Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50009568
TargetSodium-dependent dopamine transporter(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50085072(GBR-12909 | 1-{2-[(3-Fluoro-phenyl)-(4-fluoro-phen...)
Affinity DataKi:  0.360nMAssay Description:Competitive binding versus [N-methyl-3H]WIN-35428 in murine kidney cells transfected with human dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50085071(3-(4-Iodo-phenyl)-6-methyl-6-aza-bicyclo[3.2.2]non...)
Affinity DataKi:  0.480nMAssay Description:In vitro affinity determined using [3H]WIN-35428 in murine kidney cells transfected with human dopamine transporter (DAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50085071(3-(4-Iodo-phenyl)-6-methyl-6-aza-bicyclo[3.2.2]non...)
Affinity DataKi:  0.670nMAssay Description:In vitro affinity determined using [3H]citalopram in murine kidney cells transfected with human serotonin transporter (SERT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50085069(3-(4-Chloro-phenyl)-6-methyl-6-aza-bicyclo[3.2.2]n...)
Affinity DataKi:  0.900nMAssay Description:Inhibition constant against [N-methyl-3H]WIN-35428 in murine kidney cells transfected with human dopamine transporter.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50028091((1E)-5-methoxy-1-[4-(trifluoromethyl)phenyl]pentan...)
Affinity DataKi:  3.08nMAssay Description:Inhibition constant against [3H]citalopram in murine kidney cells transfected with human dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50085069(3-(4-Chloro-phenyl)-6-methyl-6-aza-bicyclo[3.2.2]n...)
Affinity DataKi:  427nMAssay Description:Inhibition constant against [3H]citalopram in murine kidney cells transfected with human serotonin transporter.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed