Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50008521
Target72 kDa type IV collagenase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074024((2S,3R)-3-(4-Methoxy-benzenesulfonyl)-2-methyl-7-p...)
Affinity DataKi:  10nMAssay Description:Inhibition of matrix metalloprotease-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074023(N-Hydroxy-3-(4-methoxy-benzenesulfonyl)-4-phenyl-b...)
Affinity DataKi:  20nMAssay Description:Inhibition of matrix metalloprotease-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074027(3-(4-Methoxy-benzenesulfonyl)-7-phenyl-heptanoic a...)
Affinity DataKi:  20nMAssay Description:Inhibition of matrix metalloprotease-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074021(3-(4-Methoxy-benzenesulfonyl)-5-phenyl-pentanoic a...)
Affinity DataKi:  30nMAssay Description:Inhibition of matrix metalloprotease-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074022(3-(4-Methoxy-benzenesulfonyl)-3-methyl-7-phenyl-he...)
Affinity DataKi:  50nMAssay Description:Inhibition of matrix metalloprotease-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074028(3-(4-Methoxy-benzenesulfonyl)-6-phenyl-hexanoic ac...)
Affinity DataKi:  50nMAssay Description:Inhibition of matrix metalloprotease-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074026(3-(4-Methoxy-benzenesulfonyl)-2-methyl-7-phenyl-he...)
Affinity DataKi:  60nMAssay Description:Inhibition of matrix metalloprotease-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074021(3-(4-Methoxy-benzenesulfonyl)-5-phenyl-pentanoic a...)
Affinity DataKi:  200nMAssay Description:Inhibition of matrix metalloprotease-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074023(N-Hydroxy-3-(4-methoxy-benzenesulfonyl)-4-phenyl-b...)
Affinity DataKi:  300nMAssay Description:Inhibition of matrix metalloprotease-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074024((2S,3R)-3-(4-Methoxy-benzenesulfonyl)-2-methyl-7-p...)
Affinity DataKi:  500nMAssay Description:Inhibition of matrix metalloprotease-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074028(3-(4-Methoxy-benzenesulfonyl)-6-phenyl-hexanoic ac...)
Affinity DataKi:  600nMAssay Description:Inhibition of matrix metalloprotease-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074026(3-(4-Methoxy-benzenesulfonyl)-2-methyl-7-phenyl-he...)
Affinity DataKi:  600nMAssay Description:Inhibition of matrix metalloprotease-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074027(3-(4-Methoxy-benzenesulfonyl)-7-phenyl-heptanoic a...)
Affinity DataKi:  700nMAssay Description:Inhibition of matrix metalloprotease-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074023(N-Hydroxy-3-(4-methoxy-benzenesulfonyl)-4-phenyl-b...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of matrix metalloprotease-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074022(3-(4-Methoxy-benzenesulfonyl)-3-methyl-7-phenyl-he...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of matrix metalloprotease-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074024((2S,3R)-3-(4-Methoxy-benzenesulfonyl)-2-methyl-7-p...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of matrix metalloprotease-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074022(3-(4-Methoxy-benzenesulfonyl)-3-methyl-7-phenyl-he...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of matrix metalloprotease-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074026(3-(4-Methoxy-benzenesulfonyl)-2-methyl-7-phenyl-he...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of matrix metalloprotease-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074028(3-(4-Methoxy-benzenesulfonyl)-6-phenyl-hexanoic ac...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of matrix metalloprotease-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074021(3-(4-Methoxy-benzenesulfonyl)-5-phenyl-pentanoic a...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of matrix metalloprotease-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074027(3-(4-Methoxy-benzenesulfonyl)-7-phenyl-heptanoic a...)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of matrix metalloprotease-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074025(3-(3,4-Dimethoxy-benzenesulfonyl)-7-phenyl-heptano...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of matrix metalloprotease-2 (MMP-2), gelatinase-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074025(3-(3,4-Dimethoxy-benzenesulfonyl)-7-phenyl-heptano...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of matrix metalloprotease-1 (MMP-1), fibroblast collagenase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50074025(3-(3,4-Dimethoxy-benzenesulfonyl)-7-phenyl-heptano...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of matrix metalloprotease-3 (MMP-3), stromelysin-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed