1193 SMILES Strings for Stearoyl-CoA desaturase

Compound Name
SMILES String
CCCCCCCCC1=C(CCCCCCCC(O)=O)C1 |c:8|
Cn1cc(Cl)nc(N2CCC(CC2)Oc2ccccc2Cl)c1=O
Cn1cc(Cl)nc(N2CCC(CC2)Oc2ccccc2C(F)(F)F)c1=O
Cn1cc(Cl)nc(N2CCC(CC2)Oc2cc(ccc2Cl)C(F)(F)F)c1=O
Cc1ccccc1OC1CCN(CC1)c1nc(Cl)cn(C)c1=O
Cn1ccnc(N2CCC(CC2)Oc2ccccc2C(F)(F)F)c1=O
Cn1cc(Cl)nc(N2CCC(CC2)Oc2cc(F)ccc2Cl)c1=O
Clc1ccccc1OC1CCN(CC1)c1nccnn1
FC(F)(F)c1ccccc1OC1CCN(CC1)c1nccnn1
FC(F)(F)c1ccc(Cl)c(OC2CCN(CC2)c2nccnn2)c1
Fc1ccc(Cl)c(OC2CCN(CC2)c2nccnn2)c1
Cc1nnc(nc1C)N1CCC(CC1)Oc1cc(ccc1Cl)C(F)(F)F
Cc1cnnc(n1)N1CCC(CC1)Oc1cc(F)ccc1Cl
Cc1cnnc(n1)N1CCC(CC1)Oc1cc(ccc1Cl)C(F)(F)F
Cc1cnnc(n1)N1CCC(CC1)Oc1ccccc1Cl
Cc1cnc(nn1)N1CCC(CC1)Oc1cc(F)ccc1Cl
[O-][N+](=O)c1ccc(Cl)c(OC2CCN(CC2)c2nccnn2)c1
Fc1cc(Br)c(OC2CCN(CC2)c2nccnn2)cc1F
[O-][N+](=O)c1ccccc1OC1CCN(CC1)c1nccnn1
FC(F)(F)c1ccccc1NC1CCN(CC1)c1nccnn1
CC1CN(CCC1Oc1cc(ccc1Cl)C(F)(F)F)c1nccnn1
CC1CN(CCC1Oc1cc(Cl)ccc1Cl)c1nccnn1
Cn1nccc(N2CCC(CC2)Oc2cc(ccc2Cl)C(F)(F)F)c1=O
FC(F)(F)c1ccc(Cl)c(OC2CCN(C2)c2nccnn2)c1
OC(=O)Cn1nnc(n1)-c1nnc(s1)N1CCC2(CC1)CCc1c(Cl)cccc1O2
OC(=O)Cn1nnc(n1)-c1cc(no1)N1CCC2(CC1)CCc1c(Cl)cccc1O2
OC(=O)Cn1nnc(n1)-c1cnc(s1)N1CCC2(CC1)CCc1c(Cl)cccc1O2
OC(=O)Cn1nnc(n1)-c1cnc(s1)N1CCC2(CC1)CC(=O)c1ccccc1O2
OC(=O)Cn1nnc(n1)-c1cnc(s1)N1CCC2(CCc3ccccc23)CC1
OC(=O)Cn1nnc(n1)-c1cnc(s1)N1CCC2(COc3ccccc23)CC1
OC(=O)Cn1nnc(n1)-c1cnc(s1)N1CCC2(CC1)C=Cc1ccccc21 |c:23|
OC(=O)Cn1nnc(n1)-c1nnc(s1)N1CCC2(CC1)CC(=O)c1ccccc1O2
OC(=O)Cn1nnc(n1)-c1cnc(s1)N1CCC2(CC1)NC(=O)c1ccccc1O2
OC(=O)Cn1nnc(n1)-c1nnc(s1)N1CCC2(CC1)Cc1ccccc1C(=O)O2
COc1cccc2OC3(CCN(CC3)c3nnc(s3)-c3nnn(CC(O)=O)n3)CCc12
OC(=O)Cn1nnc(n1)-c1nnc(s1)N1CCC2(CC1)CCc1c(O)cccc1O2
OC(=O)Cn1nnc(n1)-c1nnc(s1)N1CCC2(CC1)CC(=O)c1c(Cl)cccc1O2
OC(=O)Cn1nnc(n1)-c1cnc(s1)N1CCC2(CC1)CC(=O)c1c(Cl)cccc1O2
OC(=O)Cn1nnc(n1)-c1cc(no1)N1CCC2(CC1)CC(=O)c1c(Cl)cccc1O2
OC(=O)Cn1nnc(n1)-c1cc(no1)N1CCC2(CC1)CCc1c(OC(F)(F)F)cccc1O2
OC(=O)Cn1nnc(n1)-c1nnc(s1)N1CCC2(CC1)CCc1c(OC(F)(F)F)cccc1O2
OC(=O)Cn1nnc(n1)-c1cnc(s1)N1CCC2(CC1)CCc1c(OC(F)(F)F)cccc1O2
OC(=O)Cn1nnc(n1)-c1cc(no1)N1CCC2(CC1)CCc1c(Br)cccc1O2
OC(=O)Cn1nnc(n1)-c1cnc(s1)N1CCC2(CC1)CCc1c(Br)cccc1O2
Cc1cccc2OC3(CCN(CC3)c3ncc(s3)-c3nnn(CC(O)=O)n3)CCc12
OC(=O)Cn1nnc(n1)-c1cnc(s1)N1CCC2(CC1)Cc1cccc(Cl)c1C(=O)O2
OC(=O)Cn1nnc(n1)-c1cnc(s1)N1CCC2(CC1)NC(=O)c1c(Cl)cccc1O2
OC(=O)Cn1ccn(-c2cnc(s2)N2CCC3(CC2)CCc2c(Cl)cccc2O3)c1=O
OC(=O)Cn1nnc(n1)-c1nnc(s1)N1CCC2(CC1)CCc1c(O2)cccc1C(F)(F)F
OC(=O)Cn1nnc(n1)-c1cnc(s1)N1CCC2(CC1)CCc1c(O2)cccc1C(F)(F)F
Cc1nn(C)c(C)c1NC(=O)c1cc(on1)-c1ccco1
Cc1nn(Cc2ccccc2)c(C)c1NC(=O)c1cc(on1)-c1ccco1
Cc1nn(Cc2ccc(Cl)c(Cl)c2)c(C)c1NC(=O)c1cc(on1)-c1ccco1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)-c1ccco1
Cc1nn(Cc2ccccc2)c(C)c1NC(=O)c1cc(on1)-c1ccc2OCOc2c1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)-c1ccc2OCOc2c1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)-c1ccccc1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)-c1ccccn1
CN(Cc1cccc(F)c1)C(=O)c1cc(on1)-c1ccccc1
Cn1cc(NC(=O)c2cc(on2)-c2ccco2)cn1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(no1)-c1ccco1
CC(C)(C)OC(=O)n1cc(NC(=O)c2cc(on2)-c2ccco2)cn1
O=C(Nc1cn[nH]c1)c1cc(on1)-c1ccco1
FC(F)(F)c1ccccc1Cn1cc(NC(=O)c2cc(on2)-c2ccco2)cn1
Clc1ccc(Cn2cc(NC(=O)c3cc(on3)-c3ccco3)cn2)cc1
FC(F)(F)c1ccc(Cn2cc(NC(=O)c3cc(on3)-c3ccco3)cn2)cc1
Cc1nn(Cc2ccc(Cl)c(Cl)c2)cc1NC(=O)c1cc(on1)-c1ccco1
Fc1ccc(Cn2cc(NC(=O)c3cc(on3)-c3ccco3)cn2)cc1
Fc1ccccc1Cn1cc(NC(=O)c2cc(on2)-c2ccco2)cn1
FC(F)(F)c1cccc(Cn2cc(NC(=O)c3cc(on3)-c3ccco3)cn2)c1
Cc1c(NC(=O)c2cc(on2)-c2ccco2)cnn1Cc1ccc(Cl)c(Cl)c1
Clc1cccc(Cn2cc(NC(=O)c3cc(on3)-c3ccco3)cn2)c1
Clc1ccccc1Cn1cc(NC(=O)c2cc(on2)-c2ccco2)cn1
O=C(Nc1cnn(CCc2ccccc2)c1)c1cc(on1)-c1ccco1
O=C(Nc1cn[nH]c1)c1cc(on1)-c1ccccc1
O=C(Nc1cnn(CC2CCCCC2)c1)c1cc(on1)-c1ccco1
Cn1nc(Cc2ccc(Cl)c(Cl)c2)cc1NC(=O)c1cc(on1)-c1ccco1
Fc1ccc(Cl)c(Cn2cc(NC(=O)c3cc(on3)-c3ccco3)cn2)c1
Clc1ccc(Cn2cc(NC(=O)c3cc(on3)-c3ccco3)cn2)cc1Cl
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)-c3ccco3)cn2)c1
O=C(Nc1cnn(CC2CCOCC2)c1)c1cc(on1)-c1ccco1
Clc1ccc(CN(C(=O)c2cc(on2)-c2ccco2)c2cnn(Cc3ccc(Cl)cc3)c2)cc1
O=C(Nc1cnn(c1)-c1ccccc1)c1cc(on1)-c1ccco1
FC(F)(F)CCCn1cc(NC(=O)c2cc(on2)-c2ccco2)cn1
CC(C)(C)OC(=O)n1cc(NC(=O)c2cc(on2)-c2ccccc2)cn1
Fc1ccc(c(Cn2cc(NC(=O)c3cc(on3)-c3ccco3)cn2)c1)C(F)(F)F
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)-c1cncs1
Fc1ccccc1-c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
O=C(Nc1cnn(Cc2cccnc2)c1)c1cc(on1)-c1ccccc1
O=C(Nc1cnn(Cc2ccccn2)c1)c1cc(on1)-c1ccccc1
O=C(Nc1cnn(CC2CC2)c1)c1cc(on1)-c1ccccc1
O=C(Nc1cnn(Cc2ccc(cc2)C#N)c1)c1cc(on1)-c1ccccc1
O=C(Nc1cnn(Cc2ccc(s2)C#N)c1)c1cc(on1)-c1ccccc1
O=C(Nc1cn(Cc2ccccc2)nn1)c1cc(on1)-c1ccccc1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)-c3cnccn3)cn2)c1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)-c3ncccn3)cn2)c1
O=C(N(Cc1ccc(cc1)C#N)c1cnn(Cc2ccc(cc2)C#N)c1)c1cc(on1)-c1ccccc1
NC(=O)c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
O=C(Nc1cc(on1)-c1ccco1)c1cnn(Cc2ccccc2)c1
O=C(Nc1cnn(CC2CCOC2)c1)c1cc(on1)-c1ccccc1
CC(c1ccccc1)n1cc(NC(=O)c2cc(on2)-c2ccccc2)cn1
O=C(Nc1cnn(Cc2ccccc2)n1)c1cc(on1)-c1ccccc1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)-c3ccccc3)cn2)c1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)-c3ccccn3)cn2)c1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)-c3cccnc3)cn2)c1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)-c3ccncc3)cn2)c1
Clc1cccc(Cn2cc(NC(=O)c3cc(on3)-c3ccccn3)cn2)c1
CC(=C)c1cc(no1)C(=O)Nc1cnn(Cc2cccc(F)c2)c1
Clc1ccc(Cn2cc(cn2)C(=O)Nc2cc(on2)-c2ccco2)cc1Cl
CC(C)c1cc(no1)C(=O)Nc1cnn(Cc2cccc(F)c2)c1
Fc1ccc(Cn2cc(NC(=O)c3cc(on3)-c3ccccn3)cn2)cc1F
Fc1ccc(CN(C(=O)c2cc(on2)-c2ccccn2)c2cnn(Cc3ccc(F)c(F)c3)c2)cc1F
O=C(Nc1cnn(Cc2ccc(cn2)C#N)c1)c1cc(on1)-c1ccccc1
CC(C)(c1ccccc1)n1cc(NC(=O)c2cc(on2)-c2ccccc2)cn1
CN(C)CCC(c1ccccc1)n1cc(NC(=O)c2cc(on2)-c2ccccc2)cn1
Cc1nn(Cc2ccccc2)cc1NC(=O)c1cc(on1)-c1ccccc1
Cc1ncc(o1)-c1cc(no1)C(=O)Nc1cnn(Cc2cccc(F)c2)c1
O=C(Nc1cn(Cc2ccccc2)nc1C#N)c1cc(on1)-c1ccccc1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)-c3cncs3)cn2)c1
CSCCC(c1ccccc1)n1cc(NC(=O)c2cc(on2)-c2ccccc2)cn1
CS(=O)CCC(c1ccccc1)n1cc(NC(=O)c2cc(on2)-c2ccccc2)cn1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)-c3ccon3)cn2)c1
CSCC(c1ccccc1)n1cc(NC(=O)c2cc(on2)-c2ccccc2)cn1
Fc1ccc(c(Cn2cc(NC(=O)c3cc(on3)-c3ccccc3)cn2)c1)C(F)(F)F
CS(=O)(=O)CCC(c1ccccc1)n1cc(NC(=O)c2cc(on2)-c2ccccc2)cn1
CN(C(=O)c1cc(on1)-c1ccccc1)c1cnn(Cc2cc(F)ccc2C(F)(F)F)c1
Fc1ccc(c(Cn2cc(NC(=O)c3cc(on3)-c3ccccn3)cn2)c1)C(F)(F)F
CS(=O)CC(c1ccccc1)n1cc(NC(=O)c2cc(on2)-c2ccccc2)cn1
O=C(Nc1noc(Cc2ccccc2)n1)c1cc(on1)-c1ccccc1
CS(=O)(=O)CC(c1ccccc1)n1cc(NC(=O)c2cc(on2)-c2ccccc2)cn1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)-c3ccns3)cn2)c1
FC(F)(F)c1nn(Cc2ccccc2)cc1NC(=O)c1cc(on1)-c1ccccc1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)C3CCCCC3)cn2)c1
CC(=C)c1cc(no1)C(=O)Nc1cnn(Cc2cc(F)ccc2C(F)(F)F)c1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)C3=CCCCC3)cn2)c1 |t:19|
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)-c3cnco3)cn2)c1
CNC(=O)c1cc(no1)C(=O)Nc1cnn(Cc2cccc(F)c2)c1
Fc1ccc(C#N)c(Cn2cc(NC(=O)c3cc(on3)-c3ccccc3)cn2)c1
Cn1cccc(-c2cc(no2)C(=O)Nc2cnn(Cc3cccc(F)c3)c2)c1=O
CC(=O)c1cc(no1)C(=O)Nc1cnn(Cc2cccc(F)c2)c1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)-c3ccncn3)cn2)c1
Clc1ccccc1Cn1cc(NC(=O)c2cc(on2)-c2cccc3cn(nc23)C2COC2)cn1
Clc1ccccc1Cn1cc(NC(=O)c2cc(on2)-c2cccc3cnn(C4COC4)c23)cn1
Clc1ccccc1Cn1cc(NC(=O)c2cc(on2)-c2cccc3n(ncc23)C2COC2)cn1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)-c1cccc2cn(nc12)C1COC1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)-c1cccc2cnn(C3COC3)c12
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)-c1cccc2n(ncc12)C1COC1
Fc1cc(Cn2cc(NC(=O)c3cc(on3)-c3ccccc3)cn2)cc(c1)C#N
Fc1ccc(c(Cn2cc(NC(=O)c3cc(on3)-c3ccc(cn3)C#N)cn2)c1)C(F)(F)F
OC1(CCC1)c1cc(no1)C(=O)Nc1cnn(Cc2cccc(F)c2)c1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)N3CCOCC3)cn2)c1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)N3CCCCC3)cn2)c1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)-c3ccccc3C#N)cn2)c1
CCc1cc(no1)C(=O)Nc1cnn(Cc2cccc(F)c2)c1
Fc1cccc(Cn2cc(NC(=O)c3cc(Cl)on3)cn2)c1
Fc1cccc(Cn2cc(NC(=O)c3cc(C=C)on3)cn2)c1
Fc1ccc(c(Cn2cc(NC(=O)c3cc(on3)-c3ncccc3F)cn2)c1)C(F)(F)F
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)-c3ncccc3F)cn2)c1
COc1ccc(Cn2cc(NC(=O)c3cc(on3)-c3ccccc3)cn2)cc1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)-c1nccs1
Fc1ccccc1Cn1cc(NC(=O)c2cc(on2)-c2ccccc2)cn1
Fc1ccc(Cn2cc(NC(=O)c3cc(on3)-c3ccccc3)cn2)cc1
CN(C)CC(c1ccccc1)n1cc(NC(=O)c2cc(on2)-c2ccccc2)cn1
Fc1ccccc1-c1cc(no1)C(=O)Nc1cnn(Cc2cnccc2C(F)(F)F)c1
COC1(CCC1)c1cc(no1)C(=O)Nc1cnn(Cc2cccc(F)c2)c1
CC1(COC1)c1cc(no1)C(=O)Nc1cnn(Cc2cccc(F)c2)c1
CC(C)c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
CC(C)(C)c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)C1CC1
COC1(CCC1)c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
CC1(COC1)c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
Fc1cccnc1-c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(no1)-c1ccccc1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)-c1ccncc1
COc1ccccc1Cn1cc(NC(=O)c2cc(on2)-c2ccccc2)cn1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)-c1ccns1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)-c1cccc(c1)C#N
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)-c1ccc(cc1)C#N
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(no1)-c1ccccn1
Fc1ccccc1-c1cc(on1)C(=O)Nc1cnn(Cc2ccccc2)c1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(no1)-c1cncs1
O=C(Nc1cnn(Cc2cccc(c2)C#N)c1)c1cc(on1)-c1ccccc1
Cc1ncc(s1)-c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
Clc1cnccc1-c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)-c1ccccc1C#N
COc1ccccc1-c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
Fc1ccc(nc1)-c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
O=C(c1cnn(Cc2ccncc2)c1)c1cc(on1)-c1ccccc1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)C3COC3)cn2)c1
COCc1ncc(s1)-c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
Clc1ccccc1-c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
Cc1cnc(s1)-c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
Cc1csc(n1)-c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
Fc1cccc(c1)-c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
COc1ccc(nc1)C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)-c1cnsc1
Fc1cnccc1-c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)-c1ccncn1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)-c1cnco1
CCOC(=O)c1cc(on1)C(=O)Nc1cnn(Cc2ccccc2)c1
CC(C)(O)c1cc(on1)C(=O)Nc1cnn(Cc2ccccc2)c1
CC(=C)c1cc(on1)C(=O)Nc1cnn(Cc2ccccc2)c1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)C#C)cn2)c1
CCOC(=O)c1cc(on1)-c1cc(no1)C(=O)Nc1cnn(Cc2cccc(F)c2)c1
O=C(Nc1cnn(Cc2ccccc2)c1)c1noc2CCCCc12
Fc1ccc(-c2cc(no2)C(=O)Nc2cnn(Cc3ccccc3)c2)c(F)c1
CC(C)c1cc(on1)C(=O)Nc1cnn(Cc2ccccc2)c1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)N1CCCCC1
FC(F)(F)c1ccncc1Cn1cc(NC(=O)c2cc(on2)-c2ccccc2)cn1
CC(C)c1cc(no1)C(=O)Nc1cnn(Cc2cnccc2C(F)(F)F)c1
NC(=O)c1cc(no1)C(=O)Nc1cnn(Cc2cccc(F)c2)c1
Cc1nnc(s1)-c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
Cc1ncc(o1)-c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
Cc1nnc(o1)-c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
CC(=C)c1cc(no1)C(=O)Nc1cnn(Cc2cnccc2C(F)(F)F)c1
CC(C)c1cc(no1)C(=O)Nc1cnn(CC23CCC(CC2)CC3)c1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)-c3ccno3)cn2)c1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)C#N)cn2)c1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)-c1nncs1
FC(F)(F)c1ccncc1Cn1cc(NC(=O)c2cc(on2)-c2cnco2)cn1
Cc1ccncc1Cn1cc(NC(=O)c2cc(on2)-c2ccccc2F)cn1
COc1ccncc1Cn1cc(NC(=O)c2cc(on2)-c2ccccc2F)cn1
Fc1cccc(Cn2cc(NC(=O)c3cc(on3)-c3nncs3)cn2)c1
Cc1nnc(s1)-c1cc(no1)C(=O)Nc1cnn(Cc2cccc(F)c2)c1
CC(C)c1cc(no1)C(=O)Nc1cc2ccccn2n1
Fc1ccccc1-c1cc(no1)C(=O)Nc1cnn(Cc2cccnc2C(F)(F)F)c1
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)N1CCCC1
Cc1nnc(o1)-c1cc(no1)C(=O)Nc1cnn(Cc2cccc(F)c2)c1
Clc1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
CC(C)(C)OC(=O)Nc1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
FC(F)(F)c1ccncc1Cn1cc(NC(=O)c2cc(on2)N2CCCCC2)cn1
CN1CCN(CC1)c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
CC(=O)N1CCN(CC1)c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
CC(C)(C)OC(=O)N1CCN(CC1)c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
O[C@@H]1CCN(C1)c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1 |r|
O[C@H]1CCN(C1)c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1 |r|
CO[C@@H]1CCN(C1)c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1 |r|
CO[C@H]1CCN(C1)c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1 |r|
O=C(Nc1cnn(Cc2ccccc2)c1)c1cc(on1)N1CCNCC1
OCc1cc(no1)C(=O)Nc1cnn(Cc2cccc(F)c2)c1
Nc1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
Fc1cccc(Cn2cc(NC(=O)c3noc4CCCCc34)cn2)c1
FC(F)(F)c1ccncc1Cn1cc(NC(=O)c2noc3CCCCc23)cn1
Fc1cccc(F)c1-c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
Fc1ccccc1-c1cc(no1)C(=O)Nc1cnn(Cc2ncccc2C(F)(F)F)c1
FC(F)(F)c1ccncc1Cn1cc(NC(=O)c2cc(on2)-c2ccccn2)cn1
FC(F)(F)c1ccncc1Cn1cc(NC(=O)c2cc(on2)-c2ccco2)cn1
FC(F)(F)c1ccncc1Cn1cc(NC(=O)c2cc(on2)-c2ccc3OCOc3c2)cn1
FC(F)(F)c1ccncc1Cn1cc(NC(=O)c2cc(on2)-c2ccncn2)cn1
Cc1cnccc1-c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
FC(F)(F)c1ccncc1Cn1cc(NC(=O)c2cc(on2)-c2ccncc2)cn1
CN(C)c1cc(no1)C(=O)Nc1cnn(Cc2ccccc2)c1
O=C(N1CCC1c1ccccc1)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CC(Cc2ccccc2)C1)c1cc(on1)-c1ccco1
O=C(N1CC(C1)Oc1ccccc1)c1cc(on1)-c1ccco1
O=C(N1CC(C1)c1ccccc1)c1cc(on1)-c1ccco1
O=C(N1CC(C1)Oc1ccccc1)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CC2(C1)CN(C2)c1ccccc1)c1cc(on1)-c1ccccc1
O=C(N1CC(C1)Nc1ccccc1)c1cc(on1)-c1ccco1
O=C(N1CC(Cc2ccccc2)C1)c1cc(on1)-c1ccccc1
O=C(N1CC(C1)c1ccccc1)c1cc(on1)-c1ccccc1
O=C(N1CC(C1)Oc1ccccc1)c1cc(on1)-c1ccccc1
O=C(N1CC(C1)Nc1ccccc1)c1cc(on1)-c1ccccc1
ClCC1(CNc2ccccc2)CN(C1)C(=O)c1cc(on1)-c1ccccc1
O=C(N1CC(Cc2ccccc2)C1)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CC(C1)c1ccccc1)c1cc(on1)-c1ccc2OCOc2c1
Fc1ccccc1C1CCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
Clc1ccccc1C1CCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
Fc1cccc(c1)C1CCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CC(C1)Nc1ccccc1)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CC2(C1)CN(C2)c1ccccc1)c1cc(on1)-c1ccc2OCOc2c1
Fc1ccc(cc1)C1CCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
OC1(CC2(CN(C2)C(=O)c2cc(on2)-c2ccc3OCOc3c2)C1)c1ccccc1
O=C(N1CC2(C1)CC(=C2)c1ccccc1)c1cc(on1)-c1ccccc1 |c:8|
OC1(CC2(CN(C2)C(=O)c2cc(on2)-c2ccccc2)C1)c1ccccc1
O=C(N1CC2(CC(C2)c2ccccc2)C1)c1cc(on1)-c1ccccc1
O=C(N1CC2(CC(C2)c2ccccc2)C1)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CC(C1)c1ccccc1)c1cc(on1)-c1ccncc1
CNC(=O)c1ccc(cc1)-c1cc(no1)C(=O)N1CC(Cc2ccccc2)C1
CNC(=O)c1ccc(cc1)-c1cc(no1)C(=O)N1CC(C1)c1ccccc1
Cn1ncc2ccc(cc12)-c1cc(no1)C(=O)N1CC(C1)c1ccccc1
O=C(N1CC(C1)c1ccccc1)c1cc(on1)-c1ccccn1
O=C(N1CC(C1)c1ccccc1)c1cc(on1)-c1cccnc1
Cn1cc2ccc(cc2n1)-c1cc(no1)C(=O)N1CC(C1)c1ccccc1
COc1ccc(cc1OC)-c1cc(no1)C(=O)N1CC(C1)c1cccc(F)c1
O=C(Nc1ccccc1)C1CN(C1)C(=O)c1cc(on1)-c1ccccc1
CC1(CN(C1)C(=O)c1cc(on1)-c1ccccc1)C(=O)Nc1ccccc1
Fc1cccc(c1)C1CN(C1)C(=O)c1cc(on1)-c1ccc2OCOc2c1
O=C(NC1CN(C1)C(=O)c1cc(on1)-c1ccccc1)c1ccccc1
Clc1ccc(nc1)-c1cc(no1)C(=O)N1CC(C1)c1ccccc1
COc1ccc(nc1)-c1cc(no1)C(=O)N1CC(C1)c1ccccc1
Fc1ccc(nc1)-c1cc(no1)C(=O)N1CC(C1)c1ccccc1
FC1CN(C1)C(=O)c1cc(on1)-c1ccco1
O=C(N1CC2(C1)CCCC2)c1cc(on1)-c1ccco1
O=C(N1CC2(CCC2)C1)c1cc(on1)-c1ccco1
O=C(N1CC2(COC2)C1)c1cc(on1)-c1ccco1
O=C(N1CC(C1)c1ccccc1)c1cc(on1)N1CCOCC1
COC1CCN(CC1)c1cc(no1)C(=O)N1CC(C1)c1ccccc1
CC(C)c1cc(no1)C(=O)N1CC(C1)c1ccccc1
CC(C)c1cc(no1)C(=O)N1CC(Cc2ccccc2)C1
O=C(N1CC(C1)c1ccccc1)c1noc2CCCCc12
O=C(N1CC(Cc2ccccc2)C1)c1noc2CCCCc12
Clc1ccc(nc1)-c1cc(no1)C(=O)N1CC(Cc2ccccc2)C1
COc1ccc(nn1)-c1cc(no1)C(=O)N1CC(C1)c1ccccc1
COc1ccc(nn1)-c1cc(no1)C(=O)N1CC(Cc2ccccc2)C1
O=C(N1CC(C1)c1ccccc1)c1cc(on1)-c1ccncn1
O=C(N1CC(Cc2ccccc2)C1)c1cc(on1)-c1ccncn1
O=C(N1CC(C1)c1ccccc1)c1cc(on1)-c1cnccn1
O=C(N1CCc2ccccc2C1)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCCc2ccccc12)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCOc2ccccc12)c1cc(on1)-c1ccc2OCOc2c1
Fc1cccc2N(CCCc12)C(=O)c1cc(on1)-c1ccc2OCOc2c1
Fc1cccc2CCCN(C(=O)c3cc(on3)-c3ccc4OCOc4c3)c12
O=C(N1CCN(CC1)c1ccccc1)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCN(CC1)c1ccccc1)c1cc(on1)-c1ccccc1
CC(C)(C)OC(=O)N1CCN(CC1)C(=O)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCn2ccnc2C1)c1cc(on1)-c1ccccc1
O=C(N1CCn2ccnc2C1)c1cc(on1)-c1ccc2OCOc2c1
CC1CN(CCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1)c1ccccc1
COc1cccc(c1)N1CCN(CC1)C(=O)c1cc(on1)-c1ccc2OCOc2c1
Fc1ccc(nc1)C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
Cc1nn(C)c2cc(ccc12)-c1cc(CN2C(COC2=O)c2ccccc2)no1
COc1ccc(cc1OC)-c1cc(no1)C(=O)N1CCN(CC1)c1ccccc1
O=C(N1CCC(CC1)c1ccccc1)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCN(CC1)C(=O)c1ccncc1)c1cc(on1)-c1ccc2OCOc2c1
Fc1ccccc1N1CCN(CC1)C(=O)c1cc(on1)-c1ccc2OCOc2c1
Cc1nn(C)c2cc(ccc12)-c1cc(no1)C(=O)N1CCN(CC1)c1ccccc1
Fc1ccc(cc1)N1CCN(CC1)C(=O)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCN(C(=O)C1)c1ccccc1)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCN(CC1)C(=O)c1ccccc1)c1cc(on1)-c1ccc2OCOc2c1
Fc1cccc(c1)N1CCN(CC1)C(=O)c1cc(on1)-c1ccc2OCOc2c1
Fc1ccc(cc1)N1CCN(CC1)C(=O)c1cc(on1)-c1ccccc1
Fc1ccccc1N1CCN(CC1)C(=O)c1cc(on1)-c1ccccc1
O=C(NC1CCN(Cc2ccccc2)CC1)c1cc(on1)-c1ccco1
O=C(NC1CCN(CC1)c1ccccc1)c1cc(on1)-c1ccco1
CC(C)(C)OC(=O)N1CCC(CC1)NC(=O)c1cc(on1)-c1ccco1
O=C(N1CCC(CC1)Oc1ccccc1)c1cc(on1)-c1ccccc1
FC(F)(F)c1ccccc1C1CCN(CC1)C(=O)c1cc(on1)-c1ccccc1
CC1(CCN(CC1)C(=O)c1cc(on1)-c1ccc2OCOc2c1)c1ccccc1
O=C(N1CCC(CC1)c1ccc(cc1)C#N)c1cc(on1)-c1ccc2OCOc2c1
Fc1ccc(cc1F)C1CCN(CC1)C(=O)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCC(CC1)c1ccncc1)c1cc(on1)-c1ccc2OCOc2c1
Fc1cccc(c1)N1CCN(CC1)C(=O)c1cc(on1)-c1ccccc1
CC(C)(C)OC(=O)N1CCC2(CCN(C2)C(=O)c2cc(on2)-c2ccccc2)C1
OC1(CCN(CC1)C(=O)c1cc(on1)-c1ccccc1)c1ccccc1
Fc1ccc(Cl)c(c1)N1CCN(CC1)C(=O)c1cc(on1)-c1ccccc1
O=C(N1CCC(CC1)Oc1ccccc1)c1cc(on1)-c1ccc2OCOc2c1
Fc1ccc(Cl)c(c1)N1CCN(CC1)C(=O)c1cc(on1)-c1ccc2OCOc2c1
OC1(CCN(CC1)C(=O)c1cc(on1)-c1ccc2OCOc2c1)c1ccccc1
CNC(=O)c1ccccc1-c1cc(no1)C(=O)N1CCC(CC1)c1ccccc1
FC(F)(F)c1ccccc1C1CCN(CC1)C(=O)c1cc(on1)-c1ccc2OCOc2c1
CNC(=O)c1cccc(c1)-c1cc(no1)C(=O)N1CCC(CC1)c1ccccc1
CNC(=O)c1ccc(cc1)-c1cc(no1)C(=O)N1CCC(CC1)c1ccccc1
Fc1ccc(Cl)c(c1)C1=CCN(CC1)C(=O)c1cc(on1)-c1ccccc1 |t:9|
Fc1ccc(Cl)c(c1)C1=CCN(CC1)C(=O)c1cc(on1)-c1ccc2OCOc2c1 |t:9|
Fc1cccc(c1)C1CCN(CC1)C(=O)c1cc(on1)-c1ccccc1
Fc1ccc(Cl)c(c1)C1CCN(CC1)C(=O)c1cc(on1)-c1ccc2OCOc2c1
Fc1cccc(c1)C1CCN(CC1)C(=O)c1cc(on1)-c1ccc2OCOc2c1
Fc1ccc(Cl)c(c1)C1CCN(CC1)C(=O)c1cc(on1)-c1ccccc1
O=C(Nc1cnnc(Oc2ccccc2)c1)c1cc(on1)-c1ccccc1
O=C(Nc1ccnc(Oc2ccccc2)c1)c1cc(on1)-c1ccccc1
O=C(N1CCC(CC1)c1ccccc1)c1cc(on1)-c1ccncc1
O=C(N1CCC(CC1)c1ccccc1)c1cc(on1)-c1ccccc1
O=C(N1CCC(CC1)c1ccccc1)c1cc(on1)-c1cccnc1
O=C(N1CCC(CC1)c1ccccc1)c1cc(on1)-c1ccc(cc1)C#N
O=C(N1CCC(CC1)c1ccccc1)c1cc(on1)-c1cccc(c1)C#N
O=C(N1CCC(CC1)c1ccccc1)c1cc(on1)-c1ccccn1
CNC(=O)c1ccc(cc1)-c1cc(no1)C(=O)N1CCC(=CC1)c1ccccc1 |c:22|
COc1ccccc1-c1cc(no1)C(=O)N1CCC(CC1)c1ccccc1
CNC(=O)c1ccc(cc1)-c1cc(no1)C(=O)N1CCC(F)(CC1)c1ccccc1
O=C(N1CCC(CC1)c1cccnc1)c1cc(on1)-c1ccccc1
COC1(CCN(CC1)C(=O)c1cc(on1)-c1ccccc1)c1ccccc1
CC(=C)c1cc(no1)C(=O)N1CCC2(CC1)CCc1c(F)cccc1O2
Fc1cc(ccc1-c1cc(no1)C(=O)N1CCC(CC1)c1ccccc1)C#N
O=C(N1CCC(CC1)c1ccccc1)c1cc(on1)-c1ccccc1C#N
O=C(N1CCC[C@H]1c1ccccc1)c1cc(on1)-c1ccc2OCOc2c1 |r|
O=C(N1Cc2ccccc2C1)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCC(C1)c1ccccc1)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCC(C1)c1ccccc1)c1cc(on1)-c1ccccc1
FC(F)c1ccccc1C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
CC(C)(C)OC(=O)N1CCC(C1)NC(=O)c1cc(on1)-c1ccco1
Clc1ccccc1-c1cc(no1)C(=O)N1CCC(C1)c1ccccc1
Fc1ccc(cc1)C1CCN(C1)C(=O)c1cc(on1)-c1ccccc1
Fc1ccccc1C1CCN(C1)C(=O)c1cc(on1)-c1ccccc1
O=C(NC1CCNC1)c1cc(on1)-c1ccco1
O=C(NC1CCN(Cc2ccccc2)C1)c1cc(on1)-c1ccco1
O=C(N1CCC(C1)c1ccccc1)c1cc(on1)-c1ccco1
Fc1cccc(c1)C1CCN(C1)C(=O)c1cc(on1)-c1ccccc1
O=C(N1CCC2(CCNC2)C1)c1cc(on1)-c1ccccc1
O=C(N1CCC2(CCN(C2)c2ccccc2)C1)c1cc(on1)-c1ccccc1
CN1CCC2(CCN(C2)C(=O)c2cc(on2)-c2ccccc2)C1
O=C(NC1CCN(C1)c1ccccc1)c1cc(on1)-c1ccco1
CC(C)(C)OC(=O)N1CC2(C1)CN(C2)C(=O)c1cc(on1)-c1ccccc1
O=C(N1CC2(CNC2)C1)c1cc(on1)-c1ccccc1
FC(F)(F)c1ccccc1-c1cc(no1)C(=O)N1CCC(C1)c1ccccc1
CNC(=O)c1cc(no1)C(=O)N1CCC(C1)c1ccccc1
NC(=O)c1cc(no1)C(=O)N1CCC(C1)c1ccccc1
CC(C)c1cc(no1)C(=O)N1CCC(C1)c1ccccc1
CC(C)c1cc(no1)C(=O)N1CCC(C1)c1cccc(F)c1
O=C(N1CCC(C1)c1ccccc1)c1cc(on1)-c1ccccn1
Fc1cccc(c1)C1CCN(C1)C(=O)c1cc(on1)-c1ccccn1
Cc1cc(on1)C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCCC1c1ccccc1)c1cc(on1)-c1ccc2OCOc2c1
Cc1cccc(c1)C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
COc1ccc(cc1)C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
Cc1cc(on1)C1CCCN1C(=O)c1cc(on1)-c1ccco1
O=C(N1CCC[C@@H]1c1ccccc1)c1cc(on1)-c1ccc2OCOc2c1 |r|
COc1ccc(cc1)[C@@H]1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1 |r|
COc1ccc(cc1)[C@H]1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1 |r|
O=C(N1CCCC1c1ccccn1)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCCC1c1cccnc1)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCCC1c1ccncc1)c1cc(on1)-c1ccc2OCOc2c1
COc1ccccc1C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
COc1cccc(c1)C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
Fc1ccccc1C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
Fc1cccc(c1)C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
Fc1ccc(cc1)C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
C[C@H]1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1 |r|
C[C@@H]1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1 |r|
O=C(N1CCCC11CC1)c1cc(on1)-c1ccc2OCOc2c1
FC(F)(F)[C@H]1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1 |r|
FC(F)(F)[C@@H]1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1 |r|
COc1ccc(cc1)C1CCCN1C(=O)c1cc(on1)-c1ccc(OC)c(OC)c1
COc1ccc(cc1)C1CCCN1C(=O)c1cc(on1)-c1cccc(OC)c1
COc1ccc(cc1)C1CCCN1C(=O)c1cc(on1)-c1ccc(OC)cc1
COc1ccc(cc1)C1CCCN1C(=O)c1cc(on1)-c1ccccc1
COc1ccc(cc1)C1CCCN1C(=O)c1cc(on1)-c1ccc(F)c(F)c1
COc1ccc(cc1)C1CCCN1C(=O)c1cc(on1)-c1ccccc1OC
COc1ccc(cc1)C1CCCN1C(=O)c1cc(on1)-c1ccc(OC(F)(F)F)cc1
COc1ccc(cc1)C1CCCN1C(=O)c1cc(on1)-c1ccc(cc1)C(F)(F)F
COc1ccc(cc1)C1CCCN1C(=O)c1cc(on1)-c1ccc(OC)c(F)c1
COc1ccc(cc1)C1CCCN1C(=O)c1cc(on1)-c1ccc(F)c(OC)c1
O=C(N1CCCC1c1ccccc1)c1cc(CC2CC2)on1
O=C(N1CCC[C@@H]1c1ccccc1)c1cc(on1)-c1ccccc1 |r|
O=C(N1CCC[C@H]1c1ccccc1)c1cc(on1)-c1ccccc1 |r|
O=C(N1CCCC1c1ccccc1)c1cc(on1)-c1ccccc1
Brc1cccc(c1)C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
Brc1ccc(cc1)C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
Brc1ccccc1C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCCC1c1cccnn1)c1cc(on1)-c1ccc2OCOc2c1
COc1ccc(cc1)C1CCCN1C(=O)c1cc(on1)-c1ccc(cc1)C(F)(F)C(F)(F)F
COc1ccc(cc1)C1CCCN1C(=O)c1cc(on1)-c1ccc2OC(F)(F)Oc2c1
COc1ccc(cc1)C1CCCN1C(=O)c1cc(on1)-c1ccc2c(C)nn(C)c2c1
O=C(N1CCCC1c1ccc(cc1)C#N)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCCC1c1cccc(c1)C#N)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCOCC1c1ccccc1)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCCC1c1ccccc1C#N)c1cc(on1)-c1ccc2OCOc2c1
COc1ccc(cc1)C1CCCN1C(=O)c1cc(on1)-c1ccc2nc(oc2c1)N(C)C
COc1ccc(cc1)C1CCCN1C(=O)c1cc(on1)-c1ccc2ocnc2c1
COc1ccc(cc1)C1CCCN1C(=O)c1cc(on1)-c1ccc2ncoc2c1
O=C(N1CCC[C@H]1c1ccccc1)c1cc(on1)-c1ccccc1C#N |r|
O=C(N1CCC[C@H]1c1ccccc1)c1cc(on1)-c1cccc(c1)C#N |r|
O=C(N1CCC[C@H]1c1ccccc1)c1cc(on1)-c1ccc(cc1)C#N |r|
O=C(N1CCC[C@H]1c1ccccc1)c1cc(on1)-c1cccnc1 |r|
O=C(N1COCC1c1ccccc1)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCCC1C1CC1)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCC[C@H]1c1ccccc1)c1cc(on1)-c1ccccn1 |r|
O=C(N1CCC[C@H]1c1ccccc1)c1cc(on1)-c1ccncc1 |r|
COc1ccc(cn1)-c1cc(no1)C(=O)N1CCC[C@H]1c1ccccc1 |r|
COc1cc(on1)C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
Brc1cc(on1)C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCCC1C1CCOCC1)c1cc(on1)-c1ccc2OCOc2c1
OC1C[C@H](N(C1)C(=O)c1cc(on1)-c1ccc2OCOc2c1)c1ccccc1 |r|
COc1ccc(nc1)-c1cc(no1)C(=O)N1CCCC1c1ccccc1F
COc1ccc(nc1)-c1cc(no1)C(=O)N1CCC[C@H]1c1ccccc1 |r|
Cn1nccc1C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCCC1c1cnccn1)c1cc(on1)-c1ccc2OCOc2c1
Cc1nn(C)c2cc(ccc12)-c1cc(no1)C(=O)N1COCC1c1ccccc1
F[C@@H]1C[C@H](N(C1)C(=O)c1cc(on1)-c1ccc2OCOc2c1)c1ccccc1 |r|
O[C@H]1C[C@H](N(C1)C(=O)c1cc(on1)-c1ccc2OCOc2c1)c1ccccc1 |r|
O[C@@H]1C[C@H](N(C1)C(=O)c1cc(on1)-c1ccc2OCOc2c1)c1ccccc1 |r|
O=C(N1CCCC1c1ncco1)c1cc(on1)-c1ccc2OCOc2c1
CN1CCC(CC1)C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
Cn1ncc2cccc(C3CCCN3C(=O)c3cc(on3)-c3ccc4OCOc4c3)c12
O=C(N1CCC[C@H]1c1ccon1)c1cc(on1)-c1ccc2OCOc2c1 |r|
F[C@H]1C[C@H](N(C1)C(=O)c1cc(on1)-c1ccc2OCOc2c1)c1ccccc1 |r|
Cn1ccc(cc1=O)-c1cc(no1)C(=O)N1CCC[C@H]1c1ccccc1 |r|
Cn1cc(ccc1=O)-c1cc(no1)C(=O)N1CCC[C@H]1c1ccccc1 |r|
COc1cc(F)ccc1C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCCC1c1ncccn1)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCC[C@H]1c1ccccc1)c1cc(on1)-c1ccn2ncnc2c1 |r|
O=C(N1CCC[C@H]1c1ccccc1)c1cc(on1)-c1ccnnc1 |r|
O=C(N1CCCC1Cc1ccccc1)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCC[C@H]1c1ccccc1)c1cc(on1)-c1ccc(cn1)C#N |r|
O=C(N1CCCC1Cc1ccccc1)c1cc(on1)-c1ccccc1
COc1cccnc1C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCC[C@H]1c1ccccc1)c1noc2ccccc12 |r|
Cc1cnoc1C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCCC1c1ccncn1)c1cc(on1)-c1ccc2OCCc2c1
O=C(N1CCC[C@H]1c1ccccc1)c1cc(on1)-c1ccc2ncnn2c1 |r|
Cc1cc(no1)C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
CCOc1ccc(cc1F)-c1cc(no1)C(=O)N1CCC[C@H]1c1ccccc1 |r|
Cn1c2cc(ccc2oc1=O)-c1cc(no1)C(=O)N1CCC[C@H]1c1ccccc1 |r|
COc1ccc(cc1)-c1cc(NC(=O)[C@@H]2CCCN2c2ccccc2)on1 |r|
Cn1ccnc1C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
Brc1cccnc1C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCCC1c1ncccc1C#N)c1cc(on1)-c1ccc2OCOc2c1
Brc1ccc2c(noc2c1)C(=O)N1CCC[C@H]1c1ccccc1 |r|
O=C(N1CCC[C@H]1c1ccccc1)c1cc(on1)-c1ccc2nccnc2c1 |r|
O=C(N1CCC[C@H]1c1ccccc1)c1cc(on1)-c1ccc(=O)[nH]c1 |r|
COc1ccc(C2CCCN2C(=O)c2cc(on2)-c2ccc3OCOc3c2)c(F)c1
COc1cccc(F)c1C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
Cn1nccc1-c1ccc2c(noc2c1)C(=O)N1CCC[C@H]1c1ccccc1 |r|
O=C(Nc1ccccc1)C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCC[C@H]1c1ccccc1)c1noc2cc(ccc12)C#N |r|
Fc1cccnc1C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
Cc1nn(C)c2cc(ccc12)-c1cc(no1)C(=O)N1CCCC1c1ccnnc1
Fc1c(Br)nccc1C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
Fc1cnccc1C1CCCN1C(=O)c1cc(on1)-c1ccc2OCOc2c1
O=C(N1CCCC1c1nc2ccccc2o1)c1cc(on1)-c1ccc2OCOc2c1
Cc1nn(C)c2cc(ccc12)-c1cc(no1)C(=O)N1CCCC1c1cccnn1
O=C(N1CCC[C@H]1c1ccccc1)c1cc(on1)N1CCOCC1 |r|
Cc1nn(C)c2cc(ccc12)-c1conc1CN1C(COC1=O)c1ccccc1
Cn1nc(NC(=O)N2CC[C@@H](Oc3ccc(F)c(F)c3)C2)ccc1=O
Cn1nc(NC(=O)N2CCC(Cc3cc(F)ccc3F)CC2)ccc1=O
Cn1nc(NC(=O)N2CC[C@@H](Oc3cc(F)cc(F)c3)C2)ccc1=O
Cn1nc(NC(=O)N2CCC(Oc3cc(F)c(F)c(Cl)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CC[C@H](Oc3ccc(F)c(F)c3)C2)ccc1=O
Cn1nc(NC(=O)N2CCC(Oc3cc(F)c(F)c(C#N)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CC[C@H](Oc3cc(F)cc(F)c3)C2)ccc1=O
Cn1nc(NC(=O)N2CCC(Oc3ccc(Cl)cc3)CC2)ccc1=O
Cn1nc(NC(=O)N2CC(Oc3ccc(F)c(F)c3)C2)ccc1=O
Cn1nc(NC(=O)N2CCC(Oc3cccc(Cl)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CC(Oc3cc(F)cc(F)c3)C2)ccc1=O
Cn1nc(NC(=O)N2CCC(Cc3cc(F)c(F)c(F)c3)CC2)ccc1=O
Cn1cc(CC(=O)N2CCC(Oc3cccc(Cl)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Cc3ccc(Cl)c(F)c3)CC2)ccc1=O
Cn1nc(CC(=O)N2CCC(Oc3cccc(Cl)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Cc3ccc(F)cc3)CC2)ccc1=O
Clc1cccc(OC2CCNCC2)c1
CCn1nc(NC(=O)N2CCC(Cc3cc(F)cc(F)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Oc3cccc(Cl)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(F)(Cc3cccc(F)c3)CC2)ccc1=O
Cn1cc(OC(=O)N2CCC(Oc3cccc(Cl)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(F)(Cc3cc(F)cc(F)c3)CC2)ccc1=O
Cn1nc(OC(=O)N2CCC(Oc3cccc(Cl)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC=C(c3ccc(Cl)cc3)CC2)ccc1=O
Cn1cc(CC(=O)N2CCC(Cc3cccc(Cl)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CC=C(c3ccc(Cl)cc3)CCC2)ccc1=O
Cn1nc(CC(=O)N2CCC(Cc3cccc(Cl)c3)CC2)ccc1=O
O=C(Cc1ccc(=O)[nH]n1)N1CCC(Oc2cccc(Cl)c2)CC1
Cn1cc(NC(=O)N2CCC(Cc3cccc(Cl)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Oc3cc(F)ccc3Cl)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Cc3cccc(Cl)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Oc3ccc(F)cc3Cl)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Cc3cc(F)cc(Cl)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(COc3cccc(F)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Cc3cc(F)cc(F)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(OCc3cccc(F)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Cc3ccc(F)c(F)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(COc3ccccc3F)CC2)ccc1=O
Cn1cc(NC(=O)N2CCC(Cc3cc(F)cc(Cl)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(OCc3ccccc3F)CC2)ccc1=O
Cn1cc(NC(=O)N2CCC(Cc3cc(F)cc(F)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Oc3cccc(F)c3C(F)(F)F)CC2)ccc1=O
Cn1cc(NC(=O)N2CCC(Cc3ccc(F)c(F)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Oc3ccc(F)cc3C(F)(F)F)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Oc3ccccc3Cl)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Oc3cc(F)ccc3C(F)(F)F)CC2)ccc1=O
Cn1nc(NC(=O)C2CCN(Cc3cccc(Cl)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(COc3ccccc3Cl)CC2)ccc1=O
Cn1nc(NC(=O)N2CCN(Cc3cccc(Cl)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(COc3ccccc3C(F)(F)F)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Oc3cc(F)cc(F)c3)CC2)ccc1=O
Cn1cc(NC(=O)N2CCC(Cc3cc(F)cc(F)c3)CC2)ncc1=O
Cn1nc(NC(=O)N2CCC(Oc3ccc(F)c(F)c3)CC2)ccc1=O
Cn1cc(NC(=O)N2CCC(Cc3ccc(F)c(F)c3)CC2)ncc1=O
Cn1nc(NC(=O)N2CCC(Cc3ccc(F)c(C#N)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Cc3cc(Cl)cc(C#N)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Cc3cc(F)cc(C#N)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Oc3cccc(Cl)c3F)CC2)ccc1=O
Cn1nc(OC(=O)N2CCC(Cc3cc(F)cc(F)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Oc3cccc(C(F)(F)F)c3)CC2)ccc1=O
Cn1cc(OC(=O)N2CCC(Oc3cc(F)cc(F)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Oc3ccc(C(F)(F)F)cc3)CC2)ccc1=O
O=CN1CCC(Oc2cc(F)cc(F)c2)CC1
Cn1nc(NC(=O)N2CCC(Oc3cccc(C#N)c3Cl)CC2)ccc1=O
Cn1nc(OC(=O)N2CCC(Oc3ccc(F)c(F)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Cc3cccc(C#N)c3Cl)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(=Cc3cc(F)cc(F)c3)CC2)ccc1=O
Cn1cc(-c2nc(N3CCC(Oc4cc(F)cc(F)c4)CC3)no2)ccc1=O
Cn1nc(NC(=O)N2CCC(Cc3cccc(F)c3)CC2)ccc1=O
Cn1nc(-c2nc(N3CCC(Oc4cc(F)cc(F)c4)CC3)no2)ccc1=O
Cn1nc(NC(=O)N2CCC(Cc3cccc(Cl)c3)C2)ccc1=O
Cn1nc(-c2nc(N3CCC(Cc4cc(Cl)cc(C#N)c4)CC3)no2)ccc1=O
Cn1nc(NC(=O)N2CCC(Cc3cc(F)cc(F)c3)C2)ccc1=O
Cn1cc(-c2nc(N3CCC(Oc4cccc(F)c4Cl)CC3)no2)ccc1=O
Cn1cc(NC(=O)N2CCC(Cc3cc(F)cc(F)c3)C2)ccc1=O
Cn1nc(-c2nc(N3CCC(Oc4cccc(F)c4Cl)CC3)no2)ccc1=O
Cn1nc(NC(=O)N2CC3C(Cc4ccc(F)cc4)C3C2)ccc1=O
Cn1nc(-c2noc(N3CCC(Cc4ccc(F)c(F)c4)CC3)n2)ccc1=O
Cn1nc(NC(=O)N2CCC[C@@H](c3ccc(Cl)cc3)CC2)ccc1=O
Cn1cc(-c2noc(N3CCC(Cc4ccc(F)c(F)c4)CC3)n2)ccc1=O
Cn1nc(NC(=O)N2CCC[C@@H](c3cc(F)cc(F)c3)CC2)ccc1=O
Cn1cc(-c2noc(N3CCC(Cc4cc(F)cc(F)c4)CC3)n2)ccc1=O
Cn1nc(NC(=O)N2CC(Cc3cccc(Cl)c3)C2)ccc1=O
Cn1nc(-c2cnc(N3CCC(Cc4cc(F)cc(F)c4)CC3)o2)ccc1=O
Cn1nc(-c2nc(N3CCC(Cc4cccc(F)c4)CC3)no2)ccc1=O
Cn1nc(-c2nc(N3CCC(Cc4cccc(F)c4)CC3)no2)ccc1=O
Cn1nc(-c2noc(N3CCC(Cc4cc(F)cc(F)c4)CC3)n2)ccc1=O
Cn1cc(-c2nnc(N3CCC(Cc4cc(F)cc(F)c4)CC3)o2)ccc1=O
Cn1nc(-c2nc(N3CCC(Cc4ccccc4)CC3)no2)ccc1=O
Cn1nc(-c2nnc(N3CCC(Cc4cc(F)cc(F)c4)CC3)o2)ccc1=O
Cn1nc(-c2nc(N3CCC(Cc4ccc(F)c(F)c4)CC3)no2)ccc1=O
Cn1nc(-c2nnc(N3CCC(Cc4cc(F)cc(F)c4)CC3)s2)ccc1=O
Cn1cc(-c2nc(N3CCC(Cc4cc(F)cc(F)c4)CC3)no2)ccc1=O
Cn1nc(-c2nnc(N3CCC(Cc4cccc(F)c4)CC3)o2)ccc1=O
Cn1nc(CC(=O)N2CCC(Cc3cc(F)cc(F)c3)CC2)ccc1=O
Cn1cc(-c2nnc(N3CCC(Cc4cccc(F)c4)CC3)o2)ccc1=O
Cc1cc(NC(=O)N2CCC(Cc3cc(F)cc(F)c3)CC2)nn(C)c1=O
O=C(Cc1ccc(=O)[nH]n1)N1CCC(Cc2cccc(Cl)c2)CC1
Cc1cc(NC(=O)N2CCC(Cc3ccc(F)c(F)c3)CC2)nn(C)c1=O
O=C(Cc1ccc(=O)[nH]n1)N1CCC(Cc2cc(F)cc(F)c2)CC1
Cc1cc(NC(=O)N2CCC(Oc3cc(F)cc(F)c3)CC2)nn(C)c1=O
Cn1nc(NC(=O)N2CCC(Oc3ccc(C(F)(F)F)c(F)c3)CC2)ccc1=O
Cc1cc(NC(=O)N2CCC(Oc3ccc(F)c(F)c3)CC2)nn(C)c1=O
Cn1nc(NC(=O)N2CCC(F)(Cc3ccc(F)c(F)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Oc3cccc(Cl)c3Cl)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(F)(Cc3cccc(Cl)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Oc3cccc(F)c3Cl)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(F)(Cc3cc(F)c(F)c(Cl)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Oc3ccccc3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(O)(Cc3cccc(F)c3)CC2)ccc1=O
Cc1ccccc1OC1CCN(C(=O)Nc2ccc(=O)n(C)n2)CC1
COC1(Cc2cccc(F)c2)CCN(C(=O)Nc2ccc(=O)n(C)n2)CC1
Cn1nc(NC(=O)N2CCC(Oc3ccccc3C(F)(F)F)CC2)ccc1=O
O=c1ccc(-c2noc(N3CCC(Cc4ccc(F)c(F)c4)CC3)n2)c[nH]1
COc1ccccc1OC1CCN(C(=O)Nc2ccc(=O)n(C)n2)CC1
O=c1ccc(-c2noc(N3CCC(Cc4cc(F)cc(F)c4)CC3)n2)c[nH]1
Cn1nc(NC(=O)N2CCC(Cc3ccc(F)c(Cl)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Nc3cc(F)cc(F)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Cc3cc(F)c(F)c(Cl)c3)CC2)ccc1=O
CN(c1cc(F)cc(F)c1)C1CCN(C(=O)Nc2ccc(=O)n(C)n2)CC1
Cn1nc(NC(=O)N2CCC(Cc3cc(F)c(F)c(C#N)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Nc3cc(F)cc(Cl)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Cc3ccccc3Cl)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Nc3ccccc3C(F)(F)F)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Cc3ccc(Cl)cc3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Nc3ccccc3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Cc3cc(F)cc(F)c3Cl)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(NCc3cc(F)cc(F)c3)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(Cc3cc(F)c(F)cc3Cl)CC2)ccc1=O
Cn1cc(NC(=O)N2CCC(Nc3cc(F)cc(F)c3)CC2)ccc1=O
Cn1cc(NC(=O)N2CCC(Cc3cc(F)ccc3F)CC2)ccc1=O
Cn1nc(NC(=O)N2CCC(NCc3ccccc3C(F)(F)F)CC2)ccc1=O
Cc1ccccc1S(=O)(=O)N1CCN(CC1)c1ccc(nn1)C(=O)NCc1ccccc1
Cc1nnc(o1)-c1ccc(nn1)N1CCC(CC1)Oc1cc(F)ccc1Cl
FC(F)(F)c1ccccc1C(=O)N1CCN(CC1)c1ccc(nn1)C(=O)NCc1ccccc1
COC1(CCN(CC1)c1ccc(nn1)-c1nc(CO)no1)c1ccccc1
CC(C)(C)c1ccc(cc1)C1(CCN(CC1)c1ccc(nn1)-c1nc(CO)no1)C#N
OCc1noc(n1)-c1ccc(nn1)N1CCC(CC1)(C#N)c1ccc(cc1)[N+]([O-])=O
OCc1noc(n1)-c1ccc(nn1)N1CCC(O)(CC1)c1ccccc1
NC1(CCN(CC1)c1ccc(nn1)-c1nc(CO)no1)c1ccccc1
OCc1noc(n1)-c1ccc(nn1)N1CCC(CC1)(C#N)c1ccccc1
OCc1nsc(n1)-c1ccc(nn1)N1CCC(CC1)(c1ccc(cc1)C(F)(F)F)C(F)(F)F
OCc1nnc(o1)-c1ccc(nn1)N1CCC(CC1)(c1ccc(cc1)C(F)(F)F)C(F)(F)F
OCc1noc(n1)-c1ccc(nn1)N1CCC(CC1)(c1ccc(cc1)C(F)(F)F)C(F)(F)F
OCc1noc(n1)-c1ccc(nn1)N1CCC(CC1)(C#N)c1ccc(cc1)S(F)(F)(F)(F)F
OCc1noc(n1)-c1ccc(nn1)N1CCC(CC1)(C#N)c1ccc(cc1)C(F)(F)F
OCc1noc(n1)-c1ccc(nn1)N1CCC(CC1)(C#N)c1ccc(OC(F)(F)F)cc1
OCc1noc(n1)-c1ccc(nn1)N1CCC(CC1)(C#N)c1ccc(Cl)cc1
OCc1noc(n1)-c1ccc(nn1)N1CCC(CC1)(C#N)c1cccc(Cl)c1
OCc1noc(n1)-c1ccc(nn1)N1CCC(CC1)(C#N)c1ccccc1Cl
OCc1noc(n1)-c1ccc(nn1)N1CCC(CC1)(c1ccccc1)C(F)(F)F
OCc1nnc(s1)-c1ccc(nn1)N1CCC(CC1)(c1ccc(cc1)C(F)(F)F)C(F)(F)F
OCc1noc(n1)-c1ccc(nn1)N1CCC2(COc3ccccc23)C1
OCCc1csc(NC(=O)c2ccc(CNc3ccccc3C(F)(F)F)s2)n1
OCCc1cnc(NC(=O)c2ccc(CNc3ccccc3C(F)(F)F)cc2)s1
OC(=O)Cc1csc(NC(=O)c2ccc(CNc3ccccc3C(F)(F)F)cc2)n1
Cc1csc(NC(=O)c2ccc(CNc3cccc(Cl)c3)cc2)n1
CCCCCCc1ccccc1NCc1ccc(cc1)C(=O)Nc1nc(CC(O)=O)cs1
OCCCc1csc(NC(=O)c2ccc(CNc3ccccc3C(F)(F)F)cc2)n1
Cc1csc(NC(=O)c2ccc(CNc3ccccc3C(O)=O)cc2)n1
CCCCCCc1ccccc1NCc1ccc(s1)C(=O)Nc1nc(CCO)cs1
CCCCc1ccccc1NCc1ccc(cc1)C(=O)Nc1nc(CC(O)=O)cs1
OCCCc1nc(NC(=O)c2ccc(CNc3ccccc3C(F)(F)F)cc2)sc1CCO
OC(=O)c1cnc(NC(=O)c2ccc(CNc3ccccc3C(F)(F)F)cc2)s1
CCCc1ccccc1NCc1ccc(cc1)C(=O)Nc1nc(C)cs1
Cc1csc(NC(=O)c2ccc(COc3ccccc3Cl)cc2)n1
OC(=O)Cc1csc(NC(=O)c2ccc(CNc3ccccc3C(F)(F)F)s2)n1
Cc1csc(NC(=O)c2ccc(CNc3ccccc3C)cc2)n1
CC(C)CCc1ccccc1NCc1ccc(cc1)C(=O)Nc1nc(CCO)cs1
CCCCc1ccccc1NCc1ccc(cc1)C(=O)Nc1nc(CCO)cs1
OCCc1csc(NC(=O)c2ccc(CNc3ccccc3Cl)cc2)n1
OCc1csc(NC(=O)c2ccc(CNc3ccccc3Cl)cc2)n1
OCc1nc(NC(=O)c2ccc(CNc3ccccc3C(F)(F)F)cc2)sc1C(O)=O
OCc1cnc(NC(=O)c2ccc(CNc3ccccc3C(F)(F)F)cc2)s1
OC(=O)CCc1cnc(NC(=O)c2ccc(CNc3ccccc3C(F)(F)F)cc2)s1
OC(=O)Cc1cnc(NC(=O)c2ccc(CNc3ccccc3C(F)(F)F)cc2)s1
OCc1csc(NC(=O)c2ccc(CNc3ccccc3C(F)(F)F)cc2)n1
OC(=O)CCCc1csc(NC(=O)c2ccc(CNc3ccccc3C(F)(F)F)cc2)n1
OC(=O)CCc1csc(NC(=O)c2ccc(CNc3ccccc3C(F)(F)F)cc2)n1
Cc1csc(NC(=O)c2ccc(CNc3ccccc3C(F)(F)F)s2)n1
Cc1csc(NC(=O)N2CCC(CNc3ccccc3C(F)(F)F)CC2)n1
Cc1csc(NC(=O)c2ccc(CNc3ccccc3C)cn2)n1
COC(=O)c1ccccc1NCc1ccc(cc1)C(=O)Nc1nc(C)cs1
Cc1csc(NC(=O)c2ccc(CNc3ccc(Cl)cc3)cc2)n1
Cc1csc(NC(=O)c2ccc(CNc3ccccc3)cc2)n1
Cc1csc(NC(=O)c2ccc(CNc3ccccc3Cl)cc2)n1
Clc1ccccc1OCc1ccc(cc1)C(=O)Nc1ccncc1
OC(=O)Cc1csc(NC(=O)c2ccc(CNc3ccccc3-c3ccccc3)cc2)n1
OC(=O)Cc1csc(NC(=O)c2ccc(CNc3ccccc3Cc3ccccc3)cc2)n1
CCCCc1ccccc1NCc1ccc(s1)C(=O)Nc1nc(CC(O)=O)cs1
CCCCCCc1ccccc1NCc1ccc(s1)C(=O)Nc1nc(CC(O)=O)cs1
CCCCCCCCc1ccccc1NCc1ccc(s1)C(=O)Nc1nc(CC(O)=O)cs1
OC(=O)Cc1csc(NC(=O)c2ccc(CNc3ccccc3Cc3ccccc3)s2)n1
CCCCCCCCc1ccccc1NCc1ccc(cc1)C(=O)Nc1nc(CC(O)=O)cs1
CCCCc1ccccc1NCc1ccc(cc1)C(=O)Nc1nc(CO)cs1
OCCCc1cnc(NC(=O)c2ccc(CNc3ccccc3C(F)(F)F)cc2)s1
OCCc1csc(NC(=O)c2ccc(CNc3ccccc3C(F)(F)F)cc2)n1
Cc1ccccc1NCc1ccc(cc1)C(=O)Nc1nc(CC(O)=O)cs1
Cc1csc(NC(=O)c2ccc(CNc3ccccc3C)nc2)n1
Cc1csc(NC(=O)c2ccc(CNc3ccccc3C(F)(F)F)cc2)n1
CC(C)CCc1ccccc1NCc1ccc(cc1)C(=O)Nc1nc(CC(O)=O)cs1
OCc1csc(NC(=O)c2ccc(CNc3ccccc3C(F)(F)F)s2)n1
CC(C)CCc1ccccc1NCc1ccc(s1)C(=O)Nc1nc(CC(O)=O)cs1
OC(=O)Cc1csc(NC(=O)c2ccc(CNc3ccccc3Cl)cc2)n1
Cc1ccccc1NCc1ccc(cc1)C(=O)Nc1nc(cs1)C(O)=O
N[C@H](c1ccccc1)c1ccc(cc1)C(=O)Nc1nc2ccc(O)cc2s1 |r|
N[C@H](c1ccccc1)c1ccc(cc1)C(=O)Nc1nc2ccccc2s1 |r|
COc1ccc2nc(NC(=O)c3ccc(cc3)[C@H](N)c3ccccc3)sc2c1 |r|
COc1ccc2nc(NC(=O)c3ccc(N)cc3)sc2c1
COc1ccc2nc(NC(=O)c3ccccc3)sc2c1
COc1ccc(cc1)C(=O)Nc1nc2ccc(OC)cc2s1
COc1cccc(c1)C(=O)Nc1nc2ccc(OC)cc2s1
COc1ccc2nc(NC(=O)c3ccc(F)cc3)sc2c1
COc1ccc2nc(NC(=O)c3ccc(cc3)[N+]([O-])=O)sc2c1
COc1ccc2nc(NC(=O)c3ccc(OCc4ccccc4)cc3)sc2c1
COc1ccc2nc(NC(=O)c3ccc(Nc4ccccc4)cc3)sc2c1
COc1ccc2nc(NC(=O)c3ccc(cc3)C(=O)c3ccccc3)sc2c1
COc1ccc2nc(NC(=O)c3ccc(cc3)N=[N+]=[N-])sc2c1
COc1ccc2nc(NC(=O)c3cccc(C)c3)sc2c1
COc1ccc2nc(NC(=O)c3cccnc3)sc2c1
COc1ccc2nc(NC(=O)c3ccc(cc3)C(=O)N3CCN(C)CC3)sc2c1
COc1ccc2nc(NC(=O)c3ccc(cc3)C(=O)N3CCOCC3)sc2c1
COc1ccc2nc(NC(=O)c3ccc(cc3)C(=O)N3CCCCC3)sc2c1
COc1ccc2nc(NC(=O)c3ccc(cc3)C(=O)NCc3ccccc3)sc2c1
COc1ccc2nc(NC(=O)c3ccc(cc3)C(O)c3ccccn3)sc2c1
COc1ccc2nc(NC(=O)c3ccc(cc3)C(=O)c3ccccn3)sc2c1
COc1ccc2nc(NC(=O)c3ccc(cc3)C(=O)c3cccnc3)sc2c1
COc1ccc2nc(NC(=O)c3ccc(cc3)[C@@H](N)c3ccccc3)sc2c1 |r|
COc1ccc2nc(NC(=O)c3ccc(cc3)C(N)c3ccccc3)sc2c1
[O-][N+](=O)c1ccc(cc1)C(=O)Nc1nc2ccccc2s1
O=C(Nc1nc2ccccc2s1)c1ccc(cc1)-c1ccccc1
COc1ccc(cc1)C(=O)Nc1nc2ccccc2s1
Cc1cccc(c1)C(=O)Nc1nc2ccccc2s1
O=C(Nc1nc2ccccc2s1)c1cccnc1
O=C(Nc1nc2ccccc2s1)c1ccc(cc1)C(=O)c1ccccc1
O=C(Nc1nc2ccccc2[nH]1)c1ccc(cc1)C(=O)c1ccccc1
O=C(Nc1nc2ccccc2o1)c1ccc(cc1)C(=O)c1ccccc1
O=C(Nc1nccs1)c1ccc(cc1)C(=O)c1ccccc1
O=C(Nc1ncc(s1)-c1ccccc1)c1ccc(cc1)C(=O)c1ccccc1
O=C(Nc1nc(cs1)-c1ccccc1)c1ccc(cc1)C(=O)c1ccccc1
COc1ccc(cc1)C(=O)Nc1nc2cc(N)ccc2s1
COc1ccc2sc(NC(=O)c3ccc(cc3)[N+]([O-])=O)nc2c1
CCCOc1ccc2nc(NC(=O)c3ccc(cc3)C(=O)c3ccccc3)sc2c1
BrCCOc1ccc2nc(NC(=O)c3ccc(cc3)C(=O)c3ccccc3)sc2c1
COc1cc2sc(NC(=O)c3ccc(cc3)C(=O)c3ccccc3)nc2cc1Br
COC(=O)c1ccc2nc(NC(=O)c3ccc(cc3)C(=O)c3ccccc3)sc2c1
COc1ccc2nc(NC(=O)CCc3ccccc3)sc2c1
COc1ccc2nc(NS(=O)(=O)c3ccccc3)sc2c1
O=C(Nc1nc2ccc(OCC#C)cc2s1)c1ccc(cc1)C(=O)c1ccccc1
COc1ccc2nc(NC(=O)c3ccc(cc3)C(=O)c3ccc(OCC#C)cc3)sc2c1
COc1ccc2nc(NC(=O)c3ccc(cc3)C(=O)NCC#C)sc2c1
COc1ccc(cc1)-c1nc2ccc(NCc3ccc(Cl)c(c3)C(F)(F)F)cc2n(CCNC(C)=O)c1=O
Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1Nc1nc(-c2cccnc2)nc2c1cnn2C
COc1ccc(cc1)-c1nc2cnc(NCc3ccc(Cl)c(Cl)c3)nc2n(CCNC(C)=O)c1=O
COc1ccc(cc1)-c1nc2cnc(NCc3ccc(Cl)c(Cl)c3)nc2n(CCNS(C)(=O)=O)c1=O
COc1ccc(cc1)-c1nc2cnc(NCc3ccc(Cl)c(Cl)c3)nc2n(CCNC(=O)c2ccccc2)c1=O
COc1ccc(cc1)-c1nc2cnc(NCc3ccc(Cl)c(Cl)c3)nc2n(CCNC(=O)c2ccsc2)c1=O
COc1ccc(cc1)-c1nc2cnc(NCc3ccc(Cl)c(Cl)c3)nc2n(CCC(N)=O)c1=O
COc1ccc(cc1)-c1nc2cnc(NCc3cccc(Cl)c3)nc2n(CCNC(C)=O)c1=O
COc1ccc(cc1)-c1nc2cnc(NCc3cccc(c3)C(F)(F)F)nc2n(CCC(N)=O)c1=O
CC(=O)NCCn1c2nc(NCc3ccc(Cl)c(Cl)c3)ncc2nc(-c2cccnc2)c1=O
NC(=O)CCn1c2nc(NCc3ccc(Cl)c(Cl)c3)ncc2nc(-c2cccnc2)c1=O
NC(=O)CCn1c2nc(NCc3cccc(c3)C(F)(F)F)ncc2nc(-c2cccnc2)c1=O
Cc1ccc(cc1)-c1nc2cnc(NCc3cccc(c3)C(F)(F)F)nc2n(CCC(N)=O)c1=O
COc1ccc(cc1)-c1nc2ccc(NCc3ccc(Cl)c(Cl)c3)nc2n(CCNC(C)=O)c1=O
COc1ccc(cc1)-c1nc2ccc(NCc3ccc(Cl)cc3)nc2n(CCNC(C)=O)c1=O
COc1ccc(cc1)-c1nc2ccc(NCc3cccc(Cl)c3)nc2n(CCNC(C)=O)c1=O
COc1ccc(cc1)-c1nc2ccc(NCc3ccc(F)c(Cl)c3)nc2n(CCNC(C)=O)c1=O
COc1ccc(cc1)-c1nc2ccc(NCc3cccc(c3)C(F)(F)F)nc2n(CCNC(C)=O)c1=O
COc1ccc(cc1)-c1nc2ccc(NCc3cccc(OC(F)(F)F)c3)nc2n(CCNC(C)=O)c1=O
COc1ccc(cc1)-c1nc2ccc(NCc3ccc(cc3)C(F)(F)F)nc2n(CCNC(C)=O)c1=O
COc1ccc(cc1)-c1nc2ccc(NCc3cc(cc(c3)C(F)(F)F)C(F)(F)F)nc2n(CCNC(C)=O)c1=O
COc1ccc(cc1)-c1nc2ccc(NCc3ccc(F)c(c3)C(F)(F)F)nc2n(CCNC(C)=O)c1=O
COc1ccc(cc1)-c1nc2ccc(NCc3cc(ccn3)C(F)(F)F)nc2n(CCNC(C)=O)c1=O
COc1ccc(cc1)-c1nc2ccc(NCc3cccc(C)c3)nc2n(CCNC(C)=O)c1=O
COc1ccc(cc1)-c1nc2ccc(NCc3ccc(Cl)c(Cl)c3)nc2n(CCC(N)=O)c1=O
COc1ccc(cc1)-c1nc2ccc(NCc3cccc(c3)C(F)(F)F)nc2n(CCC(N)=O)c1=O
CNC(=O)CCn1c2nc(NCc3cccc(c3)C(F)(F)F)ccc2nc(-c2ccc(OC)cc2)c1=O
CC(=O)NCCn1c2nc(NCc3ccc(Cl)c(Cl)c3)ccc2nc(-c2cccnc2)c1=O
CC(=O)NCCn1c2nc(NCc3ccc(F)c(Cl)c3)ccc2nc(-c2cccnc2)c1=O
CC(=O)NCCn1c2nc(NCc3cccc(c3)C(F)(F)F)ccc2nc(-c2cccnc2)c1=O
COc1ccc(cc1)-c1nc2cnc(NCc3ccc(Cl)c(Cl)c3)cc2n(CCNC(C)=O)c1=O
CC(=O)NCCn1c2cc(NCc3ccc(Cl)c(Cl)c3)ncc2nc(-c2cccnc2)c1=O
CC(=O)NCCn1c2cc(NCc3ccc(Cl)c(Cl)c3)ncc2nc(-c2ccc(C)cc2)c1=O
COc1ccc(cc1)-c1nc2ccc(NCc3ccc(Cl)c(Cl)c3)cc2n(CCNC(C)=O)c1=O
COc1ccc(cc1)-c1nc2ccc(NCc3cccc(c3)C(F)(F)F)cc2n(CCNC(C)=O)c1=O
CC(=O)NCCn1c2cc(NCc3cccc(c3)C(F)(F)F)ccc2nc(-c2cccnc2)c1=O
CCc1ccc(cc1)-c1nc2ccc(NCc3cccc(c3)C(F)(F)F)cc2n(CCNC(C)=O)c1=O
COc1ccc(cc1)-c1nc2ccc(NCc3cccc(C)c3)cc2n(CCNC(C)=O)c1=O
COc1ccc(cc1)-c1nc2ccc(NCc3ccc(C)c(C)c3)cc2n(CCNC(C)=O)c1=O
COc1ccc(cc1)-c1nc2ccc(NCc3ccc(F)c(C)c3)cc2n(CCNC(C)=O)c1=O
COc1ccc(cc1)-c1nc2ccc(NCc3cc(ccn3)C(F)(F)F)cc2n(CCNC(C)=O)c1=O
Clc1ccc(CNC(=O)c2cc(NC(=O)OCc3ccccc3)ccc2Oc2cccnc2)cc1Cl
Clc1ccc(Cn2cnc3ccc(NC(=O)OCc4ccccc4)cc3c2=O)cc1Cl
Clc1ccc(Cn2cnc3ccc(NC(=O)OCc4ccccc4)cc3c2=O)cc1
Fc1ccc(Cn2cnc3ccc(NC(=O)OCc4ccccc4)cc3c2=O)cc1Cl
Cc1ccc(Cn2cnc3ccc(NC(=O)OCc4ccccc4)cc3c2=O)cc1C
Clc1ccc(Cn2cnc3ccc(NC(=O)COc4ccccc4)cc3c2=O)cc1Cl
OCC(=O)Nc1ccc2ncn(Cc3ccc(Cl)cc3)c(=O)c2c1
OCC(=O)Nc1ccc2ncn(Cc3ccc(Cl)c(c3)C(F)(F)F)c(=O)c2c1
OCC(=O)Nc1ccc2ncn(Cc3cccc(c3)-c3ccccc3)c(=O)c2c1
OCC(=O)Nc1ccc2c(c1)ncn(Cc1ccc(Cl)c(Cl)c1)c2=O
OCC(=O)Nc1cnc2ncn(Cc3ccc(Cl)c(Cl)c3)c(=O)c2c1
OC(=O)C(=O)Nc1ccc2ncn(Cc3ccc(Cl)c(Cl)c3)c(=O)c2c1
COc1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
COc1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)s1
COc1ccc(cc1OCCO)C(=O)Nc1cnc(Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)s1
COc1ccc(cc1OCCO)C(=O)Nc1ccc(Cc2cccc(c2)C(F)(F)F)s1
COc1ccc(cc1OCCO)C(=O)Nc1nnc(Cc2cccc(c2)C(F)(F)F)s1
COc1ccc(cc1OCCO)C(=O)Nc1ncc(s1)C(O)c1cccc(c1)C(F)(F)F
COc1ccc(cc1OCCO)C(=O)Nc1ncc(Oc2cccc(c2)C(F)(F)F)s1
COc1ccc(cc1OCCO)C(=O)N(C)c1ncc(Cc2cccc(c2)C(F)(F)F)s1
COc1ccc(NC(=O)c2ncc(Cc3cccc(c3)C(F)(F)F)s2)cc1OCCO
CCOc1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
COCCOc1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
CN(C)CCOc1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
OCCOc1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
CN(C)c1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
CCN(CC)c1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
CCNc1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
OCCOc1cc(ccc1N1CCOCC1)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
CC(=O)Nc1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
COc1cc(ccc1OCCO)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
COc1cc(ccc1OCC(O)=O)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
COc1cc(ccc1OCCN1CCOCC1)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
COc1ccc(cc1OCCCO)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
COc1ccc(cc1OCC(O)CO)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
COc1ccc(cc1OCC(C)O)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
COc1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2cccc(F)c2)s1
COc1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2cccc(Cl)c2)s1
COc1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2cccc(OC(F)(F)F)c2)s1
COc1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2cc(Cl)ccc2Cl)s1
COc1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2cc(Cl)cc(Cl)c2)s1
COc1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2cc(F)cc(F)c2)s1
COc1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2ccc(F)c(c2)C(F)(F)F)s1
COc1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2ccc(F)c(Cl)c2)s1
COc1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2ccc(F)c(F)c2)s1
COc1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2ccc(Cl)c(Cl)c2)s1
COc1ccc(cc1OCCO)C(=O)Nc1ncc(Cc2ccc(C)c(F)c2)s1
COc1ccc(\C=C\C(=O)Nc2ncc(Cc3cccc(c3)C(F)(F)F)s2)cc1
COc1ccc2cc(ccc2c1)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
COc1ccc(cc1OC)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
COc1cccc(c1)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
COc1ccc(cc1)C(=O)Nc1ncc(Cc2cccc(c2)C(F)(F)F)s1
OCC(=O)Nc1ccc2ncn(Cc3ccc(Cl)c(Cl)c3)c(=O)c2c1
Cc1nc2ccc(NCc3cccc(c3)C(F)(F)F)cc2n(CCNC(=O)CO)c1=O
Cc1nc2ccc(NCc3cccc(c3)C(F)(F)F)cc2n(CCNC(=O)C(O)CO)c1=O
Cc1nc2ccc(NCc3cccc(c3)C(F)(F)F)cc2n(CCNC(N)=O)c1=O
OCC(=O)NCCn1c2cc(NCc3cccc(c3)C(F)(F)F)ccc2nc(c1=O)C(F)(F)F
OCC(=O)NCCN1C(=O)COc2ccc(NCc3ccc(Cl)c(Cl)c3)cc12
CNC(=O)c1cnc(s1)N1CCN(CC1)C(=O)c1ccccc1C(F)(F)F
NC(=O)c1cnc(s1)N1CCN(CC1)C(=O)c1ccccc1C(F)(F)F
FC(F)(F)c1ccccc1C(=O)N1CCN(CC1)c1nccs1
OC(=O)c1cnc(s1)N1CCN(CC1)C(=O)c1ccccc1C(F)(F)F
FC(F)(F)c1ccccc1C(=O)N1CCN(CC1)c1ccc(nn1)C(=O)NCCc1ccccc1
FC(F)(F)c1ccccc1C(=O)N1CCN(CC1)c1ccc(nc1)C(=O)NCCc1ccccc1
FC(F)(F)c1ccccc1C(=O)N1CCN(CC1)c1ccc(cn1)C(=O)NCCc1ccccc1
FC(F)(F)c1ccccc1C(=O)N1CCN(CC1)c1ccc(cc1)C(=O)NCCc1ccccc1
O[C@@H](CNC(=O)c1ccc(nn1)N1CCN(CC1)C(=O)c1ccccc1C(F)(F)F)c1ccccc1 |r|
O[C@H](CNC(=O)c1ccc(nn1)N1CCN(CC1)C(=O)c1ccccc1C(F)(F)F)c1ccccc1 |r|
OC(CNC(=O)c1ccc(nn1)N1CCC(CC1)C(=O)c1ccccc1C(F)(F)F)c1ccccc1
Cc1ccccc1C(=O)C1CCN(CC1)c1ccc(nn1)C(=O)NCC(O)c1ccccc1
COc1ccccc1C(=O)C1CCN(CC1)c1ccc(nn1)C(=O)NCC(O)c1ccccc1
OC(CNC(=O)c1ccc(nn1)N1CCC(CC1)C(=O)c1ccccc1OC(F)(F)F)c1ccccc1
OC(CNC(=O)c1ccc(nn1)N1CCC(CC1)C(=O)c1ccccc1)c1ccccc1
OC(CNC(=O)c1ccc(nn1)N1CCC(CC1)C(=O)c1ccc(F)cc1)c1ccccc1
Cc1ccccc1C(=O)C1CCN(CC1)c1ccc(nn1)C(=O)NCC(O)c1ccccc1F
Cc1ccccc1C(=O)C1CCN(CC1)c1ccc(nn1)C(=O)NCC(O)c1cccc(F)c1
Cc1ccccc1C(=O)C1CCN(CC1)c1ccc(nn1)C(=O)NCC(O)c1ccc(F)cc1
Cc1ccccc1C(=O)C1CCN(CC1)c1ccc(nn1)C(=O)NCC(O)c1ccccn1
Cc1ccccc1C(=O)C1CCN(CC1)c1ccc(nn1)C(=O)NCC(O)c1cccnc1
Cc1ccccc1C(=O)C1CCN(CC1)c1ccc(nn1)C(=O)NCC(O)c1ccncc1
Cc1ccccc1C(=O)C1CCN(CC1)c1ccc(nn1)C(=O)NCC(O)c1ccsc1
Cc1ccccc1C(=O)C1CCN(CC1)c1ccc(nn1)C(=O)NCC(O)c1cccs1
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)CCc1ccccc1C2=O)c1ccccc1
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)Oc1ccccc1C2=O)c1ccccc1
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)CC(=O)c1ccccc1O2)c1ccccc1
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)Cc1ccccc1C(=O)O2)c1ccccc1
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)CC(O)c1ccccc1O2)c1ccccc1
COC1CC2(CCN(CC2)c2ccc(nn2)C(=O)NCC(O)c2ccccc2)Oc2ccccc12
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)Oc1ccccc1CC2O)c1ccccc1
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)Oc1ccccc1C=C2)c1ccccc1 |c:28|
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)CCc1ccccc1O2)c1ccccc1
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)Cc1ccccc1CO2)c1ccccc1
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)CC(O)c1c(F)cccc1O2)c1ccccc1
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)CC(O)c1ccc(F)cc1O2)c1ccccc1
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)CC(O)c1cccc(F)c1O2)c1ccccc1
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)CCc1c(F)cccc1O2)c1cccnc1
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)CCc1c(Cl)cccc1O2)c1cccnc1
Cc1cccc2OC3(CCN(CC3)c3ccc(nn3)C(=O)NCC(O)c3cccnc3)CCc12
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)CCc1c(O2)cccc1C(F)(F)F)c1cccnc1
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)CCc1c(F)ccc(F)c1O2)c1cccnc1
FC(F)(F)c1cccc2OC3(CCN(CC3)c3ccc(NC(=O)NCc4cccnc4)nn3)CCc12
FC(F)(F)c1cccc2OC3(CCN(CC3)c3ccc(nn3)-c3nnc(Cc4cccnc4)[nH]3)CCc12
Cn1nc(Cc2cccnc2)nc1-c1ccc(nn1)N1CCC2(CC1)CCc1c(O2)cccc1C(F)(F)F
FC(F)(F)c1cccc2OC3(CCN(CC3)c3ccc(nn3)-c3nnc(Cc4cccnc4)o3)CCc12
FC(F)(F)c1cccc2OC3(CCN(CC3)c3ccc(nn3)-c3nnc(CCc4cccnc4)o3)CCc12
FC(F)(F)c1cccc2OC3(CCN(CC3)c3ccc(nn3)-c3nnc(o3)-c3cccnc3)CCc12
NC(=O)c1cnc(s1)N1CCN(Cc2ccccc2C(F)(F)F)CC1
NC(=O)c1cnc(s1)N1CCC(CC1)Sc1ccccc1C(F)(F)F
NC(=O)c1cnc(s1)N1CCC(CC1)Oc1ccccc1C(F)(F)F
NC(=O)c1cnc(s1)N1CC[C@@H](C1)Oc1ccccc1C(F)(F)F |r|
NC(=O)c1csc(n1)N1CCC(CC1)Oc1ccccc1C(F)(F)F
NC(=O)c1nnc(s1)N1CCC(CC1)Oc1ccccc1C(F)(F)F
NC(=O)c1nnc(o1)N1CCC(CC1)Oc1ccccc1C(F)(F)F
NC(=O)c1nnc([nH]1)N1CCC(CC1)Oc1ccccc1C(F)(F)F
NC(=O)c1cc(no1)N1CCC(CC1)Oc1ccccc1C(F)(F)F
NS(=O)(=O)c1cnc(s1)N1CCC(CC1)Oc1ccccc1C(F)(F)F
FC(F)(F)c1ccccc1OC1CCN(CC1)c1ncc(s1)N1CCCC1=O
COC(=O)Nc1cnc(s1)N1CCC(CC1)Oc1ccccc1C(F)(F)F
FC(F)(F)c1ccccc1OC1CCN(CC1)c1ncc(s1)-c1ncco1
FC(F)(F)c1ccccc1OC1CCN(CC1)c1ncc(s1)-c1nnco1
FC(F)(F)c1ccccc1OC1CCN(CC1)c1ncc(s1)-c1ncon1
Cc1nc(no1)-c1cnc(s1)N1CCC(CC1)Oc1ccccc1C(F)(F)F
OCc1nc(no1)-c1cnc(s1)N1CCC(CC1)Oc1ccccc1C(F)(F)F
Fc1ccccc1-c1ccc(cc1)-c1nc2ccc(cc2[nH]1)C#N
CS(=O)(=O)c1cnc2nc([nH]c2c1)-c1ccc(cc1)-c1ccccc1F
CS(=O)(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1ccccn1
CS(=O)(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1ccc(O)cc1
CS(=O)(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1ccncc1
CS(=O)(=O)c1ccn2cc(nc2c1)-c1ccc(cc1)-c1ccccc1
CS(=O)(=O)c1ccc2nc([nH]c2c1)-c1ccc(nc1)-c1ccccc1F
CS(=O)(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1cccc(Cl)c1
CS(=O)(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1ccccc1
CS(=O)(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1ccccc1F
CS(=O)(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1cccc(F)c1
NS(=O)(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1ccccc1F
CS(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1ccccc1F
CS(=O)(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1cccs1
CS(=O)(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1ccccc1Cl
CS(=O)(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1cccc(O)c1
CC(C)(C)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1ccccc1F
CCS(=O)(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1ccccc1F
CS(=O)(=O)c1ccc2nc([nH]c2c1)-c1ccc(cc1)-c1ccoc1
Clc1cccc2OC3(CCN(CC3)c3ccc(nn3)-c3nnc(Cc4cccnc4)o3)CCc12
Fc1ccc(F)c2OC3(CCN(CC3)c3ccc(nn3)-c3nnc(Cc4cccnc4)o3)CCc12
Cc1cccc2OC3(CCN(CC3)c3ccc(nn3)-c3nnc(Cc4cccnc4)o3)CCc12
Fc1cccc2OC3(CCN(CC3)c3ccc(nn3)-c3nnc(Cc4cccnc4)o3)CCc12
C(c1nnc(o1)-c1ccc(nn1)N1CCC2(CC1)CCc1ccccc1O2)c1cccnc1
C(c1nnc(o1)-c1ccc(nn1)N1CCC2(CC1)CCc1ccccc1O2)c1ccccn1
C(c1nnc(o1)-c1ccc(nn1)N1CCC2(CC1)CCc1ccccc1O2)c1ccncc1
O=C(NCc1cccnc1)c1ccc(nn1)N1CCC2(CC1)CCc1ccccc1O2
Cc1c(ncn1Cc1ccc(Cl)cc1)C(=O)NC(N)=N
Cn1ccc(NC(=O)c2cn(Cc3cccc(OC(F)(F)F)c3)cn2)n1
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)CC(=O)c1ccccc1O2)c1cccnc1
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)CC(=O)Nc1ccccc1O2)c1ccccc1
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)CCNc1ccccc1O2)c1ccccc1
CN1CCC2(CCN(CC2)c2ccc(nn2)C(=O)NCC(O)c2ccccc2)Oc2ccccc12
CN1CCC2(CCN(CC2)c2ccc(nn2)C(=O)NCC(O)c2cccnc2)Oc2ccccc12
CCN1CCC2(CCN(CC2)c2ccc(nn2)C(=O)NCC(O)c2cccnc2)Oc2ccccc12
CC(C)N1CCC2(CCN(CC2)c2ccc(nn2)C(=O)NCC(O)c2cccnc2)Oc2ccccc12
OC(CNC(=O)c1ccc(nn1)N1CCC2(CC1)CCN(CC1CC1)c1ccccc1O2)c1cccnc1
OCCN1CCC2(CCN(CC2)c2ccc(nn2)C(=O)NCC(O)c2cccnc2)Oc2ccccc12
FC(F)(F)c1ccccc1OC1CCN(CC1)c1ncc2[nH]c(=O)[nH]c2n1
Fc1ccc(Br)c(OC2CCN(CC2)c2nc3ccccc3s2)c1
FC(F)(F)c1ccccc1OC1CCN(CC1)c1ncc2[nH]cnc2n1
Fc1ccc(Br)c(OC2CCN(CC2)c2ncc3[nH]cnc3n2)c1
Nc1nc2cnc(nc2s1)N1CCC(CC1)Oc1cc(F)ccc1Br
FC(F)(F)c1ccccc1OC1CCN(CC1)c1ncnc2nc[nH]c12
OC(=O)CCc1nc2nc(sc2c(=O)[nH]1)N1CCC(CC1)Oc1cc(F)ccc1Br
OC(=O)CNc1nc2cnc(nc2s1)N1CCC(CC1)Oc1cc(F)ccc1Br
FC(F)(F)c1ccccc1OC1CCN(CC1)c1nc2cc[nH]c(=O)c2s1
FC(F)(F)c1ccccc1OC1CCN(CC1)c1nc2nc[nH]c(=O)c2s1
FC(F)(F)c1ccccc1OC1CCN(CC1)c1nc2ncccc2s1
Cc1ncc2sc(nc2n1)N1CCC(CC1)Oc1ccccc1C(F)(F)F
Nc1ncnc2nc([nH]c12)N1CCC(CC1)Oc1ccccc1C(F)(F)F
FC(F)(F)c1ccccc1OC1CCN(CC1)c1nc2nc[nH]c2c(=O)[nH]1
Cc1nc2nc(sc2c(=O)[nH]1)N1CCC(CC1)Oc1ccccc1C(F)(F)F
OCc1nc2nc(sc2c(=O)[nH]1)N1CCC(CC1)Oc1ccccc1C(F)(F)F
OC(=O)COc1nc2cnc(nc2s1)N1CCC(CC1)Oc1cc(F)ccc1Br
NC(=O)c1cn(Cc2cc(Br)c(Br)c(Br)c2)nn1
OC(=O)Cn1nnc(n1)-c1cncc(c1)-c1cn(Cc2cc(Br)c(Br)c(Br)c2)nn1
OC(=O)Cn1nnc(n1)-c1cnc(s1)-c1cn(Cc2cc(Cl)c(Cl)c(Cl)c2)nn1
OC(=O)Cn1nnc(n1)-c1cc(no1)-c1cn(Cc2cc(Br)c(Br)c(Br)c2)nn1
OC(=O)Cn1nnc(n1)-c1cc(no1)N1CC2CN(CC2C1)c1cc(F)ccc1Cl
OC(=O)Cn1nnc(n1)-c1cnc(s1)N1CC2CN(CC2C1)c1cc(F)ccc1Cl
OC(=O)Cn1nnc(n1)-c1nnc(s1)N1CC2CN(CC2C1)c1cc(F)ccc1Cl
COc1ccc(Cl)c(c1)N1CC2CN(CC2C1)c1ncc(s1)-c1nnn(CC(O)=O)n1
OC(=O)Cn1nnc(n1)-c1cnc(s1)N1CCN(CC1)c1cc(F)ccc1Cl
OC(=O)Cn1nnc(n1)-c1cnc(s1)N1C[C@@H]2C[C@H]1CN2c1cc(F)ccc1Cl |r|
OC(=O)Cn1nnc(n1)-c1cnc(s1)N1CC2(C1)CN(C2)c1cc(F)ccc1Cl
OC(=O)Cn1nnc(n1)-c1cnc(s1)N1CC2(C1)CCN(CC2)c1cc(F)ccc1Cl
OC(=O)Cn1nnc(n1)-c1cnc(s1)N1CCC2(CN(C2)c2cc(F)ccc2Cl)CC1
OC(=O)c1cncc(c1)-c1ccc(nn1)N1CCC(CC1)Oc1cc(F)c(F)cc1Br
OC(=O)c1cncc(c1)-c1ccc(nn1)N1CCC(CC1)Oc1cc(F)ccc1Br
OC(=O)c1ccc(nc1)-c1ccc(nn1)N1CCC(CC1)Oc1cc(F)ccc1Br
OC(=O)Cc1cncc(c1)-c1ccc(nn1)N1CCC(CC1)Oc1cc(F)ccc1Br
OC(=O)c1cncc(c1)-c1cnc(nc1)N1CCC(CC1)Oc1cc(F)ccc1Br
OC(=O)c1cncc(c1)-c1cnc(cn1)N1CCC(CC1)Oc1cc(F)ccc1Br
OC(=O)c1cncc(c1)-c1ccc(nc1)N1CCC(CC1)Oc1cc(F)ccc1Br
OC(=O)c1cncc(c1)-c1cnc(nn1)N1CCC(CC1)Oc1cc(F)ccc1Br
OC(=O)c1cncc(c1)-c1ccc(nn1)N1CCC(CC1)Oc1ccccc1C(F)(F)F
OC(=O)c1cncc(c1)-c1ccc(nn1)N1CCC(CC1)Oc1ccccc1Cl
OC(=O)c1cncc(c1)-c1ccc(nn1)N1CCC(CC1)Oc1ccccc1Br
OC(=O)c1cncc(c1)-c1ccc(nn1)N1CCC(CC1)Oc1ccccc1I
OC(=O)c1cccc(c1)-c1ccc(nn1)N1CCC(CC1)Oc1ccccc1C(F)(F)F
OC(=O)c1ccc(cc1)-c1ccc(nn1)N1CCC(CC1)Oc1ccccc1C(F)(F)F
OC(=O)Cn1nnc(n1)-c1cc(no1)N1CCC(CC1)Oc1cc(F)ccc1Br
OC(=O)Cn1nnc(n1)-c1cc(OCCOc2cc(F)ccc2Br)no1
OC(=O)Cn1nnc(n1)-c1cc(OCCCOc2cc(F)ccc2Br)no1
OC(=O)Cn1nnc(n1)-c1cc(OCCCCOc2cc(F)ccc2Br)no1
OC(=O)Cn1nnc(n1)-c1cc(OCCOCc2cc(F)ccc2Br)no1
OC(=O)Cn1nnc(n1)-c1nnc(OCCCOc2cc(F)ccc2Br)s1
OC(=O)Cn1nnc(n1)-c1cnc(OCCCOc2cc(F)ccc2Br)s1
OC(=O)Cn1nnc(n1)-c1cnc(OCCCOc2cc(OC(F)(F)F)ccc2Br)s1
Cc1nc(OCCCOc2cc(F)ccc2Br)sc1-c1nnn(CC(O)=O)n1
Clc1ccccc1OC1CCN(CC1)C(=O)CNc1nccnc1C(=O)NCc1ccncc1
FC(F)(F)c1ccccc1OC1CCN(CC1)C(=O)CNc1cccnc1C(=O)NCc1cccnc1
CN(C)C(=O)c1ncccc1NCC(=O)N1CCC(CC1)Oc1ccccc1C(F)(F)F
FC(F)(F)c1ccccc1OC1CCN(CC1)C(=O)CNc1cccnc1C(=O)NCc1ccncc1
OCCNC(=O)c1ncccc1NCC(=O)N1CCC(CC1)Oc1ccccc1C(F)(F)F
CNC(=O)c1nccnc1NCC(=O)N1CCC(CC1)Nc1ccccc1C(F)(F)F
CNC(=O)c1nccnc1NCC(=O)N1CCC(CC1)Oc1c(Cl)cccc1Cl
FC(F)(F)c1ccccc1OC1CCN(CC1)C(=O)CNc1cccnc1C(=O)NCCc1ccccc1
Clc1ccccc1OC1CCN(CC1)C(=O)CNc1nccnc1C(=O)NCc1ccccc1
Clc1ccccc1OC1CCN(CC1)C(=O)CNc1ccccc1C(=O)NCc1ccccc1
Clc1ccccc1OC1CCN(CC1)C(=O)CNc1nccnc1C(=O)Nc1ccccc1
FC(F)(F)c1ccccc1OC1CCN(CC1)C(=O)CNc1cccc(n1)C(=O)NCc1ccccc1
CNC(=O)c1nccnc1NCC(=O)N1CCC(CC1)Oc1c(F)ccc(F)c1Cl
Clc1ccccc1OC1CCN(CC1)C(=O)CNc1nccnc1C#N
NC(=O)c1nccnc1NCC(=O)N1CCC(CC1)Oc1ccccc1Cl
CNC(=O)c1ncccc1NCC(=O)N1CCC(CC1)Oc1ccccc1C(F)(F)F
Clc1ccccc1OC1CCN(CC1)C(=O)CNc1nccnc1C=O
CCNC(=O)c1nccnc1NCC(=O)N1CCC(CC1)Oc1ccccc1Cl
COC(=O)c1nccnc1NCC(=O)N1CCC(CC1)Oc1ccccc1Cl
CNC(=O)c1nccnc1NCC(=O)N1CCC(CC1)Oc1ccccc1
OCCNC(=O)c1nccnc1NCC(=O)N1CCC(CC1)Oc1ccccc1Cl
CNC(=O)c1nccnc1NCC(=O)N1CCC(CC1)Oc1ccccc1Cl
Clc1ccccc1OC1CCN(CC1)C(=O)CNc1cccnc1C(=O)NCc1ccccc1
NC(=O)c1ncccc1NCC(=O)N1CCC(CC1)Oc1ccccc1C(F)(F)F
FC(F)(F)c1ccccc1OC1CCN(CC1)C(=O)CNc1cccnc1C(=O)NC1CCCC1
CC(C)CNC(=O)c1nccnc1NCC(=O)N1CCC(CC1)Oc1ccccc1Cl
CNC(=O)c1cccnc1NCC(=O)N1CCC(CC1)Oc1ccccc1C(F)(F)F
CNC(=O)c1nccnc1NCC(=O)N1CCC(CC1)C(=O)c1ccccc1
CNC(=O)c1nccnc1NCC(=O)N1CCC(CC1)Oc1c(F)cccc1F
CCCNC(=O)c1ncccc1NCC(=O)N1CCC(CC1)Oc1ccccc1C(F)(F)F
Clc1ccccc1OC1CCN(CC1)C(=O)CNc1nccnc1C(=O)NCc1cccnc1
CCNC(=O)c1ncccc1NCC(=O)N1CCC(CC1)Oc1ccccc1C(F)(F)F
CNC(=O)c1nccnc1NCC(=O)N1CCC(CC1)Oc1c(F)cccc1Cl
Clc1ccccc1OC1CCN(CC1)C(=O)CNc1nccnc1Cl
Clc1ccccc1OC1CCN(CC1)C(=O)CNc1nccnc1C(=O)NCc1ccccn1
CNC(=O)c1nccnc1NCC(=O)N1CCC(CC1)Oc1ccccc1Br
FC(F)(F)c1ccccc1OC1CCN(CC1)c1nnc(s1)-c1nnn[nH]1
Fc1ccc(Br)c(OC2CCN(CC2)c2nnc(s2)-c2nnn[nH]2)c1
OC(=O)Cn1nnc(n1)-c1nnc(s1)N1CCC(CC1)Oc1cc(F)ccc1Br
Cc1nnc(s1)-c1ccc(nn1)N1CCC(CC1)Oc1ccccc1C(F)(F)F
FC(F)(F)c1ccccc1C(=O)N1CCN(CC1)c1ccc(nn1)C(=O)Nc1ccccc1
FC(F)(F)c1ccccc1C(=O)N1CCN(CC1)c1ccc(nn1)C(=O)Nc1ccc(Cl)cc1
CCCCCCCNC(=O)c1ccc(nn1)N1CCN(CC1)C(=O)c1ccccc1C(F)(F)F
CCCCCCNC(=O)c1ccc(nn1)N1CCN(CC1)C(=O)c1ccccc1C(F)(F)F
CCCCCNC(=O)c1ccc(nn1)N1CCN(CC1)C(=O)c1ccccc1C(F)(F)F
FC(F)(F)c1ccccc1C(=O)N1CCN(CC1)c1ccc(nn1)C(=O)NCCCCC1CC1
FC(F)(F)c1ccccc1C(=O)N1CCN(CC1)c1ccc(nn1)C(=O)NCCCC1CC1
FC(F)(F)c1ccccc1C(=O)N1CCN(CC1)c1ccc(nn1)C(=O)NCCC1CC1
CC(C)CCNC(=O)c1ccc(nn1)N1CCN(CC1)C(=O)c1ccccc1C(F)(F)F
CC(C)CCNC(=O)c1ccc(cn1)N1CCN(CC1)C(=O)c1ccccc1C(F)(F)F
CCCCCCNC(=O)c1ncc(cn1)N1CCN(CC1)C(=O)c1ccccc1C(F)(F)F
CC(C)CCNC(=O)c1ccc(nc1)N1CCN(CC1)C(=O)c1ccccc1C(F)(F)F
Fc1ccc(C(=O)N2CCN(CC2)c2ccc(nn2)C(=O)NCCC2CC2)c(c1)C(F)(F)F
Fc1cccc(C(=O)N2CCN(CC2)c2ccc(nn2)C(=O)NCCC2CC2)c1C(F)(F)F
Clc1ccc(Cl)c(c1)C(=O)N1CCN(CC1)c1ccc(nn1)C(=O)NCCC1CC1
FC(F)(F)c1ccc(Cl)cc1C(=O)N1CCN(CC1)c1ccc(nn1)C(=O)NCCC1CC1
Fc1ccc(c(c1)C(=O)N1CCN(CC1)c1ccc(nn1)C(=O)NCCC1CC1)C(F)(F)F
Fc1ccc(Cl)c(c1)C(=O)N1CCN(CC1)c1ccc(nn1)C(=O)NCCC1CC1
Cc1cc(C(=O)N2CCN(CC2)c2ccc(nn2)C(=O)NCCC2CC2)c(o1)C(F)(F)F
FC(F)(F)c1nc(Cl)ncc1C(=O)N1CCN(CC1)c1ccc(nn1)C(=O)NCCC1CC1
FC(F)(F)c1occc1C(=O)N1CCN(CC1)c1ccc(nn1)C(=O)NCCC1CC1
CC(C(=O)N1CCN(CC1)c1ccc(nn1)C(=O)NCCC1CC1)(C(F)(F)F)C(F)(F)F
FC(F)(F)c1ccc(CNC(=O)c2ccc(nn2)N2CCN(CC2)C(=O)c2ccccc2C(F)(F)F)o1
Cc1ccc(CNC(=O)c2ccc(nn2)N2CCN(CC2)C(=O)c2ccccc2C(F)(F)F)o1
FC(F)(F)c1ccccc1C(=O)N1CCN(CC1)c1ccc(nn1)C(=O)NCc1nccs1
Cc1cnc(CNC(=O)c2ccc(nn2)N2CCN(CC2)C(=O)c2ccccc2C(F)(F)F)cn1
FC(F)(F)c1ccccc1C(=O)N1CCN(CC1)c1ccc(nn1)C(=O)Nc1nc2ccccc2[nH]1
FC(F)(F)c1ccccc1C(=O)N1CCN(CC1)c1ccc(nn1)C(=O)NCC(=O)c1ccccc1
CC(CNC(=O)c1ccc(nn1)N1CCN(CC1)C(=O)c1ccccc1C(F)(F)F)c1ccccc1
FC(F)(F)c1ccccc1C(=O)N1CCN(CC1)c1ccc(nn1)C(=O)NCCCc1ccccc1
FC(F)(F)c1ccccc1C(=O)c1ccc(cc1)-c1nc2ccc(cc2[nH]1)C(=O)NCc1ccc(Cl)s1
FC(F)(F)c1ccccc1C(=O)c1ccc(cc1)-c1nc2ccc(cc2[nH]1)C(=O)NCc1nccs1
FC(F)(F)c1ccccc1Oc1ccc(cc1)-c1nc2ccc(cc2[nH]1)C(=O)NCc1ccc(Cl)s1
FC(F)(F)c1ccccc1Oc1ccc(cc1)-c1nc2ccc(cc2[nH]1)C(=O)NCc1nccs1
Clc1ccccc1Oc1ccc(cc1)-c1nc2ccc(cc2[nH]1)C(=O)NCCC1CC1
Clc1ccc(CNC(=O)c2ccc3nc([nH]c3c2)-c2ccc(Oc3ccccc3Cl)cc2)s1
Clc1ccccc1Oc1ccc(cc1)-c1nc2ccc(cc2[nH]1)C(=O)NCc1nccs1
OC(c1ccc2nc([nH]c2c1)-c1ccc(OCc2ccccc2)cc1)c1ccccc1C(F)(F)F
COc1ccn(-c2nc(C)c(s2)C(=O)NCc2ccccc2)c(=O)c1
Cc1nc(sc1C(=O)NCc1ccccc1)-n1ccc(OCc2cscn2)cc1=O
Cc1nc(sc1C(=O)NCc1ccccc1)-n1ccc(CCc2ccccc2)cc1=O
Cc1nc(sc1C(=O)NCc1ccc(F)c(F)c1)-n1ccc(O)cc1=O
Cc1nc(sc1C(=O)NCc1ccccc1)-n1ccc(O)cc1=O
Cc1nc(sc1C(=O)NCc1ccc(F)cc1)-n1ccc(O)cc1=O
Cc1nc(sc1C(=O)NCc1ccccc1)-n1ccc(OCc2ccccc2)cc1=O
Cc1nc(sc1C(=O)NCc1ccccc1)-n1ccc(OCCC2CC2)cc1=O
Cc1nc(sc1C(=O)NCc1ccncc1)-n1ccc(O)cc1=O
Cc1nc(sc1C(=O)NCc1ccccc1)-n1ccc(cc1=O)-c1ccccc1
Cc1nc(sc1C(=O)NCc1ccccc1)-n1ccccc1=O
Cc1nc(sc1C(=O)NCC1CC1)-n1ccc(O)cc1=O
Cc1nc(sc1C(=O)NCc1ccccc1)-n1ccc(cc1=O)C(F)(F)F
Cc1nc(sc1C(=O)NCCC1CC1)-n1ccc(O)cc1=O
Cc1nc(sc1C(=O)NCc1ccccc1)-n1ccc(cc1=O)C1CC1
Cc1nc(sc1C(=O)NCc1ccccc1)-n1ccc(OCC2CCCO2)cc1=O
Cc1nc(sc1C(=O)NCc1ccccc1)-n1ccc(C)cc1=O
Cc1nc(sc1C(=O)NCc1cccc(F)c1)-n1ccc(O)cc1=O
Cc1nc(sc1C(=O)NCCc1ccc(F)cc1)-n1ccc(O)cc1=O
Cc1nc(sc1C(=O)NCc1cccc(F)c1)N1CCN(Cc2ccccc2)C1=O
Cc1nc(sc1C(=O)NCc1ccccc1)-c1cncc(Cc2ccccc2)n1
Cc1nc(sc1C(=O)NCc1ccccc1)-c1nnc(Cc2ccccc2)[nH]1
Cc1nc(sc1C(=O)NCc1ccccc1)-n1cc(Cc2ccccc2)nn1
Cc1nc(sc1C(=O)NCc1ccccc1)-c1cn(Cc2ccccc2)nn1
Cc1nc(sc1C(=O)NCc1ccccc1)-c1noc(Cc2ccccc2)n1
Cc1nc(sc1C(=O)NCc1ccccc1)N1C[C@@H](Cc2ccccc2)NC1=O |r|
Cc1nc(sc1C(=O)NCc1ccccc1)N1CCN(Cc2ccccc2)C1=O
Cc1nc(NC(=O)Cc2ccccc2)sc1C(=O)NCc1ccccc1
Cc1nc(sc1C(N)=O)N1CCN(Cc2ccc(F)cc2)C1=O
Cc1nc(sc1C(=O)NCc1ncco1)N1CCN(Cc2ccc(F)cc2)C1=O
Cc1nc(sc1C(=O)NCc1ccccn1)N1CCN(Cc2ccc(F)cc2)C1=O
Cc1nc(sc1C(=O)NCc1ccccn1)N1CCN(Cc2ccccc2)C1=O
CCCCN1CCN(C1=O)c1nc(C)c(s1)C(=O)NCc1cccnc1
Cc1nc(sc1C(=O)NCc1cccnc1)N1CCN(CC2CC2)C1=O
Cc1nc(sc1C(=O)NCc1cccnc1)N1CCN(CC2CCCCC2)C1=O
Cc1nc(sc1C(=O)NCc1cccnc1)N1CCN(CCCc2ccccc2)C1=O
Cc1nc(sc1C(=O)NCc1cccnc1)N1CCN(Cc2ccc(F)cc2)C1=O
Cc1nc(sc1C(=O)NCc1cccnc1)N1CCN(Cc2ccccc2)C1=O
Cc1nc(sc1C(=O)NCc1ccncc1)N1CCN(Cc2ccccc2)C1=O
Cc1nc(sc1C(=O)NCc1ccc(F)cc1)N1CCN(Cc2ccccc2)C1=O
CNC(=O)c1ccc(cn1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
CN(C)c1ccc(cn1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
COc1ccc(cn1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
Fc1ccc2CCN(C3CCN(CC3)c3ccc(nn3)-c3ccc(nc3)C(F)(F)F)c2c1
OCc1ccc(cn1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
Cc1ccc(cn1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
OC(=O)c1ccc(cc1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
Fc1ccc2CCN(C3CCN(CC3)c3ccc(nn3)-c3ccc(cc3)C(F)(F)F)c2c1
OCc1ccc(cc1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
Cc1ccc(cc1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
Cc1csc(n1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
Cc1cnc(s1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
Cc1ccc(s1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
CNC(=O)Cn1cc(cn1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
CCOCCn1cc(cn1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
OCCn1cc(cn1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
CCCn1cc(cn1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
CCn1cc(cn1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
CCOc1cnn(c1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
OCCc1cnn(c1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
OCc1cnn(c1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
Cc1cnn(c1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
OCc1cn(cn1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
Cc1cn(cn1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
Cn1cc(cn1)-c1ccc(nn1)N1CCC(CC1)n1ncc2ccc(F)cc12
Cn1cc(cn1)-c1ccc(nn1)N1CCC(CC1)n1ccc2ccc(F)cc12
Cn1cc(cn1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(cc12)C(F)(F)F
COc1ccc2CCN(C3CCN(CC3)c3ccc(nn3)-c3cnn(C)c3)c2c1
Cc1ccc2CCN(C3CCN(CC3)c3ccc(nn3)-c3cnn(C)c3)c2c1
Cn1cc(cn1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(Cl)cc12
Cn1cc(cn1)-c1ccc(nn1)N1CCC(CC1)N1CCc2cc(Cl)ccc12
Cn1cc(cn1)-c1ccc(nn1)N1CCC(CC1)N1CCc2ccc(F)cc12
Cn1cc(cn1)-c1ccc(nn1)N1CCC(CC1)N1CCc2cc(F)ccc12
Cc1nc(sc1C(=O)NCc1cccnc1)-n1cnn(Cc2ccc(cc2)C(F)(F)F)c1=O
Cc1nc(sc1C(N)=O)-n1cnn(Cc2ccc(F)cc2)c1=O
Cc1nc(sc1C(=O)NCc1cn(C)cn1)-n1cnn(Cc2ccc(F)cc2)c1=O
Cc1nc(sc1C(=O)NCc1cnn(C)c1)-n1cnn(Cc2ccc(F)cc2)c1=O
Cc1cc(CNC(=O)c2sc(nc2C)-n2cnn(Cc3ccc(F)cc3)c2=O)[nH]n1
Cc1nc(sc1C(=O)NCc1cc[nH]n1)-n1cnn(Cc2ccc(F)cc2)c1=O
Cc1ncc(CNC(=O)c2sc(nc2C)-n2cnn(Cc3ccc(F)cc3)c2=O)s1
Cc1nc(sc1C(=O)NCc1nccs1)-n1cnn(Cc2ccc(F)cc2)c1=O
Cc1nc(sc1C(=O)NCc1ncco1)-n1cnn(Cc2ccc(F)cc2)c1=O
Cc1nc(sc1C(=O)NCc1cocn1)-n1cnn(Cc2ccc(F)cc2)c1=O
Cc1nc(sc1C(=O)NCc1cnc(C)cn1)-n1cnn(Cc2ccc(F)cc2)c1=O
Cc1nc(sc1C(=O)NCc1ccccn1)-n1cnn(Cc2ccc(F)cc2)c1=O
Cc1nc(sc1C(=O)NCc1cccnc1)-n1cnn(Cc2ccc(F)cc2)c1=O
Cc1nc(sc1C(=O)NCc1cccnc1)-n1cnn(CC2CC2)c1=O
Cc1nc(sc1C(=O)NCc1cccnc1)-n1cnn(CC2CC2(F)F)c1=O
Cc1nc(sc1C(=O)NCc1cccnc1)-n1cnn(CCCC(F)(F)F)c1=O
Cc1nc(sc1C(=O)NCc1ccccn1)-n1cnn(Cc2ccc(cc2)C(F)(F)F)c1=O
CC(c1ccc(F)cc1)n1ncn(-c2nc(C)c(s2)C(=O)NCc2ccccn2)c1=O
Fc1ccc(Cn2ncn(-c3cc([nH]n3)C(=O)NCc3cccnc3)c2=O)cc1
Fc1ccc(Cn2ncn(-c3cc([nH]n3)C(=O)NCc3ccccn3)c2=O)cc1
Cc1nc(sc1C(=O)NCc1cccnc1)-n1cnn(CCOc2ccc(F)cc2)c1=O
Cc1nc(sc1C(=O)NCc1cccnc1)-n1cnn(Cc2ccc(o2)C(F)(F)F)c1=O
Cc1nc(sc1C(=O)NCc1cccnc1)-n1cnn(Cc2cc(F)cc(F)c2)c1=O