Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50009643
TargetCytosolic phospholipase A2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085993((E)-N-(((2S,4R)-4-((biphenyl-2-ylmethyl)(isobutyl)...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085984(N-[1-[2-(2,4-Difluoro-benzoyl)-benzoyl]-4-(3-isobu...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085986(N-{4-(Biphenyl-2-ylmethyl-isobutyl-amino)-1-[2-(4-...)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085987(4-(2,4-Dioxo-thiazolidin-5-ylidenemethyl)-N-[1-[2-...)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085994(N-{4-(Biphenyl-2-ylmethyl-isobutyl-amino)-1-[2-(2,...)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085980(N-{4-(Biphenyl-2-ylmethyl-isobutyl-amino)-1-[2-(4-...)
Affinity DataIC50: 21nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085997(N-{4-(2-Bromo-6-isobutyl-phenoxy)-1-[2-(2,4-difluo...)
Affinity DataIC50: 22nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085990(N-{4-(Biphenyl-2-ylmethylsulfanyl)-1-[2-(4-fluoro-...)
Affinity DataIC50: 34nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085991(N-{4-(2-Bromo-6-isobutyl-phenoxy)-1-[2-(4-fluoro-b...)
Affinity DataIC50: 38nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085983(N-{4-(Biphenyl-2-ylmethoxy)-1-[2-(2,4-difluoro-ben...)
Affinity DataIC50: 49nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085988(N-{4-(Biphenyl-2-yloxy)-1-[2-(4-fluoro-benzoyl)-be...)
Affinity DataIC50: 69nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085981(N-{4-(Biphenyl-2-ylmethylsulfanyl)-1-[2-(4-fluoro-...)
Affinity DataIC50: 72nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085982(N-{4-(Biphenyl-2-ylmethoxy)-1-[2-(4-fluoro-benzoyl...)
Affinity DataIC50: 78nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085989(N-{4-(Biphenyl-2-yloxy)-1-[2-(4-fluoro-benzoyl)-be...)
Affinity DataIC50: 83nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085985(N-{4-(Biphenyl-2-ylmethoxy)-1-[2-(4-fluoro-benzoyl...)
Affinity DataIC50: 90nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085992(N-[(2S,4R)-1-(2-Benzoyl-benzoyl)-4-(biphenyl-2-ylm...)
Affinity DataIC50: 165nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085998(1,1,1-Trifluoro-docosa-7,10,13,16-tetraen-3-one | ...)
Affinity DataIC50: 420nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085996(N-[1-(4-Benzoyl-benzoyl)-4-(biphenyl-2-ylmethoxy)-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosolic phospholipase A2(Human)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50085999(N-[1-(3-Benzoyl-benzoyl)-4-(biphenyl-2-ylmethoxy)-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed