Compile Data Set for Download or QSAR
Report error Found 233 Enz. Inhib. hit(s) with all data for entry = 50036926
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50037996(N-[1-(4-Carbamimidoyl-benzyl)-2-oxo-2-piperidin-1-...)
Affinity DataKi:  6.5nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087898(1-(3-Phenyl-2-(N-Toluene-4-sulfonyl)ureido-propion...)
Affinity DataKi:  10nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087941(N-{4-[(N-Guanidino)-sulfamoyl]-phenyl}-3-(1H-imida...)
Affinity DataKi:  10nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087955([2-(2-{4-[(N-Guanidino)-sulfamoyl]-phenylcarbamoyl...)
Affinity DataKi:  11nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087983(N-[4-(Diaminomethylene-sulfamoyl)-phenyl]-3-phenyl...)
Affinity DataKi:  12nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087903((1-Benzyl-2-{2-[4-(diaminomethylene-sulfamoyl)-phe...)
Affinity DataKi:  13nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087888(N-{4-[(N-Guanidino)-sulfamoyl]-phenyl}-3-(1H-imida...)
Affinity DataKi:  15nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087907(N-[4-(Diaminomethylene-sulfamoyl)-phenyl]-3-(1H-im...)
Affinity DataKi:  15nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087960({1-Cyclohexylmethyl-2-[2-(3-guanidino-propylcarbam...)
Affinity DataKi:  15nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087962(1-(Toluene-4-sulfonylaminocarbonyl)-pyrrolidine-2-...)
Affinity DataKi:  15nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087963([2-(2-{4-[(Amino-methoxy-methylene)-sulfamoyl]-phe...)
Affinity DataKi:  16nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087954(1-(3-Phenyl-2-(N-Toluene-4-sulfonyl)ureido-propion...)
Affinity DataKi:  18nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087998(N-[4-(Diaminomethylene-sulfamoyl)-phenyl]-3-(1H-im...)
Affinity DataKi:  18nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50038001(CHEMBL1166 | (2R,4S)-1-[5-Guanidino-2-(3-methyl-1,...)
Affinity DataKi:  19nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087994(N-{4-[(Amino-methoxy-methylene)-sulfamoyl]-phenyl}...)
Affinity DataKi:  19nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087967(N-{4-[(Amino-methoxy-methylene)-sulfamoyl]-phenyl}...)
Affinity DataKi:  21nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087965(1-(Toluene-4-sulfonylaminocarbonyl)-pyrrolidine-2-...)
Affinity DataKi:  21nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087902(1-(Toluene-4-sulfonylaminocarbonyl)-pyrrolidine-2-...)
Affinity DataKi:  27nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087953({1-[4-(Diaminomethylene-sulfamoyl)-phenylcarbamoyl...)
Affinity DataKi:  43nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087959(1-(Toluene-4-sulfonylaminocarbonyl)-pyrrolidine-2-...)
Affinity DataKi:  43nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087901(N-{4-[(N-Guanidino)-sulfamoyl]-phenyl}-3-phenyl-2-...)
Affinity DataKi:  44nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087973(1-(Toluene-4-sulfonylaminocarbonyl)-pyrrolidine-2-...)
Affinity DataKi:  48nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087886((1-{4-[(N-Guanidino)-sulfamoyl]-phenylcarbamoyl}-2...)
Affinity DataKi:  50nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087930({1-[4-(Diaminomethylene-sulfamoyl)-phenylcarbamoyl...)
Affinity DataKi:  54nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087921(N-{4-[(Amino-methoxy-methylene)-sulfamoyl]-phenyl}...)
Affinity DataKi:  60nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087969((1-{4-[(Amino-methoxy-methylene)-sulfamoyl]-phenyl...)
Affinity DataKi:  62nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087923(1-(Toluene-4-sulfonylaminocarbonyl)-pyrrolidine-2-...)
Affinity DataKi:  63nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087912(N''-[(3-aminophenyl)sulfonyl]carbonohydrazonic dia...)
Affinity DataKi:  88nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087925(N''-[(4-aminophenyl)sulfonyl]carbonohydrazonic dia...)
Affinity DataKi:  91nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50027795(2-[(dioxidosulfanyl)amino]-1,9-dihydro-6H-purin-6-...)
Affinity DataKi:  95nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087884(3-Amino-N-(amino-methoxy-methylene)-4-methoxy-benz...)
Affinity DataKi:  96nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087885(4-{[2-(diaminomethylene)hydrazino]sulfonyl}benzoic...)
Affinity DataKi:  97nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087897(N''-[(3,5-dichloro-2-hydroxyphenyl)sulfonyl]carbon...)
Affinity DataKi:  98nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087966(3-Amino-N-(amino-methoxy-methylene)-benzenesulfona...)
Affinity DataKi:  99nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087993(3-Amino-N-diaminomethylene-4-methoxy-benzenesulfon...)
Affinity DataKi:  103nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087894(4-(Diaminomethylene-sulfamoyl)-benzoic acid | CHEM...)
Affinity DataKi:  104nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087991(4-Amino-N-(amino-methoxy-methylene)-benzenesulfona...)
Affinity DataKi:  106nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087951(3-Amino-N-diaminomethylene-benzenesulfonamide | CH...)
Affinity DataKi:  107nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087890(3-{[2-(diaminomethylene)hydrazino]sulfonyl}benzoic...)
Affinity DataKi:  112nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087945(5-Dimethylamino-naphthalene-1-sulfonic acid diamin...)
Affinity DataKi:  120nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087948(3-(Diaminomethylene-sulfamoyl)-benzoic acid | CHEM...)
Affinity DataKi:  121nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087940(N''-[(pentafluorophenyl)sulfonyl]carbonohydrazonic...)
Affinity DataKi:  123nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087986(N''-(1-naphthylsulfonyl)carbonohydrazonic diamide ...)
Affinity DataKi:  125nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087976(N''-(2-naphthylsulfonyl)carbonohydrazonic diamide ...)
Affinity DataKi:  129nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087920(N''-{[5-(dimethylamino)-1-naphthyl]sulfonyl}carbon...)
Affinity DataKi:  130nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087947(Naphthalene-2-sulfonic acid diaminomethyleneamide ...)
Affinity DataKi:  132nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087933(4-[(Amino-methoxy-methylene)-sulfamoyl]-benzoic ac...)
Affinity DataKi:  133nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087937(N-Diaminomethylene-4-(4-dimethylamino-phenylazo)-b...)
Affinity DataKi:  134nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087918(Naphthalene-1-sulfonic acid diaminomethyleneamide ...)
Affinity DataKi:  136nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50087932(5-Dimethylamino-naphthalene-1-sulfonic acid amino-...)
Affinity DataKi:  138nMAssay Description:Inhibitory activity against human thrombin (using Chromozym TH as the substrate)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Displayed 1 to 50 (of 233 total ) | Next | Last >>
Jump to: