Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50036760
TargetB2 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50403371(Firazyr | HOE-140 | ICATIBANT)
Affinity DataKi:  0.0640nMAssay Description:Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50403371(Firazyr | HOE-140 | ICATIBANT)
Affinity DataKi:  0.0770nMAssay Description:Binding affinity against rat bradykinin B2 receptors expressed in CHO cells using [3H]bradykinin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50049949(2-(2-{[1-(2-{2-[2-({1-[1-(2-Amino-5-guanidino-pent...)
Affinity DataKi:  0.460nMAssay Description:Binding affinity against rat Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50049949(2-(2-{[1-(2-{2-[2-({1-[1-(2-Amino-5-guanidino-pent...)
Affinity DataKi:  0.650nMAssay Description:Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50408748(CHEMBL2112698)
Affinity DataKi:  0.700nMAssay Description:Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50408748(CHEMBL2112698)
Affinity DataKi:  6nMAssay Description:Binding affinity against rat bradykinin B2 receptors expressed in CHO cells using [3H]bradykinin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50081653([2-[2-(3-Amino-4-oxo-3,4-dihydro-2H-benzo[b][1,4]t...)
Affinity DataKi:  13nMAssay Description:Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50081652((RMP-7)H-Arg-Pro-Hyp-Gly-Ser-Pro-4-Me-Tyr(CH2NH2)-...)
Affinity DataKi:  19nMAssay Description:Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50408749(CHEMBL2111889)
Affinity DataKi:  162nMAssay Description:Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50081653([2-[2-(3-Amino-4-oxo-3,4-dihydro-2H-benzo[b][1,4]t...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against human cloned Bradykinin receptor B1 expressed in CHO cells using [3H]-bradykinin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50408748(CHEMBL2112698)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against human cloned Bradykinin receptor B1 expressed in CHO cells using [3H]-bradykinin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50408749(CHEMBL2111889)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against human cloned Bradykinin receptor B1 expressed in CHO cells using [3H]-bradykinin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed