Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50009906
TargetIntegrin alpha-4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50089019((8R,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-prop...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of VLA-4 binding to recombinant human VCAM using Ramos cell assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50089029((8R,13R)-13-[(S)-2-Acetylamino-3-(4-hydroxy-phenyl...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of VLA-4 binding to recombinant human VCAM using Solid phase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50089027((5R,8S,13S,15aR)-8-[(S)-2-Acetylamino-3-(4-hydroxy...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of VLA-4 binding to recombinant human VCAM using Solid phase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50089030((4R,12R)-12-[(S)-2-Amino-3-(4-hydroxy-phenyl)-prop...)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of VLA-4 binding to recombinant human VCAM using Ramos cell assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50089026((8R,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-prop...)
Affinity DataIC50: 5nMAssay Description:Inhibition of VLA-4 binding to recombinant human VCAM using Ramos cell assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50089029((8R,13R)-13-[(S)-2-Acetylamino-3-(4-hydroxy-phenyl...)
Affinity DataIC50: 12nMAssay Description:Inhibition of VLA-4 binding to recombinant human VCAM using Ramos cell assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50089025((8R,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-prop...)
Affinity DataIC50: 19nMAssay Description:Inhibition of VLA-4 binding to recombinant human VCAM using Solid phase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50089019((8R,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-prop...)
Affinity DataIC50: 24nMAssay Description:Inhibition of VLA-4 binding to recombinant human VCAM using Ramos cell assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50089028((4R,12R)-12-[(S)-2-Amino-3-(4-hydroxy-phenyl)-prop...)
Affinity DataIC50: 112nMAssay Description:Inhibition of VLA-4 binding to recombinant human VCAM using Ramos cell assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50089027((5R,8S,13S,15aR)-8-[(S)-2-Acetylamino-3-(4-hydroxy...)
Affinity DataIC50: 200nMAssay Description:Inhibition of VLA-4 binding to recombinant human VCAM using Ramos cell assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-4(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50089025((8R,13R)-13-[(S)-2-Amino-3-(4-hydroxy-phenyl)-prop...)
Affinity DataIC50: 480nMAssay Description:Inhibition of VLA-4 binding to recombinant human VCAM using Ramos cell assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed