Compile Data Set for Download or QSAR
Report error Found 75 Enz. Inhib. hit(s) with all data for entry = 50010248
TargetGastrin/cholecystokinin type B receptor(Rat)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092399(3-(2-{[2-(2-Benzylcarbamoyl-acetylamino)-3-(1H-ind...)
Affinity DataEC50:  3.30nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092401(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{[2-(1H-indol-3-y...)
Affinity DataEC50:  7nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092405((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-((S)-2-{[...)
Affinity DataEC50:  0.400nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092408(N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2-{[3-(1H-indol-...)
Affinity DataEC50:  0.560nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092384(N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2-{[2-(3-carboxy...)
Affinity DataEC50:  1.5nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
University of Paris

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataEC50:  0.630nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092398((S)-3-((S)-2-{[(S)-2-tert-Butoxycarbonylamino-3-(1...)
Affinity DataEC50:  1.5nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092391(3-(2-{[2-(2-Carbamoyl-acetylamino)-3-(1H-indol-3-y...)
Affinity DataEC50:  1.64nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092393(3-(2-{[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-su...)
Affinity DataEC50:  3.40nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092395(3-{2-[2-{[9-tert-Butoxycarbonylamino-3-butyl-2,5,8...)
Affinity DataEC50:  17nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092389(N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2-{[3-(1H-indol-...)
Affinity DataEC50:  2nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50024317(Tetragastrin | CHEMBL120632 | 3-{2-[2-Amino-3-(1H-...)
Affinity DataEC50:  1.40nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50002477((S)-3-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataEC50:  1nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092393(3-(2-{[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-su...)
Affinity DataKi:  0.150nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092405((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-((S)-2-{[...)
Affinity DataKi:  0.280nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092393(3-(2-{[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-su...)
Affinity DataKi:  0.310nMAssay Description:Compound was tested for binding affinity against Cholecystokinin type B receptor expressed in CHO cells on the rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092408(N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2-{[3-(1H-indol-...)
Affinity DataKi:  0.540nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
University of Paris

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.600nMAssay Description:Compound was tested for binding affinity against Cholecystokinin type B receptor expressed in CHO cells on the rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092405((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-((S)-2-{[...)
Affinity DataKi: >0.700nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092398((S)-3-((S)-2-{[(S)-2-tert-Butoxycarbonylamino-3-(1...)
Affinity DataKi: >0.700nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.700nMAssay Description:Compound was tested for binding affinity against CCK1 (cholecystokinin) receptor on guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092405((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-((S)-2-{[...)
Affinity DataKi:  0.75nMAssay Description:Compound was tested for binding affinity against Cholecystokinin type B receptor expressed in CHO cells on the rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092398((S)-3-((S)-2-{[(S)-2-tert-Butoxycarbonylamino-3-(1...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092388(3-(2-{[2-(3-tert-Butoxycarbonylamino-propionylamin...)
Affinity DataKi:  1.35nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092387(N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2-{[3-(1H-indol-...)
Affinity DataKi:  1.37nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092399(3-(2-{[2-(2-Benzylcarbamoyl-acetylamino)-3-(1H-ind...)
Affinity DataKi:  1.81nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092391(3-(2-{[2-(2-Carbamoyl-acetylamino)-3-(1H-indol-3-y...)
Affinity DataKi:  2.05nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092404(N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2-{[3-(1H-indol-...)
Affinity DataKi:  2.52nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092396(3-(2-{[2-Amino-3-(1H-indol-3-yl)-propionyl]-methyl...)
Affinity DataKi:  2.60nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092398((S)-3-((S)-2-{[(S)-2-tert-Butoxycarbonylamino-3-(1...)
Affinity DataKi:  2.60nMAssay Description:Compound was tested for binding affinity against Cholecystokinin type B receptor expressed in CHO cells on the rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092410(2-tert-Butoxycarbonylamino-N-[1-({1-[1-(1-carbamoy...)
Affinity DataKi:  2.70nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092384(N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2-{[2-(3-carboxy...)
Affinity DataKi:  3.02nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092389(N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2-{[3-(1H-indol-...)
Affinity DataKi:  3.61nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092414(N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2-{[3-(1H-indol-...)
Affinity DataKi:  3.84nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092411(2-tert-Butoxycarbonylamino-N-[1-({1-[1-(1-carbamoy...)
Affinity DataKi:  4.07nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092402(N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2-{[3-(1H-indol-...)
Affinity DataKi:  4.35nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092397(3-Amino-N-[1-({1-[1-(1-carbamoyl-2-phenyl-ethylcar...)
Affinity DataKi:  4.80nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092395(3-{2-[2-{[9-tert-Butoxycarbonylamino-3-butyl-2,5,8...)
Affinity DataKi:  6.40nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092413(3-tert-Butoxycarbonylamino-N-[1-({1-[1-(1-carbamoy...)
Affinity DataKi:  7.31nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092406(3-tert-Butoxycarbonylamino-N-[1-({1-[1-(1-carbamoy...)
Affinity DataKi:  7.76nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50002477((S)-3-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataKi:  9.40nMAssay Description:Compound was tested for binding affinity against Cholecystokinin type B receptor expressed in CHO cells on the rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092409(3-Amino-N-[1-({1-[1-(1-carbamoyl-2-phenyl-ethylcar...)
Affinity DataKi:  11.9nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092400(3-(2-{[2-(2-Amino-propionylamino)-3-(1H-indol-3-yl...)
Affinity DataKi:  15nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092401(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{[2-(1H-indol-3-y...)
Affinity DataKi:  15nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092394(3-(2-{[2-(2-Amino-acetylamino)-3-(1H-indol-3-yl)-p...)
Affinity DataKi:  18nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092401(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{[2-(1H-indol-3-y...)
Affinity DataKi:  18nMAssay Description:Compound was tested for binding affinity against Cholecystokinin type B receptor expressed in CHO cells on the rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50024317(Tetragastrin | CHEMBL120632 | 3-{2-[2-Amino-3-(1H-...)
Affinity DataKi:  19.5nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092390(3-(2-{[2-(2-Amino-propionylamino)-3-(1H-indol-3-yl...)
Affinity DataKi:  20nMAssay Description:Affinity against Cholecystokinin type A receptor on guinea pig pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50092403(N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2-{[3-(1H-indol-...)
Affinity DataKi:  23.8nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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