Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50009732
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50085904(3-Isopropyl-4-methyl-pentanoic acid 2-hydroxymethy...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [20-3H] phorbol 12,13-dibutyrate from protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50087241(3-Isopropyl-4-methyl-pentanoic acid 3-hydroxy-2-(3...)
Affinity DataKi:  29nMAssay Description:Displacement of [20-3H] phorbol 12,13-dibutyrate from protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50015677(CHEMBL55267 | 1,2-dioctanoyl-sn-glycerol | 1,2-Dio...)
Affinity DataKi:  33nMAssay Description:Displacement of [20-3H] phorbol 12,13-dibutyrate from protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50087239(Diacylglycerol derivative | CHEMBL345343)
Affinity DataKi:  39nMAssay Description:Displacement of [20-3H] phorbol 12,13-dibutyrate from protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50087237(AutoNom Name: | CHEMBL158666)
Affinity DataKi:  50nMAssay Description:Displacement of [20-3H] phorbol 12,13-dibutyrate from protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50087240((E)-Octadec-9-enoic acid (S)-1-hydroxymethyl-2-((E...)
Affinity DataKi:  87nMAssay Description:Displacement of [20-3H] phorbol 12,13-dibutyrate from protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50087238(2,2-Dimethyl-propionic acid 2-(2,2-dimethyl-propio...)
Affinity DataKi:  3.43E+3nMAssay Description:Displacement of [20-3H] phorbol 12,13-dibutyrate from protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed