Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50009169
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080842(N,N'-(acridine-3,6-diyl)bis(3-(4-methylpiperidin-1...)
Affinity DataIC50: 1.35E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080848(N,N'-(acridine-3,6-diyl)bis(3-(2-methylpiperidin-1...)
Affinity DataIC50: 2.60E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080837(3-(2-Ethyl-piperidin-1-yl)-N-{6-[3-(2-ethyl-piperi...)
Affinity DataIC50: 2.70E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080847(N,N'-(acridine-3,6-diyl)bis(3-(piperidin-1-yl)prop...)
Affinity DataIC50: 2.80E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080840(N,N'-(acridine-3,6-diyl)bis(3-(azepan-1-yl)propana...)
Affinity DataIC50: 3.10E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080850(3-[2-(2-Hydroxy-ethyl)-piperidin-1-yl]-N-(6-{3-[2-...)
Affinity DataIC50: 4.10E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080839(3-(3-Methyl-piperidin-1-yl)-N-{6-[3-(3-methyl-pipe...)
Affinity DataIC50: 4.40E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080849(3-PYRROLIDIN-1-YL-N-[6-(3-PYRROLIDIN-1-YL-PROPIONY...)
Affinity DataIC50: 5.20E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080841(N,N'-(acridine-3,6-diyl)bis(3-(2-(hydroxymethyl)pi...)
Affinity DataIC50: 5.40E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080844(N,N'-(acridine-3,6-diyl)bis(3-(diethylamino)propan...)
Affinity DataIC50: 5.80E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080845(3-(4-Hydroxy-piperidin-1-yl)-N-{6-[3-(4-hydroxy-pi...)
Affinity DataIC50: 8.00E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080851(3-Dimethylamino-N-[6-(3-dimethylamino-propionylami...)
Affinity DataIC50: 8.20E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080838(N,N'-(acridine-3,6-diyl)bis(3-(4-benzylpiperidin-1...)
Affinity DataIC50: 5.00E+4nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080852(3-Azocan-1-yl-N-[6-(3-azocan-1-yl-propionylamino)-...)
Affinity DataIC50: 5.00E+4nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080843(3-Morpholin-4-yl-N-[6-(3-morpholin-4-yl-propionyla...)
Affinity DataIC50: 5.00E+4nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080846(3,6-Bis[3-(1,3,3-trimethyl-6-azabicyclo[3.2.1]octa...)
Affinity DataIC50: 5.00E+4nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed