Compile Data Set for Download or QSAR
Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 50041033
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090430(ethyl 4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamin...)
Affinity DataIC50: 20nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090444(4-(3-Methyl-2,5-dioxo-2,5-dihydro-pyrrol-1-ylamino...)
Affinity DataIC50: 100nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090407(ethyl 4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamin...)
Affinity DataIC50: 100nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090442(3-methyl-1-(5-(2-methyl-2H-tetrazol-5-yl)-2-(thiop...)
Affinity DataIC50: 200nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090406(1-[5-(4,5-Dihydro-oxazol-2-yl)-2-thiophen-2-yl-pyr...)
Affinity DataIC50: 200nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090443(4-(3-Methyl-2,5-dioxo-2,5-dihydro-pyrrol-1-ylamino...)
Affinity DataIC50: 200nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090431(3-methyl-1-(5-(4-methyloxazol-2-yl)-2-(thiophen-2-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090420(4-(3-Methyl-2,5-dioxo-2,5-dihydro-pyrrol-1-ylamino...)
Affinity DataIC50: 200nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090450(3-methyl-1-(5-(5-methyl-1,3,4-oxadiazol-2-yl)-2-(t...)
Affinity DataIC50: 300nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090449(ethyl 2-(4-chlorophenyl)-4-(3-methyl-2,5-dioxo-2H-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090435(3-methyl-1-(5-(3-methylisoxazol-5-yl)-2-(thiophen-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090433(ethyl 2-(5-chlorothiophen-2-yl)-4-(3-methyl-2,5-di...)
Affinity DataIC50: 300nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090429(ethyl 2-(3,5-dichlorophenyl)-4-(3-methyl-2,5-dioxo...)
Affinity DataIC50: 300nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090440(4-(3-Methyl-2,5-dioxo-2,5-dihydro-pyrrol-1-ylamino...)
Affinity DataIC50: 400nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090426(ethyl 2-(4-fluorophenyl)-4-(3-methyl-2,5-dioxo-2H-...)
Affinity DataIC50: 700nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090441(2-(3-Bromo-phenyl)-4-(3-methyl-2,5-dioxo-2,5-dihyd...)
Affinity DataIC50: 700nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090421(ethyl 2-(furan-2-carbonyl)-4-(3-methyl-2,5-dioxo-2...)
Affinity DataIC50: 700nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090409(2-(4-Methoxy-phenyl)-4-(3-methyl-2,5-dioxo-2,5-dih...)
Affinity DataIC50: 900nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090408(4-(3-Methyl-2,5-dioxo-2,5-dihydro-pyrrol-1-ylamino...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090447(ethyl 2-tert-butyl-4-(3-methyl-2,5-dioxo-2H-pyrrol...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090410(ethyl 4-(methyl(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090432(2-Cyclopropyl-4-(3-methyl-2,5-dioxo-2,5-dihydro-py...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090415(ethyl 4-(3-methyl-2,5-dioxo-2,5-dihydro-1H-pyrrol-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090411(ethyl 2-(2,6-dichloropyridin-4-yl)-4-(3-methyl-2,5...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090436(ethyl 4-(methyl(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090437(2-Cyclohex-1-enylmethyl-4-(3-methyl-2,5-dioxo-2,5-...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090445(2-(4-Fluoro-phenyl)-4-[methyl-(3-methyl-2,5-dioxo-...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090439(2-Benzo[b]thiophen-2-yl-4-(3-methyl-2,5-dioxo-2,5-...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090425(4-[Acetyl-(3-methyl-2,5-dioxo-2,5-dihydro-pyrrol-1...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090428(4-(3-Methyl-2,5-dioxo-2,5-dihydro-pyrrol-1-ylamino...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090427(ethyl 2-(3-methoxyphenyl)-4-(3-methyl-2,5-dioxo-2H...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090446(ethyl 4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamin...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090423(ethyl 4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamin...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090414(ethyl 2-benzyl-4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090422(4-(3-Methyl-2,5-dioxo-2,5-dihydro-pyrrol-1-ylamino...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090417(4-(3-Methyl-2,5-dioxo-2,5-dihydro-pyrrol-1-ylamino...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090424(2-Benzenesulfonyl-4-(3-methyl-2,5-dioxo-2,5-dihydr...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090419(ethyl 4-(2,5-dioxo-2H-pyrrol-1(5H)-ylamino)-2-(tri...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090438(ethyl 2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-(3-methyl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090416(2-Ethyl-4-(3-methyl-2,5-dioxo-2,5-dihydro-pyrrol-1...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090413(ethyl 2-ethyl-4-(methyl(3-methyl-2,5-dioxo-2H-pyrr...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090434(ethyl 4-(3,4-dimethyl-2,5-dioxo-2H-pyrrol-1(5H)-yl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090418(ethyl 4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamin...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090448(2-Methyl-4-(3-methyl-2,5-dioxo-2,5-dihydro-pyrrol-...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090412(4-(2,5-Dioxo-3-phenyl-2,5-dihydro-pyrrol-1-ylamino...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed