Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50008925
TargetInositol 1,4,5-trisphosphate receptor type 3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50078572(CHEMBL297496 | {4-[(4-Dimethylamino-phenyl)-(4-{3-...)
Affinity DataKd:  1.20nMpH: 7.4Assay Description:Dissociation constant of compound was measured in IP3-binding domain(IBD) of human Inositol 1,4,5-trisphosphate receptor at pH 7.4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50078573(Phosphoric acid 3-amino-propyl ester (1R,2R,3S,4R,...)
Affinity DataKd:  1.12E+3nMpH: 7.4Assay Description:Dissociation constant of compound was measured in IP3-binding domain(IBD) of human Inositol 1,4,5-trisphosphate receptor at pH 7.4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInositol 1,4,5-trisphosphate receptor type 3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50075183(1D-myo-inositol 1,4,5-tris(dihydrogen phosphate) |...)
Affinity DataKd:  195nMpH: 7.4Assay Description:Dissociation constant of compound was measured in IP3-binding domain(IBD) of human Inositol 1,4,5-trisphosphate receptor at pH 7.4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetInositol 1,4,5-trisphosphate receptor type 3(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50078574(inositol 1,4,5-trisphosphate analogue | CHEMBL4627...)
Affinity DataKd:  188nMpH: 7.4Assay Description:Dissociation constant of compound was measured in IP3-binding domain(IBD) of human Inositol 1,4,5-trisphosphate receptor at pH 7.4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed