Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50009945
TargetB1 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089316(H-Lys-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT-OH(JMV1645) | C...)
Affinity DataKi:  0.0230nMAssay Description:Binding affinity towards human cloned B1 receptor was determined using [3H][des-Arg10-Leu9]-kallidin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089316(H-Lys-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT-OH(JMV1645) | C...)
Affinity DataKi:  9.16nMAssay Description:Binding affinity towards human cloned B2 receptor was determined using [3H]BK as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089315({3-[2-(2-{8-[2-(2,6-Diamino-hexanoylamino)-5-guani...)
Affinity DataKi:  24.1nMAssay Description:Binding affinity towards human cloned B1 receptor was determined using [3H][des-Arg10-Leu9]-kallidin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089315({3-[2-(2-{8-[2-(2,6-Diamino-hexanoylamino)-5-guani...)
Affinity DataKi:  1.19E+4nMAssay Description:Binding affinity towards human cloned B2 receptor was determined using [3H]BK as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed