Compile Data Set for Download or QSAR
Report error Found 88 Enz. Inhib. hit(s) with all data for entry = 12123
TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681377(US20240199571, Compound 37)
Affinity DataIC50: 1.73nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681401(US20240199571, Compound 82)
Affinity DataIC50: 3.01nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681376(US20240199571, Compound 36)
Affinity DataIC50: 3.44nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681359(US20240199571, Compound 14)
Affinity DataIC50: 5.37nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681427(US20240199571, Compound 112)
Affinity DataIC50: 5.84nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681361(US20240199571, Compound 18)
Affinity DataIC50: 6.60nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681360(US20240199571, Compound 16)
Affinity DataIC50: 7.51nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681394(US20240199571, Compound 72)
Affinity DataIC50: 8.56nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681428(US20240199571, Compound 116)
Affinity DataIC50: 9.27nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681432(US20240199571, Compound 120)
Affinity DataIC50: 9.40nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681410(US20240199571, Compound 92)
Affinity DataIC50: 9.81nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681425(US20240199571, Compound 110)
Affinity DataIC50: 9.84nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681413(US20240199571, Compound 95)
Affinity DataIC50: 10.1nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681387(US20240199571, Compound 57)
Affinity DataIC50: 10.4nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681424(US20240199571, Compound 109)
Affinity DataIC50: 10.7nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681395(US20240199571, Compound 73)
Affinity DataIC50: 11.8nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681416(US20240199571, Compound 98)
Affinity DataIC50: 12.6nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681409(US20240199571, Compound 91)
Affinity DataIC50: 13nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681434(US20240199571, Compound 122)
Affinity DataIC50: 13.1nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681402(US20240199571, Compound 84)
Affinity DataIC50: 13.2nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681399(US20240199571, Compound 79)
Affinity DataIC50: 13.6nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681430(US20240199571, Compound 118)
Affinity DataIC50: 13.8nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681418(US20240199571, Compound 100)
Affinity DataIC50: 14.1nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681403(US20240199571, Compound 85)
Affinity DataIC50: 14.2nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681433(US20240199571, Compound 121)
Affinity DataIC50: 14.3nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681423(US20240199571, Compound 107)
Affinity DataIC50: 15.1nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681407(US20240199571, Compound 89)
Affinity DataIC50: 15.2nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681404(US20240199571, Compound 86)
Affinity DataIC50: 16nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681422(US20240199571, Compound 104)
Affinity DataIC50: 16.6nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681417(US20240199571, Compound 99)
Affinity DataIC50: 17.4nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681426(US20240199571, Compound 111)
Affinity DataIC50: 17.6nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681431(US20240199571, Compound 119)
Affinity DataIC50: 17.7nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681411(US20240199571, Compound 93)
Affinity DataIC50: 18nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681390(US20240199571, Compound 60)
Affinity DataIC50: 18.4nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681429(US20240199571, Compound 117)
Affinity DataIC50: 19nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681364(US20240199571, Compound 21)
Affinity DataIC50: 19.4nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681363(US20240199571, Compound 20)
Affinity DataIC50: 19.4nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681368(US20240199571, Compound 26)
Affinity DataIC50: 19.6nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681400(US20240199571, Compound 80)
Affinity DataIC50: 20.2nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681388(US20240199571, Compound 58)
Affinity DataIC50: 20.4nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681414(US20240199571, Compound 96)
Affinity DataIC50: 20.6nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681421(US20240199571, Compound 103)
Affinity DataIC50: 21.6nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681375(US20240199571, Compound 35)
Affinity DataIC50: 24.6nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681405(US20240199571, Compound 87)
Affinity DataIC50: 24.8nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681415(US20240199571, Compound 97)
Affinity DataIC50: 25.3nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681372(US20240199571, Compound 31)
Affinity DataIC50: 26.7nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681435(US20240199571, Compound 123)
Affinity DataIC50: 26.7nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681383(US20240199571, Compound 50)
Affinity DataIC50: 28.3nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681419(US20240199571, Compound 101)
Affinity DataIC50: 28.7nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandPNGBDBM681397(US20240199571, Compound 75)
Affinity DataIC50: 28.9nMAssay Description:Table 1: The purpose of the assay was to test the in vitro inhibitory activity of the compounds against LSD1. The enzyme used in the assay was human ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent

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