Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50008516
TargetProteinase-activated receptor 1(Human)
University At Stony Brook

Curated by ChEMBL
LigandPNGBDBM50073994((S)-2-{(S)-2-[(S)-2-{(S)-3-(4-Fluoro-phenyl)-2-[(E...)
Affinity DataIC50: 300nMAssay Description:Human Thrombin receptor 1 (PAR-1) antagonistic ability to inhibit SFLLRN-NH2 (2.7 uM)-induced platelet aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
University At Stony Brook

Curated by ChEMBL
LigandPNGBDBM50073996((S)-2-{(S)-2-[(S)-2-[(S)-2-[3-(4-Benzoyl-phenyl)-p...)
Affinity DataIC50: 3.10E+3nMAssay Description:Human Thrombin receptor 1 (PAR-1) antagonistic ability to inhibit SFLLRN-NH2 (2.7 uM)-induced platelet aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
University At Stony Brook

Curated by ChEMBL
LigandPNGBDBM50074001((S)-2-((S)-2-{(S)-3-(4-Benzoyl-phenyl)-2-[(S)-2-{(...)
Affinity DataIC50: 3.10E+3nMAssay Description:Human Thrombin receptor 1 (PAR-1) antagonistic ability to inhibit SFLLRN-NH2 (2.7 uM)-induced platelet aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
University At Stony Brook

Curated by ChEMBL
LigandPNGBDBM50073997((2S)-5-{5-[(3aR,4R,6aS)-2-oxo-hexahydro-1H-thieno[...)
Affinity DataIC50: 3.40E+3nMAssay Description:Human Thrombin receptor 1 (PAR-1) antagonistic ability to inhibit SFLLRN-NH2 (2.7 uM)-induced platelet aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
University At Stony Brook

Curated by ChEMBL
LigandPNGBDBM50074000((S)-2-{(S)-3-(4-Benzoyl-phenyl)-2-[(S)-2-{(S)-3-(4...)
Affinity DataIC50: 6.00E+3nMAssay Description:Human Thrombin receptor 1 (PAR-1) antagonistic ability to inhibit SFLLRN-NH2 (2.7 uM)-induced platelet aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
University At Stony Brook

Curated by ChEMBL
LigandPNGBDBM50073998((S)-2-((S)-3-(4-Benzoyl-phenyl)-2-{(S)-2-[(S)-2-{(...)
Affinity DataIC50: 9.00E+3nMAssay Description:Human Thrombin receptor 1 (PAR-1) antagonistic ability to inhibit SFLLRN-NH2 (2.7 uM)-induced platelet aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
University At Stony Brook

Curated by ChEMBL
LigandPNGBDBM50073999((2S)-5-{5-[(3aR,6aS)-2-oxo-hexahydro-1H-thieno[3,4...)
Affinity DataIC50: 9.70E+3nMAssay Description:Human Thrombin receptor 1 (PAR-1) antagonistic ability to inhibit SFLLRN-NH2 (2.7 uM)-induced platelet aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
University At Stony Brook

Curated by ChEMBL
LigandPNGBDBM50073995((S)-3-(4-Benzoyl-phenyl)-2-{(S)-2-[(S)-2-{(S)-3-(4...)
Affinity DataIC50: 1.30E+4nMAssay Description:Human Thrombin receptor 1 (PAR-1) antagonistic ability to inhibit SFLLRN-NH2 (2.7 uM)-induced platelet aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed