Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50009554
TargetAlpha-1A adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084999(4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-tetrahyd...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084996(1-(3-{[4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-t...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50085000(1-{3-[(4-Benzo[1,2,5]oxadiazol-5-yl-2,5-dioxo-1,2,...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50218277(CHEMBL35520)
Affinity DataKi: <1nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50082797(4-(3,4-Difluoro-phenyl)-3-[3-(4-methoxycarbonyl-4-...)
Affinity DataKi: <1nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50085004(1-(3-{[4-(4-Nitro-phenyl)-2,5-dioxo-1,2,5,7-tetrah...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084996(1-(3-{[4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-t...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084996(1-(3-{[4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-t...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50085003(4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-tetrahyd...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084997(4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-tetrahyd...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50085002(4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-tetrahyd...)
Affinity DataKi:  9.10nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50085001(1-(4-{[4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-t...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50085005(1-{3-[(4-Benzo[1,3]dioxol-5-yl-2,5-dioxo-1,2,5,7-t...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084998(1-(2-{[4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-t...)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50085002(4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-tetrahyd...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084996(1-(3-{[4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-t...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084996(1-(3-{[4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-t...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50085004(1-(3-{[4-(4-Nitro-phenyl)-2,5-dioxo-1,2,5,7-tetrah...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50085002(4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-tetrahyd...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084999(4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-tetrahyd...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084999(4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-tetrahyd...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084996(1-(3-{[4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-t...)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084996(1-(3-{[4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-t...)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50085000(1-{3-[(4-Benzo[1,2,5]oxadiazol-5-yl-2,5-dioxo-1,2,...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084996(1-(3-{[4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-t...)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50085000(1-{3-[(4-Benzo[1,2,5]oxadiazol-5-yl-2,5-dioxo-1,2,...)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50085001(1-(4-{[4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-t...)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50085003(4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-tetrahyd...)
Affinity DataKi:  350nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50085005(1-{3-[(4-Benzo[1,3]dioxol-5-yl-2,5-dioxo-1,2,5,7-t...)
Affinity DataKi:  390nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50085004(1-(3-{[4-(4-Nitro-phenyl)-2,5-dioxo-1,2,5,7-tetrah...)
Affinity DataKi:  420nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50085001(1-(4-{[4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-t...)
Affinity DataKi:  420nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084996(1-(3-{[4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-t...)
Affinity DataKi:  430nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50085003(4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-tetrahyd...)
Affinity DataKi:  690nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084997(4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-tetrahyd...)
Affinity DataKi:  970nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084997(4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-tetrahyd...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084998(1-(2-{[4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-t...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50084998(1-(2-{[4-(3,4-Difluoro-phenyl)-2,5-dioxo-1,2,5,7-t...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1D adrenergic receptor(Human)
Synaptic Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50085005(1-{3-[(4-Benzo[1,3]dioxol-5-yl-2,5-dioxo-1,2,5,7-t...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]- prazosin from human recombinant Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed