Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50009897
TargetUrokinase-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088982(CHEMBL160253 | CHEMBL367004 | N-[1-(1-Carbamimidoy...)
Affinity DataIC50: 3.10nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088978(N-[1-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcarb...)
Affinity DataIC50: 5.10nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088984(2-Benzenesulfonylamino-N-[1-(1-carbamimidoyl-2-hyd...)
Affinity DataIC50: 10nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088979({(R)-2-[2-((S)-1-Carbamimidoyl-2-hydroxy-piperidin...)
Affinity DataIC50: 11nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088985({2-[2-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 12nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088977({1-[1-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 19nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088987({1-[1-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 23nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088986({2-[2-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 101nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088985({2-[2-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 125nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088981({1-[1-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 261nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088978(N-[1-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcarb...)
Affinity DataIC50: 275nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088982(CHEMBL160253 | CHEMBL367004 | N-[1-(1-Carbamimidoy...)
Affinity DataIC50: 367nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088979({(R)-2-[2-((S)-1-Carbamimidoyl-2-hydroxy-piperidin...)
Affinity DataIC50: 482nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088981({1-[1-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 699nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088977({1-[1-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 904nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088984(2-Benzenesulfonylamino-N-[1-(1-carbamimidoyl-2-hyd...)
Affinity DataIC50: 1.17E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088987({1-[1-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 1.46E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088983({1-[1-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088977({1-[1-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088983({1-[1-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetUrokinase-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088980({(R)-1-[(S)-1-((S)-1-Carbamimidoyl-2-hydroxy-piper...)
Affinity DataIC50: 2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088984(2-Benzenesulfonylamino-N-[1-(1-carbamimidoyl-2-hyd...)
Affinity DataIC50: 2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088979({(R)-2-[2-((S)-1-Carbamimidoyl-2-hydroxy-piperidin...)
Affinity DataIC50: 2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088987({1-[1-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088978(N-[1-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcarb...)
Affinity DataIC50: 2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088981({1-[1-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088980({(R)-1-[(S)-1-((S)-1-Carbamimidoyl-2-hydroxy-piper...)
Affinity DataIC50: 2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088982(CHEMBL160253 | CHEMBL367004 | N-[1-(1-Carbamimidoy...)
Affinity DataIC50: 2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088983({1-[1-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088986({2-[2-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088980({(R)-1-[(S)-1-((S)-1-Carbamimidoyl-2-hydroxy-piper...)
Affinity DataIC50: 2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Corvas International

Curated by ChEMBL
LigandPNGBDBM50088985({2-[2-(1-Carbamimidoyl-2-hydroxy-piperidin-3-ylcar...)
Affinity DataIC50: 2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed