Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50009523
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084713(N-[5-Amino-6-(6-hydroxy-1-pyridin-3-ylmethyl-1,2,3...)
Affinity DataIC50: 1nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50015490(NPY, human, rat | CHEMBL438945 | NPY | H-YPSKPDNPG...)
Affinity DataIC50: 3nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084712(N-{4-[(1-Allyl-6-hydroxy-1,2,3,4-tetrahydro-naphth...)
Affinity DataIC50: 5nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084693(2-(3-Benzenesulfonylamino-pyrrolidin-1-yl)-N-(6-fl...)
Affinity DataIC50: 5nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084699(2-Fluoro-N-{4-[(6-hydroxy-1-pyridin-3-ylmethyl-1,2...)
Affinity DataIC50: 7nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084701(2-(4-Benzenesulfonylamino-piperidin-1-yl)-N-(6-flu...)
Affinity DataIC50: 10nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084698(N-{4-[(6-Methoxy-1-pyridin-3-ylmethyl-1,2,3,4-tetr...)
Affinity DataIC50: 10nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084707(4-[(2-Fluoro-benzenesulfonylamino)-methyl]-cyclohe...)
Affinity DataIC50: 11nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084704(2-(3-Benzenesulfonylamino-pyrrolidin-1-yl)-N-(6-fl...)
Affinity DataIC50: 11nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084700(4-(Benzenesulfonylamino-methyl)-cyclohexanecarboxy...)
Affinity DataIC50: 11nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084703(4-[(2-Fluoro-benzenesulfonylamino)-methyl]-cyclohe...)
Affinity DataIC50: 12nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084709(2-Fluoro-N-{4-[(6-fluoro-1-pyridin-3-ylmethyl-1,2,...)
Affinity DataIC50: 19nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084694(N-{4-[(1-Allyl-6-fluoro-1,2,3,4-tetrahydro-naphtha...)
Affinity DataIC50: 21nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084692(2-Amino-6-(2-fluoro-benzenesulfonylamino)-hexanoic...)
Affinity DataIC50: 22nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084695(2-Fluoro-N-{4-[(6-methoxy-1-pyridin-3-ylmethyl-1,2...)
Affinity DataIC50: 23nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084710(N-{4-[(6-Fluoro-1-pyridin-3-ylmethyl-1,2,3,4-tetra...)
Affinity DataIC50: 27nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084706(2-(3-Benzenesulfonylamino-pyrrolidin-1-yl)-N-(6-fl...)
Affinity DataIC50: 27nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084705(4-(Benzenesulfonylamino-methyl)-cyclohexanecarboxy...)
Affinity DataIC50: 40nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084697(N-[6-(6-Methoxy-1-pyridin-3-ylmethyl-1,2,3,4-tetra...)
Affinity DataIC50: 53nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084702(4-(Benzenesulfonylamino-methyl)-cyclohexanecarboxy...)
Affinity DataIC50: 75nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084708(Naphthalene-2-sulfonic acid {4-[(6-methoxy-1-pyrid...)
Affinity DataIC50: 337nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084696(Naphthalene-2-sulfonic acid {4-[(1-benzyl-6-methox...)
Affinity DataIC50: 443nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50084711((1-Benzyl-6-methoxy-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataIC50: 900nMAssay Description:Inhibition of [125I]-PYY binding to recombinant NPY Y5 receptor on HEK293 cell membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed