Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50035052
TargetMu-type opioid receptor(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM21015([tyrosyl-3,5-3H(N)]-D-Ala2-Mephe4-glyol5-enkephali...)
Affinity DataKi:  0.530nMAssay Description:Compound was evaluated for the binding affinity of Opioid receptor mu 1 by displacing the radioligand [3H]DAMGO from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50089073(({1-[3-({1-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...)
Affinity DataKi:  720nMAssay Description:Compound was evaluated for the binding affinity of Opioid receptor mu 1 by displacing the radioligand [3H]DAMGO from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50089075(2-({1-[2-({1-[3-({1-[2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataKi:  1.44E+3nMAssay Description:Compound was evaluated for the binding affinity of Opioid receptor mu 1 by displacing the radioligand [3H]DAMGO from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50089071(({1-[2-({1-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...)
Affinity DataKi:  1.62E+3nMAssay Description:Compound was evaluated for the binding affinity of Opioid receptor mu 1 by displacing the radioligand [3H]DAMGO from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50089073(({1-[3-({1-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory concentration against [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50089075(2-({1-[2-({1-[3-({1-[2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibitory concentration against [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50089071(({1-[2-({1-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibitory concentration against [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50089072(2-({1-[2-({1-[2-({1-[2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataKi:  7.54E+3nMAssay Description:Compound was evaluated for the binding affinity of Opioid receptor mu 1 by displacing the radioligand [3H]DAMGO from rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandPNGBDBM50089072(2-({1-[2-({1-[2-({1-[2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory concentration against [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed