Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50009596
Target1-alkyl-2-acetylglycerophosphocholine esterase(Pig)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085497(2-Ethylamino-hexadecan-1-ol | 2-(ethylamino)hexade...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of secretory PLA2 activity in porcine pancreas using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target1-alkyl-2-acetylglycerophosphocholine esterase(Pig)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085496(N*1*,N*1*-Diethyl-hexadecane-1,2-diamine | N1,N1-d...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of secretory PLA2 activity in porcine pancreas using [3H]-oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085497(2-Ethylamino-hexadecan-1-ol | 2-(ethylamino)hexade...)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of secretory PLA2 activity in human recombinant synovial enzyme using [3H]oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, membrane associated(Human)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085496(N*1*,N*1*-Diethyl-hexadecane-1,2-diamine | N1,N1-d...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of secretory PLA2 activity in human recombinant synovial enzyme using [3H]oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085497(2-Ethylamino-hexadecan-1-ol | 2-(ethylamino)hexade...)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of secretory PLA2 activity in bee venom enzyme using [3H]oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085497(2-Ethylamino-hexadecan-1-ol | 2-(ethylamino)hexade...)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of secretory PLA2 activity in bee venom enzyme using [3H]oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085496(N*1*,N*1*-Diethyl-hexadecane-1,2-diamine | N1,N1-d...)
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of secretory PLA2 activity in Naja naja venom enzyme using [3H]oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Mouse)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085498(4-(1-Benzyloxymethyl-pentadecylcarbamoyl)-butyric ...)
Affinity DataIC50: 1.05E+4nMAssay Description:Effect on cytosolic Phospholipase A2 (PLA2) activity at a concentration of 100 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085496(N*1*,N*1*-Diethyl-hexadecane-1,2-diamine | N1,N1-d...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of secretory PLA2 activity in bee venom enzyme using [3H]oleate labelled membranes at a concentration of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Mouse)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085494(1,1,1-trifluoroheptadecan-2-one | 1,1,1-Trifluoro-...)
Affinity DataIC50: 1.17E+4nMAssay Description:Effect on cytosolic Phospholipase A2 (PLA2) activity at a concentration of 100 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Mouse)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085496(N*1*,N*1*-Diethyl-hexadecane-1,2-diamine | N1,N1-d...)
Affinity DataIC50: 1.19E+4nMAssay Description:Effect on cytosolic Phospholipase A2 (PLA2) activity at a concentration of 100 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Mouse)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085499(N-(1-Benzyloxymethyl-pentadecyl)-succinamic acid |...)
Affinity DataIC50: 6.28E+4nMAssay Description:Effect on cytosolic Phospholipase A2 (PLA2) activity at a concentration of 100 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Mouse)
Univ. De Valencia

Curated by ChEMBL
LigandPNGBDBM50085495((E)-3-(1-Benzyloxymethyl-pentadecylcarbamoyl)-acry...)
Affinity DataIC50: 6.95E+4nMAssay Description:Effect on cytosolic Phospholipase A2 (PLA2) activity at a concentration of 100 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed