1F
COCCNS(=O)(=O)Nc1cc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)ccn1
CNS(=O)(=O)Nc1cc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)ccn1
CNS(C)(=O)=Nc1cc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)ccn1
CNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3C)c(F)c2F)c1F
CNS(=O)(=O)Nc1cccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)c(F)c2F)c1
COCCNS(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
COCC(C)(C)NS(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
NC(=O)c1cc(Cc2cccc(NS(=O)(=O)NC[C@H]3CCCO3)c2F)c(F)c(F)c1Nc1ccc(I)cc1F |r|
CCS(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
COCCS(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CNS(=O)(=O)Nc1cccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
NS(=O)(=O)Nc1cccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CCS(=O)(=O)Nc1cccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CC1(CCC1)NS(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CC1(CCC1)NS(=O)(=O)Nc1cccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CNS(=O)(=O)Nc1cccc(Cc2cc(C(=O)NOC)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CONC(=O)c1cc(Cc2cccc(NS(N)(=O)=O)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
CONC(=O)c1cc(Cc2cccc(NS(=O)(=O)NC3(C)CCC3)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
CNS(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(cc3F)C3CC3)c(F)c2F)c1F
CNS(=O)(=O)Nc1cccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(cc3F)C3CC3)c(F)c2F)c1F
CNS(=O)(=O)Nc1cccc(Cc2cc(C(=O)NOC)c(Nc3ccc(cc3F)C3CC3)c(F)c2F)c1F
CCS(=O)(=O)Nc1cccc(Cc2cc(C(=O)NOC)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CCS(=O)(=O)Nc1cccc(Cc2cc(C(=O)NOC(C)(C)C)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
COCC1(CC1)S(=O)(=O)Nc1cccc(Cc2cc(C(=O)NOC)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
COCC1(CC1)S(=O)(=O)Nc1cccc(Cc2cc(C(=O)NOC(C)(C)C)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CONC(=O)c1cc(Cc2cccc(NS(=O)(=O)C3(C)CC3)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
CC(C)(C)ONC(=O)c1cc(Cc2cccc(NS(=O)(=O)C3(C)CC3)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
CNS(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
NC(=O)c1cc(Cc2cccc(NS(N)(=O)=O)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
CCS(=O)(=O)Nc1cccc(Cc2cc(C(=O)NOC)c(Nc3ccc(I)cc3Cl)c(F)c2F)c1F
CCS(=O)(=O)Nc1cccc(Cc2cc(C(=O)NOC(C)(C)C)c(Nc3ccc(I)cc3Cl)c(F)c2F)c1F
CCS(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3Cl)c(F)c2F)c1F
CC(C)(C)ONC(=O)c1cc(Cc2cccc(NS(=O)(=O)NC3CC3)c2F)c(F)c(F)c1Nc1ccc(I)cc1Cl
CS(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
NC(=O)c1cc(Cc2cccc(NS(=O)(=O)CC3CC3)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
NC(=O)c1cc(Cc2cccc(NS(=O)(=O)CCCF)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
CC1(CC1)S(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CC(C)CS(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CCCS(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
COCC1(CC1)S(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
NC(=O)c1cc(Cc2cccc(NS(=O)(=O)C3CCC3)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
NC(=O)c1cc(Cc2cccc(NS(=O)(=O)C3COC3)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
NC(=O)c1cc(Cc2cccc(NS(=O)(=O)C3CC3)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
NC(=O)c1cc(Cc2cccc(NS(=O)(=O)C3CCOCC3)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
CC(C)S(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CS(=O)(=O)Nc1cccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CONC(=O)c1cc(Cc2cccc(NS(C)(=O)=O)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
CNS(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1
CCS(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1
COCCS(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1
CNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(cc3F)C3CC3)c(F)c2F)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NOC)c(Nc3ccc(cc3F)C3CC3)c(F)c2F)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NOC)c(Nc3ccc(Br)cc3F)c(F)c2F)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NOC)c(Nc3ccc(Cl)cc3F)c(F)c2F)c1F
CC1(CCC1)NS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(cc3F)C3CC3)c(F)c2F)c1F
CONC(=O)c1cc(Cc2ccnc(NS(=O)(=O)NC3(C)CCC3)c2F)c(F)c(F)c1Nc1ccc(cc1F)C1CC1
CCS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(cc3F)C3CC3)c(F)c2F)c1F
CCS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NOC)c(Nc3ccc(cc3F)C3CC3)c(F)c2F)c1F
CONC(=O)c1cc(Cc2ccnc(NS(C)(=O)=O)c2F)c(F)c(F)c1Nc1ccc(cc1F)C1CC1
CNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(SC(F)F)cc3F)c(F)c2F)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc4sccc4c3)c(F)c2F)c1F
COc1ccc(COc2ccc(F)c(F)c2F)cc1
CNS(=O)(=O)Nc1nccc(Oc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CNS(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)n1
CNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)cc2F)c1F
CCNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)cc2F)c1F
NC(=O)c1cc(Cc2ccnc(NS(=O)(=O)NC3CC3)c2F)c(F)cc1Nc1ccc(I)cc1F
COCCNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)cc2F)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)n(C)c2=O)c1F
COCCNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)n(C)c2=O)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(cc3F)C3CC3)n(C)c2=O)c1F
Cn1c(Nc2ccc(cc2F)C2CC2)c(cc(Cc2ccnc(NS(=O)(=O)NC3CC3)c2F)c1=O)C(N)=O
CNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)n(C)c2=O)c1F
Cn1c(Nc2ccc(I)cc2F)c(cc(Cc2ccnc(NS(=O)(=O)NC3CC3)c2F)c1=O)C(=O)NC1CC1
COCCNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)n(C)c2=O)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NOC)c(Nc3ccc(I)cc3F)n(C)c2=O)c1F
COCCNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NOC)c(Nc3ccc(I)cc3F)n(C)c2=O)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)NOC(C)(C)C)c(Nc3ccc(I)cc3F)n(C)c2=O)c1F
Cn1c(Nc2ccc(I)cc2F)c(cc(Cc2ccnc(NS(=O)(=O)NC3CC3)c2F)c1=O)C(=O)NOC(C)(C)C
Cn1c(Nc2ccc(I)cc2F)c(cc(Cc2ccnc(NS(=O)(=O)NC3CC3)c2F)c1=O)C(N)=O
CCNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)n(C)c2=O)c1F
Cn1c(Nc2ccc(I)cc2F)c(cc(Cc2ccnc(NS(=O)(=O)NC3(C)CCC3)c2F)c1=O)C(N)=O
CNS(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)n(C)c2=O)c1F
CCNS(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)n(C)c2=O)c1F
Cn1c(Nc2ccc(I)cc2F)c(cc(Cc2cccc(NS(=O)(=O)NC3CC3)c2F)c1=O)C(N)=O
CNS(=O)(=O)Nc1cccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)n(C)c2=O)c1F
Cn1c(Nc2ccc(I)cc2F)c(cc(Cc2cccc(NS(=O)(=O)NC3CC3)c2F)c1=O)C(=O)NC1CC1
Cn1c(Nc2ccc(I)cc2F)c(cc(Cc2cccc(NS(=O)(=O)C3(C)CC3)c2F)c1=O)C(N)=O
CONC(=O)c1cc(Cc2cccc(NS(=O)(=O)C3(C)CC3)c2F)c(=O)n(C)c1Nc1ccc(I)cc1F
CCS(=O)(=O)Nc1cccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)n(C)c2=O)c1F
CCS(=O)(=O)Nc1cccc(Cc2cc(C(=O)NOC(C)(C)C)c(Nc3ccc(I)cc3F)n(C)c2=O)c1F
CCS(=O)(=O)Nc1cccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)n(C)c2=O)c1F
Cn1c(Nc2ccc(I)cc2F)c(cc(Cc2cccc(NS(=O)(=O)C3(C)CC3)c2F)c1=O)C(=O)NC1CC1
Cn1c(Nc2ccc(I)cc2F)c(cc(Cc2cccc(NS(=O)(=O)C3(C)CC3)c2F)c1=O)C(=O)NOC(C)(C)C
CCNS(=O)(=O)Nc1cccc(Cc2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)n(C)c2=O)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(=O)OC)c(Nc3ccc(I)cc3F)cn2)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)n3cncc23)c1F
CNS(=O)(=O)Nc1nccc(Cn2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2=O)c1F
CCCNS(=O)(=O)Nc1nccc(Cn2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2=O)c1F
CNS(=O)(=O)Nc1nccc(Cn2cc(C(N)=O)c(Nc3ccc(SC)cc3F)c(F)c2=O)c1F
Cc1c(Nc2ccc(I)cc2F)c(cn(Cc2ccnc(NS(=O)(=O)NC3(C)CCC3)c2F)c1=O)C(N)=O
CCS(=O)(=O)Nc1nccc(Cn2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)c(C)c2=O)c1F
CCS(=O)(=O)Nc1nccc(Cn2cc(C(=O)NOC)c(Nc3ccc(I)cc3F)c(C)c2=O)c1F
CNS(=O)(=O)Nc1nccc(Cn2cc(C(=O)NC3CC3)c(Nc3ccc(I)cc3F)c(C)c2=O)c1F
CNS(=O)(=O)Nc1nccc(Cn2cc(C(=O)NOC)c(Nc3ccc(I)cc3F)c(C)c2=O)c1F
OC[C@@H](O)CONC(=O)c1ccc(F)c(F)c1Nc1ccc(I)cc1F |r|
CNS(=O)(=O)Nc1cccc(Oc2cc(F)cc(Nc3ccc(I)cc3F)c2C(N)=O)c1
CC(C)S(=O)(=O)Nc1cccc(Oc2cncc(Nc3ccc(I)cc3F)c2C(N)=O)c1
NC(=O)c1c(Nc2ccc(I)cc2F)cncc1Oc1cccc(NS(=O)(=O)C2CC2)c1
CC1=C(C(=O)Oc2c1ccc(c2)Oc3ncccn3)Cc4ccnc(c4F)NS(=O)(=O)NC
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1cc(Cl)cc(NS(C)(=O)=O)c1)C(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1cccc(NS(C)(=O)=O)c1F)C(C)C |r|
CCCS(=O)(=O)Nc1cc(Cl)cc(c1)-c1nn(cc1-c1ccnc(NC[C@H](C)NC(=O)OC)n1)C(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1c(F)ccc(NS(C)(=O)=O)c1F)C(C)C |r,wD:5.5,(-7.74,6.48,;-6.41,5.71,;-5.08,6.48,;-5.08,8.02,;-3.74,5.71,;-3.74,4.17,;-5.08,3.4,;-2.41,3.4,;-2.41,1.86,;-1.08,1.09,;.26,1.86,;1.59,1.09,;1.59,-.45,;.26,-1.22,;-1.08,-.45,;.26,-2.76,;-.99,-3.66,;-.51,-5.13,;1.03,-5.13,;1.5,-3.66,;2.99,-3.27,;3.39,-1.78,;2.3,-.69,;4.88,-1.38,;5.97,-2.47,;5.57,-3.96,;6.66,-5.05,;6.26,-6.53,;5.86,-8.02,;4.77,-6.13,;7.74,-6.93,;4.08,-4.36,;3.68,-5.84,;-1.28,-6.46,;-.51,-7.8,;-2.82,-6.46,)|
CCCS(=O)(=O)Nc1ccc(F)c(-c2nn(cc2-c2ccnc(NC[C@H](C)NC(=O)OC)n2)C(C)C)c1F |r,wD:25.26,(6.55,-9.31,;6.95,-7.82,;5.86,-6.73,;6.26,-5.24,;4.77,-4.85,;7.74,-5.64,;6.66,-3.76,;5.57,-2.67,;5.97,-1.18,;4.88,-.09,;3.39,-.49,;2.3,.6,;2.99,-1.98,;1.5,-2.38,;1.03,-3.84,;-.51,-3.84,;-.99,-2.38,;.26,-1.47,;.26,.07,;1.59,.84,;1.59,2.38,;.26,3.15,;-1.08,2.38,;-2.41,3.15,;-2.41,4.69,;-3.74,5.46,;-5.08,4.69,;-3.74,7,;-5.08,7.77,;-5.08,9.31,;-6.41,7,;-7.74,7.77,;-1.08,.84,;-1.28,-5.17,;-.51,-6.51,;-2.82,-5.17,;4.08,-3.07,;3.68,-4.55,)|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1cc(Cl)cc(NS(C)(=O)=O)c1F)C(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1cc(F)cc(NS(C)(=O)=O)c1F)C(C)C |r|
CCn1cc(c(n1)-c1cc(Cl)cc(NS(C)(=O)=O)c1F)-c1ccnc(NC[C@H](C)NC(=O)OC)n1 |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1cc(C)cc(NS(C)(=O)=O)c1F)C(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1cc(C)cc(NS(C)(=O)=O)c1Cl)C(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1cc(F)cc(NS(C)(=O)=O)c1Cl)C(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1ccnc(NS(C)(=O)=O)c1F)C(C)C |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1ccc(F)c(NS(C)(=O)=O)c1F)C(C)C |r|
COC(=O)N[C@H](C)CNc1nccc(n1)-c1cn(nc1-c1cc(Cl)cc(NS(C)(=O)=O)c1F)C(C)C |r|
CCS(=O)(=O)Nc1c(F)ccc(-c2nn(cc2-c2ccnc(NC[C@H](C)NC(=O)OC)n2)C(C)C)c1F |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1cc(NS(C)(=O)=O)c(C)c(OC)c1)C(C)C |r|
CC(C)n1cc(c(n1)-c1cc(Cl)cc(NS(C)(=O)=O)c1F)-c1ccnc(NCCN(C)C)n1
CNc1nccc(n1)-c1cn(nc1-c1cc(Cl)cc(NS(C)(=O)=O)c1F)C(C)C
CC(C)n1cc(c(n1)-c1cc(Cl)cc(NS(C)(=O)=O)c1F)-c1ccnc(N)n1
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1c[nH]nc1-c1cc(Cl)cc(NS(C)(=O)=O)c1F |r|
COC(=O)NC[C@H](C)Nc1nccc(n1)-c1cn(nc1-c1cc(Cl)cc(NS(C)(=O)=O)c1F)C(C)C |r|
CCCS(=O)(=O)Nc1c(F)ccc(-c2nn(cc2-c2ccnc(NC[C@H](C)NC(=O)OC)n2)C(C)C)c1F |r|
COC(=O)N[C@@H](C)CNc1nccc(n1)-c1cn(nc1-c1cc(F)cc(NS(=O)(=O)C2CC2)c1F)C(C)C |r|
Cc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(COC)c23)c1F
CC(C)CS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(C)c23)c1F
COc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)CC(C)C)c3F)c12
CCCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(OC)c23)c1F
CCOc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CCCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(C)c23)c1F
CCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(OC)c23)c1F
CC(C)c1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(C)c23)c1F
COc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(C)C)c3F)c12
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(NC3CC3)c12
Oc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(NC3CCOCC3)c12
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(CC(C)C)c23)c1F
CC(C)Cc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(Cl)c12
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(N3CCOCC3)c12
COc1ccc(cn1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(OC)c23)c1F
CCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(C)c23)c1F
CC(C)CNc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(OC3CCOCC3)c12
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(O)c23)c1F
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(C#N)c12
CCNc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
COc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4cc(C)cc(C)c4)c3F)c12
CNc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
Cc1cc(C)cc(c1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(C)c23)c1F
CC(C)COc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CC(C)c1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CCCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(O)c23)c1F
Nc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CCCNc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(Cl)c23)c1F
CCCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(Cl)c23)c1F
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(NC3CCCC3)c12
COc1ccc(cc1F)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(C)c23)c1F
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(Nc3ccccc3)c12
CCCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(OCC)c23)c1F
CC(C)Nc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CCCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(NC4CC4)c23)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(NC4CC4)c23)c1F
CCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(NC(C)C)c23)c1F
OCCNc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CC(C)Nc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(C)C)c3F)c12
CC(C)Nc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4cc(C)cc(C)c4)c3F)c12
CCCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(NC4CCOCC4)c23)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(NC4CCOCC4)c23)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(Nc4ccccc4)c23)c1F
CN(C)c1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(NC3COC3)c12
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(NC(C)C)c23)c1F
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(NCC3CC3)c12
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(OCC3CC3)c12
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(NC3CCOC3)c12
CCCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(NC(C)C)c23)c1F
CCCc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(NC4COC4)c23)c1F
CN1CCC(CC1)Nc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
COCCNc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CN(C)CCNc1ncnc2[nH]cc(C(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(cc4)C(F)(F)F)c3F)c12
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncnc(NC4COC4)c23)c1F
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncnc(N3CCCC3)c12
Cn1cc(Nc2ncnc3[nH]cc(C(=O)c4c(F)ccc(NS(=O)(=O)c5ccc(cc5)C(F)(F)F)c4F)c23)cn1
CCn1cc(Nc2ncnc3[nH]cc(C(=O)c4c(F)ccc(NS(=O)(=O)c5ccc(cc5)C(F)(F)F)c4F)c23)cn1
CCCS(=O)(=O)Nc1ccc(F)c(C=O)c1F
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1C=O
Fc1ccc(NS(=O)(=O)c2ccccc2)c(F)c1C=O
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
CCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(on4)C(C)(C)C)ccc3F)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(on4)C(C)(C)C)ccc3Cl)c2cc1OC
CCOc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCOC
CCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCC
CC(C)(C)c1cc(NC(=O)Nc2cccc(Oc3ncnc4cc5OCCOc5cc34)c2)no1
COCCOc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCCCC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCC(CO)CC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCN(C)CC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCN(CCO)CC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCOCC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCN(C)CC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCOCC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCCCC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCC(CO)CC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCN(CC1)S(C)(=O)=O
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCS(=O)(=O)CC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCOCC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCN(C)CC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCC(CO)CC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCN(CCO)CC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCC(O)C1 |w:39.43|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCN(CC1)S(C)(=O)=O
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CC[C@H](O)C1 |r|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CC[C@@H](O)C1 |r|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCOCC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCN(C)CC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCC(CO)CC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCN(CCO)CC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCS(=O)(=O)CC1
COCCOc1ccc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2c1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCS(C)(=O)=O
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)F)c3)c2cc1OCCCS(C)(=O)=O
COCCOc1ccc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2c1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCS(C)(=O)=O
COCCOc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
CC(C)(C)c1cc(NC(=O)Nc2cccc(Sc3ncnc4cc(F)c(F)cc34)c2)no1
COc1ccc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2c1
COc1ccc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2c1
CCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
CCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCOC
CC(C)(C)c1cc(NC(=O)Nc2cccc(Sc3ncnc4cc5OCCOc5cc34)c2)no1
COc1cc(OC2CCOCC2)c2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2c1
CCOc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCCCC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCC(CO)CC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCN(C)CC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCN(CC1)S(C)(=O)=O
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCN(CCO)CC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCS(=O)(=O)CC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCCN1CCOCC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCCCC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCC(CO)CC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCN(C)CC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCN(CCO)CC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCN(CC1)S(C)(=O)=O
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCOCC1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCS(=O)(=O)CC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCOCC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCN(C)CC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCC(CO)CC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCN(CCO)CC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCCCC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCN(CC1)S(C)(=O)=O
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCOCC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCCCC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCN(CC1)S(C)(=O)=O
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCN(C)CC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCC(CCO)CC1
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCN1CCC(CO)CC1
COCCOc1ccc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2c1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCS(C)(=O)=O
COc1cc2nc(Cl)nc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
CC(C)(C)c1cc(NC(=O)Nc2cccc(Sc3ncnc4ccc(OCCCN5CCS(=O)(=O)CC5)cc34)c2)no1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OCCN1CCS(=O)(=O)CC1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Oc3ncnc4ccc(cc34)-c3ccc(CNCCS(C)(=O)=O)o3)c2)no1
COc1cc(OC2CCOCC2)c2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2c1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1O
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1O[C@H]1CCNC1 |r|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1O[C@H]1CCN(C)C1 |r|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1O[C@@H]1CCNC1 |r|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1O[C@@H]1CCN(C)C1 |r|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OC[C@H](O)CN1CCN(C)CC1 |r|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCC1CCNCC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCC1CCN(C)CC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1O[C@H]1CCN(CC(F)F)C1 |r|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1O[C@H]1CCN(CC(F)(F)F)C1 |r|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OC1CCN(CC(F)F)CC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1O
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1O[C@H]1CCN(C1)C(=O)OC(C)(C)C |r|
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC1CCN(C)C1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1O[C@H]1CCN(CC(F)F)C1 |r|
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC[C@@H](O)CN1CCN(C)CC1 |r|
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC[C@H](O)CN1CCN(C)CC1 |r|
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)-c4ccccc4)c3)c2cc1OC
COc1cc(NC(=O)Nc2cccc(Sc3ncnc4cc(OC)c(OC)cc34)c2)cc(c1)C(F)(F)F
COc1cc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)cc(c1)C(F)(F)F
COCCOc1cc(NC(=O)Nc2cccc(Oc3ncnc4cc(OCCOC)c(OC)cc34)c2)cc(c1)C(F)(F)F
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cccc(c4)C(C)(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cccc(c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cccc(c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C4CCOCC4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C4CC4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C#N)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C4(C)CC4)c3)c2cc1OC
COCC(C)(C)c1cc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)on1
COCCOc1cc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)cc(c1)C(F)(F)F
COCC(C)(C)c1cc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)no1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)CO)c3)c2cc1OC
COc1cc2cccc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C4CCCC4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(CC(F)(F)F)nn4-c4ccccc4)c3)c2cc1OC
COc1ccc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)cc1C(F)(F)F
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccc(OC)c(c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(Cl)cc(c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(ccn4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(ccc4Cl)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4nccc(n4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cccc(c4)C(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(ncn4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)ccc1C(F)(F)F
COCCOc1cc(NC(=O)Nc2cccc(Sc3ncnc4cc(OC)c(OC)cc34)c2)ccc1C(F)(F)F
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(cc(c4)C(F)(F)F)C(=O)N4CCOCC4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccc(c(F)c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(CN5CCOCC5)cc(c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C4(CCC4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C4(CCC4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(CF)CF)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(CF)CF)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(CF)CF)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C4CCCC4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4C)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(n(C)n4)C(F)(F)F)c3)c2cc1OC
CCOC(=O)Cn1nc(cc1NC(=O)Nc1cccc(Oc2ncnc3cc(OC)c(OC)cc23)c1)C(C)(C)C
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(CF)CF)c3)c2cc1OC
CCOC(C)(C)c1cc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)n(n1)-c1ccccc1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(n(n4)-c4ccccc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(n(n4)-c4ccccc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(F)cc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccc(cc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4ccc(cc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccc(Cl)cc4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccc(OC(F)(F)F)cc4)c3)c2cc1OC
COc1cccc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)c1
CCOc1cccc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)c1
COc1ccc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)cc1Cl
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cccc(c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccccc4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cccc(c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4ccc(c(F)c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(CN5CCOCC5)cc(c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4ccc(c(OC)c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(CF)CF)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4C)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(n(C)n4)C(F)(F)F)c3)c2cc1OC
CCOC(=O)Cn1nc(cc1NC(=O)Nc1cccc(Sc2ncnc3cc(OC)c(OC)cc23)c1)C(C)(C)C
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(CF)CF)c3)c2cc1OC
CCCOC(C)(C)c1cc(NC(=O)Nc2cccc(Sc3ncnc4cc(OC)c(OC)cc34)c2)n(n1)-c1ccccc1
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(F)cc4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc(NC(=O)Nc2cccc(Sc3ncnc4cc(OC)c(OC)cc34)c2)cc(c1)C(F)(F)F
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C4CCCC4)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)-c4ccccc4)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(cc(c4)C(F)(F)F)C(=O)N4CCOCC4)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C4CCCC4)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(n(C)n4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4C)C(C)(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(F)F)c3)c2cc1OC
CCOC(C)(C)c1cc(NC(=O)Nc2cccc(Oc3ncnc4cc(OCCOC)c(OC)cc34)c2)n(n1)-c1ccccc1
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(CF)CF)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C4CC4)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C4CCOCC4)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)COC)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C4CCCC4)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4C)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccc(c(F)c4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4ccc(c(OC)c4)C(F)(F)F)c3)c2cc1OC
CCOC(=O)Cn1nc(cc1NC(=O)Nc1cccc(Oc2ncnc3cc(OCCOC)c(OC)cc23)c1)C(C)(C)C
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(n(n4)-c4ccccc4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(F)cc4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(CF)CF)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(CF)CF)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4ccc(c(F)c4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4ccc(c(OC)c4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C4CCCC4)c3)c2cc1OC
CCOC(=O)Cn1nc(cc1NC(=O)Nc1cccc(Sc2ncnc3cc(OCCOC)c(OC)cc23)c1)C(C)(C)C
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(CF)CF)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4C)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(n(C)n4)C(F)(F)F)c3)c2cc1OC
CCOC(C)(C)c1cc(NC(=O)Nc2cccc(Sc3ncnc4cc(OCCOC)c(OC)cc34)c2)n(n1)-c1ccccc1
COCCOc1cc2ncnc(Sc3cccc(NC(=O)NC4=CC(=NC4c4ccc(F)cc4)C(F)(F)F)c3)c2cc1OC |c:24,t:22|
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C(F)(F)F)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(n(n4)-c4ccccc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)c2cc1OCCCN1CCS(=O)(=O)CC1
COc1ccc(NC(=O)Nc2cccc(Sc3ncnc4cc(OC)c(OCCCN5CCS(=O)(=O)CC5)cc34)c2)cc1C(F)(F)F
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(C)C)c3)c2cc1OCCOC
COc1cc2c(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)ncnc2cc1OCCN1CCOCC1
COc1ccc(NC(=O)Nc2cccc(Sc3ncnc4cc(OCCN5CCOCC5)c(OC)cc34)c2)cc1C(F)(F)F
COc1ccc(NC(=O)Nc2cccc(Oc3ncnc4cc(OCCN5CCOCC5)c(OC)cc34)c2)cc1C(F)(F)F
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)ncnc2cc1OCCN1CCOCC1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cnn(c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(S(=O)c3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)NC4=CC(=CC4)C(C)(C)CO)c3)c2cc1OC |c:21,t:19|
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)ncnc2cc1OCCCN1CCS(=O)(=O)CC1
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)ncnc2cc1O
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)c2cc1O
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C(F)(F)F)c3)c2cc1OC
CCOc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C(F)(F)F)c3)ncnc2cc1OC
CCOc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C(F)(F)F)c3)ncnc2cc1OC
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C(F)(F)F)c3)ncnc2cc1O
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C(F)(F)F)c3)c2cc1O
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C(F)(F)F)c3F)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(on4)C(C)(C)C(F)(F)F)ccc3F)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(C)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(no4)C(C)(C)F)c(F)cc3F)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(on4)C(C)(C)C)c(F)cc3F)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)F)c(F)cc3F)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C(C)(C)C)c(F)cc3F)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c(F)cc3F)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C(C)(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cccc(c4)C(C)(C)C#N)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cccc(c4)C(C)(C)C#N)c3)c2cc1OC
COCCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cccc(c4)C(C)(C)C#N)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4C)C(C)(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cccc(C)c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4cccc(C)c4)C(C)(C)C)c3)c2cc1OC
COCCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4cccc(C)c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C(C)(C)C)c3C)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c3C)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3C)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)F)c3C)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3C)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(no4)C(C)(C)F)ccc3F)c2cc1OC
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(on4)C(C)(CF)CF)ccc3F)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c3F)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3F)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(CF)CF)c3F)c2cc1OC
COc1cc2ncnc(Oc3ccc(Cl)c(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3ccc(Cl)c(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3ccc(Cl)c(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3ccc(Cl)c(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)CN4CCOCC4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cnccc4C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cccnc4C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)CF)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C#N)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C#N)c3)c2cc1OC
COc1cc2nc(Cl)nc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cccnc4)C(C)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)nc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cc[nH]c(=O)c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cncc(F)c4)C(C)C)c3)c2cc1OC
COc1ccc(cc1)-n1nc(cc1NC(=O)Nc1cccc(Oc2ncnc3cc(OC)c(OC)cc23)c1)C(C)(F)F
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cncc(F)c4)C(C)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(=O)[nH]c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccnc(C)c4)C(C)(C)C)c3)c2cc1OC
CCn1nc(cc1NC(=O)Nc1cccc(Sc2ncnc3cc(OC)c(OC)cc23)c1)C(C)(C)C
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cccnc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4cccnc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cncc(F)c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4cncc(F)c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(cc4)C#N)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(cc4)C#N)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4C4CCCCC4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4C4CCCCC4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4CC(C)C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4CC(C)C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4C(C)C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4C(C)C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccncc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccncc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cccc(C)c4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4Cl)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4Cl)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccn4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccn4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C4(CC4)C(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(C)cc4)C4(CC4)C(F)(F)F)c3)c2cc1OC
COc1ccc(cc1)-n1nc(cc1NC(=O)Nc1cccc(Oc2ncnc3cc(OC)c(OC)cc23)c1)C(C)C
COc1ccc(cc1)-n1nc(cc1NC(=O)Nc1cccc(Sc2ncnc3cc(OC)c(OC)cc23)c1)C(C)C
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cccnc4)C(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4cccnc4)C(C)C)c3)c2cc1OC
CCc1cc(NC(=O)Nc2cccc(Oc3ncnc4cc(OC)c(OC)cc34)c2)n(n1)-c1ccccc1
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C4CC4)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C4CC4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C4CCC4)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C4CCC4)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4Cc4ccccc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4Cc4ccccc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cccc(F)c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4cccc(F)c4)C(C)(C)C)c3)c2cc1OC
COc1ccc(cc1)-n1nc(cc1NC(=O)Nc1cccc(Oc2ncnc3cc(OC)c(OC)cc23)c1)C(C)(C)C
COc1ccc(cc1)-n1nc(cc1NC(=O)Nc1cccc(Sc2ncnc3cc(OC)c(OC)cc23)c1)C(C)(C)C
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cccc(Cl)c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4cccc(Cl)c4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(Cl)cc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(Cl)cc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3ccc(F)c(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3ccc(F)c(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(cc4)C(C)(C)C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(cc4)C(C)(C)C)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4F)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4F)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccc(cc4)C(F)(F)F)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccc(cc4)C(F)(F)F)C(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4C(F)(F)F)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4C(F)(F)F)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C4(CC4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C4(CC4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4cccc(c4)C(F)(F)F)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4cccc(c4)C(F)(F)F)C(C)(C)C)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(C)C#N)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C(F)(F)F)c3)c2cc1OC
COc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C4(CC4)C(F)(F)F)c3)c2cc1OC
CCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)F)c3)c2cc1OC
CCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)c2cc1OC
CCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(CF)CF)c3)c2cc1OC
CCOc1cc2ncnc(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c3)c2cc1OC
CCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(CF)CF)c3)c2cc1OC
CCOc1cc2ncnc(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)c2cc1OC
CCOc1cc2c(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c3)ncnc2cc1OC
CCOc1cc2c(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)F)c3)ncnc2cc1OC
CCOc1cc2c(Oc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)ncnc2cc1OC
CCOc1cc2c(Oc3cccc(NC(=O)Nc4cc(on4)C(C)(CF)CF)c3)ncnc2cc1OC
CCOc1cc2c(Sc3cccc(NC(=O)Nc4cc(no4)C(C)(C)F)c3)ncnc2cc1OC
CCOc1cc2c(Sc3cccc(NC(=O)Nc4cc(on4)C(C)(CF)CF)c3)ncnc2cc1OC
COc1cc2c(Oc3cccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)F)c3)ncnc2cc1OCCN1CCOCC1
COc1cc2ncnc(Oc3cc(NC(=O)Nc4cc(nn4-c4ccccc4)C(F)(F)F)ccc3F)c2cc1OC
COc1ccc(cn1)-n1nc(cc1NC(=O)Nc1cccc(Oc2ncnc3cc(OC)c(OC)cc23)c1)C(C)(C)C
CCc1cc(NC(=O)Nc2cccc(Sc3ncnc4cc(OC)c(OC)cc34)c2)n(n1)-c1ccccc1
CCn1nc(C#Cc2cc(ccc2C)C(=O)Nc2ccc(CN3CCN(C)CC3)c(c2)C(F)(F)F)c2c(N)ncnc12
CN1CCC(CC1)n1nc(C#Cc2cc(NC(=O)c3cccc(c3)C(F)(F)F)ccc2C)c2c(N)ncnc12
Cc1ccc(NC(=O)c2ccc(C)c(c2)C(F)(F)F)cc1C#Cc1nn([C@H]2CC[C@H](O)CC2)c2ncnc(N)c12 |r,wU:26.27,wD:29.31,(-5.46,5.4,;-3.98,5.8,;-3.58,7.29,;-2.09,7.69,;-1,6.6,;.49,7,;1.57,5.91,;1.18,4.42,;3.06,6.31,;3.46,7.79,;4.95,8.19,;6.04,7.1,;7.53,7.5,;5.64,5.62,;4.15,5.22,;6.73,4.53,;8.22,4.93,;6.33,3.04,;7.82,3.44,;-1.4,5.11,;-2.89,4.71,;-3.29,3.22,;-3.68,1.74,;-4.08,.25,;-3.18,-1,;-4.08,-2.24,;-3.68,-3.73,;-2.2,-4.13,;-1.8,-5.62,;-2.89,-6.7,;-2.49,-8.19,;-4.38,-6.31,;-4.77,-4.82,;-5.55,-1.77,;-6.88,-2.54,;-8.22,-1.77,;-8.22,-.23,;-6.88,.54,;-6.88,2.08,;-5.55,-.23,)|
CC1Nc2nc(NC(=O)c3ccc[n+](C)c3)[nH]c(=O)c2N(C1C)C(=O)c1ccc[n+](C)c1
Cn1c2[nH]c(=S)n(Cc3ccc(Cl)cc3)c2c(=O)[nH]c1=O
CSc1nc2n(C)c(=O)[nH]c(=O)c2n1Cc1ccccc1
C\C(Cl)=C/CSc1nc2n(C)c(=O)n(Cc3ccccc3)c(=O)c2n1Cc1ccccc1
Cn1c2nc(SCCO)n(Cc3ccccc3)c2c(=O)n(Cc2ccccc2)c1=O
Cn1c2nc(SCC(N)=O)n(Cc3cccc(Br)c3)c2c(=O)[nH]c1=O
CC(N=Nc1nc2n(C)c(=O)[nH]c(=O)c2n1Cc1ccccc1)c1ccc(cc1)[N+]([O-])=O |w:3.3|
Cc1cc(C)n(n1)-c1nc2n(C)c(=O)n(C)c(=O)c2n1Cc1ccccc1
C\C(Cl)=C/CSc1nc2n(C)c(=O)[nH]c(=O)c2n1CC(O)CCc1ccccc1
Cn1c2nc(N=NCc3cccc(c3)[N+]([O-])=O)n(CC=C)c2c(=O)[nH]c1=O |w:5.4|
CC(N=Nc1nc2n(C)c(=O)[nH]c(=O)c2n1C\C=C(\C)Cl)c1ccc(cc1)[N+]([O-])=O |w:3.3|
Cn1c2nc(N=NCc3cccc(c3)[N+]([O-])=O)n(Cc3ccccc3)c2c(=O)[nH]c1=O |w:5.4|
Cn1c2nc(N=NCc3ccc(cc3)[N+]([O-])=O)n(Cc3ccccc3)c2c(=O)[nH]c1=O |w:5.4|
CC(N=Nc1nc2n(C)c(=O)[nH]c(=O)c2n1Cc1ccccc1)c1ccccc1 |w:3.3|
CNC(=O)c1cc(ccn1)Oc2ccc(cc2)NC(=O)Nc3ccc(c(c3)C(F)(F)F)Cl
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccc2C(CCc2c1)N=O)-c1ccncc1
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(Cl)cc23)c1F
O=NC1CCc2cc(ccc12)-c1c[nH]nc1-c1ccncc1
Cn1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
Cn1ncc(c1-c1ccncc1)-c1ccc2C(CCc2c1)N=O
CCn1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
O=NC1CCc2cc(ccc12)-c1cn(nc1-c1ccncc1)C1CCCC1
O[C@H]1CCC[C@H]1n1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O |r|
O[C@@H]1CCC[C@H]1n1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O |r|
O[C@H]1CCC[C@H](C1)n1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O |r|
O[C@@H]1CCC[C@H](C1)n1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O |r|
COCCn1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
OCCn1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
OCCCn1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
OCC(O)Cn1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
OCC(CO)n1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
NCCn1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
CN(C)CCn1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
NCCCn1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
CN(C)CCCn1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
O=NC1CCc2cc(ccc12)-c1cn(nc1-c1ccncc1)C1CCNCC1
CN1CCC(CC1)n1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
O=NC1CCc2cc(ccc12)-c1cn(nc1-c1ccncc1)C1CCOCC1
O=NC1CCc2cc(ccc12)-c1cn(CC2CCNCC2)nc1-c1ccncc1
O=NC1CCc2cc(ccc12)-c1cn(CC2CCCNC2)nc1-c1ccncc1
CNC1CCCC(C1)n1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
Cn1cc(c(n1)-c1ccc2n(C)ncc2c1)-c1ccc2C(CCc2c1)N=O
Cn1cc(c(n1)-c1cccnc1)-c1ccc2C(CCc2c1)N=O
Cn1cc(c(n1)-c1cnco1)-c1ccc2C(CCc2c1)N=O
Cn1cc(c(n1)-c1ccnc(N)c1)-c1ccc2C(CCc2c1)N=O
Cn1cc(c(n1)-c1ccncc1O)-c1ccc2C(CCc2c1)N=O
Cn1cc(c(n1)-c1ccncn1)-c1ccc2C(CCc2c1)N=O
Cn1cc(c(n1)-c1ccncc1)-c1ccc(cc1)C(=N)NO
Cn1cc(c(n1)-c1ccncc1)-c1ccc2C(NO)=NCc2c1 |c:20|
Cn1cc(c(n1)-c1ccncc1)-c1ccc2C(NO)=NCCc2c1 |c:20|
Cn1cc(c(n1)-c1ccncc1)-c1ccc(cc1)-c1cc[nH]n1
Cc1c[nH]nc1-c1ccc(cc1)-c1cn(C)nc1-c1ccncc1
Cn1cc(c(n1)-c1ccncc1)-c1ccc-2c(Cc3c[nH]nc-23)c1
Cn1cc(c(n1)-c1ccncc1)-c1ccc2C(=O)NCc2c1
Cn1cc(c(n1)-c1ccncc1)-c1ccc2cn[nH]c2c1
Oc1cc(ccc1Cl)-c1[nH]c(nc1-c1ccncc1)-c1ccccc1
CC(COc1nccc(n1)-c1nc(c([nH]1)-c1ccc2C(CCc2c1)N=O)-c1ccncc1)N(C)C
CC(C)(CN)c1nc(c([nH]1)-c1ccc2C(CCc2c1)N=O)-c1ccncc1
O=NC1CCc2cc(ccc12)-c1[nH]c(nc1-c1ccncc1)C1CCNCC1
COCCN1CCC(CC1)c1nc(c([nH]1)-c1ccc2C(CCc2c1)N=O)-c1ccncc1
O=NC1CCc2cc(ccc12)-c1[nH]c(CN2CCOCC2)nc1-c1ccncc1
O=NC1CCc2cc(ccc12)-c1[nH]c(nc1-c1ccncc1)C(=O)NCCN1CCOCC1
CN(C)Cc1cccc(NC(=O)c2nc(c([nH]2)-c2ccc3C(CCc3c2)N=O)-c2ccncc2)c1
CN(C)CCOc1ccc(cc1)-c1cc(c(o1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
CN(C)CCOc1ccc(cc1)-c1cc(c([nH]1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
CN(C)CCOc1ccc(cc1)-c1cc(c(o1)-c1ccc2C(CCc2c1)N=O)-c1ccncc1
CN(C)CCOc1ccc(cc1)-c1cc(c([nH]1)-c1ccc2C(CCc2c1)N=O)-c1ccncc1
O=NC1CCc2cc(ccc12)-c1cc(oc1-c1ccncc1)C1CCNCC1
COCCN1CCC(CC1)c1cc(c(o1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
CN(C)CCNC(=O)c1cc(c(o1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
O=NC1CCc2cc(ccc12)-c1cc(CN2CCOCC2)oc1-c1ccncc1
CC1(CNc2c1ccc(c2)NC(=O)c3cccnc3NCc4ccncc4)C
CCN1CCN(Cc2ccc(NC(=O)Nc3ccc(Oc4cc(NC)ncn4)cc3)cc2C(F)(F)F)CC1
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(OCCN2CCOCC2)c2ccccc12)C(C)(C)C
Cn1c(Nc2ccc(cc2)C(F)(F)F)nc2cc(Oc3ccnc(c3)-c3ncc([nH]3)C(F)(F)F)ccc12
Cc1cccc(c1NC(=O)c2cnc(s2)Nc3cc(nc(n3)C)N4CCN(CC4)CCO)Cl
CN(c1ccc2c(C)n(C)nc2c1)c1ccnc(Nc2ccc(C)c(c2)S(N)(=O)=O)n1
Oc1cccc(c1)-c1nc(N2CCOCC2)c2oc3ncccc3c2n1
Oc1ccc(cc1)-c1nc(c([nH]1)-c1ccc(F)cc1)-c1ccncc1
CS(=O)c1ccc(cc1)-c1nc(c([nH]1)-c1ccc(F)cc1)-c1ccncc1
CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)CC1
Cc1nc(Cl)cc(Nc2cccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)c2)n1
Cc1nc(Nc2cccc(NC(=O)Nc3ccc(F)c(Cl)c3)c2)cc(n1)N1CCOCC1
Cc1nc(Nc2cccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)c2)cc(n1)N1CCOCC1
CN1CCN(CC1)c1cc(Nc2cccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)c2)nc(C)n1
CN(c1cccc(NC(=O)Nc2ccc(F)c(Cl)c2)c1)c1cc(nc(C)n1)N1CCOCC1
CN(c1cccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c1)c1cc(nc(C)n1)N1CCOCC1
CN(c1cccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c1)c1cc(nc(C)n1)N1CCN(C)CC1
CCN1CCN(Cc2ccc(NC(=O)c3cccc(c3)-c3ccc4nc(NC(=O)C5CC5)sc4n3)cc2C(F)(F)F)CC1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccccc3)c2c1
COc1cccc(c1)-c1ccc2ncnc(Nc3ccccc3)c2c1
Oc1ccc(cc1)-c1ccc2ncnc(Nc3ccccc3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(O)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(F)c(Cl)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(F)cc3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(Cl)cc3F)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(C)cc3F)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(c3)C(F)(F)F)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(O)cc3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(F)cc3F)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(Cl)cc3O)c2c1
COc1cccc(Nc2ncnc3ccc(cc23)-c2ccc(O)c(OC)c2)c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccccc3O)c2c1
CCS(=O)(=O)Nc1ccc(cc1)-c1ccc2ncnc(Nc3ccccc3)c2c1
COc1ccc(Nc2ncnc3ccc(cc23)-c2ccc(O)c(OC)c2)cc1O
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(c3)S(N)(=O)=O)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(C)c(O)c3)c2c1
COc1cc(ccc1O)-c1cc2c(Nc3cccc(O)c3)ncnc2cc1OC
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccccc3C(N)=O)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(cc3O)C(O)=O)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(c3)C(N)=O)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(c3)[N+]([O-])=O)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(N)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc4OCOc4c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc4cn[nH]c4c3)c2c1
COc1cc(ccc1O)-c1cc2c(Nc3ccc(C)c(O)c3)ncnc2cc1OC
COc1cc(ccc1O)-c1cc2c(Nc3cc(O)ccc3Cl)ncnc2cc1OC
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(NC(C)=O)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(NC(=O)C(F)(F)F)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(cc3)S(N)(=O)=O)c2c1
COc1cc2ncnc(Nc3cccc(O)c3)c2cc1-c1ccc(O)cc1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(F)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(O)c3C)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc4nc[nH]c4c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(NS(C)(=O)=O)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cc(O)ccc3F)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cc(O)ccc3Cl)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(O)c3Cl)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cc(O)c(Cl)cc3Cl)c2c1
Oc1ccc(cc1)-c1ccc2ncnc(Nc3cccc(O)c3)c2c1
Oc1cccc(Nc2ncnc3ccc(cc23)-c2cccc(O)c2)c1
COc1ccc(cc1)-c1ccc2ncnc(Nc3cccc(O)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc4nn[nH]c4c3)c2c1
COc1cccc(c1)-c1ccc2ncnc(Nc3cccc(O)c3)c2c1
COc1cc2ncnc(Nc3cccc(O)c3)c2cc1-c1ccc(N)cc1
Nc1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
CC(=O)Nc1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
CS(=O)(=O)Nc1cccc(c1)-c1ccc2ncnc(Nc3cccc(O)c3)c2c1
CS(=O)(=O)Nc1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1cccc(-c2ccc3ncnc(Nc4cccc5[nH]ncc45)c3c2)c1F
COc1ccc(cc1F)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(cc1Cl)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(c(C)c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(cc1C)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
Fc1ccc(cc1Cl)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
Clc1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
Fc1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc4nn[nH]c34)c2c1
COc1cc(ccc1F)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
Fc1ccc(cc1F)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
N(c1cccc2[nH]ncc12)c1ncnc2ccc(cc12)-c1ccccc1
FC(F)(F)c1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
[C-]#[N+]c1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(cc1OC)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
CN(C)c1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
Fc1ccccc1-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
[O-][N+](=O)c1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
CCOc1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
OCc1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
CS(=O)(=O)Nc1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
C1Oc2ccc(cc2O1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
NC(=O)c1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(cc1C=O)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc4n(C)ncc34)c2c1
COc1cc(ccc1O)-c1ccc2nccc(Nc3cccc(O)c3)c2c1
COc1cc(ccc1O)-c1ccc2nccc(Nc3cc(O)ccc3F)c2c1
N#Cc1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1cc(ccc1O)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
Cc1ccc(F)cc1-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1cccc(-c2ccc3ncnc(Nc4cccc5[nH]ncc45)c3c2)c1OC
CN(C)c1ccc(cc1)-c1ccc2ncnc(Nc3cccc(O)c3)c2c1
O=S(=O)Nc1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
CCS(=O)(=O)Nc1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
CCCS(=O)(=O)Nc1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
CS(=O)(=O)c1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1cccc(-c2ccc3nccc(Nc4cccc5[nH]ncc45)c3c2)c1F
COc1ccc(cc1F)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(cc1OC)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
N#Cc1cccc(c1)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(cc1Cl)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(cc1C=O)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
NC(=O)c1cccc(c1)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc(OC(F)F)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccccc3F)c2c1
CS(=O)(=O)c1ccc(cc1)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
Nc1ccc(cc1)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
CCCS(=O)(=O)Nc1cccc(c1)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
COc1cccc(c1)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
Oc1ccc(cc1)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
Fc1ccccc1-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc4[nH]nc(Cl)c34)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cccc4[nH]c(=O)[nH]c34)c2c1
COc1cc(ccc1O)-c1ccc2nccc(Nc3cc(NS(C)(=O)=O)ccc3F)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cc(NS(C)(=O)=O)ccc3F)c2c1
Oc1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
Oc1cccc(Nc2ncnc3ccc(cc23)-c2ccccc2)c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3c(F)cccc3F)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3c(F)ccc4[nH]ncc34)c2c1
Nc1ccc(F)c(c1)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
Nc1ccc(F)c(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
Oc1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1cccc(c1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(cc1)-c1ccc2ncnc(Nc3cccc4[nH]ncc34)c2c1
Oc1cccc(c1)-c1ccc2nccc(Nc3cccc4[nH]ncc34)c2c1
COc1ccc(cc1)-c1ccc2ncnc(Oc3cccc(O)c3)c2c1
N(c1cccc2[nH]ncc12)c1ncnc2ccc(cc12)-c1ccc2[nH]ncc2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cc(O)ccc3C)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cc(O)c(C)cc3F)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(Cl)c(O)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cc(O)c(F)cc3F)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3cc(O)c(Cl)cc3F)c2c1
Oc1cc(Nc2ncnc3ccc(cc23)-c2ccc(Cl)cc2)c(F)cc1F
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(F)c(O)c3)c2c1
COc1cc(ccc1O)-c1ccc2ncnc(Nc3ccc(F)c(O)c3F)c2c1
Oc1c(F)ccc(Nc2ncnc3ccc(cc23)-c2ccc3[nH]ncc3c2)c1F
Oc1c(F)ccc(Nc2ncnc3ccc(cc23)-c2ccc(Cl)cc2)c1F
Cc1ccc2c(Nc3ccc(Cl)cc3)nccc2c1NC(=O)c1csc2c(N)ncnc12
COc1ccc(Nc2nccc3c(NC(=O)c4csc5c(N)ncnc45)c(C)ccc23)cc1
Cc1ccc2c(Nc3cccc(Cl)c3)nccc2c1NC(=O)c1csc2c(N)ncnc12
Cc1ccc2c(Nc3ccc(OC(F)F)cc3)nccc2c1NC(=O)c1csc2c(N)ncnc12
CN(C)Cc1cc(Nc2nccc3c(NC(=O)c4csc5c(N)ncnc45)c(C)ccc23)ccc1Cl
CC(=O)c1ccc(Nc2nccc3c(NC(=O)c4csc5c(N)ncnc45)c(C)ccc23)cc1
Cc1ccc2c(Nc3ccc(F)c(Cl)c3)nccc2c1NC(=O)c1csc2c(N)ncnc12
Cc1ccc2c(c1NC(=O)c3csc4c3ncnc4N)ccnc2Nc5cccc(c5F)Cl
CNc1cc2nc(C)c(cc2cn1)-c1cc(NC(=O)NCCC(C)(C)C)ccc1F
CNc1cc2nc(C)c(cc2cn1)-c1cc(NC(=O)NCCC(C)(C)F)c(F)cc1C
CC(C)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Fc1ccc(NS(=O)(=O)c2cccc(c2)C(F)(F)F)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)c2cccs2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Fc1ccc(NS(=O)(=O)c2ccc(Cl)c(Cl)c2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)c2cc3ccccc3o2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)c2ccc(Cl)cc2F)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
[O-][N+](=O)c1ccccc1CS(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
COc1ccc(cc1OC)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Fc1ccc(NS(=O)(=O)C2CCCCC2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)c2ccc(OC(F)(F)F)cc2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(c(c1)C(F)(F)F)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Cc1c(Cl)cccc1S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Fc1ccc(NS(=O)(=O)c2ccco2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
COC(=O)c1sccc1S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Fc1ccc(NS(=O)(=O)c2ccsc2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)c2ccoc2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)C2CC2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Cc1nc(C)c(s1)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Fc1ccc(NS(=O)(=O)N2CCOCC2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Cn1cnc(c1)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Cc1ccc(o1)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Fc1ccc(NS(=O)(=O)c2occc2C2OCCO2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Cc1cc(c(C)o1)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Cc1cc(c(o1)C(F)(F)F)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Cc1cccc(Cl)c1S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Fc1ccc(cc1Cl)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Fc1ccc(NS(=O)(=O)c2cccc(Cl)c2F)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)c2cccnc2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Cc1ccccc1S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Fc1ccc(NS(=O)(=O)c2ccccc2Cl)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)c2cccc(Cl)c2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)c2ccccc2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)c2cccc3CCOc23)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)c2cccc3ccoc23)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)c2cccc3CCCOc23)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Cc1nc2ccc(cc2s1)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Cn1ccc2cc(ccc12)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Cn1ccc2c(cccc12)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Cn1ccc2cccc(c12)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Cn1cc(cn1)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Fc1ccc(NS(=O)(=O)c2ccc(Cl)s2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(ncn1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(ncn1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1=O
Cc1ccc(cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1=O)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1=O
Cc1ccc(cc1-c1cc(nc(n1)N1CCOCC1)N1CCS(=O)(=O)CC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCS(=O)(=O)CC1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1nc(cc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(cc1-c1nc(cc(n1)N1CCOCC1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2Cl)C2(CC2)C#N)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
CN(C)c1cncc(c1)C(=O)Nc1ccc(C)c(c1)-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cncc(c2)C(C)(C)C)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
CN(C)Cc1cc(cc(c1)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
CCN1CCN(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(OC(F)(F)F)c2)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)S(C)(=O)=O)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cc(no2)C(C)(C)C)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cc(on2)C(C)(C)C)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2csc(n2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)S(C)(=O)=O)N1CCOCC1
CCNc1nc(cc(n1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CC2(COC2)C1)N1CCOCC1
CNc1nc(cc(n1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(NCCO)n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCC(O)C1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)-n1ccnc1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(OCCO)n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(NS(C)(=O)=O)n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCCC1=O)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)-n1cc(nn1)C(C)(C)O)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(N)n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(NC(CO)CO)n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(OCCO)n1)N1CCOCC1
CC(=C)c1cc(nc(n1)N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
CC(=C)c1cc(nc(n1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C)N1CCOCC1
CC(C)c1cc(nc(n1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C)N1CCOCC1
CC(C)c1cc(nc(n1)N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOC(C)(C)C1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CC2(COC2)C1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CCOC[C@H]1CO |r|
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1C2CCC1COC2
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CCCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CC2CC1CO2
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)N1CC2CCC(C1)O2
C[C@@H]1CN(CCO1)c1cc(nc(n1)N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C |r|
C[C@H]1CN(CCO1)c1cc(nc(n1)N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C |r|
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(OC2CCOCC2)nc(n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1nc(nc(N2CCOCC2)c1C)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(cnn1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(cnn1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(n1)N1CCOCC1)C(F)(F)F
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(cc1-c1ccnc(c1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccnn2)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)S(C)(=O)=O)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cnccn2)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cncnc2)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnnc2)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)F)cc1-c1ccnc(c1)N1CCOCC1
CN(C)c1cc(cc(n1)N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1ccnc(c1)N1CCO[C@H](CO)C1 |r|
C[C@@H]1CO[C@H](CN(C)C)CN1c1cc(ccn1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C |r|
C[C@H]1CO[C@@H](CN(C)C)CN1c1cc(ccn1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C |r|
CN(C)c1cncc(c1)C(=O)Nc1cnc(C)c(c1)-c1ccnc(c1)N1CCOCC1
C[C@@H]1COCCN1c1cc(ccn1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C |r|
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1ccnc(c1)N1CCO[C@H](CO)C1 |r|
CNC[C@@H]1CN(CCO1)c1cc(ccn1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C |r|
CC(=O)NC[C@@H]1CN(CCO1)c1cc(ccn1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C |r|
COC(=O)NC[C@@H]1CN(CCO1)c1cc(ccn1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C |r|
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1ccnc(c1)N1CCO[C@H](CNC(=O)CO)C1 |r|
COc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1ccnc(c1)N1CCOCC1
CC(F)(F)c1cc(ccn1)C(=O)Nc1c[nH]c(=O)c(c1)-c1ccnc(c1)N1CCOCC1
FC(F)(F)c1cc(ccn1)C(=O)Nc1c[nH]c(=O)c(c1)-c1ccnc(c1)N1CCOCC1
CC(C)(C#N)c1cc(ccn1)C(=O)Nc1c[nH]c(=O)c(c1)-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N)nc(c1)N1CCOCC1
CCn1cc(cc(c1=O)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1ccnc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1ccnc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1ccnc(c1)N1CCOCC1
COc1ccc(cc1C(F)(F)F)C(=O)Nc1cnc(C)c(c1)-c1ccnc(c1)N1CCOCC1
COc1cc(ccc1F)C(=O)Nc1cnc(C)c(c1)-c1ccnc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)F)cc1-c1ccnc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1ccnc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(C)(F)F)cc1-c1ccnc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1ccnc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)S(C)(=O)=O)cc1-c1ccnc(c1)N1CCOCC1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(nc(c1)N1CCOCC1)C1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(c1)N1CCOCC1)C1CCOCC1
OCc1ccc(cc1-c1ccnc(c1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F
FC(F)c1ccc(cc1-c1ccnc(c1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F
FCc1ccc(cc1-c1ccnc(c1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(cc1-c1cc(nc(c1)N1CCOCC1)N1CCOCC1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(nc(c1)-c1cnn(C)c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1-c1cc(nc(c1)N1CCOCC1)C1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(NCCO)nc(c1)N1CCOCC1
CCn1cc(cc(c1=O)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cncc(n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1c[nH]c(=O)c(n1)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1c[nH]c(=O)c(n1)N1CCOCC1
COc1ncc(cc1-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(cn(C)c1=O)N1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(cn(C)c1=O)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(c[nH]c1=O)N1CCOCC1
COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C
COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C
COc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cnc1C
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(c1)C1CCOCC1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(OC2CCOCC2)c(c1)N1CCOCC1
CC(C)n1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C
CC(C)n1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
CC(C)Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
Cc1ccc(cc1-c1cc(N2CCOCC2)c(=O)n(C)c1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(CCO)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(CCO)c1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(CCO)c1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cnc(OCCO)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1c[nH]c(=O)c(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(CC#N)c1
C[C@H](C#N)n1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C |r|
C[C@@H](C#N)n1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C |r|
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(CCS(C)(=O)=O)c1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(CCS(C)(=O)=O)c1
C[C@H](Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C)C#N |r|
C[C@@H](Oc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C)C#N |r|
Cc1ccc(cc1-c1cc(N2CCOCC2)c(=O)n(CCS(C)(=O)=O)c1)C(=O)Nc1cccc(c1)C(F)(F)F
CCn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
CCn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C
CCn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)ccc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(F)(F)F)ccc1C
CCn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C
CCOc1ncc(cc1N1CCOCC1)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)n(C)c(=O)c1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(cc1-c1cc(N2CCOCC2)c(=O)n(C)n1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ncc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ncc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
CCn1cc(nc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cn(CC(F)F)c(=O)c(n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
CN(C)Cc1cc(cc(c1)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
CCN1CCN(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
CN(C)c1cncc(c1)C(=O)Nc1ccc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cc(cc(c2)S(C)(=O)=O)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
COc1ccc(cc1C(F)(F)F)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
COc1cc(ccc1F)C(=O)Nc1cnc(C)c(c1)-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2ccnc(c2)S(C)(=O)=O)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2)S(C)(=O)=O)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2)C(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc(N2CCOCC2)c(=O)n(C)n1
Cn1cc(cc(N2CCOCC2)c1=O)-c1cc(ccc1C(F)F)C(=O)Nc1cccc(c1)C(F)(F)F
COC(=O)NCCn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)cnc1C
COC(=O)NCCn1cc(cc(N2CCOCC2)c1=O)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
COc1cc(nc(c1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(=O)cc([nH]1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2n1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CC3CC(C2)O3)c(=O)n(C)c1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc2nccn2c(n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cn2ccnc2c(n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1nc(N2CCOCC2)c2sccc2n1
C[C@@H]1COCCN1c1nc(cn2ccnc12)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C |r|
Cc1ccc(NC(=O)c2ccnc(c2)C(C)(C)C#N)cc1-c1cc2[nH]cnc2c(n1)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2oc(=O)[nH]c2c1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc(cc2[nH]c(=O)oc12)N1CCOCC1
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1cc2[nH]cnc2c(n1)N1CCOCC1
C[C@@H]1COCCN1c1nc(cc2[nH]cnc12)-c1cc(NC(=O)c2ccnc(c2)C(C)(C)C#N)ccc1C |r|
C[C@@H]1COCCN1c1nc(cc2[nH]cnc12)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C |r|
Cc1ncc(NC(=O)c2cc(cc(c2)S(C)(=O)=O)C(F)(F)F)cc1-c1ccnc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)F)cc1-c1cc(N2CCOCC2)c(=O)n(C)c1
CCN1CCN(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1ccnc(c1)N1CCOCC1
CSc1nc(N)cc(Oc2ccc(cc2)-c2nnc(Nc3cccc(c3)C(F)(F)F)[nH]2)n1
O=C1CCc2c(Oc3ccc4CC5C(C5c4c3)c3nc4ccccc4[nH]3)ccnc2N1
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Cc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
O=C1CCc2c(Oc3ccc4CC5C(C5c4c3)c3nc4ccccc4s3)ccnc2N1
O=C1CCc2c(Oc3ccc4OC5C(C5c4c3)c3nc4ccccc4[nH]3)ccnc2N1
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
FC(F)(F)c1ccc2nc([nH]c2c1)C1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
FC(F)(F)c1ccc2nc([nH]c2c1)C1[C@@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@H]12 |r|
Clc1cc2nc([nH]c2cc1Cl)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Clc1cc2nc([nH]c2cc1Cl)C1[C@@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@H]12 |r|
Clc1cc2nc([nH]c2cc1Cl)C1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
Cc1cc2[nH]c(nc2cc1F)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Cc1cc2[nH]c(nc2cc1F)C1[C@@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@H]12 |r|
Cc1cc2[nH]c(nc2cc1F)C1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
FC(F)(F)c1cc2[nH]c(nc2cc1Cl)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
FC(F)(F)c1cc2[nH]c(nc2cc1Cl)C1[C@@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@H]12 |r|
FC(F)(F)c1cc2[nH]c(nc2cc1Cl)C1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
O=C1CCc2c(Oc3ccc4OC5C(C5c4c3)c3nc4ccc(cc4[nH]3)C#N)ccnc2N1
Fc1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Cc1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
O=C1CCc2c(Oc3ccc4OC5C(C5c4c3)c3nc4ccncc4[nH]3)ccnc2N1
FC(F)(F)c1cc(Cl)c2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Fc1cc2nc([nH]c2cc1F)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Clc1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Brc1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
FC(F)(F)Oc1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Cn1c(nc2ccccc12)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
COc1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Fc1cc2[nH]c(nc2cc1Cl)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
FC(F)(F)c1cccc2nc([nH]c12)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Fc1cccc2nc([nH]c12)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
CC(C)(C)c1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
O=C1CCc2c(Oc3ccc4OC5C(C5c4c3)c3nc4cc5CCCc5cc4[nH]3)ccnc2N1
NC(=O)c1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Cn1c(nc2ccc(cc12)C(F)(F)F)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Cn1c(nc2cc(ccc12)C(F)(F)F)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Oc3c(cccc3Oc3ccnc4NC(=O)CCc34)C12
Clc1cccc2nc([nH]c12)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Oc1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
O=C1CCc2c(Oc3ccc4OC5C(C5c4c3)c3nc4ccc(cc4[nH]3)-c3ccccc3)ccnc2N1
O=C1CCc2c(Oc3ccc4OC5C(C5c4c3)c3nc(no3)-c3ccccc3)ccnc2N1
O=C1CCc2c(Oc3ccc4OC5C(C5c4c3)c3nc(c[nH]3)-c3ccccc3)ccnc2N1
O=C1CCc2c(Oc3ccc4OC5C(C5c4c3)c3nc(c[nH]3)-c3ccncc3)ccnc2N1
Clc1ccccc1-c1c[nH]c(n1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
FC(F)(F)c1c[nH]c(n1)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
OCCn1c(nc2cc(ccc12)C(F)(F)F)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
Cc1cc(Oc2ccnc3NC(=O)CCc23)cc2C3C(Oc12)C3c1nc2ccc(cc2[nH]1)C(F)(F)F
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Oc3cc(Cl)c(Oc4ccnc5NC(=O)CCc45)cc3C12
Cc1cc2nc([nH]c2cc1F)C1C2Oc3cc(Cl)c(Oc4ccnc5NC(=O)CCc45)cc3C12
CNC(=O)c1cc(Oc2ccc3OC4C(C4c3c2)c2nc3ccc(cc3[nH]2)C(F)(F)F)ccn1
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccncn4)cc3C12
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5[nH]ccc45)cc3C12
FC(F)(F)c1c[nH]c(n1)-c1cc(Oc2ccc3OC4C(C4c3c2)c2nc3ccc(cc3[nH]2)C(F)(F)F)ccn1
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ncnc5[nH]cnc45)cc3C12
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccncc4)cc3C12
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4ccnc5NC(=O)OCc45)cc3C12
FC(F)(F)c1ccc2nc([nH]c2c1)C1C2Oc3ccc(Oc4c(Cl)cnc5NC(=O)CCc45)cc3C12
OC(=O)C1C2Cc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
OC(=O)C1C2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3C12
CN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
CN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(C)(C)C
CN(C)CCN(C)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCN(CC1)C(C)(C)C)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCN(CC1)C1CCCC1)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCN(CC=C)CC1)C(=O)Nc1cc(on1)C(C)(C)C
CCN1CCC2(CCN(C2)c2cncc(c2)-c2cn(nn2)-c2cc(ccc2C)C(=O)Nc2cc(on2)C(C)(C)C)C1
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCN(CC2CCCO2)CC1)C(=O)Nc1cc(on1)C(C)(C)C
CN(C)CC1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
CN(C1CCOC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(NC2CCOC2)c1)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(NC(C)(C)C)c1)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCOCC1)C(=O)Nc1cc(n[nH]1)C(C)(C)C
CC(C)Nc1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
CC1CN(CCN1C)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCN(CCN2CCOCC2)CC1)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCCOCC1)C(=O)Nc1cc(on1)C(C)(C)C
CN(C)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCC1)C(=O)Nc1cc(on1)C(C)(C)C
COCC(C)Nc1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(NCC(F)(F)F)c1)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(NCCF)c1)C(=O)Nc1cc(on1)C(C)(C)C
C[C@H]1CN(C[C@@H](C)O1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C |r|
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCOCC1)C(=O)Nc1cc(nn1C)C(C)(C)C
CN(CC1CCCO1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCN(CC1)C1CC1)C(=O)Nc1cc(on1)C(C)(C)C
CCCCN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(NC2CC2)c1)C(=O)Nc1cc(on1)C(C)(C)C
CN(C1CCOCC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
CNc1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCN(CC(F)(F)F)CC1)C(=O)Nc1cc(on1)C(C)(C)C
CC1CN(CC(C)N1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
CCN1CCN(CC1C)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(NCC2CCCO2)c1)C(=O)Nc1cc(on1)C(C)(C)C
CC(C)N(C)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
COCCNc1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
CC(C)N1CCN(CC1C)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(NC2CCOCC2)c1)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCCC1)C(=O)Nc1cc(on1)C(C)(C)C
COCCCN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
CCCN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCCCC1)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(NC2CCCC2)c1)C(=O)Nc1cc(on1)C(C)(C)C
CC(C)N1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
COCCN1C(C)CN(CC1C)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
CN(C)CCNc1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCOCC1)C(=O)Nc1cc(on1)C(C)(C)C
CCN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
CCOCCN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
CC(C)CN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
CN(C)C1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
CC(C)N1CCCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
COCCN(C)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(NCC(F)F)c1)C(=O)Nc1cc(on1)C(C)(C)C
CN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(nn1C)C(C)(C)C
CCN(C)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCC1)C(=O)Nc1cc(ccn1)C(F)(F)F
Cc1ccc(cc1-n1cc(nn1)-c1cncc(NCC2CCCO2)c1)C(=O)Nc1cc(ccn1)C(F)(F)F
CN(CC1CCCO1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F
CN(C)C1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F
COCCN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F
CN(C)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F
CN1CCC(C1)Nc1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCCCC1)C(=O)Nc1cc(ccn1)C(F)(F)F
CN(CCN1CCCC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F
Cc1ccc(cc1-n1cc(nn1)-c1cncc(NC2CC2)c1)C(=O)Nc1cc(ccn1)C(F)(F)F
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCCOCC1)C(=O)Nc1cc(ccn1)C(F)(F)F
CN(C1CCOC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F
CN(C1CCOCC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F
Cc1ccc(cc1-n1cc(nn1)-c1cncc(NC2CCOC2)c1)C(=O)Nc1cc(ccn1)C(F)(F)F
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1C[C@@H]2C[C@H]1CN2)C(=O)Nc1cc(ccn1)C(F)(F)F |r|
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCOCC1)C(=O)Nc1cc(ccn1)C(F)(F)F
COCCN(C)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F
CN(C1CCN(C)CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F
CN(C)C1CCN(C1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F
CN1CCC(CC1)Nc1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCNCC1)C(=O)Nc1cc(ccn1)C(F)(F)F
CN(C1CCN(C)C1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F
CN(C)[C@H]1CCN(C1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F |r|
CN(C)[C@@H]1CCN(C1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F |r|
Cc1ccc(cc1-n1cc(nn1)-c1cncc(NC2CCOCC2)c1)C(=O)Nc1cc(ccn1)C(F)(F)F
CN1C[C@@H]2C[C@H]1CN2c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F |r|
CN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F
Cc1ccc(cc1-n1cc(nn1)-c1cncc(c1)N1CCCC1)C(=O)Nc1cc(ccn1)C(F)(F)F
CN(C)CCNc1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F
CN(C)CCN(C)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F
CCN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F
CC(C)N1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(ccn1)C(F)(F)F
CN1CCN(CC1)C1CCN(C1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
CN1CCN(CC1)C1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
CN1CCCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
CC(C)N1CCN(CC1)C1CCN(C1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
CN1CCN(CC1)C1CN(C1)c1cncc(c1)-c1cn(nn1)-c1cc(ccc1C)C(=O)Nc1cc(on1)C(C)(C)C
Cc1ccc(NC(=O)c2cc(ccn2)C(F)(F)F)cc1-n1cc(nn1)-c1cncc(c1)N1CCOCC1
CC(C)NCc1cc(oc1C(C)(C)C)C(=O)Nc1ccc(C)c(c1)-n1cc(nn1)-c1cncc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccc(o2)C(C)(C)C)cc1-n1cc(nn1)-c1cncc(c1)N1CCN(CC1)C(C)(C)C
Cc1ccc(NC(=O)c2cc(nn2C)C(C)(C)C)cc1-n1cc(nn1)-c1cncc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cc(on2)C(C)(C)C)cc1-n1cc(nn1)-c1cncc(c1)N1CCOCC1
CN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(NC(=O)c2cc(nn2C)C(C)(C)C)ccc1C
CN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(NC(=O)c2cc(ccn2)C(F)(F)F)ccc1C
CN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(NC(=O)c2cc(on2)C(C)(C)C)ccc1C
Cc1cc(nn1C(C)(C)C)C(=O)Nc1ccc(C)c(c1)-n1cc(nn1)-c1cncc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2cc(CN3CCCC3)c(o2)C(C)(C)C)cc1-n1cc(nn1)-c1cncc(c1)N1CCOCC1
Cc1ccc(NC(=O)c2ccc(s2)C(C)(C)C)cc1-n1cc(nn1)-c1cncc(c1)N1CCOCC1
Cc1oc(cc1C(=O)Nc1ccc(C)c(c1)-n1cc(nn1)-c1cncc(c1)N1CCOCC1)C(C)(C)C
Cc1ccc(NC(=O)c2ccc(o2)C(C)(C)C)cc1-n1cc(nn1)-c1cncc(c1)N1CCOCC1
CCN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(NC(=O)c2ccc(o2)C(C)(C)C)ccc1C
CN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(NC(=O)c2ccc(o2)C(C)(C)C)ccc1C
Cc1ccc(NC(=O)c2ccc(o2)C(C)(C)C)cc1-n1cc(nn1)-c1cncc(c1)N1CCN(CC2CC2)CC1
COCCCN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(NC(=O)c2ccc(o2)C(C)(C)C)ccc1C
Cc1ccc(NC(=O)c2ccc(o2)C(C)(C)C)cc1-n1cc(nn1)-c1cncc(c1)N1CCN(CC=C)CC1
CC(C)CN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(NC(=O)c2ccc(o2)C(C)(C)C)ccc1C
Cc1ccc(NC(=O)c2ccc(o2)C(C)(C)C)cc1-n1cc(nn1)-c1cncc(c1)N1CCNCC1
CCOCCN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(NC(=O)c2ccc(o2)C(C)(C)C)ccc1C
Cc1ccc(NC(=O)c2ccc(s2)C(C)(C)C)cc1-n1cc(nn1)-c1cncc(c1)N1CCN(CC1)C(=O)OC(C)(C)C
Cc1ccc(NC(=O)c2ccc(s2)C(C)(C)C)cc1-n1cc(nn1)-c1cncc(c1)N1CCNCC1
CCCN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(NC(=O)c2ccc(s2)C(C)(C)C)ccc1C
CN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(NC(=O)c2ccc(s2)C(C)(C)C)ccc1C
CCN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(NC(=O)c2ccc(s2)C(C)(C)C)ccc1C
CCOCCN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(NC(=O)c2ccc(s2)C(C)(C)C)ccc1C
Cc1ccc(NC(=O)c2ccc(s2)C(C)(C)C)cc1-n1cc(nn1)-c1cncc(c1)N1CCN(CC1)C(C)(C)C
CC(C)CN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(NC(=O)c2ccc(s2)C(C)(C)C)ccc1C
Cc1ccc(NC(=O)c2ccc(s2)C(C)(C)C)cc1-n1cc(nn1)-c1cncc(c1)N1CCN(CC2CC2)CC1
Cc1ccc(NC(=O)c2ccc(s2)C(C)(C)C)cc1-n1cc(nn1)-c1cncc(c1)N1CCN(CC=C)CC1
COCCCN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(NC(=O)c2ccc(s2)C(C)(C)C)ccc1C
Cc1cc(nn1C(C)(C)C)C(=O)Nc1ccc(C)c(c1)-n1cc(nn1)-c1cncc(c1)N1CCN(CC1)C1CC1
CCN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(NC(=O)c2cc(C)n(n2)C(C)(C)C)ccc1C
CC(C)N1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(NC(=O)c2cc(C)n(n2)C(C)(C)C)ccc1C
CCCN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(NC(=O)c2cc(C)n(n2)C(C)(C)C)ccc1C
CN1CCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(NC(=O)c2cc(C)n(n2)C(C)(C)C)ccc1C
CN1CCCN(CC1)c1cncc(c1)-c1cn(nn1)-c1cc(NC(=O)c2cc(C)n(n2)C(C)(C)C)ccc1C
Cc1ccc(NC(=O)c2cc(CNC(C)(C)C)c(o2)C(C)(C)C)cc1-n1cc(nn1)-c1cncc(c1)N1CCOCC1
CN1CCC(CC1)NCc1cc(oc1C(C)(C)C)C(=O)Nc1ccc(C)c(c1)-n1cc(nn1)-c1cncc(c1)N1CCOCC1
CN1CCN(Cc2cc(oc2C(C)(C)C)C(=O)Nc2ccc(C)c(c2)-n2cc(nn2)-c2cncc(c2)N2CCOCC2)CC1
CN(C)CCN(C)Cc1cc(oc1C(C)(C)C)C(=O)Nc1ccc(C)c(c1)-n1cc(nn1)-c1cncc(c1)N1CCOCC1
CN(C)Cc1cc(oc1C(C)(C)C)C(=O)Nc1ccc(C)c(c1)-n1cc(nn1)-c1cncc(c1)N1CCOCC1
CN(C)CCNCc1cc(oc1C(C)(C)C)C(=O)Nc1ccc(C)c(c1)-n1cc(nn1)-c1cncc(c1)N1CCOCC1
Cc1cc(Oc2cc(NC(=O)C3CC3)ncn2)ccc1NC(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3cc(NC(=O)C4CC4)ncn3)cc2)ccc1Cl
Fc1cc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)ccc1Oc1cc(NC(=O)C2CC2)ncn1
Fc1cc(Oc2cc(NC(=O)C3CC3)ncn2)ccc1NC(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
Cc1cc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)ccc1Oc1cc(NC(=O)C2CC2)ncn1
Cc1cc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)cnc1Oc1ccnc(NC(=O)C2CC2)c1
FC(F)(F)c1cc(NC(=O)Nc2cnc(Oc3ccnc(NC(=O)C4CC4)c3)c(Cl)c2)ccc1Cl
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)nc2)ccc1Cl
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cn2)ccc1Cl
Fc1cc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)ccc1Oc1ccnc(NC(=O)C2CC2)c1
Cc1cc(Oc2ccnc(NC(=O)C3CC3)c2)ccc1NC(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
Fc1cc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)cc(Oc2ccnc(NC(=O)C3CC3)c2)c1
Fc1cc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)cnc1Oc1ccnc(NC(=O)C2CC2)c1
CC1(CC1)C(=O)Nc1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)cc2F)ccn1
Fc1cc(Oc2ccnc(NC(=O)C3CC3)c2)ccc1NC(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
Cc1ccc(Oc2ccnc(NC(=O)C3CC3)c2)cc1NC(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
Cc1cc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)ccc1Oc1ccnc(NC(=O)C2CC2)c1
Fc1cc(Oc2ccnc(NC(=O)C3CC3)c2)ccc1NC(=O)Nc1cccc(OC(F)(F)F)c1
CC(F)(F)c1cc(F)cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2F)c1
CS(=O)(=O)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)cc(c1)C(F)(F)F
CN1CCC(C1)Oc1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)cc(c1)C(F)(F)F
CC1CN(C(=O)O1)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)cc(c1)C(F)(F)F
CC(=O)Nc1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)cc(c1)C(F)(F)F
CC1CN(CC(C)O1)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)cc(c1)C(F)(F)F
CN(C)C1CCN(C1)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)cc(c1)C(F)(F)F
OC1CCN(CC1)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)cc(c1)C(F)(F)F
Fc1cc(NC(=O)Nc2cc(cc(c2)C(F)(F)F)N2CCCC2=O)ccc1Oc1ccnc(NC(=O)C2CC2)c1
CC(F)(F)c1cncc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)c1
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2ccnc(NC(=O)C3CC3)c2)c(F)c1)C1CC1
Fc1c[nH]c2ccc(NC(=O)Nc3ccc(Oc4ccnc(NC(=O)C5CC5)c4)c(F)c3)cc12
Fc1cc(NC(=O)Nc2cccc(c2)C(F)(F)F)ccc1Oc1ccnc(NC(=O)C2CC2)c1
Fc1cc(NC(=O)Nc2ccc(C#N)c(c2)C(F)(F)F)ccc1Oc1ccnc(NC(=O)C2CC2)c1
Fc1cc(NC(=O)Nc2ccc(Cl)c(OC(F)(F)F)c2)ccc1Oc1ccnc(NC(=O)C2CC2)c1
CN1CCN(Cc2cc(NC(=O)Nc3ccc(Oc4ccnc(NC(=O)C5CC5)c4)cc3)cc(c2)C(F)(F)F)CC1
CC(F)(F)c1cncc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2)c1
Cc1cc(Oc2cc(NC(=O)C3CC3)ncn2)ccc1NC(=O)Nc1ccc(F)c(c1)C(F)(F)F
Cc1cc(Oc2cc(NC(=O)C3CC3)ncn2)ccc1NC(=O)Nc1cccc(c1)C(F)(F)F
Cc1cc(Oc2cc(NC(=O)C3CC3)ncn2)ccc1NC(=O)Nc1ccc(Cl)c(c1)C(C)(F)F
CC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3cc(NC(=O)C4CC4)ncn3)c(F)c2)ccc1Cl
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2cc(NC(=O)C3CC3)ncn2)cc1F)C(F)(F)F
Fc1cc(Oc2cc(NC(=O)C3CC3)ncn2)ccc1NC(=O)Nc1cccc(c1)C(F)(F)F
CC(F)(F)c1ccc(F)c(NC(=O)Nc2ccc(Oc3cc(NC(=O)C4CC4)ncn3)cc2F)c1
CC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3cc(NC(=O)C4CC4)ncn3)cc2F)ccc1Cl
Cc1cc(NC(=O)Nc2cc(ccc2F)C(C)(F)F)ccc1Oc1cc(NC(=O)C2CC2)ncn1
Cc1cc(NC(=O)Nc2ccc(F)c(c2)C(C)(F)F)ccc1Oc1cc(NC(=O)C2CC2)ncn1
Cc1cc(NC(=O)Nc2cc(ccc2F)C(F)(F)F)cnc1Oc1ccnc(NC(=O)C2CC2)c1
COc1ccc(NC(=O)Nc2cnc(Oc3ccnc(NC(=O)C4CC4)c3)c(C)c2)cc1C(F)(F)F
CC(C)Oc1cc(NC(=O)Nc2cnc(Oc3ccnc(NC(=O)C4CC4)c3)c(C)c2)cc(c1)C(F)(F)F
Cc1cc(Oc2ccnc(NC(=O)C3CC3)c2)ncc1NC(=O)Nc1cc(ccc1F)C(F)(F)F
Cc1cc(Oc2ccnc(NC(=O)C3CC3)c2)ncc1NC(=O)Nc1cc(ccc1F)C(C)(F)F
CS(=O)(=O)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)nc2)cc(c1)C(F)(F)F
CN1CCC(CC1)Nc1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)nc2)cc(c1)C(F)(F)F
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)nc2)cc(c1)N1CCS(=O)(=O)CC1
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cn2)ccc1C#N
CS(=O)(=O)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cn2)cc(c1)C(F)(F)F
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2)ccc1Cl
Fc1ccc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2)cc1C(F)(F)F
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2)ccc1C#N
Fc1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2)cc(c1)C(F)(F)F
FC(F)(F)c1ccc(Cl)c(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2)c1
CN1CCC(CC1)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2)cc(c1)C(F)(F)F
FC(F)(F)c1cccc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2)c1
CS(=O)(=O)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2)cc(c1)C(F)(F)F
FC(F)(F)Oc1cccc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2)c1
CC(F)(F)c1ccnc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2)c1
CC(F)(F)c1ccc(F)c(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2)c1
CC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2)ccc1Cl
FC1(F)CCOc2ccc(NC(=O)Nc3ccc(Oc4ccnc(NC(=O)C5CC5)c4)cc3)cc12
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2)cc(c1)C#N
Fc1ccc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)cc1C(F)(F)F
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2ccnc(NC(=O)C3CC3)c2)c(F)c1)C(F)(F)F
Fc1cc(NC(=O)Nc2cc(ccc2Cl)C(F)(F)F)ccc1Oc1ccnc(NC(=O)C2CC2)c1
Fc1cc(NC(=O)Nc2cc(cc(c2)C(F)(F)F)-c2ccncc2)ccc1Oc1ccnc(NC(=O)C2CC2)c1
CN1CCC(CC1)Nc1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)cc(c1)C(F)(F)F
CC1CN(CCO1)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)cc(c1)C(F)(F)F
Fc1cc(NC(=O)Nc2cc(NC(=O)C=C)cc(c2)C(F)(F)F)ccc1Oc1ccnc(NC(=O)C2CC2)c1
CN1CCC(CC1)Oc1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)cc(c1)C(F)(F)F
CS(=O)(=O)Nc1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)cc(c1)C(F)(F)F
Fc1cc(NC(=O)Nc2cc(cc(c2)C(F)(F)F)N2CCS(=O)(=O)CC2)ccc1Oc1ccnc(NC(=O)C2CC2)c1
CN1CCN(Cc2cc(NC(=O)Nc3ccc(Oc4ccnc(NC(=O)C5CC5)c4)c(F)c3)cc(c2)C(F)(F)F)CC1
CN1CCC(CC1)Nc1ccc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)cc1C(F)(F)F
Fc1cc(NC(=O)Nc2cc(ncn2)C(F)(F)F)ccc1Oc1ccnc(NC(=O)C2CC2)c1
Fc1cc(NC(=O)Nc2cccc(OC(F)(F)F)c2)ccc1Oc1ccnc(NC(=O)C2CC2)c1
Fc1cc(NC(=O)Nc2ccc(OC(F)(F)F)cc2)ccc1Oc1ccnc(NC(=O)C2CC2)c1
CC(F)(F)c1ccc(F)c(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)c1
CC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)ccc1Cl
CC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)ccc1F
Fc1ccc(Cl)cc1NC(=O)Nc1ccc(Oc2ccnc(NC(=O)C3CC3)c2)c(F)c1
Fc1cc(NC(=O)Nc2cc(cc(c2)C(F)(F)F)-c2cccnc2)ccc1Oc1ccnc(NC(=O)C2CC2)c1
CC(C)Nc1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)cc(c1)C(F)(F)F
CN1CCC(CC1)Oc1ccc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)cc1C(F)(F)F
Fc1cc(NC(=O)Nc2cc(cc(c2)C(F)(F)F)N2CCOCC2)ccc1Oc1ccnc(NC(=O)C2CC2)c1
Fc1cc(NC(=O)Nc2cc(cc(c2)C(F)(F)F)C#N)ccc1Oc1ccnc(NC(=O)C2CC2)c1
Cc1cc(Oc2ccnc(NC(=O)C3CC3)c2)ccc1NC(=O)Nc1ccc(F)c(c1)C(F)(F)F
Cc1cc(Oc2ccnc(NC(=O)C3CC3)c2)ccc1NC(=O)Nc1cccc(c1)C(F)(F)F
Cc1cc(Oc2ccnc(NC(=O)C3CC3)c2)ccc1NC(=O)Nc1cccc(OC(F)(F)F)c1
Cc1cc(Oc2ccnc(NC(=O)C3CC3)c2)ccc1NC(=O)Nc1cc(OC(F)(F)F)ccc1F
Cc1cc(Oc2ccnc(NC(=O)C3CC3)c2)ccc1NC(=O)Nc1ccc(F)c(OC(F)(F)F)c1
Cc1cc(Oc2ccnc(NC(=O)C3CC3)c2)ccc1NC(=O)Nc1ccc(Cl)c(c1)C(C)(F)F
Fc1ccc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2F)cc1C(F)(F)F
Fc1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2F)cc(c1)C(F)(F)F
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2ccnc(NC(=O)C3CC3)c2)cc1F)C(F)(F)F
Fc1cc(Oc2ccnc(NC(=O)C3CC3)c2)ccc1NC(=O)Nc1cc(ccc1Cl)C(F)(F)F
Fc1cc(Oc2ccnc(NC(=O)C3CC3)c2)ccc1NC(=O)Nc1cccc(c1)C(F)(F)F
Fc1cc(Oc2ccnc(NC(=O)C3CC3)c2)ccc1NC(=O)Nc1cc(cc(c1)C(F)(F)F)N1CC(F)(F)C1
Fc1ccc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2F)cc1OC(F)(F)F
CC(F)(F)c1ccnc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2F)c1
CC(F)(F)c1cccc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2F)c1
CC(F)(F)c1ccc(F)c(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2F)c1
CC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2F)ccc1Cl
CC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2F)ccc1F
Fc1cc(Oc2ccnc(NC(=O)C3CC3)c2)ccc1NC(=O)Nc1ccc(C#N)c(Cl)c1
Cc1ccc(Oc2ccnc(NC(=O)C3CC3)c2)cc1NC(=O)Nc1cc(F)cc(c1)C(F)(F)F
Cc1ccc(Oc2ccnc(NC(=O)C3CC3)c2)cc1NC(=O)Nc1cc(ccc1F)C(F)(F)F
Cc1ccc(Oc2ccnc(NC(=O)C3CC3)c2)cc1NC(=O)Nc1cc(ccc1F)C(C)(F)F
Cc1cc(NC(=O)Nc2ccc(F)c(c2)C(F)(F)F)ccc1Oc1ccnc(NC(=O)C2CC2)c1
Cc1cc(NC(=O)Nc2cccc(c2)C(F)(F)F)ccc1Oc1ccnc(NC(=O)C2CC2)c1
Cc1cc(NC(=O)Nc2cccc(OC(F)(F)F)c2)ccc1Oc1ccnc(NC(=O)C2CC2)c1
Cc1cc(NC(=O)Nc2cc(ccc2F)C(C)(F)F)ccc1Oc1ccnc(NC(=O)C2CC2)c1
Cc1cc(NC(=O)Nc2ccc(Cl)c(c2)C(C)(F)F)ccc1Oc1ccnc(NC(=O)C2CC2)c1
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2)cc(OCC2CNC2)c1
Nc1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)c(F)c2)cc(c1)C(F)(F)F
CN1CC(C1)Oc1cc(NC(=O)Nc2ccc(Oc3ccnc(NC(=O)C4CC4)c3)cc2)cc(c1)C(F)(F)F
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1NC(=O)c1cccc2c(N)nccc12
Nc1c(c(nn1-c1c(Cl)cc(Cl)cc1Cl)-c1ccncc1)-c1ccc(F)cc1 |(-1,-2.52,;-1.47,-1.05,;-2.94,-.58,;-2.94,.96,;-1.47,1.44,;-.56,.19,;.98,.19,;1.74,1.52,;.97,2.85,;3.28,1.52,;4.06,.18,;5.6,.18,;3.29,-1.15,;1.75,-1.15,;.97,-2.48,;-4.18,1.87,;-4.2,3.41,;-5.54,4.16,;-6.87,3.37,;-6.84,1.82,;-5.5,1.08,;-4.18,-1.48,;-5.52,-.72,;-6.85,-1.5,;-6.84,-3.04,;-8.17,-3.82,;-5.49,-3.8,;-4.17,-3.02,)|
CN1CCN(CCNc2nccc(n2)-c2c(nc3occn23)-c2cccc(O)c2)S1(=O)=O
CCN1CCN(CCNc2nccc(n2)-c2c(nc3occn23)-c2cccc(O)c2)S1(=O)=O
COc1ccc(cc1)S(=O)(=O)NCCNc1nccc(n1)-c1c(nc2sccn12)-c1ccccc1
COc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc(cc2)C(F)(F)F)n1
Oc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc(F)cc2)n1
Oc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccc(F)cc2)n1
Oc1c(Br)cc(C=C2C(=O)Nc3ccc(I)cc23)cc1Br
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(Cl)cc2)c1F
Nc1ncnc2n(CC3SSCC3O)nc(-c3ccc(Oc4ccccc4)cc3)c12
Nc1ncnc2n(C[C@@H]3SSC[C@@H]3O)nc(-c3ccc(Oc4ccccc4)cc3)c12 |r|
Nc1ncnc2n(C[C@H]3SSC[C@H]3O)nc(-c3ccc(Oc4ccccc4)cc3)c12 |r|
COc1cc2ncnc(Nc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)c(Cl)c3)c2c2OCCOc12
COc1cc2ncnc(Nc3ccc(NC(=O)Nc4cccc(c4)S(C)(=O)=O)c(Cl)c3)c2c2OCCOc12
COc1cc2ncnc(Oc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)cc3)c2c2OCCOc12
COc1cc2ncnc(Oc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)c(F)c3)c2c2OCCOc12
COc1cc2ncnc(Oc3ccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)cc3)c2c2OCCOc12
COCCOc1cc2ncnc(Nc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)c(Cl)c3)c2c2OCCOc12
COCCOc1cc2ncnc(Oc3ccc(NC(=O)NC4CC4)c(Cl)c3)c2c2OCCOc12
COCCOc1cc2ncnc(Oc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)cc3)c2c2OCCOc12
COCCOc1cc2ncnc(Oc3ccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)cc3)c2c2OCCOc12
COCCOc1cc2ncnc(Oc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)c(F)c3)c2c2OCCOc12
COCCOc1cc2ncnc(Oc3ccc(NC(=O)Nc4ccc(F)cc4F)c(F)c3)c2c2OCCOc12
COCCOc1cc2ncnc(Oc3ccc(NC(=O)Nc4cccc(OC)c4)cc3)c2c2OCCOc12
Clc1cc(Oc2ncnc3cc(OCCCN4CCCC4)c4OCCOc4c23)ccc1NC(=O)NC1CC1
Clc1cc(Oc2ncnc3cc(OCCCN4CCOCC4)c4OCCOc4c23)ccc1NC(=O)NC1CC1
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2ncnc3cc(OCCCN4CCOCC4)c4OCCOc4c23)cc1)C(F)(F)F
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ncnc4cc(OCCCN5CCOCC5)c5OCCOc5c34)cc2)ccc1Cl
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2ncnc3cc(OCCCN4CCOCC4)c4OCCOc4c23)c(F)c1)C(F)(F)F
Fc1cc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)ccc1Oc1ncnc2cc(OCCCN3CCOCC3)c3OCCOc3c12
CCN1CCN(CCNc2nccc(n2)-c2c(nc3sccn23)-c2ccc(F)c(O)c2)S1(=O)=O
COc1cc(ccc1F)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccc(F)cc2)n1
Nc1cc(ccc1F)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccc(F)cc2)n1
Cc1ccc2c(Nc3ccc(O)c(Cl)c3F)nccc2c1NC(=O)c1csc2c(N)ncnc12 |$;;;;;;N;;;;;;;;;;;;;;;;;;;;;;;;;;;$|
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4cccc(Cl)c4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(csc23)C(=O)Nc2c(C)ccc3c(Cc4cccc(c4)C(F)(F)F)nccc23)c(OC)c1
Cc1ccc2c(nccc2c1NC(=O)c1csc2c(N)ncnc12)C(=O)c1cccc(c1)C(F)(F)F
Cc1ccc2c(nccc2c1NC(=O)c1csc2c(N)ncnc12)C(O)c1cccc(c1)C(F)(F)F
Cc1ccc2c(nccc2c1NC(=O)c1csc2c(N)ncnc12)C(O)c1ccc(Cl)cc1F
COc1ccc(CNc2ncnc3c(csc23)C(=O)Nc2c(C)ccc3c(nccc23)C(C)Oc2ccccc2)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4cccc(Cl)c4)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4ccccc4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4ccc(Cl)cc4F)nccc23)c(OC)c1
Cc1ccc2c(Nc3cccc(c3)C(F)(F)F)nccc2c1NC(=O)c1cnc2c(N)ncnn12
COc1ccc(CNc2ncnc3c(cc(F)cc23)C(=O)Nc2c(C)ccc3c(Nc4cccc(Cl)c4F)nccc23)c(OC)c1
Cc1ccc2c(Nc3ccc(F)c(Cl)c3)nccc2c1NC(=O)c1cnc2c(N)ncnn12
COc1ccc(Nc2nccc3c(NC(=O)c4cccc5c(NCc6ccc(OC)cc6OC)ncnc45)c(C)ccc23)c(F)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4ccc(F)cc4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4cc(Cl)ccc4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cc(F)cc23)C(=O)Nc2c(C)ccc3c(Nc4ccc(F)cc4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4cc(ccc4F)S(C)(=O)=O)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4cc(F)c(F)cc4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(F)ccc3c(Nc4cccc(Cl)c4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(ccc(F)c23)C(=O)Nc2c(C)ccc3c(Nc4cccc(Cl)c4F)nccc23)c(OC)c1
COc1ccc(CNc2ncnc3c(cccc23)C(=O)Nc2c(C)ccc3c(Nc4c(F)cc(F)cc4F)nccc23)c(OC)c1
Cc1cc(F)c(NC(=O)N2CC[C@@H](CC(F)(F)F)C2)cc1-c1cc(N2CCOCC2)c2nn(C)cc2c1 |r|
Cc1n(C)nc2c(cc(cc12)-c1cc(NC(=O)N2CC[C@@H](CC(F)(F)F)C2)c(F)cc1C)N1CCOCC1 |r|
Cc1cc(F)c(NC(=O)N2CC[C@@H](CC(F)(F)F)C2)cc1-c1cc(N2CCOCC2)c2nccn2c1 |r|
Cc1cc(F)c(NC(=O)N2CC=C(C2)C(F)(F)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2c1 |c:11|
Cc1cc(F)c(NC(=O)N2CCC(C2)C(F)(F)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nc3CCOCc3n2c1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nc3CCC(O)Cc3n2c1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nc3COCCc3n2c1
Cc1ccc(NC(=O)N2CC[C@@H](CC(F)(F)F)C2)cc1-c1cc(N2CC3CCC(C2)O3)c2nccn2c1 |r|
Cc1cc(F)c(NC(=O)c2ccn(c2)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)[C@@H]2CCN(CC(F)(F)F)C2)cc1-c1cc(N2CCOCC2)c2nccn2c1 |r|
Cc1cc(F)c(NC(=O)N2CCOC(C2)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)N2CCC(C2)C2(CC2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)c2cn(cc2F)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)c2cn(cn2)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)N2CC=C(C2)C2(C)CC2)cc1-c1cc(N2CCOCC2)c2nccn2c1 |c:11|
Cc1cc(F)c(NC(=O)c2cncc(c2)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1ccc(NC(=O)c2cnn(c2F)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)N2CCC(C2)C(C)(C)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2c1
CCc1nc2cc(cc(N3CCOCC3)n2n1)-c1cc(C(=O)Nc2cn(nc2F)C(C)(C)C)c(F)cc1C
Cc1cc(F)c(NC(=O)c2cncc(c2)C(C)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)c2cn(nn2)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
CC(C(F)F)C1CCN(C1)C(=O)Nc1cc(c(C)cc1F)-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)N2CCC(F)(C2)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1ccc(NC(=O)c2cc(ncc2F)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
CC(C)(C)n1ncc(C(=O)Nc2cc(c(Cl)cc2F)-c2cc(N3CCOCC3)c3nccn3c2)c1F
Fc1cc(F)c(cc1NC(=O)N1CC[C@@H](CC(F)(F)F)C1)-c1cc(N2CCOCC2)c2nccn2c1 |r|
Cc1cc(F)c(NC(=O)c2cnn(c2F)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
CC(C)(C)n1ncc(C(=O)Nc2ccc(Cl)c(c2)-c2cc(N3CCOCC3)c3nccn3c2)c1F
Cc1cc(F)c(NC(=O)c2cnn(c2F)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2ncc(F)n2c1
Cc1cc(F)c(N)cc1-c1cc(N2CCOCC2)c2nccn2c1
CC(C(F)F)c1cc(ccn1)C(=O)Nc1cc(c(C)cc1F)-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)c2cn(c(F)n2)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
CC(C)C1CN(CC1F)C(=O)Nc1cc(c(C)cc1F)-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)N2CCC(C2)C(F)(F)C2CC2)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)c2cnn(c2)C(C)(C)C(F)F)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)c2cnn(c2)C(F)C(C)(C)F)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)c2cnn(c2)C(C)(C)C(F)(F)F)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1ncc(NC(=O)c2cnn(c2F)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cnc(NC(=O)c2cnn(c2F)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cn2cc(cc(N3CCOCC3)c2n1)-c1cc(NC(=O)c2cn(cn2)C(C)(C)C)c(F)cc1C
Cc1cc(F)c(NC(=O)c2nn(cc2F)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1ccc(NC(=O)c2nn(cc2F)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cn2cc(cc(N3CCOCC3)c2n1)-c1cc(NC(=O)c2cnn(c2F)C(C)(C)C)c(F)cc1C
Cc1cn2cc(cc(N3CCOCC3)c2n1)-c1cc(NC(=O)c2cn(c(F)n2)C(C)(C)C)c(F)cc1C
CC(C)(C)n1cc(nc1F)C(=O)Nc1cc(c(Cl)cc1F)-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)c2cnn(c2F)C(C)(C)C)cc1-c1cc(C2=CCOCC2)c2nccn2c1 |t:26|
Cc1c(F)c(F)c(NC(=O)c2cnn(c2F)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)c2ncn(c2F)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)c2cnn(c2F)C(C)(C)C)cc1-c1cc(N2CCOCC2)n2nccc2c1
Cc1cc(F)c(NC(=O)c2cnn(c2)C23CC(C2)C3)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)c2ccnc(c2)N2CCCC2)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)c2cnn(c2F)C(C)(C)C)cc1-c1cc(N2CC3CCC(C2)O3)c2nccn2c1
Cc1cc(F)c(NC(=O)c2cnn(c2F)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2ncnn2c1
Cc1cc(F)c(NC(=O)c2cnc(o2)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)c2coc(n2)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1ccc(NC(=O)c2cnc(o2)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)c2cnn(n2)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)c2ccnc(c2)C23CC(C2)C3)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)c2cnn(c2F)C(C)(C)C)cc1-c1cc(N2CCOCC2)n2ncnc2c1
Cc1cc(F)c(cc1-c1cc(N2CCOCC2)c2nccn2c1)C(=O)Nc1cnn(c1)C(C)(C)C
Cc1cc(F)c(cc1-c1cc(N2CCOCC2)c2nccn2c1)C(=O)Nc1cccc(c1)C(C)(C)C
CC(C)n1ccc2c(ccnc12)C(=O)Nc1cc(c(C)cc1F)-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(NC(=O)c2cnn(c2F)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nnnn2c1
CC(C)(C)n1ncc(C(=O)Nc2cc(c(Cl)cn2)-c2cc(N3CCOCC3)c3nccn3c2)c1F
Cc1cc(F)c(NC(=O)c2cnn(c2F)C(C)(C)C)cc1-c1cn2ccnc2c(n1)N1CCOCC1
Cc1cc(F)c(NC(=O)c2cnn(c2F)C(C)(C)C)cc1-c1cc(c2nccn2c1)C12CC1COCC2
Cc1cc(F)c(NC(=O)c2cnn(c2F)C(C)(C)C)cc1-c1cc(N2CCOCC2)c2nccn2n1
Cc1cc(F)c(NC(=O)c2cc(F)n(c2)C2(C)CC2)cc1-c1cc(N2CCOCC2)c2nccn2c1
Cc1cc(F)c(cc1-c1cc(N2CCOCC2)c2nccn2c1)C(=O)Nc1cnn(c1F)C(C)(C)C
Cc1cc(F)c(cc1-c1cc(N2CCOCC2)c2nccn2n1)C(=O)Nc1cnn(c1F)C(C)(C)C
CN(c1cc(ccn1)C(=O)Nc1cc(c(C)cc1F)-c1cc(N2CCOCC2)c2nccn2c1)C(F)(F)F
Cc1cn2nc(cc(N3CCOCC3)c2n1)-c1cc(NC(=O)c2cnn(c2F)C(C)(C)C)c(F)cc1C
Cc1cn2cc(cc(N3CCOCC3)c2n1)-c1cc(C(=O)Nc2cnn(c2F)C(C)(C)C)c(F)cc1C
Cc1nc2c(cc(cn2c1F)-c1cc(NC(=O)c2cnn(c2F)C(C)(C)C)c(F)cc1C)N1CCOCC1
Cc1nc2c(cc(cn2c1F)-c1cc(NC(=O)c2cnn(c2F)C(C)(C)C)ccc1C)N1CCOCC1
Cc1nc2c(cc(cn2c1F)-c1cc(C(=O)Nc2cnn(c2F)C(C)(C)C)c(F)cc1C)N1CCOCC1
Cc1nc2cc(cc(N3CCOCC3)n2n1)-c1cc(NC(=O)c2cnn(c2F)C(C)(C)C)c(F)cc1C
Cc1nc2cc(cc(N3CCOCC3)n2n1)-c1cc(C(=O)Nc2cnn(c2F)C(C)(C)C)c(F)cc1C
Cc1nc2c(cc(cn2n1)-c1cc(C(=O)Nc2cnn(c2F)C(C)(C)C)c(F)cc1C)N1CCOCC1
Cc1nc2cc(cc(N3CCOCC3)n2n1)-c1cc(NC(=O)c2cnc(o2)C(C)(C)C)c(F)cc1C
Cc1nc2cc(cc(N3CCOCC3)n2n1)-c1cc(NC(=O)c2coc(n2)C(C)(C)C)c(F)cc1C
Cc1nc2c(cc(cn2n1)-c1cc(NC(=O)c2cnc(o2)C(C)(C)C)c(F)cc1C)N1CCOCC1
Cc1nc2c(cc(cn2n1)-c1cc(NC(=O)c2coc(n2)C(C)(C)C)c(F)cc1C)N1CCOCC1
Cc1nc2c(cc(cn2n1)-c1cc(NC(=O)c2cnn(n2)C(C)(C)C)c(F)cc1C)N1CCOCC1
Cc1cc(F)c(NC(=O)c2cnc(o2)C(C)(C)C)cc1-c1cc(N2CCOCC2)n2nc(nc2c1)C1CC1
CCc1nc2cc(cc(N3CCOCC3)n2n1)-c1cc(NC(=O)c2cnc(o2)C(C)(C)C)c(F)cc1C
CCc1nc2cc(cc(N3CCOCC3)n2n1)-c1cc(C(=O)Nc2cnn(c2F)C(C)(C)C)c(F)cc1C
Cc1cc(F)c(cc1-c1cc(N2CCOCC2)n2nc(nc2c1)C1CC1)C(=O)Nc1cnn(c1F)C(C)(C)C
CC(C)c1nc2c(cc(cn2n1)-c1cc(C(=O)Nc2cnn(c2F)C(C)(C)C)c(F)cc1C)N1CCOCC1
CN(C)c1nc2c(cc(cn2n1)-c1cc(C(=O)Nc2cnn(c2F)C(C)(C)C)c(F)cc1C)N1CCOCC1
Cc1nc2c(cc(cn2n1)-c1cc(C(=O)Nc2cn(nc2F)C2(C)CC2)c(F)cc1C)N1CCOCC1
CNS(=O)(=O)Nc1cccc(Cc2c(CC(=O)NOCCO)c3ccc(Oc4ncccn4)cc3oc2=O)c1F
CNS(=O)(=O)NCC(=O)N(Cc1cc(C(=O)NOCCO)c(Nc2ccc(I)cc2F)c(F)c1F)OC
[#6]-[#7]S(=O)(=O)[#7-]([Na+])-c1nccc(-[#6]-c2cc(-[#6](-[#7])=O)c(-[#7]-c3ccc(cc3F)-[#6]-3-[#6]-[#6]-3)c(F)c2F)c1F
NC(=O)c1cc(Cc2ccnc(NS(=O)(=O)NC3C4CCOC34)c2F)c(F)c(F)c1Nc1ccc(I)cc1F
CNS(C)(=O)=Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)c(F)c2F)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc4sccc4c3F)c(F)c2F)c1F
CNS(=O)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)cn2)c1F
Cn1cnc2ccc(Oc3c(F)ccc(NS(=O)(=O)N4CC[C@@H](F)C4)c3C#N)cc2c1=O
Cn1cnc2ccc(Oc3c(F)ccc(NS(=O)(=O)N4CC[C@H](F)C4)c3C#N)cc2c1=O
CCCS(=O)(=O)Nc1ccc(F)c(Oc2ccc3ncn(C)c(=O)c3c2)c1C#N
CN(C)S(=O)(=O)Nc1ccc(Cl)c(Oc2ccc3ncn(C)c(=O)c3c2)c1C#N
Cn1cnc2ccc(Oc3c(Cl)ccc(NS(=O)(=O)N4CCCC4)c3C#N)cc2c1=O
CN(C)S(=O)(=O)Nc1ccc(Cl)c(Oc2ccc3ncn(C)c(=O)c3c2)c1F
Cn1cnc2ccc(Oc3c(Cl)ccc(NS(=O)(=O)N4CCCC4)c3F)cc2c1=O
CNS(=O)(=O)Nc1nccc(Oc2cc(C(N)=O)c(Nc3ccc(I)cc3F)cc2F)c1F
CNS(=C)(=O)Nc1nccc(Cc2cc(C(N)=O)c(Nc3ccc(I)cc3F)n(C)c2=O)c1F
COc6ccc(S(=O)(=O)Nc5ccc(F)c(Nc3ncnc4ccc(n2cnc1c(C(N)=O)cccc12)nc34)c5F)c(C)c6
Nc5nc(c4ccc3ncnc(Nc2c(F)ccc(NS(=O)(=O)c1ccccc1Cl)c2F)c3n4)cs5
CN(C)C(=O)c5cn(c4ccc3ncnc(Nc2c(F)ccc(NS(=O)(=O)c1ccccc1Cl)c2F)c3n4)c6cccc(N)c56
Nc1cccc2c1nnn2c6ccc5ncnc(Nc4c(F)ccc(NS(=O)(=O)c3cccc(Cl)c3Cl)c4F)c5n6
Nc1cccc3c1c(C(=O)N2CCOCC2)cn3c7ccc6ncnc(Nc5c(F)ccc(NS(=O)(=O)c4ccccc4Cl)c5F)c6n7
Cc1c(Cl)cccc1S(=O)(=O)Nc6ccc(F)c(Nc4ncnc5ccc(n3cnc2c(O)cccc23)nc45)c6F
Cc1c(Cl)cccc1S(=O)(=O)Nc6ccc(F)c(Nc4ncnc5ccc(n3nnc2c(O)cccc23)nc45)c6F
O=C(Nc1cccc2c1ncn2c6ccc5ncnc(Nc4c(F)ccc(NS(=O)(=O)c3ccccc3Cl)c4F)c5n6)N7CCOCC7
CN(C)C(=O)Nc1cccc2c1ncn2-c1ccc2ncnc(Nc3c(F)ccc(CS(=O)(=O)c4ccccc4Cl)c3F)c2n1
O=S(=O)(Nc6ccc(F)c(Nc4ncnc5ccc(n3cc(c1ncc[nH]1)c2ccccc23)nc45)c6F)c7cccc(Cl)c7Cl
O=S(=O)(Nc6ccc(F)c(Nc4ncnc5ccc(n3nc(c1nnc(O)o1)c2ccccc23)nc45)c6F)c7cccc(Cl)c7Cl
CN(C)c7nnc(c5nn(c4ccc3ncnc(Nc2c(F)ccc(NS(=O)(=O)c1cccc(Cl)c1Cl)c2F)c3n4)c6ccccc56)o7
O=S(=O)(Nc6ccc(F)c(Nc4ncnc5ccc(n3nc(c1ncc[nH]1)c2ccccc23)nc45)c6F)c7ccccc7Cl
NCC(=O)c5cn(c4ccc3ncnc(Nc2c(F)ccc(NS(=O)(=O)c1ccccc1Cl)c2F)c3n4)c6ccccc56
CN(C)CC(=O)c5cn(c4ccc3ncnc(Nc2c(F)ccc(NS(=O)(=O)c1ccccc1Cl)c2Cl)c3n4)c6ccccc56
Cc1c(F)cccc1S(=O)(=O)Nc6ccc(F)c(Nc4ncnc5ccc(n3cnc2c(C#N)cccc23)nc45)c6F
Cc1c(F)cccc1S(=O)(=O)Nc6ccc(F)c(Nc4ncnc5ccc(n3ncc2CCN(CCO)Cc23)nc45)c6F
Cc1c(F)cccc1S(=O)(=O)Nc5ccc(F)c(Nc3ncnc4ccc(n2cnc(/C=C/C#N)c2)nc34)c5F
Cc1c(F)cccc1S(=O)(=O)Nc6ccc(F)c(Nc4ncnc5ccc(n3cnc2c(CO)cccc23)nc45)c6F
Cc1c(F)cccc1S(=O)(=O)Nc5ccc(F)c(Nc3ncnc4ccc(n2cnc(CCC#N)c2)nc34)c5F
Nc1nccc2c1ncn2c6ccc5ncnc(Nc4c(F)ccc(NS(=O)(=O)c3cccc(Cl)c3Cl)c4F)c5n6
Cc1nc(N)ccc1S(=O)(=O)Nc6ccc(F)c(Nc4ncnc5ccc(n3cnc2c(N)cccc23)nc45)c6F
Cc1c(F)cccc1S(=O)(=O)Nc6ccc(F)c(Nc4ncnc5ccc(n3cc2c(CCCN2C)n3)nc45)c6F
CC(=O)N6CCCc5nn(c4ccc3ncnc(Nc2c(F)ccc(NS(=O)(=O)c1cccc(F)c1C)c2F)c3n4)cc56
Cc1c(F)cccc1S(=O)(=O)Nc6ccc(F)c(Nc4ncnc5ccc(n3cc2c(CCCN2CCN)n3)nc45)c6F
Cc1cc(N)ccc1S(=O)(=O)Nc6ccc(F)c(Nc4ncnc5ccc(n3cnc2c(N)cccc23)nc45)c6F
COCCN(CCOC)c1cccc2c1ncn2c6ccc5ncnc(Nc4c(F)ccc(NS(=O)(=O)c3cccc(F)c3C)c4F)c5n6
CN(C)CCN(C)S(=O)(=O)c5ccn(c4ccc3ncnc(Nc2c(F)ccc(NS(=O)(=O)c1cccc(Cl)c1Cl)c2F)c3n4)c5
Cc1c(F)cccc1S(=O)(=O)Nc6ccc(F)c(Nc4ncnc5ccc(n3cc2c(CCCN2CCCO)n3)nc45)c6F
Cc1c(F)cccc1S(=O)(=O)Nc6ccc(F)c(Nc4ncnc5ccc(n3cc2c(CCCN2C(=O)CN)n3)nc45)c6F
Cc1c(F)cccc1S(=O)(=O)Nc6ccc(F)c(Nc4ncnc5ccc(n3ncc2CCN(CCN)Cc23)nc45)c6F
Cc1c(F)cccc1S(=O)(=O)Nc7ccc(F)c(Nc5ncnc6ccc(n4cnc3c(c2cnccc2N)cccc34)nc56)c7F
Cc1c(F)cccc1S(=O)(=O)Nc7ccc(F)c(Nc5ncnc6ccc(n4cnc3c(c2cccnc2N)cccc34)nc56)c7F
Cc1c(F)cccc1S(=O)(=O)Nc6ccc(F)c(Nc4ncnc5ccc(n2ncc3c2CCCN3CCO)nc45)c6F
O=S(=O)(Nc6ccc(F)c(Nc4ncnc5ccc(n3cc(S(=O)(=O)C1CCNCC1)c2ccccc23)nc45)c6F)c7cccc(Cl)c7Cl
CN7CCC(S(=O)(=O)c5cn(c4ccc3ncnc(Nc2c(F)ccc(NS(=O)(=O)c1cccc(Cl)c1Cl)c2F)c3n4)c6ccccc56)CC7
CP(C)(=O)c1cn(-c2ccc3ncnc(Nc4c(F)ccc(NS(=O)(=O)c5cccc(Cl)c5Cl)c4F)c3n2)c2ccccc12
COCCC(=O)Nc1cn(-c2ccc3ncnc(Nc4c(F)ccc(NS(=O)(=O)c5cccc(Cl)c5Cl)c4F)c3n2)c2ccccc12
CN(C)CCCS(=O)(=O)c1cn(-c2ccc3ncnc(Nc4c(F)ccc(NS(=O)(=O)c5cccc(Cl)c5Cl)c4F)c3n2)c2ccccc12
CC(=O)N1CCCc2nn(-c3ccc4ncnc(Nc5c(F)ccc(NS(=O)(=O)c6cccc(Cl)c6Cl)c5F)c4n3)cc21
O=S(=O)(Nc1ccc(F)c(Nc2ncnc3ccc(-n4cc(CC5CCN(CC(F)F)CS5(=O)=O)c5ccccc54)nc23)c1F)c1cccc(Cl)c1Cl
CC(C)(CC(F)F)S(=O)(=O)c1cn(-c2ccc3ncnc(Nc4c(F)ccc(NS(=O)(=O)c5cccc(Cl)c5Cl)c4F)c3n2)c2ccccc12
O=C(c1cn(-c2ccc3ncnc(Nc4c(F)ccc(NS(=O)(=O)c5cccc(Cl)c5Cl)c4F)c3n2)c2ccccc12)C1CCOC1
C[P-](=O)(=O)c1cn(-c2ccc3ncnc(Nc4c(F)ccc(NS(=O)(=O)c5cccc(Cl)c5Cl)c4F)c3n2)c2cccc(N)c12
O=S(=O)(Nc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5nccnc54)nc23)c1F)c1cccc(Cl)c1Cl
O=C1CCCN1c1cn(-c2ccc3ncnc(Nc4c(F)ccc(NS(=O)(=O)c5cccc(Cl)c5Cl)c4F)c3n2)c2ccccc12
O=S(=O)(Nc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5c(N6CC[C@@H](O)C6)nccc54)nc23)c1F)c1cccc(Cl)c1Cl
CCOc1nccc2c1ncn2-c1ccc2ncnc(Nc3c(F)ccc(NS(=O)(=O)c4cccc(Cl)c4Cl)c3F)c2n1
O=S(=O)(Nc1ccc(F)c(Nc2ncnc3ccc(-n4cc(N5CCCCS5(=O)=O)c5ccccc54)nc23)c1F)c1cccc(Cl)c1Cl
CC(C)(C#N)c1cccc2c1ncn2-c1ccc2ncnc(Nc3c(F)ccc(NS(=O)(=O)c4cccc(Cl)c4Cl)c3F)c2n1
CS(=O)(=O)c1cccc2c1ncn2-c1ccc2ncnc(Nc3c(F)ccc(NS(=O)(=O)c4cccc(Cl)c4Cl)c3F)c2n1
COCCOc1nccc2c1ncn2-c1ccc2ncnc(Nc3c(F)ccc(NS(=O)(=O)c4cccc(Cl)c4Cl)c3F)c2n1
CC7(O)CCN(c1cccc2c1ccn2c6ccc5ncnc(Nc4c(F)ccc(NS(=O)(=O)c3cccc(Cl)c3Cl)c4F)c5n6)CC7
CCOc1cccc2c1ncn2c6ccc5ncnc(Nc4c(F)ccc(NS(=O)(=O)c3cccc(Cl)c3Cl)c4F)c5n6
Cc1c(F)cccc1S(=O)(=O)Nc6ccc(F)c(Nc4ncnc5ccc(n3ncc2CCN(CC(N)=O)Cc23)nc45)c6F
O=S(=O)(Nc4ccc(F)c(Nc2ncnc3ccc(c1cscn1)nc23)c4F)c5cccc(Cl)c5Cl
O=S(=O)(Nc5ccc(F)c(Nc3ncnc4ccc(c1cnn2CCCCCCc12)nc34)c5F)c6cccc(Cl)c6Cl
CC5=NC=C(c4ccc3ncnc(Nc2c(F)ccc(NS(=O)(=O)c1cccc(Cl)c1Cl)c2F)c3n4)C5
CN6CCN(c5ncc(c4ccc3ncnc(Nc2c(F)ccc(NS(=O)(=O)c1cccc(Cl)c1Cl)c2F)c3n4)s5)CC6
O=S(=O)(Nc6ccc(F)c(Nc4ncnc5ccc(n3nnc2c(N1CCNCC1)cccc23)nc45)c6F)c7cccc(Cl)c7Cl
O=S7(=O)CCN(c1cccc2c1ncn2c6ccc5ncnc(Nc4c(F)ccc(NS(=O)(=O)c3cccc(Cl)c3Cl)c4F)c5n6)CC7
O=S(=O)(Nc5ccc(F)c(n4cnc3c(N2CCC1(CCCC1O)CC2)cccc34)c5F)c6cccc(Cl)c6Cl
O=S(=O)(Nc6ccc(F)c(Nc4ncnc5ccc(n3cnc2c(C1CCNCC1)cccc23)nc45)c6F)c7cccc(Cl)c7Cl
O=S(=O)(Nc7ccc(F)c(Nc5ncnc6ccc(n4ncc3c(C2CCC1(CCCC1O)CC2)cccc34)nc56)c7F)c8cccc(Cl)c8Cl
CC(C)C7(O)CCN(c1cccc2c1ccn2c6ccc5ncnc(Nc4c(F)ccc(NS(=O)(=O)c3cccc(Cl)c3Cl)c4F)c5n6)CC7
CCCOc1cccc2c1nnn2c6ccc5ncnc(Nc4c(F)ccc(NS(=O)(=O)c3cccc(Cl)c3Cl)c4F)c5n6
O=S(=O)(Nc6ccc(F)c(Nc4ncnc5ccc(n3cnc2c(C1CCN(CCO)CC1)cccc23)nc45)c6F)c7cccc(Cl)c7Cl
COc1ccc(S(=O)(=O)Nc2ccc(F)c(Nc3ncnc4ccc(-n5cnc6ccccc65)nc34)c2F)cc1
COc1ccc(S(=O)(=O)Nc2ccc(F)c(Nc3ncnc4ccc(-n5cnc6ccccc65)nc34)c2F)c(F)c1
COc1ccc(S(=O)(=O)Nc2ccc(F)c(Nc3ncnc4ccc(-n5cnc6ccccc65)nc34)c2F)c(C)c1
O=S(=O)(Nc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5ccccc54)nc23)c1F)c1ccc(Cl)cc1Cl
COc1ccc(S(=O)(=O)Nc2ccc(F)c(Nc3ncnc4ccc(-n5cnc6ccccc65)nc34)c2F)c(Cl)c1
Cc1ccc(S(=O)(=O)Nc2ccc(F)c(Nc3ncnc4ccc(-n5cnc6ccccc65)nc34)c2F)c(C)c1
O=S(=O)(Nc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5ccccc54)nc23)c1F)c1ccccc1Cl
Cc1ccccc1S(=O)(=O)Nc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5ccccc54)nc23)c1F
CCc1ccc(S(=O)(=O)Nc2ccc(F)c(Nc3ncnc4ccc(-n5cnc6ccccc65)nc34)c2F)cc1
COc1ccc(S(=O)(=O)Nc2ccc(F)c(Nc3ncnc4ccc(-n5cnc6ccccc65)nc34)c2F)cc1OC
O=S(=O)(Nc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5ccccc54)nc23)c1F)c1ccccc1C(F)(F)F
O=S(=O)(Nc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5ccccc54)nc23)c1F)c1ccc2c(c1)OCO2
O=S(=O)(Nc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5ccccc54)nc23)c1F)c1sccc1Cl
O=S(=O)(Nc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5ccccc54)nc23)c1F)c1cccc(Cl)c1Cl
Cc1c(Cl)cccc1S(=O)(=O)Nc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5ccccc54)nc23)c1F
O=S(=O)(Nc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5ccccc54)nc23)c1F)c1ccccc1Br
O=S(=O)(Nc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5ccccc54)nc23)c1F)c1ccc(F)cc1Cl
O=S(=O)(Nc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5ccccc54)nc23)c1F)c1c(F)cccc1Cl
O=S(=O)(Nc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5ccccc54)nc23)c1F)c1cc(Cl)ccc1Cl
Cc1ccc(C)c(S(=O)(=O)Nc2ccc(F)c(Nc3ncnc4ccc(-n5cnc6ccccc65)nc34)c2F)c1
Cc1cccc(Cl)c1S(=O)(=O)Nc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5ccccc54)nc23)c1F
Cc1cccc(S(=O)(=O)Nc2ccc(F)c(Nc3ncnc4ccc(-n5cnc6ccccc65)nc34)c2F)c1C
Cc1ccc(S(=O)(=O)Nc2ccc(F)c(Nc3ncnc4ccc(-n5cnc6ccccc65)nc34)c2F)c(Cl)c1
Cc1c(F)cccc1S(=O)(=O)Nc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5ccccc54)nc23)c1F
CO[C@@H]1CCN(S(=O)(=O)Nc2ccc(F)c(Nc3ncnc4ccc(-n5cnc6ccccc65)nc34)c2F)C1
CCc1ccc(S(=O)(=O)Nc2ccc(F)c(Nc3ncnc4ccc(-n5cnc6ccccc65)nc34)c2F)c(C)c1Cl
COc1ccc(S(=O)(=O)Nc2ccc(F)c(Nc3ncnc4ccc(-n5cnc6ccccc65)nc34)c2F)c(C)c1F
Cc1cccc(S(=O)(=O)Nc2ccc(F)c(Nc3ncnc4ccc(-n5cnc6ccccc65)nc34)c2F)c1Cl
Cc1c(Cl)csc1S(=O)(=O)Nc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5ccccc54)nc23)c1F
Cc1csc(S(=O)(=O)Cc2ccc(F)c(Nc3ncnc4ccc(-n5cnc6ccccc65)nc34)c2F)c1Cl
O=S(=O)(Cc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5ccccc54)nc23)c1F)c1scc(Cl)c1Cl
O=S(=O)(Cc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5ccccc54)nc23)c1F)c1cccc(Cl)c1C(F)(F)F
O=S(=O)(Cc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5ccccc54)nc23)c1F)c1cccc(F)c1C(F)(F)F
Cc1scc(S(=O)(=O)Nc2ccc(F)c(Nc3ncnc4ccc(-n5cnc6ccccc65)nc34)c2F)c1C
Cc1c(S(=O)(=O)Nc2ccc(F)c(Nc3ncnc4ccc(-n5cnc6ccccc65)nc34)c2F)ccc(F)c1F
Cc1ccc(S(=O)(=O)Nc2ccc(F)c(Nc3ncnc4ccc(-n5cnc6ccccc65)nc34)c2F)c(C)c1F
Cc1c(S(=O)(=O)Nc2ccc(F)c(Nc3ncnc4ccc(-n5cnc6ccccc65)nc34)c2F)ccc(Cl)c1F
O=S(=O)(Nc1ccc(F)c(Nc2ncnc3ccc(-n4cnc5ccccc54)nc23)c1F)c1ccc(C(F)(F)F)cc1Cl
CNS(=O)(=O)c1ccc(OC)c(Nc2cc(Nc3ccc(Cl)cn3)ncn2)c1
CNS(=O)(=O)c1ccc(c(Nc2cc(Nc3ccc(Cl)cn3)ncn2)c1)S(C)(=O)=O
CCS(=O)(=O)c1ccc(cc1Nc1cc(Nc2ccc(Cl)cn2)ncn1)S(=O)(=O)NC
CNS(=O)(=O)c1ccc(c(Nc2cc(Nc3ccc(Cl)cn3)ncn2)c1)S(=O)(=O)C(C)C
CNS(=O)(=O)c1ccc(OCC(F)(F)F)c(Nc2cc(Nc3ccc(Cl)cn3)ncn2)c1
CNS(=O)(=O)c1ccc(c(Nc2cc(Nc3ccc(Cl)cn3)ncn2)c1)S(=O)(=O)C(C)(C)C
CNc1cc(ncn1)C1(CC1)C(=O)Nc1cc(ccc1C)C(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
CNc1cc(ncn1)C1(CC1)C(=O)Nc1cc(ccc1C)C(=O)Nc1ccc(OCC2CCN(C)CC2)c(c1)C(F)(F)F
CNc1cc(ncn1)C1(CC1)C(=O)Nc1cc(ccc1C)C(=O)Nc1ccc(OCCCN2CCOCC2)c(c1)C(F)(F)F
CN(C)CCCNc1cc(ncn1)C1(CC1)C(=O)Nc1cc(ccc1C)C(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
Cc1ccc(cc1NC(=O)C1(CC1)c1cc(NCCN2CCCCC2)ncn1)C(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
CN1CCC(CNc2cc(ncn2)C2(CC2)C(=O)Nc2cc(ccc2C)C(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)CC1
CN1CCN(CCCNc2cc(ncn2)C2(CC2)C(=O)Nc2cc(ccc2C)C(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)CC1
CNc1nccc(n1)C1(CC1)C(=O)Nc1cc(ccc1C)C(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
CNc1cc(ncn1)C1(CC1)C(=O)Nc1cc(ccc1C)C(=O)Nc1ccc(OC2CCN(C)CC2)c(c1)C(F)(F)F
Cc1ccc(cc1NC(=O)C1(CC1)c1cc(NCCN2CCCC2)ncn1)C(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
COc1n[nH]c2ncc(cc12)C#Cc1c(F)ccc(NS(=O)(=O)c2ccccc2)c1F
COc1n[nH]c2ncc(cc12)C#Cc1c(F)ccc(NS(=O)(=O)c2ccccc2Cl)c1F
COc1n[nH]c2ncc(cc12)C#Cc1c(F)ccc(NS(=O)(=O)c2cccc(Cl)c2)c1F
COc1n[nH]c2ncc(cc12)C#Cc1c(F)ccc(NS(=O)(=O)c2ccc(Cl)cc2)c1F
COc1n[nH]c2ncc(cc12)C#Cc1c(F)ccc(NS(=O)(=O)c2cccc(C)c2)c1F
COc1n[nH]c2ncc(cc12)C#Cc1c(F)ccc(NS(=O)(=O)c2cccc(OC)c2)c1F
COc1c2cc(cnc2[nH]n1)C#Cc3c(ccc(c3F)NS(=O)(=O)c4cccc(c4)Br)F
COc1n[nH]c2ncc(cc12)C#Cc1c(F)ccc(NS(=O)(=O)c2cccc(c2)C#N)c1F
Fc1ccc(NS(=O)(=O)c2cccc(Cl)c2)c(F)c1C#Cc1cnc2[nH]ccc2c1
Fc1ccc(NS(=O)(=O)c2cccc(Cl)c2)c(F)c1C#Cc1ccc2[nH]ncc2c1
Fc1ccc(NS(=O)(=O)c2cccc(Cl)c2)c(F)c1C#Cc1cnc2[nH]nc(OC3CCCC3)c2c1
COc1n[nH]c2ncc(cc12)C#Cc1c(F)ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)c1F
CC(C)Oc1n[nH]c2ncc(cc12)C#Cc1c(F)ccc(NS(=O)(=O)c2cccc(Cl)c2)c1F
Fc1ccc(NS(=O)(=O)c2cccc(Cl)c2)c(F)c1C#Cc1cnc2[nH]ncc2c1
Cn1ncc2cc(cnc12)C#Cc1c(F)ccc(NS(=O)(=O)c2cccc(Cl)c2)c1F
Clc1cccc(NC(=O)Nc2ccc(cc2)-c2ccc(NC(=O)C=C)nc2)c1
Nc1n[nH]c2cccc(-c3ccc(NC(=S)Nc4cc(Br)ccc4OC(F)(F)F)cc3)c12
Cn1ccc2c(Oc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)cc3)ncnc12
Cn1ncc2c(Oc3ccc4n(C)c(Nc5ccc(Cl)cc5)nc4c3)ncnc12
Cc1ccc(Nc2nc3cc(Oc4ncnc5n(C)ncc45)ccc3n2C)cc1
Cn1ncc2c(Oc3ccc4n(C)c(Nc5ccc(Br)cc5)nc4c3)ncnc12
Cn1ncc2c(Oc3ccc4n(C)c(Nc5ccc(F)cc5)nc4c3)ncnc12
Cn1ncc2c(Oc3ccc4n(C)c(Nc5ccc(Cl)c(Cl)c5)nc4c3)ncnc12
Cn1ncc2c(Oc3ccc4n(C)c(Nc5cccc(c5)C(F)(F)F)nc4c3)ncnc12
Cn1ncc2c(Oc3ccc4n(C)c(Nc5ccc(cc5)C(F)(F)F)nc4c3)ncnc12
Cn1ncc2c(Oc3ccc4n(C)c(Nc5ccc(OC(F)(F)F)cc5)nc4c3)ncnc12
CNC(=O)c1cc(Oc2ccc(cc2)C2=NNC(C2)c2cccc(Br)c2)ccn1 |t:15|
CNC(=O)c1cc(Oc2ccc(cc2)C2=NNC(C2)c2ccc(OC)cc2)ccn1 |t:15|
CNC(=O)c1cc(Oc2ccc(cc2)C2=NNC(C2)c2ccccc2)ccn1 |t:15|
CNC(=O)c1cc(Oc2ccc(cc2)C2CC(=NN2)c2ccc(cc2)[N+]([O-])=O)ccn1 |c:17|
CC(=O)Nc1cn2cc(ccc2n1)-c1cc(NC(=O)c2cc(ccn2)C(F)(F)F)ccc1C
CC(=O)Nc1cn2cc(ccc2n1)-c1cc(NC(=O)c2cccc(Cl)c2)ccc1C
CC(=O)Nc1cn2cc(ccc2n1)-c1cc(NC(=O)c2cccc(n2)C(F)(F)F)ccc1C
CC(=O)Nc1cn2cc(ccc2n1)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
CC(=O)Nc1cn2cc(ccc2n1)-c1cc(NC(=O)c2cccc(c2)C(C)(C)C)ccc1C
C[C@H]1CN(C)CCN1c1cc(cc(c1)C(F)(F)F)C(=O)Nc1ccc(C)c(c1)-c1ccc2nc(NC(C)=O)cn2c1 |r|
CC(=O)Nc1cn2cc(ccc2n1)-c1cc(NC(=O)c2ccccc2)ccc1C
CN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)Nc2ccc(C)c(c2)-c2ccc3nc(NC(C)=O)cn3c2)CC1
c1cc2c(cc1C(F)(F)F)nc([nH]2)[C@H]3[C@H]4[C@@H]3Oc5c4cc(cc5)Oc6ccnc7c6CCC(=O)N7
F[C@H]1CCN(C1)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F |r|
Cc1ccc(NC(=O)c2cccc(c2)C(C)(C)C#C)cc1Nc1ccc2ncn(C)c(=O)c2c1
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-n1cc(-c2cncnc2)c2nc(ccc12)N(C)C1CCN(CC)CC1 |(23.77,-37.37,;22.26,-37.06,;21.77,-35.6,;20.26,-35.29,;19.86,-36.78,;18.77,-35.69,;19.78,-33.84,;18.27,-33.53,;17.24,-34.69,;15.73,-34.38,;15.25,-32.92,;13.74,-32.6,;16.28,-31.77,;17.78,-32.07,;18.8,-30.92,;15.79,-30.31,;16.69,-29.06,;15.78,-27.82,;16.25,-26.36,;17.75,-26.03,;18.22,-24.57,;17.18,-23.43,;15.67,-23.76,;15.21,-25.23,;14.32,-28.3,;12.98,-27.54,;11.65,-28.31,;11.65,-29.85,;12.98,-30.63,;14.33,-29.85,;10.32,-27.54,;10.32,-26,;8.99,-28.31,;7.65,-27.54,;6.32,-28.3,;6.32,-29.84,;4.98,-30.61,;3.65,-29.83,;7.65,-30.62,;8.99,-29.85,)|
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2cnc(nc2)C2CC2)c1F
FC(F)(F)c1ccc2nc([nH]c2c1)[C@H]1[C@@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@H]12 |r|
CSc1cc(Oc2ccnc3[nH]c(=O)cnc23)ccc1NC(=O)Nc1cc(nn1-c1ccccc1)C(C)(C)C
CC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)cnc34)cc2F)n(n1)-c1ccccc1
C[C@H](NC(=O)c1ncnc(N)c1Cl)c1ncc(s1)C(=O)Nc1cc(c(Cl)cn1)C(F)(F)F |r|
COC(=O)Nc1nc2cc(ccc2[nH]1)C1(O)N(C(=O)c2ccccc12)c1cc(Cl)ccc1C
CC(C)(C)c1nc(c(s1)c2ccnc(n2)N)c3cccc(c3F)NS(=O)(=O)c4c(cccc4F)F
OCCn1cc(c(n1)-c1ccncc1)-c1ccc2\C(CCc2c1)=N\O
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccc2\C(CCc2c1)=N\O)-c1ccncc1
CC(C)(N)c1cc(cc(c1)C(F)(F)F)C(=O)NC1CCc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1
COc1cccc(c1)-n1cc(NC(=O)Cn2ccc(n2)-c2ccccn2)cn1
O=C(Cn1ccc2ccccc12)Nc1cnn(c1)-c1ccccc1
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccccc2)c1F
Clc1cccc(c1)-c1ccn(CC(=O)Nc2cnn(Cc3ccccc3)c2)n1
CCn1cc(NC(=O)Cn2ccc(n2)-c2ccccn2)cn1
Cn1cc(NC(=O)Cn2ccc(n2)-c2cccc(Cl)c2)cn1
COc1cccc(c1)-n1cc(NC(=O)Cn2ccc3ccccc23)cn1
COc1ccc(cc1)-n1cc(NC(=O)Cn2ccc3ccccc23)cn1
Cc1ccc(cc1)-n1cc(NC(=O)Cn2ccc3ccccc23)cn1
CCn1cc(NC(=O)Cn2ccc3ccccc23)cn1
COc1ccc(cc1)-n1cc(NC(=O)Cc2ccc(OC)c(OC)c2)cn1
COc1ccc(CC(=O)Nc2cnn(c2)-c2ccc(C)cc2)cc1OC
COc1ccc(CC(=O)Nc2cnn(Cc3ccccc3)c2)cc1OC
CCn1cc(NC(=O)Cc2ccc(OC)c(OC)c2)cn1
COc1ccc(CC(=O)Nc2cnn(C)c2)cc1OC
CCn1cc(NC(=O)Cn2ccc(n2)-c2cccc(Cl)c2)cn1
O=C(Cn1ccc(n1)-c1ccccn1)Nc1cnn(c1)-c1ccccc1
Cn1cc(NC(=O)Cn2ccc3ccccc23)cn1
Cn1cc(NC(=O)Cn2ccc(n2)-c2ccccn2)cn1
COc1cccc(c1)-n1cc(NC(=O)Cc2ccc(OC)c(OC)c2)cn1
COc1ccc(cc1)-n1cc(NC(=O)Cn2ccc(n2)-c2cccc(Cl)c2)cn1
O=C(Cn1ccc(n1)-c1ccccn1)Nc1cnn(Cc2ccccc2)c1
O=C(Cn1ccc2ccccc12)Nc1cnn(Cc2ccccc2)c1
COc1ccc(CC(=O)Nc2cnn(c2)-c2ccccc2)cc1OC
COc1ccc(cc1)-n1cc(NC(=O)Cn2ccc(n2)-c2ccccn2)cn1
Cc1c([nH]c2ccc(Cl)cc12)C(=O)NC(CO)Cc1ccccc1
COCCOc1cc2c(cc1OCCOC)ncnc2Nc3cccc(c3)C#C
CCc1c([nH]c2ccc(cc12)C(F)(F)F)C(=O)NC(CO)Cc1ccccc1
OCC(Cc1ccccc1)NC(=O)c1cc2cc(Cl)ccc2[nH]1
Clc1ccc2c(cc3n2cc(Cc2ccccc2)[nH]c3=O)c1
Cc1c2cc(Cl)ccc2n2cc(Cc3ccccc3)[nH]c(=O)c12
CCc1c2cc(ccc2n2cc(Cc3ccccc3)[nH]c(=O)c12)C(F)(F)F
O=C(Nc1cccc(c1)C(=O)Nc1ccc2[nH]ncc2c1)c1ccc(Oc2ccccc2)cc1
Brc1ccc(cc1)C(=O)Nc1cccc(c1)C(=O)Nc1ccc2[nH]ncc2c1
Clc1ccc(cc1)C(=O)Nc1cccc(c1)C(=O)Nc1ccc2[nH]ccc2c1
Fc1cccc(c1)C(=O)Nc1cccc(c1)C(=O)Nc1ccc2[nH]ncc2c1
Fc1ccc(cc1)C(=O)Nc1cccc(c1)C(=O)Nc1ccc2[nH]ncc2c1
Clc1ccc(cc1)C(=O)Nc1cccc(c1)C(=O)Nc1ccc2[nH]ncc2c1
FC(F)(F)c1ccc(cc1)C(=O)Nc1cccc(c1)C(=O)Nc1ccc2[nH]ncc2c1
Cc1cccc(n1)C(=O)Nc1cccc(c1)C(=O)Nc1ccc2[nH]ncc2c1
Clc1cccc(n1)C(=O)Nc1cccc(c1)C(=O)Nc1ccc2[nH]ncc2c1
Clc1cccc(OC(=O)Nc2cccc(c2)C(=O)Nc2ccc3[nH]ccc3c2)c1
O=C(Nc1cccc(c1)C(=O)Nc1ccc2[nH]ccc2c1)c1ccccc1
O=C(Nc1cccc(c1)C(=O)Nc1ccc2[nH]ccc2c1)c1ccc(Oc2ccccc2)cc1
Clc1cccc(n1)C(=O)Nc1cccc(c1)C(=O)Nc1ccc2[nH]ccc2c1
O=C(Nc1cccc(c1)C(=O)Nc1ccc2[nH]ncc2c1)c1ccccc1
CC(C)(C)c1ccc(cc1)C(=O)Nc1cccc(c1)C(=O)Nc1ccc2[nH]ncc2c1
Clc1ccnc(c1)C(=O)Nc1cccc(c1)C(=O)Nc1ccc2[nH]ncc2c1
Brc1ccc(nc1)C(=O)Nc1cccc(c1)C(=O)Nc1ccc2[nH]ncc2c1
O=C(Nc1ccc2[nH]ccc2c1)c1cccc(NC(=O)c2ccccn2)c1
Clc1cccc(c1)C(=O)Nc1cccc(c1)C(=O)Nc1ccc2[nH]ncc2c1
O=C(Nc1ccc2[nH]ncc2c1)c1cccc(NC(=O)c2ccccn2)c1
CNC(=O)c1ccc(Sc2ccc(NC(=O)Nc3ccc(F)c(c3)C(F)(F)F)cc2)nc1
CNC(=O)c1ccc(Sc2cccc(NC(=S)Nc3ccc(OC(F)(F)F)cc3)c2)nc1
CNC(=O)c1ccc(Sc2cccc(NC(=S)Nc3ccc(F)c(F)c3)c2)nc1
CNC(=O)c1ccc(Sc2cccc(NC(=S)Nc3cccc(c3)C(F)(F)F)c2)nc1
CNC(=O)c1ccc(Sc2ccc(NC(=S)Nc3ccc(Cl)cc3)cc2)nc1
CNC(=O)c1ccc(Sc2ccc(NC(=S)Nc3cccc(C)c3)cc2)nc1
CNC(=O)c1ccc(Sc2ccc(NC(=S)Nc3cccc(c3)C(F)(F)F)cc2)nc1
CNC(=O)c1ccc(Sc2ccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)cc2)nc1
CNC(=O)c1ccc(Sc2cccc(NC(=S)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)c2)nc1
CNC(=O)c1ccc(Sc2cccc(NC(=S)Nc3ccc(F)c(Cl)c3)c2)nc1
CNC(=O)c1ccc(Sc2cccc(NC(=S)Nc3ccc(Cl)c(c3)C(F)(F)F)c2)nc1
CNC(=O)c1ccc(Sc2cccc(NC(=S)Nc3ccc(F)c(c3)C(F)(F)F)c2)nc1
CNC(=O)c1ccc(Sc2ccc(NC(=S)Nc3ccc(F)c(c3)C(F)(F)F)cc2)nc1
CNC(=O)c1ccc(Sc2ccc(NC(=S)Nc3ccc(Cl)c(c3)C(F)(F)F)cc2)nc1
CNC(=O)c1ccc(Sc2ccc(NC(=S)Nc3ccc(F)c(F)c3)cc2)nc1
CNC(=O)c1ccc(Sc2ccc(NC(=S)Nc3ccc(OC(F)(F)F)cc3)cc2)nc1
CNC(=O)c1ccc(Sc2cccc(NC(=S)Nc3ccc(Cl)cc3)c2)nc1
CNC(=O)c1ccc(Sc2ccc(NC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)cc2)nc1
CC(C)n1nc(C#Cc2cccc3cc(ncc23)-c2cccc(c2)C(F)(F)F)c2c(N)ncnc12
CC(C)n1nc(C#Cc2cccc3cc(ncc23)-c2ccc(Cl)c(c2)C(F)(F)F)c2c(N)ncnc12
CC(C)n1nc(C#Cc2cccc3cc(ncc23)-c2ccc(CN3CCN(C)CC3)cc2)c2c(N)ncnc12
CC(C)n1nc(C#Cc2cccc3cc(ncc23)-c2ccc(Cl)cc2)c2c(N)ncnc12
CC(C)n1nc(C#Cc2cccc(NC(=O)c3cccc(c3)C(F)(F)F)c2)c2c(N)ncnc12
CC(C)n1nc(C#Cc2c(C)ccc3cc(ncc23)-c2cccc(c2)C(F)(F)F)c2c(N)ncnc12
CCn1nc(C#Cc2cccc3cc(ncc23)-c2cccc(c2)C(F)(F)F)c2c(N)ncnc12
CC(C)n1nc(C#Cc2cccc3cc(ncc23)-c2ccc(C)cc2)c2c(N)ncnc12
NCCCCCCC(=S)N\N=C1/CC2(CCCCC2)Oc2c1ccc1ccccc21
Clc1ccc(NC(=O)N\N=C2/CC3(CCCC3)Oc3ccccc23)cc1
O=C(N\N=C1/CC2(CCCCC2)Oc2c1ccc1ccccc21)C1C2CC3CC(C2)CC1C3 |TLB:32:31:29:25.26.27,THB:27:26:23:30.28.29,27:28:23:25.32.26,1:23:29:25.26.27,32:26:23.31.30:29,(33.82,-4.03,;33.82,-5.57,;35.16,-6.34,;36.49,-5.57,;37.83,-6.33,;37.83,-7.88,;39.16,-8.64,;37.83,-9.4,;37.82,-10.94,;39.14,-11.72,;40.48,-10.95,;40.49,-9.41,;40.51,-7.87,;40.49,-6.33,;39.15,-5.56,;39.16,-4.01,;40.49,-3.24,;41.83,-4.01,;43.15,-3.23,;44.49,-3.99,;44.5,-5.54,;43.16,-6.32,;41.83,-5.55,;32.49,-6.34,;31.27,-7.59,;29.96,-7.08,;28.55,-7.4,;28.51,-8.93,;29.9,-9.53,;31.25,-9.08,;30.96,-8.32,;30.99,-6.73,;29.59,-6.14,)|
Fc1ccc(Oc2ccc3nc(NC(=O)COCCOCCOCCOCCOCC(=O)Nc4nc5ccc(Oc6ccc(F)c(NC(=O)Cc7cccc(c7)C(F)(F)F)c6)c(C#N)c5s4)sc3c2C#N)cc1NC(=O)Cc1cccc(c1)C(F)(F)F
Fc1ccc(Oc2ccc3nc(NC(=O)COCCOCCOCC(=O)Nc4nccs4)sc3c2C#N)cc1NC(=O)Cc1cccc(c1)C(F)(F)F
c1cc(cc(c1)C(F)(F)F)CC(=O)Nc2cc(ccc2F)Oc3ccc4c(c3C#N)sc(n4)NC(=O)C5CC5
COCCOCC(=O)Nc1nc2ccc(Oc3ccc(F)c(NC(=O)Cc4cccc(c4)C(F)(F)F)c3)c(C#N)c2s1
Fc1ccc(Oc2ccc3nc(NC(=O)COCCOCCOCC(=O)Nc4nc5ccc(Oc6ccc(F)c(NC(=O)Cc7cccc(c7)C(F)(F)F)c6)c(C#N)c5s4)sc3c2C#N)cc1NC(=O)Cc1cccc(c1)C(F)(F)F
Fc1ccc(Oc2ccc3nc(NC(=O)COCCOCCOCCOCCOCCOCCOCC(=O)Nc4nc5ccc(Oc6ccc(F)c(NC(=O)Cc7cccc(c7)C(F)(F)F)c6)c(C#N)c5s4)sc3c2C#N)cc1NC(=O)Cc1cccc(c1)C(F)(F)F
Fc1ccc(Oc2ccc3nc(NC(=O)COCCOCCOCCOCC(=O)Nc4nc5ccc(Oc6ccc(F)c(NC(=O)Cc7cccc(c7)C(F)(F)F)c6)c(C#N)c5s4)sc3c2C#N)cc1NC(=O)Cc1cccc(c1)C(F)(F)F
Fc1ccc(Oc2ccc3nc(NC(=O)COCC(=O)Nc4nc5ccc(Oc6ccc(F)c(NC(=O)Cc7cccc(c7)C(F)(F)F)c6)c(C#N)c5s4)sc3c2C#N)cc1NC(=O)Cc1cccc(c1)C(F)(F)F
Cc1nc2ccc(c(C)c2c(=O)[nH]1)-c1ccnc2ccccc12
C[C@@]12[C@@H]([C@@H](C[C@@H](O1)n3c4ccccc4c5c3c6n2c7ccccc7c6c8c5C(=O)NC8)NC)OC
S=C(Nc1ccccc1)N1N=C(CC1c1ccc2OCCOc2c1)c1cccs1 |c:11|
Clc1ccc(cc1Cl)C1=NN(C(C1)c1ccc2OCCOc2c1)C(=S)Nc1ccccc1 |t:9|
Clc1ccc(cc1)C1=NN(C(C1)c1ccc2OCCOc2c1)C(=S)Nc1ccccc1 |t:8|
COc1ccccc1C1=NN(C(C1)c1ccc2OCCOc2c1)C(=S)Nc1ccccc1 |t:9|
Cc1ccc(cc1C)C1=NN(C(C1)c1ccc2OCCOc2c1)C(=S)Nc1ccccc1 |t:9|
Cc1ccc(cc1)C1=NN(C(C1)c1ccc2OCCOc2c1)C(=S)Nc1ccccc1 |t:8|
Brc1ccccc1C1=NN(C(C1)c1ccc2OCCOc2c1)C(=S)Nc1ccccc1 |t:8|
Clc1cccc(c1)C1=NN(C(C1)c1ccc2OCCOc2c1)C(=S)Nc1ccccc1 |t:8|
Fc1ccc(cc1)C1=NN(C(C1)c1ccc2OCCOc2c1)C(=S)Nc1ccccc1 |t:8|
CSc1ccc(cc1)C1=NN(C(C1)c1ccc2OCCOc2c1)C(=S)Nc1ccccc1 |t:9|
S=C(Nc1ccccc1)N1N=C(CC1c1ccc2OCCOc2c1)c1ccc(OCc2ccccc2)cc1 |c:11|
[O-][N+](=O)c1ccc(cc1)C1=NN(C(C1)c1ccc2OCCOc2c1)C(=S)Nc1ccccc1 |t:10|
COc1cccc(c1)C1=NN(C(C1)c1ccc2OCCOc2c1)C(=S)Nc1ccccc1 |t:9|
FC(F)(F)c1ccc(cc1)C1=NN(C(C1)c1ccc2OCCOc2c1)C(=S)Nc1ccccc1 |t:11|
S=C(Nc1ccccc1)N1N=C(CC1c1ccc2OCCOc2c1)c1ccccc1 |c:11|
Brc1ccc(cc1)C1=NN(C(C1)c1ccc2OCCOc2c1)C(=S)Nc1ccccc1 |t:8|
COc1ccc(cc1)-c1nc2sc(cn2n1)-c1ccc(Cl)cc1
CNC(=O)c1cc(Cn2ccc3cc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)ccc23)ccn1
CN1CCN(CCNc2nccc(n2)C2(CC2)C(=O)Nc2cc(ccc2C)C(=O)Nc2ccc(c(Cl)c2)C(F)(F)F)CC1
CN1CCN(CCCNc2cc(ncn2)C2(CC2)C(=O)Nc2cc(ccc2C)C(=O)Nc2ccc(c(Cl)c2)C(F)(F)F)CC1
COc1cc2c3c(n[nH]c3ncc2cc1-c1c(F)ccc(NS(=O)(=O)CCCF)c1F)C1CC1 |(22.49,-22.5,;23.83,-23.27,;23.84,-24.81,;22.53,-25.58,;22.53,-27.1,;21.19,-27.89,;19.72,-27.42,;18.82,-28.66,;19.73,-29.91,;21.19,-29.43,;22.54,-30.19,;23.87,-29.43,;23.86,-27.88,;25.18,-27.1,;25.18,-25.57,;26.51,-24.81,;27.85,-25.57,;27.85,-27.11,;29.18,-24.8,;29.17,-23.26,;27.83,-22.49,;27.82,-20.94,;29.14,-20.17,;28.36,-18.83,;29.91,-18.82,;30.49,-20.93,;31.82,-20.15,;33.16,-20.92,;34.49,-20.14,;26.5,-23.27,;25.16,-22.5,;19.24,-25.95,;19.55,-24.45,;18.09,-24.93,)|
Fc1ccc(cc1)-c1nc2sccn2c1-c1ccnc(NC2CCCN(C2)S(=O)(=O)c2ccc(F)cc2)n1
Oc1ccc(cc1)S(=O)(=O)NCCNc1nccc(n1)-c1c(nc2sccn12)-c1ccc(F)cc1
CNC(=O)c1cc(Cn2cc(F)c3cc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)ccc23)ccn1
CNc1ncc2cc(c(C)nc2n1)-c1cc(NC(=O)NCCC(C)(C)C)c(F)cc1C
CNc1cc2n(C3CCOC3)c(=O)c(cc2cn1)-c1ccc(F)c(NC(=O)Nc2cc(no2)C(C)(C)C)c1
COc1cc(O)c(C(O)=O)c(c1)C1=C(C)C[C@@H](O)C1=O |r,wD:16.17,c:13,(10.48,-22.79,;11.26,-21.46,;10.49,-20.12,;11.26,-18.8,;10.49,-17.47,;11.26,-16.14,;8.97,-17.47,;8.2,-16.14,;8.96,-14.8,;6.65,-16.13,;8.21,-18.79,;8.97,-20.12,;6.66,-18.79,;5.76,-17.54,;4.98,-16.2,;4.29,-18.01,;4.29,-19.55,;3.04,-20.45,;5.75,-20.03,;6.22,-21.5,)|
COc1cc2c(C(=O)OC22C(C)CC(=O)C2=O)c(O)c1
COc1cc(O)c2c(c1)c1c(C)cc(O)cc1oc2=O
Cc1cc(O)cc2oc(=O)c3c(O)cc(OS(O)(=O)=O)cc3c12
Cc1cc(O)cc2oc(=O)c3c(O)cc(O)cc3c12
COc1cc(O)c2c(c1)-c1cc(O)c(O)cc1COC2=O
[H][C@]12[C@@H](O)CC(=O)c3c(O)ccc(-c4ccc(O)c5C(=O)CC[C@]1(O)c45)c23 |r|
COc1cc(O)c(C(O)=O)c(c1)-c1cc(O)c(O)cc1C
COc1cc(O)c2c(c1)c1c(C)cc(O)c(O)c1oc2=O
Cc1cc(O)c(O)cc1-c1cc(O)cc(O)c1C(O)=O
FC(F)(F)c1cccc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)c3ccccc23)c1
Fc1cc(Oc2ccnc3[nH]c(=O)[nH]c23)ccc1NC(=O)Nc1cccc(SC(F)(F)F)c1
Cn1c2c(Oc3ccc(NC(=O)Nc4cccc(c4)C(F)(F)F)c4ccccc34)ccnc2[nH]c1=O
Fc1cc(Oc2ccnc3[nH]c(=O)[nH]c23)ccc1NC(=O)Nc1cccc(c1)C(F)(F)F
FC(F)(F)c1ccc(N2CCOCC2)c(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)c3ccccc23)c1
Cn1c2c(Oc3ccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c4ccccc34)ccnc2[nH]c1=O
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2Cl)ccc1Cl
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2C(F)(F)F)ccc1Cl
Cn1c2c(Oc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)c4ccccc34)ccnc2[nH]c1=O
Cn1c2c(Oc3ccc(NC(=O)Nc4cccc(SC(F)(F)F)c4)c4ccccc34)ccnc2[nH]c1=O
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)c3ccccc23)ccc1Cl
Cc1cc(Oc2ccnc3[nH]c(=O)[nH]c23)ccc1NC(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)c2ccccc12)C(F)(F)F
Fc1cc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)ccc1Oc1ccnc2[nH]c(=O)[nH]c12
CSc1cc(Oc2ccnc3[nH]c(=O)[nH]c23)ccc1NC(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
Cn1c2c(Oc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)c(F)c3)ccnc2[nH]c1=O
Cn1c2c(Oc3ccc(NC(=O)Nc4cccc(c4)C(C)(C)C)c4ccccc34)ccnc2[nH]c1=O
CSc1cc(Oc2ccnc3[nH]c(=O)[nH]c23)ccc1NC(=O)Nc1cccc(c1)C(F)(F)F
CS(=O)(=O)c1cc(Oc2ccnc3[nH]c(=O)[nH]c23)ccc1NC(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
CC(C)(C)c1cccc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)c3ccccc23)c1
Cn1c2nccc(Oc3ccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c4ccccc34)c2[nH]c1=O
Fc1cc(Oc2ccnc3[nH]c(=O)[nH]c23)ccc1NC(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)ccc1Cl
CN(C)c1cc(Oc2ccnc3[nH]c(=O)[nH]c23)ccc1NC(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
Cn1c2c(Oc3ccc(NC(=O)c4cccc(OC(F)(F)F)c4)c4ccccc34)ccnc2[nH]c1=O
COc1cc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)ccc1Oc1ccnc2[nH]c(=O)[nH]c12
Cc1cc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)ccc1Oc1ccnc2[nH]c(=O)[nH]c12
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2-c2ccccc2)ccc1Cl
FC(F)(F)Oc1cccc(CC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)c3ccccc23)c1
COc1cc(Oc2ccnc3[nH]c(=O)[nH]c23)ccc1NC(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
Fc1ccc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)c3ccccc23)cc1F
Fc1cccc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)c3ccccc23)c1
Cn1c2c(Oc3ccc(NC(=O)c4cccc(SC(F)(F)F)c4)c4ccccc34)ccnc2[nH]c1=O
Fc1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2F)cc(c1)C(F)(F)F
CSc1cc(Oc2ccnc3[nH]c(=O)[nH]c23)ccc1NC(=O)Nc1cc(ccc1F)C(F)(F)F
Cc1c(C)c(Oc2ccnc3[nH]c(=O)[nH]c23)ccc1NC(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
Cn1c2nccc(Oc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)c4ccccc34)c2[nH]c1=O
COc1cc(NC(=O)Nc2cccc(c2)C(F)(F)F)ccc1Oc1ccnc2[nH]c(=O)[nH]c12
FC(F)(F)c1cccc(CC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)c3ccccc23)c1
Cn1c2nccc(Oc3ccc(NC(=O)Nc4cccc(c4)C(C)(C)C)c4ccccc34)c2[nH]c1=O
COc1cc(O)c2C(=O)C3=C([C@@H](O)[C@](C)(O)[C@H](O)[C@H]3O)C(=O)c2c1 |r,t:9|
COc1cc(O)c2C(=O)C3=C([C@@H](O)[C@](C)(O)[C@H](O)[C@H]3O)C(=O)c2c1-c1c(O)c2C(=O)c3cc(O)c(C)cc3C(=O)c2cc1OC |r,wU:18.19,11.11,13.13,wD:16.16,t:9,(-6.62,-6.52,;-5.29,-5.75,;-3.96,-6.52,;-3.96,-8.06,;-2.63,-8.83,;-2.63,-10.37,;-1.3,-8.07,;.04,-8.83,;.05,-10.37,;1.38,-8.06,;1.38,-6.5,;2.72,-5.72,;2.71,-4.19,;4.06,-6.5,;4.82,-5.16,;5.38,-7.27,;4.07,-8.06,;5.4,-8.82,;2.72,-8.83,;2.72,-10.37,;.03,-5.73,;.02,-4.19,;-1.3,-6.52,;-2.63,-5.75,;-2.6,-3.5,;-1.27,-2.73,;.06,-3.5,;-1.26,-1.19,;.06,-.41,;1.4,-1.16,;.05,1.13,;1.37,1.91,;1.36,3.45,;2.68,4.23,;.01,4.21,;-.01,5.74,;-1.31,3.42,;-1.29,1.89,;-2.62,1.11,;-3.96,1.87,;-2.6,-.43,;-3.93,-1.19,;-3.93,-2.74,;-5.26,-3.5,;-6.59,-2.73,)|
COc1cc(O)c2C(=O)c3cc(O)c(C)cc3C(=O)c2c1
COc1cc(O)c2C(=O)c3c(O)c(O)c(C)cc3C(=O)c2c1
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Sc2ccnc3[nH]c(=O)[nH]c23)cc1)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3n(C)c(=O)n(C)c23)cc1F)C(C)(C)C
Cc1ccc(cn1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3n(C)c(=O)[nH]c23)cc1F)C(C)(C)C
CC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2F)n(n1)-c1ccccc1
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3n(C)c(=O)[nH]c23)c2ccccc12)C(C)(C)C
Cn1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3n(C)c(=O)[nH]c23)c2ccccc12)C(C)(C)C
Cn1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)n(C)c23)c2ccccc12)C(C)(C)C
Cn1c2c(Oc3ccc(NC(=O)Nc4cc(nn4-c4cccnc4)C(C)(C)C)c4ccccc34)ccnc2[nH]c1=O
Cn1c2c(Oc3ccc(NC(=O)Nc4cc(nn4-c4ccc(F)cc4)C(C)(C)C)c4ccccc34)ccnc2[nH]c1=O
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)c2ccccc12)C(C)(C)C
CC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)c3ccccc23)n(n1)-c1ccc(F)cc1
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3n(C)c(=O)n(C)c23)cc1)C(C)(C)C
Cn1c2nccc(Oc3ccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)cc3)c2[nH]c1=O
Cn1c2c(Oc3ccc(NC(=O)Nc4cc(nn4-c4cccnc4)C(C)(C)C)cc3)ccnc2[nH]c1=O
Cn1c2c(Oc3ccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)cc3)ccnc2[nH]c1=O
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)n(C)c23)cc1)C(F)(F)F
Cn1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)n(C)c23)cc1)C(C)(C)C
O=C(Nc1nnc(s1)C1CCCO1)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1
CC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)n(n1)-c1ccccc1
CC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)n(n1)-c1ccc(Cl)cc1
CC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)n(n1)-c1ccc(F)cc1
CC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)n(n1)-c1ccc(F)cc1F
CC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)n(Cc2ccccc2)n1
CC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)n(n1)C(C)(C)C
CSc1cc(Oc2ccnc3[nH]c(=O)[nH]c23)ccc1NC(=O)Nc1cc(nn1-c1ccc(C)cc1)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1F)C(C)(C)C
Cn1c2nccc(Oc3ccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c4ccccc34)c2[nH]c1=O
Cn1c2c(Oc3ccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c4ccccc34)ccnc2[nH]c1=O
Cn1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)c2ccccc12)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3n(C)c(=O)[nH]c23)cc1)C(C)(C)C
Cn1c2c(Oc3ccc(NC(=O)Nc4cc(nn4-c4ccc(F)cc4)C(C)(C)C)cc3)ccnc2[nH]c1=O
CC(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)n(n1)-c1ccccc1
Cc1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)n(n1)-c1ccc(Cl)cc1
Cn1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1)C(C)(C)C
CCCn1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1)C(C)(C)C
Cn1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3n(C)c(=O)[nH]c23)cc1)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)[nH]c23)cc1)C(C)(C)C
Cn1c2nccc(Oc3ccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c(F)c3)c2n(C)c1=O
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)n(C)c23)cc1)C(C)(C)C
Cn1c2c(Oc3ccc(NC(=O)Nc4cc(nn4-c4ccccc4)C4CC4)cc3)ccnc2[nH]c1=O
CC(C)(C)c1cc(NC(=O)Nc2ccc(Sc3ccnc4[nH]c(=O)[nH]c34)cc2)n(n1)-c1ccccc1
CC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)c3ccccc23)n(n1)-c1ccccc1
CC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)n(n1)-c1ccccn1
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)n(C)c23)c2ccccc12)C(C)(C)C
CC(C)(C)c1csc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)[nH]c34)cc2)n1
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2ccnc3ncc(=O)[nH]c23)cc1F)C(F)(F)F
Cc1nc2nccc(Oc3ccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c(F)c3)c2[nH]c1=O
Nc1nc2c(Oc3ccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c(F)c3)ccnc2[nH]c1=O
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]nnc23)cc1F)C(F)(F)F
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]cnc23)cc1F)C(F)(F)F
CN(C)Cc1nc2c(Oc3ccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c(F)c3)ccnc2[nH]1
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)c(=O)[nH]c34)cc2)ccc1Cl
Fc1cc(Oc2ccnc3[nH]c(=O)cnc23)ccc1NC(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
Cn1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)cnc23)cc1F)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)cnc23)cc1F)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)c(=O)[nH]c23)cc1F)C(C)(C)C
CSc1cc(Oc2ccnc3[nH]c(=O)cnc23)ccc1NC(=O)Nc1cc(ccc1F)C(F)(F)F
CSc1cc(Oc2ccnc3[nH]c(=O)c(=O)[nH]c23)ccc1NC(=O)Nc1cc(ccc1F)C(F)(F)F
CSc1cc(Oc2ccnc3[nH]c(=O)c(C)nc23)ccc1NC(=O)Nc1cc(ccc1F)C(F)(F)F
CSc1cc(Oc2ccnc3[nH]c(=O)c(C)nc23)ccc1NC(=O)Nc1cc(nn1-c1ccc(C)cc1)C(C)(C)C
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)c(nc23)C(F)(F)F)c2ccccc12)C(F)(F)F
CC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)cnc34)c3ccccc23)n(n1)-c1ccccc1
Cc1nc2c(Oc3ccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c4ccccc34)ccnc2[nH]c1=O
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)cnc23)c2ccccc12)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)c(C)nc23)c2ccccc12)C(C)(C)C
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2ccnc3ncc(=O)[nH]c23)cc1)C(F)(F)F
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3ncc(=O)[nH]c23)cc1)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3nc(N)c(=O)[nH]c23)cc1F)C(C)(C)C
CSc1cc(Oc2ccnc3ncc(=O)[nH]c23)ccc1NC(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
CSc1cc(Oc2ccnc3ncc(=O)[nH]c23)ccc1NC(=O)Nc1cc(nn1-c1ccccc1)C(C)(C)C
Cc1nc2nccc(Oc3ccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c4ccccc34)c2[nH]c1=O
Nc1nc2nccc(Oc3ccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c4ccccc34)c2[nH]c1=O
CC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc4ncc(=O)[nH]c34)c3ccccc23)n(n1)-c1ccccc1
Cc1nc2nccc(Oc3ccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c4ccccc34)c2[nH]c1=O
CN(C)c1nc2c(Oc3ccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c(F)c3)ccnc2[nH]1
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3NC(=O)CNc23)cc1F)C(C)(C)C
Fc1ccc(cc1NC(=O)Nc1cccc(Oc2ccnc3[nH]c(=O)cnc23)c1)C(F)(F)F
Fc1ccc(cc1NC(=O)Nc1cccc(Oc2ccnc3ncc(=O)[nH]c23)c1)C(F)(F)F
CC(C)(C)c1cc(NC(=O)Nc2cccc(Oc3ccnc4ncc(=O)[nH]c34)c2)n(n1)-c1ccccc1
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1cccc(Oc2ccnc3[nH]c(=O)cnc23)c1)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1cccc(Oc2ccnc3[nH]c(=O)c(C)nc23)c1)C(C)(C)C
FC(F)(F)Oc1cccc(c1)C(=O)Nc1cccc(Oc2ccnc3ncc(=O)[nH]c23)c1
CC(C)(C)c1cccc(c1)C(=O)Nc1cccc(Oc2ccnc3ncc(=O)[nH]c23)c1
Cc1nc2c(Oc3cccc(NC(=O)c4cccc(c4)C(C)(C)C)c3)ccnc2[nH]c1=O
CN1CCN(CC1)c1cnc2c(Oc3ccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c(F)c3)ccnc2n1
CN1CCN(CC1)c1cnc2c(Oc3ccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c(F)c3)ccnc2n1
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2ccnc3nc(cnc23)N2CCOCC2)cc1F)C(F)(F)F
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3nc(cnc23)N2CCOCC2)cc1F)C(C)(C)C
CNc1cnc2c(Oc3ccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c(F)c3)ccnc2n1
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)cnc23)cc1F)C(F)(F)F
Nc1nc2nccc(Oc3ccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c(F)c3)c2[nH]c1=O
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(S)nc23)cc1F)C(F)(F)F
CN(C)c1nc2c(Oc3ccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c(F)c3)ccnc2[nH]1
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)cnc34)cc2)ccc1Cl
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)c(N)nc23)cc1F)C(C)(C)C
CSc1cc(Oc2ccnc3[nH]c(=O)cnc23)ccc1NC(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
CSc1cc(Oc2ccnc3[nH]c(=O)c(C)nc23)ccc1NC(=O)Nc1cc(nn1-c1ccccc1)C(C)(C)C
Cc1nc2c(Oc3ccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c4ccccc34)ccnc2[nH]c1=O
CC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)c(N)nc34)c3ccccc23)n(n1)-c1ccccc1
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)c(N)nc23)c2ccccc12)C(C)(C)C
Fc1cc(Oc2ccnc3ncc(=O)[nH]c23)ccc1NC(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
CC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc4ncc(=O)[nH]c34)cc2F)n(n1)-c1ccccc1
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2ccnc3ncc(=O)[nH]c23)c2ccccc12)C(F)(F)F
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2ccnc3nc(c(=O)[nH]c23)C(F)(F)F)c2ccccc12)C(F)(F)F
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(S)nc23)cc1F)C(C)(C)C
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2ccnc3NCC(=O)Nc23)cc1)C(F)(F)F
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1cccc(Oc2ccnc3ncc(=O)[nH]c23)c1)C(C)(C)C
CC(C)(C)c1cc(NC(=O)c2cccc(Oc3ccnc4[nH]c(=O)cnc34)c2)n(n1)-c1ccccc1
CN(C)c1cnc2c(Oc3ccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c(F)c3)ccnc2n1
CN(C)c1cnc2c(Oc3ccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c(F)c3)ccnc2n1
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccnc4ncc(=O)[nH]c34)cc2)ccc1Cl
FC(F)(F)Oc1cccc(c1)C(=O)Nc1cccc(Oc2ccnc3[nH]c(=O)cnc23)c1
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]nnc23)cc1F)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3nc(C)c(=O)[nH]c23)c2ccccc12)C(C)(C)C
CC(C)(C)c1cc(NC(=O)Nc2cccc(Oc3ccnc4[nH]c(=O)cnc34)c2)n(n1)-c1ccccc1
CC(C)(C)c1cccc(c1)C(=O)Nc1cccc(Oc2ccnc3[nH]c(=O)cnc23)c1
Cc1nc2c(Oc3ccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c(F)c3)ccnc2[nH]c1=O
CSc1cc(Oc2ccnc3[nH]c(=O)c(=O)[nH]c23)ccc1NC(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
CSc1cc(Oc2ccnc3[nH]c(=O)cnc23)ccc1NC(=O)Nc1cc(nn1-c1ccc(C)cc1)C(C)(C)C
Nc1nc2c(Oc3ccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c4ccccc34)ccnc2[nH]c1=O
CSc1cc(Oc2ccnc3ncc(=O)[nH]c23)ccc1NC(=O)Nc1cc(ccc1F)C(F)(F)F
Fc1ccc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)c(=O)[nH]c23)cc1F)C(F)(F)F
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(Oc2ccnc3[nH]c(=O)cnc23)cc1)C(C)(C)C
Cc1nc2nccc(Oc3ccc(NC(=O)Nc4cc(nn4-c4ccccc4)C(C)(C)C)c(F)c3)c2[nH]c1=O
CC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc4nc(cnc34)N3CCOCC3)cc2F)n(n1)-c1ccccc1
CC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc4nc(N)c(=O)[nH]c34)c3ccccc23)n(n1)-c1ccccc1
Oc1nc2c(Oc3cccc(NC(=O)c4cccc(OC(F)(F)F)c4)c3)ccnc2[nH]c1=O
CC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc4[nH]c(=O)c(=O)[nH]c34)cc2F)n(n1)-c1ccccc1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc(cc1)-c1cc[nH]n1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc(cc1)-c1n[nH]cc1C
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc(cc1)-c1n[nH]cc1Cl
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2-c3[nH]ncc3CCc2c1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2c3[nH]ncc3ccc2c1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc-2c(Cc3nn[nH]c-23)c1
CN1CCN(CC1)c1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc-2c(Cc3cn[nH]c-23)c1
CN(C)CCN1CCN(CC1)C(=O)c1cc(c(o1)-c1ccncc1)-c1ccc-2c(Cc3cn[nH]c-23)c1
O=C(N1CCNCC1)c1cc(c(o1)-c1ccncc1)-c1ccc-2c(Cc3cn[nH]c-23)c1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc-2c(Cc3cn[nH]c-23)c1
O=C(N1CCOCC1)c1cc(c(o1)-c1ccncc1)-c1ccc-2c(Cc3cn[nH]c-23)c1
CN1CCN(CC1)C(=O)c1cc(c(o1)-c1ccncc1)-c1ccc-2c(Cc3cn[nH]c-23)c1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2C3=NNC(=O)CC3Cc2c1 |t:30|
CN(C)CCN1CCN(CC1)C(=O)c1cc(c(o1)-c1ccncc1)-c1ccc-2c(Cc3cnn(C)c-23)c1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc(cc1)-c1n[nH]cc1C#N
C1c2cn[nH]c2-c2ccc(cc12)-c1nc([nH]c1-c1ccncc1)C1CCNCC1
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NS(=O)(=O)NCC(F)F)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NS(=O)(=O)C4CC4)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NS(=O)(=O)CC4CC4)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NS(=O)(=O)CCCF)c3F)cc12
CCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(OC)c3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]ccc3c2)c1C
CCCS(=O)(=O)Nc1cc(F)c(F)c(C(=O)Nc2cnc3[nH]ccc3c2)c1F
CCCS(=O)(=O)Nc1cc(F)cc(C(=O)Nc2cnc3[nH]ccc3c2)c1F
CCCS(=O)(=O)Nc1cccc(C(=O)Nc2cnc3[nH]ccc3c2)c1F
CCCS(=O)(=O)Nc1ccc(Cl)c(C(=O)Nc2cnc3[nH]ccc3c2)c1Cl
CCCS(=O)(=O)Nc1ccc(OC)c(C(=O)Nc2cnc3[nH]nc(OC)c3c2)c1F
CCCS(=O)(=O)Nc1ccc(Cl)c(c1)C(=O)Nc1cnc2[nH]nc(OC)c2c1
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NS(=O)(=O)c4ccco4)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NS(=O)(=O)c4cccs4)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NS(=O)(=O)c4ccccn4)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NS(=O)(=O)c4ccc(F)cc4)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NS(=O)(=O)c4cccc(F)c4)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NS(=O)(=O)c4ccccc4)c3F)cc12
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(O[C@@H]4CCOC4)c3c2)c1F |r|
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(OCC)c3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]cc(c3c2)C(F)(F)F)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]cc(I)c3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(CC)c3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(I)c3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(Br)c3c2)c1F
Fc1ccc(NS(=O)(=O)N2CCCC2)c(F)c1C(=O)Nc1cnc2[nH]ccc2c1
CN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]ccc3c2)c1F
Fc1ccc(NS(=O)(=O)C2CC2)c(F)c1C(=O)Nc1cnc2[nH]ccc2c1
Fc1ccc(NS(=O)(=O)CC2CC2)c(F)c1C(=O)Nc1cnc2[nH]ccc2c1
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NS(=O)(=O)N4CCCC4)c3F)cc12
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(OC)c3c2)c1F
CCCS(=O)(=O)Nc1cccc(C(=O)Nc2cnc3[nH]nc(OC)c3c2)c1F
CCCS(=O)(=O)Nc1ccc(Cl)c(C(=O)Nc2cnc3[nH]nc(OC)c3c2)c1F
CCNS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(OC)c3c2)c1F
CCCS(=O)(=O)Nc1cc(F)c(F)c(C(=O)Nc2cnc3[nH]nc(OC)c3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(OC)c3c2)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]ccc3c2)c1F
FCCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]ccc3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(c1)C(=O)Nc1cnc2[nH]ccc2c1
CCCS(=O)(=O)Nc1ccc(F)c(c1)C(=O)Nc1cnc2[nH]nc(OC)c2c1
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]ccc3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(c3c2)C(F)(F)F)c1F
Fc1ccc(NS(=O)(=O)CCC(F)(F)F)c(F)c1C(=O)Nc1cnc2[nH]ccc2c1
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NS(=O)(=O)c4ccccc4F)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NS(=O)(=O)c4cccnc4)c3F)cc12
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(OCC4CCC4)c3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]cc(C)c3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(C)c3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]ncc3c2)c1F
CCCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]ccc3c2)c1F
CCCS(=O)(=O)Nc1ccc(Cl)c(C(=O)Nc2cnc3[nH]nc(OC)c3c2)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(OC)c3c2)c1C(F)(F)F
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NS(=O)(=O)NC(C)C)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NS(=O)(=O)CC(C)C)c3F)cc12
CCCS(=O)(=O)Nc1ccc(C)c(C(=O)Nc2cnc3[nH]ccc3c2)c1F
CCCS(=O)(=O)Nc1ccc(Cl)c(c1)C(=O)Nc1cnc2[nH]ccc2c1
CCCS(=O)(=O)Nc1cc(F)cc(C(=O)Nc2cnc3[nH]nc(OC)c3c2)c1F
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NS(=O)(=O)Cc4ccccc4)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NS(=O)(=O)c4cn(C)cn4)c3F)cc12
CCCS(=O)(=O)Nc1ccc(Cl)c(C(=O)Nc2cnc3[nH]ccc3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(OC)c3c2)c1OC
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(OCC4COC4)c3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]cc(Br)c3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(OCC(F)(F)F)c3c2)c1F
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NS(=O)(=O)N(C)C)c3F)cc12
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]cc(CC)c3c2)c1F
CC(C)CS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]ccc3c2)c1F
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NS(=O)(=O)c4cc(F)ccc4F)c3F)cc12
Fc1ccc(NS(=O)(=O)CC(F)(F)F)c(F)c1C(=O)Nc1cnc2[nH]ccc2c1
COc1cc2ncnc(Nc3ccc(NC(=O)Nc4cc(on4)C(C)(C)C)cc3)c2cc1OC
COc1cc2ncnc(Nc3cccc(NC(=O)Nc4cc(on4)C(C)(C)C)c3)c2cc1OC
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(C(C)C)c3c2)c1F
CC(C)CS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(C4CC4)c3c2)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(C4CC4)c3c2)c1F
FCCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(C4CC4)c3c2)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(C4CC4)c3c2)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(OC)c3c2)c1Cl
CCCS(=O)(=O)Nc1ccc(Cl)c(C(=O)Nc2cnc3[nH]ncc3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]cnc3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2ccc(N)nc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cccnc2)c1F
CCCS(=O)(=O)Nc1ccc(c(c1F)C(=O)Nc2cc(c(nc2)N)Br)F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(N(C)C)c3c2)c1F
CNC(=O)c1cc(Oc2ccc3nc(Nc4cccc(c4)C(C)(C)C)ccc3c2)ccn1
CCc1ccccc1Nc1ncc2cc(Oc3ccnc(c3)C(=O)NC)ccc2n1
CNC(=O)c1cc(Oc2ccc3nc(Nc4cccc(Br)c4)ncc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4cccc(c4)C(C)(C)C)ncc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4cccc(c4)C(F)(F)F)ncc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4ccc(F)cc4)ncc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4ccc(Br)cc4)ncc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4ccc(cc4)C(C)C)ncc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4ccc(OC)cc4)ncc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4ccc(OC(F)(F)F)cc4)ncc3c2)ccn1
OCCNC(=O)c1cc(Oc2ccc3nc(Nc4ccc(Br)cc4)ncc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4ccccc4Br)ncc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4ccccc4Oc4ccccc4)ncc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4cccc(c4)C(C)C)ncc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4ccc(Oc5ccccc5)cc4)ncc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4cccc(c4)C(C)(C)C)cnc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4ccccc4)ncc3c2)ccn1
Brc1ccc(Nc2ncc3cc(Oc4ccnc(c4)C(=O)NCCN4CCCCC4)ccc3n2)cc1
CNC(=O)c1cc(Oc2ccc3nc(Nc4cccc(OC(F)(F)F)c4)ncc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4ccc(cc4)-c4cccnc4)ncc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4cccc(Cl)c4)ncc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(Nc4ccc(cc4)C(F)(F)F)ncc3c2)ccn1
[O-][N+](=O)c1ccc(\C=C(/C(=O)c2ccccc2)S(=O)(=O)Cc2ccccc2)cc1
[O-][N+](=O)c1ccc(\C=C(/C(=O)c2ccc(Cl)cc2)S(=O)(=O)Cc2ccccc2)cc1
Fc1ccc(\C=C(/C(=O)c2ccc(Cl)cc2)S(=O)(=O)Cc2ccccc2)cc1
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1cc2cnc(Nc3ccccc3)nc2n(C)c1=O |(14.17,-24.55,;12.84,-23.77,;11.5,-24.55,;10.18,-23.78,;9.4,-22.44,;10.94,-22.44,;8.85,-24.56,;7.52,-23.79,;7.51,-22.24,;6.17,-21.48,;4.84,-22.24,;3.51,-21.48,;4.84,-23.79,;6.18,-24.56,;6.18,-26.1,;3.51,-24.56,;2.18,-23.78,;.85,-24.55,;-.47,-23.77,;-1.8,-24.54,;-1.8,-26.08,;-3.13,-26.85,;-4.47,-26.08,;-4.46,-24.54,;-5.79,-23.77,;-7.13,-24.54,;-7.13,-26.09,;-5.79,-26.85,;-.48,-26.84,;.84,-26.08,;2.18,-26.85,;2.18,-28.39,;3.51,-26.09,;4.85,-26.85,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1ccc2ccncc2c1
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1ccc2ccncc2n1
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1cc2cncc(Br)c2cn1
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1cc2cnccc2c(=O)n1C |(47.93,-11.02,;46.6,-10.25,;45.26,-11.02,;43.94,-10.25,;43.15,-8.91,;44.69,-8.91,;42.6,-11.03,;41.27,-10.26,;41.26,-8.71,;39.92,-7.94,;38.59,-8.71,;37.26,-7.94,;38.59,-10.26,;39.93,-11.03,;39.93,-12.57,;37.26,-11.02,;35.93,-10.25,;34.6,-11.02,;33.28,-10.24,;31.94,-11.01,;31.94,-12.55,;33.27,-13.31,;34.59,-12.55,;35.93,-13.32,;35.93,-14.87,;37.26,-12.56,;38.59,-13.33,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1ccc2nc(N)ncc2c1
CCCS(=O)(=O)Nc1cccc(c1)-c1cc2cnc(N)nc2n(C)c1=O
CCCS(=O)(=O)Nc1ccc(F)c(c1)-c1ccc2nc(N)ncc2c1
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1cc2cnc(N)nc2n(C)c1=O |(9.34,-.05,;8.01,.72,;6.67,-.05,;5.35,.71,;4.57,2.06,;6.11,2.06,;4.01,-.06,;2.68,.71,;2.67,2.26,;1.34,3.02,;.01,2.25,;-1.32,3.02,;.01,.71,;1.34,-.07,;1.34,-1.61,;-1.32,-.06,;-2.65,.72,;-3.98,-.05,;-5.31,.72,;-6.64,-.04,;-6.64,-1.58,;-7.97,-2.35,;-5.31,-2.34,;-3.99,-1.59,;-2.65,-2.36,;-2.65,-3.9,;-1.32,-1.59,;.02,-2.36,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1cc2cnc(NCC3CC3)nc2n(C)c1=O |(56.32,-.34,;54.99,.43,;53.65,-.34,;52.32,.43,;51.54,1.77,;53.08,1.77,;51,-.35,;49.66,.42,;49.66,1.97,;48.32,2.73,;46.99,1.97,;45.65,2.73,;46.99,.42,;48.32,-.35,;48.32,-1.89,;45.65,-.35,;44.33,.43,;42.99,-.34,;41.67,.44,;40.34,-.33,;40.34,-1.87,;39.01,-2.64,;37.67,-1.87,;36.34,-2.64,;34.8,-2.65,;35.57,-3.98,;41.66,-2.63,;42.98,-1.87,;44.32,-2.64,;44.32,-4.18,;45.65,-1.88,;46.99,-2.64,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1cc2cnc(NCCO)nc2n(C)c1=O |(10.92,-12.49,;9.59,-11.72,;8.25,-12.5,;6.93,-11.73,;6.15,-10.38,;7.69,-10.38,;5.59,-12.51,;4.27,-11.73,;4.26,-10.18,;2.92,-9.42,;1.59,-10.19,;.26,-9.42,;1.59,-11.73,;2.93,-12.51,;2.93,-14.05,;.25,-12.5,;-1.07,-11.72,;-2.4,-12.49,;-3.73,-11.72,;-5.05,-12.49,;-5.05,-14.03,;-6.39,-14.79,;-7.72,-14.03,;-9.06,-14.79,;-10.39,-14.03,;-3.73,-14.79,;-2.41,-14.03,;-1.07,-14.8,;-1.07,-16.34,;.26,-14.03,;1.59,-14.8,)|
CCCS(=O)(=O)Nc1ccc(c(c1F)C2=Cc3cnc(nc3N(C2=O)C)NCCCO)F
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1cc2cnc(NC3CCOCC3)nc2n(C)c1=O |(59.79,-12.06,;58.46,-11.29,;57.12,-12.06,;55.8,-11.3,;55.02,-9.95,;56.56,-9.95,;54.46,-12.07,;53.14,-11.3,;53.13,-9.75,;51.79,-8.99,;50.46,-9.76,;49.13,-8.99,;50.46,-11.3,;51.8,-12.08,;51.8,-13.62,;49.12,-12.07,;47.8,-11.29,;46.47,-12.06,;45.14,-11.29,;43.82,-12.05,;43.82,-13.59,;42.48,-14.36,;41.15,-13.6,;41.15,-12.06,;39.83,-11.29,;38.49,-12.05,;38.48,-13.6,;39.82,-14.37,;45.14,-14.35,;46.46,-13.6,;47.8,-14.37,;47.8,-15.91,;49.13,-13.6,;50.46,-14.37,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1cc2cnc(Nc3cccnc3)nc2n(C)c1=O |(39.5,-24.7,;38.16,-23.92,;36.83,-24.7,;35.5,-23.93,;34.72,-22.59,;36.26,-22.59,;34.17,-24.71,;32.84,-23.94,;32.83,-22.39,;31.49,-21.63,;30.16,-22.39,;28.83,-21.63,;30.16,-23.94,;31.5,-24.71,;31.5,-26.25,;28.83,-24.71,;27.5,-23.93,;26.17,-24.7,;24.84,-23.92,;23.52,-24.69,;23.52,-26.23,;22.18,-27,;20.85,-26.23,;19.53,-27,;18.19,-26.24,;18.19,-24.7,;19.52,-23.92,;20.86,-24.69,;24.84,-26.99,;26.16,-26.23,;27.5,-27,;27.5,-28.54,;28.83,-26.24,;30.17,-27,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1cc2cnccc2n(CCc2ccccc2)c1=O |(8.36,-21.46,;7.02,-20.69,;5.69,-21.46,;4.37,-20.7,;3.58,-19.35,;5.12,-19.35,;3.03,-21.47,;1.7,-20.7,;1.69,-19.15,;.35,-18.39,;-.98,-19.16,;-2.31,-18.39,;-.98,-20.7,;.36,-21.47,;.36,-23.02,;-2.31,-21.47,;-3.64,-20.69,;-4.97,-21.46,;-6.29,-20.69,;-7.62,-21.45,;-7.62,-22.99,;-6.3,-23.76,;-4.98,-22.99,;-3.64,-23.77,;-3.64,-25.31,;-2.3,-26.08,;-2.3,-27.62,;-3.64,-28.39,;-3.64,-29.93,;-2.3,-30.7,;-.97,-29.92,;-.97,-28.38,;-2.31,-23,;-.97,-23.77,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1cc2cnc(NC)nc2n(C)c1=O |(31.39,-.05,;30.06,.72,;28.72,-.05,;27.4,.71,;26.62,2.06,;28.16,2.06,;26.07,-.06,;24.73,.71,;24.73,2.26,;23.39,3.02,;22.06,2.25,;20.73,3.02,;22.06,.71,;23.4,-.07,;23.39,-1.61,;20.72,-.06,;19.4,.72,;18.07,-.05,;16.75,.72,;15.42,-.04,;15.42,-1.58,;14.08,-2.35,;12.75,-1.59,;16.74,-2.34,;18.06,-1.59,;19.4,-2.36,;19.4,-3.9,;20.73,-1.59,;22.06,-2.36,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1cc2cnccc2cn1
CCCS(=O)(=O)Nc1ccc(C)c(c1)-c1ccc2nc(N)ncc2c1
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1cc2cnc(Nc3cnn(C)c3)nc2n(C)c1=O |(13.75,-37.45,;12.42,-36.67,;11.08,-37.45,;9.76,-36.68,;8.98,-35.34,;10.52,-35.34,;8.42,-37.46,;7.09,-36.69,;7.08,-35.14,;5.74,-34.38,;4.42,-35.14,;3.08,-34.38,;4.42,-36.69,;5.75,-37.46,;5.75,-39,;3.08,-37.46,;1.76,-36.68,;.43,-37.45,;-.9,-36.67,;-2.23,-37.44,;-2.23,-38.98,;-3.57,-39.75,;-4.82,-38.87,;-4.86,-37.33,;-6.33,-36.88,;-7.21,-38.15,;-8.75,-38.18,;-6.28,-39.37,;-.91,-39.74,;.42,-38.98,;1.76,-39.75,;1.76,-41.29,;3.09,-38.99,;4.42,-39.75,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1ccc2cc(N)ncc2c1
CCCS(=O)(=O)Nc1ccc(F)c(-c2cc3ccncc3[nH]2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc(nn3c2)N2CCOCC2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc(nn3c2)C(F)(F)F)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3occc3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc[nH]c3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3ccnn3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc(CC)nn3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc(nn3c2)C2CC2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc(nn3c2)N2CCCC2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc(OCC)nn3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc(OCCOC)nn3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc(nn3c2)-c2ccc(F)cc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc(nn3c2)-c2cccnc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3ccccc3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc(nn3c2)C2CCCC2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc(NC)nn3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc(NC(C)C)nn3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc(OC)nn3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc(nn3c2)-c2ccccc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc(nn3c2)-c2cccc(F)c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc(C)nn3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc(OC(C)C)nn3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3nccn3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc(nn3c2)-c2cnn(C)c2)c1F
CC(C)(C)OC(=O)Nc1cc(Oc2ccc3nc(NC(=O)C4CC4)sc3n2)ccc1F
[#8-]-[#7+](=O)-c1ccc(cc1)-c1ccc(\[#6]=[#6]-2\[#6](=O)-[#7]-[#6](=S)-[#7]-[#6]-2=O)o1
[#8-]-[#7+](=O)-c1ccccc1-c1ccc(\[#6]=[#6]-2\[#6](=O)-[#7]-[#6](=S)-[#7]-[#6]-2=O)o1
OC(=O)c1ccc(cc1)-c1ccc(\C=C2\C(=O)NC(=S)N(C2=O)c2cccc(Cl)c2Cl)o1
OC(=O)c1ccc(cc1)-c1ccc(\C=C2\C(=O)NC(=S)N(C2=O)c2ccc(Br)cc2)o1
OC(=O)c1ccc(cc1Cl)-c1ccc(\C=C2\C(=O)NC(=S)N(C2=O)c2ccc(Br)cc2)o1
Cc1ccc(cc1)N1C(=S)NC(=O)\C(=C\c2ccc(o2)-c2ccc(cc2)C(O)=O)C1=O
Cc1ccc(cc1)N1C(=S)NC(=O)\C(=C\c2ccc(o2)-c2cccc(c2)C(O)=O)C1=O
COC(=O)c1ccccc1-c1ccc(\C=C2\C(=O)NC(=S)N(C2=O)c2ccc(C)cc2)o1
CCOC(=O)c1ccccc1-c1ccc(\C=C2\C(=O)NC(=S)N(C2=O)c2ccc(C)cc2)o1
Cc1ccc(cc1)N1C(=S)NC(=O)\C(=C\c2ccc(CN(CCC#N)S(C)(=O)=O)o2)C1=O
CS(=O)(=O)N(CCC#N)Cc1ccc(\C=C2\C(=O)NC(=S)N(C2=O)c2ccc(Br)cc2)o1
CCOc1ccc(cc1)N1C(=S)NC(=O)\C(=C\c2ccc(CN(CCC#N)S(C)(=O)=O)o2)C1=O
Cc1cccc(c1)N1C(=S)NC(=O)\C(=C\c2ccc(CN(CCC#N)S(C)(=O)=O)o2)C1=O
O=[#6]1-[#7]-[#6](=S)-[#7]-[#6](=O)\[#6]-1=[#6]/c1ccc(o1)-c1ccccc1C#N
Cc1c(Cl)cccc1N1C(=S)NC(=O)\C(=C\c2ccc(o2)-c2ccc(cc2)C(O)=O)C1=O
OC(=O)c1ccccc1-c1ccc(\C=C2\C(=O)NC(=S)N(C2=O)c2ccc(Br)cc2)o1
Cc1ccc(cc1)N1C(=S)NC(=O)\C(=C\c2ccc(o2)-c2ccc(F)cc2)C1=O
COc1cccc(c1)N1C(=S)NC(=O)\C(=C\c2ccc(CN(CCC#N)S(C)(=O)=O)o2)C1=O
[#8-]-[#7+](=O)-c1cccc(c1)-c1ccc(\[#6]=[#6]-2\[#6](=O)-[#7]-[#6](=S)-[#7]-[#6]-2=O)o1
OC(=O)c1cccc(c1)-c1ccc(\C=C2\C(=O)NC(=S)N(C2=O)c2ccc(Br)cc2)o1
Cc1ccc(cc1Cl)N1C(=S)NC(=O)\C(=C\c2ccc(CN(CCC#N)S(C)(=O)=O)o2)C1=O
[#6]-[#8]-c1ccc(\[#6]=[#6]-2\[#6](=O)-[#7]-[#6](=S)-[#7]-[#6]-2=O)cc1-[#8]-[#6](=O)-c1ccccc1
Cc1ccc(cc1)N1C(=S)NC(=O)\C(=C\c2ccc(o2)-c2ccc(C(O)=O)c(Cl)c2)C1=O
CS(=O)(=O)N(CCC#N)Cc1ccc(\C=C2\C(=O)NC(=S)N(C2=O)c2ccc(Cl)c(Cl)c2)o1
O=C(Nc1ccccc1)Nc1cccc(c1)C(=O)Nc1cnc2[nH]ncc2c1
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NC(=O)c4cccc(c4)C(C)(C)C#N)c3F)cc12
CC(C)(C#N)c1cccc(c1)C(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]ncc3c2)c1F
COc1n[nH]c2ncc(NC(=O)c3cccc(NC(=O)c4cccc(c4)C(C)(C)C#N)c3)cc12
COc1n[nH]c2ncc(NC(=O)c3cccc(NC(=O)c4cccc(c4)C(C)(C)C#N)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3cc(NC(=O)c4cccc(c4)C(C)(C)C#N)ccc3Cl)cc12
COc1n[nH]c2ncc(NC(=O)c3cc(ccc3C)C(=O)Nc3cccc(c3)C(F)(F)F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(NC(=O)c4ccccc4)c3F)cc12
CC(C)(C#N)c1cccc(c1)C(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]ccc3c2)c1F
COc1n[nH]c2ncc(NC(=O)c3cc(NC(=O)c4cccc(c4)C(C)(C)C#N)ccc3C)cc12
COc1n[nH]c2ncc(NC(=O)c3cccc(c3)C(=O)Nc3ccccc3)cc12
COc1n[nH]c2ncc(NC(=O)c3cc(NC(=O)c4cccc(c4)C(C)(C)C#N)ccc3F)cc12
COc1n[nH]c2ncc(NC(=O)c3cc(NC(=O)c4ccc(Cl)c(c4)C(F)(F)F)ccc3F)cc12
CC(C)(C#N)c1cccc(c1)C(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]nc(C4CC4)c3c2)c1F
COc1cc(cnc1N)-c1nn(cc1-c1ccnc(NC[C@H](C)O)n1)C(C)C |r|
C[S+]([O-])c1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc(F)cc1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2c(O)c(F)ccc2c1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2c(O)cccc2c1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2c(csc2c1)C(O)C(F)(F)F
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc(Cl)c(Cl)c1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2cc(F)ccc2c1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2c(cc[nH]c2=O)c1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2ccc(=O)[nH]c2c1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2ccc(O)cc2c1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2c(csc2c1)[S+](C)[O-]
CCC[S+]([O-])c1csc2cc(ccc12)-c1nc([nH]c1-c1ccncc1)-c1ccc(OCCN(C)C)cc1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2c(csc2c1)[C@@H](O)C(F)(F)F |r|
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2c(csc2c1)C(O)C(F)(F)C(F)(F)F
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2c(C=O)csc2c1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc(F)c(Cl)c1
CCCSc1csc2cc(ccc12)-c1nc([nH]c1-c1ccncc1)-c1ccc(OCCN(C)C)cc1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2[nH]c(=O)ccc2c1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2c(CO)coc2c1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2cc(O)ccc2c1
CCC(O)c1csc2cc(ccc12)-c1nc([nH]c1-c1ccncc1)-c1ccc(OCCN(C)C)cc1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2c(N)nccc2c1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2c(O)c(Cl)ccc2c1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2sc(cc2c1)C(O)C(F)(F)F
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2c(CO)csc2c1
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2c(coc2c1)C(N)=O
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc(cc1)C(O)C(F)(F)F
CN(C)CCOc1ccc(cc1)-c1nc(c([nH]1)-c1ccncc1)-c1ccc2cc(ccc2c1)C(O)=O
CSc1csc2cc(ccc12)-c1nc([nH]c1-c1ccncc1)-c1ccc(OCCN(C)C)cc1
CCOC(=O)c1sc(NC(=O)c2ccc(OCC)cc2)c(C#N)c1C
CCOC(=O)c1sc(NC(=O)c2cc(OC)cc(OC)c2)c(C#N)c1C
CCOC(=O)c1sc(NC(=O)c2ccccc2C)c(C#N)c1C
CCOC(=O)c1sc(NC(=O)c2ccc(F)cc2)c(C(=O)Nc2ccccc2)c1C
Brc1ccc(cc1)-c1ccc(\[#6]=[#6]-2\[#6](=O)-[#7]-[#6](=S)-[#7]-[#6]-2=O)o1
CCOC(=O)c1sc(NC(=O)c2ccc(Cl)c(c2)[N+]([O-])=O)c(C#N)c1C
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2ccccc2Br)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccccc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2ccccc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)C2CCC2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)C(C)C)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2cccnc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2cccc(OC)c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2ccc(cc2)C#N)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2ccc(OC)cc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2ccc(Cl)c(Cl)c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2ccccc2Cl)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2cccc(Br)c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(Cl)cc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)C2CCCNC2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)C2CCNCC2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2ccc(cc2)S(C)(=O)=O)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2ccc(C)cc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3cc(nn3c2)-c2ccc(Cl)cc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2ccncc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2ccc(F)c(F)c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2ccc(OC(F)(F)F)cc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2ccc(F)cc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(CC)nc3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2cccc(Cl)c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2ccccc2F)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)C(C)(C)C)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2ccc(Br)cc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2ccc(Cl)cc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2ccc(cc2)C(F)(F)F)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(C)nc3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(cc3c2)-c2ccc(F)cc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2cccc(F)c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)Nc2cnc3[nH]c(nc3c2)-c2cccc(c2)C(F)(F)F)c1F
CC(C)n1c(C)nc2c(F)cc(cc12)-c1nc(Nc2ccc3CN(CCN(C)C)CCc3n2)ncc1F
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3nccnc3c2)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(Cc4ccccc4)c(=O)c3c2)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(N(CC)c2ccc3ncn(C)c(=O)c3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncnc(NC)c3c2)c1Cl
CCCS(=O)(=O)Nc1ccc(Cl)c(Nc2ccc3ncn(C)c(=O)c3c2)c1F
CCCS(=O)(=O)Nc1ccc(Cl)c(N(C)c2ccc3ncn(C)c(=O)c3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncnc(OC)c3c2)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(-c4cnn(C)c4)c(=O)c3c2)c1Cl
CCCS(=O)(=O)Nc1ccc(Cl)c(Nc2ccc3ncn(C)c(=O)c3c2)c1C#N
CCCS(=O)(=O)Nc1ccc(F)c(N(C)c2ccc3ncn(C)c(=O)c3c2)c1Cl
Cc1ccc(cc1Nc2ccc3c(c2)C(=O)N(C=N3)C)NC(=O)c4cccc(c4)C(C)(C)C#N
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncncc3c2)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncnc(N(C)C)c3c2)c1Cl
CCCS(=O)(=O)Nc1cccc(c1C#N)Nc2ccc3c(c2)C(=O)N(C=N3)C
CCCS(=O)(=O)Nc1ccc(F)c(N(CC)c2ccc3ncn(C)c(=O)c3c2)c1Cl
CCCS(=O)(=O)Nc1cccc(Oc2ccc3ncn(C)c(=O)c3c2)c1C#N
CCCS(=O)(=O)Nc1ccc(C)c(Nc2ccc3ncn(C)c(=O)c3c2)c1
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncncc3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2)c1F
CCCS(=O)(=O)Nc1ccc(c(c1F)N(C)c2ccc3c(c2)C(=O)N(C=N3)C)F
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncccc3c2)c1F
CCCS(=O)(=O)Nc1ccc(Cl)c(Oc2ccc3ncn(C)c(=O)c3c2)c1C#N
CNC(=O)c1cc(Oc2ccc3nc(NC(=O)Nc4ccc(Cl)c(Cl)c4)sc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(NC(=O)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F)sc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)sc3c2)ccn1
CNC(=O)c1cc(Oc2ccc3nc(NC(=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)sc3c2)ccn1
COc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c1
COc1ccc(cc1Cl)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
Oc1c(Br)cc(\C=C2/C(=O)Nc3ccc(I)cc23)cc1Br
Cc1ccc(cc1NC(=O)c2ccc3c(c2)ccc(n3)C)NC(=O)c4ccc5c(c4)OCCO5
CC(C)(C)N1CCN(Cc2ccc3cc(ccc3n2)C(=O)Nc2cc(NC(=O)c3ccc4OCCOc4c3)ccc2Cl)CC1
Cc1ccc(NC(=O)c2ccc3OCCOc3c2)cc1NC(=O)c1ccc2nc(OCCN3CCCC3)ccc2c1
CN1CCC(CC1)Oc1ccc(NC(=O)c2ccc(C)c(NC(=O)C3(CC3)c3ncnc4[nH]ccc34)c2)cc1C(F)(F)F
CN1CCC(COc2ccc(NC(=O)c3ccc(C)c(NC(=O)C(C)(C)c4ncnc5[nH]ccc45)c3)cc2C(F)(F)F)CC1
Cc1ccc(cc1NC(=O)C1(CC1)c1ncnc2[nH]ccc12)C(=O)Nc1ccccc1
Cc1ccc(cc1NC(=O)C1(CC1)c1ncnc2[nH]cnc12)C(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
Cc1ccc(cc1NC(=O)C1(CC1)c1ncnc2[nH]ccc12)C(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
Cc1ccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)cc1NC(=O)C1(CC1)c1ncnc2[nH]ccc12
Cc1ccc(cc1NC(=O)C1(CC1)c1ncnc2[nH]ccc12)C(=O)Nc1cccc(F)c1
Cc1ccc(cc1NC(=O)C1(CC1)c1ncnc2[nH]ccc12)C(=O)Nc1cccc(Cl)c1
Cc1ccc(cc1NC(=O)C1(CC1)c1ncnc2[nH]ccc12)C(=O)Nc1ccc(N2CCOCC2)c(c1)C(F)(F)F
Cc1ccc(cc1NC(=O)C(C)(C)c1ncnc2[nH]ccc12)C(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
Cc1ccc(cc1NC(=O)C1(CC1)c1ncnc2[nH]ccc12)C(=O)Nc1ccc(F)cc1
CN1CCC(COc2ccc(NC(=O)c3ccc(C)c(NC(=O)C4(CC4)c4ncnc5[nH]ccc45)c3)cc2C(F)(F)F)CC1
CN1CCN(CC1)c1ccc(NC(=O)c2ccc(C)c(NC(=O)C3(CC3)c3ncnc4[nH]ccc34)c2)cc1C(F)(F)F
Cc1ccc(NC(=O)c2ccc(Cl)c(c2)C(F)(F)F)cc1NC(=O)C1(CC1)c1ncnc2[nH]ccc12
Cc1ccc(cc1NC(=O)C1(CC1)c1ncnc2[nH]ccc12)C(=O)Nc1ccc(Cl)cc1
Cc1ccc(cc1NC(=O)C1(CC1)c1ncnc2[nH]ccc12)C(=O)Nc1ccc(OCCCN2CCOCC2)c(c1)C(F)(F)F
CN1CC[C@H]1CCc1ccc(C)cc1NC(=O)Nc1cccc(Oc2ccc3nc[nH]c(=O)c3c2)c1 |r|
Cc1ccc(cc1)-c1cc([nH]n1)-c1cccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c1
Cc1nccn1-c1cc(cc(c1)C(F)(F)F)C(=O)Nc1cccc(c1)-c1cc(n[nH]1)-c1ccc(C)cc1
CC(C)c1cc([nH]n1)-c1cccc(NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c1
CC(C)c1cc([nH]n1)-c1cccc(NC(=O)Nc2cccc(c2)C(F)(F)F)c1
Cc1cn(cn1)-c1cc(cc(c1)C(F)(F)F)C(=O)Nc1cccc(c1)-c1cc(n[nH]1)-c1ccc(C)cc1
Cc1ccc(cc1)-c1cc([nH]n1)-c1cccc(NC(=O)c2ccc(c(c2)N2CCOCC2)C(F)(F)F)c1
Cc1ccc(cc1)-c1cc([nH]n1)-c1cccc(NC(=O)c2cc(cc(c2)C(F)(F)F)N2CCOCC2)c1
CC(C)c1cc([nH]n1)-c1cccc(NC(=O)c2cc(cc(c2)C(F)(F)F)N2CCOCC2)c1
CC(C)c1cc([nH]n1)-c1cccc(NC(=O)c2cc(cc(c2)C(F)(F)F)N2CCN(C)CC2)c1
CC(C)c1cc([nH]n1)-c1cccc(NC(=O)c2cc(cc(c2)C(F)(F)F)-n2cnc(C)c2)c1
CC(C)c1cc([nH]n1)-c1cccc(NC(=O)Nc2ccc(Cl)c(Cl)c2)c1
Cc1ccc(cc1)-c1cc([nH]n1)-c1cccc(NC(=O)c2ccc3ccccc3n2)c1
CC(C)c1cc([nH]n1)-c1cccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(OCCO)nc(c1)N1CCOCC1
COc1n[nH]c2ncc(cc12)-c1cn(nn1)-c1c(Cl)ccc(NS(=O)(=O)c2cccc(Cl)c2)c1Cl
COc1n[nH]c2ncc(cc12)-c1cn(nn1)-c1c(F)ccc(NS(=O)(=O)c2ccc3ccccc3c2)c1F
COc1n[nH]c2ncc(cc12)-c1cn(nn1)-c1c(F)ccc(NS(=O)(=O)c2cccc(c2)-c2ccccc2)c1F
COc1n[nH]c2ncc(cc12)-c1cn(nn1)-c1c(F)ccc(NS(=O)(=O)c2cccc(c2)C(C)C)c1F
COc1n[nH]c2ncc(cc12)-c1cn(nn1)-c1c(F)ccc(NS(=O)(=O)c2cccc(OC)c2)c1F
COc1n[nH]c2ncc(cc12)-c1cn(nn1)-c1c(F)ccc(NS(=O)(=O)c2ccccc2)c1F
COc1n[nH]c2ncc(cc12)-c1cn(nn1)-c1c(F)ccc(NC(=O)Nc2cccc(Cl)c2)c1F
COc1n[nH]c2ncc(cc12)-c1cn(nn1)-c1c(F)ccc(NC(=O)Cc2cccc(Cl)c2)c1F
COc1n[nH]c2ncc(cc12)-c1cn(nn1)-c1cc(NS(=O)(=O)c2cccc(Cl)c2)ccc1F
COc1n[nH]c2ncc(cc12)-c1cn(nn1)-c1cccc(NS(=O)(=O)c2cccc(Cl)c2)c1
Nc1ccc(cn1)-c1cn(nn1)-c1c(F)ccc(NS(=O)(=O)c2cccc(Cl)c2)c1F
COc1n[nH]c2ncc(cc12)-c1nc(no1)-c1c(F)ccc(NS(=O)(=O)c2cccc(Cl)c2)c1F
COc1n[nH]c2ncc(cc12)-c1ncc([nH]1)-c1c(F)ccc(NS(=O)(=O)c2cccc(Cl)c2)c1F
COc1n[nH]c2ncc(cc12)-c1cn(nn1)-c1c(F)ccc(NC(=O)c2cccc(Cl)c2)c1F
COc1n[nH]c2ncc(cc12)-c1cn(nn1)-c1c(F)ccc(NS(=O)(=O)c2cccc(Cl)c2)c1F
COc1n[nH]c2ncc(cc12)-c1cn(nn1)-c1c(F)ccc(NS(=O)(=O)c2cccc3ccccc23)c1F
COc1n[nH]c2ncc(cc12)-c1cn(nn1)-c1c(F)ccc(NS(=O)(=O)c2cccc(Br)c2)c1F
COc1n[nH]c2ncc(cc12)-c1cn(nn1)-c1cccc(NS(=O)(=O)c2cccc(Cl)c2)c1F
Nc1ncc(cn1)-c1cn(nn1)-c1c(F)ccc(NS(=O)(=O)c2cccc(Cl)c2)c1F
COc1n[nH]c2ncc(cc12)-c1cn(nn1)-c1c(F)ccc(NS(=O)(=O)c2cccc(c2)C#N)c1F
COc1n[nH]c2ncc(cc12)-c1nnc(o1)-c1c(F)ccc(NS(=O)(=O)c2cccc(Cl)c2)c1F
COc1n[nH]c2ncc(cc12)-c1cn(nn1)-c1c(F)ccc(NS(=O)(=O)c2cccc(C)c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-n1cc(-c2cncnc2)c2nc(ccc12)N(C)C1CCN(CC1)C(=O)CCOCCOCCOCCNc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12 |(-10.34,9.68,;-9.01,10.47,;-7.68,9.7,;-6.34,10.46,;-7.12,11.8,;-5.58,11.81,;-5.02,9.7,;-5.02,8.16,;-6.35,7.39,;-6.35,5.84,;-5.01,5.08,;-5.01,3.54,;-3.67,5.85,;-3.68,7.38,;-2.36,8.16,;-2.34,5.09,;-.93,5.72,;.12,4.57,;1.65,4.75,;2.55,3.5,;4.08,3.66,;4.7,5.08,;3.79,6.33,;2.26,6.16,;-.66,3.25,;-.17,1.79,;-1.2,.66,;-2.71,.96,;-3.18,2.42,;-2.16,3.56,;-.7,-.82,;-1.73,-1.97,;.81,-1.13,;1.29,-2.58,;2.79,-2.9,;3.82,-1.75,;3.34,-.29,;1.83,.05,;5.33,-2.07,;6.35,-.92,;5.81,-3.53,;7.32,-3.84,;7.8,-5.31,;9.3,-5.62,;9.78,-7.09,;11.29,-7.4,;11.77,-8.86,;13.28,-9.18,;13.76,-10.64,;15.27,-10.96,;15.75,-12.42,;17.25,-12.74,;17.73,-14.2,;16.71,-15.34,;17.18,-16.8,;18.69,-17.12,;19.72,-15.96,;21.25,-15.94,;22.17,-17.18,;21.71,-14.48,;23.17,-14,;24.32,-15.02,;25.78,-14.54,;26.09,-13.03,;27.55,-12.55,;24.94,-12.01,;23.47,-12.49,;22.32,-11.47,;20.47,-13.59,;20.45,-12.05,;19.24,-14.5,)|
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(CNC(=O)CCCCNc3ccc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4c3)cc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(CNC(=O)CCCCNc3ccc4C(=O)N(C5CCC(=O)N(C)C5=O)C(=O)c4c3)cc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-n1cc(-c2cncnc2)c2nc(ccc12)N(C)C1CCN(CC1)C(=O)CCOCCOCCOCCNc1cccc2C(=O)N(C3CCC(=O)N(C)C3=O)C(=O)c12 |(-10.34,9.68,;-9.01,10.47,;-7.68,9.7,;-6.34,10.46,;-7.12,11.8,;-5.58,11.81,;-5.02,9.7,;-5.02,8.16,;-6.35,7.39,;-6.35,5.84,;-5.01,5.08,;-5.01,3.54,;-3.67,5.85,;-3.68,7.38,;-2.36,8.16,;-2.34,5.09,;-.93,5.72,;.12,4.57,;1.65,4.75,;2.55,3.5,;4.08,3.66,;4.7,5.08,;3.79,6.33,;2.26,6.16,;-.66,3.25,;-.17,1.79,;-1.2,.66,;-2.71,.96,;-3.18,2.42,;-2.16,3.56,;-.7,-.82,;-1.73,-1.97,;.81,-1.13,;1.29,-2.58,;2.79,-2.9,;3.82,-1.75,;3.34,-.29,;1.83,.05,;5.33,-2.07,;6.35,-.92,;5.81,-3.53,;7.32,-3.84,;7.8,-5.31,;9.3,-5.62,;9.78,-7.09,;11.29,-7.4,;11.77,-8.86,;13.28,-9.18,;13.76,-10.64,;15.27,-10.96,;15.75,-12.42,;17.25,-12.74,;17.73,-14.2,;16.71,-15.34,;17.18,-16.8,;18.69,-17.12,;19.72,-15.96,;21.25,-15.94,;22.17,-17.18,;21.71,-14.48,;23.17,-13.99,;24.32,-15.02,;25.78,-14.54,;26.09,-13.03,;27.55,-12.55,;24.94,-12,;25.25,-10.5,;23.47,-12.49,;22.32,-11.47,;20.47,-13.59,;20.45,-12.05,;19.24,-14.5,)|
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(\N=N/c4ccc(OC)cc4)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(\N=N\c4ccccc4)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(\N=N\c4ccc(OC)cc4)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(\N=N\c4ccccc4F)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(\N=N\c4ccc(C)cc4)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(\N=N\c4ccc(F)cc4)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(\N=N\c4ccccc4OC)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(\N=N/c4ccccc4)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3cccc(c3)\N=N/c3ccc(OC)cc3)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(\N=N/c4ccc(F)cc4)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(\N=N/c4ccccc4C)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(\N=N\c4ccccc4C)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(\N=N/c4ccccc4F)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(\N=N/c4ccccc4OC)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3c(F)ccc(\N=N/c4ccc(C)cc4)c3F)cc12
COc1n[nH]c2ncc(NC(=O)c3cccc(c3)\N=N\c3ccc(OC)cc3)cc12
CCn1c2c(c(n1)C#Cc3c(ccc4c3ccnc4Nc5ccc(cc5)Cl)C)c(ncn2)N
CC(C)n1nc(C#Cc2cccc3c(Nc4cccc(c4)C(F)(F)F)nccc23)c2c(N)ncnc12
CC(C)n1nc(C#Cc2cccc3c(Nc4cccc(c4)C(F)(F)F)ncnc23)c2c(N)ncnc12
CC(C)n1nc(C#Cc2cccc3c(Nc4cc(cc(c4)C(F)(F)F)-n4cnc(C)c4)nccc23)c2c(N)ncnc12
CC(C)n1nc(C#Cc2cccc3c(Oc4cccc(c4)C(F)(F)F)nccc23)c2c(N)ncnc12
CC(C)n1nc(C#Cc2c(C)ccc3c(Nc4cccc(c4)C(F)(F)F)nccc23)c2c(N)ncnc12
CCCn1nc(C#Cc2cccc3c(Nc4cccc(c4)C(F)(F)F)nccc23)c2c(N)ncnc12
CC(C)n1nc(C#Cc2cccc3c(Nc4ccc(Cl)cc4)nccc23)c2c(N)ncnc12
CC(C)n1nc(C#Cc2cccc3c(Nc4ccc(Cl)c(c4)C(F)(F)F)nccc23)c2c(N)ncnc12
CC(C)n1nc(C#Cc2cccc3c(Nc4cccc(c4)C(F)(F)F)cccc23)c2c(N)ncnc12
CC(C)n1nc(C#Cc2cccc3c(Nc4ccc(C)c(c4)C(F)(F)F)nccc23)c2c(N)ncnc12
CCn1nc(C#Cc2cccc3c(Nc4cccc(c4)C(F)(F)F)nccc23)c2c(N)ncnc12
CN(C)c1ccc(cc1)C(=O)Nc1cccc(NC(=O)COc2ccc3c(c2)occc3=O)c1
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)CN)C(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CO)C(=O)N[C@@H]([C@@H](C)O)C(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)C(C)C)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)NC(CCC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)C(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCSC)C(=O)NCC(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](C)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)CN)C(C)C)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CO)C(=O)N[C@@H]([C@@H](C)O)C(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)CN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CCSC)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)CN)C(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CO)C(=O)N[C@@H]([C@@H](C)O)C(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)CN)C(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CO)C(=O)N[C@@H]([C@@H](C)O)C(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)CN)C(C)C)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CO)C(=O)N[C@@H]([C@@H](C)O)C(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)CN)C(C)C)[C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CO)C(=O)N[C@@H]([C@@H](C)O)C(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)CN)C(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)C(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)C(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(N)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](C)NC(=O)[C@@H](N)C(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)C(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(O)=O |r|
CSCC[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)C(C)C)[C@@H](C)O)C(C)C)C(=O)NCC(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)C(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)NCC(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](N)CC(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(O)=O |r|
CSCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc2cnc[nH]2)NC(=O)[C@H](CCCNC(N)=N)NC(=O)C(CCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC1=O)C(C)C |r|
CSCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](Cc2cnc[nH]2)NC(=O)[C@H](CCCNC(N)=N)NC(=O)C(CCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC1=O)C(C)C |r|
CSCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](Cc2cnc[nH]2)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC1=O)C(C)C |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)CN)C(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CO)C(=O)N[C@@H]([C@@H](C)O)C(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)CN)C(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CO)C(=O)N[C@@H]([C@@H](C)O)C(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)CN)C(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)NC(CCC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CO)C(=O)N[C@@H]([C@@H](C)O)C(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)C(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(O)=O |r|
CC[C@H](C)[C@@H]1NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc2cnc[nH]2)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC1=O)C(=O)N[C@@H](CCSC)C(O)=O)NC(=O)[C@@H](N)C(C)C)[C@@H](C)O)C(C)C |r|
CSCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc2cnc[nH]2)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)CNC1=O)C(C)C |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)C(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)C(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)CC(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)CN)C(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CO)C(=O)N[C@@H]([C@@H](C)O)C(O)=O |r|
CC[C@H](C)[C@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)C(C)C)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCSC)C(=O)NCC(O)=O |r|
CNC(=O)c1cc(Oc2ccc(NC(=O)c3ccc(Cl)cc3)cc2)ccc1N
CNC(=O)c1cc(Oc2ccc(NC(=O)c3ccccc3)cc2)ccc1N
CNC(=O)c1cc(Oc2ccc(NC(=O)c3ccc(Cl)c(c3)C(F)(F)F)cc2)ccc1N
CNC(=O)c1cc(Oc2ccc(NC(=O)c3ccc(OC)cc3)cc2)ccc1N
CNC(=O)c1cc(Oc2ccc(NC(=O)c3ccc(N)cc3)cc2)ccc1N
CNC(=O)c1cc(Oc2ccc(NC(=O)c3ccc4ccccc4c3)cc2)ccc1N
NC(=O)c1cc(Oc2ccc(NC(=O)c3ccc(Cl)c(c3)C(F)(F)F)cc2)ccc1N
CCNC(=O)c1cc(Oc2ccc(NC(=O)c3ccc(Cl)c(c3)C(F)(F)F)cc2)ccc1N
CN(C)C(=O)c1cc(Oc2ccc(NC(=O)c3ccc(Cl)c(c3)C(F)(F)F)cc2)ccc1N
CNC(=O)c1cc(Oc2ccc(NC(=O)c3cccc(N)c3)cc2)ccc1N
CNC(=O)c1cc(Oc2ccc(NC(=O)c3ccc(F)cc3)cc2)ccc1N
CNC(=O)c1cc(Oc2ccc(NC(=O)c3cccc(O)c3)cc2)ccc1N
CNC(=O)c1cc(Oc2ccc(NC(=O)c3cccnc3)cc2)ccc1N
CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)c(F)c2)ccn1
CC(=O)c1ccc(Nc2ccnc(SCC(=O)c3ccc(cc3)-c3ccccc3)n2)cc1
OC(=O)c1ccc(Nc2ccnc(SCC(=O)c3ccc(Cl)cc3)n2)cc1
CCOC(=O)c1ccc(Nc2ccnc(SCC(=O)c3ccc(OC)cc3)n2)cc1
COc1ccc(cc1)C(=O)CSc1nccc(Nc2ccc(cc2)N2CCOCC2)n1
CC(=O)c1ccc(Nc2ccnc(SCC(=O)c3ccc(Cl)cc3)n2)cc1
OC(=O)c1ccc(Nc2ccnc(SCC(=O)c3ccc(cc3)C#N)n2)cc1
CCOC(=O)c1ccc(Nc2ccnc(SCC(=O)c3ccc(cc3)[N+]([O-])=O)n2)cc1
CCOC(=O)c1ccc(Nc2ccnc(SCC(=O)c3ccc(cc3)C#N)n2)cc1
Fc1ccc(cc1)C(=O)CSc1nccc(Nc2ccc(cc2)N2CCOCC2)n1
CNC(=O)c1cc(Oc2cccc3nc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)ccc23)ccn1
COc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)c2ccccc2)c1
COc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)Nc2ccccc2)c1
Oc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c1
Oc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
Oc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c1
Oc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)c2ccc(N3CCOCC3)c(c2)C(F)(F)F)c1
Oc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)c2ccc(Cl)c(Cl)c2)c1
COc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)c2ccc(N3CCOCC3)c(c2)C(F)(F)F)c1
COc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
COc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)c2ccc(Cl)c(Cl)c2)c1
Oc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c1
Oc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)Nc2cccc(c2)C(F)(F)F)c1
Oc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)Nc2ccccc2)c1
COc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)Nc2cccc(c2)C(F)(F)F)c1
Oc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)c2ccccc2)c1
Oc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)Nc2ccc(Cl)c(Cl)c2)c1
COc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c1
COc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)Nc2ccc(Cl)c(Cl)c2)c1
COc1cc(Cl)cc(c1)-c1nn(cc1-c1ccncc1)-c1cccc(NC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c1
FC(F)(F)CNC(=O)c1cc(cs1)-c1cnn2cc(cnc12)-c1ccc(OCCN2CCCCC2)cc1
Cc1sc(cc1-c1cnn2cc(Cl)cnc12)C(=O)N[C@@H]1[C@H](N)CCCC1(F)F |r|
Cn1cc(cn1)-c1cnc2c(cnn2c1)-c1csc(c1)C(=O)NCC(F)(F)F
Cn1cc(cn1)-c1cnc2c(cnn2c1)-c1csc(c1)C(=O)N[C@@H]1CCCC[C@@H]1N |r|
C[C@@H]1C[C@H]1C(=O)N1CCN(C[C@H]1C)c1cnc(C#N)c(n1)-c1cnn(C)c1 |r|
COC(=O)c1ccc2\C(=C(\Nc3ccc(cc3)-n3c(C)ccc3CN3CCN(C)CC3)c3ccccc3)C(=O)Nc2c1
O=S(=O)(NCCCNc1nccc(n1)-n1ccc2cccnc12)c1ccccc1
Fc1ccc(cc1)S(=O)(=O)NCCCNc1nccc(n1)-n1ccc2cccnc12
Brc1ccc(cc1)S(=O)(=O)NCCCNc1nccc(n1)-n1ccc2cccnc12
COc1ccc(cc1)S(=O)(=O)NCCCNc1nccc(n1)-n1ccc2cccnc12
FC(F)(F)c1cccc(c1)S(=O)(=O)NCCCNc1nccc(n1)-n1ccc2cccnc12
Cc1ccc(cc1)S(=O)(=O)NCCCNc1nccc(n1)-n1ccc2cccnc12
Brc1cccc(c1)S(=O)(=O)NCCCNc1nccc(n1)-n1ccc2cccnc12
Fc1ccc(NC(=O)Nc2ccc(cc2)C(F)(F)F)c(F)c1C(=O)c1c[nH]c2ncccc12
Cc1ccc(NC(=O)Nc2ccc(F)c(C(=O)c3c[nH]c4ncccc34)c2F)cc1
Fc1ccc(NC(=O)Nc2ccc(Br)cc2)c(F)c1C(=O)c1c[nH]c2ncc(Br)cc12
Fc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNC(=O)c2ccccc2)n1
Fc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNC(=O)c2c(F)cccc2F)n1
Fc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNC(=O)c2ccc(Cl)cc2)n1
Fc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc(cc2)C(F)(F)F)n1
Fc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccc(cc2)C(F)(F)F)n1
Cc1ccc(cc1)S(=O)(=O)NCCCNc1nccc(n1)-c1c(nc2sccn12)-c1cccc(F)c1
COc1ccc(cc1)S(=O)(=O)NCCCNc1nccc(n1)-c1c(nc2sccn12)-c1cccc(F)c1
Fc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccc(Cl)cc2)n1
Fc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccc(Br)cc2)n1
c1cc2c(c(c1)C(=O)Nc3c(ccc(c3F)NS(=O)(=O)N4CCCC4)Cl)ncnc2N
Cc1nn(C)cc1-c1cc(C(=O)Nc2c(Cl)ccc(NS(=O)(=O)c3ccccc3Cl)c2F)c2ncnc(N)c2c1
Cc1cc(C(=O)Nc2c(Cl)ccc(NS(=O)(=O)c3cc(F)ccc3F)c2F)c2ncnc(NCCN)c2c1
Cc1cc(C(=O)Nc2c(Cl)ccc(NS(=O)(=O)c3cc(F)ccc3F)c2F)c2ncnc(N[C@@H]3CCCNC3)c2c1 |r|
Cc1cc(C(=O)Nc2c(Cl)ccc(NS(=O)(=O)c3cc(F)ccc3F)c2F)c2ncnc(N[C@H]3CC[C@H](N)CC3)c2c1
c1cc(c(cc1F)S(=O)(=O)Nc2ccc(c(c2F)NC(=O)c3csc4c3ncnc4NC5CCC(CC5)N)Cl)F
N[C@H]1CC[C@@H](CC1)Nc1ncnc2c(csc12)C(=O)Nc1c(Cl)ccc(NS(=O)(=O)Cc2ccccc2)c1F
N[C@H]1CC[C@@H](CC1)Nc1ncnc2c(csc12)C(=O)Nc1c(Cl)ccc(NS(=O)(=O)c2ccccc2Cl)c1F |r,wU:1.0,wD:4.7,(2.27,-26,;3.78,-26.32,;4.8,-25.18,;6.3,-25.5,;6.78,-26.96,;5.75,-28.11,;4.24,-27.79,;8.29,-27.28,;9.32,-26.13,;8.84,-24.68,;9.87,-23.53,;11.37,-23.86,;11.85,-25.31,;13.24,-25.93,;13.09,-27.47,;11.58,-27.79,;10.81,-26.45,;14.58,-25.16,;14.58,-23.62,;15.91,-25.93,;17.25,-25.17,;17.25,-23.62,;15.91,-22.85,;18.58,-22.85,;19.91,-23.61,;19.92,-25.16,;21.25,-25.93,;22.58,-25.15,;21.8,-23.82,;23.35,-23.81,;23.92,-25.93,;23.91,-27.47,;25.25,-28.25,;26.59,-27.47,;26.59,-25.92,;25.25,-25.15,;25.24,-23.61,;18.58,-25.94,;18.58,-27.48,)|
COc1cc2c(Oc3ccc(NC(=O)NN4C(SCC4=O)c4c(F)cccc4F)cc3)ccnc2cc1OC1CCN(CC1)C(=O)NC(C)C
COc1cccc2nc(Nc3cccc(NC(=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)c3)ccc12
COc1cccc2nc(Nc3cccc(NC(=O)c4ccc(N5CCN(C)CC5)c(c4)C(F)(F)F)c3)ccc12
COc1cccc2nc(Nc3cccc(NC(=O)c4ccc(N5CCOCC5)c(c4)C(F)(F)F)c3)ccc12
CCN1CCN(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1cccc(Nc2ccc3c(OC)cccc3n2)c1
COc1cccc2nc(Nc3cccc(NC(=O)c4cc(cc(c4)C(F)(F)F)N4CCOCC4)c3)ccc12
COc1cccc2nc(Nc3cccc(NC(=O)c4cc(cc(c4)C(F)(F)F)-n4cnc(C)c4)c3)ccc12
Cc1cc(c(cc1Nc2ccc3c(c2F)C(=O)N(C=N3)C)NC(=O)NCCC(C)(C)C)F
CNc1ncc2cc(-c3cc(NC(=O)NCCC(C)(C)C)c(F)cc3C)c(=O)n(C)c2n1
Cc1cc(F)c(NC(=O)NCCC(C)(C)C)cc1-c1ccc2cc(N)ncc2c1
Cc1cc(F)c(NC(=O)NCCC(C)(C)C)cc1-c1ccc2c(cnn(C)c2=O)c1
Cc1cc(F)c(cc1-c1ccc2c(cnn(C)c2=O)c1)C(=O)NCCCC(C)(C)C
Cc1cc(F)c(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1-c1ccc2c(cnn(C)c2=O)c1
Cc1cc(F)c(NC(=O)c2cccc(c2)C(C)(C)C#N)cc1-c1cnc2c(cnn(C)c2=O)c1
Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCCNS(=O)(=O)c2cccc(F)c2)n1
Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCCNS(=O)(=O)c2ccc(cc2)C(F)(F)F)n1
COc1ccc(cc1)S(=O)(=O)NCCCCNc1nccc(n1)-c1c(nc2sccn12)-c1cccc(N)c1
Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCCNS(=O)(=O)c2ccc(Cl)cc2)n1
Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2cccc(F)c2)n1
Cc1ccc(cc1)S(=O)(=O)NCCNc1nccc(n1)-c1c(nc2sccn12)-c1cccc(N)c1
Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc(cc2)C(F)(F)F)n1
COc1ccc(cc1)S(=O)(=O)NCCNc1nccc(n1)-c1c(nc2sccn12)-c1cccc(N)c1
Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc(Cl)cc2)n1
Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCCNS(=O)(=O)c2ccc(Br)cc2)n1
Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2cccc3ccccc23)n1
Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc(F)cc2)n1
Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc(Br)cc2)n1
Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCCNS(=O)(=O)c2ccc(F)cc2)n1
Nc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCCNS(=O)(=O)c2cccc3ccccc23)n1
Oc1cc(ccc1F)-c1nc([nH]c1-c1ccnc(NCCCNS(=O)(=O)c2ccccc2)n1)-c1ccccc1
Oc1cc(ccc1F)-c1nc([nH]c1-c1ccnc(NCCCNS(=O)(=O)c2ccc(Br)cc2)n1)-c1ccccc1
Oc1cc(ccc1F)-c1nc([nH]c1-c1ccnc(NCCCNS(=O)(=O)c2cccc(F)c2)n1)-c1ccccc1
Cc1ccc(cc1)S(=O)(=O)NCCCNc1nccc(n1)-c1[nH]c(nc1-c1ccc(F)c(O)c1)-c1ccccc1
COc1ccc(cc1)S(=O)(=O)NCCCNc1nccc(n1)-c1[nH]c(nc1-c1ccc(F)c(O)c1)-c1ccccc1
Oc1cc(ccc1Cl)-c1nc([nH]c1-c1ccnc(NCCCNS(=O)(=O)c2ccccc2)n1)-c1ccccc1
Oc1cc(ccc1Cl)-c1nc([nH]c1-c1ccnc(NCCCNS(=O)(=O)c2ccc(Br)cc2)n1)-c1ccccc1
Oc1cc(ccc1Cl)-c1nc([nH]c1-c1ccnc(NCCCNS(=O)(=O)c2cccc(F)c2)n1)-c1ccccc1
Cc1ccc(cc1)S(=O)(=O)NCCCNc1nccc(n1)-c1[nH]c(nc1-c1ccc(Cl)c(O)c1)-c1ccccc1
COc1ccc(cc1)S(=O)(=O)NCCCNc1nccc(n1)-c1[nH]c(nc1-c1ccc(Cl)c(O)c1)-c1ccccc1
Oc1ccc(cc1)S(=O)(=O)NCCNc1cc(ccn1)-c1[nH]c(nc1-c1cccc(O)c1)-c1ccccc1
CC(C)(C)c1cc(NC(=O)Nc2ccc(Nc3ncnc4NCCCOc34)cc2)no1
Nc1n[nH]c2cccc(C#Cc3cccc(NC(=O)c4ccc(N5CCOCC5)c(c4)C(F)(F)F)c3)c12
NS(=O)(=O)c1ccc(cc1)-c1cnc2[nH]nc(C(=O)c3c(F)ccc(NS(=O)(=O)Cc4ccccc4)c3F)c2c1
Nc1ccc(cc1)-c1cnc2[nH]nc(C(=O)c3c(F)ccc(NS(=O)(=O)Cc4ccccc4)c3F)c2c1
O=S1(=O)CC2(OCCO2)c2cc3nccc(Nc4ccc5scnc5c4)c3cc12
Cc1cc(Oc2ccccc2)ccc1-n1c2ccnc3sc(C(=O)N[C@@H]4CCN(C4)C(=O)C=C)c([nH]c1=O)c23 |r,wD:25.26,(-1,4.5,;-2.28,3.77,;-3.62,4.54,;-4.95,3.77,;-6.28,4.54,;-7.62,3.77,;-8.95,4.54,;-10.28,3.77,;-10.28,2.23,;-8.95,1.46,;-7.62,2.23,;-4.95,2.23,;-3.62,1.46,;-2.28,2.23,;-.95,1.46,;-.95,-.08,;-2.28,-.85,;-2.28,-2.39,;-.95,-3.16,;.39,-2.39,;1.85,-2.87,;2.76,-1.62,;4.29,-1.65,;5.09,-.33,;5.04,-3,;6.58,-3,;7.49,-1.75,;8.95,-2.23,;8.95,-3.77,;7.49,-4.24,;10.28,-4.54,;10.28,-6.08,;11.62,-3.77,;11.62,-2.23,;1.72,-.08,;1.72,1.46,;.39,2.23,;.39,3.77,;.39,-.85,)|
CC(C)Oc1cc(F)ccc1Nc1ncnc2ccc(nc12)-c1ccc(cc1)C(=O)N1CCNCC1
C(Oc1cccc(c1)-c1nc2sccn2c1-c1ccncn1)c1ccccc1
CS(=O)(=O)c1nccc(n1)-c1c(nc2sccn12)-c1cccc(OCc2ccccc2)c1
c1cc(cc(c1)NC(=O)Nc2ccc(cc2)Oc3ccncc3)C(F)(F)F
FC(F)(F)c1cccc(NC(=O)Nc2ccc(Oc3ccncn3)cc2)c1
FC(F)(F)c1cccc(NC(=O)Nc2ccc(Oc3ccnc4ccccc34)cc2)c1
FC(F)(F)c1cccc(NC(=O)Nc2ccc(Oc3ncnc4ccccc34)cc2)c1
COc1ccc2ncnc(Oc3ccc(NC(=O)Nc4cccc(c4)C(F)(F)F)cc3)c2c1
COc1cc2ncnc(Oc3ccc(NC(=O)Nc4cccc(c4)C(F)(F)F)cc3)c2cc1OC
Cc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2)c2ccccc2n1
FC(F)(F)c1cccc(NC(=O)Nc2ccc(Oc3ccnc4[nH]ccc34)cc2)c1
FC(F)(F)c1cccc(NC(=O)Nc2ccc(Oc3ncnc4[nH]ccc34)cc2)c1
CNc1nccc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2)n1
CNc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2)ncn1
Nc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2)ncn1
CN(C)c1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2)ncn1
Oc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2)ncn1
COc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2)ncn1
Cc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2)ncn1
CCNc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2)ncn1
CC(C)Nc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2)ncn1
CCCNc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2)ncn1
CC(C)CNc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2)ncn1
OCCNc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2)ncn1
C[C@@H](O)CNc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2)ncn1 |r|
C[C@H](O)CNc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2)ncn1 |r|
CC(C)(O)CNc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2)ncn1
CC(=O)Nc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2)ncn1
OC(=O)Cc1cccc(Nc2cc(Oc3ccc(NC(=O)Nc4cccc(c4)C(F)(F)F)cc3)ncn2)c1
FC(F)(F)c1cccc(NC(=O)Nc2ccc(Oc3cc(Nc4cccc(CN5CCCC5)c4)ncn3)cc2)c1
CNc1cc(Oc2ccc(NC(=O)Nc3ccccc3)cc2)ncn1
CNc1cc(Oc2ccc(NC(=O)Nc3cccc(C)c3)cc2)ncn1
CNc1cc(Oc2ccc(NC(=O)Nc3cccc(CF)c3)cc2)ncn1
CNc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)F)cc2)ncn1
CCc1cccc(NC(=O)Nc2ccc(Oc3cc(NC)ncn3)cc2)c1
CNc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(C)F)cc2)ncn1
CNc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(C)(F)F)cc2)ncn1
CNc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(C)(C)C)cc2)ncn1
CNc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2F)ncn1
CNc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)c(F)c2)ncn1
CNc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)c(F)c2F)ncn1
CNc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2Cl)ncn1
CNc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)c3ccccc23)ncn1
CNc1cc(Oc2c(C)cc(NC(=O)Nc3cccc(c3)C(F)(F)F)c3ccccc23)ncn1
CNc1cc(Oc2ccc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2C)ncn1
CNc1cc(Oc2c(C)cc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2C)ncn1
CNc1cc(Oc2cc(C)c(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2C)ncn1
CNc1cc(ncn1)Oc2c(cc(cc2Cl)NC(=O)Nc3cccc(c3)C(F)(F)F)Cl
CNc1cc(Oc2c(F)cc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2F)ncn1
CNc1cc(Oc2c(C)cc(NC(=O)Nc3cccc(c3)C(F)(F)F)cc2Cl)ncn1
CCc1cc(NC(=O)Nc2cccc(c2)C(F)(F)F)cc(Cl)c1Oc1cc(NC)ncn1
CNS(=O)(=O)c1ccc(N(C)C)c(Nc2ncnc3[nH]ccc23)c1
CNS(=O)(=O)c1ccc(N(C)C)c(Nc2ncnc3cc(OC)c(OC)cc23)c1
COc1n[nH]c2ncc(NC(=O)c3cc(NC(=O)NCCC(C)(C)C)c(F)cc3C)cc12
CNc1cc(ncn1)-c1cccnc1Nc1cc(NC(=O)NCCC(C)(C)C)c(F)cc1C
CN(C(=O)Nc1cc(NC(=O)NCCC(C)(C)C)c(F)cc1C)c1cc(N)ncn1
Cc1cc(F)c(NC(=O)NCCC(C)(C)C)cc1NC(=O)c1cccc2c(N)ncnc12
Cc1cc(F)c(NC(=O)NCCC(C)(C)C)cc1Nc1ccc2ncn(C)c(=O)c2c1
Cc1cccc(n1)-c1n[nH]cc1-c1ccc2ncccc2n1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1ccc2NC(=O)CC3(CCOCC3)Oc2c1
Cc1ccc(NC(=O)c2cc(cnn2)C(F)(F)F)cc1-c1ccc2NC(=O)CC3(CCOCC3)Oc2c1
COc1ccc(CNc2ccc3n(cnc3c2)-c2ccccc2)cc1OC
COc1cc(CNc2ccc3n(cnc3c2)-c2ccccc2)ccc1OCCO
Fc1ccc(cc1)S(=O)(=O)NCCNc1nccc(n1)-c1c(nc2sccn12)-c1ccccc1
Cc1ccc(cc1)S(=O)(=O)NCCNc1nccc(n1)-c1c(nc2sccn12)-c1ccccc1
Fc1ccc(cc1)S(=O)(=O)NCCCNc1nccc(n1)-c1c(nc2sccn12)-c1ccccc1
COc1ccc(cc1)S(=O)(=O)NCCCNc1nccc(n1)-c1c(nc2sccn12)-c1ccccc1
Cc1ccc(cc1)S(=O)(=O)NCCCNc1nccc(n1)-c1c(nc2sccn12)-c1ccccc1
COc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccccc2)n1
COc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc(F)cc2)n1
COc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2cccc(F)c2)n1
COc1ccc(cc1)S(=O)(=O)NCCNc1nccc(n1)-c1c(nc2sccn12)-c1cccc(OC)c1
COc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc(C)cc2)n1
COc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc3ccccc3c2)n1
COc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccccc2)n1
COc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccc(F)cc2)n1
COc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2cccc(F)c2)n1
COc1ccc(cc1)S(=O)(=O)NCCCNc1nccc(n1)-c1c(nc2sccn12)-c1cccc(OC)c1
COc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccc(C)cc2)n1
COc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccc3ccccc3c2)n1
COc1ccc(cc1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc(F)cc2)n1
COc1ccc(cc1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc(OC)cc2)n1
COc1ccc(cc1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc(C)cc2)n1
COc1ccc(cc1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2cccc3ccccc23)n1
Oc1ccc(cc1)S(=O)(=O)NCCNc1nccc(n1)-c1c(nc2sccn12)-c1ccccc1
Oc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccccc2)n1
Cc1ccc(cc1)S(=O)(=O)NCCNc1nccc(n1)-c1c(nc2sccn12)-c1cccc(O)c1
Oc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccccc2)n1
Oc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2cccc(F)c2)n1
Cc1ccc(cc1)S(=O)(=O)NCCCNc1nccc(n1)-c1c(nc2sccn12)-c1cccc(O)c1
Oc1ccc(cc1)-c1nc2sccn2c1-c1ccnc(NCCNS(=O)(=O)c2ccc(O)cc2)n1
Cc1ccc(cc1)S(=O)(=O)NCCNc1nccc(n1)-c1c(nc2sccn12)-c1ccc(O)cc1
COc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCN2CCN(C)S2(=O)=O)n1
COc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCN2CCN(Cc3ccccc3)S2(=O)=O)n1
COc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCN2CC(C)(C)NS2(=O)=O)n1
COc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCN2CCCN(C)S2(=O)=O)n1
COc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCN2CCNS2(=O)=O)n1
COc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCN2CCCNS2(=O)=O)n1
COc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCN2CCCN(C(=O)OC(C)(C)C)S2(=O)=O)n1
CN1CCN(CCNc2nccc(n2)-c2c(nc3sccn23)-c2cccc(O)c2)S1(=O)=O
Oc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCN2CCN(Cc3ccccc3)S2(=O)=O)n1
CC1(C)CN(CCNc2nccc(n2)-c2c(nc3sccn23)-c2cccc(O)c2)S(=O)(=O)N1
CN1CCCN(CCNc2nccc(n2)-c2c(nc3sccn23)-c2cccc(O)c2)S1(=O)=O
Oc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCN2CCNS2(=O)=O)n1
Oc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCN2CCCNS2(=O)=O)n1
CC(C)(C)OC(=O)N1CCCN(CCNc2nccc(n2)-c2c(nc3sccn23)-c2cccc(O)c2)S1(=O)=O
Oc1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCNC(=O)c2ccccc2)n1
[O-][N+](=O)c1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccc(F)cc2)n1
[O-][N+](=O)c1cccc(c1)-c1nc2sccn2c1-c1ccnc(NCCCNS(=O)(=O)c2cccc(F)c2)n1
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C(=O)NCCOCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(cc2)-c2scnc2C)C(C)(C)C)c1F |r|
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C(=O)NCCOCCOCCOCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(cc2)-c2scnc2C)C(C)(C)C)c1F |r|
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C(=O)NCCCCCCOCCCCCOCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(cc2)-c2scnc2C)C(C)(C)C)c1F |r|
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(CNC(=O)CCCCOCCCCOCCCCOc3cc(ccc3CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3Cc4ccccc4C3=O)-c3scnc3C)cc2)c1F |r|
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(cc2)C(=O)NCCOCCOCCOCCOc2cc(ccc2CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)-c2scnc2C)c1F |r|
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(CNC(=O)CCCCOCCOCCOCCOc3cc(ccc3CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3Cc4ccccc4C3=O)-c3scnc3C)cc2)c1F |r|
COCC1CN(C1)C1CCN(CC1)c1cc(OC)c(Nc2ncc(Br)c(Nc3ccc4OCCOc4c3P(C)(C)=O)n2)cc1C
COc1cc(CN(c2ccc(F)c(C#Cc3cnc4[nH]nc(-c5ccc(F)cc5)c4c3)c2F)S(=O)(=O)c2cccnc2)c(cc1OC)[N+]([O-])=O
Fc1ccc(cc1)-c1n[nH]c2ncc(cc12)C#Cc1c(F)ccc(NS(=O)(=O)c2cccnc2)c1F
CC(C)S(=O)(=O)N1Cc2nc(nc(N3CCOCC3C)c2C1)-c1c[nH]c2ccccc12
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1ccc2C(=O)NC3(CCOCC3)Oc2c1
CC(=O)Nc1cccc(c1)-c1cncc(NCc2cc(C)n[nH]2)n1
CC(=O)Nc1cccc(c1)-c1cncc(NCCc2ccccc2)n1
CC(=O)Nc1cccc(c1)-c1cncc(Nc2nc(cs2)C(C)(C)C)n1
CC(=O)Nc1cccc(c1)-c1cncc(Nc2cccc(Cl)c2)n1
CC(=O)Nc1cccc(c1)-c1cncc(NCc2ccc3OCOc3c2)n1
CC(=O)Nc1cccc(c1)-c1cncc(NCc2cc(C)on2)n1
COc1cc(Nc2cncc(n2)-c2cccc(NC(C)=O)c2)cc(OC)c1
CC(=O)Nc1cccc(c1)-c1cncc(Nc2ccc3OCOc3c2)n1
CC(=O)Nc1cccc(c1)-c1cncc(Nc2ccc3OC(F)(F)C(F)(F)Oc3c2)n1
COc1cc(Nc2cncc(n2)-c2cccc(NC(C)=O)c2)cc(OC)c1OC
COc1cc(CNc2cncc(n2)-c2cccc(NC(C)=O)c2)cc(OC)c1OC
CC(=O)Nc1cccc(c1)-c1cncc(Nc2ccc3OCCOc3c2)n1
CC(=O)Nc1cccc(c1)-c1cncc(NCCCc2ccccc2)n1
COc1ccc(Nc2cncc(n2)-c2cccc(NC(C)=O)c2)cc1OC
CC(=O)Nc1cccc(c1)-c1cncc(NCCOc2ccccc2)n1
COc1cccc(Nc2cncc(n2)-c2cccc(NC(C)=O)c2)c1
CC(=O)Nc1cccc(c1)-c1cncc(NCc2ccoc2)n1
CC(=O)Nc1cccc(c1)-c1cncc(Nc2cccc3OC(F)(F)C(F)(F)Oc23)n1
CC(=O)Nc1cccc(c1)-c1cncc(Nc2ccc3OC(F)(F)Oc3c2)n1
CC(=O)Nc1cccc(c1)-c1cncc(NCc2cccc(F)c2)n1
CC(=O)Nc1cccc(c1)-c1cncc(NCc2ccc(F)c(Cl)c2)n1
CN(Nc1cncc(n1)-c1cccc(NC(C)=O)c1)c1ccccc1
CC(=O)Nc1cccc(c1)-c1cncc(Nc2cccc(c2)-c2cnco2)n1
COc1ccc(Nc2cncc(n2)-c2cccc(NC(C)=O)c2)c(OC)c1
CC(=O)Nc1cccc(c1)-c1cncc(Nc2ccccc2)n1
CC(=O)Nc1cccc(c1)-c1cncc(NCc2ccccn2)n1
COc1ccc(OCCNc2cncc(n2)-c2cccc(NC(C)=O)c2)cc1
CC(=O)Nc1cccc(c1)-c1cncc(Nc2ccc(cc2)N2CCOCC2)n1
CC(=O)Nc1cccc(c1)-c1cncc(Nc2ccc(OC(F)(F)F)cc2)n1
CC(=O)Nc1cccc(c1)-c1cncc(Nc2cc(Cl)nc(Cl)c2)n1
CC(=O)Nc1cccc(c1)-c1cncc(Nc2ccc3OCCCOc3c2)n1
CC(=O)Nc1cccc(c1)-c1cncc(Nc2ccc(cc2)S(=O)(=O)N2CCOCC2)n1
CC(=O)Nc1cccc(c1)-c1cncc(Nc2cccc(OCCN)c2)n1
CC(=O)Nc1cccc(c1)-c1cncc(Nc2ccc3COC(=O)c3c2)n1
CC(=O)Nc1cccc(c1)-c1cncc(Nc2cccc(O)c2)n1
COc1ccccc1Nc1cncc(n1)-c1cccc(NC(C)=O)c1
CC(=O)Nc1cccc(c1)-c1cncc(NCc2ccccc2)n1
COc1ccc(Nc2cncc(n2)-c2cccc(NC(C)=O)c2)cc1
CC(=O)Nc1cccc(c1)-c1cncc(NCc2ccc3OCCOc3c2)n1
CC(=O)Nc1cccc(c1)-c1cncc(Nc2ccc(F)c(Cl)c2)n1
Nc1nccc(n1)-c1sc(nc1-c1cccc(NS(=O)(=O)c2cc(F)ccc2F)c1F)C1CCN1
Nc1nccc(n1)-c1sc(nc1-c1cccc(NS(=O)(=O)c2cc(F)ccc2F)c1F)C1CCCN1
Nc1nccc(n1)-c1sc(nc1-c1cccc(NS(=O)(=O)c2cc(F)ccc2F)c1F)C1CCCCN1
Nc1nccc(n1)-c1sc(nc1-c1cccc(NS(=O)(=O)c2cc(F)ccc2F)c1F)C1CNCCN1
CC(C)(C)c1nc(c(s1)-c1ccnc(N)n1)-c1cc(Cl)cc(NS(=O)(=O)c2cc(F)ccc2F)c1F
Nc1nccc(n1)-c1sc(nc1-c1cc(Cl)cc(NS(=O)(=O)c2cc(F)ccc2F)c1F)C1COCCN1
Nc1nccc(n1)-c1sc(nc1-c1cccc(NS(=O)(=O)c2cc(F)ccc2F)c1F)C1CCN(CC1)C1CC1
Nc1nccc(n1)-c1sc(nc1-c1cccc(NS(=O)(=O)c2cc(F)ccc2F)c1F)C1CCCNC1
Nc1nccc(n1)-c1sc(nc1-c1cccc(NS(=O)(=O)c2cc(F)ccc2F)c1F)C1COCCN1
NCCCc1nc(c(s1)-c1ccnc(N)n1)-c1cccc(NS(=O)(=O)c2cc(F)ccc2F)c1F
CC(=O)Nc1nccc(n1)-c1sc(CCCN)nc1-c1cccc(NS(=O)(=O)c2cc(F)ccc2F)c1F
CCN(C)S(=O)(=O)Nc1cccc(c1)-c1nc(sc1-c1ccnc(N)n1)C(C)(C)C
C[C@@H]1COCCN1c1nc(nc2ccc(cc12)-c1ccnn1C)-c1cccc2[nH]ccc12 |r|
FC(F)(F)c1ccc(NC(=O)Nc2ccc(Oc3ccc(cc3)C(=O)c3ncc[nH]3)cc2)cc1Cl
COc1ccc(NC(=O)Nc2ccc(Oc3ccc(cc3)C(=O)c3ncc[nH]3)cc2)cc1
Fc1ccc(NS(=O)(=O)c2ccoc2)c(F)c1Nc1ccccc1-c1ncnc2[nH]cnc12
CCCCN1CCN(CC1)Oc1cc2nccc(Oc3ccc(NS(=O)(=O)c4cc(F)ccc4F)cc3F)c2cc1OC
CN1CCN(CCNc2nccc(n2)C2(CC2)C(=O)Nc2cc(ccc2C)C(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)CC1
Oc1cccc(c1)-c1nn(cc1-c1ccnc(NCCCNS(=O)(=O)c2ccc(Cl)cc2)c1)-c1ccccc1
Cc1nn(c(Cl)c1Nc1ccc(cc1)C(F)(F)F)-c1ccccc1
COc1ccc(cc1)-n1cc(NC(=O)c2cccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)c2)cn1
Cc1ccc(cc1)C1=NN=C(NC(=S)Nc2ccc(Cl)cc2)SC1 |t:8,10|
FC(F)(F)c1cc(NC(=O)Nc2ccc(Oc3ccc(cc3)C(=O)c3ncc[nH]3)cc2)ccc1Cl
Cc1nccn1-c1cc(cc(c1)C(F)(F)F)C(=O)Nc1cccc(c1)-c1cc([nH]n1)C(=O)OCCN1CCOCC1
[H][C@@]12C[C@@H](COC)C(NN)[C@@]1(C)CC[C@]1([H])c3ccc(O)cc3CC[C@@]21[H] |r|
CN(C)CCOc1ccc(cc1)-c1n\c(c([nH]1)=C1C=CNC=C1)=c1/ccc2=C(CCc2c1)N=O |c:20,23,t:29,(10.25,3.39,;8.71,3.39,;7.94,4.72,;7.94,2.06,;6.4,2.06,;5.63,.72,;4.09,.72,;3.32,2.06,;1.77,2.06,;1.01,.72,;1.78,-.61,;3.32,-.61,;-.53,.72,;-1.43,-.53,;-2.9,-.05,;-2.9,1.49,;-1.43,1.96,;-4.23,2.26,;-5.57,1.49,;-6.9,2.26,;-6.9,3.8,;-5.57,4.57,;-4.23,3.81,;-4.23,-.82,;-4.23,-2.36,;-5.57,-3.13,;-6.9,-2.36,;-8.36,-2.84,;-9.27,-1.59,;-8.36,-.35,;-6.9,-.82,;-5.57,-.05,;-8.76,-4.32,;-10.25,-4.72,)|
COc1ccc(cc1)-n1cc(Nc2cccc3[nH]ncc23)cn1
Cc1ccc(cc1)-n1cc(NC(=O)c2c[nH]c3ccccc23)cn1
COc1cc(ccc1Cl)-c1nn(cc1-c1ccncc1)-c1ccc(NC(=O)CN2CCOCC2)cc1
COC(=O)c1ccccc1-c1ccc(\C=C\[N+]([O-])=O)o1
COc1cccc(c1)-c1nn(cc1-c1ccncc1)-c1ccccc1
Cn1ncc2c(Oc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)cc3)ncnc12
CC(=O)Nc1cc(ccn1)-c1sc(nc1-c1cccc(NS(=O)(=O)c2cc(F)ccc2F)c1F)C1CCN(CC1)C1CC1
CCC[S+]([O-])Nc1ccc(F)c(Cc2c[nH]c3nc(N)n(C)c(=O)c23)c1F
CC(C)[S+]([O-])Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(C)cc23)c1F
Fc1cccc(c1)-c1nc2occn2c1-c1ccnc(NCCCNS(=O)(=O)c2ccccc2)n1
COc1ccc(cc1)-c1n[nH]c(\N=C\c2ccc(O)c(OC)c2)n1
OCCn1cc(c(n1)-c1ccncc1)-c1ccc2\C(CCc2c1)=N/O
CN(C1CCN(CC1)C(=O)c1ccccc1)c1nc(nc(n1)-c1cnc(N)nc1)N1CCOCC1
COc1cccc(c1)-c1nn(cc1-c1ccnc(NCCCNC(=O)Nc2ccc(Cl)c(Cl)c2)c1)-c1ccccc1
Fc1ccc(NS(=O)(=O)c2cccc(c2)-c2ccccc2)c(F)c1-n1cc(nn1)-c1cnc2[nH]nc(OC3CCN(C3)C(=O)C=C)c2c1
Fc1ccc(NS(=O)(=O)c2ccccc2)c(F)c1-n1cc(nn1)-c1cnc2[nH]nc(OC3CCN(C3)C(=O)C=C)c2c1
O=C(Nc1ccccc1)N1CCN(CC1)c1nnc(Cc2ccccc2)c2ccccc12
COc1ccc(NC(=O)N2CCN(CC2)c2nnc(Cc3ccccc3)c3ccccc23)cc1
Clc1ccc(NC(=O)N2CCN(CC2)c2nnc(Cc3ccccc3)c3ccccc23)cc1
FC(F)(F)c1cc(NC(=O)N2CCN(CC2)c2nnc(Cc3ccccc3)c3ccccc23)ccc1Cl
COc1ccc(Cc2nnc(N3CCN(CC3)C(=O)Nc3ccccc3)c3ccccc23)cc1
COc1ccc(Cc2nnc(N3CCN(CC3)C(=O)Nc3ccc(OC)cc3)c3ccccc23)cc1
COc1ccc(Cc2nnc(N3CCN(CC3)C(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)c3ccccc23)cc1
S=C(Nc1ccccc1)N1CCN(CC1)c1nnc(Cc2ccccc2)c2ccccc12
COc1cccc(NC(=S)N2CCN(CC2)c2nnc(Cc3ccccc3)c3ccccc23)c1
COc1ccc(NC(=S)N2CCN(CC2)c2nnc(Cc3ccccc3)c3ccccc23)cc1
Clc1cccc(NC(=S)N2CCN(CC2)c2nnc(Cc3ccccc3)c3ccccc23)c1
Clc1ccc(NC(=S)N2CCN(CC2)c2nnc(Cc3ccccc3)c3ccccc23)cc1
COc1ccc(Cc2nnc(N3CCN(CC3)C(=S)Nc3ccccc3)c3ccccc23)cc1
COc1ccc(Cc2nnc(N3CCN(CC3)C(=S)Nc3ccc(OC)cc3)c3ccccc23)cc1
COc1ccc(Cc2nnc(N3CCN(CC3)C(=S)Nc3cccc(Cl)c3)c3ccccc23)cc1
COc1ccc(Cc2nnc(N3CCN(CC3)C(=S)Nc3ccc(Cl)cc3)c3ccccc23)cc1
O=C(N1CCN(CC1)c1nnc(Cc2ccccc2)c2ccccc12)c1ccccc1
COc1ccc(cc1)C(=O)N1CCN(CC1)c1nnc(Cc2ccccc2)c2ccccc12
Clc1ccc(cc1)C(=O)N1CCN(CC1)c1nnc(Cc2ccccc2)c2ccccc12
COc1ccc(Cc2nnc(N3CCN(CC3)C(=O)c3ccccc3)c3ccccc23)cc1
COc1cncc(c1)-c1cn(nn1)-c1c(F)ccc(NS(=O)(=O)C(C)C)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(N)cc2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(NC(=O)COCCOCCNC(=O)CCCCC[N+]3=C(C=CC=CC=C4/N(C)c5ccccc5C4(C)C)C(C)(C)c4ccccc34)cc2)c1F
COc1ccc(\C=C/c2cc(OC)c(OC)c(OC)c2)cc1NC(=O)CCC(=O)N[C@@H](CCCNC(N)=N)C(O)=O |r|
Nc1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
OCCOCCNc1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
FC1(F)Oc2ccc(NC(=O)c3ccccc3NCc3ccnc(NC(=O)NCc4ccccc4)c3)cc2O1
CNC(=O)Nc1ccc(CNc2ncsc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)cn1
CNC(=O)Nc1ccc(CNc2c(cnn2C)C(=O)Nc2ccc(SC(F)(F)F)cc2)cn1
FC1(F)Oc2ccc(NC(=O)c3ccccc3NCc3ccnc(c3)C3=NCCN3)cc2O1 |t:27|
NC(=O)c1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
FC1(F)Oc2ccc(NC(=O)c3ncsc3NCc3ccncc3)cc2OC1(F)F
FC1(F)Oc2ccc(NC(=O)c3ccccc3NCc3ccnc(c3)C(=O)NC3CC3)cc2O1
CCNC(=O)Nc1ccc(CNc2ncsc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)cn1
CNc1nccc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)n1
CNC(=O)Nc1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
CNC(=O)c1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
CNC(=O)Nc1ccc(CNc2c(cnn2C)C(=O)Nc2ccc3OC(F)(F)C(F)(F)Oc3c2)cn1
OCCNc1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
FC1(F)Oc2ccc(NC(=O)c3ccccc3NCc3ccncc3)cc2OC1(F)F
COCCNC(=O)c1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
FC1(F)Oc2ccc(NC(=O)c3ccccc3NCc3ccnc(NC(=O)Nc4ccc5CCCc5c4)c3)cc2O1
COCCCNc1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
CCN(CC)CCCNC(=O)c1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
CNC(=O)c1cc(CNc2c(cnn2C)C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
FC1(F)Oc2ccc(NC(=O)c3ccccc3NCc3ccnc(NC(=O)Nc4ccccc4)c3)cc2O1
COCCCNC(=O)c1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
COCCNc1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
OCCNC(=O)c1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
CCNC(=O)Nc1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
CCN(CC)CCNC(=O)c1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
CNC(=O)c1cc(CNc2ncsc2C(=O)Nc2ccc3OC(F)(F)C(F)(F)Oc3c2)ccn1
FC1(F)Oc2ccc(NC(=O)c3ccccc3NCc3ccnc(c3)C(=O)NCCCN3CCOCC3)cc2O1
FC1(F)Oc2ccc(NC(=O)c3ccccc3NCc3ccnc(NCCCn4ccnc4)c3)cc2O1
CS(=O)(=O)Nc1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
CNC(=O)c1cc(CNc2ccsc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
CN(C)c1nccc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)n1
OCCCNc1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
FC1(F)Oc2ccc(NC(=O)c3ccccc3NCc3ccnc(c3)C#N)cc2O1
CCNC(=O)c1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
CNC(=O)c1cc(CNc2ncsc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
CS(=O)(=O)CCNC(=O)c1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
FC1(F)Oc2ccc(NC(=O)c3ccccc3NCc3ccnc(NCCc4cnc[nH]4)c3)cc2O1
CNc1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
CC(=O)Nc1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
NC(=S)c1cc(CNc2ccccc2C(=O)Nc2ccc3OC(F)(F)Oc3c2)ccn1
CCN(C)S(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(Cl)cc2)c1F
CC(C)(C#N)c1cccc(c1)C(=O)Nc2ccc(c(c2F)C(=O)c3c[nH]c4c3cc(cn4)Cl)F
O=C(CSc1nc2sc3c(c2c(=O)n1-c1ccc(Cl)cc1)CCCC3)NNC(=O)Nc1cccc(C(F)(F)F)c1
O=C(CSc1nc2sc3c(c2c(=O)n1-c1ccc(Cl)cc1)CCCC3)NNC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1
O=C(CSc1nc2ccccc2c(=O)n1-c1ccc(Cl)cc1)Nc1ccc(-c2nc3ccccc3[nH]2)cc1
COc1ccc(-n2c(SCC(=O)Nc3ccc(-c4nc5ccccc5[nH]4)cc3)nc3ccccc3c2=O)cc1
NC(=O)CCn1cc(nn1)-c1ccc2ncnc(Nc3cc(O)c(F)cc3F)c2c1
Cc1ccc(-c2ccnc(-c3ccnc4[nH]ccc34)n2)c(C)n1
Cc1ccc(NC(=O)N2CCO[C@H](C(F)(F)F)C2)cc1-c1cc(OCCO)nc(N2CCOCC2)c1
Cc1ccc(NC(=O)N2CCO[C@@H](C(F)(F)F)C2)cc1-c1cc(OCCO)nc(N2CCOCC2)c1
Cc1ccc(NC(=O)N2CC[C@@H](C(F)(F)F)C2)cc1-c1cc(OCCO)nc(N2CCOCC2)c1
Cc1ccc(NC(=O)N2CC[C@H](C(F)(F)F)C2)cc1-c1cc(OCCO)nc(N2CCOCC2)c1
Cc1ccc(NC(=O)N2CC[C@@H](CC(F)(F)F)C2)cc1-c1cc(OCCO)nc(N2CCOCC2)c1
Cc1ccc(NC(=O)N2CC[C@@H](CC(F)(F)F)C2)cc1-c1cc(OC[C@@H](C)O)nc(N2CCOCC2)c1
Cc1ccc(NC(=O)N2CC[C@@H](CC(F)(F)F)C2)cc1-c1cc(OCC(C)(C)O)nc(N2CCOCC2)c1
Cc1ccc(NC(=O)N2CC[C@@H](CC(F)(F)F)C2)cc1-c1cc(O[C@@H](C)CO)nc(N2CCOCC2)c1
Cc1ccc(NC(=O)N2CC[C@@H](CC(F)(F)F)C2)cc1-c1cc(O[C@H](C)CO)nc(N2CCOCC2)c1
C[C@H](CO)Nc1cc(cc(n1)N1CCOCC1)-c1cc(NC(=O)N2CC[C@@H](CC(F)(F)F)C2)ccc1C |r|
C/C(=NO)c1ccc(NC(=O)c2cc(-c3ccc(S(C)(=O)=O)cc3)nc3ccccc23)cc1
COCCOc1cc2c(cc1OCCOC)ncnc2Nc3cccc(c3)C#C
C=CCn1c(SCC(=O)Nc2ccc(C(=O)/C=C/c3ccc(Cl)cc3)cc2)nnc1-c1cc(-c2ccccc2)nc2ccccc12
O=C(Nc1cc(-c2ccc(Br)cc2)[nH]n1)c1ccnc(F)c1
OCCn1cc(-c2ccc3c(c2)C/C(=NO)C3)c(-c2ccncc2)n1
CCCS(=O)(=O)Nc1ccc(F)c(Oc2ccc3ncn(C)c(=O)c3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(Sc2ccc3ncn(C)c(=O)c3c2)c1F
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2F)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2Cl)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2OC)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(CC)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C(C)C)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(CC4CC4)c(=O)c3c2C)c1Cl
CCCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C4CC4)c(=O)c3c2C)c1Cl
Cc1c(ccc2c1C(=O)N(C=N2)C)Nc3c(ccc(c3Cl)NS(=O)(=O)CCCF)F
CCS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
CC(C)CS(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
Cc1c(Nc2c(F)ccc(NS(=O)(=O)CC3CC3)c2Cl)ccc2ncn(C)c(=O)c12
CCC(C)S(=O)(=O)Nc1ccc(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
Cc1c(Nc2c(F)ccc(NS(=O)(=O)C3CC3)c2Cl)ccc2ncn(C)c(=O)c12
Cc1ccc(NC(=O)c2cccc(C(F)(F)F)c2)cc1-n1cc(-c2cncc(N3CCOCC3)c2)cn1
C[C@H](c1ncc(s1)C(=O)Nc2cc(c(cn2)Cl)C(F)(F)F)NC(=O)c3c(c(ncn3)N)Cl
Fc1ccccc1NC(=O)N[C@@H]1[C@H]2Oc3ccc(Oc4ccnc5NC(=O)CCc45)cc3[C@@H]12 |r|
CC(C)C(=O)Nc1ccc(-c2nc(-c3cccc(O)c3)c(-c3ccnc(Br)c3)[nH]2)cc1
CCCS(=O)(=O)Nc1cc(F)c(F)c(Nc2ccc3ncn(C)c(=O)c3c2C)c1Cl
CC(C)[C@@H]1NC(=O)[C@H](Cc2cnc[nH]2)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](N)CCCCNC(=O)CC[C@@H](C(N)O)NC(=O)[C@H](C)NC1=O
CNS(=O)(=O)Nc1cccc(Cn2cnc3c(F)c(Nc4ccc(C5CC5)cc4F)c(C(=O)NOCCO)cc32)c1
CCNS(=O)(=O)Nc1cccc(Cn2cnc3c(F)c(Nc4ccc(C5CC5)cc4F)c(C(=O)NOCCO)cc32)c1
CNS(=O)(=O)Nc1cccc(Cn2cnc3c(F)c(Nc4ccc(C5CC5)cc4F)c(C(=O)NOCCO)cc32)c1F
CCNS(=O)(=O)Nc1cccc(Cn2cnc3c(F)c(Nc4ccc(C5CC5)cc4F)c(C(=O)NOCCO)cc32)c1F
CNS(=O)(=O)Nc1cccc(Cn2cnc3c(F)c(Nc4ccc(I)cc4F)c(C(=O)NOCCO)cc32)c1F
CC(C)(C)c1nc(-c2cccc(NS(=O)(=O)c3c(F)cccc3F)c2F)c(-c2ccnc(NCCCCCCC(=O)NO)n2)s1
O=C(CCCCCCNc1nccc(-c2sc(-c3ccccc3)nc2-c2cccc(NS(=O)(=O)c3c(F)cccc3F)c2F)n1)NO
COc1ccc(-c2c(C#N)c(N)nc3sc(C(N)=O)c(N)c23)cc1OC
N#Cc1c(N)nc2sc(C(N)=O)c(N)c2c1-c1ccc(Cl)cc1
Cn1cc(-c2cccc(NC(=O)c3cc4c(nc3O[C@H]3C[C@@H](O)C3)OC(C)(C)C4)n2)cn1
O=C(Nc1ccc(-c2ccc3c(=O)[nH]cnc3c2)cc1)Nc1ccc(F)c(F)c1
N#Cc1c(-c2ccc(Cl)cc2Cl)cc(-c2c[nH]c3ccccc23)[nH]c1=O
C[C@@H](C(F)(F)F)N(Cc1ccc(cc1)F)C(=O)CN2C(=O)[C@]3(CCc4c3ccc(c4)NC(=O)NC)OC2=O
Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1Nc1nc(-c2cccnc2)nc2nn(C)cc12
Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1Nc1nc(-c2cccnc2)nc2c1cnn2C
CC[C@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2N(C)C1=O |r|
CCOc1cc(ccc1Nc2ncc3c(n2)N(c4ccccc4C(=O)N3C)C)N5CCC(CC5)O
Cc1cn(CCN2CCN(CC2)c2ccccc2-c2cc(cc(c2)C(=O)NCCCN2CCCC2)C#N)c2ccccc12
CCc1cc(Nc2nccc(n2)-c2c(nc3ccccn23)-c2ccc(OC)c(c2)C(=O)Nc2c(F)cccc2F)c(OC)cc1N1CCC(CC1)N1CCN(CC1)S(C)(=O)=O
CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3cc(nn3-c3ccc4ncccc4c3)C(C)(C)C)c(F)c2)ccn1
c1cc(c(cc1I)F)Nc2c(ccc(c2F)F)C(=O)N3CC(C3)([C@@H]4CCCCN4)O
CCN1CCN(Cc2ccc(Nc3ncc(F)c(n3)-c3cc(F)c4nc(C)n(C(C)C)c4c3)nc2)CC1
CCN1CCN(CC1)Cc2ccc(cc2C(F)(F)F)NC(=O)c3ccc(c(c3)Oc4ccnc5c4cc[nH]5)C
CCN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(/C=C/c4cnc5[nH]ccc5c4OC)c3)cc2C(F)(F)F)CC1
O=C(NCC#N)c1ccc(cc1)-c1ccnc(Nc2ccc(cc2)N2CCOCC2)n1
CC[C@@H]1CN(C[C@@H]1c1cnc2cnc3[nH]ccc3n12)C(=O)NCC(F)(F)F |r|
CCN1CCN(CC\C=C\c2ccc3c(Nc4ccc(Sc5nccn5C)c(Cl)c4)c(cnc3c2)C#N)CC1
Oc1cc(CNC=C2C(=O)NC(=O)c3ccc(I)cc23)ccc1-c1ccoc1 |w:6.5|
COc1c(NC(=O)Nc2ccc(-c3ccc(CN4CCOCC4)nc3)c3ccccc23)cc(cc1NS(C)(=O)=O)C(C)(C)C
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2ccnn12
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)Nc2cc(ccc2Cl)C(F)(F)F)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)Nc2ccc(F)c(c2)C(F)(F)F)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)Nc2ccc(C)c(c2)C(F)(F)F)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)Nc2cccc(Cl)c2)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)Nc2ccccc2C(F)(F)F)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)Nc2ccc(cc2)C(F)(F)F)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)Nc2cccc(c2)C(F)(F)F)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cc(ccc2Cl)C(F)(F)F)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cc(ccc2C)C(F)(F)F)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2ccc(Cl)c(c2)C(F)(F)F)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2ccc(OC)c(c2)C(F)(F)F)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2ccc(C)c(c2)C(F)(F)F)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2ccc(cc2)C(F)(F)F)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(OC(F)(F)F)c2)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C#N)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(Br)c2)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(Cl)c2)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(OC)c2)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(C)c2)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2ccccc2)c1
CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
COCCCNC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c1
FC(F)(F)c1cc(NC(=O)Nc2cccc(c2)-c2ccnc3c(cnn23)C(=O)NCCN2CCOCC2)ccc1Cl
CCN(CC)CCNC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2c(cnn12)C(=O)NCCN1CCOCC1
CN(C)CCNC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
CNC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
NC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
CN(C)CCOC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
FC(F)(F)COC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
COC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
OC(=O)c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2c(cnn12)C#N
CCOC(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc(OC)c1 |THB:13:11:5:7.8|
CCOC(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(Cl)c(OC)c1 |THB:13:11:5:7.8|
CCOC(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc(O)c1 |THB:13:11:5:7.8|
COc1cccc(c1)-c1c(nn2c(ccnc12)C1CC2CCC(C1)N2)-c1ccncc1 |TLB:12:17:24:20.21|
COc1cc(ccc1Cl)-c1c(nn2c(ccnc12)C1CC2CCC(C1)N2)-c1ccncc1 |TLB:13:18:25:21.22|
Oc1cccc(c1)-c1c(nn2c(ccnc12)C1CC2CCC(C1)N2)-c1ccncc1 |TLB:11:16:23:19.20|
Oc1cc(ccc1Cl)-c1c(nn2c(ccnc12)C1CC2CCC(C1)N2)-c1ccncc1 |TLB:12:17:24:20.21|
CCN1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(Cl)c(OC)c1 |THB:10:8:2:4.5|
CCN1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(Cl)c(O)c1 |THB:10:8:2:4.5|
CCN1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(C#N)c(O)c1 |THB:10:8:2:4.5|
CCN1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(F)c(O)c1 |THB:10:8:2:4.5|
CC(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(Cl)c(O)c1 |THB:11:9:3:5.6|
CCOC(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(F)c(F)c1 |THB:13:11:5:7.8|
CCOC(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(cc1)-c1nnco1 |THB:13:11:5:7.8|
CCOC(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc2cc[nH]c2c1 |THB:13:11:5:7.8|
CCOC(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ccc12 |THB:13:11:5:7.8,(14.43,.28,;13.11,-.51,;11.77,.23,;10.45,-.56,;9.1,.18,;10.47,-2.1,;9.94,-3.57,;8.42,-4.25,;9.79,-4.21,;10.98,-3.35,;12.52,-4.19,;11.98,-5.67,;11.54,-4.48,;11.98,-7.21,;10.65,-7.98,;10.65,-9.52,;11.99,-10.29,;13.32,-9.52,;14.79,-9.99,;15.7,-8.74,;14.79,-7.49,;13.32,-7.97,;17.24,-8.74,;18.01,-10.08,;19.54,-10.08,;20.31,-8.74,;19.54,-7.4,;18,-7.41,;15.4,-11.41,;14.47,-12.63,;15.07,-14.06,;16.6,-14.25,;17.53,-13.02,;19.08,-12.88,;19.42,-11.36,;18.09,-10.57,;16.92,-11.59,)|
CCOC(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc2CC(=O)Nc2c1 |THB:13:11:5:7.8|
CCOC(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]c(=O)[nH]c12 |THB:13:11:5:7.8,(-.79,-20.79,;-2.11,-21.58,;-3.46,-20.84,;-4.78,-21.63,;-6.12,-20.89,;-4.75,-23.17,;-5.28,-24.64,;-6.81,-25.32,;-5.43,-25.28,;-4.24,-24.42,;-2.7,-25.27,;-3.24,-26.74,;-3.69,-25.55,;-3.24,-28.28,;-4.57,-29.05,;-4.57,-30.59,;-3.24,-31.37,;-1.9,-30.59,;-.43,-31.07,;.48,-29.82,;-.43,-28.56,;-1.9,-29.04,;2.02,-29.81,;2.79,-31.15,;4.33,-31.15,;5.1,-29.82,;4.32,-28.48,;2.78,-28.49,;-.36,-32.61,;-1.66,-33.43,;-1.6,-34.97,;-.24,-35.69,;1.07,-34.87,;2.57,-35.28,;3.42,-33.99,;4.96,-33.92,;2.45,-32.77,;1,-33.32,)|
CCOC(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |THB:13:11:5:7.8,(16.08,-21.46,;14.76,-22.25,;13.41,-21.51,;12.09,-22.3,;10.75,-21.56,;12.12,-23.84,;11.59,-25.31,;10.07,-25.99,;11.44,-25.95,;12.63,-25.09,;14.17,-25.94,;13.63,-27.41,;13.18,-26.22,;13.63,-28.95,;12.3,-29.72,;12.3,-31.26,;13.63,-32.03,;14.97,-31.26,;16.44,-31.73,;17.35,-30.49,;16.44,-29.23,;14.97,-29.71,;18.88,-30.48,;19.65,-31.82,;21.19,-31.82,;21.96,-30.48,;21.18,-29.15,;19.65,-29.15,;16.51,-33.27,;15.21,-34.09,;15.27,-35.64,;16.63,-36.35,;17.94,-35.53,;19.43,-35.94,;20.29,-34.65,;19.32,-33.44,;17.87,-33.98,)|
OC(=O)[C@H]1CCCN1C(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wU:3.2,THB:18:16:10:12.13,(28.67,-19.29,;28.61,-20.83,;27.25,-21.54,;29.91,-21.65,;31.37,-21.16,;32.29,-22.4,;31.39,-23.66,;29.92,-23.2,;28.69,-24.11,;27.34,-23.37,;28.71,-25.65,;28.18,-27.12,;26.66,-27.8,;28.03,-27.77,;29.22,-26.9,;30.76,-27.75,;30.22,-29.22,;29.78,-28.03,;30.22,-30.76,;28.89,-31.53,;28.89,-33.08,;30.23,-33.85,;31.56,-33.08,;33.03,-33.55,;33.94,-32.3,;33.03,-31.05,;31.56,-31.53,;35.48,-32.3,;36.25,-33.63,;37.79,-33.63,;38.56,-32.3,;37.78,-30.96,;36.24,-30.97,;33.1,-35.09,;31.8,-35.91,;31.86,-37.45,;33.22,-38.17,;34.53,-37.35,;36.03,-37.76,;36.88,-36.47,;35.91,-35.26,;34.46,-35.8,)|
CS(=O)(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |THB:12:10:4:6.7,(-3.77,1.28,;-5.1,.49,;-6.44,-.27,;-6.43,1.27,;-5.06,-1.05,;-5.6,-2.52,;-7.12,-3.2,;-5.75,-3.16,;-4.56,-2.3,;-3.02,-3.14,;-3.56,-4.62,;-4,-3.43,;-3.56,-6.16,;-4.88,-6.93,;-4.89,-8.47,;-3.55,-9.24,;-2.22,-8.47,;-.75,-8.94,;.16,-7.69,;-.75,-6.44,;-2.22,-6.92,;1.7,-7.69,;2.47,-9.03,;4,-9.03,;4.77,-7.69,;4,-6.35,;2.46,-6.36,;-.68,-10.48,;-1.98,-11.3,;-1.92,-12.84,;-.56,-13.56,;.75,-12.74,;2.25,-13.15,;3.1,-11.86,;2.13,-10.65,;.68,-11.19,)|
CN(C)C(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |THB:13:11:5:7.8,(13.39,-1.4,;12.04,-.65,;12.02,.89,;10.72,-1.45,;9.38,-.7,;10.75,-2.98,;10.22,-4.45,;8.7,-5.13,;10.07,-5.1,;11.26,-4.23,;12.8,-5.08,;12.26,-6.55,;11.81,-5.36,;12.26,-8.09,;10.93,-8.86,;10.93,-10.4,;12.26,-11.17,;13.6,-10.4,;15.07,-10.88,;15.98,-9.63,;15.07,-8.37,;13.6,-8.85,;17.51,-9.62,;18.28,-10.96,;19.82,-10.96,;20.59,-9.63,;19.81,-8.29,;18.28,-8.3,;15.14,-12.41,;13.84,-13.24,;13.9,-14.78,;15.26,-15.5,;16.57,-14.67,;18.06,-15.09,;18.92,-13.79,;17.95,-12.58,;16.5,-13.13,)|
CCNC(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |THB:13:11:5:7.8,(29.22,-.78,;27.9,-1.58,;26.56,-.83,;25.24,-1.63,;23.89,-.88,;25.27,-3.16,;24.73,-4.63,;23.21,-5.31,;24.58,-5.28,;25.77,-4.41,;27.31,-5.26,;26.77,-6.73,;26.33,-5.54,;26.78,-8.27,;25.45,-9.04,;25.45,-10.58,;26.78,-11.35,;28.11,-10.58,;29.59,-11.06,;30.5,-9.81,;29.58,-8.55,;28.11,-9.03,;32.03,-9.8,;32.8,-11.14,;34.34,-11.14,;35.11,-9.81,;34.33,-8.47,;32.79,-8.48,;29.65,-12.6,;28.35,-13.42,;28.41,-14.96,;29.77,-15.68,;31.08,-14.85,;32.58,-15.27,;33.43,-13.97,;32.47,-12.76,;31.01,-13.31,)|
CC(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |THB:11:9:3:5.6,(42.06,-.04,;40.74,-.83,;39.39,-.09,;40.77,-2.37,;40.23,-3.84,;38.71,-4.52,;40.08,-4.48,;41.27,-3.62,;42.81,-4.47,;42.27,-5.94,;41.83,-4.75,;42.28,-7.48,;40.95,-8.25,;40.95,-9.79,;42.28,-10.56,;43.61,-9.79,;45.09,-10.26,;46,-9.02,;45.08,-7.76,;43.61,-8.24,;47.53,-9.01,;48.3,-10.35,;49.84,-10.35,;50.61,-9.01,;49.83,-7.68,;48.29,-7.68,;45.15,-11.8,;43.85,-12.62,;43.91,-14.17,;45.27,-14.88,;46.58,-14.06,;48.08,-14.47,;48.93,-13.18,;47.97,-11.97,;46.51,-12.51,)|
OCCN1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |THB:11:9:3:5.6,(-4.35,-23.89,;-5.7,-23.15,;-7.02,-23.94,;-6.99,-25.48,;-7.53,-26.95,;-9.05,-27.63,;-7.68,-27.59,;-6.48,-26.73,;-4.95,-27.58,;-5.49,-29.05,;-5.93,-27.86,;-5.48,-30.59,;-6.81,-31.36,;-6.81,-32.9,;-5.48,-33.67,;-4.15,-32.9,;-2.67,-33.38,;-1.76,-32.13,;-2.68,-30.87,;-4.15,-31.35,;-.23,-32.12,;.54,-33.46,;2.08,-33.46,;2.85,-32.12,;2.07,-30.79,;.53,-30.79,;-2.61,-34.91,;-3.91,-35.73,;-3.85,-37.28,;-2.49,-37.99,;-1.18,-37.17,;.32,-37.58,;1.17,-36.29,;.21,-35.08,;-1.25,-35.62,)|
CC(C)(C)OC(=O)[C@H]1CCCN1C(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wU:7.6,THB:22:20:14:16.17,(10.21,-19.41,;10,-20.93,;8.57,-21.52,;8.74,-20.04,;11.22,-21.88,;11.15,-23.42,;9.79,-24.13,;12.45,-24.24,;13.91,-23.75,;14.83,-24.99,;13.93,-26.25,;12.47,-25.79,;11.23,-26.71,;9.88,-25.96,;11.26,-28.24,;10.72,-29.71,;9.2,-30.39,;10.57,-30.36,;11.76,-29.49,;13.3,-30.34,;12.76,-31.81,;12.32,-30.62,;12.77,-33.35,;11.44,-34.12,;11.43,-35.67,;12.77,-36.44,;14.1,-35.67,;15.58,-36.14,;16.49,-34.89,;15.58,-33.64,;14.1,-34.12,;18.02,-34.89,;18.79,-36.22,;20.33,-36.22,;21.1,-34.89,;20.32,-33.55,;18.79,-33.56,;15.64,-37.68,;14.34,-38.5,;14.4,-40.05,;15.77,-40.76,;17.07,-39.94,;18.57,-40.35,;19.42,-39.06,;18.46,-37.85,;17.01,-38.39,)|
CCN1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |THB:10:8:2:4.5,(30.67,-24,;29.35,-24.8,;29.38,-26.34,;28.85,-27.8,;27.32,-28.48,;28.7,-28.45,;29.89,-27.59,;31.43,-28.43,;30.88,-29.9,;30.44,-28.71,;30.89,-31.44,;29.56,-32.21,;29.56,-33.76,;30.89,-34.53,;32.22,-33.76,;33.7,-34.23,;34.61,-32.98,;33.7,-31.73,;32.22,-32.21,;36.14,-32.98,;36.91,-34.31,;38.45,-34.31,;39.22,-32.98,;38.44,-31.64,;36.9,-31.65,;33.76,-35.77,;32.47,-36.59,;32.52,-38.13,;33.89,-38.85,;35.2,-38.03,;36.69,-38.44,;37.54,-37.15,;36.58,-35.93,;35.13,-36.48,)|
CC(C)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |THB:11:9:3:5.6,(-4.36,3.26,;-5.68,2.47,;-7.03,3.22,;-5.65,.93,;-6.19,-.53,;-7.71,-1.21,;-6.34,-1.18,;-5.15,-.32,;-3.61,-1.16,;-4.15,-2.63,;-4.59,-1.45,;-4.15,-4.17,;-5.47,-4.94,;-5.48,-6.49,;-4.14,-7.26,;-2.81,-6.49,;-1.34,-6.96,;-.43,-5.71,;-1.34,-4.46,;-2.81,-4.94,;1.11,-5.71,;1.88,-7.04,;3.41,-7.04,;4.18,-5.71,;3.41,-4.37,;1.87,-4.38,;-1.27,-8.5,;-2.57,-9.32,;-2.51,-10.86,;-1.15,-11.58,;.16,-10.76,;1.66,-11.17,;2.51,-9.88,;1.54,-8.66,;.09,-9.21,)|
CC(=O)CN1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |THB:12:10:4:6.7,(13.66,1.58,;12.31,2.32,;12.28,3.86,;10.99,1.53,;11.02,-.01,;10.48,-1.47,;8.96,-2.16,;10.33,-2.12,;11.53,-1.26,;13.07,-2.1,;12.52,-3.58,;12.08,-2.39,;12.53,-5.11,;11.2,-5.88,;11.2,-7.43,;12.53,-8.2,;13.86,-7.43,;15.34,-7.9,;16.25,-6.65,;15.34,-5.4,;13.86,-5.88,;17.78,-6.65,;18.55,-7.98,;20.09,-7.98,;20.86,-6.65,;20.08,-5.31,;18.54,-5.32,;15.4,-9.44,;14.1,-10.26,;14.16,-11.8,;15.53,-12.52,;16.83,-11.7,;18.33,-12.11,;19.18,-10.82,;18.22,-9.61,;16.77,-10.15,)|
CCOC(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(Cl)c2[nH]ncc12 |THB:13:11:5:7.8,(29.95,2.2,;28.63,1.41,;27.29,2.16,;25.97,1.36,;24.62,2.11,;26,-.18,;25.46,-1.65,;23.94,-2.33,;25.31,-2.29,;26.51,-1.43,;28.04,-2.27,;27.5,-3.75,;27.06,-2.56,;27.51,-5.29,;26.18,-6.06,;26.18,-7.6,;27.51,-8.37,;28.84,-7.6,;30.32,-8.07,;31.23,-6.82,;30.31,-5.57,;28.84,-6.05,;32.76,-6.82,;33.53,-8.16,;35.07,-8.16,;35.84,-6.82,;35.06,-5.48,;33.52,-5.49,;30.38,-9.61,;29.08,-10.43,;29.14,-11.97,;30.5,-12.69,;30.56,-14.23,;31.81,-11.87,;33.31,-12.28,;34.16,-10.99,;33.2,-9.78,;31.74,-10.32,)|
CCN1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(Cl)c2[nH]ncc12 |THB:10:8:2:4.5,(-4.54,-15.7,;-5.86,-16.5,;-5.83,-18.03,;-6.37,-19.5,;-7.89,-20.18,;-6.52,-20.15,;-5.33,-19.28,;-3.79,-20.13,;-4.33,-21.6,;-4.77,-20.41,;-4.33,-23.14,;-5.65,-23.91,;-5.66,-25.45,;-4.32,-26.22,;-2.99,-25.45,;-1.52,-25.93,;-.6,-24.68,;-1.52,-23.42,;-2.99,-23.9,;.93,-24.68,;1.7,-26.01,;3.23,-26.01,;4.01,-24.68,;3.23,-23.34,;1.69,-23.35,;-1.45,-27.47,;-2.75,-28.29,;-2.69,-29.83,;-1.33,-30.55,;-1.27,-32.09,;-.02,-29.73,;1.48,-30.14,;2.33,-28.84,;1.36,-27.63,;-.09,-28.18,)|
CCOC(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(F)c2[nH]ncc12 |THB:13:11:5:7.8,(15.45,-16.9,;14.13,-17.7,;12.78,-16.95,;11.46,-17.75,;10.11,-17,;11.49,-19.29,;10.96,-20.75,;9.44,-21.43,;10.81,-21.4,;12,-20.54,;13.54,-21.38,;13,-22.85,;12.55,-21.67,;13,-24.39,;11.67,-25.16,;11.67,-26.71,;13,-27.48,;14.34,-26.71,;15.81,-27.18,;16.72,-25.93,;15.81,-24.68,;14.34,-25.16,;18.26,-25.93,;19.02,-27.26,;20.56,-27.26,;21.33,-25.93,;20.55,-24.59,;19.02,-24.6,;15.88,-28.72,;14.58,-29.54,;14.64,-31.08,;16,-31.8,;16.06,-33.34,;17.31,-30.98,;18.8,-31.39,;19.66,-30.1,;18.69,-28.88,;17.24,-29.43,)|
Fc1ccc(-c2c(nn3c(ccnc23)C2CC3CCC(C2)N3)-c2ccncc2)c2cn[nH]c12 |TLB:9:14:21:17.18,(31.91,-31.64,;31.85,-30.1,;30.48,-29.38,;30.43,-27.84,;31.72,-27.02,;31.66,-25.48,;32.57,-24.24,;31.66,-22.98,;30.18,-23.46,;28.85,-22.7,;27.52,-23.47,;27.52,-25.01,;28.85,-25.78,;30.18,-25.01,;28.84,-21.16,;28.4,-19.97,;26.81,-19.06,;25.29,-19.74,;26.66,-19.7,;27.85,-18.84,;29.39,-19.69,;27.34,-17.59,;34.1,-24.23,;34.87,-25.57,;36.41,-25.57,;37.18,-24.23,;36.4,-22.9,;34.86,-22.9,;33.09,-27.73,;34.54,-27.19,;35.5,-28.4,;34.65,-29.69,;33.16,-29.28,)|
CCOC(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(c2[nH]ncc12)C(F)(F)F |THB:13:11:5:7.8,(.29,-34.91,;-1.03,-35.7,;-2.38,-34.96,;-3.7,-35.75,;-5.05,-35.01,;-3.67,-37.29,;-4.2,-38.76,;-5.73,-39.44,;-4.35,-39.41,;-3.16,-38.54,;-1.62,-39.39,;-2.16,-40.86,;-2.61,-39.67,;-2.16,-42.4,;-3.49,-43.17,;-3.49,-44.72,;-2.15,-45.49,;-.82,-44.72,;.65,-45.19,;1.56,-43.94,;.65,-42.69,;-.82,-43.17,;3.1,-43.94,;3.87,-45.28,;5.41,-45.28,;6.18,-43.94,;5.4,-42.6,;3.86,-42.61,;.72,-46.73,;-.58,-47.55,;-.52,-49.1,;.84,-49.81,;2.15,-48.99,;3.65,-49.4,;4.5,-48.11,;3.53,-46.9,;2.08,-47.44,;.9,-51.35,;-.4,-52.17,;2.26,-52.07,;.89,-52.89,)|
CCN1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(c2[nH]ncc12)C(F)(F)F |THB:10:8:2:4.5,(12.5,-34.61,;11.19,-35.41,;11.21,-36.95,;10.68,-38.41,;9.16,-39.09,;10.53,-39.06,;11.72,-38.2,;13.26,-39.04,;12.72,-40.51,;12.27,-39.33,;12.72,-42.05,;11.39,-42.82,;11.39,-44.37,;12.72,-45.14,;14.06,-44.37,;15.53,-44.84,;16.44,-43.59,;15.53,-42.34,;14.06,-42.82,;17.97,-43.59,;18.74,-44.92,;20.28,-44.92,;21.05,-43.59,;20.27,-42.25,;18.74,-42.26,;15.6,-46.38,;14.3,-47.2,;14.36,-48.74,;15.72,-49.46,;17.03,-48.64,;18.52,-49.05,;19.38,-47.76,;18.41,-46.54,;16.96,-47.09,;15.78,-51,;14.48,-51.82,;17.14,-51.72,;15.76,-52.72,)|
CCOC(=O)N1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(C)c2[nH]ncc12 |THB:13:11:5:7.8,(-1.88,2.01,;-3.2,1.22,;-4.55,1.96,;-5.86,1.17,;-7.21,1.91,;-5.83,-.37,;-6.37,-1.84,;-7.89,-2.52,;-6.52,-2.48,;-5.33,-1.62,;-3.79,-2.47,;-4.33,-3.94,;-4.77,-2.75,;-4.33,-5.48,;-5.65,-6.25,;-5.66,-7.79,;-4.32,-8.56,;-2.99,-7.79,;-1.52,-8.27,;-.6,-7.02,;-1.52,-5.76,;-2.99,-6.24,;.93,-7.01,;1.7,-8.35,;3.23,-8.35,;4.01,-7.02,;3.23,-5.68,;1.69,-5.68,;-1.45,-9.8,;-2.75,-10.63,;-2.69,-12.17,;-1.33,-12.89,;-1.27,-14.42,;-.02,-12.06,;1.48,-12.48,;2.33,-11.18,;1.36,-9.97,;-.09,-10.51,)|
CCN1C2CCC1CC(C2)c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(C)c2[nH]ncc12 |THB:10:8:2:4.5,(10.62,1.13,;9.3,.33,;9.33,-1.21,;8.8,-2.67,;7.28,-3.35,;8.65,-3.32,;9.84,-2.45,;11.38,-3.3,;10.84,-4.77,;10.39,-3.58,;10.84,-6.31,;9.51,-7.08,;9.51,-8.63,;10.84,-9.4,;12.18,-8.63,;13.65,-9.1,;14.56,-7.85,;13.65,-6.6,;12.17,-7.07,;16.09,-7.85,;16.86,-9.18,;18.4,-9.18,;19.17,-7.85,;18.39,-6.51,;16.86,-6.52,;13.72,-10.64,;12.42,-11.46,;12.48,-13,;13.84,-13.72,;13.9,-15.26,;15.15,-12.9,;16.64,-13.31,;17.5,-12.01,;16.53,-10.8,;15.08,-11.35,)|
CCOC(=O)N1C2CCC1CC(C2)c1c(C)cnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |THB:13:11:5:7.8,(5.99,.06,;4.67,-.73,;3.32,.01,;2,-.78,;.65,-.04,;2.03,-2.32,;1.5,-3.79,;-.02,-4.47,;1.35,-4.44,;2.54,-3.57,;4.08,-4.42,;3.54,-5.89,;3.09,-4.7,;3.54,-7.43,;2.21,-8.2,;.88,-7.43,;2.21,-9.74,;3.54,-10.51,;4.88,-9.74,;6.35,-10.22,;7.26,-8.97,;6.35,-7.71,;4.88,-8.19,;8.79,-8.97,;9.56,-10.3,;11.1,-10.3,;11.87,-8.97,;11.09,-7.63,;9.56,-7.64,;6.42,-11.76,;5.12,-12.58,;5.18,-14.12,;6.54,-14.84,;7.85,-14.02,;9.34,-14.43,;10.2,-13.13,;9.23,-11.92,;7.78,-12.47,)|
COC(=O)C1CC2N(C)C1Cc1cnc3c(c(nn3c21)-c1ccncc1)-c1ccc(Cl)c(O)c1 |TLB:12:11:7:4.5,THB:18:19:7:4.5|
CN1C2Cc3cnc4c(c(nn4c3C1CC2CO)-c1ccncc1)-c1ccc(Cl)c(O)c1 |TLB:11:12:1:15.14,THB:5:4:1:15.14|
CN1C2Cc3cnc4c(c(nn4c3C1CC2S(=O)(=O)c1ccccc1)-c1ccncc1)-c1ccc(Cl)c(O)c1 |TLB:11:12:1:15.14,THB:5:4:1:15.14|
Fc1c(NC(=O)c2cccc(OC(F)(F)F)c2)cc(Oc2cccc3[nH]c(=O)[nH]c23)c(F)c1F
CC(C)(C)c1cc(NC(=O)c2cccc(Oc3cccc4[nH]c(=O)[nH]c34)c2)n(n1)-c1ccccc1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Oc3cccc4[nH]c(=O)[nH]c34)c2)n(n1)-c1ccccc1
[H][C@]12CN(c3ccc(c(C)c3)-c3ccnc4c(c(nn34)-c3ccncc3)-c3cccc(O)c3)[C@]([H])(CN1)C2 |r|
CN1C2CCC1CN(C2)c1ccc(cc1)-c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(Cl)c(O)c1 |TLB:0:1:3.4:8.7.6|
[H][C@]12CN(c3ccc(c(F)c3)-c3ccnc4c(c(nn34)-c3ccncc3)-c3cccc(O)c3)[C@]([H])(CN1C)C2 |r|
[H][C@]12CN(c3ccc(c(C)c3)-c3ccnc4c(c(nn34)-c3ccncc3)-c3ccc(F)c(O)c3)[C@]([H])(CN1C)C2 |r|
[H][C@]12CN(c3ccc(c(C)c3)-c3ccnc4c(c(nn34)-c3ccncc3)-c3cccc(O)c3)[C@]([H])(CN1C)C2 |r|
[H][C@]12CN(c3ccc(c(F)c3)-c3ccnc4c(c(nn34)-c3ccncc3)-c3cccc(O)c3)[C@]([H])(CN1)C2 |r|
[H][C@]12CN(c3ccc(c(Cl)c3)-c3ccnc4c(c(nn34)-c3ccncc3)-c3cccc(O)c3)[C@]([H])(CN1)C2 |r|
[H][C@]12CN(c3ccc(cc3)-c3ccnc4c(c(nn34)-c3ccncc3)-c3ccc(F)c(O)c3)[C@]([H])(CN1)C2 |r|
[H][C@]12CN(c3ccc(c(Cl)c3)-c3ccnc4c(c(nn34)-c3ccncc3)-c3cccc(O)c3)[C@]([H])(CN1C)C2 |r|
[H][C@]12CN(c3ccc(cc3)-c3ccnc4c(c(nn34)-c3ccncc3)-c3ccc(F)c(O)c3)[C@]([H])(CN1C)C2 |r|
CN1C2CCC1CN(C2)c1ccc(cc1)-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc(O)c1 |TLB:0:1:3.4:8.7.6|
COc1cccc(c1)-c1c(nn2c(ccnc12)-c1ccc(cc1)N1CC2CCC(C1)N2C)-c1ccncc1 |TLB:31:30:26.27:24.23.29|
COc1cc(ccc1Cl)-c1c(nn2c(ccnc12)-c1ccc(cc1)N1CC2CCC(C1)N2C)-c1ccncc1 |TLB:32:31:27.28:25.24.30|
Oc1cccc(c1)-c1c(nn2c(ccnc12)-c1ccc(NCC23CCN(CC2)CC3)cc1)-c1ccncc1
Oc1cccc(c1)-c1c(nn2c(ccnc12)-c1ccc(N[C@@H]2CN3CCC2CC3)cc1)-c1ccncc1 |r,wD:21.23,(12.65,-48.79,;13.43,-47.46,;14.97,-47.48,;15.75,-46.14,;14.99,-44.81,;13.46,-44.8,;12.67,-46.12,;12.72,-43.45,;13.63,-42.21,;12.73,-40.96,;11.26,-41.43,;9.93,-40.66,;8.59,-41.43,;8.59,-42.96,;9.92,-43.74,;11.26,-42.97,;9.93,-39.13,;8.6,-38.36,;8.6,-36.81,;9.93,-36.04,;9.95,-34.5,;11.3,-33.75,;11.33,-32.2,;12.68,-31.45,;14,-32.25,;13.98,-33.79,;12.63,-34.54,;13.14,-33.23,;11.85,-32.65,;11.27,-36.81,;11.28,-38.36,;15.17,-42.22,;15.93,-43.56,;17.47,-43.57,;18.25,-42.24,;17.47,-40.9,;15.94,-40.9,)|
Oc1cccc(c1)-c1c(nn2c(ccnc12)-c1ccc(N[C@H]2CN3CCC2CC3)cc1)-c1ccncc1 |r,wU:21.23,(27.09,-49.36,;27.87,-48.04,;29.41,-48.05,;30.19,-46.72,;29.43,-45.38,;27.9,-45.37,;27.11,-46.7,;27.16,-44.03,;28.07,-42.79,;27.17,-41.54,;25.71,-42,;24.37,-41.24,;23.04,-42,;23.03,-43.54,;24.36,-44.31,;25.7,-43.54,;24.37,-39.7,;23.04,-38.93,;23.05,-37.39,;24.37,-36.62,;24.39,-35.08,;25.74,-34.33,;25.77,-32.78,;27.12,-32.02,;28.45,-32.82,;28.42,-34.36,;27.07,-35.12,;27.58,-33.8,;26.3,-33.23,;25.71,-37.38,;25.72,-38.93,;29.61,-42.8,;30.37,-44.14,;31.91,-44.15,;32.69,-42.82,;31.92,-41.48,;30.38,-41.47,)|
Oc1cccc(c1)-c1c(nn2c(ccnc12)-c1ccc(cc1)N1C[C@@H]2C[C@H]1CN2)-c1ccncc1 |r|
CN1C[C@@H]2C[C@H]1CN2c1ccc(cc1)-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc(O)c1 |r|
CCN1C[C@@H]2C[C@H]1CN2c1ccc(cc1)-c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(F)c(O)c1 |r|
CC(=O)N1C[C@@H]2C[C@H]1CN2c1ccc(cc1)-c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(F)c(O)c1 |r|
COc1cccc(c1)-c1c(nn2c(ccnc12)-c1ccc(cc1)N1C[C@@H]2C[C@H]1CN2)-c1ccncc1 |r|
COc1cccc(c1)-c1c(nn2c(ccnc12)-c1ccc(cc1F)N1C[C@@H]2C[C@H]1CN2)-c1ccncc1 |r|
COc1cc(ccc1F)-c1c(nn2c(ccnc12)-c1ccc(cc1)N1C[C@@H]2C[C@H]1CN2)-c1ccncc1 |r|
COc1cccc(c1)-c1c(nn2c(ccnc12)-c1ccc(cc1)N1C[C@@H]2C[C@H]1CN2C)-c1ccncc1 |r|
COc1cc(ccc1F)-c1c(nn2c(ccnc12)-c1ccc(cc1)N1C[C@@H]2C[C@H]1CN2C)-c1ccncc1 |r|
COc1cc(ccc1F)-c1c(nn2c(ccnc12)-c1ccc(cc1C)N1C[C@@H]2C[C@H]1CN2C)-c1ccncc1 |r|
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2c(cnn12)C#CCCCN1CCOCC1
CN1CCN(CCCC#Cc2cnn3c(ccnc23)-c2cccc(NC(=O)c3cccc(c3)C(F)(F)F)c2)CC1
CN(C)c1ccc(cc1)-c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
CN(C)S(=O)(=O)c1ccc(cc1)-c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
NC(=O)c1cccc(c1)-c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
COCCOCC(=O)Nc1ccc(cc1)-c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
CN(C)CC(=O)Nc1ccc(cc1)-c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
CN(C)CC(=O)Nc1cccc(c1)-c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
CN(C)CCc1ccccc1-c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
CN(C)CCc1cccc(c1)-c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
CN(C)CCc1ccc(cc1)-c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
CN(C)Cc1ccccc1-c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
CN(C)Cc1cccc(c1)-c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
CN(C)Cc1ccc(cc1)-c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2c(cnn12)-c1ccc(CN2CCCC2)cc1
CN1CCN(Cc2ccc(cc2)-c2cnn3c(ccnc23)-c2cccc(NC(=O)c3cccc(c3)C(F)(F)F)c2)CC1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2c(cnn12)-c1cccnc1
Nc1ccc(cn1)-c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
CN(C)CCNc1ccc(cn1)-c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
CN1CCN(CC1)c1ccc(cn1)-c1cnn2c(ccnc12)-c1cccc(NC(=O)c2cccc(c2)C(F)(F)F)c1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2c(cnn12)-c1cnc(nc1)N1CCOCC1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2c(cnn12)-c1cn[nH]c1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2c(cnn12)-c1cnn(CCN2CCCC2)c1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2c(cnn12)-c1ccoc1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2c(cnn12)-c1coc(CN2CCCC2)c1
CCN1CCN(Cc2cc(co2)-c2cnn3c(ccnc23)-c2cccc(NC(=O)c3cccc(c3)C(F)(F)F)c2)CC1
Fc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1ccnc2c(cnn12)-c1cn[nH]c1
FC(F)(F)c1cccc(c1)C(=O)Nc1ccc(Cl)c(c1)-c1ccnc2c(cnn12)-c1cn[nH]c1
COc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1-c1ccnc2c(cnn12)-c1cn[nH]c1
CN1CCN(CC1)c1ccc(cn1)-c1cnn2c(ccnc12)-c1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1F
Cc1c(C#N)c(N)[nH]c2c(C#N)c(=C)c(=Cc3ccc(O)cc3)c12 |w:15.15|
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2cc(nn12)-c1cccc(c1)C(F)(F)F
COc1ccc(cc1)-c1cc2nccc(-c3cccc(NC(=O)c4cccc(c4)C(F)(F)F)c3)n2n1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2cc(nn12)-c1cccs1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2cc(nn12)-c1c[nH]cn1
Cn1cncc1-c1cc2nccc(-c3cccc(NC(=O)c4cccc(c4)C(F)(F)F)c3)n2n1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2cc(nn12)-c1ccncc1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2cc(nn12)-c1cccnc1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2cc(nn12)N1CCNCC1
CN1CCN(CC1)c1cc2nccc(-c3cccc(NC(=O)c4cccc(c4)C(F)(F)F)c3)n2n1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2cc(nn12)N1CCOCC1
Clc1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2cc(nn12)-c1ccncc1
COc1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2cc(nn12)-c1ccncc1
Clc1ccc(cc1Cl)C(=O)Nc1cccc(c1)-c1ccnc2cc(nn12)-c1ccncc1
FC(F)(F)c1cc(ccc1Cl)C(=O)Nc1cccc(c1)-c1ccnc2cc(nn12)-c1ccncc1
FC(F)(F)c1cccc(NC(=O)Nc2cccc(c2)-c2ccnc3cc(nn23)-c2ccncc2)c1
FC(F)(F)c1cc(NC(=O)Nc2cccc(c2)-c2ccnc3cc(nn23)-c2ccncc2)ccc1Cl
CN(C)CCNc1cc(ccn1)-c1cc2nccc(-c3cccc(NC(=O)c4cccc(c4)C(F)(F)F)c3)n2n1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2cc(nn12)-c1ccnc(NCCN2CCOCC2)c1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2cc(nn12)-c1ccnc(NCCCN2CCOCC2)c1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2cc(nn12)-c1ccnc(NCCN2CCCC2)c1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2cc(nn12)-c1ccnc(NCCCN2CCCC2)c1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2cc(nn12)-c1ccnc(NCCCN2CCCC2=O)c1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ccnc2cc(nn12)-c1ccnc(NCCCc2ncc[nH]2)c1
OC1CCN(CCNc2cc(ccn2)-c2cc3nccc(-c4cccc(NC(=O)c5cccc(c5)C(F)(F)F)c4)n3n2)CC1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ncnc2cc(sc12)-c1cccnc1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ncnc2cc(sc12)-c1ccncc1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ncnc2sc(cc12)-c1cccnc1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1ncnc2sc(cc12)-c1ccncc1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1c(cnc2cc(sc12)-c1cccnc1)C#N
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1c(cnc2cc(sc12)-c1ccncc1)C#N
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1c(cnc2sc(cc12)-c1cccnc1)C#N
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(c1)-c1c(cnc2sc(cc12)-c1ccncc1)C#N
CNC(=O)c1cc(Oc2ccc(NC(=O)c3ccc(CN4CCN(C)CC4)cc3)cc2)ccn1
CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(OCCN3CCOCC3)c3ccccc23)CC1
Cc1ccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)cc1Nc1nccc(n1)-c1cccnc1
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(C)c(Nc2nccc(n2)-c2cccnc2)c1)C(C)(C)C
CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3cc(nn3-c3ccc(C)cc3)C(C)(C)C)cc2)ccn1
CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3ccc(CN4CCN(C)CC4)cc3)cc2)ccn1
FC(F)(F)c1cc(NC(=O)Nc2ccc(OCCN3CCOCC3)cc2)ccc1Cl
C[C@@]12[C@](C[C@@H](O1)n3c4ccccc4c5c3c6n2c7ccccc7c6c8c5C(=O)NC8)(CO)O
C[C@@]12[C@@H]([C@@H](C[C@@H](O1)n3c4ccccc4c5c3c6n2c7ccccc7c6c8c5C(=O)NC8)N(C)C(=O)c9ccccc9)OC
CC(C)(C)c1cc(NC(=O)Nc2ccc(cc2)-c2cn3c(n2)sc2cc(OCCN4CCOCC4)ccc32)no1
COc1cc2c(ncnc2cc1OCCCN1CCCCC1)N1CCN(CC1)C(=O)Nc1ccc(OC(C)C)cc1
CO[C@@H]1[C@@H](C[C@H]2O[C@]1(C)n1c3ccccc3c3c4[C@H](O)NC(=O)c4c4c5ccccc5n2c4c13)N(C)C(=O)c1ccccc1 |r|
CCN(CC)CCNC(=O)c1c(C)[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c1C
Cn1ccc2c1c(ncn2)Oc3ccc(c(c3)F)NC(=O)Nc4cccc(c4)C(F)(F)F
CC(C)(C)c1cc(NC(=O)Nc2cccc(Cl)c2Cl)n(n1)-c1cccc(CC(N)=O)c1
[H][C@]12CN(c3cc(F)c(c(F)c3)-c3ccnc4c(c(nn34)-c3ccncc3)-c3cccc4[nH]ncc34)[C@]([H])(CN1C1CCC1)C2 |r,wU:36.42,1.0,(4.86,-17.8,;3.77,-18.9,;3.78,-20.44,;2.44,-21.22,;2.45,-22.75,;1.12,-23.53,;1.13,-25.07,;-.2,-25.85,;2.46,-25.83,;3.8,-25.06,;5.13,-25.82,;3.79,-23.52,;2.47,-27.37,;1.14,-28.14,;1.14,-29.68,;2.47,-30.45,;3.81,-29.68,;5.28,-30.16,;6.19,-28.9,;5.28,-27.65,;3.81,-28.13,;7.73,-28.9,;8.5,-30.24,;10.04,-30.24,;10.81,-28.9,;10.03,-27.56,;8.5,-27.57,;5.76,-31.62,;7.26,-31.94,;7.74,-33.4,;6.71,-34.55,;5.2,-34.23,;3.95,-35.13,;2.71,-34.22,;3.2,-32.76,;4.73,-32.77,;1.11,-20.46,;-.44,-20.45,;1.1,-18.92,;2.43,-18.13,;2.43,-16.59,;3.51,-15.5,;2.42,-14.42,;1.33,-15.51,;2.19,-19.36,)|
[H][C@]12CN(c3ccc(c(F)c3)-c3ccnc4c(c(nn34)-c3ccncc3)-c3ccc(F)c4[nH]ncc34)[C@]([H])(CN1C)C2 |r,wU:36.42,1.0,(5.96,-12.33,;4.87,-13.43,;4.88,-14.97,;3.54,-15.75,;3.55,-17.28,;4.89,-18.05,;4.89,-19.59,;3.56,-20.36,;2.23,-19.6,;.9,-20.38,;2.22,-18.06,;3.57,-21.9,;2.24,-22.67,;2.24,-24.21,;3.57,-24.98,;4.91,-24.21,;6.38,-24.69,;7.29,-23.44,;6.38,-22.18,;4.91,-22.66,;8.83,-23.43,;9.6,-24.77,;11.14,-24.77,;11.91,-23.43,;11.13,-22.09,;9.6,-22.1,;6.86,-26.15,;8.36,-26.47,;8.84,-27.93,;7.81,-29.09,;8.29,-30.55,;6.3,-28.76,;5.05,-29.66,;3.81,-28.75,;4.3,-27.29,;5.83,-27.3,;2.21,-14.99,;.66,-14.98,;2.2,-13.45,;3.53,-12.67,;3.53,-11.12,;3.29,-13.89,)|
[H][C@]12CN(c3cc(F)c(c(F)c3)-c3ccnc4c(c(nn34)-c3ccncc3)-c3cccc4[nH]ncc34)[C@]([H])(CN1CC(C)C)C2 |r,wU:36.42,1.0,(21.41,.41,;20.33,-.69,;20.34,-2.23,;19,-3.01,;19.01,-4.54,;17.67,-5.32,;17.69,-6.86,;16.35,-7.64,;19.02,-7.62,;20.35,-6.85,;21.69,-7.62,;20.35,-5.31,;19.03,-9.16,;17.7,-9.93,;17.7,-11.48,;19.03,-12.25,;20.37,-11.47,;21.84,-11.95,;22.75,-10.7,;21.84,-9.44,;20.36,-9.92,;24.29,-10.69,;25.06,-12.03,;26.6,-12.03,;27.37,-10.7,;26.59,-9.36,;25.06,-9.36,;22.32,-13.42,;23.82,-13.73,;24.3,-15.19,;23.27,-16.35,;21.76,-16.03,;20.51,-16.92,;19.27,-16.01,;19.75,-14.56,;21.29,-14.56,;17.67,-2.25,;16.12,-2.25,;17.66,-.71,;18.99,.07,;18.98,1.62,;20.31,2.39,;20.31,3.93,;21.65,1.63,;18.75,-1.15,)|
[H][C@]12CN(c3ccc(c(C)c3)-c3ccnc4c(c(nn34)-c3ccncc3)-c3ccc(F)c4[nH]ncc34)[C@]([H])(CN1C)C2 |r,wU:36.42,1.0,(-6.99,-8.62,;-8.07,-9.72,;-8.07,-11.26,;-9.4,-12.03,;-9.39,-13.57,;-8.05,-14.33,;-8.05,-15.87,;-9.39,-16.65,;-10.72,-15.89,;-12.05,-16.66,;-10.73,-14.35,;-9.38,-18.18,;-10.71,-18.95,;-10.71,-20.5,;-9.37,-21.27,;-8.04,-20.5,;-6.56,-20.98,;-5.65,-19.72,;-6.56,-18.47,;-8.04,-18.95,;-4.11,-19.72,;-3.34,-21.06,;-1.8,-21.06,;-1.03,-19.72,;-1.81,-18.38,;-3.35,-18.39,;-6.09,-22.44,;-4.59,-22.76,;-4.11,-24.22,;-5.14,-25.37,;-4.66,-26.84,;-6.65,-25.05,;-7.89,-25.95,;-9.13,-25.04,;-8.65,-23.58,;-7.11,-23.59,;-10.73,-11.27,;-12.28,-11.27,;-10.75,-9.74,;-9.41,-8.95,;-9.42,-7.41,;-9.65,-10.17,)|
[H][C@]12CN(c3cc(F)c(c(F)c3)-c3ccnc4c(c(nn34)-c3ccncc3)-c3cccc4[nH]ncc34)[C@]([H])(CN1C(C)C)C2 |r,wU:36.42,1.0,(9.92,3.92,;8.84,2.82,;8.84,1.28,;7.51,.5,;7.52,-1.03,;6.18,-1.82,;6.19,-3.35,;4.86,-4.13,;7.52,-4.11,;8.86,-3.34,;10.2,-4.11,;8.85,-1.8,;7.53,-5.65,;6.2,-6.42,;6.2,-7.97,;7.54,-8.74,;8.87,-7.97,;10.35,-8.44,;11.26,-7.19,;10.34,-5.93,;8.87,-6.41,;12.79,-7.19,;13.56,-8.52,;15.1,-8.52,;15.88,-7.19,;15.1,-5.85,;13.56,-5.85,;10.82,-9.91,;12.32,-10.22,;12.8,-11.68,;11.77,-12.84,;10.26,-12.52,;9.02,-13.41,;7.78,-12.51,;8.26,-11.05,;9.79,-11.06,;6.17,1.26,;4.63,1.26,;6.16,2.8,;7.5,3.58,;7.49,5.12,;8.82,5.9,;6.15,5.89,;7.26,2.36,)|
[H][C@]12CN(c3ccc(c(Br)c3)-c3ccnc4c(c(nn34)-c3ccncc3)-c3cccc4[nH]ncc34)[C@]([H])(CN1C)C2 |r,wU:35.41,1.0,(-8.28,-15.09,;-9.36,-16.19,;-9.36,-17.73,;-10.69,-18.5,;-10.68,-20.03,;-9.35,-20.8,;-9.34,-22.34,;-10.68,-23.12,;-12.01,-22.36,;-13.34,-23.13,;-12.03,-20.82,;-10.67,-24.65,;-12.01,-25.42,;-12.01,-26.97,;-10.67,-27.74,;-9.33,-26.97,;-7.86,-27.45,;-6.94,-26.19,;-7.86,-24.94,;-9.33,-25.42,;-5.41,-26.19,;-4.64,-27.53,;-3.1,-27.53,;-2.33,-26.19,;-3.1,-24.85,;-4.64,-24.86,;-7.38,-28.91,;-5.88,-29.23,;-5.4,-30.69,;-6.43,-31.84,;-7.94,-31.52,;-9.19,-32.42,;-10.42,-31.51,;-9.94,-30.05,;-8.41,-30.06,;-12.04,-17.74,;-13.58,-17.74,;-12.05,-16.21,;-10.7,-15.42,;-10.71,-13.88,;-10.94,-16.64,)|
[H][C@]12CN(c3cc(F)c(c(F)c3)-c3ccnc4c(c(nn34)-c3ccncc3)-c3cccc4[nH]ncc34)[C@]([H])(CN1CC)C2 |r,wU:36.42,1.0,(-2.84,3.86,;-3.92,2.75,;-3.91,1.21,;-5.25,.44,;-5.24,-1.09,;-6.58,-1.88,;-6.57,-3.41,;-7.9,-4.19,;-5.23,-4.18,;-3.9,-3.4,;-2.56,-4.17,;-3.9,-1.86,;-5.22,-5.71,;-6.55,-6.48,;-6.55,-8.03,;-5.22,-8.8,;-3.89,-8.03,;-2.41,-8.51,;-1.5,-7.25,;-2.41,-6,;-3.89,-6.48,;.04,-7.25,;.81,-8.59,;2.35,-8.59,;3.12,-7.25,;2.34,-5.91,;.8,-5.92,;-1.93,-9.97,;-.43,-10.29,;.05,-11.75,;-.98,-12.9,;-2.49,-12.58,;-3.74,-13.48,;-4.98,-12.57,;-4.5,-11.11,;-2.96,-11.12,;-6.58,1.2,;-8.13,1.2,;-6.59,2.74,;-5.26,3.52,;-5.27,5.06,;-3.94,5.84,;-5.5,2.3,)|
[H][C@]12CN(c3ccc(c(Cl)c3)-c3ccnc4c(c(nn34)-c3ccncc3)-c3cccc4[nH]ncc34)[C@]([H])(CN1C)C2 |r,wU:35.41,1.0,(38.98,4.96,;37.9,3.86,;37.9,2.32,;36.57,1.54,;36.58,.01,;37.92,-.76,;37.92,-2.3,;36.58,-3.07,;35.25,-2.31,;33.92,-3.09,;35.24,-.77,;36.59,-4.61,;35.26,-5.38,;35.26,-6.93,;36.6,-7.7,;37.93,-6.92,;39.41,-7.4,;40.32,-6.15,;39.41,-4.89,;37.93,-5.37,;41.86,-6.14,;42.63,-7.48,;44.17,-7.48,;44.94,-6.15,;44.16,-4.81,;42.62,-4.81,;39.88,-8.87,;41.39,-9.18,;41.87,-10.64,;40.83,-11.8,;39.32,-11.48,;38.08,-12.37,;36.84,-11.46,;37.32,-10.01,;38.86,-10.01,;35.24,2.3,;33.69,2.3,;35.22,3.84,;36.56,4.62,;36.55,6.17,;36.32,3.4,)|
CN1C[C@@H]2C[C@H]1CN2c1cccc(c1)-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wU:3.3,5.4,(10.64,4.14,;11.97,3.38,;11.98,1.83,;13.31,1.06,;12.91,2.55,;13.31,4.15,;14.64,3.37,;14.64,1.83,;15.98,1.07,;17.32,1.85,;18.66,1.09,;18.66,-.45,;17.32,-1.23,;16,-.47,;17.33,-2.76,;16,-3.53,;16,-5.08,;17.34,-5.85,;18.67,-5.08,;20.15,-5.56,;21.06,-4.3,;20.15,-3.05,;18.67,-3.53,;22.6,-4.3,;23.37,-5.64,;24.91,-5.64,;25.68,-4.3,;24.9,-2.96,;23.36,-2.97,;20.62,-7.02,;22.12,-7.34,;22.61,-8.8,;21.57,-9.95,;20.06,-9.63,;18.82,-10.53,;17.58,-9.62,;18.06,-8.16,;19.6,-8.17,)|
C(N1C[C@@H]2C[C@H]1CO2)c1ccc(cc1)-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wU:5.4,3.3,(16.44,2.06,;17.77,2.83,;19.1,2.05,;20.44,2.8,;19.27,3.96,;17.78,4.37,;19.12,5.13,;20.46,4.35,;16.45,.52,;17.78,-.25,;17.79,-1.79,;16.45,-2.57,;15.12,-1.8,;15.11,-.27,;16.46,-4.1,;15.13,-4.87,;15.13,-6.42,;16.47,-7.19,;17.8,-6.42,;19.27,-6.9,;20.19,-5.64,;19.27,-4.39,;17.8,-4.87,;21.72,-5.64,;22.49,-6.98,;24.03,-6.98,;24.81,-5.64,;24.03,-4.3,;22.49,-4.31,;19.75,-8.36,;21.25,-8.68,;21.73,-10.14,;20.7,-11.29,;19.19,-10.97,;17.95,-11.87,;16.71,-10.96,;17.19,-9.5,;18.72,-9.51,)|
CN1C[C@@H]2C[C@H]1CN2c1c(F)cc(cc1F)-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wU:3.3,5.4,(36.72,-34.69,;36.73,-36.23,;35.39,-37.02,;35.41,-38.56,;36.49,-37.45,;38.07,-37,;38.08,-38.54,;36.74,-39.31,;36.75,-40.85,;38.09,-41.62,;39.42,-40.84,;38.09,-43.16,;36.76,-43.93,;35.42,-43.17,;35.41,-41.63,;34.07,-40.87,;36.77,-45.47,;35.44,-46.24,;35.43,-47.78,;36.77,-48.55,;38.1,-47.78,;39.58,-48.26,;40.49,-47,;39.58,-45.75,;38.1,-46.23,;42.03,-47,;42.8,-48.34,;44.34,-48.34,;45.11,-47,;44.33,-45.66,;42.79,-45.67,;40.05,-49.72,;41.56,-50.04,;42.04,-51.5,;41,-52.65,;39.5,-52.33,;38.25,-53.23,;37.01,-52.32,;37.49,-50.86,;39.03,-50.87,)|
CN(C)c1cc(ccc1-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12)N1C[C@@H]2C[C@H]1CN2C |r,wU:37.42,35.41,(6.85,-21.06,;8.19,-21.82,;8.2,-23.36,;9.52,-21.04,;9.51,-19.5,;10.85,-18.72,;12.19,-19.49,;12.19,-21.03,;10.85,-21.8,;10.86,-23.34,;9.53,-24.11,;9.53,-25.66,;10.87,-26.43,;12.2,-25.66,;13.68,-26.13,;14.59,-24.88,;13.68,-23.62,;12.2,-24.1,;16.13,-24.88,;16.9,-26.21,;18.44,-26.21,;19.21,-24.88,;18.43,-23.54,;16.89,-23.54,;14.15,-27.6,;15.65,-27.91,;16.14,-29.37,;15.1,-30.53,;13.59,-30.21,;12.35,-31.1,;11.11,-30.2,;11.59,-28.74,;13.13,-28.75,;10.84,-17.19,;12.17,-16.41,;12.17,-14.87,;10.59,-15.33,;9.51,-16.43,;9.49,-14.89,;10.83,-14.11,;10.82,-12.57,)|
C(N1C[C@@H]2C[C@@H]1CN2)c1ccc(cc1)-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wU:3.3,wD:5.4,(3.49,-2.92,;4.83,-2.15,;6.16,-2.93,;7.49,-2.16,;6.31,-1.02,;4.82,-.62,;6.15,.15,;7.71,-.52,;3.5,-4.46,;4.84,-5.23,;4.84,-6.77,;3.5,-7.54,;2.18,-6.79,;2.16,-5.24,;3.52,-9.08,;2.19,-9.85,;2.18,-11.4,;3.52,-12.17,;4.85,-11.39,;6.33,-11.87,;7.24,-10.61,;6.33,-9.37,;4.85,-9.84,;8.77,-10.62,;9.54,-11.95,;11.08,-11.95,;11.85,-10.62,;11.08,-9.27,;9.53,-9.28,;6.8,-13.34,;8.3,-13.65,;8.79,-15.11,;7.75,-16.26,;6.24,-15.94,;4.99,-16.84,;3.75,-15.93,;4.23,-14.46,;5.77,-14.47,)|
CN1C[C@@H]2C[C@H]1CN2c1ccc(cc1C(F)(F)F)-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wU:3.3,5.4,(34.33,-13.96,;34.34,-15.5,;33,-16.29,;33.02,-17.82,;34.1,-16.72,;35.68,-16.27,;35.69,-17.81,;34.35,-18.58,;34.36,-20.12,;35.7,-20.88,;35.7,-22.42,;34.37,-23.2,;33.03,-22.44,;33.02,-20.9,;31.68,-20.14,;31.67,-18.59,;30.35,-20.92,;30.34,-19.36,;34.38,-24.73,;33.05,-25.5,;33.04,-27.05,;34.38,-27.82,;35.71,-27.05,;37.19,-27.53,;38.1,-26.27,;37.19,-25.02,;35.71,-25.5,;39.64,-26.27,;40.41,-27.61,;41.95,-27.61,;42.72,-26.27,;41.94,-24.93,;40.4,-24.94,;37.66,-28.99,;39.17,-29.31,;39.65,-30.77,;38.61,-31.92,;37.11,-31.6,;35.86,-32.5,;34.62,-31.59,;35.1,-30.13,;36.64,-30.14,)|
CN1C[C@@H]2C[C@H]1CN2c1ccc(cc1F)-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wU:3.3,5.4,(22.69,-13.24,;22.7,-14.78,;21.37,-15.56,;21.38,-17.1,;22.46,-16,;24.04,-15.54,;24.05,-17.08,;22.71,-17.86,;22.72,-19.39,;24.06,-20.16,;24.06,-21.7,;22.73,-22.47,;21.39,-21.71,;21.38,-20.17,;20.04,-19.41,;22.74,-24.01,;21.41,-24.78,;21.4,-26.33,;22.74,-27.1,;24.07,-26.32,;25.55,-26.8,;26.46,-25.55,;25.55,-24.29,;24.07,-24.77,;28,-25.54,;28.77,-26.88,;30.31,-26.88,;31.08,-25.55,;30.3,-24.21,;28.76,-24.21,;26.02,-28.27,;27.53,-28.58,;28.01,-30.04,;26.98,-31.2,;25.47,-30.88,;24.22,-31.77,;22.98,-30.87,;23.46,-29.41,;25,-29.41,)|
CN1C[C@@H]2C[C@H]1CC2c1cc(F)ccc1-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wU:3.3,5.4,(-2.11,-1.77,;-.77,-1,;.57,-1.77,;1.9,-.99,;.41,-.6,;-.78,.54,;.56,1.32,;1.89,.54,;3.22,1.31,;3.2,2.85,;4.53,3.63,;4.53,5.17,;5.87,2.86,;5.88,1.32,;4.54,.55,;4.55,-.99,;3.22,-1.76,;3.22,-3.31,;4.55,-4.08,;5.89,-3.3,;7.36,-3.78,;8.27,-2.53,;7.36,-1.27,;5.89,-1.75,;9.81,-2.52,;10.58,-3.86,;12.12,-3.86,;12.89,-2.53,;12.12,-1.19,;10.58,-1.19,;7.84,-5.25,;9.34,-5.56,;9.82,-7.02,;8.79,-8.18,;7.28,-7.86,;6.03,-8.75,;4.8,-7.84,;5.28,-6.39,;6.81,-6.39,)|
CN1C[C@@H]2C[C@H]1CN2c1ccc(-c2ccnc3c(c(nn23)-c2ccncc2)-c2cccc3[nH]ncc23)c(c1)C(F)(F)F |r,wU:3.3,5.4,(-.03,-12.85,;-.02,-14.39,;-1.36,-15.18,;-1.35,-16.72,;-.26,-15.62,;1.32,-15.16,;1.32,-16.7,;-.01,-17.47,;-0,-19.01,;1.33,-19.78,;1.34,-21.32,;0,-22.09,;.01,-23.62,;-1.32,-24.4,;-1.32,-25.94,;.02,-26.71,;1.35,-25.94,;2.82,-26.42,;3.74,-25.16,;2.82,-23.91,;1.35,-24.39,;5.27,-25.16,;6.04,-26.5,;7.58,-26.5,;8.35,-25.16,;7.58,-23.82,;6.04,-23.83,;3.3,-27.88,;4.8,-28.2,;5.28,-29.66,;4.25,-30.81,;2.74,-30.49,;1.49,-31.39,;.26,-30.48,;.74,-29.02,;2.27,-29.03,;-1.33,-21.33,;-1.34,-19.79,;-2.66,-22.11,;-4,-21.34,;-2.65,-23.65,;-4.16,-22.5,)|
Fc1cc(CN2C[C@@H]3C[C@H]2CO3)ccc1-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wU:9.8,7.7,(25.62,-2.98,;26.95,-2.2,;26.94,-.66,;28.28,.12,;28.27,1.66,;29.6,2.44,;30.93,1.65,;32.27,2.41,;31.1,3.56,;29.61,3.97,;30.95,4.73,;32.29,3.95,;29.61,-.65,;29.62,-2.19,;28.28,-2.96,;28.29,-4.5,;26.96,-5.27,;26.96,-6.82,;28.3,-7.59,;29.63,-6.81,;31.1,-7.29,;32.02,-6.04,;31.1,-4.78,;29.63,-5.26,;33.55,-6.03,;34.32,-7.37,;35.86,-7.37,;36.64,-6.04,;35.86,-4.7,;34.32,-4.7,;31.58,-8.76,;33.08,-9.07,;33.56,-10.53,;32.53,-11.69,;31.02,-11.37,;29.78,-12.26,;28.54,-11.35,;29.02,-9.9,;30.55,-9.9,)|
CN1C[C@@H]2C[C@H]1CN2c1ccc(cc1)-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wU:3.3,5.4,(-9.85,7.04,;-9.84,5.5,;-11.18,4.71,;-11.16,3.17,;-10.08,4.27,;-8.5,4.73,;-8.5,3.19,;-9.83,2.41,;-9.82,.88,;-8.48,.11,;-8.48,-1.43,;-9.82,-2.2,;-11.15,-1.44,;-11.16,.1,;-9.81,-3.74,;-11.14,-4.51,;-11.14,-6.05,;-9.8,-6.82,;-8.47,-6.05,;-6.99,-6.53,;-6.08,-5.28,;-6.99,-4.02,;-8.47,-4.5,;-4.54,-5.27,;-3.77,-6.61,;-2.23,-6.61,;-1.46,-5.27,;-2.24,-3.93,;-3.78,-3.94,;-6.52,-7.99,;-5.02,-8.31,;-4.53,-9.77,;-5.57,-10.93,;-7.08,-10.6,;-8.32,-11.5,;-9.56,-10.59,;-9.08,-9.13,;-7.54,-9.14,)|
CN1C[C@@H]2C[C@H]1CN2c1ccc(-c2ccnc3c(c(nn23)-c2ccncc2)-c2cccc3[nH]ncc23)c2ccccc12 |r,wU:3.3,5.4,(15.66,4.33,;15.67,2.79,;14.34,2,;14.34,.46,;15.43,1.56,;17.01,2.02,;17.01,.48,;15.68,-.3,;15.69,-1.83,;17.03,-2.6,;17.03,-4.14,;15.69,-4.91,;15.7,-6.45,;14.37,-7.22,;14.38,-8.76,;15.71,-9.54,;17.04,-8.76,;18.52,-9.24,;19.43,-7.99,;18.52,-6.73,;17.04,-7.21,;20.97,-7.98,;21.74,-9.32,;23.28,-9.32,;24.05,-7.98,;23.27,-6.65,;21.73,-6.65,;18.99,-10.7,;20.5,-11.02,;20.98,-12.48,;19.94,-13.64,;18.43,-13.32,;17.19,-14.21,;15.95,-13.3,;16.43,-11.85,;17.97,-11.85,;14.37,-4.15,;13.06,-4.93,;11.72,-4.19,;11.69,-2.65,;13.01,-1.87,;14.35,-2.61,)|
Fc1cc(CN2C3COCC2COC3)ccc1-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |(13.8,-22.79,;15.13,-22.01,;15.12,-20.47,;16.4,-19.69,;16.45,-18.15,;17.8,-17.42,;18.65,-16.43,;18.72,-14.73,;20.2,-14.56,;19.38,-15.46,;19.29,-17.23,;21.11,-17.39,;21.5,-15.89,;20.4,-16.61,;17.79,-20.46,;17.8,-22,;16.46,-22.77,;16.47,-24.31,;15.14,-25.08,;15.14,-26.62,;16.47,-27.39,;17.81,-26.62,;19.28,-27.1,;20.19,-25.84,;19.28,-24.59,;17.81,-25.07,;21.73,-25.84,;22.5,-27.18,;24.04,-27.18,;24.81,-25.84,;24.03,-24.5,;22.5,-24.51,;19.76,-28.56,;21.26,-28.88,;21.74,-30.34,;20.71,-31.49,;19.2,-31.17,;17.95,-32.07,;16.71,-31.16,;17.2,-29.7,;18.73,-29.71,)|
CN1C[C@@H]2CC[C@H]1CN2c1ccc(cc1)-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wD:6.6,3.9,(-6.71,3.85,;-6.7,2.31,;-8.04,1.53,;-8.03,-.01,;-7.27,1.33,;-6.47,.46,;-5.36,1.55,;-5.36,.01,;-6.69,-.77,;-6.69,-2.3,;-5.35,-3.07,;-5.34,-4.61,;-6.68,-5.39,;-8.01,-4.62,;-8.02,-3.09,;-6.67,-6.92,;-8,-7.69,;-8,-9.24,;-6.67,-10.01,;-5.33,-9.24,;-3.86,-9.72,;-2.94,-8.46,;-3.86,-7.21,;-5.33,-7.69,;-1.41,-8.46,;-.64,-9.8,;.9,-9.8,;1.68,-8.46,;.9,-7.12,;-.64,-7.13,;-3.38,-11.18,;-1.88,-11.5,;-1.4,-12.96,;-2.43,-14.11,;-3.94,-13.79,;-5.19,-14.69,;-6.42,-13.78,;-5.94,-12.32,;-4.41,-12.33,)|
CN1C[C@@H]2C[C@H]1CN2c1ccc(c(F)c1F)-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wU:3.3,5.4,(1.07,-33.28,;1.07,-34.82,;-.26,-35.61,;-.25,-37.15,;.83,-36.05,;2.41,-35.59,;2.42,-37.13,;1.08,-37.91,;1.09,-39.44,;2.43,-40.21,;2.44,-41.75,;1.1,-42.52,;-.23,-41.76,;-1.56,-42.54,;-.24,-40.22,;-1.58,-39.46,;1.11,-44.06,;-.22,-44.83,;-.22,-46.37,;1.11,-47.14,;2.45,-46.37,;3.92,-46.85,;4.83,-45.6,;3.92,-44.34,;2.45,-44.82,;6.37,-45.59,;7.14,-46.93,;8.68,-46.93,;9.45,-45.59,;8.67,-44.25,;7.14,-44.26,;4.4,-48.31,;5.9,-48.63,;6.38,-50.09,;5.35,-51.25,;3.84,-50.92,;2.59,-51.82,;1.35,-50.91,;1.84,-49.45,;3.37,-49.46,)|
Fc1cc(CN2C[C@H]3C[C@@H]2CO3)ccc1-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wD:9.8,7.7,(-13.19,-23.21,;-11.86,-22.44,;-11.88,-20.9,;-10.53,-20.12,;-10.54,-18.57,;-9.21,-17.8,;-7.88,-18.58,;-6.54,-17.83,;-7.7,-16.67,;-9.19,-16.26,;-7.86,-15.5,;-6.52,-16.28,;-9.19,-20.88,;-9.19,-22.42,;-10.52,-23.2,;-10.51,-24.73,;-11.85,-25.5,;-11.85,-27.05,;-10.51,-27.82,;-9.18,-27.05,;-7.7,-27.53,;-6.79,-26.27,;-7.7,-25.02,;-9.18,-25.5,;-5.25,-26.27,;-4.48,-27.61,;-2.94,-27.61,;-2.17,-26.27,;-2.95,-24.93,;-4.49,-24.94,;-7.23,-28.99,;-5.72,-29.31,;-5.24,-30.77,;-6.27,-31.92,;-7.78,-31.6,;-9.03,-32.5,;-10.27,-31.59,;-9.79,-30.13,;-8.25,-30.14,)|
CN1C[C@@H]2C[C@H]1CN2c1ccc(c(C)c1)-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wU:3.3,5.4,(14.11,6.43,;14.12,4.89,;12.79,4.1,;12.8,2.57,;13.88,3.67,;15.46,4.12,;15.47,2.58,;14.13,1.81,;14.14,.27,;15.48,-.49,;15.48,-2.03,;14.15,-2.81,;12.81,-2.05,;11.48,-2.82,;12.8,-.51,;14.16,-4.34,;12.83,-5.11,;12.83,-6.66,;14.16,-7.43,;15.49,-6.66,;16.97,-7.14,;17.88,-5.88,;16.97,-4.63,;15.49,-5.11,;19.42,-5.88,;20.19,-7.22,;21.73,-7.22,;22.5,-5.88,;21.72,-4.54,;20.18,-4.55,;17.45,-8.6,;18.95,-8.92,;19.43,-10.38,;18.4,-11.53,;16.89,-11.21,;15.64,-12.11,;14.4,-11.2,;14.88,-9.74,;16.42,-9.75,)|
CN1C[C@@H]2C[C@H]1CN2c1ccc(cc1)-c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(F)c2[nH]ncc12 |r,wU:3.3,5.4,(28.5,5.92,;28.51,4.38,;27.17,3.6,;27.18,2.06,;28.27,3.16,;29.85,3.62,;29.85,2.08,;28.52,1.3,;28.53,-.23,;29.86,-1,;29.87,-2.54,;28.53,-3.31,;27.2,-2.55,;27.19,-1.01,;28.54,-4.85,;27.21,-5.62,;27.21,-7.17,;28.55,-7.94,;29.88,-7.16,;31.36,-7.64,;32.27,-6.39,;31.35,-5.13,;29.88,-5.61,;33.8,-6.38,;34.57,-7.72,;36.11,-7.72,;36.89,-6.39,;36.11,-5.05,;34.57,-5.05,;31.83,-9.11,;33.33,-9.42,;33.81,-10.88,;32.78,-12.04,;33.26,-13.5,;31.27,-11.72,;30.03,-12.61,;28.79,-11.71,;29.27,-10.25,;30.8,-10.25,)|
CN1C[C@@H]2CC[C@H]1CN2c1ccc(c(F)c1)-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wD:6.6,3.9,(4.83,5.26,;4.84,3.71,;3.5,2.93,;3.51,1.39,;4.27,2.73,;5.07,1.86,;6.17,2.95,;6.18,1.41,;4.85,.63,;4.85,-.9,;6.19,-1.67,;6.2,-3.21,;4.86,-3.98,;3.53,-3.22,;2.2,-4,;3.52,-1.68,;4.87,-5.52,;3.54,-6.29,;3.54,-7.84,;4.87,-8.61,;6.21,-7.84,;7.68,-8.31,;8.59,-7.06,;7.68,-5.8,;6.21,-6.28,;10.13,-7.06,;10.9,-8.39,;12.44,-8.39,;13.22,-7.06,;12.44,-5.72,;10.9,-5.72,;8.16,-9.78,;9.66,-10.09,;10.14,-11.55,;9.11,-12.71,;7.6,-12.39,;6.35,-13.29,;5.12,-12.38,;5.6,-10.92,;7.13,-10.93,)|
CN1C[C@@H]2C[C@H]1CN2c1cc(F)c(cc1F)-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wU:3.3,5.4,(12.11,-32.8,;12.12,-34.34,;10.78,-35.12,;10.8,-36.66,;11.88,-35.56,;13.46,-35.1,;13.47,-36.64,;12.13,-37.42,;12.14,-38.95,;10.8,-39.73,;10.81,-41.27,;9.48,-42.05,;12.15,-42.03,;13.48,-41.26,;13.48,-39.72,;14.81,-38.95,;12.16,-43.57,;10.83,-44.34,;10.82,-45.89,;12.16,-46.66,;13.49,-45.88,;14.97,-46.36,;15.88,-45.11,;14.97,-43.85,;13.49,-44.33,;17.42,-45.1,;18.19,-46.44,;19.73,-46.44,;20.5,-45.11,;19.72,-43.77,;18.18,-43.77,;15.44,-47.83,;16.95,-48.14,;17.43,-49.6,;16.39,-50.76,;14.88,-50.44,;13.64,-51.33,;12.4,-50.42,;12.88,-48.97,;14.42,-48.97,)|
CN1C[C@@H]2C[C@H]1CN2c1c(F)c(F)c(c(F)c1F)-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wU:3.3,5.4,(-7.9,5.85,;-7.89,4.3,;-9.22,3.52,;-9.21,1.98,;-8.13,3.08,;-6.55,3.54,;-6.54,2,;-7.88,1.22,;-7.87,-.31,;-6.53,-1.08,;-5.2,-.3,;-6.53,-2.62,;-5.19,-3.39,;-7.86,-3.39,;-9.19,-2.63,;-10.52,-3.41,;-9.2,-1.09,;-10.54,-.33,;-7.85,-4.93,;-9.18,-5.7,;-9.18,-7.24,;-7.85,-8.02,;-6.51,-7.24,;-5.04,-7.72,;-4.13,-6.47,;-5.04,-5.21,;-6.51,-5.69,;-2.59,-6.46,;-1.82,-7.8,;-.28,-7.8,;.49,-6.46,;-.29,-5.13,;-1.82,-5.13,;-4.56,-9.19,;-3.06,-9.5,;-2.58,-10.96,;-3.61,-12.12,;-5.12,-11.8,;-6.37,-12.69,;-7.61,-11.78,;-7.13,-10.33,;-5.59,-10.33,)|
CN1C[C@@H]2C[C@H]1CN2c1ccc(c(F)c1)-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wU:3.3,5.4,(25.08,5.67,;25.09,4.13,;23.75,3.34,;23.77,1.8,;24.85,2.9,;26.43,3.36,;26.44,1.82,;25.1,1.04,;25.11,-.49,;26.45,-1.26,;26.45,-2.8,;25.12,-3.57,;23.78,-2.81,;22.45,-3.59,;23.77,-1.27,;25.13,-5.11,;23.8,-5.88,;23.79,-7.42,;25.13,-8.19,;26.46,-7.42,;27.94,-7.9,;28.85,-6.65,;27.94,-5.39,;26.46,-5.87,;30.39,-6.64,;31.16,-7.98,;32.7,-7.98,;33.47,-6.64,;32.69,-5.3,;31.15,-5.31,;28.41,-9.36,;29.92,-9.68,;30.4,-11.14,;29.36,-12.29,;27.85,-11.97,;26.61,-12.87,;25.37,-11.96,;25.85,-10.5,;27.39,-10.51,)|
CN1C[C@@H]2C[C@H]1CN2c1cc(F)c(c(F)c1)-c1ccnc2c(c(nn12)-c1ccncc1)-c1cccc2[nH]ncc12 |r,wU:3.3,5.4,(24.13,-33.61,;24.13,-35.15,;22.8,-35.94,;22.81,-37.47,;23.89,-36.37,;25.47,-35.92,;25.48,-37.46,;24.14,-38.23,;24.15,-39.77,;22.82,-40.55,;22.83,-42.09,;21.5,-42.86,;24.16,-42.85,;25.5,-42.07,;26.83,-42.84,;25.49,-40.53,;24.17,-44.38,;22.84,-45.15,;22.84,-46.7,;24.17,-47.47,;25.51,-46.7,;26.98,-47.18,;27.89,-45.92,;26.98,-44.67,;25.51,-45.15,;29.43,-45.92,;30.2,-47.26,;31.74,-47.26,;32.51,-45.92,;31.73,-44.58,;30.2,-44.59,;27.46,-48.64,;28.96,-48.96,;29.44,-50.42,;28.41,-51.57,;26.9,-51.25,;25.65,-52.15,;24.41,-51.24,;24.9,-49.78,;26.43,-49.79,)|
CN1C[C@@H]2C[C@H]1CN2c1cc(F)c(c(F)c1)-c1ccnc2c(c(nn12)-c1ccncc1)-c1ccc(F)c2[nH]ncc12 |r,wU:3.3,5.4,(16.85,-11.72,;16.86,-13.27,;15.53,-14.05,;15.54,-15.59,;16.62,-14.49,;18.2,-14.03,;18.21,-15.57,;16.87,-16.35,;16.88,-17.88,;15.54,-18.66,;15.55,-20.2,;14.22,-20.98,;16.89,-20.96,;18.22,-20.19,;19.56,-20.96,;18.22,-18.65,;16.9,-22.5,;15.57,-23.27,;15.57,-24.82,;16.9,-25.59,;18.24,-24.81,;19.71,-25.29,;20.62,-24.04,;19.71,-22.78,;18.23,-23.26,;22.16,-24.03,;22.93,-25.37,;24.47,-25.37,;25.24,-24.04,;24.46,-22.7,;22.92,-22.7,;20.19,-26.76,;21.69,-27.07,;22.17,-28.53,;21.14,-29.69,;21.62,-31.15,;19.63,-29.37,;18.38,-30.26,;17.14,-29.36,;17.62,-27.9,;19.16,-27.9,)|
COc1ccc2cc([nH]c2c1)-c1n[nH]c2cccnc12
c1cc(c(cc1[N+](=O)[O-])Cl)NC(=O)c2cc(ccc2O)Cl
CN(C)Cc1cc(cc(c1)C(F)(F)F)C(=O)N[C@@H]1CCc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1 |r|
CC(C)(N)c1cc(cc(c1)C(F)(F)F)C(=O)N[C@@H]1CCc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1 |r|
Oc1ccccc1C1CC(=NN1C(=O)c1ccc(s1)-c1ccccn1)c1cccnc1 |c:10|
CCc1c[nH]nc1-c1ccc(cc1)-c1cn(C)nc1-c1ccncc1
Cn1cc(c(n1)-c1ccncc1)-c1ccc2-c3n[nH]cc3CCc2c1
Cn1cc(c(n1)-c1ccncc1)-c1ccc2-c3cn[nH]c3CCc2c1
Cn1cc(c(n1)-c1ccncc1)-c1ccc2c(cc3[nH][nH]nc23)c1
Cn1cc(c(n1)-c1ccncc1)-c1ccc(cc1)-c1c[nH]nn1
Cn1cc(c(n1)-c1ccncc1)-c1ccc(cc1)-c1cc[nH]c1
CNC(=O)c1ccc(cc1)-c1cn(C)nc1-c1ccncc1
Cn1cc(c(n1)-c1ccncc1)-c1ccc(cc1)S(N)(=O)=O
Cn1cc(c(n1)-c1ccncc1)-c1cccc2[nH]ncc12
Cn1cc(c(n1)-c1ccncc1)-c1ccc2[nH]ncc2c1
Cn1cc(c(n1)-c1ccncc1)-c1ccc2[nH]ccc2c1
Cn1cc(c(n1)-c1ccncc1)-c1ccc2cc[nH]c2c1
Cn1cc(c(n1)-c1ccncc1)-c1ccc2c(O)cccc2c1
Cn1cc(c(n1)-c1ccncc1)-c1ccc2cc(O)ccc2c1
Cn1cc(N)c(n1)-c1ccncc1
Cn1cc(O)c(n1)-c1ccncc1
C1c2c[nH]nc2-c2ccc(cc12)-c1cn(nc1-c1ccncc1)C1CCNCC1
CN1CCC(CC1)n1cc(c(n1)-c1ccncc1)-c1ccc-2c(Cc3c[nH]nc-23)c1
C1CC2CC(CC1N2)n1cc(c(n1)-c1ccncc1)-c1ccc-2c(Cc3c[nH]nc-23)c1
C1c2c[nH]nc2-c2ccc(cc12)-c1cn(nc1-c1ccncc1)C1CCCNC1
C1c2c[nH]nc2-c2ccc(cc12)-c1cn(nc1-c1ccncc1)C1CCCNCC1
N[C@H]1CC[C@@H](CC1)n1cc(c(n1)-c1ccncc1)-c1ccc-2c(Cc3c[nH]nc-23)c1 |r,wU:4.7,wD:1.0,(6.31,.76,;4.77,.77,;4.01,2.11,;2.46,2.11,;1.7,.78,;2.46,-.56,;3.99,-.56,;.16,.79,;-.74,2.03,;-2.21,1.56,;-2.21,.02,;-.74,-.46,;-3.46,-.88,;-4.79,-.12,;-6.12,-.89,;-6.12,-2.43,;-4.79,-3.2,;-3.45,-2.43,;-3.53,2.33,;-3.52,3.87,;-4.85,4.64,;-6.19,3.88,;-6.19,2.33,;-7.66,1.85,;-8.57,3.1,;-10.04,3.56,;-10.05,5.11,;-8.59,5.6,;-7.67,4.35,;-4.86,1.56,)|
N[C@H]1CC[C@H](CC1)n1cc(c(n1)-c1ccncc1)-c1ccc-2c(Cc3c[nH]nc-23)c1 |r,wD:4.7,1.0,(30.59,1.1,;29.05,1.11,;28.29,2.45,;26.74,2.46,;25.98,1.13,;26.74,-.21,;28.27,-.22,;24.44,1.13,;23.54,2.37,;22.07,1.9,;22.07,.37,;23.54,-.12,;20.82,-.54,;19.49,.23,;18.16,-.54,;18.16,-2.09,;19.49,-2.86,;20.83,-2.09,;20.74,2.68,;20.76,4.21,;19.43,4.99,;18.09,4.22,;18.09,2.67,;16.62,2.19,;15.71,3.44,;14.24,3.91,;14.23,5.45,;15.69,5.94,;16.61,4.69,;19.42,1.91,)|
CNCCn1cc(c(n1)-c1ccncc1)-c1ccc-2c(Cc3c[nH]nc-23)c1
O[C@@H]1CCC[C@@H](C1)n1cc(c(n1)-c1ccncc1)-c1ccc-2c(Cc3c[nH]nc-23)c1 |r|
C1c2c[nH]nc2-c2ccc(cc12)-c1cn(nc1-c1ccncc1)-c1ccccc1
O[C@@H]1CNCC[C@H]1n1cc(c(n1)-c1ccncc1)-c1ccc-2c(Cc3c[nH]nc-23)c1 |r|
C1c2c[nH]nc2-c2ccc(cc12)-c1cn(nc1-c1ccncc1)C1CC2COCC(C1)N2
F[C@@H]1CNCC[C@H]1n1cc(c(n1)-c1ccncc1)-c1ccc-2c(Cc3c[nH]nc-23)c1 |r|
F[C@H]1CNCC[C@H]1n1cc(c(n1)-c1ccncc1)-c1ccc-2c(Cc3c[nH]nc-23)c1 |r|
F[C@H]1CCNC[C@H]1n1cc(c(n1)-c1ccncc1)-c1ccc-2c(Cc3c[nH]nc-23)c1 |r|
F[C@H]1CNCC[C@@H]1n1cc(c(n1)-c1ccncc1)-c1ccc-2c(Cc3c[nH]nc-23)c1 |r|
CNC(=O)c1ncc(C#Cc2cc(ccc2C)C(=O)Nc2ccc(CN3CCN(CCO)CC3)c(c2)C(F)(F)F)n1C
CCOC(=O)c1cccc(Nc2nc(N)nc3nc[nH]c23)c1
NC(=O)c1ccc(Nc2nnc(-c3ccc(O)cc3)c3ccccc23)cc1
Nc1ccccc1Oc1ccc(cc1)-c1nc(N)nc(N)n1
Cc1ccc(\C=C\c2nc(N)nc(n2)-c2ccccc2O)o1
Oc1ccc(cc1)\N=C1/NC(=O)\C(S1)=C\c1c[nH]c2ccccc12
Cc1ccc(CNC(=O)c2c(N)n(-c3cccc(O)c3)c3nc4ccccc4nc23)cc1
CN1CCN(CC1)CC(=O)N(C)c2ccc(cc2)N/C(=C\3/c4ccc(cc4NC3=O)C(=O)OC)/c5ccccc5
CN1CCN(CC1)c1ccc2nc([nH]c2c1)-c1c(N)c2c(F)cccc2[nH]c1=O
CCOc1cc2ncc(C#N)c(Nc3ccc(OCc4ccccn4)c(Cl)c3)c2cc1NC(=O)\C=C\CN(C)C
Cc1cn(cn1)-c1cc(NC(=O)c2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)cc(c1)C(F)(F)F
C[C@@H]1CCN(C[C@@H]1N(C)c1ncnc2[nH]ccc12)C(=O)CC#N |r|
CN1CC[C@@H]([C@H](O)C1)c1c(O)cc(O)c2c1oc(cc2=O)-c1ccccc1Cl |r|
Clc1ccc(Nc2nnc(Cc3ccncc3)c3ccccc23)cc1
COc1cc2c(cc1OCCCN3CCOCC3)c(ncn2)Nc4ccc(c(c4)Cl)F
CN1c2c(cnc(n2)Nc3cccc(c3)SC)C=C(C1=O)c4c(cccc4Cl)Cl
Cc1ccc(F)c(NC(=O)Nc2ccc(cc2)-c2cccc3[nH]nc(N)c23)c1
COc1ccc(c(c1C(=O)c2cnc(nc2N)NC3CCN(CC3)S(=O)(=O)C)F)F
Cc1cnc2c(NCCN)nc3ccc(C)cc3n12
C=CC(=O)Nc1cc2c(cc1OCCCN3CCOCC3)ncnc2Nc4ccc(c(c4)Cl)F
CCN(CCCOc1ccc2c(c1)ncnc2Nc3cc(n[nH]3)CC(=O)Nc4cccc(c4)F)CCO
CC1(C(=O)Nc2c(ccc(n2)Nc3c(cnc(n3)Nc4cc(c(c(c4)OC)OC)OC)F)O1)C
CC(C)(C)c1cnc(o1)CSc2cnc(s2)NC(=O)C3CCNCC3
Cn1cc(cn1)-c1ccc2nnc(Sc3ccc4ncccc4c3)n2n1
Cc1cnc(nc1Nc2cccc(c2)S(=O)(=O)NC(C)(C)C)Nc3ccc(cc3)OCCN4CCCC4
CN(C)C[C@@H]1CCn2cc(C3=C(C(=O)NC3=O)c3cn(CCO1)c1ccccc31)c1ccccc21 |r,t:10|
c1cc(c(c(c1)Cl)C2=C3C=CC(=NN3C=NC2=O)Sc4ccc(cc4F)F)Cl
COc1cc2c(Oc3ccc(NC(=O)C4(CC4)C(=O)NC4=CCC(F)C=C4)cc3F)ccnc2cc1OCCCN1CCOCC1 |c:26,t:21|
C[C@@H](Oc1cc(sc1C(N)=O)-n1cnc2ccc(CN3CCN(C)CC3)cc12)c1ccccc1C(F)(F)F |r|
Cc1ccc(cc1Nc2nc(cs2)c3cccnc3)NC(=O)c4ccc(cc4)CN5CCN(CC5)C
O=C(N1CCNCC1)c1ccc(\C=C\c2n[nH]c3ccccc23)cc1
CN(C)CC(=O)N1CCC(CC1)c1ccc(NC(=O)c2ncc([nH]2)C#N)c(c1)C1=CCCCC1 |t:31|
COc1cc(Oc2ccnc3cc(OC)c(OC)cc23)ccc1NC(=O)NC(C)c1nccs1
CN1CCN(CC1)CCCOc2cc3c(cc2OC)c(c(cn3)C#N)Nc4cc(c(cc4Cl)Cl)OC
CN1CCC(CC1)COc2cc3c(cc2OC)c(ncn3)Nc4ccc(cc4F)Br
CN1CCN(CC1)c1cc(Nc2cc(C)n[nH]2)nc(Sc2ccc(NC(=O)C3CC3)cc2)n1
Cn1cnc2c1cc(c(c2F)Nc3ccc(cc3Cl)Br)C(=O)NOCCO
Nc1nc(N)c2nc(-c3cccc(O)c3)c(nc2n1)-c1cccc(O)c1
CNC(=O)c1ccccc1Sc2ccc3c(c2)[nH]nc3/C=C/c4ccccn4
Fc1ccc(C(=O)NOCC2CC2)c(Nc2ccc(I)cc2Cl)c1F
OC(=O)c1ccc(Nc2ncc3CN=C(c4cc(Cl)ccc4-c3n2)c2c(F)cccc2F)cc1 |c:13|
CN(C)C/C=C/C(=O)Nc1cc2c(cc1O[C@H]3CCOC3)ncnc2Nc4ccc(c(c4)Cl)F
C[C@@H](O)COc1cn2ncnc(Oc3ccc4[nH]c(C)cc4c3F)c2c1C
COc1ccc(cc1)COc2ccc(cc2OC)Cc3cnc(nc3N)N
Clc1cccc(Cl)c1C(=O)Nc1cn[nH]c1C(=O)NC1CCNCC1
CC(C)n1nc(-c2cc3cc(O)ccc3[nH]2)c2c(N)ncnc12
Cc1[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c(C)c1C(=O)NC[C@H](O)CN1CCOCC1
CNC(=O)c1c(F)cccc1Nc1nc(Nc2cc3N(CCc3cc2OC)C(=O)CN(C)C)nc2[nH]ccc12
CC(C)S(=O)(=O)c1ccccc1Nc2c(cnc(n2)Nc3ccc(cc3OC)N4CCC(CC4)N5CCN(CC5)C)Cl
Cc1[nH]c(\C=C2/C(=O)Nc3ccc(cc23)S(=O)(=O)Cc2c(Cl)cccc2Cl)c(C)c1C(=O)N1CCC[C@@H]1CN1CCCC1 |r|
c1c[nH]c2c1c(ncn2)c3cnn(c3)[C@H](CC#N)C4CCCC4
COc1c(Cl)cc2c3ccncc3[nH]c2c1NC(=O)c1cccnc1C
CS(=O)(=O)N1CCN(Cc2cc3nc(nc(N4CCOCC4)c3s2)-c2cccc3[nH]ncc23)CC1
COc1cc2c(Oc3ccc4[nH]c(C)cc4c3F)ncnc2cc1OCCCN1CCCC1
Cn1cc(C2=C(C(=O)NC2=O)c2cn(C3CCN(Cc4ccccn4)CC3)c3ccccc23)c2ccccc12 |t:4|
Cc1n[nH]c2ccc(cc12)-c1cncc(OC[C@@H](N)Cc2ccccc2)c1 |r|
CCn1c(nc2c(ncc(OC[C@H]3CCCNC3)c12)C#CC(C)(C)O)-c1nonc1N |r|
C[C@@H](Oc1cc(cnc1N)-c1cnn(c1)C1CCNCC1)c1c(Cl)ccc(F)c1Cl |r|
CS(=O)(=O)CCNCc1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
CC(C)(CC(=O)NCCn1ccc2c1c(ncn2)Nc3ccc(c(c3)Cl)Oc4cccc(c4)C(F)(F)F)O
NC(=O)c1ccc2[nH]cc(-c3cccc(O)c3)c2c1
Oc1cccc(c1)-c1c[nH]c2cc3C(=O)NC(=O)c3cc12
Oc1cccc(Nc2cc3C(=O)NC(=O)c3cc2Nc2cccc(O)c2)c1
Oc1cccc(Nc2cc3C(=O)NC(=O)c3cc2Nc2ccccc2)c1
Oc1cccc(Nc2cc3c(cc2Nc2ccccc2)c(=O)[nH][nH]c3=O)c1
Oc1cccc(Nc2cc3c(cc2Nc2cccc(O)c2)c(=O)[nH][nH]c3=O)c1
Clc1cccc(c1)C(=O)Nc1cccc(Nc2cc3C(=O)NC(=O)c3cc2Cl)c1
Clc1cc2C(=O)NC(=O)c2cc1Nc1cccc(NC(=O)c2cccc(Br)c2)c1
Clc1cc2C(=O)NC(=O)c2cc1Nc1cccc(NC(=O)c2cccc(I)c2)c1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(Nc2cc3C(=O)NC(=O)c3cc2Cl)c1
FC(F)(F)Oc1cccc(c1)C(=O)Nc1cccc(Nc2cc3C(=O)NC(=O)c3cc2Cl)c1
Clc1cc2C(=O)NC(=O)c2cc1Nc1cccc(NC(=O)c2cccc(c2)C#N)c1
Cn1nc(cc1C(=O)Nc1cccc(Nc2cc3C(=O)NC(=O)c3cc2Cl)c1)C(C)(C)C
Clc1cccc(c1)C(=O)Nc1cccc(Nc2cc3c(cc2Cl)c(=O)[nH][nH]c3=O)c1
Clc1cc2c(cc1Nc1cccc(NC(=O)c3cccc(Br)c3)c1)c(=O)[nH][nH]c2=O
Clc1cc2c(cc1Nc1cccc(NC(=O)c3cccc(I)c3)c1)c(=O)[nH][nH]c2=O
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(Nc2cc3c(cc2Cl)c(=O)[nH][nH]c3=O)c1
FC(F)(F)Oc1cccc(c1)C(=O)Nc1cccc(Nc2cc3c(cc2Cl)c(=O)[nH][nH]c3=O)c1
Clc1cc2c(cc1Nc1cccc(NC(=O)c3cccc(c3)C#N)c1)c(=O)[nH][nH]c2=O
Cn1nc(cc1C(=O)Nc1cccc(Nc2cc3c(cc2Cl)c(=O)[nH][nH]c3=O)c1)C(C)(C)C
COc1cncc(c1)-c1nc(NC(C)(C)CO)nc2sc(C(N)=O)c(N)c12
COc1cncc(c1)-c1nc(N[C@H](C)CO)nc2sc(C(N)=O)c(N)c12 |r|
NC(=O)c1sc2ncnc(-c3cccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)c3)c2c1N
CC(C)(CO)Nc1nc(-c2cccc(NC(=O)Nc3ccc(cc3)C(F)(F)F)c2)c2c(N)c(sc2n1)C(N)=O
CC(C)(CO)Nc1nc(-c2cccc(O)c2F)c2c(N)c(sc2n1)C(N)=O
CC(C)(CO)Nc1nc(-c2cc(O)cc(Cl)c2)c2c(N)c(sc2n1)C(N)=O
NC(=O)c1sc2nc(NC3CC3)nc(-c3cccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)c3)c2c1N
Cc1ccc(NC(=O)Nc2cccc(c2)-c2nc(NC3CC3)nc3sc(C(N)=O)c(N)c23)cc1
NC(=O)c1sc2nc(NC3CC3)nc(-c3cccc(NC(=O)Nc4ccccc4)c3)c2c1N
COc1cncc(c1)-c1nc(NC2CC2)nc2sc(C(N)=O)c(N)c12
NC(=O)c1sc2nc(NC3CC3)nc(-c3cccc(O)c3F)c2c1N
Cc1ccc(cc1O)-c1nc(NC2CC2)nc2sc(C(N)=O)c(N)c12
NC(=O)c1sc2nc(NC3CC3)nc(-c3ccc(Cl)c(O)c3)c2c1N
NC(=O)c1sc2nc(NC3CC3)nc(-c3cc(O)cc(Cl)c3)c2c1N
COc1cccc(c1)-c1nc(NC2CC2)nc2sc(C(N)=O)c(N)c12
NC(=O)c1sc2nc(NC3CC3)nc(-c3ccc(O)cc3)c2c1N
NC(=O)c1sc2nc(NC3CC3)nc(-c3cccc(O)c3)c2c1N
C[C@H](CO)Cc1nc(-c2ccc(Cl)c(Cl)c2)c2c(N)c(sc2n1)C(N)=O |r|
C[C@H](CO)Oc1nc(-c2ccc(Cl)c(Cl)c2)c2c(N)c(sc2n1)C(N)=O |r|
CC(C)(CO)Nc1nc(-c2ccc(Cl)c(Cl)c2)c2c(N)c(sc2n1)C(N)=O
C[C@H](CO)Nc1nc(-c2ccc(Cl)c(Cl)c2)c2c(N)c(sc2n1)C(N)=O |r|
NCCNc1nc(-c2ccc(Cl)c(Cl)c2)c2c(N)c(sc2n1)C(N)=O
NC(=O)c1sc2nc(NCCO)nc(-c3ccc(Cl)c(Cl)c3)c2c1N
NC(=O)c1sc2nc(N)nc(-c3ccc(Cl)c(Cl)c3)c2c1N
NC(=O)c1sc2ncnc(-c3ccc(Cl)c(Cl)c3)c2c1N
NC(=O)c1sc2nc(NC3CC3)nc(-c3ccc(Cl)c(Cl)c3)c2c1N
Cc1ccc(Nc2nncc3c(cccc23)-c2ccc(O)cc2)cc1
NC(=O)COc1ccc(Nc2nncc3c(cccc23)-c2ccc(O)cc2)cc1
COc1ccc(Nc2nncc3c(cccc23)-c2ccc(O)cc2)cc1
Oc1ccc(cc1)-c1cccc2c(Nc3cccc(O)c3)nncc12
NS(=O)(=O)c1ccc(Nc2nncc3c(cccc23)-c2ccc(O)cc2)cc1
NC(=O)Cc1ccc(Nc2nncc3c(cccc23)-c2ccc(O)cc2)cc1
CN(C)C(=O)Cc1ccc(cc1)-c1cccc2c(Nc3cccc(O)c3)nncc12
OC(=O)c1ccc(Nc2ncnc3nc[nH]c23)cc1
Nc1nc(Nc2cccc(O)c2)c2[nH]cnc2n1
Nc1nc(Nc2cccc(Br)c2)c2[nH]cnc2n1
CCC(=O)c1cccc(Nc2nc(N)nc3nc[nH]c23)c1
COc1ccc(Nc2nc(N)nc3nc[nH]c23)cc1OC
Nc1nc(Nc2cccc(F)c2)c2[nH]cnc2n1
Nc1nc(Nc2ccc(F)c(Cl)c2)c2[nH]cnc2n1
COc1cc(Nc2nc(N)nc3nc[nH]c23)cc(OC)c1OC
Nc1nc(Nc2ccc(Cl)c(Cl)c2)c2[nH]cnc2n1
COc1ccc(OC)c(Nc2nc(N)nc3nc[nH]c23)c1
Nc1nc(Nc2cccc(Cl)c2)c2[nH]cnc2n1
Nc1nc(Nc2cccc(c2)C(F)(F)F)c2[nH]cnc2n1
C1COc2cc(Nc3nc(Nc4ccc5OCCOc5c4)c4[nH]cnc4n3)ccc2O1
COc1cc(Nc2nc(N)nc3nc[nH]c23)cc(OC)c1
Nc1nc(Nc2ccccc2O)c2[nH]cnc2n1
CC(=O)Nc1ccc(Nc2ncnc3nc[nH]c23)cc1
Cn1c(Nc2ccc(cc2)C(F)(F)F)nc2ccc(Oc3ccnc(c3)-c3c[nH]c(n3)C(F)(F)F)cc12
CC(C)n1c2CCCC(=O)c2c2C(=O)c3ccccc3-c12
c1c2c-3c(c(c1O)O)OC(=O)c4c3c(c(c(c4)O)O)OC2=O
O=NCc1ccc(cc1)-c1[nH]c(nc1-c1ccncc1)-c1ccccc1
Clc1cc(ccc1CN=O)-c1[nH]c(nc1-c1ccncc1)-c1ccccc1
CC(C)(CNS(C)(=O)=O)c1nc(c([nH]1)-c1ccc(Cl)c(O)c1)-c1ccncc1
CC(C)(C)c1nc(c([nH]1)-c1ccc(F)cc1)-c1ccncc1
c1ccc(cc1)c2[nH]c(c(n2)c3ccncc3)c4cccc(c4)O
Nc1nccc(n1)-c1nc([nH]c1-c1ccc(Cl)c(O)c1)-c1ccccc1
CC(C)(CNC(=O)Nc1ccc(Cl)cc1)c1nc(c([nH]1)-c1ccc(Cl)c(O)c1)-c1ccncc1
Oc1ccc(cc1)-c1[nH]c(nc1-c1ccncc1)-c1ccccc1
Oc1cc(ccc1Cl)-c1[nH]c(nc1-c1ccncc1)-c1cccnc1
Oc1cc(ccc1Cl)-c1[nH]cnc1-c1ccncc1
Oc1cc(ccc1Cl)-c1[nH]c(nc1-c1ccncn1)-c1ccccc1
Oc1cc(ccc1Cl)-c1[nH]c(nc1-c1cccnc1)-c1ccccc1
Oc1cc(ccc1Cl)-c1[nH]c(nc1-c1ccncc1)-c1ccco1
OCc1cccc(c1)-c1[nH]c(nc1-c1ccncc1)-c1ccccc1
OCc1ccc(cc1O)-c1[nH]c(nc1-c1ccncc1)-c1ccccc1
O=NC1CCCc2cc(ccc12)-c1[nH]c(nc1-c1ccncc1)-c1ccccc1
NCc1ccc(cc1)-c1nc(c([nH]1)-c1ccc(Cl)c(O)c1)-c1ccncc1
Oc1cc(ccc1Cl)-c1[nH]c(nc1-c1ccnnc1)-c1ccccc1
CC(C)(CN)c1nc(c([nH]1)-c1ccc(Cl)c(O)c1)-c1ccncc1
OC1CCc2cc(ccc12)-c1[nH]c(nc1-c1ccncc1)-c1ccccc1
CC(C)(C)c1nc(c([nH]1)-c1ccc(Cl)c(O)c1)-c1ccncc1
O=NC1CCc2cc(ccc12)-c1[nH]c(nc1-c1ccncc1)-c1ccccc1
ONC(=N)c1ccc(cc1)-c1[nH]c(nc1-c1ccncc1)-c1ccccc1
Oc1cc(ccc1CN=O)-c1[nH]c(nc1-c1ccncc1)-c1ccccc1
CN(C)CCCNC(=O)c1nc(c([nH]1)-c1ccc(Cl)c(O)c1)-c1ccncc1
COc1cccc(c1)-c1[nH]c(nc1-c1ccncc1)-c1ccccc1
CC(N=O)c1ccc(cc1)-c1[nH]c(nc1-c1ccncc1)-c1ccccc1
Oc1cc(ccc1Cl)-c1[nH]c(nc1-c1ccccc1)-c1ccccc1
OCc1ccc(cc1Cl)-c1[nH]c(nc1-c1ccncc1)-c1ccccc1
OCc1ccc(cc1)-c1[nH]c(nc1-c1ccncc1)-c1ccccc1
Cc1cccc(c1N2c3nc4ccccc4n3-c5c(cnc(n5)Nc6ccc(cc6)N7CCN(CC7)C)C2=O)C
FC(F)(F)c1cc(NC(=O)Nc2cccc(c2)-c2[nH]c(nc2-c2ccnc(NCCN3CCNC3=O)n2)C2CC2)ccc1Cl
Clc1ccc(CS(=O)(=O)Nc2cccc(c2)-c2[nH]c(nc2-c2ccnc(NCCN3CCNC3=O)n2)C2CC2)cc1Cl
NC(=O)c1cccc(Nc2nccc(n2)-c2nc([nH]c2-c2cccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)c2)C2CC2)c1
CNc1nccc(n1)-c1nc([nH]c1-c1cccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c1)C1CC1
Clc1ccc(CC(=O)Nc2cccc(c2)-c2[nH]c(nc2-c2ccnc(NCCN3CCNC3=O)n2)C2CC2)cc1
FC(F)(F)c1nc(c([nH]1)-c1cccc(NC(=O)Cc2ccc(Cl)cc2)c1)-c1ccnc(NCCN2CCNC2=O)n1
CC(C)(C)NC(=O)NCCNc1nccc(n1)-c1nc([nH]c1-c1ccccc1Cl)C1CC1
Clc1ccc(Cl)c(c1)-c1[nH]c(nc1-c1ccnc(NCCN2CCNC2=O)n1)C1CC1
CNc1nccc(n1)-c1nc([nH]c1-c1cccc(NS(=O)(=O)Cc2ccc(Cl)c(Cl)c2)c1)C1CC1
NC(=O)c1cccc(Nc2nccc(n2)-c2nc([nH]c2-c2cccc(NS(=O)(=O)Cc3ccc(Cl)c(Cl)c3)c2)C2CC2)c1
CNc1nccc(n1)-c1nc([nH]c1-c1cccc(NC(=O)Cc2ccc(Cl)cc2)c1)C1CC1
NC(=O)c1cccc(Nc2nccc(n2)-c2nc([nH]c2-c2cccc(NC(=O)Cc3ccc(Cl)cc3)c2)C2CC2)c1
CNc1nccc(n1)-c1nc([nH]c1-c1cccc(NC(=O)Cc2ccc(Cl)cc2)c1)C(F)(F)F
NC(=O)c1cccc(Nc2nccc(n2)-c2nc([nH]c2-c2cccc(NC(=O)Cc3ccc(Cl)cc3)c2)C(F)(F)F)c1
CCn1cc(c(n1)-c1cccc(NC(=S)Nc2ccccc2)c1)-c1ccnc2[nH]ccc12
CCn1cc(c(n1)-c1cccc(NC(=O)Nc2ccccc2)c1)-c1ccnc2[nH]c(cc12)C(O)=O
CCOC(=O)c1cc2c(ccnc2[nH]1)-c1cn(CC)nc1-c1cccc(NC(=O)Nc2ccccc2)c1
CCn1cc(c(n1)-c1cccc(NC(=O)Nc2ccccc2)c1)-c1ccnc2[nH]cc(Br)c12
CCn1cc(c(n1)-c1cccc(NC(=O)Nc2cccc(OC)c2)c1)-c1ccnc2[nH]ccc12
CCn1cc(c(n1)-c1cccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c1)-c1ccnc2[nH]ccc12
CCn1cc(c(n1)-c1cccc(NC(=O)Nc2cc(ccc2F)C(F)(F)F)c1)-c1ccnc2[nH]ccc12
CCn1cc(c(n1)-c1cccc(NC(=O)Nc2cccc(Cl)c2)c1)-c1ccnc2[nH]ccc12
CCn1cc(c(n1)-c1cccc(NC(=O)Nc2ccc(cc2)C(F)(F)F)c1)-c1ccnc2[nH]ccc12
CCn1cc(c(n1)-c1cccc(NC(=O)Nc2c(F)cccc2F)c1)-c1ccnc2[nH]ccc12
CCn1cc(c(n1)-c1cccc(NC(=O)Nc2ccccc2Cl)c1)-c1ccnc2[nH]ccc12
CCn1cc(c(n1)-c1cccc(NC(=O)Nc2ccc(OCc3ccccc3)cc2)c1)-c1ccnc2[nH]ccc12
CCn1cc(c(n1)-c1cccc(NC(=O)NCc2ccccc2)c1)-c1ccnc2[nH]ccc12
CCn1cc(c(n1)-c1cccc(NC(=O)NC2CCCCC2)c1)-c1ccnc2[nH]ccc12
CCn1cc(c(n1)-c1cccc(NC(=O)Nc2ccccc2)c1)-c1ccnc2[nH]ccc12
OC1Nc2ccc(I)cc2C1=Cc1cc(Br)c(O)c(Br)c1
CN(C)c1cccc(c1)C(=O)Nc1ccc(C)c(NC(=O)c2ccc(O)cc2)c1
COCC(=O)NC\C=C\c1ccc2ncnc(Nc3ccc(Oc4ccc(C)nc4)c(C)c3)c2c1
NC(=O)c1ccc(cc1)-c1nc(c([nH]1)-c1ccc2OCOc2c1)-c1ccccn1
CCOc1cc2c(cc1NC(=O)/C=C/CN(C)C)c(c(cn2)C#N)Nc3ccc(c(c3)Cl)F
CC[C@H](CO)Nc1nc(NCc2ccccc2)c2ncn(C(C)C)c2n1 |r|
c1cc(c(c(c1)F)C(=O)n2c(nc(n2)Nc3ccc(cc3)S(=O)(=O)N)N)F
Nc1ncnc2c(csc12)C(=O)Nc1c(Cl)ccc(NS(=O)(=O)CCCF)c1F
CC(C)(N)C(=O)NCCn1ccc2ncnc(Nc3ccc(Oc4cccc5sncc45)c(Cl)c3)c12
CCCNS(=O)(=O)c1ccc2[nH]c3c(nccc3c2c1)C(N)=O
CCN(CC)CCCNS(=O)(=O)c1ccc2[nH]c3c(nccc3c2c1)C(N)=O
NC(=O)c1nccc2c3cc(ccc3[nH]c12)S(=O)(=O)NCCCO
CC(O)CNS(=O)(=O)c1ccc2[nH]c3c(nccc3c2c1)C(N)=O
CN(C)CCCNS(=O)(=O)c1ccc2[nH]c3c(nccc3c2c1)C(N)=O
COC(CNS(=O)(=O)c1ccc2[nH]c3c(nccc3c2c1)C(N)=O)OC
NC(=O)c1nccc2c3cc(ccc3[nH]c12)S(=O)(=O)NCC(O)CO
NC(=O)c1nccc2c3cc(ccc3[nH]c12)S(=O)(=O)NCCO
COCCCNS(=O)(=O)c1ccc2[nH]c3c(nccc3c2c1)C(N)=O
NC(=O)c1nccc2c3cc(ccc3[nH]c12)S(=O)(=O)NC1CC1
NC(=O)c1nccc2c3cc(ccc3[nH]c12)S(=O)(=O)Nc1ccccc1
Cc1ccc(NS(=O)(=O)c2ccc3[nH]c4c(nccc4c3c2)C(N)=O)cc1
NC(=O)c1nccc2c3cc(ccc3[nH]c12)S(=O)(=O)Nc1ccc(F)cc1
NC(=O)c1nccc2c3cc(ccc3[nH]c12)S(=O)(=O)Nc1ccccn1
NC(=O)c1nccc2c3cc(ccc3[nH]c12)S(N)(=O)=O
NS(=O)(=O)c1ccc2[nH]c3cnccc3c2c1
CC(=O)NS(=O)(=O)c1ccc2[nH]c3cnccc3c2c1
NC(=O)c1nccc2c3cc(ccc3[nH]c12)S(=O)(=O)Nc1nccs1
CC(C)(C(=O)NCCn1ccc2ncnc(Nc3ccc(Oc4cccc(Cl)c4)c(Cl)c3)c12)S(C)(=O)=O
Cc1ccc2c(Nc3ccc(Cl)cc3)nccc2c1Nc1ncccc1-c1ncnc2nc[nH]c12
CC(C)(C)NS(=O)(=O)c1cncc(c1)-c1ccn2nc(N)nc2c1
CC(C)(C#N)Oc1cccc(c1Cl)C(=O)Nc2cc(ccc2F)N(C)c3ccc4c(n3)sc(n4)NC(=O)C5CC5
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(Oc2ccc3nccn3n2)c1
CC(C)(C)c1ccc(cc1)C(=O)Nc2cn3cc(ccc3n2)n4ccnc4
COc1cc2CCN=C(c3ccc(Cl)c(Cl)c3)c2cc1Cl |t:7|
COc1cc2CCN=C(c3cccc(Cl)c3)c2cc1Cl |t:7|
c1ccnc(c1)N[C@@H](c2ccco2)c3cc(c4cccnc4c3O)Cl
Oc1c(ccc2cccnc12)C(Nc1cccnc1)c1ccsc1
COc1ccc(cc1)C(N1CCOCC1)c1ccc2cccnc2c1O
Cc1cc(C)c2c(n1)sn(C(=O)c1cccs1)c2=O
Fc1ccc(cc1)C(=O)\C=C\S(=O)(=O)c1ccc(Cl)cc1
COc1cc(cc(Br)c1O)C(Nc1ccccn1)c1cc(Cl)c2cccnc2c1O
Oc1c(Sc2nnc[nH]2)cc(NS(=O)(=O)c2cccs2)c2ccccc12
O=C1C(Sc2nnc[nH]2)=CC(=NS(=O)(=O)c2cccs2)c2ccccc12 |w:11.12,c:9|
Oc1ccc(NS(=O)(=O)c2cccs2)c2ccccc12
Oc1c(Cl)cc(NS(=O)(=O)c2cccs2)c2ccccc12
Oc1c(Br)cc(NS(=O)(=O)c2cccs2)c2ccccc12
Oc1c(Sc2ncc[nH]2)cc(NS(=O)(=O)c2cccs2)c2ccccc12
Oc1c(Sc2ccccn2)cc(NS(=O)(=O)c2cccs2)c2ccccc12
Cn1nnnc1Sc1cc(NS(=O)(=O)c2cccs2)c2ccccc2c1O
Oc1c(Sc2ccccc2)cc(NS(=O)(=O)c2cccs2)c2ccccc12
Oc1c(Sc2cnn[nH]2)cc(NS(=O)(=O)c2cccs2)c2ccccc12
CC(=O)N1CCc2cc(ccc12)S(=O)(=O)Nc1cc(Sc2nnc[nH]2)c(O)c2ccccc12
Oc1c(Sc2nnc[nH]2)cc(NS(=O)(=O)c2ccc(cc2)C(F)(F)F)c2ccccc12
CCCCCCCCS(=O)(=O)Nc1cc(Sc2nnc[nH]2)c(O)c2ccccc12
Oc1c(Sc2nnc[nH]2)cc(NS(=O)(=O)c2c(F)ccc(N(Cc3ccccc3)Cc3ccccc3)c2F)c2ccccc12
Oc1c(Sc2nnc[nH]2)cc(NS(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)c2ccccc12
Oc1ccc(O)n1-c1ccc(F)c(c1F)S(=O)(=O)Nc1cc(Sc2nnc[nH]2)c(O)c2ccccc12 |(36.55,-5.4,;36.24,-6.91,;37.27,-8.05,;36.51,-9.39,;35,-9.07,;33.87,-10.11,;34.83,-7.55,;33.49,-6.78,;32.16,-7.56,;30.83,-6.8,;30.83,-5.27,;29.5,-4.5,;32.16,-4.5,;33.48,-5.26,;34.81,-4.48,;32.16,-2.97,;30.83,-2.21,;30.82,-3.74,;33.48,-2.2,;33.48,-.67,;34.82,.11,;34.81,1.68,;36.14,2.46,;37.48,1.7,;38.88,2.34,;39.92,1.2,;39.16,-.14,;37.65,.17,;33.47,2.44,;33.46,3.97,;32.13,1.67,;30.78,2.43,;29.44,1.66,;29.44,.1,;30.78,-.68,;32.13,.11,)|
Oc1c(Sc2nnc[nH]2)cc(NS(=O)(=O)c2ccc(cc2)-c2ccccc2)c2ccccc12
Oc1c(Sc2nnc[nH]2)cc(NS(=O)(=O)c2ccc3ccccc3c2)c2ccccc12
CCCCCCCCCCS(=O)(=O)Nc1cc(Sc2nnc[nH]2)c(O)c2ccccc12
Nc1ncc(-c2cccnc2)c2scc(-c3cccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)c3)c12
Nc1ncc(-c2cccnc2)c2scc(-c3cccc(NC(=O)Nc4cc(ccc4F)C(F)(F)F)c3)c12
Nc1ncc(-c2cccnc2)c2scc(-c3cccc(NC(=O)Nc4ccc(cc4)C(F)(F)F)c3)c12
Nc1ncc(-c2cccnc2)c2scc(-c3cccc(NC(=O)Nc4ccc(OCc5ccccc5)cc4)c3)c12
Nc1ncc(-c2cccnc2)c2scc(-c3cccc(NC(=O)Nc4c(F)cccc4F)c3)c12
COc1cccc(NC(=O)Nc2cccc(c2)-c2csc3c(cnc(N)c23)-c2cccnc2)c1
Nc1ncc(-c2cccnc2)c2scc(-c3cccc(NC(=O)Nc4ccccc4)c3)c12
Nc1ncc(-c2cccnc2)c2scc(-c3cccc(NC(=O)NCc4ccccc4)c3)c12
Nc1ncc(-c2cccnc2)c2scc(-c3cccc(NC(=O)NC4CCCCC4)c3)c12
Cc1noc(C)c1NC(=O)Nc1cccc(c1)-c1csc2c(cnc(N)c12)-c1cccnc1
Nc1ncc(-c2cccnc2)c2scc(-c3cccc(NC(=O)Cc4cccs4)c3)c12
Nc1ncc(-c2cccnc2)c2scc(-c3cccc(NC(=O)Cc4ccccc4)c3)c12
Nc1ncc(-c2cccnc2)c2scc(-c3cccc(NC(=O)c4cccc(c4)C(F)(F)F)c3)c12
Nc1ncc(-c2cccnc2)c2scc(-c3cccc(NC(=O)c4cc(F)ccc4F)c3)c12
Nc1ncc(-c2cccnc2)c2scc(-c3cccc(NC(=O)c4ccccc4)c3)c12
Nc1ncc(-c2cccnc2)c2scc(-c3cccc(NC(=O)C4CCCCC4)c3)c12
CC(C)(C)NC(=O)Nc1cccc(c1)-c1csc2c(cnc(N)c12)-c1cccnc1
Cn1cccc1C(=O)Nc1cccc(c1)-c1csc2c(cnc(N)c12)-c1cccnc1
Nc1cccc(c1)-c1csc2c(cnc(N)c12)-c1cccnc1
Nc1ncc(-c2cccnc2)c2scc(-c3cccc(NS(=O)(=O)c4ccccc4)c3)c12
COCCNC(=O)c1ccc(Nc2ncc3cc(ccc3n2)-c2ccncc2)cc1
c1cc(c2ccsc2c1)Oc3ccc(cc3Cl)Nc4c5c(ncn4)NCCC(=C5)C(=O)NCCO
Cc1cc(n(n1)C)C(=O)Nc2cccc(c2)Oc3ccc4nc(cn4n3)NC(=O)C5CC5
Fc1cccc(c1)C(=O)Nc1cccc(Oc2ccc3nc(NC(=O)C4CC4)cn3n2)c1
Cc1cc(C(=O)Nc2cccc(Oc3ccc4nc(NC(=O)C5CC5)sc4c3)c2)n(C)n1
Cc1cc(C(=O)Nc2cccc(Oc3ccc4nc(NC(=O)C5CC5)sc4n3)c2)n(C)n1
Cc1cc(C(=O)Nc2cccc(Oc3ccc4nc(NC(=O)C5CC5)cn4c3)c2)n(C)n1
Cc1cc(C(=O)Nc2cccc(Oc3ccc4nc(NC(=O)C5CC5)nn4c3)c2)n(C)n1
Cc1cc(C(=O)Nc2cc(Oc3ccc4nc(NC(=O)C5CC5)nn4c3)ccc2F)n(C)n1
CC(C)(C)NC(c1ccc(Cl)cc1)c1ccc(cc1)-c1cn[nH]c1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(Oc2ccc3nc(NC(=O)C4CCOCC4)cn3n2)c1
O=[#6]1-[#7]-[#6](=S)-[#7]-[#6](=O)\[#6]-1=[#6]/c1ccc(o1)-c1ccc2-[#8]-[#6]-[#8]-c2c1
O\N=C1/CCc2cc(ccc12)-c1cn(nc1-c1ccncc1)C1CCNCC1
CN1CCC(CC1)n1cc(c(n1)-c1ccncc1)-c1ccc2\C(CCc2c1)=N\O
O\N=C1/CCc2cc(ccc12)-c1cn(nc1-c1ccncc1)C1CCOCC1
CCN(CCO)CCCOc1ccc2c(Nc3cccc(NC(=O)Nc4ccc(F)c(Cl)c4)c3)ncnc2c1
CC(NC(=O)c1cccc(c1)-c1ccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)cc1)c1ccccc1
COc1ccc(Oc2cc(C)c(-c3csc(NC(=O)c4ccnc(F)c4)n3)c(C)c2)cc1
CC(C)N1CCN(CC(=O)Nc2cc(Oc3ccc4n(C)c(Nc5cc(ccc5F)C(F)(F)F)nc4c3)ccn2)CC1
CN1CCC(CC1)C(=O)Nc1cc(Oc2ccc3n(C)c(Nc4cccc(c4)C(C)(C)C)nc3c2)ccn1
CC(=O)Nc1cc(Oc2ccc3n(C)c(Nc4ccc(cc4)C(F)(F)F)nc3c2)ccn1
CCc1ccc(Nc2nc3cc(Oc4ccnc(NC(C)=O)c4)ccc3n2C)cc1
CC(=O)Nc1cc(Oc2ccc3n(C)c(Nc4cccc(OC(F)(F)F)c4)nc3c2)ccn1
CC(=O)Nc1cc(Oc2ccc3n(C)c(Nc4cccc(c4)C(C)(C)C)nc3c2)ccn1
CC(C)N1CCC(CC1)C(=O)Nc1cc(Oc2ccc3n(C)c(Nc4cc(ccc4F)C(F)(F)F)nc3c2)ccn1
Cn1c(Nc2cccc(c2)C(C)(C)C)nc2cc(Oc3ccnc(NC(=O)C4CCNCC4)c3)ccc12
CC(=O)Nc1cc(Oc2ccc3n(C)c(Nc4ccc(OC(F)(F)F)cc4)nc3c2)ccn1
CC(=O)Nc1cc(Oc2ccc3n(C)c(Nc4ccc(cc4)C(C)(C)C)nc3c2)ccn1
CC(C)c1cccc(Nc2nc3cc(Oc4ccnc(NC(C)=O)c4)ccc3n2C)c1
CCN1CCN(CC(=O)Nc2cc(Oc3ccc4n(C)c(Nc5cc(ccc5F)C(F)(F)F)nc4c3)ccn2)CC1
CC(C)N1CCC(CC1)C(=O)Nc1cc(Oc2ccc3n(C)c(Nc4cccc(c4)C(C)(C)C)nc3c2)ccn1
CC(=O)Nc1cc(Oc2ccc3n(C)c(Nc4cc(ccc4F)C(F)(F)F)nc3c2)ccn1
CC(C)c1ccc(Nc2nc3cc(Oc4ccnc(NC(C)=O)c4)ccc3n2C)cc1
CC(=O)Nc1cc(Oc2ccc3n(C)c(Nc4cccc(c4)C(F)(F)F)nc3c2)ccn1
CCc1cccc(Nc2nc3cc(Oc4ccnc(NC(C)=O)c4)ccc3n2C)c1
CC(=O)c1ccc(cc1)N2CCN(CC2)C(=O)CN3CC[C@H](C3)C(=O)Nc4ccc(c(c4)Cl)O
Cc1cc(\C=N\NC(=O)Nc2ccc(cc2)-c2nc(N3CCOCC3)c3sccc3n2)cc(C)c1O
FC(F)(F)c1cc(NC(=O)Nc2cccc(Nc3ncccc3-c3ncnc4[nH]cnc34)c2)ccc1Cl
Cc1ccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)cc1Nc1ncccc1-c1ncnc2[nH]cnc12
FC(F)(F)c1cc(NC(=O)c2cccc(Nc3ncccc3-c3ncnc4[nH]cnc34)c2)ccc1Cl
Cc1ccc(cc1Nc1ncccc1-c1ncnc2[nH]cnc12)C(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
Cc1ccc(cc1Nc1ncccc1-c1ncnc2[nH]cnc12)C(=O)Nc1cccc(c1)C(F)(F)F
CC(C)c1cccc(NC(=O)c2ccc(C)c(Nc3ncccc3-c3ncnc4[nH]cnc34)c2)c1
Cc1ccc(cc1Nc1ncccc1-c1ncnc2[nH]cnc12)C(=O)Nc1cccc(c1)C#N
Cc1ccc(cc1Nc1ncccc1-c1ncnc2[nH]cnc12)C(=O)Nc1cccc(F)c1
Cc1cc(NC(=O)c2ccc(C)c(Nc3ncccc3-c3ncnc4[nH]cnc34)c2)ccc1Cl
Cc1ccc(cc1Nc1ncccc1-c1ncnc2[nH]cnc12)C(=O)Nc1cccc(Cl)c1
Cc1ccc(cc1Nc1ncccc1-c1ncnc2[nH]cnc12)C(=O)Nc1ccc(Cl)c(Br)c1
Cc1ccc(cc1Nc1ncccc1-c1ncnc2[nH]cnc12)C(=O)Nc1ccc(cc1)C(F)(F)F
FC(F)(F)c1cc(NC(=O)c2ccc(Cl)c(Nc3ncccc3-c3ncnc4[nH]cnc34)c2)ccc1Cl
FC(F)(F)c1cccc(NC(=O)c2ccc(Cl)c(Nc3ncccc3-c3ncnc4[nH]cnc34)c2)c1
CC(C)c1cccc(NC(=O)c2ccc(Cl)c(Nc3ncccc3-c3ncnc4[nH]cnc34)c2)c1
Clc1ccc(NC(=O)c2ccc(Cl)c(Nc3ncccc3-c3ncnc4[nH]cnc34)c2)cc1Cl
Fc1ccc(cc1Nc1ncccc1-c1ncnc2[nH]cnc12)C(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
FC(F)(F)c1cc(ccc1Cl)C(=O)Nc1cccc(Nc2ncccc2-c2ncnc3[nH]cnc23)c1
Cc1ccc(NC(=O)c2ccc(Cl)c(c2)C(F)(F)F)cc1Nc1ncccc1-c1ncnc2[nH]cnc12
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1Nc1ncccc1-c1ncnc2[nH]cnc12
Cc1ccc(NC(=O)c2cccc(c2)C#N)cc1Nc1ncccc1-c1ncnc2[nH]cnc12
Cc1cc(ccc1Cl)C(=O)Nc1ccc(C)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1
Cc1ccc(NC(=O)c2cccc(Cl)c2)cc1Nc1ncccc1-c1ncnc2[nH]cnc12
COc1cccc(c1)C(=O)Nc1ccc(C)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1
CN(C)c1cccc(c1)C(=O)Nc1ccc(C)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1
CC(C)c1cccc(NC(=O)c2ccc(C)c(Nc3ncccc3-c3ncnc4n(C)cnc34)c2)c1
O=C(Nc1cccc(Nc2ncccc2-c2ncnc3[nH]cnc23)c1)C1CC1
CC(=O)Nc1cc(Nc2ncccc2-c2ncnc3[nH]cnc23)ccc1Cl
C[C@H](O)CNc1nccc(n1)-n1ccnc1Cc1cccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c1 |r|
CCN(CC)CCCNc1nc(nc2ccsc12)-c1ccc(NC(=O)Nc2ccc(Cl)cc2)cc1
COc1ccc(cc1)C(=O)Nc1ccc(C)c(c1)C(=O)Nc1ccc(nc1)-c1ncc[nH]1
FC(F)(F)c1cc(ccc1Cl)C(=O)Nc1ccc(Cl)c(c1)C(=O)Nc1ccc(nc1)-c1ncc[nH]1
COc1cccc(c1)C(=O)Nc1ccc(C)c(c1)C(=O)Nc1ccc(nc1)-c1ncc[nH]1
FC(F)(F)c1cc(NC(=O)c2ccc(Cl)c(c2)C(=O)Nc2ccc(nc2)-c2ncc[nH]2)ccc1Cl
CNc1ncc2ccc(Oc3c(C)ccc(C(=O)c4c(-c5ccccc5)n(C)n(-c5ccccc5)c4=O)c3N)cc2n1
Cn1cc(-c2ccc3N(CC(=O)c4cc(F)cc(c4)C(F)(F)F)CCc3c2)c2c(N)ncnc12
CNc1ncc2cc(ccc2n1)-c1c(C)ccc(C(=O)Nc2ccc(OC)c(c2)C(F)(F)F)c1N
COc1cc2nccc(Oc3ccc(NC(=O)c4c(-c5ccccc5)n(C)n(-c5ccccc5)c4=O)nc3)c2cc1OC
CNc1ncc2ccc(Oc3cc(ccc3C)C(=O)c3c(-c4ccccc4)n(C)n(-c4ccccc4)c3=O)cc2n1
CNc1ncc2ccc(Oc3cc(ccc3N)C(=O)c3c(-c4ccccc4)n(C)n(-c4ccccc4)c3=O)cc2n1
CNc1ncc2ccc(Oc3cc(ccc3Cl)C(=O)c3c(-c4ccccc4)n(C)n(-c4ccccc4)c3=O)cc2n1
CNc1ncc2c(F)cc(Oc3c(C)ccc(C(=O)c4c(-c5ccccc5)n(C)n(-c5ccccc5)c4=O)c3N)cc2n1
CNc1ncc2c(Cl)cc(Oc3c(C)ccc(C(=O)c4c(-c5ccccc5)n(C)n(-c5ccccc5)c4=O)c3N)cc2n1
Cc1ncc2ccc(Oc3c(C)ccc(C(=O)c4c(-c5ccccc5)n(C)n(-c5ccccc5)c4=O)c3N)cc2n1
Cc1nc2cc(ccc2s1)-c1c(C)ccc(C(=O)c2c(-c3ccccc3)n(C)n(-c3ccccc3)c2=O)c1N
Cc1nc2ccc(cc2s1)-c1c(C)ccc(C(=O)c2c(-c3ccccc3)n(C)n(-c3ccccc3)c2=O)c1N
CNc1nc2ccc(cc2s1)-c1c(C)ccc(C(=O)c2c(-c3ccccc3)n(C)n(-c3ccccc3)c2=O)c1N
Cc1ccc(C(=O)c2c(-c3ccccc3)n(C)n(-c3ccccc3)c2=O)c(N)c1-c1ccc2nc(N)sc2c1
Cc1ccc(C(=O)c2c(-c3ccccc3)n(C)n(-c3ccccc3)c2=O)c(N)c1-c1ccc2nc(CF)sc2c1
Cc1ccc(C(=O)c2c(-c3ccccc3)n(C)n(-c3ccccc3)c2=O)c(N)c1-c1ccc2nc(sc2c1)C(F)F
Cc1ccc(C(=O)c2c(-c3ccccc3)n(C)n(-c3ccccc3)c2=O)c(N)c1-c1ccc2nc(sc2c1)C(F)(F)F
Cc1ccc2cc(ccc2n1)-c1c(C)ccc(C(=O)c2c(-c3ccccc3)n(C)n(-c3ccccc3)c2=O)c1N
Cc1nc(N)c2c(cn(C)c2n1)-c1ccc2N(CC(=O)c3cc(F)cc(c3)C(F)(F)F)CCc2c1
CCCS(=O)(=O)Nc1cc(F)c(C(=O)c2c[nH]c3ncc(Cl)cc23)c(F)c1
CCN(C)S(=O)(=O)Nc1cc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(Cl)cc2)c(F)c1
CCCS(=O)(=O)Nc1cc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(Cl)cc2)c(F)c1
CCN(C)S(=O)(=O)Nc1cc(F)c(C(=O)c2c[nH]c3ncc(Cl)cc23)c(F)c1
Fc1ccc(NS(=O)(=O)c2cccnc2)c(F)c1C#Cc1cnc2[nH]nc(-c3ccc(Cl)cc3)c2c1
Fc1ccc(NS(=O)(=O)c2cccnc2)c(F)c1C#Cc1cnc2[nH]nc(-c3cccc(Cl)c3)c2c1
Fc1ccc(NS(=O)(=O)c2cccnc2)c(F)c1C#Cc1cnc2[nH]nc(-c3ccccc3Cl)c2c1
Fc1ccc(NS(=O)(=O)c2cccnc2)c(F)c1C#Cc1cnc2[nH]nc(-c3ccncc3)c2c1
Fc1ccc(NS(=O)(=O)c2cccnc2)c(F)c1C#Cc1cnc2[nH]nc(-c3ccccc3)c2c1
Fc1ccc(NS(=O)(=O)c2cccnc2)c(F)c1C#Cc1cnc2[nH]nc(C3CC3)c2c1
Cc1n[nH]c2ncc(cc12)C#Cc1c(F)ccc(NS(=O)(=O)c2cccnc2)c1F
CCOc1n[nH]c2ncc(cc12)C#Cc1c(F)ccc(NS(=O)(=O)c2cccnc2)c1F
COc1n[nH]c2ncc(cc12)C#Cc1c(F)ccc(NS(=O)(=O)c2cccnc2)c1F
Fc1ccc(NS(=O)(=O)c2cccnc2)c(F)c1C#Cc1cnc2ccnn2c1
Fc1ccc(NS(=O)(=O)c2cccnc2)c(F)c1C#Cc1ccc2[nH]ncc2c1
Fc1ccc(NS(=O)(=O)c2cccnc2)c(F)c1C#Cc1cnc2[nH]ccc2c1
Fc1ccc(NS(=O)(=O)c2cccnc2)c(F)c1C#Cc1cnc2[nH]ncc2c1
Fc1ccc(NS(=O)(=O)c2ccccn2)c(F)c1C#Cc1cnc2[nH]ncc2c1
Fc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(C#Cc2cnc3[nH]ncc3c2)c1F
Fc1cccc(c1)S(=O)(=O)Nc1ccc(F)c(C#Cc2cnc3[nH]ncc3c2)c1F
Fc1ccccc1S(=O)(=O)Nc1ccc(F)c(C#Cc2cnc3[nH]ncc3c2)c1F
Fc1ccc(NS(=O)(=O)c2ccccc2)c(F)c1C#Cc1cnc2[nH]ncc2c1
N#Cc1ccc(cc1)-c1cnc2ccc(NCc3ccccc3)nn12
OC1CCN(CC1)c1cc(ccn1)-c1cnc2ccc(nn12)N1CCC[C@@H]1c1cccc(F)c1 |r|
OC(=O)CN1CCN(CC1)c1cc(ccn1)-c1cnc2ccc(nn12)N1CCC[C@@H]1c1cccc(F)c1 |r|
CNc1ncc2cc(cnc2n1)-c1cc(NC(=O)NCCC(C)(C)C)c(F)cc1C
CNc1cc2nc(C)c(cc2cn1)-c1cc(NC(=O)NCCC(C)(C)C)c(F)cc1C
CNc1cc2nc(C)c(cc2cn1)-c1ccc(F)c(NC(=O)NCCC(C)(C)C)c1
CNc1ncc2cc(c(C)nc2n1)-c1ccc(F)c(NC(=O)NCCC(C)(C)C)c1
CNc1cc2nc(C)c(cc2cn1)-c1cc(NC(=O)NCCC(C)(C)C)ccc1C
CNc1cc2nc(C)c(cc2cn1)-c1cc(NC(=O)NC[C@@H](O)C(C)(C)C)c(F)cc1C |r|
CCn1c2cc(NC)ncc2cc(-c2cc(NC(=O)NCCC(C)(C)C)c(F)cc2C)c1=O
CCn1c2cc(NC)ncc2cc(-c2ccc(F)c(NC(=O)Nc3cc(no3)C(C)(C)C)c2)c1=O
CNc1cc2n([C@H]3CCOC3)c(=O)c(cc2cn1)-c1ccc(F)c(NC(=O)Nc2cc(no2)C(C)(C)C)c1 |r|
Cc1cc(F)c(NC(=O)NCCC(C)(C)C)cc1-c1cc2cnc(N)nc2nc1C
COc1cc(cc(OC)c1OC)-c1nc(c[nH]c1=O)-c1c[nH]c2ccccc12
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]c4ccccc4c23)c1
CNS(=O)(=O)c1ccc(N2CCOCC2)c(Nc2ncnc3[nH]c(cc23)-c2cccc(c2)C(F)(F)F)c1
CNS(=O)(=O)c1cccc(c1)Nc2c3c([nH]cn3)ncn2
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]ccc23)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]cc(C)c23)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]cc(C(C)C)c23)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]cc(CC(C)C)c23)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]cc(F)c23)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]cc(Cl)c23)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]cc(Br)c23)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]cc(-c4ccccc4)c23)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]cc(-c4ccccc4Cl)c23)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]cc(-c4cccc(Cl)c4)c23)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]cc(-c4ccc(Cl)cc4)c23)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]cc(-c4ccc(OC)cc4)c23)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]cc(-c4ccncc4)c23)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]cc(-c4ccc(CN)cc4)c23)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]cc(-c4ccc(cc4)C(O)=O)c23)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]c(Br)cc23)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]c(cc23)-c2ccccc2)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]c(cc23)-c2ccccc2C)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]c(cc23)-c2cccc(C)c2)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]c(cc23)-c2ccc(C)cc2)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]c(cc23)-c2cccc(c2)C(F)(F)F)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]c(cc23)-c2ccc(O)cc2)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]c(cc23)-c2ccncc2)c1
CNS(=O)(=O)c1cccc(Nc2ncnc3[nH]c(cc23)C(O)=O)c1
CNS(=O)(=O)c1ccc(Cl)c(Nc2ncnc3[nH]ccc23)c1
CNc1ccc(cc1Nc1ncnc2[nH]ccc12)S(=O)(=O)NC
CNS(=O)(=O)c1ccc(N2CCOCC2)c(Nc2ncnc3[nH]ccc23)c1
CNS(=O)(=O)c1ccc(N(C)C)c(Nc2ncnc3[nH]cc(C)c23)c1
CNS(=O)(=O)c1ccc(N(C)C)c(Nc2ncnc3[nH]cc(Br)c23)c1
CNS(=O)(=O)c1ccc(N2CCOCC2)c(Nc2ncnc3[nH]cc(C)c23)c1
CNS(=O)(=O)c1ccc(c(c1)Nc2c3c(c[nH]c3ncn2)Br)N4CCOCC4
CNS(=O)(=O)c1ccc(N(C)C)c(Nc2ncnc3[nH]c(Br)cc23)c1
CNS(=O)(=O)c1ccc(N(C)C)c(Nc2ncnc3[nH]c(cc23)-c2cccc(c2)C(F)(F)F)c1
CNS(=O)(=O)c1ccc(N2CCOCC2)c(Nc2ncnc3[nH]c(Br)cc23)c1
CN1CCN(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1ccc(C)c(NC(=O)c2cnoc2C)c1
Cn1c(Nc2cccc(c2)C(C)(C)C)nc2cc(Oc3ccnc(c3)-c3ncc[nH]3)ccc12
CNC(=O)c1cc(Oc2ccc3n(C)c(Nc4cccc(c4)C(C)(C)C)nc3c2)ccn1
Cn1c(Nc2cccc(c2)C(C)(C)C)nc2cc(Oc3ccnc(c3)-c3ncc([nH]3)-c3ccccc3)ccc12
Cn1c(Nc2cccc(c2)C(C)(C)C)nc2cc(Oc3ccnc(c3)-c3ncc([nH]3)C(F)(F)F)ccc12
Cn1c(Nc2ccc(cc2)C(C)(C)C)nc2cc(Oc3ccnc(c3)-c3ncc([nH]3)C(F)(F)F)ccc12
Cn1c(Nc2cc(ccc2F)C(C)(C)C)nc2cc(Oc3ccnc(c3)-c3ncc([nH]3)C(F)(F)F)ccc12
Cn1c(Nc2cccc(c2)C(F)(F)F)nc2cc(Oc3ccnc(c3)-c3ncc([nH]3)C(F)(F)F)ccc12
Cn1c(Nc2cc(ccc2F)C(F)(F)F)nc2cc(Oc3ccnc(c3)-c3ncc([nH]3)C(F)(F)F)ccc12
Cc1cnc([nH]1)-c1cc(Oc2ccc3n(C)c(Nc4cc(ccc4F)C(F)(F)F)nc3c2)ccn1
Cn1c2nc(Nc3ccc4[nH]ccc4c3)ncc2cc(c1=O)S(=O)(=O)c1ccc(F)cc1F
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1ccc2cc(NC[C@@H](C)NC(=O)OC)ncc2c1 |r|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1ccc2cc(NC[C@H](C)NC(=O)OC)ncc2c1 |r|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1cc2cnc(N)cc2cc1OC |(-13.09,.93,;-12.02,1.55,;-10.69,.78,;-9.35,1.54,;-9.35,2.78,;-8.28,2.16,;-8.02,.77,;-6.68,1.54,;-6.68,3.08,;-5.35,3.85,;-4.01,3.08,;-2.95,3.7,;-4.01,1.54,;-5.35,.77,;-5.35,-.46,;-2.68,.77,;-1.33,1.54,;,.77,;1.33,1.54,;2.66,.77,;2.66,-.77,;3.73,-1.38,;1.33,-1.54,;,-.77,;-1.33,-1.54,;-2.68,-.77,;-4.01,-1.54,;-4.01,-2.77,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1cc2cnc(NC[C@H](C)NC(=O)OC)cc2cc1OC |r,wU:23.24,(-13.09,.93,;-12.02,1.55,;-10.69,.78,;-9.35,1.54,;-9.35,2.78,;-8.28,2.16,;-8.02,.77,;-6.68,1.54,;-6.68,3.08,;-5.35,3.85,;-4.01,3.08,;-2.95,3.7,;-4.01,1.54,;-5.35,.77,;-5.35,-.46,;-2.68,.77,;-1.33,1.54,;,.77,;1.33,1.54,;2.66,.77,;2.66,-.77,;4,-1.54,;5.33,-.76,;6.67,-1.53,;6.67,-2.76,;8,-.76,;9.34,-1.53,;9.34,-2.76,;10.67,-.75,;11.74,-1.37,;1.33,-1.54,;,-.77,;-1.33,-1.54,;-2.68,-.77,;-4.01,-1.54,;-4.01,-2.77,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1cc2cnc(NC[C@H](C)NC(=O)OC)cc2cc1CC |r,wU:23.24,(-13.09,.93,;-12.02,1.55,;-10.69,.78,;-9.35,1.54,;-9.35,2.78,;-8.28,2.16,;-8.02,.77,;-6.68,1.54,;-6.68,3.08,;-5.35,3.85,;-4.01,3.08,;-2.95,3.7,;-4.01,1.54,;-5.35,.77,;-5.35,-.46,;-2.68,.77,;-1.33,1.54,;,.77,;1.33,1.54,;2.66,.77,;2.66,-.77,;4,-1.54,;5.33,-.76,;6.67,-1.53,;6.67,-2.76,;8,-.76,;9.34,-1.53,;9.34,-2.76,;10.67,-.75,;11.74,-1.37,;1.33,-1.54,;,-.77,;-1.33,-1.54,;-2.68,-.77,;-4.01,-1.54,;-4.01,-2.77,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1cc2cnc3[nH]ncc3c2cc1OC |(-13.75,-1.62,;-12.68,-2.23,;-11.35,-1.45,;-10.01,-2.22,;-10,-3.45,;-8.94,-2.83,;-8.68,-1.44,;-7.34,-2.2,;-7.34,-3.74,;-6,-4.5,;-4.67,-3.73,;-3.6,-4.34,;-4.67,-2.19,;-6.01,-1.42,;-6.02,-.19,;-3.35,-1.39,;-2,-2.11,;-.68,-1.39,;.66,-2.11,;2,-1.39,;2,.15,;3.17,1.19,;2.53,2.6,;.98,2.43,;.66,.92,;-.68,.15,;-2,.92,;-3.35,.15,;-4.69,.92,;-4.69,2.16,)|
COc1cc2c3c(n[nH]c3ncc2cc1-c1c(F)ccc(NS(=O)(=O)CCCF)c1Cl)C1CC1 |(-4.69,2.16,;-4.69,.92,;-3.35,.15,;-2,.92,;-.68,.15,;.66,.92,;.98,2.43,;2.53,2.6,;3.17,1.19,;2,.15,;2,-1.39,;.66,-2.11,;-.68,-1.39,;-2,-2.11,;-3.35,-1.39,;-4.67,-2.19,;-4.67,-3.73,;-3.6,-4.34,;-6,-4.5,;-7.34,-3.74,;-7.34,-2.2,;-8.68,-1.44,;-10.01,-2.22,;-10,-3.45,;-8.94,-2.83,;-11.35,-1.45,;-12.68,-2.23,;-14.02,-1.47,;-15.08,-2.09,;-6.01,-1.42,;-6.02,-.19,;-.05,3.57,;-.44,4.98,;-1.49,3.85,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1Cl)-c1cc2cnc3[nH]nc(C4CC4)c3c2cc1OC |(-13.75,-1.62,;-12.68,-2.23,;-11.35,-1.45,;-10.01,-2.22,;-10,-3.45,;-8.94,-2.83,;-8.68,-1.44,;-7.34,-2.2,;-7.34,-3.74,;-6,-4.5,;-4.67,-3.73,;-3.6,-4.34,;-4.67,-2.19,;-6.01,-1.42,;-6.02,-.19,;-3.35,-1.39,;-2,-2.11,;-.68,-1.39,;.66,-2.11,;2,-1.39,;2,.15,;3.17,1.19,;2.53,2.6,;.98,2.43,;-.05,3.57,;-.44,4.98,;-1.49,3.85,;.66,.92,;-.68,.15,;-2,.92,;-3.35,.15,;-4.69,.92,;-4.69,2.16,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1F)-c1cc2cnc3[nH]nc(C4CC4)c3c2cc1OC |(-13.75,-1.62,;-12.68,-2.23,;-11.35,-1.45,;-10.01,-2.22,;-10,-3.45,;-8.94,-2.83,;-8.68,-1.44,;-7.34,-2.2,;-7.34,-3.74,;-6,-4.5,;-4.67,-3.73,;-3.6,-4.34,;-4.67,-2.19,;-6.01,-1.42,;-6.02,-.19,;-3.35,-1.39,;-2,-2.11,;-.68,-1.39,;.66,-2.11,;2,-1.39,;2,.15,;3.17,1.19,;2.53,2.6,;.98,2.43,;-.05,3.57,;-.44,4.98,;-1.49,3.85,;.66,.92,;-.68,.15,;-2,.92,;-3.35,.15,;-4.69,.92,;-4.69,2.16,)|
CCCS(=O)(=O)Nc1ccc(F)c(c1Cl)-c1cc2cnc3[nH]ncc3c2cc1OC |(-13.75,-1.62,;-12.68,-2.23,;-11.35,-1.45,;-10.01,-2.22,;-10,-3.45,;-8.94,-2.83,;-8.68,-1.44,;-7.34,-2.2,;-7.34,-3.74,;-6,-4.5,;-4.67,-3.73,;-3.6,-4.34,;-4.67,-2.19,;-6.01,-1.42,;-6.02,-.19,;-3.35,-1.39,;-2,-2.11,;-.68,-1.39,;.66,-2.11,;2,-1.39,;2,.15,;3.17,1.19,;2.53,2.6,;.98,2.43,;.66,.92,;-.68,.15,;-2,.92,;-3.35,.15,;-4.69,.92,;-4.69,2.16,)|
COc1cc2c3cn[nH]c3ncc2cc1-c1c(F)ccc(NS(=O)(=O)CCCF)c1Cl |(-4.68,2.16,;-4.69,.92,;-3.35,.15,;-2,.92,;-.68,.15,;.66,.92,;.98,2.43,;2.53,2.6,;3.17,1.19,;2,.15,;2,-1.39,;.66,-2.11,;-.68,-1.39,;-2,-2.11,;-3.35,-1.39,;-4.67,-2.19,;-4.67,-3.73,;-3.6,-4.34,;-6,-4.5,;-7.33,-3.74,;-7.34,-2.2,;-8.68,-1.44,;-10.01,-2.21,;-10,-3.45,;-8.94,-2.82,;-11.35,-1.45,;-12.68,-2.23,;-14.02,-1.47,;-15.08,-2.09,;-6.01,-1.42,;-6.01,-.19,)|
CCCS(=O)(=O)Nc1ccc(Cl)c(c1Cl)-c1cc2cnc3[nH]ncc3c2cc1OC |(-13.75,-1.62,;-12.68,-2.23,;-11.35,-1.45,;-10.01,-2.22,;-10,-3.45,;-8.94,-2.83,;-8.68,-1.44,;-7.34,-2.2,;-7.34,-3.74,;-6,-4.5,;-4.67,-3.73,;-3.6,-4.34,;-4.67,-2.19,;-6.01,-1.42,;-6.02,-.19,;-3.35,-1.39,;-2,-2.11,;-.68,-1.39,;.66,-2.11,;2,-1.39,;2,.15,;3.17,1.19,;2.53,2.6,;.98,2.43,;.66,.92,;-.68,.15,;-2,.92,;-3.35,.15,;-4.69,.92,;-4.69,2.16,)|
CCCCS(=O)(=O)Nc1ccc(F)c(c1Cl)-c1cc2cnc3[nH]nc(C4CC4)c3c2cc1OC |(-15.08,-2.09,;-14.02,-1.47,;-12.68,-2.23,;-11.35,-1.45,;-10.01,-2.22,;-10,-3.45,;-8.94,-2.83,;-8.68,-1.44,;-7.34,-2.2,;-7.34,-3.74,;-6,-4.5,;-4.67,-3.73,;-3.6,-4.34,;-4.67,-2.19,;-6.01,-1.42,;-6.02,-.19,;-3.35,-1.39,;-2,-2.11,;-.68,-1.39,;.66,-2.11,;2,-1.39,;2,.15,;3.17,1.19,;2.53,2.6,;.98,2.43,;-.05,3.57,;-.44,4.98,;-1.49,3.85,;.66,.92,;-.68,.15,;-2,.92,;-3.35,.15,;-4.69,.92,;-4.69,2.16,)|
CCNCc1cc(cc(c1)C(F)(F)F)C(=O)N[C@@H]1CCc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1
NCc1cc(cc(c1)C(F)(F)F)C(=O)N[C@@H]1CCc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1
NC1(CCC1)c1cc(cc(c1)C(F)(F)F)C(=O)N[C@@H]1CCc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1
N[C@H](CO)c1cc(cc(c1)C(F)(F)F)C(=O)N[C@@H]1CCc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1
OC1(CNC1)c1cc(cc(c1)C(F)(F)F)C(=O)N[C@@H]1CCc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1
OCC1COCCN1Cc1cc(cc(c1)C(F)(F)F)C(=O)N[C@@H]1CCc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1 |r|
FC(F)(F)c1cc(cc(c1)-c1cnc[nH]1)C(=O)N[C@@H]1CCc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1 |r|
FC(F)(F)c1cc(cc(c1)-c1cc[nH]n1)C(=O)N[C@@H]1CCc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1 |r|
FC(F)(F)c1cc(cc(c1)-c1cn[nH]c1)C(=O)N[C@@H]1CCc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1
Cn1cnc(c1)-c1cc(cc(c1)C(F)(F)F)C(=O)N[C@@H]1CCc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1
Cn1nccc1-c1cc(cc(c1)C(F)(F)F)C(=O)N[C@@H]1CCc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1
Cn1cc(cn1)-c1cc(cc(c1)C(F)(F)F)C(=O)N[C@@H]1CCc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1
FC(F)(F)c1cccc(c1)C(=O)N[C@@H]1CCc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1 |r|
CNCc1cc(cc(c1)C(F)(F)F)C(=O)N[C@@H]1CCc2ccc(Oc3ccnc4NC(=O)CCc34)cc2C1 |r|
C[C@H](NC(=O)c1[nH]nc2cc(NCc3cccc(NC(=O)c4cc(cc(c4)C(F)(F)F)-n4cncc4C)c3)ccc12)C(N)=O |r|
FC(F)(F)c1cc(ccc1Cl)C(=O)Nc1cccc(c1)-c1cnc2c(NC(=O)c3cc(Cl)cc(Cl)c3)nccn12
Fc1ccc(NC(=O)Nc2cccc(c2)-c2cnc3c(NC(=O)c4cc(Cl)cc(Cl)c4)nccn23)c(F)c1
FC(F)(F)c1cc(NC(=O)Nc2cccc(c2)-c2cnc3c(NC(=O)c4cc(Cl)cc(Cl)c4)nccn23)ccc1Cl
FC(F)(F)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1nccn2c(cnc12)-c1cccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c1
Fc1ccc(cc1C(F)(F)F)C(=O)Nc1nccn2c(cnc12)-c1cccc(NC(=O)Nc2ccc(Cl)c(c2)C(F)(F)F)c1
Cc1n[nH]c(C)c1S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
CC(C)(C)CS(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Fc1ccc(NS(=O)(=O)Cc2ccccc2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
CCC(C)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
CCCC(C)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Fc1ccc(NS(=O)(=O)C2CCC2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Cc1ccc2c(Nc3ccc(Cl)cc3)nccc2c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)c2ccccc2F)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1cccc(c1)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Fc1ccc(cc1)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Fc1ccc(NS(=O)(=O)c2ccccn2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)c2nccs2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)c2cn[nH]c2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
CS(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Fc1ccc(NS(=O)(=O)CC(F)(F)F)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
CC(C)CS(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Fc1ccc(NS(=O)(=O)CC2CC2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)C2CCCC2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)C2CCOC2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)C2CCOCC2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
CN(C)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
CCN(C)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
CCN(CC)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F
Fc1ccc(NS(=O)(=O)N2CCCC2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
Fc1ccc(NS(=O)(=O)N2CCCCC2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
O[C@H]1CCN(C1)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F |r|
O[C@@H]1CCN(C1)S(=O)(=O)Nc1ccc(F)c(Nc2ncccc2-c2ncnc3[nH]cnc23)c1F |r|
Fc1ccc(NS(=O)(=O)N2CCNCC2)c(F)c1Nc1ncccc1-c1ncnc2[nH]cnc12
CC(=O)Nc1cc(Nc2cccc(NC(=O)c3cccc(c3)C3CC3)c2)ccn1
O=C(Nc1cc(Nc2cccc(NC(=O)c3cccc(c3)C3(CC3)C#N)c2)ccn1)C1CC1
CC(C)(C#N)c1cccc(c1)C(=O)Nc1cccc(Nc2ccnc(NC(=O)C3CC3)c2)c1
O=C(Nc1cc(Nc2cccc(NC(=O)c3cccc(c3)C3CC3)c2)ccn1)C1CC1
CC(C)(C)c1cccc(c1)C(=O)Nc1cccc(Nc2ccnc(NC(=O)C3CC3)c2)c1
CC(C)c1cccc(c1)C(=O)Nc1cccc(Nc2ccnc(NC(=O)C3CC3)c2)c1
O=C(Nc1cc(Nc2cccc(NC(=O)c3cccc(c3)C3CC3)c2)ccn1)C1CCCCC1
O=C(Nc1cc(Nc2cccc(NC(=O)c3cccc(c3)C3CC3)c2)ccn1)C1CCCC1
O=C(Nc1cc(Nc2cccc(NC(=O)c3cccc(c3)C3CC3)c2)ccn1)C1CCC1
CC(C)(C)C(=O)Nc1cc(Nc2cccc(NC(=O)c3cccc(c3)C3CC3)c2)ccn1
CC(C)C(=O)Nc1cc(Nc2cccc(NC(=O)c3cccc(c3)C3CC3)c2)ccn1
CCC(=O)Nc1cc(Nc2cccc(NC(=O)c3cccc(c3)C3CC3)c2)ccn1
CCc1cccc(c1)C(=O)Nc1cccc(Nc2ccnc(NC(=O)C3CC3)c2)c1
Cc1cccc(c1)C(=O)Nc1cccc(Nc2ccnc(NC(=O)C3CC3)c2)c1
O=C(Nc1cc(Nc2cccc(NC(=O)c3cccc(c3)C#N)c2)ccn1)C1CC1
[O-][N+](=O)c1cccc(c1)C(=O)Nc1cccc(Nc2ccnc(NC(=O)C3CC3)c2)c1
Clc1cccc(c1)C(=O)Nc1cccc(Nc2ccnc(NC(=O)C3CC3)c2)c1
FC(F)(F)c1ccc(cc1)C(=O)Nc1cccc(Nc2ccnc(NC(=O)C3CC3)c2)c1
FC(F)(F)c1ccccc1C(=O)Nc1cccc(Nc2ccnc(NC(=O)C3CC3)c2)c1
FC(F)(F)c1cccc(c1)C(=O)Nc1cccc(Nc2ccnc(NC(=O)C3CC3)c2)c1
Clc1ccc(cc1Cl)C1CC(=NN1c1ccccc1)c1ccc2OCCOc2c1 |c:11|
CN(C)c1ccc(cc1)C1CC(=NN1c1ccccc1)c1ccc2OCCOc2c1 |c:12|
C(Oc1ccc(cc1)C1CC(=NN1c1ccccc1)c1ccc2OCCOc2c1)c1ccccc1 |c:11|
Clc1cccc(c1)C1CC(=NN1c1ccccc1)c1ccc2OCCOc2c1 |c:10|
C(Oc1cccc(c1)C1CC(=NN1c1ccccc1)c1ccc2OCCOc2c1)c1ccccc1 |c:11|
COc1cccc(c1)C1CC(=NN1c1ccccc1)c1ccc2OCCOc2c1 |c:11|
c1ccc(cc1)Nc2c[nH]c3c2cccn3
COC(=O)c1cc2cc(NCc3cc(NC(=O)c4cc(cc(c4)C(F)(F)F)-n4cnc(C)c4)ccc3C)cnc2[nH]1
CCOc1cc2ncnc(Nc3cc(ccc3OCC(F)(F)F)S(=O)(=O)NC)c2cc1OC
CNS(=O)(=O)c1ccc(OCC(F)(F)F)c(Nc2ncnc3cc(OC(C)C)c(OC)cc23)c1
CNS(=O)(=O)c1ccc(OCC(F)(F)F)c(Nc2ncnc3cc(OCCCOC)ccc23)c1
CNS(=O)(=O)c1ccc(OCC(F)(F)F)c(Nc2ncnc3cc(OCCCN4CCOCC4)ccc23)c1
CNS(=O)(=O)c1ccc(c(c1)Nc2c3c(c[nH]c3ncn2)Cl)N4CCOCC4
CNS(=O)(=O)c1ccc(N(C)C)c(Nc2ncnc3ccccc23)c1
CNS(=O)(=O)c1ccc(N(C)C)c(Nc2ncnc3ccsc23)c1
CNS(=O)(=O)c1ccc(N(C)C)c(Nc2ncnc3ccn(C)c23)c1
CNS(=O)(=O)c1ccc(N(C)C)c(Nc2ncnc3cc[nH]c23)c1
CNS(=O)(=O)c1ccc(N(C)C)c(Nc2ncnc3ccc(OC)cc23)c1
CNS(=O)(=O)c1ccc(N(C)C)c(Nc2ncnc3ccc(N)cc23)c1
CNc1ccc2ncnc(Nc3cc(ccc3N(C)C)S(=O)(=O)NC)c2c1
CNS(=O)(=O)c1ccc(N(C)C)c(Nc2ncnc3cc(N)ccc23)c1
CNc1ccc2c(Nc3cc(ccc3N(C)C)S(=O)(=O)NC)ncnc2c1
CNS(=O)(=O)c1ccc(N(C)C)c(Nc2ncnc3cc(OCCCOC)ccc23)c1
CNS(=O)(=O)c1ccc(N(C)C)c(Nc2ncnc3cc(OCCCN4CCOCC4)ccc23)c1
CNS(=O)(=O)c1ccc(N(C)C)c(Nc2ncnc3cc(OC)cc(OC)c23)c1
CNS(=O)(=O)c1ccc(OCC(F)(F)F)c(Nc2ncnc3cc(OC)c(OC)cc23)c1
CNS(=O)(=O)c1ccc(OCC(F)(F)F)c(Nc2ncnc3cc(OC)cc(OC)c23)c1
CNS(=O)(=O)c1ccc(OCC(F)(F)F)c(Nc2ncnc3cc(OC)c(OC)c(OC)c23)c1
CS(=O)(=O)Nc1cccc(Cn2c(=O)oc3cc(OC(=O)c4ccccc4)ccc3c2=O)c1F
COc1ccc2c(c1)oc(=O)n(Cc1cccc(NS(=O)(=O)NCCC#N)c1F)c2=O
CCCC(=O)Oc1ccc2c(c1)oc(=O)n(Cc1cccc(NS(=O)(=O)NC)c1F)c2=O
CNS(=O)(=O)Nc1cccc(Cn2c(=O)oc3cc(OC(C)=O)ccc3c2=O)c1F
CCC(=O)Oc1ccc2c(c1)oc(=O)n(Cc1cccc(NS(=O)(=O)NC)c1F)c2=O
CNS(=O)(=O)Nc1cccc(Cn2c(=O)oc3cc(OC(=O)C(C)C)ccc3c2=O)c1F
CNS(=O)(=O)Nc1cccc(Cn2c(=O)oc3cc(OS(C)(=O)=O)ccc3c2=O)c1F
CCS(=O)(=O)Oc1ccc2c(c1)oc(=O)n(Cc1cccc(NS(=O)(=O)NC)c1F)c2=O
CN(C)C(=O)Oc1ccc2c(c1)oc(=O)n(Cc1cccc(NS(=O)(=O)NCc3ccccc3)c1F)c2=O
CN(C)C(=O)Oc1ccc2c(c1)oc(=O)n(Cc1cccc(NS(=O)(=O)Nc3ccccc3)c1F)c2=O
CC(C)NS(=O)(=O)Nc1cccc(Cn2c(=O)oc3cc(OC(=O)N(C)C)ccc3c2=O)c1F
CN(C)C(=O)Oc1ccc2c(c1)oc(=O)n(Cc1cccc(NS(=O)(=O)NCCC#N)c1F)c2=O
CN(C)C(=O)Oc1ccc2c(c1)oc(=O)n(Cc1cccc(NS(=O)(=O)NCC(F)(F)F)c1F)c2=O
CNS(=O)(=O)Nc1cccc(Cn2c(=O)oc3cc(OC(=O)N(C)C)ccc3c2=O)c1F
CN(C)C(=O)Oc1ccc2c(c1)oc(=O)n(Cc1cccc(NS(N)(=O)=O)c1F)c2=O
CCS(=O)(=O)Nc1cccc(Cn2c(=O)oc3cc(OC(=O)N(C)C)ccc3c2=O)c1F
CN(C)C(=O)Oc1ccc2oc(=O)n(Cc3cccc(NS(C)(=O)=O)c3F)c(=O)c2c1
CN(C)C(=O)Oc1ccc2c(c1)oc(=O)n(Cc1cccc(NC(C)=O)c1)c2=O
CN(C)C(=O)Oc1ccc2c(c1)oc(=O)n(Cc1ccc(F)c(NS(C)(=O)=O)c1)c2=O
CN(C)C(=O)Oc1ccc2c(c1)oc(=O)n(Cc1cccc(NS(C)(=O)=O)c1F)c2=O
CN(C)C(=O)Oc1ccc2c(c1)oc(=O)n(Cc1ccc(NS(C)(=O)=O)cc1)c2=O
CN(C)C(=O)Oc1ccc2c(c1)oc(=O)n(Cc1ccccc1NS(C)(=O)=O)c2=O
CN(C)C(=O)Oc1ccc2c(c1)oc(=O)n(Cc1cccc(NS(C)(=O)=O)c1)c2=O
CN(C)C(=O)Oc1ccc2c(c1)oc(=O)n(Cc1cccc(c1)[N+]([O-])=O)c2=O
CN(C)C(=O)Oc1ccc2c(c1)oc(=O)n(Cc1ccc(F)cc1)c2=O
CN(C)C(=O)Oc1ccc2c(c1)oc(=O)n(Cc1ccccc1F)c2=O
CN(C)C(=O)Oc1ccc2c(C)c(Cc3ccc(F)cc3)c(=O)oc2c1
Nc1ccccc1SC(=N)C(C#N)C(C#N)C(=N)Sc1ccccc1N
CNC(=O)c1cc(Oc2ccc(cc2)C(=O)\C=C\c2ccccc2)ccn1
CNC(=O)c1cc(Oc2ccc(cc2)C(=O)\C=C\c2cc(OC)c(OC)c(OC)c2)ccn1
CNC(=O)c1cc(Oc2ccc(cc2)C(=O)\C=C\c2cccc(Br)c2)ccn1
CNC(=O)c1cc(Oc2ccc(\C=C\C(=O)c3ccc(F)cc3)cc2)ccn1
CC1(C)C(=O)N([C@H]2CCc3c2cccc3O)c2nc(Nc3ccccc3)ncc12 |r|
COc1cc2cc(Oc3ccc(NC(=O)Nc4ccc(Cl)c(c4)C(F)(F)F)cc3)c(C)nc2cc1OC
CC1(C)OCC(=O)Nc2cc(Nc3nc(NCC(F)(F)F)c4occc4n3)ccc12
CCCNC(=O)c1ccc(Nc2nc(NCC(F)(F)F)c3cc[nH]c3n2)cc1