Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50008745
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076782(N-Cyclopropylmethyl-N-ethyl-2,5-dimethyl-N'-(2,4,6...)
Affinity DataKi:  2nMAssay Description:Antagonistic activity for Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50058163(CHEMBL9946 | CP 154,526 | CP-154526 | N-butyl-N-et...)
Affinity DataKi:  2.70nMAssay Description:Antagonistic activity for Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50074458([3-(2-Bromo-4,6-dimethoxy-phenyl)-5-methyl-3H-[1,2...)
Affinity DataKi:  3.5nMAssay Description:Antagonistic activity for Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50074456(CHEMBL10504 | SC241 | [3-(2-Bromo-4-isopropyl-phen...)
Affinity DataKi:  3.70nMAssay Description:Antagonistic activity for Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076779((2-Bromo-4-isopropyl-phenyl)-ethyl-[4-methyl-6-(2-...)
Affinity DataKi:  5.5nMAssay Description:Antagonistic activity for Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076785(2,5,6-Trimethyl-4-(2-trifluoromethyl-phenyl)-7-(2,...)
Affinity DataKi:  9.70nMAssay Description:Antagonistic activity for Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076786(3-(2-Bromo-4,6-dimethoxy-phenyl)-5-methyl-7-(2-tri...)
Affinity DataKi:  21nMAssay Description:Antagonistic activity for Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076780((2-Bromo-4,6-dimethoxy-phenyl)-[2-methyl-5-nitro-6...)
Affinity DataKi:  23nMAssay Description:Antagonistic activity for Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076777(9-(2-Bromo-4,6-dimethoxy-phenyl)-2,8-dimethyl-6-(2...)
Affinity DataKi:  32nMAssay Description:Antagonistic activity for Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076783(6-Methyl-3-methylsulfanyl-1-(2,4,6-trichloro-pheny...)
Affinity DataKi:  33nMAssay Description:Antagonistic activity for Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076784(N*4*-(2-Bromo-4,6-dimethoxy-phenyl)-2-methyl-6-(2-...)
Affinity DataKi:  60nMAssay Description:Antagonistic activity for Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076787(9-(2-Bromo-4,6-dimethoxy-phenyl)-2,7-dimethyl-6-(2...)
Affinity DataKi:  96nMAssay Description:Antagonistic activity for Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076778(5-Methyl-7-(2-trifluoromethyl-phenyl)-3-(2,4,6-tri...)
Affinity DataKi:  168nMAssay Description:Antagonistic activity for Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50076781(9-(2-Bromo-4,6-dimethoxy-phenyl)-2-methyl-6-(2-tri...)
Affinity DataKi:  202nMAssay Description:Antagonistic activity for Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed