Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50008777
TargetNeutrophil elastase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50077013(2-(6-Methoxy-3,4-dihydro-naphthalen-1-yl)-benzo[d]...)
Affinity DataIC50: 610nMAssay Description:In vitro inhibitory activity against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50077014(CHEMBL24450 | cid_296003 | 2-Furan-2-yl-benzo[d][1...)
Affinity DataIC50: 5.50E+3nMAssay Description:In vitro inhibitory activity against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50077012(((E)-2-Cyclooct-1-enyl)-benzo[d][1,3]oxazin-4-one ...)
Affinity DataIC50: 7.00E+3nMAssay Description:In vitro inhibitory activity against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50077011(2-Phenyl-benzo[d][1,3]oxazin-4-one | CHEMBL24449 |...)
Affinity DataIC50: 1.70E+4nMAssay Description:In vitro inhibitory activity against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50077014(CHEMBL24450 | cid_296003 | 2-Furan-2-yl-benzo[d][1...)
Affinity DataKi:  1.78E+3nMAssay Description:pKi against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50077011(2-Phenyl-benzo[d][1,3]oxazin-4-one | CHEMBL24449 |...)
Affinity DataKi:  9.55E+3nMAssay Description:pKi against human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed