Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50008591
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075089(Sodium; [2-(4-chloro-benzenesulfonylamino)-indan-5...)
Affinity DataIC50: 2.20nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075088(Sodium; {2-[(4-chloro-benzenesulfonylamino)-methyl...)
Affinity DataIC50: 3nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075086(Sodium; [2-(benzenesulfonylamino-methyl)-indan-5-y...)
Affinity DataIC50: 13nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075091(Sodium; 3-{2-[(4-chloro-benzenesulfonylamino)-meth...)
Affinity DataIC50: 15nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075077(Sodium; {2-[(naphthalene-2-sulfonylamino)-methyl]-...)
Affinity DataIC50: 22nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075082(Sodium; 2-[(4-chloro-benzenesulfonylamino)-methyl]...)
Affinity DataIC50: 26nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075094(Sodium; {2-[2-(4-chloro-benzenesulfonylamino)-ethy...)
Affinity DataIC50: 32nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075093(Sodium; 5-{2-[(4-chloro-benzenesulfonylamino)-meth...)
Affinity DataIC50: 36nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002805(CHEMBL71685 | (daltroban){4-[2-(4-Chloro-benzenesu...)
Affinity DataIC50: 37nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075079(Sodium; 4-{2-[(4-chloro-benzenesulfonylamino)-meth...)
Affinity DataIC50: 39nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075096(Sodium; 2-[2-(4-chloro-benzenesulfonylamino)-ethyl...)
Affinity DataIC50: 66nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075092(Sodium; 2-[3-(4-chloro-benzenesulfonylamino)-propy...)
Affinity DataIC50: 85nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075076(Sodium; {2-[(thiophene-2-sulfonylamino)-methyl]-in...)
Affinity DataIC50: 85nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075085(Sodium; {2-[(4-chloro-benzenesulfonylamino)-methyl...)
Affinity DataIC50: 141nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075091(Sodium; 3-{2-[(4-chloro-benzenesulfonylamino)-meth...)
Affinity DataIC50: 160nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075090(Sodium; {2-[(naphthalene-1-sulfonylamino)-methyl]-...)
Affinity DataIC50: 295nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075085(Sodium; {2-[(4-chloro-benzenesulfonylamino)-methyl...)
Affinity DataIC50: 320nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075088(Sodium; {2-[(4-chloro-benzenesulfonylamino)-methyl...)
Affinity DataIC50: 360nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075089(Sodium; [2-(4-chloro-benzenesulfonylamino)-indan-5...)
Affinity DataIC50: 360nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002805(CHEMBL71685 | (daltroban){4-[2-(4-Chloro-benzenesu...)
Affinity DataIC50: 460nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075081(Sodium; 2-[4-(4-chloro-benzenesulfonylamino)-butyl...)
Affinity DataIC50: 479nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075084(Sodium; {2-[3-(4-chloro-benzenesulfonylamino)-prop...)
Affinity DataIC50: 513nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075077(Sodium; {2-[(naphthalene-2-sulfonylamino)-methyl]-...)
Affinity DataIC50: 950nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075095(Sodium; {2-[4-(4-chloro-benzenesulfonylamino)-buty...)
Affinity DataIC50: 977nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075086(Sodium; [2-(benzenesulfonylamino-methyl)-indan-5-y...)
Affinity DataIC50: 1.02E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075080(Sodium; [2-(cyclohexanesulfonylamino-methyl)-indan...)
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075082(Sodium; 2-[(4-chloro-benzenesulfonylamino)-methyl]...)
Affinity DataIC50: 1.32E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075079(Sodium; 4-{2-[(4-chloro-benzenesulfonylamino)-meth...)
Affinity DataIC50: 1.34E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075083(Sodium; {2-[(pentane-1-sulfonylamino)-methyl]-inda...)
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075094(Sodium; {2-[2-(4-chloro-benzenesulfonylamino)-ethy...)
Affinity DataIC50: 1.48E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075087(Sodium; {2-[(pyridine-3-sulfonylamino)-methyl]-ind...)
Affinity DataIC50: 1.90E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075076(Sodium; {2-[(thiophene-2-sulfonylamino)-methyl]-in...)
Affinity DataIC50: 2.81E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075093(Sodium; 5-{2-[(4-chloro-benzenesulfonylamino)-meth...)
Affinity DataIC50: 2.88E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075078(Sodium; [2-(phenylmethanesulfonylamino-methyl)-ind...)
Affinity DataIC50: 5.90E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075092(Sodium; 2-[3-(4-chloro-benzenesulfonylamino)-propy...)
Affinity DataIC50: 6.60E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075096(Sodium; 2-[2-(4-chloro-benzenesulfonylamino)-ethyl...)
Affinity DataIC50: 7.76E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075080(Sodium; [2-(cyclohexanesulfonylamino-methyl)-indan...)
Affinity DataIC50: 1.78E+4nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075090(Sodium; {2-[(naphthalene-1-sulfonylamino)-methyl]-...)
Affinity DataIC50: 4.79E+4nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075084(Sodium; {2-[3-(4-chloro-benzenesulfonylamino)-prop...)
Affinity DataIC50: 7.23E+4nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075083(Sodium; {2-[(pentane-1-sulfonylamino)-methyl]-inda...)
Affinity DataIC50: 7.76E+4nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075087(Sodium; {2-[(pyridine-3-sulfonylamino)-methyl]-ind...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075095(Sodium; {2-[4-(4-chloro-benzenesulfonylamino)-buty...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075081(Sodium; 2-[4-(4-chloro-benzenesulfonylamino)-butyl...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Zeria Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50075078(Sodium; [2-(phenylmethanesulfonylamino-methyl)-ind...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro thromboxane A2 antagonistic activity on aggregation of rabbit platelets induced by U-46,619 (4 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed