Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50010252
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092455(1-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 1.40nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092453(N-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 1.80nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092421(1-(2,6-Dichloro-phenyl)-3-{2-[1-(2,3-dihydro-benzo...)
Affinity DataIC50: 2.30nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092440(1-Benzoyl-3-{2-[1-(2,3-dihydro-benzo[1,4]dioxin-2-...)
Affinity DataIC50: 2.60nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092425(2-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 3.80nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092452(1-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 4.5nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092434(1-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092431(2-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092419(1-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092423(1-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 11nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092443(3-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 11.5nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092427(1-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 15nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092446(1-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 15nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092429(3-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 16nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092457(N-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 24nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092456(N-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 24nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092445(N-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 25nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092448(Phenyl-carbamic acid 2-[1-(2,3-dihydro-benzo[1,4]d...)
Affinity DataIC50: 26nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092439(3-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 28nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092438(N-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 30nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092437(1-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 32nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092451(1-Cyclohexyl-3-{2-[1-(2,3-dihydro-benzo[1,4]dioxin...)
Affinity DataIC50: 35nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092430(1-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 36nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092428(1-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 38nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092426(N-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 41nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092420(1-Benzyl-3-{2-[1-(2,3-dihydro-benzo[1,4]dioxin-2-y...)
Affinity DataIC50: 45nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092442(Benzothiazol-2-yl-[1-(2,3-dihydro-benzo[1,4]dioxin...)
Affinity DataIC50: 50nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092458(N-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 50nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092432({2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-pi...)
Affinity DataIC50: 52nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092449(1-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 80nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092422(1-{3-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 90nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092424(1-Benzoyl-3-{2-[1-(2,3-dihydro-benzo[1,4]dioxin-2-...)
Affinity DataIC50: 120nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092454(1-(2,6-Diethoxy-phenyl)-3-{2-[1-(2,3-dihydro-benzo...)
Affinity DataIC50: 135nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092447(1-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 210nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092435(1-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 320nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092417(1-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 480nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092436(3-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-pip...)
Affinity DataIC50: 550nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092441(1-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-pip...)
Affinity DataIC50: 750nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092418(1-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-pip...)
Affinity DataIC50: 750nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50092450(N-{2-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-...)
Affinity DataIC50: 800nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataIC50: 1.13E+3nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50019848(CHEMBL10316 | Idazoxan | US8633208, Idazoxan | 4,5...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of specific binding of [3H]-YM 09151-2 to Dopamine receptor D2 site in rat striatal tissue.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed